5[(pyrazol-4-yl)carbonyl]benzazolone as herbicide

Abstract

Pyrazolylbenzazolones of the formula I 1

Description

[0001] The present invention relates to 5-[(pyrazol-4-yl)carbonyl]-benzazolones (hereinbelow: benzazolones), to compositions comprising such compounds, and to the use of the benzazolones or of the compositions comprising them for controlling harmful plants.

[0002] WO 96/05197 discloses saccharin derivatives having herbicidal action which are substituted on the benzene ring of the saccharin skeleton by a (5-hydroxypyrazol-4-yl)carbonyl radical. WO 97/30993 and WO 97/09327 disclose dioxothiochromane derivatives and dihydrobenzothiophene derivatives having herbicidal action which likewise have a (5-hydroxypyrazol-4-yl)-carbonyl radical on the benzene ring of the sulfur heterocycle.

[0003] WO 97/08164 discloses, inter alia, benzo-fused derivatives of γ-butyrolactam having herbicidal action which likewise have a (5-hydroxypyrazol-4-yl)carbonyl radical.

[0004] JP 10130627 describes, inter alia, herbicides based on pyrazole derivatives of the formula (a) 2

[0005] in which R1 is C1-C4-alkyl or C2-C4-alkenyl, R2 is preferably hydrogen or methyl, Q is preferably hydrogen, n-propylsulfonyl, tolylsulfonyl or cyclohexylsulfonyl. X is C1-C4-(halo)alkyl, C2-C4-alkoxyalkyl, halogen, C1-C4-(halo)alkoxy. Z is O, SOr or NR3 where r=0 to 2, where R3 is hydrogen, C1-C4-(halo)alkyl, C1-C4-(halo)alkylsulfonyl or C1-C4-alkylcarbonyl. Y is oxygen or a substituent on the alkylene chain. D is a substituted or unsubstituted C1-C3-alkylene chain and p is an integer from 0 to 3. The variable m is an integer from zero to six, and n is an integer from zero to two.

[0006] However, the herbicidal properties of the compounds known from the publications mentioned and their compatibility with crop plants do not meet all of the criteria required from herbicides.

[0007] PCT/EP 00/04040 discloses 4-(3′,4′-heterocyclylbenzoyl)pyrazoles. Heterocyclic radicals mentioned are, inter alia, benzoxazolyl, benzimidazolyl, benzothiazolyl and benzotriazinyl. The compounds have herbicidal action.

[0008] It is an object of the present invention to provide novel compounds having herbicidal action which preferably have greater activity than the herbicidal substances of the prior art and/or better selectivity for harmful plants.

[0009] We have found that this object is achieved by 5-[(pyrazol-4-yl)-carbonyl]benzazolones of the formula I defined below.

[0010] Consequently, the present invention relates to pyrazolylcarbonyl-benzazolones of the formula I 3

[0011] in which A, R1, R2, R3 and Pz are as defined below:

[0012] A is O, S, SO, SO2 or NR6;

[0013] R1 is halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-hydroxyalkyl,

[0014] C1-C4-alkoxy-C1-C4-alkyl, C1-C4-haloalkoxy-C1-C4-alkyl,

[0015] C1-C4-haloalkylthio-C1-C4-alkyl, C1-C4-alkylthio-C1-C4-alkyl,

[0016] C1-C4-alkylsulfonyl-C1-C4-alkyl, C1-C4-haloalkylsulfonyl-C1-C4-alkyl, C1-C4-alkoxy, C1-C4-hydroxyalkoxy,

[0017] C1-C4-haloalkoxy, C1-C4-alkoxy-C1-C4-alkoxy, C1-C4-haloalkoxy-C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-haloalkylthio,

[0018] C1-C4-alkylsulfonyl, C1-C4-haloalkylsulfonyl;

[0019] R2 is hydrogen, hydroxyl, nitro, amino, C1-C6-alkylamino,

[0020] di(C1-C6-alkyl)amino, cyano, CHO, C1-C6-alkoxy, C1-C6-alkyl,

[0021] C1-C6-hydroxyalkyl, C1-C6-haloalkyl, C1-C6-alkoxy-C1-C6-alkyl,

[0022] C1-C6-haloalkoxy-C1-C6-alkyl, C2-C6-alkenyl, C2-C6-haloalkenyl,

[0023] C1-C6-haloalkoxy-C2-C6-alkenyl, C1-C6-alkoxy-C2-C6-alkenyl,

[0024] C2-C6-alkynyl, C2-C6-haloalkynyl, C1-C6-haloalkoxy-C2-C6-alkynyl, C1-C6-alkoxy-C2-C6-alkynyl, C1-C6-alkylsulfonyl,

[0025] C1-C6-haloalkylsulfonyl, (C1-C6-alkyl)carbonyl,

[0026] C1-C6-haloalkylcarbonyl, hydroxycarbonyl-C1-C4-alkyl,

[0027] C1-C6-alkoxycarbonyl-C1-C6-alkyl,

[0028] a radical of the formula C(O)OR4, CON(R5)2 or C(═NOR4a)R4b,

[0029] aryl, aryl-C1-C4-alkyl, arylsulfonyl, arylcarbonyl,

[0030] C3-C6-cycloalkyl, C3-C6-cycloalkenyl,

[0031] 3-, 4-, 5-, 6- or 7-membered heterocyclyl,

[0032] 3-, 4-, 5-, 6- or 7-membered heterocyclyl-C1-C6-alkyl,

[0033] where each aryl, cycloalkyl, cycloalkenyl and each heterocyclyl radical may be unsubstituted or may carry one, two, three or four substituents, in each case selected from the group consisting of halogen, C1-C4-haloalkyl, C1-C4-alkoxy and C1-C4-haloalkoxy;

[0034] R3 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy-C1-C4-alkyl, C1-C4-haloalkoxy-C1-C4-alkyl or halogen;

[0035] in which

[0036] R4 is C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy-C1-C6-alkyl, C1-C6-haloalkoxy-C1-C6-alkyl,

[0037] C2-C6-alkenyl, C2-C6-haloalkenyl, C1-C6-haloalkoxy-C2-C6-alkenyl, C1-C6-alkoxy-C2-C6-alkenyl,

[0038] C2-C6-alkynyl, C2-C6-haloalkynyl, C1-C6-haloalkoxy-C2-C6-alkynyl, C1-C6-alkoxy-C2-C6-alkynyl;

[0039] R4a, R4b independently of one another may have the meanings mentioned for R4, and R4b may be hydrogen;

[0040] R5 independently of one another are hydrogen,

[0041] C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy-C1-C6-alkyl, (C1-C6-haloalkoxy)-C1-C6-alkyl,

[0042] C2-C6-alkenyl, C2-C6-haloalkenyl, C1-C6-haloalkyl-C2-C6-alkenyl, C1-C6-haloalkoxy-C2-C6-alkenyl,

[0043] C1-C6-alkoxy-C2-C6-alkenyl, C2-C6-alkynyl,

[0044] C2-C6-haloalkynyl, C1-C6-haloalkyl-C2-C6-alkynyl,

[0045] C1-C6-haloalkoxy-C2-C6-alkynyl, C1-C6-alkoxy-C2-C6-alkynyl, or together form a 3- to 7-membered heterocycle which may be partially or fully halogenated and/or may carry one, two or three substituents selected from the group consisting of

[0046] C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy,

[0047] C1-C6-haloalkoxy;

[0048] R6 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-halo-alkoxy-C1-C4-alkyl, C1-C4-alkoxy-C1-C4-alkyl; and

[0049] Pz is a radical of the formula IIa or IIb, 4

[0050] in which the variables R7, R8 and R9 are as defined below:

[0051] R7 is hydroxyl, mercapto, halogen, OR10, SR10, SOR11, SO2R11,

[0052] OSO2R11, P(O)R12R13, OP(O)R12R13, P(S)R12R13, OP(S)R12R13,

[0053] NR14R15, ONR14R15 or N-bonded heterocyclyl which may be partially or fully halogenated and/or may carry one, two or three of the following radicals: nitro, cyano, C1-C4-alkyl,

[0054] C1-C4-haloalkyl, C1-C4-alkoxy or C1-C4-haloalkoxy;

[0055] R8 is hydrogen, C1-C6-alkyl, C3-C6-cycloalkyl, C1-C6-haloalkyl,

[0056] hydroxyl, C1-C6-alkoxy or C1-C6-haloalkoxy;

[0057] R9 is hydrogen, halogen, C1-C6-alkyl, C3-C6-cycloalkyl,

[0058] C1-C6-haloalkyl, hydroxyl, C1-C6-alkoxy, C1-C6-haloalkoxy,

[0059] C1-C6-alkylthio or C1-C6-haloalkylthio;

[0060] where

[0061] R10 is C1-C6-alkyl, C3-C6-alkenyl, C3-C6-haloalkenyl,

[0062] C3-C6-alkynyl, C3-C6-haloalkynyl, C3-C6-cycloalkyl,

[0063] C1-C6-alkylcarbonyl, C2-C6-alkenylcarbonyl,

[0064] C2-C6-alkynylcarbonyl, C3-C6-cycloalkylcarbonyl,

[0065] C1-C6-alkoxycarbonyl, C3-C6-alkenyloxycarbonyl,

[0066] C3-C6-alkynyloxycarbonyl, C1-C6-alkylthiocarbonyl,

[0067] C1-C6-alkylaminocarbonyl, C3-C6-alkenylaminocarbonyl,

[0068] C3-C6-alkynylaminocarbonyl, N,N-di(C1-C6-alkyl)amino-carbonyl, N—(C3-C6-alkenyl)-N—(C1-C6-alkyl)amino-carbonyl, N—(C3-C6-alkynyl)-N—(C1-C6-alkyl)amino-carbonyl, N—(C1-C6-alkoxy)-N—(C1-C6-alkyl)amino-carbonyl, N—(C3-C6-alkenyl)-N—(C1-C6-alkoxy)amino-carbonyl, N—(C3-C6-alkynyl)-N—(C1-C6-alkoxy)amino-carbonyl, di(C1-C6-alkyl)aminothiocarbonyl or

[0069] C1-C6-alkoxyimino-C1-C6-alkyl, where the alkyl, cycloalkyl and alkoxy radicals mentioned may be partially or fully halogenated and/or may carry one, two or three of the following groups: cyano,

[0070] C1-C4-alkoxy, C1-C4-alkylthio, di(C1-C4-alkyl)amino,

[0071] C1-C4-alkylcarbonyl, C1-C4-alkoxycarbonyl,

[0072] C1-C4-alkoxy-C1-C4-alkoxycarbonyl,

[0073] C1-C4-alkylaminocarbonyl, di(C1-C4-alkyl)-aminocarbonyl, aminocarbonyl, C1-C4-alkylcarbonyloxy or C3-C6-cycloalkyl;

[0074] is phenyl, phenyl-C1-C6-alkyl, phenylcarbonyl-C1-C6-alkyl, phenylcarbonyl, phenoxycarbonyl,

[0075] phenyloxythiocarbonyl, phenylaminocarbonyl,

[0076] N—(C1-C6-alkyl)-N-(phenyl)aminocarbonyl, phenyl-C2-C6-alkenylcarbonyl, heterocyclyl, heterocyclyl-C1-C6-alkyl, heterocyclylcarbonyl-C1-C6-alkyl,

[0077] heterocyclylcarbonyl, heterocyclyloxycarbonyl,

[0078] heterocyclyloxythiocarbonyl, heterocyclylaminocarbonyl, N—(C1-C6-alkyl)-N-(heterocyclyl)aminocarbonyl, or heterocyclyl-C2-C6-alkenylcarbonyl,

[0079] where the phenyl and the heterocyclyl radical of the 18 lastmentioned substituents may be partially or fully halogenated and/or may carry one, two or three of the following radicals: nitro, cyano, C1-C4-alkyl,

[0080] C1-C4-haloalkyl, C1-C4-alkoxy or C1-C4-haloalkoxy;

[0081] R11 is C1-C6-alkyl, C3-C6-alkenyl, C3-C6-alkynyl or C3-C6-cycloalkyl, where the four radicals mentioned may be partially or fully halogenated and/or may carry one, two or three of the following groups:

[0082] cyano, C1-C4-alkoxy, C1-C4-haloalkoxy,

[0083] C1-C4-alkylthio, C1-C4-haloalkylthio,

[0084] C1-C4-alkylcarbonyl, C1-C4-alkoxycarbonyl or C1-C4-haloalkoxycarbonyl;

[0085] is phenyl, phenyl-C1-C6-alkyl, heterocyclyl or heterocyclyl-C1-C6-alkyl, where the phenyl and the heterocyclyl radical of the lastmentioned substituents may be partially or fully halogenated and/or may carry one, two or three of the following radicals: nitro, cyano, C1-C4-alkyl, C1-C4-haloalkyl,

[0086] C1-C4-alkoxy, C1-C4-haloalkoxy or

[0087] C1-C4-alkoxycarbonyl;

[0088] R12, R13 independently of one another are hydrogen, hydroxyl,

[0089] C1-C6-alkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenyl-C1-C4-alkyl or phenoxy, where the three lastmentioned substituents may be partially or fully halogenated and/or may carry one, two or three of the following radicals: nitro, cyano, C1-C4-alkyl,

[0090] C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy or

[0091] C1-C4-alkoxycarbonyl;

[0092] R14 is hydrogen, C1-C6-alkyl, C3-C6-alkenyl,

[0093] C3-C6-haloalkenyl, C3-C6-alkynyl, C3-C6-haloalkynyl,

[0094] C3-C6-cycloalkyl, C1-C6-alkylcarbonyl, hydroxyl,

[0095] C1-C6-alkoxy, C3-C6-alkenyloxy, C3-C6-alkynyloxy,

[0096] amino, C1-C6-alkylamino, di(C1-C6-alkyl)amino or C1-C6-alkylcarbonylamino, where the alkyl, cycloalkyl and alkoxy radicals mentioned may be partially or fully halogenated and/or may carry one, two or three of the following radicals: cyano, C1-C4-alkoxycarbonyl, C1-C4-alkylaminocarbonyl, di(C1-C4-alkyl)-aminocarbonyl or C3-C6-cycloalkyl;

[0097] is phenyl, phenyl-C1-C4-alkyl, phenylcarbonyl,

[0098] heterocyclyl, heterocyclyl-C1-C4-alkyl or

[0099] heterocyclylcarbonyl, where the phenyl or

[0100] heterocyclyl radical of the six lastmentioned substituents may be partially or fully halogenated and/or may carry one, two or three of the following radicals: nitro, cyano, C1-C4-alkyl, C1-C4-haloalkyl,

[0101] C1-C4-alkoxy or C1-C4-haloalkoxy; and

[0102] R15 is hydrogen, C1-C6-alkyl or C3-C6-alkenyl,

[0103] C3-C6-alkynyl;

[0104] and their agriculturally useful salts.

[0105] Furthermore we have found herbicidal compositions which comprise the pyrazolyl derivatives of the formula I and have very good herbicidal action. Moreover, we have found methods for controlling undesirable vegetation using the pyrazolyl derivatives of the formula I.

[0106] Depending on the substitution pattern, the compounds of the formula I may contain one or more chiral centers, in which case they are present as enantiomers or diasteromer mixtures. The invention provides both the pure enantiomers or diastereomers and their mixtures.

[0107] The compounds of the formula I may also be present in the form of their agriculturally useful salts, the type of salt generally being immaterial. In general, the salts of those cations and the acid addition salts of those acids are suitable whose cations and anions, respectively, do not negatively affect the herbicidal action of the compounds I.

