Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems

Industry

CPC
A61K31/4985

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Parent Industries

AHUMAN NECESSITIES A61Medical science A61KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES A61K31/00Medicinal preparations containing organic active ingredients

Current Industry

A61K31/4985Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems

Industries

Patents Grantslast 30 patents

Information Patent Grant
BCL-2 inhibitors
- Patent number 12,220,419
- Issue date Feb 11, 2025
- Newave Pharmaceutical Inc.
- Yi Chen
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Pyrazino[1′,2′:1,5]pyrazolo[4,3-c] [2,6] naphthyridine compounds as...
- Patent number 12,215,107
- Issue date Feb 4, 2025
- KING FAISAL UNIVERSITY
- Christophe Tratrat
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Spirocyclic 2,3-dihydro-7-azaindole compounds and uses thereof
- Patent number 12,208,088
- Issue date Jan 28, 2025
- Genentech, Inc.
- Sushant Malhotra
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Anti-cancer nuclear hormone receptor-targeting compounds
- Patent number 12,208,141
- Issue date Jan 28, 2025
- NUVATION BIO INC.
- David Hung
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Combination therapies
- Patent number 12,208,099
- Issue date Jan 28, 2025
- MIRATI THERAPEUTICS, INC.
- Ruth Wei Aranda
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Substituted indole Mcl-1 inhibitors
- Patent number 12,195,472
- Issue date Jan 14, 2025
- Vanderbilt University
- Taekyu Lee
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Organic compounds
- Patent number 12,194,044
- Issue date Jan 14, 2025
- 1NTRA-CELLULAR THERAP1ES, 1NC.
- Wei Yao
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Five- and six-membered compound, and preparation method therefor an...
- Patent number 12,195,479
- Issue date Jan 14, 2025
- HANGZHOU POLYMED BIOPHARMACEUTICALS, INC.
- Jason Shaoyun Xiang
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Antiproliferative compounds and second active agents for combined use
- Patent number 12,186,311
- Issue date Jan 7, 2025
- Celgene Corporation
- Lilly L. Wong
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Liquid oral formulations for sildenafil
- Patent number 12,186,321
- Issue date Jan 7, 2025
- LIQMEDS WORLDWIDE LIMITED
- Jinal Pandya
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Imidazo[1,5-a]pyrido[4,3-e]pyrazines as CK2 inhibitors
- Patent number 12,187,726
- Issue date Jan 7, 2025
- KING FAISAL UNIVERSITY
- Christophe Tratrat
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Sleep improving agent
- Patent number 12,186,312
- Issue date Jan 7, 2025
- Amino Up Co., Ltd.
- Kazunori Goto
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Liquid oral formulations for tadalafil
- Patent number 12,186,322
- Issue date Jan 7, 2025
- LIQMEDS WORLDWIDE LIMITED
- Jinal Pandya
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Imidazopiperazine inhibitors of transcription activating proteins
- Patent number 12,186,324
- Issue date Jan 7, 2025
- Board of Regents, The University of Texas System
- Kang Le
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Regimens for treating HIV infections and aids
- Patent number 12,178,815
- Issue date Dec 31, 2024
- VIIV HEALTHCARE COMPANY
- Herta Crauwels
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Uses of DPP IV inhibitors
- Patent number 12,171,767
- Issue date Dec 24, 2024
- Boehringer Ingelheim International GmbH
- Klaus Dugi
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
PAPD5 inhibitors and methods of use thereof
- Patent number 12,171,755
- Issue date Dec 24, 2024
- Children's Medical Center Corporation
- Suneet Agarwal
- C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information Patent Grant
Treatment of a disease of the gastrointestinal tract with a JAK or...
- Patent number 12,171,764
- Issue date Dec 24, 2024
- BIORA THERAPEUTICS, INC.
- Mitchell Lawrence Jones
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Sulfoximine glycosidase inhibitors
- Patent number 12,157,734
- Issue date Dec 3, 2024
- Asceneuron SA
- Anna Quattropani
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Oral film formulation for modulating absorption profile
- Patent number 12,156,937
- Issue date Dec 3, 2024
- INTELGENX CORP.
- Nadine Paiement
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Process for preparing substituted pyrazolo[1,5-a]pyrazines
- Patent number 12,150,941
- Issue date Nov 26, 2024
- SUMITOMO PHARMA CO., LTD.
- Yohei Ikuma
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Compositions and methods
- Patent number 12,144,808
- Issue date Nov 19, 2024
- INTRA-CELLULAR THERAPIES, INC.
- Peng Li
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Substituted indole Mcl-1 inhibitors
- Patent number 12,144,816
- Issue date Nov 19, 2024
- Vanderbilt University
- Taekyu Lee
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Compositions comprising macrocycle derivatives incorporating bridge...
- Patent number 12,139,481
- Issue date Nov 12, 2024
- Southwestern Oklahoma State University
- Timothy J. Hubin
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Positive allosteric modulators of the muscarinic acetylcholine rece...
- Patent number 12,139,498
- Issue date Nov 12, 2024
- Vanderbilt University
- Craig W. Lindsley
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Pyrazolo[3,4-b]pyrazine SHP2 phosphatase inhibitors and methods of...
- Patent number 12,138,263
- Issue date Nov 12, 2024
- Relay Therapeutics, Inc.
- Alexander M. Taylor
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Pharmaceutical compositions
- Patent number 12,138,264
- Issue date Nov 12, 2024
- VIIV HEALTHCARE COMPANY
- Deepak B. Mundhra
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Diketopiperazine derivatives as calcium ATPase inhibitor for enhanc...
- Patent number 12,139,491
- Issue date Nov 12, 2024
- HOLOSMEDIC
- Ki Cheong Park
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Heating unit for use in a drug delivery device
- Patent number 12,138,383
- Issue date Nov 12, 2024
- Alexza Pharmaceuticals, Inc.
- Martin J. Wensley
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Treatment of erectile dysfunction and other indications
- Patent number 12,138,268
- Issue date Nov 12, 2024
- Strategic Science & Technologies, LLC
- Eric T. Fossel
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE

Patents Applicationslast 30 patents

Information Patent Application
POLYMORPH OF KRAS INHIBITOR, PREPARATION METHOD THEREFOR, AND USE T...
- Publication number 20250051333
- Publication date Feb 13, 2025
- GENFLEET THERAPEUTICS (SHANGHAI) INC.
- Fusheng ZHOU
- C07 - ORGANIC CHEMISTRY
Information Patent Application
TREATMENT OF NEUROLOGICAL DISORDERS
- Publication number 20250049790
- Publication date Feb 13, 2025
- PRAXIS PRECISION MEDICINES, INC.
- Michael Kristopher Mathieu Kahlig
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
PARP INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE...
- Publication number 20250051324
- Publication date Feb 13, 2025
- KEYTHERA (SUZHOU) BIO-PHARMACEUTICALS CO., LIMITED
- Yongqi DENG
- C07 - ORGANIC CHEMISTRY
Information Patent Application
METHODS OF TREATING ALOPECIA ARAETA
- Publication number 20250049789
- Publication date Feb 13, 2025
- ABBVIE INC.
- Andrea Chiricozzi
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
SOS1 Inhibitor With Pyrido-Fused Six-Membered Ring Structure
- Publication number 20250042857
- Publication date Feb 6, 2025
- HAIHE BIOPHARMA CO., LTD.
- Dongsheng LI
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
HETEROCYCLIC SUBSTITUTED 1,3,4-THIADIAZOLE AND PYRIDAZINE COMPOUNDS...
- Publication number 20250042879
- Publication date Feb 6, 2025
- Rgenta Therapeutics, Inc.
- Travis T. Wager
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
BRUTON'S TYROSINE KINASE INHIBITORS AS ANTIVIRAL AGENTS
- Publication number 20250041308
- Publication date Feb 6, 2025
- University of Florida Research Foundation, Incorporated
- Michael MCINTOSH
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
Combination Therapy Comprising A2A/A2B and PD-1/PD-L1 Inhibitors
- Publication number 20250041310
- Publication date Feb 6, 2025
- INCYTE CORPORATION
- Hui Wang
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
POLYMORPH FORMS OF A 5H-PYRROLO[2,3-b]PYRAZINE DERIVATIVE, METHODS...
- Publication number 20250042909
- Publication date Feb 6, 2025
- BeiGene, Ltd.
- Hui Chen
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
AN IGF1R INHIBITOR AND AN AKT INHIBITOR FOR USE IN THE TREATMENT OF...
- Publication number 20250041293
- Publication date Feb 6, 2025
- Genome Research Limited
- Elizabeth Coker
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
Synergistic compositions for use in the treatment of cancer
- Publication number 20250041294
- Publication date Feb 6, 2025
- Sartar Therapeutics Oy
- Harri Sihto
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
Compounds and Compositions as C-Kit Kinase Inhibitors
- Publication number 20250034138
- Publication date Jan 30, 2025
- Enanta Pharmaceuticals, Inc.
- Peilin XU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-...
- Publication number 20250034157
- Publication date Jan 30, 2025
- ABBVIE INC.
- Ayman Allian
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE PARP INHIBITOR AND USE...
- Publication number 20250034168
- Publication date Jan 30, 2025
- XIZANG HAISCO PHARMACEUTICAL CO., LTD.
- Yao LI
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES T...
- Publication number 20250034170
- Publication date Jan 30, 2025
- Vanqua Bio, Inc.
- Kevin Hunt
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
THERAPEUTIC TARGETS AND AGENTS FOR THE TREATMENT OF POSTTRAUMATIC S...
- Publication number 20250032484
- Publication date Jan 30, 2025
- The United States Government as Represented by the Department of Veterans Aff...
- Brian Shiner
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
APPLICATION OF IMIDAZO [1,2-A] PYRAZINE COMPOUNDS OR THEIR PHARMACE...
- Publication number 20250032485
- Publication date Jan 30, 2025
- GUANGZHOU MEDICAL UNIVERSITY
- XIYONG YU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
TREATMENT OF HIDRADENITIS WITH JAK INHIBITORS
- Publication number 20250032492
- Publication date Jan 30, 2025
- Pfizer Inc.
- Andrew FENSOME
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
WRN INHIBITORS
- Publication number 20250034136
- Publication date Jan 30, 2025
- Nimbus Wadjet, Inc.
- Derun Li
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
COMPOSITIONS AND METHODS FOR TREATING WITH A COMBINATION OF ALTERNA...
- Publication number 20250032788
- Publication date Jan 30, 2025
- Novocure GmbH
- Eyal Dor-On
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
REGULATING T CELL IMMUNE RESPONSE THROUGH IGF-I RECEPTOR (IGF-1R)
- Publication number 20250034264
- Publication date Jan 30, 2025
- The Regents of the University of Michigan
- Terry J. Smith
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
BTK INHIBITORS
- Publication number 20250034150
- Publication date Jan 30, 2025
- Biogen MA Inc.
- Brian T. Hopkins
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
METHODS FOR TREATING ALZHEIMER DISEASE AND FOR REDUCING AMYLOID BET...
- Publication number 20250025468
- Publication date Jan 23, 2025
- ARIBIO CO., LTD.
- Jai Jun Choung
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
TREATMENT OF NEURODEGENERATIVE DISEASES VIA ADMINISTRATION OF BUNTA...
- Publication number 20250025444
- Publication date Jan 23, 2025
- ANNOVIS BIO, INC.
- Maria Maccecchini
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
N-(5-SUBSTITUTED-[(1,3,4-THIADIAZOLYL) OR (THIAZOLYL)])(SUBSTITUTED...
- Publication number 20250026748
- Publication date Jan 23, 2025
- Repare Therapeutics Inc.
- Bingcan LIU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
COMPOUNDS AND METHODS FOR TREATING CORONA VIRUSES
- Publication number 20250025443
- Publication date Jan 23, 2025
- Clear Creek Bio, Inc.
- John K. DICKSON
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
PHARMACEUTICAL COMPOSITIONS
- Publication number 20250017924
- Publication date Jan 16, 2025
- ViiV Healthcare Company
- Deepak B. Mundhra
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
PHARMACEUTICAL COMPOSITIONS
- Publication number 20250017923
- Publication date Jan 16, 2025
- ViiV Healthcare Company
- Deepak B. Mundhra
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
PI3K-ALPHA INHIBITORS AND METHODS OF USE THEREOF
- Publication number 20250019380
- Publication date Jan 16, 2025
- Relay Therapeutics, Inc.
- Alessandro BOEZIO
- C07 - ORGANIC CHEMISTRY
Information Patent Application
Antiviral Therapy
- Publication number 20250017939
- Publication date Jan 16, 2025
- ViiV Healthcare Company
- Mark Richard Underwood
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE

Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems

Industry

Parent Industries

Current Industry

Patents Grantslast 30 patents

BCL-2 inhibitors

Pyrazino[1′,2′:1,5]pyrazolo[4,3-c] [2,6] naphthyridine compounds as...

Spirocyclic 2,3-dihydro-7-azaindole compounds and uses thereof

Anti-cancer nuclear hormone receptor-targeting compounds

Combination therapies

Substituted indole Mcl-1 inhibitors

Organic compounds

Five- and six-membered compound, and preparation method therefor an...

Antiproliferative compounds and second active agents for combined use

Liquid oral formulations for sildenafil

Imidazo[1,5-a]pyrido[4,3-e]pyrazines as CK2 inhibitors

Sleep improving agent

Liquid oral formulations for tadalafil

Imidazopiperazine inhibitors of transcription activating proteins

Regimens for treating HIV infections and aids

Uses of DPP IV inhibitors

PAPD5 inhibitors and methods of use thereof

Treatment of a disease of the gastrointestinal tract with a JAK or...

Sulfoximine glycosidase inhibitors

Oral film formulation for modulating absorption profile

Process for preparing substituted pyrazolo[1,5-a]pyrazines

Compositions and methods

Substituted indole Mcl-1 inhibitors

Compositions comprising macrocycle derivatives incorporating bridge...

Positive allosteric modulators of the muscarinic acetylcholine rece...

Pyrazolo[3,4-b]pyrazine SHP2 phosphatase inhibitors and methods of...

Pharmaceutical compositions

Diketopiperazine derivatives as calcium ATPase inhibitor for enhanc...

Heating unit for use in a drug delivery device

Treatment of erectile dysfunction and other indications

Patents Applicationslast 30 patents

POLYMORPH OF KRAS INHIBITOR, PREPARATION METHOD THEREFOR, AND USE T...

TREATMENT OF NEUROLOGICAL DISORDERS

PARP INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE...

METHODS OF TREATING ALOPECIA ARAETA

SOS1 Inhibitor With Pyrido-Fused Six-Membered Ring Structure

HETEROCYCLIC SUBSTITUTED 1,3,4-THIADIAZOLE AND PYRIDAZINE COMPOUNDS...

BRUTON'S TYROSINE KINASE INHIBITORS AS ANTIVIRAL AGENTS

Combination Therapy Comprising A2A/A2B and PD-1/PD-L1 Inhibitors

POLYMORPH FORMS OF A 5H-PYRROLO[2,3-b]PYRAZINE DERIVATIVE, METHODS...

AN IGF1R INHIBITOR AND AN AKT INHIBITOR FOR USE IN THE TREATMENT OF...

Synergistic compositions for use in the treatment of cancer

Compounds and Compositions as C-Kit Kinase Inhibitors

PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-...

NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE PARP INHIBITOR AND USE...

SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES T...

THERAPEUTIC TARGETS AND AGENTS FOR THE TREATMENT OF POSTTRAUMATIC S...

APPLICATION OF IMIDAZO [1,2-A] PYRAZINE COMPOUNDS OR THEIR PHARMACE...

TREATMENT OF HIDRADENITIS WITH JAK INHIBITORS

WRN INHIBITORS

COMPOSITIONS AND METHODS FOR TREATING WITH A COMBINATION OF ALTERNA...

REGULATING T CELL IMMUNE RESPONSE THROUGH IGF-I RECEPTOR (IGF-1R)

BTK INHIBITORS

METHODS FOR TREATING ALZHEIMER DISEASE AND FOR REDUCING AMYLOID BET...

TREATMENT OF NEURODEGENERATIVE DISEASES VIA ADMINISTRATION OF BUNTA...

N-(5-SUBSTITUTED-[(1,3,4-THIADIAZOLYL) OR (THIAZOLYL)])(SUBSTITUTED...

COMPOUNDS AND METHODS FOR TREATING CORONA VIRUSES

PHARMACEUTICAL COMPOSITIONS

PHARMACEUTICAL COMPOSITIONS

PI3K-ALPHA INHIBITORS AND METHODS OF USE THEREOF

Antiviral Therapy