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non condensed and containing further heterocyclic rings
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A61K31/4155
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HUMAN NECESSITIES
A61
Medical science
A61K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
A61K31/00
Medicinal preparations containing organic active ingredients
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A61K31/4155
non condensed and containing further heterocyclic rings
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Patents Grants
last 30 patents
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Patent Grant
Small molecule inhibitors of lactate dehydrogenase and methods of u...
Patent number
12,365,653
Issue date
Jul 22, 2025
THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF...
David J. Maloney
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
6-hydroxy-8-oxatricyclo[3.2.1.02,4]octane-2-carboxamide derivatives...
Patent number
12,365,692
Issue date
Jul 22, 2025
Novartis AG
James Paul Lajiness
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Acyl sulfonamides for treating cancer
Patent number
12,357,603
Issue date
Jul 15, 2025
Bayer Aktiengesellschaft
Léa Aurelie Bouché
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
JAK1 pathway inhibitors for the treatment of cytokine-related disor...
Patent number
12,336,998
Issue date
Jun 24, 2025
Incyte Corporation
Michael O'Neill Montgomery
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Coumarin-modified androgens for the treatment of prostate cancer
Patent number
12,337,004
Issue date
Jun 24, 2025
Health Research, Inc.
James L. Mohler
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted heterocyclyl derivatives as CDK inhibitors
Patent number
12,331,023
Issue date
Jun 17, 2025
AURIGENE ONCOLOGY LIMITED
Susanta Samajdar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pharmaceutical composition of darolutamide
Patent number
12,329,742
Issue date
Jun 17, 2025
Orion Corporation
Susanna Ilmonen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pharmaceutical combination and composition, and combination prepara...
Patent number
12,318,366
Issue date
Jun 3, 2025
Hua Medicine (Shanghai) Ltd.
Li Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Inhibition of dipeptide repeat proteins
Patent number
12,318,365
Issue date
Jun 3, 2025
ALS THERAPY DEVELOPMENT INSTITUTE
Fernando G. Vieira
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
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Patent Grant
Methods and compositions for the prevention and treatment of hearin...
Patent number
12,318,391
Issue date
Jun 3, 2025
St. Jude Children's Research Hospital, Inc.
Jian Zuo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Methods and compositions for unsilencing imprinted genes
Patent number
12,310,947
Issue date
May 27, 2025
The University of North Carolina at Chapel Hill
Benjamin D. Philpot
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Anti-androgens for the treatment of metastatic castration-sensitive...
Patent number
12,303,497
Issue date
May 20, 2025
Aragon Pharmaceuticals, Inc.
Margaret K. Yu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Charged ion channel blockers and methods for use
Patent number
12,303,496
Issue date
May 20, 2025
Nocion Therapeutics, Inc.
Bridget McCarthy Cole
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Inhibitors of receptor interacting protein kinase I for the treatme...
Patent number
12,286,406
Issue date
Apr 29, 2025
Board of Regents, The University of Texas System
Richard T. Lewis
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Inhibiting monoacylglycerol lipase (MAGL)
Patent number
12,286,421
Issue date
Apr 29, 2025
Psy Therapeutics, Inc.
Jacob Matthew Hooker
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Combination comprising HDAC inhibitor and CD137 agonist for cancer...
Patent number
12,285,410
Issue date
Apr 29, 2025
4SC AG
Svetlana Hamm
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
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Patent Grant
Compounds and compositions for inducing chondrogenesis
Patent number
12,280,041
Issue date
Apr 22, 2025
Novartis AG
Ha-Soon Choi
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Grant
JAK1 pathway inhibitors for the treatment of prurigo nodularis
Patent number
12,268,667
Issue date
Apr 8, 2025
Incyte Corporation
Paul Smith
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Autotaxin inhibitor compounds
Patent number
12,268,668
Issue date
Apr 8, 2025
SABRE THERAPEUTICS LLC
John Howard Hutchinson
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Carboxylic acid aromatic amides as antagonists of bradykinin B1 rec...
Patent number
12,239,630
Issue date
Mar 4, 2025
Bayer Pharma Aktiengesellschaft
Stefan Baeurle
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Neuroprotective disruption of Kv2.1/syntaxin interaction by small m...