[0108] Suitable cations are, in particular, ions of the alkali metals, preferably lithium, sodium and potassium, of the alkaline earth metals, preferably calcium and magnesium, and of the transition metals, preferably manganese, copper, zinc and iron, and also ammonium, where, if desired, one to four hydrogen atoms may be replaced by C1-C4-alkyl, hydroxy-C1-C4-alkyl, C1-C4-alkoxy-C1-C4-alkyl, hydroxy-C1-C4-alkoxy-C1-C4-alkyl, phenyl or benzyl, preferably ammonium, dimethylammonium, diisopropylammonium, tetramethylammonium, tetrabutylammonium, 2-(2-hydroxyeth-1-oxy)-eth-1-ylammonium, di(2-hydroxyeth-1-yl)ammonium, trimethylbenzylammonium, furthermore phosphonium ions, sulfonium ions, preferably tri(C1-C4-alkyl)sulfonium, and sulfoxonium ions, preferably tri(C1-C4-alkyl)sulfoxonium.

[0109] Anions of useful acid addition salts are primarily chloride, bromide, fluoride, hydrogen sulfate, sulfate, dihydrogen phosphate, hydrogen phosphate, nitrate, bicarbonate, carbonate, hexafluorosilicate, hexafluorophosphate, benzoate and the anions of C1-C4-alkanoic acids, preferably formate, acetate, propionate and butyrate.

[0110] For R7=hydroxyl or mercapto {Z=O,S}, IIa also represents the tautomeric forms IIa′ and IIa″ 5

[0111] and IIb also represents the tautomeric forms IIb′ and IIb″ 6

[0112] The organic molecular moieties mentioned for the substituents R1 to R15 or as radicals on phenyl and heterocyclyl radicals are collective terms for individual enumerations of the particular group members. All hydrocarbon chains, i.e. all alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, N-alkylamino, N,N-dialkylamino, N-haloalkylamino, N-alkoxyamino, N-alkoxy-N-alkylamino, N-alkylcarbonylamino, alkylcarbonyl, haloalkylcarbonyl, alkoxycarbonyl, haloalkoxycarbonyl, alkylthiocarbonyl, alkylcarbonyloxy, alkylaminocarbonyl, dialkylaminocarbonyl, dialkylaminothiocarbonyl, alkoxyalkyl, hydroxyalkoxyalkyl, alkoxyiminoalkyl, phenylalkylcarbonyl, heterocyclylalkylcarbonyl, phenylalkenylcarbonyl, heterocyclylalkenylcarbonyl, N-alkoxy-N-alkylaminocarbonyl, N-alkyl-N-phenylaminocarbonyl, N-alkyl-N-heterocyclylaminocarbonyl, phenylalkyl, heterocyclylalkyl, phenylcarbonylalkyl, heterocyclylcarbonyl-alkyl, alkoxyalkoxycarbonyl, alkenylcarbonyl, alkenyloxycarbonyl, alkenylaminocarbonyl, N-alkenyl-N-alkylaminocarbonyl, N-alkenyl-N-alkoxyaminocarbonyl, alkynylcarbonyl, alkynyloxycarbonyl, alkynylaminocarbonyl, N-alkynyl-N-alkylaminocarbonyl, N-alkynyl-N-alkoxyaminocarbonyl, alkenyl, alkynyl, haloalkenyl, haloalkynyl, alkenyloxy, alkynyloxy, alkanediyl, alkenediyl, alkadienediyl or alkynediyl moieties can be straight-chain or branched. Unless indicated otherwise, halogenated substituents preferably carry one to five identical or different halogen atoms. The expression halogen represents in each case fluorine, chlorine, bromine or iodine.

[0113] Examples of other meanings are:

[0114] C1-C4-alkyl: for example methyl, ethyl, propyl, 1-methylethyl,

[0115] butyl, 1-methylpropyl, 2-methylpropyl or 1,1-dimethylethyl;

[0116] C1-C4-haloalkyl: a C1-C4-alkyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example,

[0117] chloromethyl, dichloromethyl, trichloromethyl, fluoromethyl,

[0118] difluoromethyl, trifluoromethyl, chlorofluoromethyl,

[0119] dichlorofluoromethyl, chlorodifluoromethyl, 2-fluoroethyl,

[0120] 2-chloroethyl, 2-bromoethyl, 2-iodoethyl, 2,2-difluoroethyl,

[0121] 2,2,2-trifluoroethyl, 2-chloro-2-fluoroethyl,

[0122] 2-chloro-2,2-difluoroethyl, 2,2-dichloro-2-fluoroethyl,

[0123] 2,2,2-trichloroethyl, pentafluoroethyl, 2-fluoropropyl,

[0124] 3-fluoropropyl, 2,2-difluoropropyl, 2,3-difluoropropyl,

[0125] 2-chloropropyl, 3-chloropropyl, 2,3-dichloropropyl,

[0126] 2-bromopropyl, 3-bromopropyl, 3,3,3-trifluoropropyl,

[0127] 3,3,3-trichloropropyl, 2,2,3,3,3-pentafluoropropyl,

[0128] heptafluoropropyl, 1-(fluoromethyl)-2-fluoroethyl,

[0129] 1-(chloromethyl)-2-chloroethyl, 1-(bromomethyl)-2-bromoethyl,

[0130] 4-fluorobutyl, 4-chlorobutyl, 4-bromobutyl or

[0131] nonafluorobutyl;

[0132] C1-C6-alkyl, and the alkyl moieties of C1-C6-alkylamino,

[0133] di(C1-C6-alkyl)amino, N—(C1-C6-alkoxy)-N—(C1-C6-alkyl)aminocarbonyl, N—(C3-C6-alkenyl)-N—(C1-C6-alkyl)-aminocarbonyl,

[0134] (C3-C6-alkynyl)-N—(C1-C6-alkyl)aminocarbonyl, N—(C1-C6-alkyl)-N-phenylaminocarbonyl, and also N—(C1-C6-alkyl)-N-heterocyclylamino-carbonyl: C1-C4-alkyl as mentioned above,

[0135] and also, for example, n-pentyl, 1-methylbutyl,

[0136] 2-methylbutyl, 3-methylbutyl, 2,2-dimethylpropyl,

[0137] 1-ethylpropyl, hexyl, 1,1-dimethylpropyl, 1,2-dimethylpropyl,

[0138] 1-methylpentyl, 2-methylpentyl, 3-methylpentyl,

[0139] 4-methylpentyl, 1,1-dimethylbutyl, 1,2-dimethylbutyl,

[0140] 1,3-dimethylbutyl, 2,2-dimethylbutyl, 2,3-dimethylbutyl,

[0141] 3,3-dimethylbutyl, 1-ethylbutyl, 2-ethylbutyl,

[0142] 1,1,2-trimethylpropyl, 1-ethyl-1-methylpropyl or

[0143] 1-ethyl-3-methylpropyl;

[0144] C1-C6-haloalkyl, and the haloalkyl moieties of

[0145] N—C1-C6-haloalkylamino: C1-C4-haloalkyl, as mentioned above,

[0146] and also, for example, 5-fluoropentyl, 5-chloropentyl,

[0147] 5-bromopentyl, 5-iodopentyl, undecafluoropentyl,

[0148] 6-fluorohexyl, 6-chlorohexyl, 6-bromohexyl, 6-iodohexyl or

[0149] dodecafluorohexyl;

[0150] C1-C4-alkoxy and the alkoxy moieties of hydroxy-C1-C4-alkoxy-C1-C4-alkyl, C1-C4-alkoxy-C1-C4-alkoxycarbonyl: for example

[0151] methoxy, ethoxy, propoxy, 1-methylethoxy, butoxy,

[0152] 1-methylpropoxy, 2-methylpropoxy or 1,1-dimethylethoxy;

[0153] C1-C6-alkoxy, and the alkoxy moieties of

[0154] C1-C6-alkoxy-C3-C6-alkenyl, C1-C6-alkoxy-C3-C6-alkynyl,

[0155] C1-C6-alkoxy-C2-C6-alkenyl, C1-C6-alkoxy-C2-C6-alkynyl,

[0156] N—C1-C6-alkoxyamino, N—(C1-C6-alkoxy)-N—(C1-C6-alkyl)amino,

[0157] C1-C6-alkoxyimino-C1-C6-alkyl, (C1-C6-alkoxy) (C1-C6-alkylthio)methyl, N—(C1-C6-alkoxy)-N—(C1-C6-alkyl)aminocarbonyl,

[0158] N—(C3-C6-alkenyl)-N—(C1-C6-alkoxy)aminocarbonyl and

[0159] N—(C3-C6-alkynyl)-N—(C1-C6-alkoxy)aminocarbonyl: C1-C4-alkoxy as mentioned above, and also, for example, pentoxy,

[0160] 1-methylbutoxy, 2-methylbutoxy, 3-methylbutoxy, 1,1-dimethylpropoxy, 1,2-dimethylpropoxy, 2,2-dimethylpropoxy,

[0161] 1-ethylpropoxy, hexoxy, 1-methylpentoxy, 2-methylpentoxy,

[0162] 3-methylpentoxy, 4-methylpentoxy, 1,1-dimethylbutoxy,

[0163] 1,2-dimethylbutoxy, 1,3-dimethylbutoxy, 2,2-dimethylbutoxy,

[0164] 2,3-dimethylbutoxy, 3,3-dimethylbutoxy, 1-ethylbutoxy,

[0165] 2-ethylbutoxy, 1,1,2-trimethylpropoxy,

[0166] 1,2,2-trimethylpropoxy, 1-ethyl-1-methylpropoxy or

[0167] 1-ethyl-2-methylpropoxy;

[0168] C1-C4-haloalkoxy and the haloalkoxy moieties of

[0169] C1-C4-haloalkoxy-C1-C4-alkyl, C1-C4-haloalkoxy-C1-C4-alkoxy,

[0170] C1-C4-haloalkoxy-C1-C6-alkyl, C1-C4-haloalkoxy-C1-C6-alkoxy,

[0171] C1-C4-haloalkoxy-C3-C6-alkenyl, C1-C4-haloalkoxy-C3-C6-alkynyl: a

[0172] C1-C4-alkoxy radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example, fluoromethoxy, difluoromethoxy,

[0173] trifluoromethoxy, chlorodifluoromethoxy, bromodifluoromethoxy, 2-fluoroethoxy, 2-chloroethoxy, 2-bromomethoxy,

[0174] 2-iodoethoxy, 2,2-difluoroethoxy, 2,2,2-trifluoroethoxy,

[0175] 2-chloro-2-fluoroethoxy, 2-chloro-2,2-difluoroethoxy,

[0176] 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy,

[0177] pentafluoroethoxy, 2-fluoropropoxy, 3-fluoropropoxy,

[0178] 2-chloropropoxy, 3-chloropropoxy, 2-bromopropoxy,

[0179] 3-bromopropoxy, 2,2-difluoropropoxy, 2,3-difluoropropoxy,

[0180] 2,3-dichloropropoxy, 3,3,3-trifluoropropoxy, 3,3,3-trichloro-propoxy, 2,2,3,3,3-pentafluoropropoxy, heptafluoropropoxy,

[0181] 1-(fluoromethyl)-2-fluoroethoxy, 1-(chloromethyl)-2-chloro-ethoxy, 1-(bromomethyl)-2-bromoethoxy, 4-fluorobutoxy,

[0182] 4-chlorobutoxy, 4-bromobutoxy or nonafluorobutoxy;

[0183] C1-C6-haloalkoxy: C1-C4-haloalkoxy as mentioned above, and also, for example, 5-fluoropentoxy, 5-chloropentoxy,

[0184] 5-bromopentoxy, 5-iodopentoxy, undecafluoropentoxy,

[0185] 6-fluorohexoxy, 6-chlorohexoxy, 6-bromohexoxy, 6-iodohexoxy

[0186] or dodecafluorohexoxy;

[0187] C1-C4-alkylthio (C1-C4-alkylsulfanyl: C1-C4-alkyl-S—): for example methylthio, ethylthio, propylthio, 1-methylethylthio,

[0188] butylthio, 1-methylpropylthio, 2-methylpropylthio or

[0189] 1,1-dimethylethylthio;

[0190] C1-C6-alkylthio, and the alkylthio moieties of

[0191] C1-C6-alkylthiocarbonyl: C1-C4-alkylthio as mentioned above, and also, for example, pentylthio, 1-methylbutylthio,

[0192] 2-methylbutylthio, 3-methylbutylthio, 2,2-dimethylpropylthio,

[0193] 1-ethylpropylthio, hexylthio, 1,1-dimethylpropylthio,

[0194] 1,2-dimethylpropylthio, 1-methylpentylthio,

[0195] 2-methylpentylthio, 3-methylpentylthio, 4-methylpentylthio,

[0196] 1,1-dimethylbutylthio, 1,2-dimethylbutylthio,

[0197] 1,3-dimethylbutylthio, 2,2-dimethylbutylthio,

[0198] 2,3-dimethylbutylthio, 3,3-dimethylbutylthio,

[0199] 1-ethylbutylthio, 2-ethylbutylthio, 1,1,2-trimethyl-propylthio, 1,2,2-trimethylpropylthio, 1-ethyl-1-methyl-propylthio or 1-ethyl-2-methylpropylthio;

[0200] C1-C4-haloalkylthio and the haloalkylthio moieties of

[0201] C1-C4-haloalkylthio-C1-C4-alkyl: a C1-C4-alkylthio radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example,

[0202] fluoromethylthio, difluoromethylthio, trifluoromethylthio,

[0203] chlorodifluoromethylthio, bromodifluoromethylthio,

[0204] 2-fluoroethylthio, 2-chloroethylthio, 2-bromoethylthio,

[0205] 2-iodoethylthio, 2,2-difluoroethylthio, 2,2,2-trifluoroethylthio, 2,2,2-trichloroethylthio, 2-chloro-2-fluoroethylthio, 2-chloro-2,2-difluoroethylthio, 2,2-dichloro2-fluoroethylthio, pentafluoroethylthio, 2-fluoropropylthio,

[0206] 3-fluoropropylthio, 2-chloropropylthio, 3-chloropropylthio,

[0207] 2-bromopropylthio, 3-bromopropylthio, 2,2-difluoropropylthio,

[0208] 2,3-difluoropropylthio, 2,3-dichloropropylthio,

[0209] 3,3,3-trifluoropropylthio, 3,3,3-trichloropropylthio,

[0210] 2,2,3,3,3-pentafluoropropylthio, heptafluoropropylthio,

[0211] 1-(fluoromethyl)-2-fluoroethylthio, 1-(chloromethyl)-2-chloroethylthio, 1-(bromomethyl)-2-bromoethylthio,

[0212] 4-fluorobutylthio, 4-chlorobutylthio, 4-bromobutylthio or nonafluorobutylthio;

[0213] C1-C6-haloalkylthio: C1-C4-haloalkylthio as mentioned above,

[0214] and also 5-fluoropentylthio, 5-chloropentylthio,

[0215] 5-bromopentylthio, 5-iodopentylthio, undecafluoropentylthio,

[0216] 6-fluorohexylthio, 6-chlorohexylthio, 6-bromohexylthio,

[0217] 6-iodohexylthio or dodecafluorohexylthio;

[0218] C1-C4-alkylsulfinyl (C1-C4-alkyl-S(═O)—): for example,

[0219] methylsulfinyl, ethylsulfinyl, propylsulfinyl,

[0220] 1-methylethylsulfinyl, butylsulfinyl, 1-methylpropylsulfinyl,

[0221] 2-methylpropylsulfinyl or 1,1-dimethylethylsulfinyl;

[0222] C1-C6-alkylsulfinyl: C1-C4-alkylsulfinyl as mentioned above,

[0223] and also pentylsulfinyl, 1-methylbutylsulfinyl,

[0224] 2-methylbutylsulfinyl, 3-methylbutylsulfinyl,

[0225] 2,2-dimethylpropylsulfinyl, 1-ethylpropylsulfinyl,

[0226] 1,1-dimethylpropylsulfinyl, 1,2-dimethylpropylsulfinyl,

[0227] hexylsulfinyl, 1-methylpentylsulfinyl, 2-methylpentyl-sulfinyl, 3-methylpentylsulfinyl, 4-methylpentylsulfinyl,

