CA 121:255787, Hatano, 1994.* |
Lakhani, CA 109:149419, 1988.* |
Lakhani, CA 117:48192, 1991.* |
Vostrova, CA 91:193127, 1979.* |
Giardina et al., (1997) “Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 1. Identification of The 4-Quinolinecarboxamide Framework”, Journal of Medicinal Chemistry, vol. 40, pp. 1794-1807. |
Raveglia et al., (1997) “A Nobel Synthesis of 3-Halo-2-phenylquinoline-4-carboxylic Acids”, J. Heterocyclic Chem. vol. 34 pp. 557-559 . |
Giardina et al., (1998) “Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 2. Identification of (S)-N-(1-Phenylpropyl)-3-hydroxy-2-phenylquinoline-4-carboxamide (SB 223412)”, Journal of Medicinal Chemistry. |
Sarau et al., (1997) “Nonpeptide Tachykinin receptor Antagonists: I. Pharmacological and Pharmacokinetic Characterization of SB 223412, a Novel, Potent and Selective Neurkinin-3 Receptor Antagonist”, The Journal of pharmacology and Experimental Therapeutics, vol. 281, No. 3, pp. 1303-1311. |
Giardina et al., (1997) “Lead generation and lead optimization processes in the discovery of selective nonpeptide neurokinin receptor antagonists” Drugs of the Future, vol. 22, No. 11, 1235-1257. |
Giardinia et al. (1999) “Replacement of the quinoline system in 2-phenyl-4-quinolincarboxamide NK-3 receptor antagonists”, IL Farmaco, vol. 54, pp. 364-374. |
Raveglia et al., “Quinoline NK-3 Receptor Antagonists: Chemical Strategies to Prevent (æ-1) Metabolic Oxidation”, pp. 62, 1982. |
Giardina et al., “2-Pheny-4-quinolinecarboxamides: A Novel Class of Potent and Selective Non-Peptide Competitive Antagonists for the Human Neurokinin-3 Receptor”, Journal of Medicinal Chemistry, vol. 39, No. 12, pp. 2281-2284, 1993. |
Piero Savarino et al., “Assembled systems (X-azolopyridine)(quinoline). Bases and Salts.”, Journal of Heterocyclic Chemistry, vol. 29, 1992, pp. 185-192, XP002144891. |
Giardina et al., “Reliable And Efficient Synthesis of SR 142801”, Bioorg. Med. Chem. Lett., 6(19), (1996), 2307-2310. |