Patent number
12,226,400
Issue date
Feb 18, 2025
University of Pittsburgh of the Commonwealth System of Higher Education
Elias Aizenman
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds useful as kinase inhibitors
Patent number
12,220,401
Issue date
Feb 11, 2025
Loxo Oncology, Inc.
Nicolas Guisot
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted indole Mcl-1 inhibitors
Patent number
12,195,472
Issue date
Jan 14, 2025
Vanderbilt University
Taekyu Lee
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
MCT4 inhibitors for treating disease
Patent number
12,187,682
Issue date
Jan 7, 2025
Vettore, LLC
Kenneth Mark Parnell
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Uses of indolinone compounds
Patent number
12,161,626
Issue date
Dec 10, 2024
Oncternal Therapeutics, Inc.
Brian Lannutti
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
JAK1 pathway inhibitors for the treatment of gastrointestinal disease
Patent number
12,150,943
Issue date
Nov 26, 2024
Incyte Corporation
Krishnaswamy Yeleswaram
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds and radioligands for targeting neurotensin receptor and u...
Patent number
12,145,926
Issue date
Nov 19, 2024
Full-Life Technologies HK Limited
Fa Liu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
ACSS2 inhibitors and methods of use thereof
Patent number
12,133,852
Issue date
Nov 5, 2024
EpiVario, Inc.
Philippe Nakache
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
AUTOTAC chimeric compound, and composition for preventing, ameliora...
Patent number
12,129,218
Issue date
Oct 29, 2024
AUTOTAC INC.
Yong Tae Kwon
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Fap-activated therapeutic agents, and uses related thereto
Patent number
12,121,505
Issue date
Oct 22, 2024
BACH BIOSCIENCES, LLC
William W. Bachovchin
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
COMBINATION THERAPY FOR TREATING CANCER
Publication number
20250235448
Publication date
Jul 24, 2025
AstraZeneca AB
Sabina Chiara COSULICH
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLYL COMPOUNDS AS KV7 CHANNEL ACTIVATORS
Publication number
20250230152
Publication date
Jul 17, 2025
BIOHAVEN THERAPEUTICS LTD.
Lynn RESNICK
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DISTINCT CD8+ T CELL PROGRAMMING IN THE TUMOR MICROENVIRONMENT CONT...
Publication number
20250228915
Publication date
Jul 17, 2025
Ohio State Innovation Foundation
Zihai LI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
2,3-DIHYDROBENZO[B][1,4]DIOXIN-6-YL CONTAINING COMPOUNDS USEFUL AS...
Publication number
20250230153
Publication date
Jul 17, 2025
Bristol-Myers Squibb Company
Timothy P. Connolly
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL BENZOTHIOPHENE DERIVATIVE AND USE THEREOF AS BET INHIBITOR
Publication number
20250221977
Publication date
Jul 10, 2025
BENOBIO CO., LTD.
In Hyun LEE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INHIBITORS OF RECEPTOR INTERACTING PROTEIN KINASE I FOR THE TREATME...
Publication number
20250214942
Publication date
Jul 3, 2025
Board of Regents, The University of Texas System
Richard T. LEWIS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ERCC1-XPF COMPLEX INHIBITOR COMPOUNDS AND THE USE THEREOF IN THE TR...
Publication number
20250213584
Publication date
Jul 3, 2025
FUNDAÇÃO D. ANNA DE SOMMER CHAMPALIMAUD E DR. CARLOS MONTEZ CHAMPALIMAUD
Nuno José DE CASTILHO MONTEIRO GIL
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
T-TYPE CALCIUM CHANNEL MODULATORS COMPRISING AN AZASPIRONONANE CORE...
Publication number
20250214932
Publication date
Jul 3, 2025
PRAXIS PRECISION MEDICINES, INC.
Ricardo Lira
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INHIBITING MONOACYLGLYCEROL LIPASE (MAGL)
Publication number
20250214974
Publication date
Jul 3, 2025
Psy Therapeutics, Inc.
Jacob Matthew Hooker
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHODS AND PROCESSES FOR THE PREPARATION OF MCT4 INHIBITORS
Publication number
20250206723
Publication date
Jun 26, 2025
Vettore, LLC
Jon LAWSON
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
JAK1 PATHWAY INHIBITORS FOR THE TREATMENT OF PRURIGO NODULARIS
Publication number
20250195476
Publication date
Jun 19, 2025
INCYTE CORPORATION
Paul Smith
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CDK2 INHIBITOR AND PREPARATION METHOD AND USE THEREOF
Publication number
20250195475
Publication date
Jun 19, 2025
INVENTISBIO CO., LTD.