[0228] 1,1-dimethylbutylsulfinyl, 1,2-dimethylbutylsulfinyl,

[0229] 1,3-dimethylbutylsulfinyl, 2,2-dimethylbutylsulfinyl,

[0230] 2,3-dimethylbutylsulfinyl, 3,3-dimethylbutylsulfinyl,

[0231] 1-ethylbutylsulfinyl, 2-ethylbutylsulfinyl,

[0232] 1,1,2-trimethylpropylsulfinyl, 1,2,2-trimethylpropylsulfinyl,

[0233] 1-ethyl-1-methylpropylsulfinyl or

[0234] 1-ethyl-2-methylpropylsulfinyl;

[0235] C1-C4-haloalkylsulfinyl: a C1-C4-alkylsulfinyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example,

[0236] fluoromethylsulfinyl, difluoromethylsulfinyl,

[0237] trifluoromethylsulfinyl, chlorodifluoromethylsulfinyl,

[0238] bromodifluoromethylsulfinyl, 2-fluoroethylsulfinyl,

[0239] 2-chloroethylsulfinyl, 2-bromoethylsulfinyl,

[0240] 2-iodoethylsulfinyl, 2,2-difluoroethylsulfinyl,

[0241] 2,2,2-trifluoroethylsulfinyl, 2,2,2-trichloroethylsulfinyl,

[0242] 2-chloro-2-fluoroethylsulfinyl, 2-chloro-2,2-difluoro-ethylsulfinyl, 2,2-dichloro-2-fluoroethylsulfinyl,

[0243] pentafluoroethylsulfinyl, 2-fluoropropylsulfinyl,

[0244] 3-fluoropropylsulfinyl, 2-chloropropylsulfinyl,

[0245] 3-chloropropylsulfinyl, 2-bromopropylsulfinyl,

[0246] 3-bromopropylsulfinyl, 2,2-difluoropropylsulfinyl,

[0247] 2,3-difluoropropylsulfinyl, 2,3-dichloropropylsulfinyl,

[0248] 3,3,3-trifluoropropylsulfinyl, 3,3,3-trichloropropylsulfinyl,

[0249] 2,2,3,3,3-pentafluoropropylsulfinyl, heptafluoropropyl-sulfinyl, 1-(fluoromethyl)-2-fluoroethylsulfinyl,

[0250] 1-(chloromethyl)-2-chloroethylsulfinyl, 1-(bromomethyl)-2-bromoethylsulfinyl, 4-fluorobutylsulfinyl,

[0251] 4-chlorobutylsulfinyl, 4-bromobutylsulfinyl or

[0252] nonafluorobutylsulfinyl;

[0253] C1-C6-haloalkylsulfinyl: C1-C4-haloalkylsulfinyl as mentioned above, and also 5-fluoropentylsulfinyl,

[0254] 5-chloropentylsulfinyl, 5-bromopentylsulfinyl,

[0255] 5-iodopentylsulfinyl, undecafluoropentylsulfinyl,

[0256] 6-fluorohexylsulfinyl, 6-chlorohexylsulfinyl,

[0257] 6-bromohexylsulfinyl, 6-iodohexylsulfinyl or

[0258] dodecafluorohexylsulfinyl;

[0259] C1-C4-alkylsulfonyl (C1-C4-alkyl-S(═O)2—) and the alkylsulfonyl moieties of C1-C4-alkylsulfonyl-C1-C4-alkyl: for example methylsulfonyl, ethylsulfonyl, propylsulfonyl,

[0260] 1-methylethylsulfonyl, butylsulfonyl, 1-methylpropylsulfonyl,

[0261] 2-methylpropylsulfonyl or 1,1-dimethylethylsulfonyl;

[0262] C1-C6-alkylsulfonyl: C1-C4-alkylsulfonyl, as mentioned above,

[0263] and also pentylsulfonyl, 1-methylbutylsulfonyl,

[0264] 2-methylbutylsulfonyl, 3-methylbutylsulfonyl,

[0265] 1,1-dimethylpropylsulfonyl, 1,2-dimethylpropylsulfonyl,

[0266] 2,2-dimethylpropylsulfonyl, 1-ethylpropylsulfonyl,

[0267] hexylsulfonyl, 1-methylpentylsulfonyl,

[0268] 2-methylpentylsulfonyl, 3-methylpentylsulfonyl,

[0269] 4-methylpentylsulfonyl, 1,1-dimethylbutylsulfonyl,

[0270] 1,2-dimethylbutylsulfonyl, 1,3-dimethylbutylsulfonyl,

[0271] 2,2-dimethylbutylsulfonyl, 2,3-dimethylbutylsulfonyl,

[0272] 3,3-dimethylbutylsulfonyl, 1-ethylbutylsulfonyl,

[0273] 2-ethylbutylsulfonyl, 1,1,2-trimethylpropylsulfonyl,

[0274] 1,2,2-trimethylpropylsulfonyl, 1-ethyl-1-methylpropylsulfonyl

[0275] or 1-ethyl-2-methylpropylsulfonyl;

[0276] C1-C4-haloalkylsulfonyl: a C1-C4-alkylsulfonyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, and also the haloalkylsulfonyl of C1-C4-haloalkylsulfonyl-C1-C4-alkyl: for example, fluoromethylsulfonyl, difluoromethylsulfonyl,

[0277] trifluoromethylsulfonyl, chlorodifluoromethylsulfonyl,

[0278] bromodifluoromethylsulfonyl, 2-fluoroethylsulfonyl,

[0279] 2-chloroethylsulfonyl, 2-bromoethylsulfonyl,

[0280] 2-iodoethylsulfonyl, 2,2-difluoroethylsulfonyl,

[0281] 2,2,2-trifluoroethylsulfonyl, 2-chloro-2-fluoroethylsulfonyl,

[0282] 2-chloro-2,2-difluoroethylsulfonyl, 2,2-dichloro-2-fluoroethylsulfonyl, 2,2,2-trichloroethylsulfonyl,

[0283] pentafluoroethylsulfonyl, 2-fluoropropylsulfonyl,

[0284] 3-fluoropropylsulfonyl, 2-chloropropylsulfonyl,

[0285] 3-chloropropylsulfonyl, 2-bromopropylsulfonyl,

[0286] 3-bromopropylsulfonyl, 2,2-difluoropropylsulfonyl,

[0287] 2,3-difluoropropylsulfonyl, 2,3-dichloropropylsulfonyl,

[0288] 3,3,3-trifluoropropylsulfonyl, 3,3,3-trichloropropylsulfonyl,

[0289] 2,2,3,3,3-pentafluoropropylsulfonyl, heptafluoropropylsulfonyl, 1-(fluoromethyl)-2-fluoroethylsulfonyl,

[0290] 1-(chloromethyl)-2-chloroethylsulfonyl, 1-(bromomethyl)-2-bromoethylsulfonyl, 4-fluorobutylsulfonyl,

[0291] 4-chlorobutylsulfonyl, 4-bromobutylsulfonyl or

[0292] nonafluorobutylsulfonyl;

[0293] C1-C6-haloalkylsulfonyl and the haloalkylsulfonyl moieties of C1-C6-haloalkylsulfonyl-C1-C6-alkyl: C1-C4-haloalkylsulfonyl as mentioned above, and also 5-fluoropentylsulfonyl,

[0294] 5-chloropentylsulfonyl, 5-bromopentylsulfonyl,

[0295] 5-iodopentylsulfonyl, 6-fluorohexylsulfonyl,

[0296] 6-bromohexylsulfonyl, 6-iodohexylsulfonyl or

[0297] dodecafluorohexylsulfonyl;

[0298] C1-C6-alkylamino: methylamino, ethylamino, propylamino,

[0299] 1-methylethylamino, butylamino, 1-methylpropylamino,

[0300] 2-methylpropylamino, 1,1-dimethylethylamino, pentylamino,

[0301] 1-methylbutylamino, 2-methylbutylamino, 3-methylbutylamino,

[0302] 2,2-dimethylpropylamino, 1-ethylpropylamino, hexylamino,

[0303] 1,1-dimethylpropylamino, 1,2-dimethylpropylamino,

[0304] 1-methylpentylamino, 2-methylpentylamino,

[0305] 3-methylpentylamino, 4-methylpentylamino,

[0306] 1,1-dimethylbutylamino, 1,2-dimethylbutylamino,

[0307] 1,3-dimethylbutylamino, 2,2-dimethylbutylamino,

[0308] 2,3-dimethylbutylamino, 3,3-dimethylbutylamino,

[0309] 1-ethylbutylamino, 2-ethylbutylamino,

[0310] 1,1,2-trimethylpropylamino, 1,2,2-trimethylpropylamino,

[0311] 1-ethyl-1-methylpropylamino or 1-ethyl-2-methylpropylamino;

[0312] di(C1-C4-alkyl)amino: for example N,N-dimethylamino,

[0313] N,N-diethylamino, N,N-dipropylamino, N,N-di(1-methylethyl)-amino, N,N-dibutylamino, N,N-di(1-methylpropyl)amino,

[0314] N,N-di(2-methylpropyl)amino, N,N-di(1,1-dimethylethyl)amino,

[0315] N-ethyl-N-methylamino, N-methyl-N-propylamino,

[0316] N-methyl-N-(1-methylethyl)amino, N-butyl-N-methylamino,

[0317] N-methyl-N-(1-methylpropyl)amino, N-methyl-N-(2-methylpropyl)amino, N-(1,1-dimethylethyl)-N-methylamino,

[0318] N-ethyl-N-propylamino, N-ethyl-N-(1-methylethyl)amino,

[0319] N-butyl-N-ethylamino, N-ethyl-N-(1-methylpropyl)amino,

[0320] N-ethyl-N-(2-methylpropyl)amino, N-ethyl-N-(1,1-dimethyl-ethyl)amino, N-(1-methylethyl)-N-propylamino,

[0321] N-butyl-N-propylamino, N-(1-methylpropyl)-N-propylamino,

[0322] N-(2-methylpropyl)-N-propylamino, N-(1,1-dimethylethyl)-N-propylamino, N-butyl-N-(1-methylethyl)amino,

[0323] N-(1-methylethyl)-N-(1-methylpropyl)amino, N-(1-methylethyl)-N-(2-methylpropyl)amino, N-(1,1-dimethylethyl)-N-(1-methylethyl)amino, N-butyl-N-(1-methylpropyl)amino,

[0324] N-butyl-N-(2-methylpropyl)amino, N-butyl-N-(1,1-dimethyl-ethyl)amino, N-(1-methylpropyl)-N-(2-methylpropyl)amino,

[0325] N-(1,1-dimethylethyl)-N-(1-methylpropyl)amino or

[0326] N-(1,1-dimethylethyl)-N-(2-methylpropyl)amino;

[0327] di(C1-C6-alkyl)amino: di(C1-C4-alkyl)amino as mentioned above,

[0328] and also N,N-dipentylamino, N,N-dihexylamino,

[0329] N-methyl-N-pentylamino, N-ethyl-N-pentylamino,

[0330] N-methyl-N-hexylamino or N-ethyl-N-hexylamino;

[0331] C1-C4-alkylcarbonyl: for example methylcarbonyl,

[0332] ethylcarbonyl, propylcarbonyl, 1-methylethylcarbonyl,

[0333] butylcarbonyl, 1-methylpropylcarbonyl, 2-methylpropylcarbonyl

[0334] or 1,1-dimethylethylcarbonyl;

[0335] C1-C6-alkylcarbonyl, and the alkylcarbonyl radicals of C1-C6-alkylcarbonylamino: C1-C4-alkylcarbonyl as mentioned above, and also, for example, pentylcarbonyl,

[0336] 1-methylbutylcarbonyl, 2-methylbutylcarbonyl,

[0337] 3-methylbutylcarbonyl, 2,2-dimethylpropylcarbonyl,

[0338] 1-ethylpropylcarbonyl, hexylcarbonyl, 1,1-dimethylpropyl-carbonyl, 1,2-dimethylpropylcarbonyl, 1-methylpentylcarbonyl,

[0339] 2-methylpentylcarbonyl, 3-methylpentylcarbonyl,

[0340] 4-methylpentylcarbonyl, 1,1-dimethylbutylcarbonyl,

[0341] 1,2-dimethylbutylcarbonyl, 1,3-dimethylbutylcarbonyl,

[0342] 2,2-dimethylbutylcarbonyl, 2,3-dimethylbutylcarbonyl,

[0343] 3,3-dimethylbutylcarbonyl, 1-ethylbutylcarbonyl,

[0344] 2-ethylbutylcarbonyl, 1,1,2-trimethylpropylcarbonyl,

[0345] 1,2,2-trimethylpropylcarbonyl, 1-ethyl-1-methylpropylcarbonyl

[0346] or 1-ethyl-2-methylpropylcarbonyl;

[0347] C1-C4-haloalkylcarbonyl: a C1-C4-alkylcarbonyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e. for example,

[0348] chloroacetyl, dichloroacetyl, trichloroacetyl, fluoroacetyl,

[0349] difluoroacetyl, trifluoroacetyl, chlorofluoroacetyl,

[0350] dichlorofluoroacetyl, chlorodifluoroacetyl, 2-fluoroethyl-carbonyl, 2-chloroethylcarbonyl, 2-bromoethylcarbonyl,

[0351] 2-iodoethylcarbonyl, 2,2-difluoroethylcarbonyl,

[0352] 2,2,2-trifluoroethylcarbonyl, 2-chloro-2-fluoroethylcarbonyl,

[0353] 2-chloro-2,2-difluoroethylcarbonyl, 2,2-dichloro-2-fluoroethylcarbonyl, 2,2,2-trichloroethylcarbonyl,

[0354] pentafluoroethylcarbonyl, 2-fluoropropylcarbonyl,

[0355] 3-fluoropropylcarbonyl, 2,2-difluoropropylcarbonyl,

[0356] 2,3-difluoropropylcarbonyl, 2-chloropropylcarbonyl,

[0357] 3-chloropropylcarbonyl, 2,3-dichloropropylcarbonyl,

[0358] 2-bromopropylcarbonyl, 3-bromopropylcarbonyl,

[0359] 3,3,3-trifluoropropylcarbonyl, 3,3,3-trichloropropylcarbonyl,

[0360] 2,2,3,3,3-pentafluoropropylcarbonyl, heptafluoropropyl-carbonyl, 1-(fluoromethyl)-2-fluoroethylcarbonyl,

[0361] 1-(chloromethyl)-2-chloroethylcarbonyl, 1-(bromomethyl)-2-bromoethylcarbonyl, 4-fluorobutylcarbonyl,

[0362] 4-chlorobutylcarbonyl, 4-bromobutylcarbonyl or

[0363] nonafluorobutylcarbonyl;

[0364] C1-C6-haloalkylcarbonyl: a C1-C4-haloalkylcarbonyl radical as mentioned above, and also 5-fluoropentylcarbonyl,

[0365] 5-chloropentylcarbonyl, 5-bromopentylcarbonyl,

[0366] perfluoropentylcarbonyl, 6-fluorohexylcarbonyl,

[0367] 6-chlorohexylcarbonyl, 6-bromohexylcarbonyl or

[0368] perfluorohexylcarbonyl;

[0369] C1-C4-alkoxycarbonyl: for example methoxycarbonyl,

[0370] ethoxycarbonyl, propoxycarbonyl, 1-methylethoxycarbonyl,

[0371] butoxycarbonyl, 1-methylpropoxycarbonyl,

[0372] 2-methylpropoxycarbonyl or 1,1-dimethylethoxycarbonyl;

[0373] C1-C6-alkoxycarbonyl and also the alkoxycarbonyl moieties of C1-C6-alkoxycarbonyl-C1-C6-alkyl: C1-C4-alkoxycarbonyl as mentioned above, and also, for example, pentoxycarbonyl,

[0374] 1-methylbutoxy-carbonyl, 2-methylbutoxycarbonyl, 3-methylbutoxycarbonyl,

[0375] 2,2-dimethylpropoxycarbonyl, 1-ethylpropoxycarbonyl,

[0376] hexoxycarbonyl, 1,1-dimethylpropoxycarbonyl,

[0377] 1,2-dimethylpropoxycarbonyl, 1-methylpentoxycarbonyl,

[0378] 2-methylpentoxycarbonyl, 3-methylpentoxycarbonyl,

[0379] 4-methylpentoxycarbonyl, 1,1-dimethylbutoxycarbonyl,

[0380] 1,2-dimethylbutoxycarbonyl, 1,3-dimethylbutoxycarbonyl,

[0381] 2,2-dimethylbutoxycarbonyl, 2,3-dimethylbutoxycarbonyl,

[0382] 3,3-dimethylbutoxycarbonyl, 1-ethylbutoxycarbonyl,

[0383] 2-ethylbutoxycarbonyl, 1,1,2-trimethylpropoxycarbonyl,

[0384] 1,2,2-trimethylpropoxycarbonyl, 1-ethyl-1-methylpropoxy-carbonyl or 1-ethyl-2-methylpropoxycarbonyl;

[0385] C1-C4-haloalkoxycarbonyl: a C1-C4-alkoxycarbonyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example

[0386] fluoromethoxycarbonyl, difluoromethoxycarbonyl,

[0387] trifluoromethoxycarbonyl, chlorodifluoromethoxycarbonyl,

[0388] bromodifluoromethoxycarbonyl, 2-fluoroethoxycarbonyl,

[0389] 2-chloroethoxycarbonyl, 2-bromoethoxycarbonyl,

[0390] 2-iodoethoxycarbonyl, 2,2-difluoroethoxycarbonyl,

[0391] 2,2,2-trifluoroethoxycarbonyl, 2-chloro-2-fluoroethoxy-carbonyl, 2-chloro-2,2-difluoroethoxycarbonyl,

[0392] 2,2-dichloro-2-fluoroethoxycarbonyl, 2,2,2-trichloroethoxycarbonyl, pentafluoroethoxycarbonyl, 2-fluoropropoxycarbonyl,

[0393] 3-fluoropropoxycarbonyl, 2-chloropropoxycarbonyl,

[0394] 3-chloropropoxycarbonyl, 2-bromopropoxycarbonyl,

[0395] 3-bromopropoxycarbonyl, 2,2-difluoropropoxycarbonyl,

[0396] 2,3-difluoropropoxycarbonyl, 2,3-dichloropropoxycarbonyl,

[0397] 3,3,3-trifluoropropoxycarbonyl, 3,3,3-trichloropropoxycarbonyl, 2,2,3,3,3-pentafluoropropoxycarbonyl,

[0398] heptafluoropropoxycarbonyl, 1-(fluoromethyl)-2-fluoroethoxycarbonyl, 1-(chloromethyl)-2-chloroethoxycarbonyl,

[0399] 1-(bromomethyl)-2-bromoethoxycarbonyl,

[0400] 4-fluorobutoxycarbonyl, 4-chlorobutoxycarbonyl,

[0401] 4-bromobutoxycarbonyl or 4-iodobutoxycarbonyl;

[0402] C1-C6-haloalkoxycarbonyl: a C1-C4-haloalkoxycarbonyl radical as mentioned above, and also 5-fluoropentoxycarbonyl,

[0403] 5-chloropentoxycarbonyl, 5-bromopentoxycarbonyl,

[0404] 6-fluorohexoxycarbonyl, 6-chlorohexoxycarbonyl or

[0405] 6-bromohexoxycarbonyl;

[0406] (C1-C4-alkyl)carbonyloxy: acetyloxy, ethylcarbonyloxy,

[0407] propylcarbonyloxy, 1-methylethylcarbonyloxy,

[0408] butylcarbonyloxy, 1-methylpropylcarbonyloxy,

[0409] 2-methylpropylcarbonyloxy or 1,1-dimethylethylcarbonyloxy;

[0410] (C1-C4-alkylamino)carbonyl: for example methylaminocarbonyl,

[0411] ethylaminocarbonyl, propylaminocarbonyl,

[0412] 1-methylethylaminocarbonyl, butylaminocarbonyl,

[0413] 1-methylpropylaminocarbonyl, 2-methylpropylaminocarbonyl or

[0414] 1,1-dimethylethylaminocarbonyl;

[0415] (C1-C6-alkylamino)carbonyl: (C1-C4-alkylamino)carbonyl as mentioned above, and also, for example, pentylaminocarbonyl,

[0416] 1-methylbutylaminocarbonyl, 2-methylbutylaminocarbonyl,

[0417] 3-methylbutylaminocarbonyl, 2,2-dimethylpropylaminocarbonyl,

[0418] 1-ethylpropylaminocarbonyl, hexylaminocarbonyl,

[0419] 1,1-dimethylpropylaminocarbonyl, 1,2-dimethylpropylamino-carbonyl, 1-methylpentylaminocarbonyl, 2-methylpentylamino-carbonyl, 3-methylpentylaminocarbonyl, 4-methylpentylamino-carbonyl, 1,1-dimethylbutylaminocarbonyl, 1,2-dimethylbutylamino-carbonyl, 1,3-dimethylbutylaminocarbonyl, 2,2-dimethyl-butylaminocarbonyl, 2,3-dimethylbutylaminocarbonyl,

[0420] 3,3-dimethylbutylaminocarbonyl, 1-ethylbutylaminocarbonyl,

[0421] 2-ethylbutylaminocarbonyl, 1,1,2-trimethylpropylamino-carbonyl, 1,2,2-trimethylpropylaminocarbonyl,

[0422] 1-ethyl-1-methylpropylaminocarbonyl or

[0423] 1-ethyl-2-methylpropylaminocarbonyl;

[0424] di(C1-C4-alkyl)aminocarbonyl: for example

[0425] N,N-dimethylaminocarbonyl, N,N-diethylaminocarbonyl,

[0426] N,N-di(1-methylethyl)aminocarbonyl, N,N-dipropylamino-carbonyl, N,N-dibutylaminocarbonyl, N,N-di(1-methylpropyl)-aminocarbonyl, N,N-di(2-methylpropyl)aminocarbonyl,

[0427] N,N-di(1,1-dimethylethyl)aminocarbonyl, N-ethyl-N-methyl-aminocarbonyl, N-methyl-N-propylaminocarbonyl,

[0428] N-methyl-N-(1-methylethyl)aminocarbonyl, N-butyl-N-methyl-aminocarbonyl, N-methyl-N-(1-methylpropyl)aminocarbonyl,

[0429] N-methyl-N-(2-methylpropyl)aminocarbonyl,

[0430] N-(1,1-dimethylethyl)-N-methylaminocarbonyl,

[0431] N-ethyl-N-propylaminocarbonyl, N-ethyl-N-(1-methylethyl)-aminocarbonyl, N-butyl-N-ethylaminocarbonyl,

[0432] N-ethyl-N-(1-methylpropyl)aminocarbonyl, N-ethyl-N-(2-methyl-propyl)aminocarbonyl, N-ethyl-N-(1,1-dimethylethyl)amino-carbonyl, N-(1-methylethyl)-N-propylaminocarbonyl,

[0433] N-butyl-N-propylaminocarbonyl, N-(1-methylpropyl)-N-propyl-aminocarbonyl, N-(2-methylpropyl)-N-propylaminocarbonyl,

[0434] N-(1,1-dimethylethyl)-N-propylaminocarbonyl,

[0435] N-butyl-N-(1-methylethyl)aminocarbonyl, N-(1-methylethyl)-N-(1-methylpropyl)aminocarbonyl, N-(1-methylethyl)-N-(2-methylpropyl)aminocarbonyl, N-(1,1-dimethylethyl)-N-(1-methylethyl)aminocarbonyl, N-butyl-N-(1-methylpropyl)aminocarbonyl,

[0436] N-butyl-N-(2-methylpropyl)aminocarbonyl,

[0437] N-butyl-N-(1,1-dimethylethyl)aminocarbonyl,

[0438] N-(1-methylpropyl)-N-(2-methylpropyl)aminocarbonyl,

[0439] N-(1,1-dimethylethyl)-N-(1-methylpropyl)aminocarbonyl or N-(1,1-dimethylethyl)-N-(2-methylpropyl)aminocarbonyl;

[0440] di(C1-C6-alkyl)aminocarbonyl: di(C1-C4-alkyl)aminocarbonyl as mentioned above, and also, for example, N-methyl-N-pentyl-aminocarbonyl,

[0441] N-methyl-N-(1-methylbutyl)aminocarbonyl, N-methyl-N-(2-methylbutyl)aminocarbonyl, N-methyl-N-(3-methylbutyl)aminocarbonyl, N-methyl-N-(2,2-dimethyl-propyl)aminocarbonyl, N-methyl-N-(1-ethylpropyl)-aminocarbonyl, N-methyl-N-hexylaminocarbonyl,

[0442] N-methyl-N-(1,1-dimethylpropyl)aminocarbonyl,

[0443] N-methyl-N-(1,2-dimethylpropyl)aminocarbonyl,

[0444] N-methyl-N-(1-methylpentyl)aminocarbonyl,

[0445] N-methyl-N-(2-methylpentyl)aminocarbonyl,

[0446] N-methyl-N-(3-methylpentyl)aminocarbonyl,

[0447] N-methyl-N-(4-methylpentyl)aminocarbonyl,

[0448] N-methyl-N-(1,1-dimethylbutyl)aminocarbonyl,

[0449] N-methyl-N-(1,2-dimethylbutyl)aminocarbonyl,

[0450] N-methyl-N-(1,3-dimethylbutyl)aminocarbonyl,

[0451] N-methyl-N-(2,2-dimethylbutyl)aminocarbonyl,

[0452] N-methyl-N-(2,3-dimethylbutyl)aminocarbonyl,

[0453] N-methyl-N-(3,3-dimethylbutyl)aminocarbonyl,

[0454] N-methyl-N-(1-ethylbutyl)aminocarbonyl,

[0455] N-methyl-N-(2-ethylbutyl)aminocarbonyl,

[0456] N-methyl-N-(1,1,2-trimethylpropyl)aminocarbonyl,

[0457] N-methyl-N-(1,2,2-trimethylpropyl)aminocarbonyl,

[0458] N-methyl-N-(1-ethyl-1-methylpropyl)aminocarbonyl,

[0459] N-methyl-N-(1-ethyl-2-methylpropyl)aminocarbonyl,

[0460] N-ethyl-N-pentylaminocarbonyl,

[0461] N-ethyl-N-(1-methylbutyl)aminocarbonyl,

[0462] N-ethyl-N-(2-methylbutyl)aminocarbonyl,

[0463] N-ethyl-N-(3-methylbutyl)aminocarbonyl,

[0464] N-ethyl-N-(2,2-dimethylpropyl)aminocarbonyl,

[0465] N-ethyl-N-(1-ethylpropyl)aminocarbonyl,

[0466] N-ethyl-N-hexylaminocarbonyl,

[0467] N-ethyl-N-(1,1-dimethylpropyl)aminocarbonyl,

[0468] N-ethyl-N-(1,2-dimethylpropyl)aminocarbonyl,

[0469] N-ethyl-N-(1-methylpentyl)aminocarbonyl,

[0470] N-ethyl-N-(2-methylpentyl)aminocarbonyl,

[0471] N-ethyl-N-(3-methylpentyl)aminocarbonyl,

[0472] N-ethyl-N-(4-methylpentyl)aminocarbonyl,

[0473] N-ethyl-N-(1,1-dimethylbutyl)aminocarbonyl,

[0474] N-ethyl-N-(1,2-dimethylbutyl)aminocarbonyl,

[0475] N-ethyl-N-(1,3-dimethylbutyl)aminocarbonyl,

[0476] N-ethyl-N-(2,2-dimethylbutyl)aminocarbonyl,

[0477] N-ethyl-N-(2,3-dimethylbutyl)aminocarbonyl,

[0478] N-ethyl-N-(3,3-dimethylbutyl)aminocarbonyl,

[0479] N-ethyl-N-(1-ethylbutyl)aminocarbonyl,

[0480] N-ethyl-N-(2-ethylbutyl)aminocarbonyl,

[0481] N-ethyl-N-(1,1,2-trimethylpropyl)aminocarbonyl,

[0482] N-ethyl-N-(1,2,2-trimethylpropyl)aminocarbonyl,

[0483] N-ethyl-N-(1-ethyl-1-methylpropyl)aminocarbonyl,

[0484] N-ethyl-N-(1-ethyl-2-methylpropyl)aminocarbonyl,

[0485] N-propyl-N-pentylaminocarbonyl,

[0486] N-butyl-N-pentylaminocarbonyl, N,N-dipentylaminocarbonyl,

[0487] N-propyl-N-hexylaminocarbonyl, N-butyl-N-hexylaminocarbonyl,

[0488] N-pentyl-N-hexylaminocarbonyl or N,N-dihexylaminocarbonyl;

[0489] di(C1-C6-alkyl)aminothiocarbonyl: for example

[0490] N,N-dimethylaminothiocarbonyl, N,N-diethylaminothiocarbonyl,

[0491] N,N-di(1-methylethyl)aminothiocarbonyl,

[0492] N,N-dipropylaminothiocarbonyl, N,N-dibutylaminothiocarbonyl,

[0493] N,N-di(1-methylpropyl)aminothiocarbonyl,

[0494] N,N-di(2-methylpropyl)aminothiocarbonyl,

[0495] N,N-di(1,1-dimethylethyl)aminothiocarbonyl,

[0496] N-ethyl-N-methylaminothiocarbonyl,

[0497] N-methyl-N-propylaminothiocarbonyl,

[0498] N-methyl-N-(1-methylethyl)aminothiocarbonyl,

[0499] N-butyl-N-methylaminothiocarbonyl,

[0500] N-methyl-N-(1-methylpropyl)aminothiocarbonyl,

[0501] N-methyl-N-(2-methylpropyl)aminothiocarbonyl,

[0502] N-(1,1-dimethylethyl)-N-methylaminothiocarbonyl,

[0503] N-ethyl-N-propylaminothiocarbonyl,

[0504] N-ethyl-N-(1-methylethyl)aminothiocarbonyl,

[0505] N-butyl-N-ethylaminothiocarbonyl,

[0506] N-ethyl-N-(1-methylpropyl)aminothiocarbonyl,

[0507] N-ethyl-N-(2-methylpropyl)aminothiocarbonyl,

[0508] N-ethyl-N-(1,1-dimethylethyl)aminothiocarbonyl,

[0509] N-(1-methylethyl)-N-propylaminothiocarbonyl,

[0510] N-butyl-N-propylaminothiocarbonyl,

[0511] N-(1-methylpropyl)-N-propylaminothiocarbonyl,

[0512] N-(2-methylpropyl)-N-propylaminothiocarbonyl,

[0513] N-(1,1-dimethylethyl)-N-propylaminothiocarbonyl,

[0514] N-butyl-N-(1-methylethyl)aminothiocarbonyl,

[0515] N-(1-methylethyl)-N-(1-methylpropyl)aminothiocarbonyl,

[0516] N-(1-methylethyl)-N-(2-methylpropyl)aminothiocarbonyl,

[0517] N-(1,1-dimethylethyl)-N-(1-methylethyl)aminothiocarbonyl,

[0518] N-butyl-N-(1-methylpropyl)aminothiocarbonyl,

[0519] N-butyl-N-(2-methylpropyl)aminothiocarbonyl,

[0520] N-butyl-N-(1,1-dimethylethyl)aminothiocarbonyl,

[0521] N-(1-methylpropyl)-N-(2-methylpropyl)aminothiocarbonyl,

[0522] N-(1,1-dimethylethyl)-N-(1-methylpropyl)aminothiocarbonyl,

[0523] N-(1,1-dimethylethyl)-N-(2-methylpropyl)aminothiocarbonyl,

[0524] N-methyl-N-pentylaminothiocarbonyl,

[0525] N-methyl-N-(1-methylbutyl)aminothiocarbonyl,

[0526] N-methyl-N-(2-methylbutyl)aminothiocarbonyl,

[0527] N-methyl-N-(3-methylbutyl)aminothiocarbonyl,

[0528] N-methyl-N-(2,2-dimethylpropyl)aminothiocarbonyl,

[0529] N-methyl-N-(1-ethylpropyl)aminothiocarbonyl,

[0530] N-methyl-N-hexylaminothiocarbonyl,

[0531] N-methyl-N-(1,1-dimethylpropyl)aminothiocarbonyl,

[0532] N-methyl-N-(1,2-dimethylpropyl)aminothiocarbonyl,

[0533] N-methyl-N-(1-methylpentyl)aminothiocarbonyl,

[0534] N-methyl-N-(2-methylpentyl)aminothiocarbonyl,

[0535] N-methyl-N-(3-methylpentyl)aminothiocarbonyl,

[0536] N-methyl-N-(4-methylpentyl)aminothiocarbonyl,

[0537] N-methyl-N-(1,1-dimethylbutyl)aminothiocarbonyl,

[0538] N-methyl-N-(1,2-dimethylbutyl)aminothiocarbonyl,

[0539] N-methyl-N-(1,3-dimethylbutyl)aminothiocarbonyl,

[0540] N-methyl-N-(2,2-dimethylbutyl)aminothiocarbonyl,

[0541] N-methyl-N-(2,3-dimethylbutyl)aminothiocarbonyl,

[0542] N-methyl-N-(3,3-dimethylbutyl)aminothiocarbonyl,

[0543] N-methyl-N-(1-ethylbutyl)aminothiocarbonyl,

[0544] N-methyl-N-(2-ethylbutyl)aminothiocarbonyl,

[0545] N-methyl-N-ethyl-N-(1,1,2-trimethylpropyl)aminothiocarbonyl,

[0546] N-methyl-N-(1,2,2-trimethylpropyl)aminothiocarbonyl,

[0547] N-methyl-N-(1-ethyl-1-methylpropyl)aminothiocarbonyl,

[0548] N-methyl-N-(1-ethyl-2-methylpropyl)aminothiocarbonyl,

[0549] N-ethyl-N-pentylaminothiocarbonyl,

[0550] N-ethyl-N-(1-methylbutyl)aminothiocarbonyl,

[0551] N-ethyl-N-(2-methylbutyl)aminothiocarbonyl,

[0552] N-ethyl-N-(3-methylbutyl)aminothiocarbonyl,

[0553] N-ethyl-N-(2,2-dimethylpropyl)aminothiocarbonyl,

[0554] N-ethyl-N-(1-ethylpropyl)aminothiocarbonyl,

[0555] N-ethyl-N-hexylaminothiocarbonyl,

[0556] N-ethyl-N-(1,1-dimethylpropyl)aminothiocarbonyl,

[0557] N-ethyl-N-(1,2-dimethylpropyl)aminothiocarbonyl,

[0558] N-ethyl-N-(1-methylpentyl)aminothiocarbonyl,

[0559] N-ethyl-N-(2-methylpentyl)aminothiocarbonyl,

[0560] N-ethyl-N-(3-methylpentyl)aminothiocarbonyl,

[0561] N-ethyl-N-(4-methylpentyl)aminothiocarbonyl,

[0562] N-ethyl-N-(1,1-dimethylbutyl)aminothiocarbonyl,

[0563] N-ethyl-N-(1,2-dimethylbutyl)aminothiocarbonyl,

[0564] N-ethyl-N-(1,3-dimethylbutyl)aminothiocarbonyl,

[0565] N-ethyl-N-(2,2-dimethylbutyl)aminothiocarbonyl,

[0566] N-ethyl-N-(2,3-dimethylbutyl)aminothiocarbonyl,

[0567] N-ethyl-N-(3,3-dimethylbutyl)aminothiocarbonyl,

[0568] N-ethyl-N-(1-ethylbutyl)aminothiocarbonyl,

[0569] N-ethyl-N-(2-ethylbutyl)aminothiocarbonyl,

[0570] N-ethyl-N-(1,1,2-trimethylpropyl)aminothiocarbonyl,

[0571] N-ethyl-N-(1,2,2-trimethylpropyl)aminothiocarbonyl,

[0572] N-ethyl-N-(1-ethyl-1-methylpropyl)aminothiocarbonyl,

[0573] N-ethyl-N-(1-ethyl-2-methylpropyl)aminothiocarbonyl,

[0574] N-propyl-N-pentylaminothiocarbonyl,

[0575] N-butyl-N-pentylaminothiocarbonyl,

[0576] N,N-dipentylaminothiocarbonyl,

[0577] N-propyl-N-hexylaminothiocarbonyl,

[0578] N-butyl-N-hexylaminothiocarbonyl,

[0579] N-pentyl-N-hexylaminothiocarbonyl or

[0580] N,N-dihexylaminothiocarbonyl;

[0581] C1-C6-hydroxyalkyl: C1-C6-alkyl which is substituted by one to three OH groups, for example hydroxymethyl, 1-hydroxyethyl,

[0582] 2-hydroxyethyl, 1,2-bishydroxyethyl, 1-hydroxypropyl,

[0583] 2-hydroxypropyl, 3-hydroxypropyl, 4-hydroxybutyl,

[0584] 2,2-dimethyl-3-hydroxypropyl;

[0585] phenyl-C1-C6-alkyl: C1-C6-alkyl which is substituted by a phenyl radical, for example benzyl, 1-phenylethyl and 2-phenylethyl, where the phenyl radical may, in the manner mentioned, be partially or fully halogenated or may carry one to three of the substituents mentioned above for phenyl; correspondingly, heterocyclyl-C1-C6-alkyl is a C1-C6-alkyl which is substituted by a heterocyclyl radical;

[0586] C1-C6-alkoxy-C1-C6-alkyl: C1-C6-alkyl which is substituted by C1-C6-alkoxy as mentioned above, i.e., for example,

[0587] methoxymethyl, ethoxymethyl, propoxymethyl, (1-methylethoxy)-methyl, butoxymethyl, (1-methylpropoxy)methyl,

[0588] (2-methylpropoxy)methyl, (1,1-dimethylethoxy)methyl,

[0589] 2-(methoxy)ethyl, 2-(ethoxy)ethyl, 2-(propoxy)ethyl,

[0590] 2-(1-methylethoxy)ethyl, 2-(butoxy)ethyl,

[0591] 2-(1-methylpropoxy)ethyl, 2-(2-methylpropoxy)ethyl,

[0592] 2-(1,1-dimethylethoxy)ethyl, 2-(methoxy)propyl,

[0593] 2-(ethoxy)propyl, 2-(propoxy)propyl, 2-(1-methylethoxy)-propyl, 2-(butoxy)propyl, 2-(1-methylpropoxy)propyl,

[0594] 2-(2-methylpropoxy)propyl, 2-(1,1-dimethylethoxy)propyl,

[0595] 3-(methoxy)propyl, 3-(ethoxy)propyl, 3-(propoxy)propyl,

[0596] 3-(1-methylethoxy)propyl, 3-(butoxy)propyl,

[0597] 3-(1-methylpropoxy)propyl, 3-(2-methylpropoxy)propyl,

[0598] 3-(1,1-dimethylethoxy)propyl, 2-(methoxy)butyl,

[0599] 2-(ethoxy)butyl, 2-(propoxy)butyl, 2-(1-methylethoxy)butyl,

[0600] 2-(butoxy)butyl, 2-(1-methylpropoxy)butyl,

[0601] 2-(2-methylpropoxy)butyl, 2-(1,1-dimethylethoxy)butyl,

[0602] 3-(methoxy)butyl, 3-(ethoxy)butyl, 3-(propoxy)butyl,

[0603] 3-(1-methylethoxy)butyl, 3-(butoxy)butyl,

[0604] 3-(1-methylpropoxy)butyl, 3-(2-methylpropoxy)butyl,

[0605] 3-(1,1-dimethylethoxy)butyl, 4-(methoxy)butyl,

[0606] 4-(ethoxy)butyl, 4-(propoxy)butyl, 4-(1-methylethoxy)butyl,

[0607] 4-(butoxy)butyl, 4-(1-methylpropoxy)butyl,

[0608] 4-(2-methylpropoxy)butyl or 4-(1,1-dimethylethoxy)butyl;

[0609] C1-C6-alkoxy-C1-C6-alkoxy, and the alkoxyalkoxy moieties of C1-C6-alkoxy-C1-C6-alkoxycarbonyl: C1-C6-alkoxy which is substituted by C1-C6-alkoxy as mentioned above, i.e, for example, methoxymethoxy, ethoxymethoxy, propoxymethoxy,

[0610] (1-methylethoxy)methoxy, butoxymethoxy, (1-methylpropoxy)-methoxy, (2-methylpropoxy)methoxy, (1,1-dimethylethoxy)-methoxy, 2-(methoxy)ethoxy, 2-(ethoxy)ethoxy,

[0611] 2-(propoxy)ethoxy, 2-(1-methylethoxy)ethoxy,

[0612] 2-(butoxy)ethoxy, 2-(1-methylpropoxy)ethoxy,

[0613] 2-(2-methylpropoxy)ethoxy, 2-(1,1-dimethylethoxy)ethoxy,

[0614] 2-(methoxy)propoxy, 2-(ethoxy)propoxy, 2-(propoxy)propoxy,

[0615] 2-(1-methylethoxy)propoxy, 2-(butoxy)propoxy,

[0616] 2-(1-methylpropoxy)propoxy, 2-(2-methylpropoxy)propoxy,

[0617] 2-(1,1-dimethylethoxy)propoxy, 3-(methoxy)propoxy,

[0618] 3-(ethoxy)propoxy, 3-(propoxy)propoxy, 3-(1-methylethoxy)-propoxy, 3-(butoxy)propoxy, 3-(1-methylpropoxy)propoxy,

[0619] 3-(2-methylpropoxy)propoxy, 3-(1,1-dimethylethoxy)propoxy,

[0620] 2-(methoxy)butoxy, 2-(ethoxy)butoxy, 2-(propoxy)-butoxy,

[0621] 2-(1-methylethoxy)butoxy, 2-(butoxy)butoxy,

[0622] 2-(1-methylpropoxy)butoxy, 2-(2-methylpropoxy)butoxy,

[0623] 2-(1,1-dimethylethoxy)butoxy, 3-(methoxy)butoxy,

[0624] 3-(ethoxy)butoxy, 3-(propoxy)butoxy, 3-(1-methylethoxy)butoxy, 3-(butoxy)butoxy, 3-(1-methylpropoxy)butoxy,

[0625] 3-(2-methylpropoxy)butoxy, 3-(1,1-dimethylethoxy)butoxy,

[0626] 4-(methoxy)butoxy, 4-(ethoxy)butoxy, 4-(propoxy)butoxy,

[0627] 4-(1-methylethoxy)butoxy, 4-(butoxy)butoxy,

[0628] 4-(1-methylpropoxy)butoxy, 4-(2-methylpropoxy)butoxy or

[0629] 4-(1,1-dimethylethoxy)butoxy;

[0630] C3-C6-alkenyl, and the alkenyl moieties of

[0631] C3-C6-alkenylcarbonyl, C3-C6-alkenyloxy,

[0632] C3-C6-alkenyloxycarbonyl, C3-C6-alkenylaminocarbonyl,

[0633] N—(C3-C6-alkenyl)-N—(C1-C6-alkyl)aminocarbonyl,

[0634] N—(C3-C6-alkenyl)-N—(C1-C6-alkoxy)aminocarbonyl: for example

[0635] prop-1-en-3-yl, but-1-en-4-yl, 1-methylprop-2-en-1-yl,

[0636] 2-methylprop-2-en-1-yl, 2-buten-1-yl, 1-penten-3-yl,

[0637] 1-penten-4-yl, 2-penten-4-yl, 1-methylbut-2-en-1-yl,

[0638] 2-methylbut-2-en-1-yl, 3-methylbut-2-en-1-yl,

[0639] 1-methylbut-3-en-1-yl, 2-methylbut-3-en-1-yl,

[0640] 3-methyl-but-3-en-1-yl, 1,1-dimethylprop-2-en-1-yl,

[0641] 1,2-dimethylprop-2-en-1-yl, 1-ethylprop-2-en-1-yl,

[0642] hex-3-en-1-yl, hex-4-en-1-yl, hex-5-en-1-yl,

[0643] 1-methylpent-3-en-1-yl, 2-methylpent-3-en-1-yl,

[0644] 3-methylpent-3-en-1-yl, 4-methylpent-3-en-1-yl,

[0645] 1-methylpent-4-en-1-yl, 2-methylpent-4-en-1-yl,

[0646] 3-methylpent-4-en-1-yl, 4-methylpent-4-en-1-yl,

[0647] 1,1-dimethylbut-2-en-1-yl, 1,1-dimethylbut-3-en-1-yl,

[0648] 1,2-dimethylbut-2-en-1-yl, 1,2-dimethylbut-3-en-1-yl,

[0649] 1,3-dimethylbut-2-en-1-yl, 1,3-dimethylbut-3-en-1-yl,

[0650] 2,2-dimethylbut-3-en-1-yl, 2,3-dimethylbut-2-en-1-yl,

[0651] 2,3-dimethylbut-3-en-1-yl, 3,3-dimethylbut-2-en-1-yl,

[0652] 1-ethylbut-2-en-1-yl, 1-ethylbut-3-en-1-yl,

[0653] 2-ethylbut-2-en-1-yl, 2-ethylbut-3-en-1-yl,

[0654] 1,1,2-trimethylprop-2-en-1-yl, 1-ethyl-1-methylprop-2-en-1-yl

[0655] or 1-ethyl-2-methylprop-2-en-1-yl;

[0656] C2-C6-alkenyl, and the alkenyl moieties of C2-C6-alkenylcarbonyl, phenyl-C2-C6-alkenylcarbonyl and heterocyclyl-C2-C6-alkenylcarbonyl: C3-C6-alkenyl as mentioned above, and also ethenyl;

[0657] C3-C6-haloalkenyl: a C3-C6-alkenyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example,

[0658] 2-chloroallyl, 3-chloroallyl, 2,3-dichloroallyl,

[0659] 3,3-dichloroallyl, 2,3,3-trichloroallyl,

[0660] 2,3-dichlorobut-2-enyl, 2-bromoallyl, 3-bromoallyl,

[0661] 2,3-dibromoallyl, 3,3-dibromoallyl, 2,3,3-tribromoallyl or

[0662] 2,3-dibromobut-2-enyl;

[0663] C3-C6-alkynyl, and the alkynyl moieties of

[0664] C3-C6-alkynylcarbonyl, C3-C6-alkynyloxy,

[0665] C3-C6-alkynyloxycarbonyl, C3-C6-alkynylaminocarbonyl,

[0666] N—(C3-C6-alkynyl)-N—(C1-C6-alkyl)aminocarbonyl,

[0667] N—(C3-C6-alkynyl)-N—(C1-C6-alkoxy)aminocarbonyl: for example

[0668] propargyl, but-1-yn-3-yl, but-1-yn-4-yl, but-2-yn-1-yl,

[0669] pent-1-yn-3-yl, pent-1-yn-4-yl, pent-1-yn-5-yl,

[0670] pent-2-yn-1-yl, pent-2-yn-4-yl, pent-2-yn-5-yl,

[0671] 3-methylbut-1-yn-3-yl, 3-methylbut-1-yn-4-yl, hex-1-yn-3-yl,

[0672] hex-1-yn-4-yl, hex-1-yn-5-yl, hex-1-yn-6-yl, hex-2-yn-1-yl,

[0673] hex-2-yn-4-yl, hex-2-yn-5-yl, hex-2-yn-6-yl, hex-3-yn-1-yl,

[0674] hex-3-yn-2-yl, 3-methylpent-1-yn-3-yl,

[0675] 3-methylpent-1-yn-4-yl, 3-methylpent-1-yn-5-yl,

[0676] 4-methylpent-2-yn-4-yl or 4-methylpent-2-yn-5-yl;

[0677] C2-C6-alkynyl, and the alkynyl moieties of C2-C6-alkynylcarbonyl: C3-C6-alkynyl as mentioned above, and also ethynyl;

[0678] C3-C6-haloalkynyl: a C3-C6-alkynyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example,

[0679] 1,1-difluoroprop-2-yn-1-yl, 3-iodoprop-2-yn-1-yl,

[0680] 4-fluorobut-2-yn-1-yl, 4-chlorobut-2-yn-1-yl,

[0681] 1,1-difluorobut-2-yn-1-yl, 4-iodobut-3-yn-1-yl,

[0682] 5-fluoropent-3-yn-1-yl, 5-iodopent-4-yn-1-yl,

[0683] 6-fluorohex-4-yn-1-yl or 6-iodohex-5-yn-1-yl;

[0684] C1-C6-alkanediyl: methanediyl, ethane-1,1-diyl,

[0685] ethane-1,2-diyl, propane-1,1-diyl, propane-1,2-diyl,

[0686] propane-1,3-diyl, propane-2,2-diyl, butane-1,1-diyl,

[0687] butane-1,2-diyl, butane-1,3-diyl, butane-1,4-diyl,

[0688] 2-methylpropane-1,3-diyl, 2-methylpropane-1,2-diyl,

[0689] 2-methylpropane-1,1-diyl, 1-methylpropane-1,2-diyl,

[0690] 1-methylpropane-2,2-diyl, 1-methylpropane-1,1-diyl,

[0691] pentane-1,1-diyl, pentane-1,2-diyl, pentane-1,3-diyl,

[0692] pentane-1,5-diyl, pentane-2,3-diyl, pentane-2,2-diyl,

[0693] 1-methylbutane-1,1-diyl, 1-methylbutane-1,2-diyl,

[0694] 1-methylbutane-1,3-diyl, 1-methylbutane-1,4-diyl,

[0695] 2-methylbutane-1,1-diyl, 2-methylbutane-1,2-diyl,

[0696] 2-methylbutane-1,3-diyl, 2-methylbutane-1,4-diyl,

[0697] 2,2-dimethylpropane-1,1-diyl, 2,2-dimethylpropane-1,3-diyl,

[0698] 1,1-dimethylpropane-1,3-diyl, 1,1-dimethylpropane-1,2-diyl,

[0699] 2,3-dimethylpropane-1,3-diyl, 2,3-dimethylpropane-1,2-diyl,

[0700] 1,3-dimethylpropane-1,3-diyl, hexane-1,1-diyl,

[0701] hexane-1,2-diyl, hexane-1,3-diyl, hexane-1,4-diyl,

[0702] hexane-1,5-diyl, hexane-1,6-diyl, hexane-2,5-diyl,

[0703] 2-methylpentane-1,1-diyl, 1-methylpentane-1,2-diyl,

[0704] 1-methylpentane-1,3-diyl, 1-methylpentane-1,4-diyl,

[0705] 1-methylpentane-1,5-diyl, 2-methylpentane-1,1-diyl,

[0706] 2-methylpentane-1,2-diyl, 2-methylpentane-1,3-diyl,

[0707] 2-methylpentane-1,4-diyl, 2-methylpentane-1,5-diyl,

[0708] 3-methylpentane-1,1-diyl, 3-methylpentane-1,2-diyl,

[0709] 3-methylpentane-1,3-diyl, 3-methylpentane-1,4-diyl,

[0710] 3-methylpentane-1,5-diyl, 1,1-dimethylbutane-1,2-diyl,

[0711] 1,1-dimethylbutane-1,3-diyl, 1,1-dimethylbutane-1,4-diyl,

[0712] 1,2-dimethylbutane-1,1-diyl, 1,2-dimethylbutane-1,2-diyl,

[0713] 1,2-dimethylbutane-1,3-diyl, 1,2-dimethylbutane-1,4-diyl,

[0714] 1,3-dimethylbutane-1,1-diyl, 1,3-dimethylbutane-1,2-diyl,

[0715] 1,3-dimethylbutane-1,3-diyl, 1,3-dimethylbutane-1,4-diyl,

[0716] 1-ethylbutane-1,1-diyl, 1-ethylbutane-1,2-diyl,

[0717] 1-ethylbutane-1,3-diyl, 1-ethylbutane-1,4-diyl,

[0718] 2-ethylbutane-1,1-diyl, 2-ethylbutane-1,2-diyl,

[0719] 2-ethylbutane-1,3-diyl, 2-ethylbutane-1,4-diyl,

[0720] 2-ethylbutane-2,3-diyl, 2,2-dimethylbutane-1,1-diyl,

[0721] 2,2-dimethylbutane-1,3-diyl, 2,2-dimethylbutane-1,4-diyl,

[0722] 1-isopropylpropane-1,1-diyl, 1-isopropylpropane-1,2-diyl,

[0723] 1-isopropylpropane-1,3-diyl, 2-isopropylpropane-1,1-diyl,

[0724] 2-isopropylpropane-1,2-diyl, 2-isopropylpropane-1,3-diyl,

[0725] 1,2,3-trimethylpropane-1,1-diyl, 1,2,3-trimethylpropane1,2-diyl or 1,2,3-trimethylpropane-1,3-diyl;

[0726] C2-C6-alkenediyl: ethene-1,1-diyl, ethene-1,2-diyl,

[0727] 1-propene-1,1-diyl, 1-propene-1,2-diyl, 1-propene-1,3-diyl,

[0728] 2-propene-1,1-diyl, 2-propene-1,2-diyl, 2-propene-1,3-diyl,

[0729] 1-butene-1,1-diyl, 1-butene-1,2-diyl, 1-butene-1,3-diyl,

[0730] 1-butene-1,4-diyl, 2-butene-1,1-diyl, 2-butene-1,2-diyl,

[0731] 2-butene-1,3-diyl, 2-butene-1,4-diyl, 3-butene-1,1-diyl,

[0732] 3-butene-1,2-diyl, 3-butene-1,3-diyl, 3-butene-1,4-diyl,

[0733] 1-methyl-1-propene-1,2-diyl, 1-methyl-1-propene-1,3-diyl,

[0734] 1-methyl-2-propene-1,1-diyl, 1-methyl-2-propene-1,2-diyl,

[0735] 1-methyl-2-propene-1,3-diyl, 2-methyl-1,1-propene-1,1-diyl,

[0736] 2-methyl-1-propene-1,3-diyl, 3-butene-1,1-diyl,

[0737] 3-butene-1,2-diyl, 3-butene-1,3-diyl, 3-butene-1,4-diyl,

[0738] 1-pentene-1,1-diyl, 1-pentene-1,2-diyl, 1-pentene-1,3-diyl,

[0739] 1-pentene-1,4-diyl, 1-pentene-1,5-diyl, 1-hexene-1,1-diyl,

[0740] 1-hexene-1,2-diyl, 1-hexene-1,3-diyl, 1-hexene-1,4-diyl,

[0741] 1-hexene-1,5-diyl or 1-hexene-1,6-diyl;

[0742] C2-C6-alkadienediyl: 1,3-butadiene-1,1-diyl,

[0743] 1,3-butadiene-1,2-diyl, 1,3-butadiene-1,3-diyl,

[0744] 1,3-butadiene-1,4-diyl, 1,3-pentadiene-1,1-diyl,

[0745] 1,3-pentadiene-1,2-diyl, 1,3-pentadiene-1,3-diyl,

[0746] 1,3-pentadiene-1,4-diyl, 1,3-pentadiene-1,5-diyl,

[0747] 2,4-pentadiene-1,1-diyl, 2,4-pentadiene-1,2-diyl,

[0748] 2,4-pentadiene-1,3-diyl, 2,4-pentadiene-1,4-diyl,

[0749] 2,4-pentadiene-1,5-diyl, 1-methyl-1,3-butadiene-1,4-diyl,

[0750] 1,3-hexadiene-1,1-diyl, 1,3-hexadiene-1,2-diyl,

[0751] 1,3-hexadiene-1,3-diyl, 1,3-hexadiene-1,4-diyl,

[0752] 1,3-hexadiene-1,5-diyl, 1,3-hexadiene-1,6-diyl,

[0753] 1-methyl-1,3-pentadiene-1,2-diyl, 1-methyl-1,3-pentadiene-1,3-diyl, 1-methyl-1,3-pentadiene-1,4-diyl or

[0754] 1-methyl-1,3-pentadiene-1,5-diyl;

[0755] C2-C6-alkynediyl: ethyne-1,2-diyl, 1-propyne-1,3-diyl,

[0756] 2-propyne-1,1-diyl, 2-propyne-1,3-diyl, 1-butyne-1,3-diyl,

[0757] 1-butyne-1,4-diyl, 2-butyne-1,1-diyl, 2-butyne-1,4-diyl,

[0758] 1-methyl-2-propyne-1,1-diyl, 1-methyl-2-propyne-1,3-diyl,

[0759] 1-pentyne-1,3-diyl, 1-pentyne-1,4-diyl, 1-pentyne-1,5-diyl,

[0760] 2-pentyne-1,1-diyl, 2-pentyne-1,4-diyl, 2-pentyne-1,5-diyl,

[0761] 3-pentyne-1,1-diyl, 3-pentyne-1,2-diyl, 3-pentyne-1,5-diyl,

[0762] 4-pentyne-1,1-diyl, 4-pentyne-1,2-diyl, 4-pentyne-1,3-diyl,

[0763] 4-pentyne-1,5-diyl, 1-hexyne-1,3-diyl, 1-hexyne-1,4-diyl,

[0764] 1-hexyne-1,5-diyl, 1-hexyne-1,6-diyl, 2-hexyne-1,1-diyl,

[0765] 2-hexyne-1,4-diyl, 2-hexyne-1,5-diyl, 2-hexyne-1,6-diyl,

[0766] 3-hexyne-1,1-diyl, 3-hexyne-1,2-diyl, 3-hexyne-1,5-diyl,

[0767] 3-hexyne-1,6-diyl, 4-hexyne-1,1-diyl, 4-hexyne-1,2-diyl,

[0768] 4-hexyne-1,3-diyl, 4-hexyne-1,6-diyl, 5-hexyne-1,1-diyl,

[0769] 5-hexyne-1,2-diyl, 5-hexyne-1,3-diyl, 5-hexyne-1,4-diyl or

[0770] 5-hexyne-1,6-diyl;

[0771] C3-C6-cycloalkyl, and the cycloalkyl moieties of C3-C6-cycloalkylamino and C3-C6-cycloalkylcarbonyl: for example cyclopropyl, cyclobutyl, cyclopentyl or cyclohexyl;

[0772] aryl is understood as meaning carbocyclic aromatic compounds such as phenyl or naphthyl;

[0773] a 3- to 7-membered heterocycle is understood as meaning a saturated, partially saturated or unsaturated 3-, 4-, 5-, 6- or 7-membered heterocyclic ring which contains one, two, three or four identical or different heteroatoms selected from the following group: oxygen, sulfur or nitrogen, i.e., for example,

[0774] C-bonded 5-membered rings such as:

[0775] tetrahydrofuran-2-yl, tetrahydrofuran-3-yl,

[0776] tetrahydrothien-2-yl, tetrahydrothien-3-yl,

[0777] tetrahydropyrrol-2-yl, tetrahydropyrrol-3-yl,

[0778] 2,3-dihydrofuran-2-yl, 2,3-dihydrofuran-3-yl,

[0779] 2,5-dihydrofuran-2-yl, 2,5-dihydrofuran-3-yl,

[0780] 4,5-dihydrofuran-2-yl, 4,5-dihydrofuran-3-yl,

[0781] 2,3-dihydrothien-2-yl, 2,3-dihydrothien-3-yl,

[0782] 2,5-dihydrothien-2-yl, 2,5-dihydrothien-3-yl,

[0783] 4,5-dihydrothien-2-yl, 4,5-dihydrothien-3-yl,

[0784] 2,3-dihydro-1H-pyrrol-2-yl, 2,3-dihydro-1H-pyrrol-3-yl,

[0785] 2,5-dihydro-1H-pyrrol-2-yl, 2,5-dihydro-1H-pyrrol-3-yl,

[0786] 4,5-dihydro-1H-pyrrol-2-yl, 4,5-dihydro-1H-pyrrol-3-yl,

[0787] 3,4-dihydro-2H-pyrrol-2-yl, 3,4-dihydro-2H-pyrrol-3-yl,

[0788] 3,4-dihydro-5H-pyrrol-2-yl, 3,4-dihydro-5H-pyrrol-3-yl,

[0789] 2-furyl, 3-furyl, 2-thienyl, 3-thienyl, pyrrol-2-yl,

[0790] pyrrol-3-yl, tetrahydropyrazol-3-yl, tetrahydropyrazol-4-yl,

[0791] tetrahydroisoxazol-3-yl, tetrahydroisoxazol-4-yl,

[0792] tetrahydroisoxazol-5-yl, 1,2-oxathiolan-3-yl,

[0793] 1,2-oxathiolan-4-yl, 1,2-oxathiolan-5-yl,

[0794] tetrahydroisothiazol-3-yl, tetrahydroisothiazol-4-yl,

[0795] tetrahydroisothiazol-5-yl, 1,2-dithiolan-3-yl,

[0796] 1,2-dithiolan-4-yl, tetrahydroimidazol-2-yl,

[0797] tetrahydroimidazol-4-yl, tetrahydrooxazol-2-yl,

[0798] tetrahydrooxazol-4-yl, tetrahydrooxazol-5-yl,

[0799] tetrahydrothiazol-2-yl, tetrahydrothiazol-4-yl,

[0800] tetrahydrothiazol-5-yl, 1,3-dioxolan-2-yl,

[0801] 1,3-dioxolan-4-yl, 1,3-oxathiolan-2-yl, 1,3-oxathiolan-4-yl,

[0802] 1,3-oxathiolan-5-yl, 1,3-dithiolan-2-yl, 1,3-dithiolan-4-yl,

[0803] 4,5-dihydro-1H-pyrazol-3-yl, 4,5-dihydro-1H-pyrazol-4-yl,

[0804] 4,5-dihydro-1H-pyrazol-5-yl, 2,5-dihydro-1H-pyrazol-3-yl,

[0805] 2,5-dihydro-1H-pyrazol-4-yl, 2,5-dihydro-1H-pyrazol-5-yl,

[0806] 4,5-dihydroisoxazol-3-yl, 4,5-dihydroisoxazol-4-yl,

[0807] 4,5-dihydroisoxazol-5-yl, 2,5-dihydroisoxazol-3-yl,

[0808] 2,5-dihydroisoxazol-4-yl, 2,5-dihydroisoxazol-5-yl,

[0809] 2,3-dihydroisoxazol-3-yl, 2,3-dihydroisoxazol-4-yl,

[0810] 2,3-dihydroisoxazol-5-yl, 4,5-dihydroisothiazol-3-yl,

[0811] 4,5-dihydroisothiazol-4-yl, 4,5-dihydroisothiazol-5-yl,

[0812] 2,5-dihydroisothiazol-3-yl, 2,5-dihydroisothiazol-4-yl,

[0813] 2,5-dihydroisothiazol-5-yl, 2,3-dihydroisothiazol-3-yl,

[0814] 2,3-dihydroisothiazol-4-yl, 2,3-dihydroisothiazol-5-yl,

[0815] Δ3-1,2-dithiol-3-yl, Δ3-1,2-dithiol-4-yl,

[0816] Δ3-1,2-dithiol-5-yl, 4,5-dihydro-1H-imidazol-2-yl,

[0817] 4,5-dihydro-1H-imidazol-4-yl, 4,5-dihydro-1H-imidazol-5-yl,

[0818] 2,5-dihydro-1H-imidazol-2-yl, 2,5-dihydro-1H-imidazol-4-yl,

[0819] 2,5-dihydro-1H-imidazol-5-yl, 2,3-dihydro-1H-imidazol-2-yl,

[0820] 2,3-dihydro-1H-imidazol-4-yl, 4,5-dihydrooxazol-2-yl,

[0821] 4,5-dihydrooxazol-4-yl, 4,5-dihydrooxazol-5-yl,

[0822] 2,5-dihydrooxazol-2-yl, 2,5-dihydrooxazol-4-yl,

[0823] 2,5-dihydrooxazol-5-yl, 2,3-dihydrooxazol-2-yl,

[0824] 2,3-dihydrooxazol-4-yl, 2,3-dihydrooxazol-5-yl,

[0825] 4,5-dihydrothiazol-2-yl, 4,5-dihydrothiazol-4-yl,

[0826] 4,5-dihydrothiazol-5-yl, 2,5-dihydrothiazol-2-yl,

[0827] 2,5-dihydrothiazol-4-yl, 2,5-dihydrothiazol-5-yl,

[0828] 2,3-dihydrothiazol-2-yl, 2,3-dihydrothiazol-4-yl,

[0829] 2,3-dihydrothiazol-5-yl, 1,3-dioxol-2-yl, 1,3-dioxol-4-yl,

[0830] 1,3-dithiol-2-yl, 1,3-dithiol-4-yl, 1,3-oxathiol-2-yl,

[0831] 1,3-oxathiol-4-yl, 1,3-oxathiol-5-yl, pyrazol-3-yl,

[0832] pyrazol-4-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl,

[0833] isothiazol-3-yl, isothiazol-4-yl, isothiazol-5-yl,

[0834] imidazol-2-yl, imidazol-4-yl, oxazol-2-yl, oxazol-4-yl,

[0835] oxazol-5-yl, thiazol-2-yl, thiazol-4-yl, thiazol-5-yl,

[0836] 1,2,3-Δ2-oxadiazolin-4-yl, 1,2,3-Δ2-oxadiazolin-5-yl,

[0837] 1,2,4-Δ4-oxadiazolin-3-yl, 1,2,4-Δ4-oxadiazolin-5-yl,

[0838] 1,2,4-Δ2-oxadiazolin-3-yl, 1,2,4-Δ2-oxadiazolin-5-yl,

[0839] 1,2,4-Δ3-oxadiazolin-3-yl, 1,2,4-Δ3-oxadiazolin-5-yl,

[0840] 1,3,4-Δ2-oxadiazolin-2-yl, 1,3,4-Δ2-oxadiazolin-5-yl,

[0841] 1,3,4-Δ3-oxadiazolin-2-yl, 1,3,4-oxadiazolin-2-yl,

[0842] 1,2,4-Δ4-thiadiazolin-3-yl, 1,2,4-Δ4-thiadiazolin-5-yl,

[0843] 1,2,4-Δ3-thiadiazolin-3-yl, 1,2,4-Δ3-thiadiazolin-5-yl,

[0844] 1,2,4-Δ2-thiadiazolin-3-yl, 1,2,4-Δ2-thiadiazolin-5-yl,

[0845] 1,3,4-Δ2-thiadiazolin-2-yl, 1,3,4-Δ2-thiadiazolin-5-yl,

[0846] 1,3,4-Δ3-thiadiazolin-2-yl, 1,3,4-thiadiazolin-2-yl,

[0847] 1,3,2-dioxathiolan-4-yl, 1,2,3-Δ2-triazolin-4-yl,

[0848] 1,2,3-Δ2-triazolin-5-yl, 1,2,4-Δ2-triazolin-3-yl,

[0849] 1,2,4-Δ2-triazolin-5-yl, 1,2,4-Δ3-triazolin-3-yl,

[0850] 1,2,4-Δ3-triazolin-5-yl, 1,2,4-Δ1-triazolin-2-yl,

[0851] 1,2,4-triazolin-3-yl, 3H-1,2,4-dithiazol-5-yl,

[0852] 2H-1,3,4-dithiazol-5-yl, 2H-1,3,4-oxathiazol-5-yl,

[0853] 1,2,3-oxadiazol-4-yl, 1,2,3-oxadiazol-5-yl,

[0854] 1,2,4-oxadiazol-3-yl, 1,2,4-oxadiazol-5-yl,

[0855] 1,3,4-oxadiazol-2-yl, 1,2,3-thiadiazol-4-yl,

[0856] 1,2,3-thiadiazol-5-yl, 1,2,4-thiadiazol-3-yl,

[0857] 1,2,4-thiadiazol-5-yl, 1,3,4-thiadiazol-2-yl,

[0858] 1,2,3-triazol-4-yl, 1,2,4-triazol-3-yl, tetrazol-5-yl;

[0859] C-bonded 6-membered rings such as:

