Balakrishna, et al., “Inhibition of Hepatitis B Virus by a Novel L-Nucleoside, 2′-Fluoro-5-Methyl—L-arabinofuranosyl Uracil,” Antimicrobial Agents and Chemotherapy, Feb. 1996, pp. 380-356. |
Borthwick, et al., “Synthesis and Enzymatic Resolution of Carbocyclic 2′-Ara-fluoro-Guanosine: A Potent New Anti-Herpetic Agent,” J. Chem. Soc., Chem. Commun, 1988. |
Cheng, et al., Journal of Biological Chemistry, vol. 267(20), pp. 13938-13942 (1992). |
Chu, et al., “Use of 2′-Fluoro-5-methyl—L-arabinofuranosyluracil as a Novel Antiviral Agent for Hepatitis B Virus and Epstein-Barr Virus” Antimicrobial Agents and Chemotherapy, Apr. 1995 pp. 979-981. |
Furman, et al., “The Anti-Hepatitis B Virus Activities, Cytotoxicities, and Anabolic Profiles of the (−) and (+) Enantiomers of cis-5-Fluoro-I-[2-(Hydroxymethyl)-1,3-oxathiolane-5-yl]-Cytosine” Antimicrobial Agents and Chemotherapy, Dec. 1992, pp. 2686-2692. |
Martin, et al., “Synthesis and Antiviral Activity of Monofluoro and Difluoro Analogues of Pyrimidine Deoxyribonucleosides against Human Immunodeficiency Virus (HIV-1),” J. Med., Chem. 1990, 33, 2137-2145. |
Schinazi, et al, Mutations in retroviral genes associated with drug resistance, International Antiviral News, 1997. |
Schinazi, et al., “Selective Inhibition of Human Immunodeficiency viruses by Racemates and Enantiomers of cis-5-Fluoro-I-[2-(Hydroxymethyl)-1,3-Oxathiolane-5-yl]Cytosine” Antimicrobial Agents and Chemotherapy, Nov. 1992, pp. 2423-2431. |
Sterzycki, et al., “Synthesis and Anti-HIV Activity of Several 2′-Fluoro-Containing Pyrimidine Nucleosides,” J. Med. Chem. 1990. |
Su, T.S., et al., “Synthesis and Antiviral Effects of Several 1-(2-Deoxy-2-fluoro-B-D-arabinofuranosyl)-5-alkyluracils. Some Structure-Activity Relationships,” J. Med. Chem., 1986, 29, 151-154. |
Wantanabe, et al., “Synthesis and Anti-HIV Activity of 2′-“Up”-Fluoro Analogues of Active Anti-Aids Nucleosides 3′-Azido-3′-deoxythymidine (AZT) and 2′,3′-dideoxycytidine (DDC),” J. Med. Chem. 1990, 33, 2145-2150. |
Siddiqui MA et al., Tetrahed. Letters, vol. 39 No. 13 Mar. 26, 1998. |
Toyota, A., et al., Tetrahedron vol. 51, No. 32, pp. 8783-8798, 1995. |
Yoahimura, Y., et al., J. Org. Chem., 1999, 64, 7912-7920. |
Marquez, V.E., et al., Nucleosides & Nucleotides, 14(3-5), 555-558 (1995). |
Machida, H., et al., Antiviral Research, 39(1998) p. 129-137. |
Wantanabe, et al., “Synthesis and Anti-HIV Activity of 2'-“Up”-Fluoro Analogues of Active Anti-Aids Nucleosides 3'-Azido-3'-deoxythymidine (AZT) and 2',3'-dideoxycytidine (DDC),” J. Med. Chem. 1990, 33, 2145-2150. |