Yanxin YU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SMALL MOLECULE MODULATORS OF IL-17
Publication number
20250197378
Publication date
Jun 19, 2025
Leo Pharma A/S
Mark David ANDREWS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ACSS2 INHIBITORS AND METHODS OF USE THEREOF
Publication number
20250186433
Publication date
Jun 12, 2025
EpiVario, Inc.
Philippe NAKACHE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ORAL COMPLEMENT FACTOR D INHIBITORS
Publication number
20250186391
Publication date
Jun 12, 2025
BIOCRYST PHARMACEUTICALS, INC.
Pravin L. Kotian
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Biphenyl and Phenylpyridine Compounds
Publication number
20250188030
Publication date
Jun 12, 2025
Pfizer Inc.
Joyann Susan DONALDSON
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLE MEMBRANE-ASSOCIATED TYROSINE-AND THREONINE-SPECIFIC CDC2-I...
Publication number
20250188094
Publication date
Jun 12, 2025
INSILICO MEDICINE IP LIMITED
Xiao DING
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMBINATION TREATMENT FOR CANCER
Publication number
20250177352
Publication date
Jun 5, 2025
LAEKNA LIMITED
Chris LU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CRYSTALLINE FORM OF DAROLUTAMIDE
Publication number
20250179025
Publication date
Jun 5, 2025
QUÍMICA SINTÉTICA, S.A.
GIUSEPPE BARRECA
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF
Publication number
20250179013
Publication date
Jun 5, 2025
Accent Therapeutics, Inc.
Matthew H. Daniels
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CYCLOALKYL OR HETEROCYCLYL SUBSTITUTED HETEROARYL COMPOUND, AND COM...
Publication number
20250179027
Publication date
Jun 5, 2025
Shenzhen TargetRx, Inc.
Yihan Wang
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SALTS OF HETEROCYCLIC INHIBITORS OF MONOCARBOXYLATE TRANSPORTER 4 F...
Publication number
20250179049
Publication date
Jun 5, 2025
Vettore, LLC
Jon LAWSON
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ANTIBACTERIAL AGENTS
Publication number
20250179008
Publication date
Jun 5, 2025
TAXIS PHARMACEUTICALS, INC.
David Ryall Brown
A01 - AGRICULTURE FORESTRY ANIMAL HUSBANDRY HUNTING TRAPPING FISHING
Information
Patent Application
PYRAZOLYL COMPOUNDS AS KV7 CHANNEL ACTIVATORS
Publication number
20250171429
Publication date
May 29, 2025
BIOHAVEN THERAPEUTICS LTD.
Lynn RESNICK
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ALLOSTERIC STING MODULATORS AND METHODS OF USE
Publication number
20250170120
Publication date
May 29, 2025
The Board of Regents of the University of Texas System
Yong LU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
EMOPAMIL-BINDING PROTEIN INHIBITORS AND USES THEREOF
Publication number
20250171463
Publication date
May 29, 2025
Biogen MA Inc.
Martin Himmelbauer
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLYL COMPOUNDS AS KV7 CHANNEL ACTIVATORS
Publication number
20250171405
Publication date
May 29, 2025
BIOHAVEN THERAPEUTICS LTD.
Lynn RESNICK
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MONOACYLGLYCEROL LIPASE INHIBITORS AND USE THEREOF FOR THE TREATMEN...
Publication number
20250170100
Publication date
May 29, 2025
Psy Therapeutics, Inc.
Jacob Matthew Hooker
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLYL COMPOUNDS AS KV7 CHANNEL ACTIVATORS
Publication number
20250171430
Publication date
May 29, 2025
BIOHAVEN THERAPEUTICS LTD.
Lynn RESNICK
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MONOACYLGLYCEROL LIPASE INHIBITORS AND USE THEREOF FOR THE TREATMEN...
Publication number
20250170101
Publication date
May 29, 2025
Psy Therapeutics, Inc.
Jacob Matthew Hooker
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE