Pyrazines or piperazines forming part of bridged ring systems

Industry

CPC
A61K31/4995

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Parent Industries

AHUMAN NECESSITIES A61Medical science A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES A61K31/00Medicinal preparations containing organic active ingredients

Current Industry

A61K31/4995Pyrazines or piperazines forming part of bridged ring systems

Industries

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Patents Grantslast 30 patents

Information Patent Grant
Bile acid recycling inhibitors for treatment of hypercholemia and c...
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- Issue date Nov 19, 2024
- Shire Human Genetic Therapies, Inc.
- Bronislava Gedulin
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Information Patent Grant
Compositions comprising macrocycle derivatives incorporating bridge...
- Patent number 12,139,481
- Issue date Nov 12, 2024
- Southwestern Oklahoma State University
- Timothy J. Hubin
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Bicyclic heterocycles as FGFR inhibitors
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- Issue date Sep 10, 2024
- Incyte Corporation
- Oleg Vechorkin
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Substituted 1H-pyrazolo[4,3-c]pyridines and derivatives as EGFR inh...
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- Issue date Aug 20, 2024
- Boehringer Ingelheim International GmbH
- Harald Engelhardt
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Information Patent Grant
Methods of treatment
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- Issue date Jun 25, 2024
- BOW RIVER LLC
- Sundar Srinivasan
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors
- Patent number 11,998,545
- Issue date Jun 4, 2024
- Array Biopharma Inc.
- Steven W. Andrews
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Methods of treatment
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- Issue date May 7, 2024
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- Sundar Srinivasan
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Information Patent Grant
Methods for treating cholestasis
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- Issue date Mar 5, 2024
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- Thomas Jaecklin
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Information Patent Grant
Compositions and use of varenicline for treating dry eye
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- Issue date Feb 27, 2024
- Oyster Point Pharma, Inc.
- Douglas Michael Ackermann
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Information Patent Grant
Compositions and use of varenicline for treating dry eye
- Patent number 11,903,942
- Issue date Feb 20, 2024
- Oyster Point Pharma, Inc.
- Douglas Michael Ackermann
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Compositions and use of varenicline for treating dry eye
- Patent number 11,903,941
- Issue date Feb 20, 2024
- Oyster Point Pharma, Inc.
- Douglas Michael Ackermann
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Compositions and use of varenicline for treating dry eye
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- Issue date Feb 20, 2024
- Oyster Point Pharma, Inc.
- Douglas Michael Ackermann
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Information Patent Grant
Methods of treatment
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- Sundar Srinivasan
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Information Patent Grant
Methods of treating cancer
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Information Patent Grant
KDM1A inhibitors for the treatment of disease
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- Issue date Oct 3, 2023
- Imago Biosciences, Inc.
- Hugh Y. Rienhoff
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Information Patent Grant
Muscarinic acetylcholine M1 receptor antagonists
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- Issue date Sep 12, 2023
- Pipeline Therapeutics, Inc.
- Yifeng Xiong
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Methods of treatment
- Patent number 11,730,724
- Issue date Aug 22, 2023
- BOW RIVER LLC
- Sundar Srinivasan
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Halogenation of complex organic compounds
- Patent number 11,692,176
- Issue date Jul 4, 2023
- Regents of the University of Michigan
- David H. Sherman
- C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information Patent Grant
Aromatic heterocyclic compound, and pharmaceutical composition and...
- Patent number 11,679,108
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- GUANGZHOU HENOVCOM BIOSCIENCE CO., LTD.
- Jiancun Zhang
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Combinations of estrogen receptor degraders and cyclin-dependent ki...
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Information Patent Grant
Asymmetric bisaminoquinolines and bisaminoquinolines with varied li...
- Patent number 11,639,335
- Issue date May 2, 2023
- The Trustees of the University of Pennsylvania
- Ravi K. Amaravadi
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Bicyclic heterocycles as FGFR inhibitors
- Patent number 11,607,416
- Issue date Mar 21, 2023
- Incyte Corporation
- Oleg Vechorkin
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Combination therapy with an antitumor alkaloid
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- Issue date Feb 28, 2023
- Pharma Mar, S.A.
- Victoria Moneo Ocaña
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Information Patent Grant
Substituted pyridines and methods of use
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- Issue date Feb 28, 2023
- Theravance Biopharma R&D IP, LLC
- Christina Owens
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Methods for treating cholestasis
- Patent number 11,497,745
- Issue date Nov 15, 2022
- MIRUM PHARMACEUTICALS, INC.
- Thomas Jaecklin
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Chemokine CXCR4 receptor modulators and uses related thereto
- Patent number 11,497,744
- Issue date Nov 15, 2022
- Emory University
- Dennis Liotta
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Methods of treating lung cancer with CYP3A4 substrate drugs
- Patent number 11,491,152
- Issue date Nov 8, 2022
- BOW RIVER LLC
- Sundar Srinivasan
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Treatment of cancers having alterations within the SWI/SNF chromati...
- Patent number 11,433,068
- Issue date Sep 6, 2022
- The General Hospital Corporation
- David E. Fisher
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Methods of treatment
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- Issue date Aug 23, 2022
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- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Bile acid recycling inhibitors for treatment of pediatric cholestat...
- Patent number 11,376,251
- Issue date Jul 5, 2022
- Shire Human Genetic Therapies, Inc.
- Bronislava Gedulin
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE

Patents Applicationslast 30 patents

Information Patent Application
TRICYCLIC DERIVATIVE AND PREPARATION METHOD THEREFOR AND APPLICATIO...
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- Gang DENG
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Information Patent Application
5,6,7,8-TETRAHYDRO-2,6-NAPHTHYRIDINE DERIVATIVES AS CANCER THERAPEU...
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Substituted Pyrazolopyridines
- Publication number 20250051363
- Publication date Feb 13, 2025
- Neuro3 Therapeutics, Inc.
- Mark Seefeld
- C07 - ORGANIC CHEMISTRY
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SOS1 Inhibitor With Pyrido-Fused Six-Membered Ring Structure
- Publication number 20250042857
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- HAIHE BIOPHARMA CO., LTD.
- Dongsheng LI
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
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COMBINATION THERAPY FOR TREATMENT OF CANCER
- Publication number 20250041313
- Publication date Feb 6, 2025
- CITY OF HOPE
- Ravi Salgia
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
1,4-DIHETEROCYCLIC SUBSTITUTED AROMATIC RING OR AROMATIC HETEROCYCL...
- Publication number 20250034116
- Publication date Jan 30, 2025
- BeBetter Med Inc.
- Xiong CAI
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE PARP INHIBITOR AND USE...
- Publication number 20250034168
- Publication date Jan 30, 2025
- XIZANG HAISCO PHARMACEUTICAL CO., LTD.
- Yao LI
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
METHODS OF TREATMENT
- Publication number 20250032482
- Publication date Jan 30, 2025
- Bow River LLC
- Sundar SRINIVASAN
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
DIAZABICYCLOOCTANE DERIVATIVES USEFUL AS MATRIX METALLOPROTEINASE I...
- Publication number 20250026761
- Publication date Jan 23, 2025
- VASA THERAPEUTICS SPÓLKA Z OGRANICZONA ODPOWIEDZIALNOSCIA
- Benjamin Anthony Pratt
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
CBL-B INHIBITORS AND METHODS OF USE THEREOF
- Publication number 20250011318
- Publication date Jan 9, 2025
- ARCUS BIOSCIENCES, INC.
- Srikanth Kumar Gangam
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
6-SUBSTITUTED INDOLE COMPOUNDS
- Publication number 20250002471
- Publication date Jan 2, 2025
- GILEAD SCIENCES, INC.
- Stephen E. Ammann
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
Compounds for the Degradation of EGFR Kinase
- Publication number 20240425523
- Publication date Dec 26, 2024
- BEIGENE SWITZERLAND GMBH
- Huaqing Liu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
PARG INHIBITORY COMPOUNDS
- Publication number 20240425498
- Publication date Dec 26, 2024
- FORX THERAPEUTICS AG
- Ulrich Luecking
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
LURBINECTEDIN AND ATEZOLIZUMAB COMBINATIONS
- Publication number 20240415834
- Publication date Dec 19, 2024
- Pharma Mar, s.a.
- Luis Gonzaga Paz-Ares Rodriguez
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
COMPOUND FOR DEGRADATION OF BCL-2 FAMILY PROTEINS AND MEDICAL APPLI...
- Publication number 20240408085
- Publication date Dec 12, 2024
- XIZANG HAISCO PHARMACEUTICAL CO., LTD.
- Chen ZHANG
- C07 - ORGANIC CHEMISTRY
Information Patent Application
Methods of Treating Lymphedema
- Publication number 20240398793
- Publication date Dec 5, 2024
- CELLTAXIS, LLC
- Stanley Glenn ROCKSON
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
SYNTHESIS AND APPLICATION OF PHOSPHATASE DEGRADER
- Publication number 20240383908
- Publication date Nov 21, 2024
- HINOVA PHARMACEUTICALS INC.
- Lei FAN
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
GLUCAGON-LIKE PEPTIDE-1 RECEPTOR MODULATORS AND USES THEREOF
- Publication number 20240382471
- Publication date Nov 21, 2024
- Hepagene Therapeutics (HK) Limited
- Xiaodong Xu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
ANTI-VIRAL COMPOUNDS
- Publication number 20240383852
- Publication date Nov 21, 2024
- INFEX Therapeutics Limited
- James Kirkham
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
SUBSTITUTED TETRAHYDROFURAN-2-CARBOXAMIDES AS MODULATORS OF SODIUM...
- Publication number 20240368135
- Publication date Nov 7, 2024
- VERTEX PHARMACEUTICALS INCORPORATED
- Elizabeth Mary BECK
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
Macrocyclic Compounds Having ENT1 Inhibiting Activity
- Publication number 20240368183
- Publication date Nov 7, 2024
- ITEOS BELGIUM S.A.
- Michael Deligny
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
SUBSTITUTED 1H-PYRAZOLO[4,3-C]PYRIDINES AND DERIVATIVES AS EGFR INH...
- Publication number 20240358688
- Publication date Oct 31, 2024
- Boehringer Ingelheim International GmbH
- Harald ENGELHARDT
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
NOVEL PARP7 INHIBITOR AND USE THEREOF
- Publication number 20240351997
- Publication date Oct 24, 2024
- SHANGHAI QILU PHARMACEUTICAL RESEARCH AND DEVELOPMENT CENTRE LTD.
- Xiaoxia YAN
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
HALO-SUBSTITUTED AMINO PYRIDINE COMPOUNDS AS INHIBITORS OF THE HAEM...
- Publication number 20240343704
- Publication date Oct 17, 2024
- ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
- Anh Chau
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
ANALOGS FOR THE TREATMENT OF DISEASE
- Publication number 20240336611
- Publication date Oct 10, 2024
- Insilico Medicine IP Limited
- Aleksandrs ZAVORONKOVS
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
FACTOR XIIA INHIBITORS
- Publication number 20240327412
- Publication date Oct 3, 2024
- KALVISTA PHARMACEUTICALS LIMITED
- Rebecca Louise DAVIE
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
PYRAZOLYL DERIVATIVES AS INHIBITORS OF THE KRAS MUTANT PROTEIN
- Publication number 20240317721
- Publication date Sep 26, 2024
- Novartis AG
- Claudio BOMIO-CONFAGLIA
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
HYDROISOQUINOLINE OR HYDRONAPHTHYRIDINE COMPOUNDS FOR THE TREATMENT...
- Publication number 20240317735
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- Hoffmann-La Roche Inc.
- Fabian DEY
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
NOVEL MACROCYCLIC AMINOPYRAZOLE COMPOUNDS AS CDK2 INHIBITORS
- Publication number 20240317777
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- Accutar Biotechnology Inc.
- Xiangzhu Wang
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Information Patent Application
BROMODOMAIN INHIBITORS FOR CANCER THERAPY
- Publication number 20240316043
- Publication date Sep 26, 2024
- UNIVERSITY OF TENNESSEE RESEARCH FOUNDATION
- Duane Miller
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE

Pyrazines or piperazines forming part of bridged ring systems

Industry

Parent Industries

Current Industry

Patents Grantslast 30 patents

Bile acid recycling inhibitors for treatment of hypercholemia and c...

Compositions comprising macrocycle derivatives incorporating bridge...

Bicyclic heterocycles as FGFR inhibitors

Substituted 1H-pyrazolo[4,3-c]pyridines and derivatives as EGFR inh...

Methods of treatment

Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors

Methods of treatment

Methods for treating cholestasis

Compositions and use of varenicline for treating dry eye

Compositions and use of varenicline for treating dry eye

Compositions and use of varenicline for treating dry eye

Compositions and use of varenicline for treating dry eye

Methods of treatment

Methods of treating cancer

KDM1A inhibitors for the treatment of disease

Muscarinic acetylcholine M1 receptor antagonists

Methods of treatment

Halogenation of complex organic compounds

Aromatic heterocyclic compound, and pharmaceutical composition and...

Combinations of estrogen receptor degraders and cyclin-dependent ki...

Asymmetric bisaminoquinolines and bisaminoquinolines with varied li...

Bicyclic heterocycles as FGFR inhibitors

Combination therapy with an antitumor alkaloid

Substituted pyridines and methods of use

Methods for treating cholestasis

Chemokine CXCR4 receptor modulators and uses related thereto

Methods of treating lung cancer with CYP3A4 substrate drugs

Treatment of cancers having alterations within the SWI/SNF chromati...

Methods of treatment

Bile acid recycling inhibitors for treatment of pediatric cholestat...

Patents Applicationslast 30 patents

TRICYCLIC DERIVATIVE AND PREPARATION METHOD THEREFOR AND APPLICATIO...

5,6,7,8-TETRAHYDRO-2,6-NAPHTHYRIDINE DERIVATIVES AS CANCER THERAPEU...

Substituted Pyrazolopyridines

SOS1 Inhibitor With Pyrido-Fused Six-Membered Ring Structure

COMBINATION THERAPY FOR TREATMENT OF CANCER

1,4-DIHETEROCYCLIC SUBSTITUTED AROMATIC RING OR AROMATIC HETEROCYCL...

NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE PARP INHIBITOR AND USE...

METHODS OF TREATMENT

DIAZABICYCLOOCTANE DERIVATIVES USEFUL AS MATRIX METALLOPROTEINASE I...

CBL-B INHIBITORS AND METHODS OF USE THEREOF

6-SUBSTITUTED INDOLE COMPOUNDS

Compounds for the Degradation of EGFR Kinase

PARG INHIBITORY COMPOUNDS

LURBINECTEDIN AND ATEZOLIZUMAB COMBINATIONS

COMPOUND FOR DEGRADATION OF BCL-2 FAMILY PROTEINS AND MEDICAL APPLI...

Methods of Treating Lymphedema

SYNTHESIS AND APPLICATION OF PHOSPHATASE DEGRADER

GLUCAGON-LIKE PEPTIDE-1 RECEPTOR MODULATORS AND USES THEREOF

ANTI-VIRAL COMPOUNDS

SUBSTITUTED TETRAHYDROFURAN-2-CARBOXAMIDES AS MODULATORS OF SODIUM...

Macrocyclic Compounds Having ENT1 Inhibiting Activity

SUBSTITUTED 1H-PYRAZOLO[4,3-C]PYRIDINES AND DERIVATIVES AS EGFR INH...

NOVEL PARP7 INHIBITOR AND USE THEREOF

HALO-SUBSTITUTED AMINO PYRIDINE COMPOUNDS AS INHIBITORS OF THE HAEM...

ANALOGS FOR THE TREATMENT OF DISEASE

FACTOR XIIA INHIBITORS

PYRAZOLYL DERIVATIVES AS INHIBITORS OF THE KRAS MUTANT PROTEIN

HYDROISOQUINOLINE OR HYDRONAPHTHYRIDINE COMPOUNDS FOR THE TREATMENT...

NOVEL MACROCYCLIC AMINOPYRAZOLE COMPOUNDS AS CDK2 INHIBITORS

BROMODOMAIN INHIBITORS FOR CANCER THERAPY