[0860] tetrahydropyran-2-yl, tetrahydropyran-3-yl,

[0861] tetrahydropyran-4-yl, piperidin-2-yl, piperidin-3-yl,

[0862] piperidin-4-yl, tetrahydrothiopyran-2-yl,

[0863] tetrahydrothiopyran-3-yl, tetrahydrothiopyran-4-yl,

[0864] 2H-3,4-dihydropyran-6-yl, 2H-3,4-dihydropyran-5-yl,

[0865] 2H-3,4-dihydropyran-4-yl, 2H-3,4-dihydropyran-3-yl,

[0866] 2H-3,4-dihydropyran-2-yl, 2H-3,4-dihydropyran-6-yl,

[0867] 2H-3,4-dihydrothiopyran-5-yl, 2H-3,4-dihydrothiopyran-4-yl,

[0868] 2H-3,4-dihydropyran-3-yl, 2H-3,4-dihydropyran-2-yl,

[0869] 1,2,3,4-tetrahydropyridin-6-yl,

[0870] 1,2,3,4-tetrahydropyridin-5-yl,

[0871] 1,2,3,4-tetrahydropyridin-4-yl,

[0872] 1,2,3,4-tetrahydropyridin-3-yl,

[0873] 1,2,3,4-tetrahydropyridin-2-yl, 2H-5,6-dihydropyran-2-yl,

[0874] 2H-5,6-dihydropyran-3-yl, 2H-5,6-dihydropyran-4-yl,

[0875] 2H-5,6-dihydropyran-5-yl, 2H-5,6-dihydropyran-6-yl,

[0876] 2H-5,6-dihydrothiopyran-2-yl, 2H-5,6-dihydrothiopyran-3-yl,

[0877] 2H-5,6-dihydrothiopyran-4-yl, 2H-5,6-dihydrothiopyran-5-yl,

[0878] 2H-5,6-dihydrothiopyran-6-yl, 1,2,5,6-tetrahydropyridin-2-yl,

[0879] 1,2,5,6-tetrahydropyridin-3-yl,

[0880] 1,2,5,6-tetrahydropyridin-4-yl,

[0881] 1,2,5,6-tetrahydropyridin-5-yl,

[0882] 1,2,5,6-tetrahydropyridin-6-yl,

[0883] 2,3,4,5-tetrahydropyridin-2-yl,

[0884] 2,3,4,5-tetrahydropyridin-3-yl,

[0885] 2,3,4,5-tetrahydropyridin-4-yl,

[0886] 2,3,4,5-tetrahydropyridin-5-yl,

[0887] 2,3,4,5-tetrahydropyridin-6-yl, 4H-pyran-2-yl, 4H-pyran-3-yl,

[0888] 4H-pyran-4-yl, 4H-thiopyran-2-yl, 4H-thiopyran-3-yl,

[0889] 4H-thiopyran-4-yl, 1,4-dihydropyridin-2-yl,

[0890] 1,4-dihydropyridin-3-yl, 1,4-dihydropyridin-4-yl,

[0891] 2H-pyran-2-yl, 2H-pyran-3-yl, 2H-pyran-4-yl, 2H-pyran-5-yl,

[0892] 2H-pyran-6-yl, 2H-thiopyran-2-yl, 2H-thiopyran-3-yl,

[0893] 2H-thiopyran-4-yl, 2H-thiopyran-5-yl, 2H-thiopyran-6-yl,

[0894] 1,2-dihydropyridin-2-yl, 1,2-dihydropyridin-3-yl,

[0895] 1,2-dihydropyridin-4-yl, 1,2-dihydropyridin-5-yl,

[0896] 1,2-dihydropyridin-6-yl, 3,4-dihydropyridin-2-yl,

[0897] 3,4-dihydropyridin-3-yl, 3,4-dihydropyridin-4-yl,

[0898] 3,4-dihydropyridin-5-yl, 3,4-dihydropyridin-6-yl,

[0899] 2,5-dihydropyridin-2-yl, 2,5-dihydropyridin-3-yl,

[0900] 2,5-dihydropyridin-4-yl, 2,5-dihydropyridin-5-yl,

[0901] 2,5-dihydropyridin-6-yl, 2,3-dihydropyridin-2-yl,

[0902] 2,3-dihydropyridin-3-yl, 2,3-dihydropyridin-4-yl,

[0903] 2,3-dihydropyridin-5-yl, 2,3-dihydropyridin-6-yl,

[0904] pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, 1,3-dioxan-2-yl,

[0905] 1,3-dioxan-4-yl, 1,3-dioxan-5-yl, 1,4-dioxan-2-yl,

[0906] 1,3-dithian-2-yl, 1,3-dithian-4-yl, 1,3-dithian-5-yl,

[0907] 1,4-dithian-2-yl, 1,3-oxathian-2-yl, 1,3-oxathian-4-yl,

[0908] 1,3-oxathian-5-yl, 1,3-oxathian-6-yl, 1,4-oxathian-2-yl,

[0909] 1,4-oxathian-3-yl, 1,2-dithian-3-yl, 1,2-dithian-4-yl,

[0910] hexahydropyrimidin-2-yl, hexahydropyrimidin-4-yl,

[0911] hexahydropyrimidin-5-yl, hexahydropyrazin-2-yl,

[0912] hexahydropyridazin-3-yl, hexahydropyridazin-4-yl,

[0913] tetrahydro-1,3-oxazin-2-yl, tetrahydro-1,3-oxazin-4-yl,

[0914] tetrahydro-1,3-oxazin-5-yl, tetrahydro-1,3-oxazin-6-yl,

[0915] tetrahydro-1,3-thiazin-2-yl, tetrahydro-1,3-thiazin-4-yl,

[0916] tetrahydro-1,3-thiazin-5-yl, tetrahydro-1,3-thiazin-6-yl,

[0917] tetrahydro-1,4-thiazin-2-yl, tetrahydro-1,4-thiazin-3-yl,

[0918] tetrahydro-1,4-oxazin-2-yl, tetrahydro-1,4-oxazin-3-yl,

[0919] tetrahydro-1,2-oxazin-3-yl, tetrahydro-1,2-oxazin-4-yl,

[0920] tetrahydro-1,2-oxazin-5-yl, tetrahydro-1,2-oxazin-6-yl,

[0921] 2H-5,6-dihydro-1,2-oxazin-3-yl,

[0922] 2H-5,6-dihydro-1,2-oxazin-4-yl,

[0923] 2H-5,6-dihydro-1,2-oxazin-5-yl,

[0924] 2H-5,6-dihydro-1,2-oxazin-6-yl,

[0925] 2H-5,6-dihydro-1,2-thiazin-3-yl,

[0926] 2H-5,6-dihydro-1,2-thiazin-4-yl,

[0927] 2H-5,6-dihydro-1,2-thiazin-5-yl,

[0928] 2H-5,6-dihydro-1,2-thiazin-6-yl,

[0929] 4H-5,6-dihydro-1,2-oxazin-3-yl,

[0930] 4H-5,6-dihydro-1,2-oxazin-4-yl,

[0931] 4H-5,6-dihydro-1,2-oxazin-5-yl,

[0932] 4H-5,6-dihydro-1,2-oxazin-6-yl,

[0933] 4H-5,6-dihydro-1,2-thiazin-3-yl,

[0934] 4H-5,6-dihydro-1,2-thiazin-4-yl,

[0935] 4H-5,6-dihydro-1,2-thiazin-5-yl,

[0936] 4H-5,6-dihydro-1,2-thiazin-6-yl,

[0937] 2H-3,6-dihydro-1,2-oxazin-3-yl,

[0938] 2H-3,6-dihydro-1,2-oxazin-4-yl,

[0939] 2H-3,6-dihydro-1,2-oxazin-5-yl,

[0940] 2H-3,6-dihydro-1,2-oxazin-6-yl,

[0941] 2H-3,6-dihydro-1,2-thiazin-3-yl,

[0942] 2H-3,6-dihydro-1,2-thiazin-4-yl,

[0943] 2H-3,6-dihydro-1,2-thiazin-5-yl,

[0944] 2H-3,6-dihydro-1,2-thiazin-6-yl,

[0945] 2H-3,4-dihydro-1,2-oxazin-3-yl,

[0946] 2H-3,4-dihydro-1,2-oxazin-4-yl,

[0947] 2H-3,4-dihydro-1,2-oxazin-5-yl,

[0948] 2H-3,4-dihydro-1,2-oxazin-6-yl,

[0949] 2H-3,4-dihydro-1,2-thiazin-3-yl,

[0950] 2H-3,4-dihydro-1,2-thiazin-4-yl,

[0951] 2H-3,4-dihydro-1,2-thiazin-5-yl,

[0952] 2H-3,4-dihydro-1,2-thiazin-6-yl,

[0953] 2,3,4,5-tetrahydropyridazin-3-yl,

[0954] 2,3,4,5-tetrahydropyridazin-4-yl,

[0955] 2,3,4,5-tetrahydropyridazin-5-yl,

[0956] 2,3,4,5-tetrahydropyridazin-6-yl,

[0957] 3,4,5,6-tetrahydropyridazin-3-yl,

[0958] 3,4,5,6-tetrahydropyridazin-4-yl,

[0959] 1,2,5,6-tetrahydropyridazin-3-yl,

[0960] 1,2,5,6-tetrahydropyridazin-4-yl,

[0961] 1,2,5,6-tetrahydropyridazin-5-yl,

[0962] 1,2,5,6-tetrahydropyridazin-6-yl,

[0963] 1,2,3,6-tetrahydropyridazin-3-yl,

[0964] 1,2,3,6-tetrahydropyridazin-4-yl,

[0965] 4H-5,6-dihydro-1,3-oxazin-2-yl,

[0966] 4H-5,6-dihydro-1,3-oxazin-4-yl,

[0967] 4H-5,6-dihydro-1,3-oxazin-5-yl,

[0968] 4H-5,6-dihydro-1,3-oxazin-6-yl,

[0969] 4H-5,6-dihydro-1,3-thiazin-2-yl,

[0970] 4H-5,6-dihydro-1,3-thiazin-4-yl,

[0971] 4H-5,6-dihydro-1,3-thiazin-5-yl,

[0972] 4H-5,6-dihydro-1,3-thiazin-6-yl,

[0973] 3,4,5,6-tetrahydropyrimidin-2-yl,

[0974] 3,4,5,6-tetrahydropyrimidin-4-yl,

[0975] 3,4,5,6-tetrahydropyrimidin-5-yl,

[0976] 3,4,5,6-tetrahydropyrimidin-6-yl,

[0977] 1,2,3,4-tetrahydropyrazin-2-yl,

[0978] 1,2,3,4-tetrahydropyrazin-5-yl,

[0979] 1,2,3,4-tetrahydropyrimidin-2-yl,

[0980] 1,2,3,4-tetrahydropyrimidin-4-yl,

[0981] 1,2,3,4-tetrahydropyrimidin-5-yl,

[0982] 1,2,3,4-tetrahydropyrimidin-6-yl,

[0983] 2,3-dihydro-1,4-thiazin-2-yl, 2,3-dihydro-1,4-thiazin-3-yl,

[0984] 2,3-dihydro-1,4-thiazin-5-yl, 2,3-dihydro-1,4-thiazin-6-yl,

[0985] 2H-1,2-oxazin-3-yl, 2H-1,2-oxazin-4-yl, 2H-1,2-oxazin-5-yl,

[0986] 2H-1,2-oxazin-6-yl, 2H-1,2-thiazin-3-yl, 2H-1,2-thiazin-4-yl,

[0987] 2H-1,2-thiazin-5-yl, 2H-1,2-thiazin-6-yl, 4H-1,2-oxazin-3-yl,

[0988] 4H-1,2-oxazin-4-yl, 4H-1,2-oxazin-5-yl, 4H-1,2-oxazin-6-yl,

[0989] 4H-1,2-thiazin-3-yl, 4H-1,2-thiazin-4-yl,

[0990] 4H-1,2-thiazin-5-yl, 4H-1,2-thiazin-6-yl, 6H-1,2-oxazin-3-yl,

[0991] 6H-1,2-oxazin-4-yl, 6H-1,2-oxazin-5-yl, 6H-1,2-oxazin-6-yl,

[0992] 6H-1,2-thiazin-3-yl, 6H-1,2-thiazin-4-yl,

[0993] 6H-1,2-thiazin-5-yl, 6H-1,2-thiazin-6-yl, 2H-1,3-oxazin-2-yl,

[0994] 2H-1,3-oxazin-4-yl, 2H-1,3-oxazin-5-yl, 2H-1,3-oxazin-6-yl,

[0995] 2H-1,3-thiazin-2-yl, 2H-1,3-thiazin-4-yl,

[0996] 2H-1,3-thiazin-5-yl, 2H-1,3-thiazin-6-yl, 4H-1,3-oxazin-2-yl,

[0997] 4H-1,3-oxazin-4-yl, 4H-1,3-oxazin-5-yl, 4H-1,3-oxazin-6-yl,

[0998] 4H-1,3-thiazin-2-yl, 4H-1,3-thiazin-4-yl,

[0999] 4H-1,3-thiazin-5-yl, 4H-1,3-thiazin-6-yl, 6H-1,3-oxazin-2-yl,

[1000] 6H-1,3-oxazin-4-yl, 6H-1,3-oxazin-5-yl, 6H-1,3-oxazin-6-yl,

[1001] 6H-1,3-thiazin-2-yl, 6H-1,3-oxazin-4-yl, 6H-1,3-oxazin-5-yl,

[1002] 6H-1,3-thiazin-6-yl, 2H-1,4-oxazin-2-yl, 2H-1,4-oxazin-3-yl,

[1003] 2H-1,4-oxazin-5-yl, 2H-1,4-oxazin-6-yl, 2H-1,4-thiazin-2-yl,

[1004] 2H-1,4-thiazin-3-yl, 2H-1,4-thiazin-5-yl,

[1005] 2H-1,4-thiazin-6-yl, 4H-1,4-oxazin-2-yl, 4H-1,4-oxazin-3-yl,

[1006] 4H-1,4-thiazin-2-yl, 4H-1,4-thiazin-3-yl,

[1007] 1,4-dihydropyridazin-3-yl, 1,4-dihydropyridazin-4-yl,

[1008] 1,4-dihydropyridazin-5-yl, 1,4-dihydropyridazin-6-yl,

[1009] 1,4-dihydropyrazin-2-yl, 1,2-dihydropyrazin-2-yl,

[1010] 1,2-dihydropyrazin-3-yl, 1,2-dihydropyrazin-5-yl,

[1011] 1,2-dihydropyrazin-6-yl, 1,4-dihydropyrimidin-2-yl,

[1012] 1,4-dihydropyrimidin-4-yl, 1,4-dihydropyrimidin-5-yl,

[1013] 1,4-dihydropyrimidin-6-yl, 3,4-dihydropyrimidin-2-yl,

[1014] 3,4-dihydropyrimidin-4-yl, 3,4-dihydropyrimidin-5-yl,

[1015] 3,4-dihydropyrimidin-6-yl, pyridazin-3-yl, pyridazin-4-yl,

[1016] pyrimidin-2-yl, pyrimidin-4-yl, pyrimidin-5-yl, pyrazin-2-yl,

[1017] 1,3,5-triazin-2-yl, 1,2,4-triazin-3-yl, 1,2,4-triazin-5-yl,

[1018] 1,2,4-triazin-6-yl or 1,2,4,5-tetrazin-3-yl;

[1019] +P2

[1020] N-bonded 5-membered rings such as:

[1021] tetrahydropyrrol-1-yl, 2,3-dihydro-1H-pyrrol-1-yl,

[1022] 2,5-dihydro-1H-pyrrol-1-yl, pyrrol-1-yl,

[1023] tetrahydropyrazol-1-yl, tetrahydroisoxazol-2-yl,

[1024] tetrahydroisothiazol-2-yl, tetrahydroimidazol-1-yl,

[1025] tetrahydrooxazol-3-yl, tetrahydrothiazol-3-yl,

[1026] 4,5-dihydro-1H-pyrazol-1-yl, 2,5-dihydro-1H-pyrazol-1-yl,

[1027] 2,3-dihydro-1H-pyrazol-1-yl, 2,5-dihydroisoxazol-2-yl,

[1028] 2,3-dihydroisoxazol-2-yl, 2,5-dihydroisothiazol-2-yl,

[1029] 2,3-dihydroisoxazol-2-yl, 4,5-dihydro-1H-imidazol-1-yl,

[1030] 2,5-dihydro-1H-imidazol-1-yl, 2,3-dihydro-1H-imidazol-1-yl,

[1031] 2,3-dihydrooxazol-3-yl, 2,3-dihydrothiazol-3-yl,

[1032] pyrazol-1-yl, imidazol-1-yl, 1,2,4-Δ4-oxadiazolin-2-yl,

[1033] 1,2,4-Δ2-oxadiazolin-4-yl, 1,2,4-Δ3-oxadiazolin-2-yl,

[1034] 1,3,4-Δ2-oxadiazolin-4-yl, 1,2,4-Δ5-thiadiazolin-2-yl,

[1035] 1,2,4-Δ3-thiadiazolin-2-yl, 1,2,4-Δ2-thiadiazolin-4-yl,

[1036] 1,3,4-Δ2-thiadiazolin-4-yl, 1,2,3-Δ2-triazolin-1-yl,

[1037] 1,2,4-Δ2-triazolin-1-yl, 1,2,4-Δ2-triazolin-4-yl,

[1038] 1,2,4-Δ3-triazolin-1-yl, 1,2,4-Δ1-triazolin-4-yl,

[1039] 1,2,3-triazol-1-yl, 1,2,4-triazol-1-yl, tetrazol-1-yl;

[1040] N-bonded 6-membered rings such as:

[1041] piperidin-1-yl, 1,2,3,4-tetrahydropyridin-1-yl,

[1042] 1,2,5,6-tetrahydropyridin-1-yl, 1,4-dihydropyridin-1-yl,

[1043] 1,2-dihydropyridin-1-yl, hexahydropyrimidin-1-yl,

[1044] hexahydropyrazin-1-yl, hexahydropyridazin-1-yl,

[1045] tetrahydro-1,3-oxazin-3-yl, tetrahydro-1,3-thiazin-3-yl,

[1046] tetrahydro-1,4-thiazin-4-yl, tetrahydro-1,4-oxazin-4-yl

[1047] (morpholinyl), tetrahydro-1,2-oxazin-2-yl,

[1048] 2H-5,6-dihydro-1,2-oxazin-2-yl,

[1049] 2H-5,6-dihydro-1,2-thiazin-2-yl,

[1050] 2H-3,6-dihydro-1,2-oxazin-2-yl,

[1051] 2H-3,6-dihydro-1,2-thiazin-2-yl,

[1052] 2H-3,4-dihydro-1,2-thiazin-2-yl,

[1053] 2,3,4,5-tetrahydropyridazin-2-yl,

[1054] 1,2,5,6-tetrahydropyridazin-1-yl,

[1055] 1,2,5,6-tetrahydropyridazin-2-yl,

[1056] 1,2,3,6-tetrahydropyridazin-1-yl,

[1057] 3,4,5,6-tetrahydropyrimidin-3-yl,

[1058] 1,2,3,4-tetrahydropyrazin-1-yl,

[1059] 1,2,3,4-tetrahydropyrimidin-1-yl,

[1060] 1,2,3,4-tetrahydropyrimidin-3-yl,

[1061] 2,3-dihydro-1,4-thiazin-4-yl, 2H-1,2-oxazin-2-yl,

[1062] 2H-1,2-thiazin-2-yl, 4H-1,4-oxazin-4-yl, 4H-1,4-thiazin-4-yl,

[1063] 1,4-dihydropyridazin-1-yl, 1,4-dihydropyrazin-1-yl,

[1064] 1,2-dihydropyrazin-1-yl, 1,4-dihydropyrimidin-1-yl or

[1065] 3,4-dihydropyrimidin-3-yl;

[1066] and also N-bonded cyclic imides such as:

[1067] phthalimide, tetrahydrophthalimide, succinimide, maleimide,

[1068] glutarimide, 5-oxotriazolin-1-yl,

[1069] 5-oxo-1,3,4-oxadiazolin-4-yl or

[1070] 2,4-dioxo(1H,3H)pyrimidin-3-yl;

[1071] where, if appropriate, the sulfur of the heterocycles mentioned may be oxidized to S═O or S(═O)2

[1072] and where a bicyclic ring system may be formed with a fused-on phenyl ring or with a C3-C6-carbocycle or with a further 5- to 6-membered heterocycle.

[1073] All phenyl rings or heterocyclyl radicals and all phenyl components in phenoxy, phenylalkyl, phenylcarbonylalkyl, phenylcarbonyl, phenylalkenylcarbonyl, phenoxycarbonyl, phenyloxythiocarbonyl, phenylaminocarbonyl and N-alkyl-N-phenylaminocarbonyl, phenylsulfonyl or phenoxysulfonyl or heterocyclyl components in heterocyclyloxy, heterocyclylalkyl, heterocyclylcarbonylalkyl, heterocyclylcarbonyl, heterocyclyloxythiocarbonyl, heterocyclylalkenylcarbonyl, heterocyclyloxycarbonyl, heterocyclylaminocarbonyl, N-alkyl-N-heterocyclylaminocarbonyl, heterocyclylsulfonyl or heterocyclyloxysulfonyl are, unless stated otherwise, preferably unsubstituted, or they carry one, two or three halogen atoms and/or a nitro group, a cyano radical and/or one or two methyl, trifluoromethyl, methoxy or trifluoromethoxy substituents.

[1074] With respect to the use of the compounds of the formula I according to the invention as herbicides, the variables A, R1 to R15 preferably have the following meanings, in each case on their own or in combination:

[1075] A is S, SO2, O or NR6, where R6 is as defined above. R6 is preferably not hydrogen. R6 is in particular C1-C4-alkyl and very particularly preferably methyl. In a first group of particularly preferred compounds I, A is O or NR6, where R6 is as defined above. In another group of particularly preferred compounds, A is S or SO2.

[1076] R1 is halogen, C1-C4-alkyl, C1-C4-alkoxy, in particular methyl, methoxy or chlorine.

[1077] R2 has the abovementioned meanings other than hydrogen, and is in particular

[1078] C1-C4-alkyl, C1-C4-haloalkyl, hydroxyl, C1-C4-alkoxy,

[1079] C1-C4-alkylsulfonyl, C1-C4-haloalkylsulfonyl, hydroxycarbonyl-C1-C4-alkyl, C(═N—O(—C1-C4-alkyl) )-(C1-C4-alkyl), NH2,

[1080] C1-C4-alkylamino, di(C1-C4-alkyl)amino, phenyl, phenylcarbonyl or benzyl, where the phenyl rings of the three lastmentioned substituents may be substituted by one or two halogen atoms, methoxy groups or methyl groups, cyano, C1-C4-alkylcarbonyl,

[1081] C1-C4-haloalkylcarbonyl, C1-C4-alkoxycarbonyl,

[1082] C1-C4-alkoxycarbonyl-C1-C4-alkyl, C3-C6-alkenyl, C3-C6-alkynyl,

[1083] 1,3-dioxolan-2-yl, 1,3-dithiolan-2-yl, 1,3-dioxan-2-yl,

[1084] 1,3-dithian-2-yl, oxazolin-2-yl, oxazolidin-2-yl,

[1085] 4,5-dihydroisoxazol-3-yl, 4,5-dihydroisoxazol-4-yl,

[1086] isoxazol-3-yl, isoxazol-4-yl, methyl or ethyl substituted by one of the heterocycles mentioned above, such as in

[1087] (1,3-dioxolan-2-yl)methyl, (1,3-dithiolan-2-yl)methyl,

[1088] (1,3-dioxan-2-yl)methyl, (1,3-dithian-2-yl)methyl,

[1089] (oxazolin-2-yl)methyl, (oxazolidin-2-yl)methyl,

[1090] (4,5-dihydroisoxazol-3-yl)methyl,

[1091] (4,5-dihydroisoxazol-4-yl)methyl, (isoxazol-3-yl)methyl,

[1092] (isoxazol-4-yl)methyl, 2-(1,3-dioxolan-2-yl)ethyl,

[1093] 2-(1,3-dithiolan-2-yl)ethyl, 2-(1,3-dioxan-2-yl)ethyl,

[1094] 2-(1,3-dithian-2-yl)ethyl, 2-(oxazolin-2-yl)ethyl,

[1095] 2-(oxazolidin-2-yl)ethyl, 2-(4,5-dihydroisoxazol-3-yl)ethyl,

[1096] (4,5-dihydroisoxazol-4-yl)ethyl, 2-(isoxazol-3-yl)ethyl,

[1097] 2-(isoxazol-4-yl)ethyl, where the abovementioned heterocycles may be mono-, di- or trisubstituted by C1-C4-alkyl, in particular methyl;

[1098] and is especially C1-C4-alkyl, C3-C6-alkenyl, methoxymethyl, CF3, CHF2, CN, OH, OCH3, NH2, NHCH3, N(CH3)2, C1-C4-alkoxycarbonyl, acetyl, trifluoroacetyl, C(═NOCH3)CH3, SO2CH3, SO2CF3, CH2CO2H, C1-C4-alkoxycarbonyl-C1-C4-alkyl, cyclopropyl, cyclopentyl, cyclohexyl, 4,5-dihydroisoxazol-3-yl, 4,5-dihydroisoxazol-4-yl, isoxazol-3-yl, isoxazol-4-yl, where the abovementioned heterocycles may be monosubstituted by methyl, is phenyl, benzyl, benzoyl, 2-pyridyl.

[1099] R2 is particularly preferably C1-C4-alkyl or C3-C6-alkenyl. Particular preference is also given to those compounds I in which R2 is C3-C6-alkynyl, (1,3-dioxolan-2-yl)methyl, 2-(1,3-dioxolan-2-yl)ethyl or benzyl where the phenyl ring may be unsubstituted or carry 1 or 2 substituents, selected from the group consisting of halogen, methyl and methoxy.

[1100] R3 is C1-C4-alkyl, halogen and in particular hydrogen.

[1101] In especially prefered compounds I, A is O or S, R1 is methyl, R3 is hydrogen and R3 is a substituent different from hydrogen, in particular one of the substituents mentioned above as being preferred and specifically C1-C6-alkyl, C3-C6-alkynyl, C3-C6-alkenyl, (1,3-dioxolan-2-yl)methyl, 2-(1,3-dioxolan-2-yl)ethyl or benzyl where the phenyl ring may be unsubstituted or may carry 1 or 2 substituents selected from the group consisting of halogen, methyl and methoxy.

[1102] R7 is hydroxyl, halogen, OR10, SR10, SO2R11, OSO2R11, NR14R15, ONR14R15 or N-bonded heterocyclyl which may be partially or fully halogenated and/or may carry one, two or three of the following radicals: nitro, cyano, C1-C4-alkyl,

[1103] C1-C4-haloalkyl, C1-C4-alkoxy or C1-C4-haloalkoxy; in particular hydroxyl, OR10 and OSO2R11, especially hydroxyl,

[1104] C1-C4-alkyloxy, O—CH2-phenyl, phenylcarbonyloxy, 2-, 3- or

[1105] 4-fluorophenylcarbonyloxy, cyclopropylcarbonyloxy,

[1106] C1-C4-sulfonyloxy, phenylsulfonyloxy and 2-, 3- or

[1107] 4-methylphenylsulfonyloxy;

[1108] R8 is C1-C6-alkyl, C3-C6-cycloalkyl, in particular C1-C4-alkyl and cyclopropyl; and

[1109] R9 is hydrogen or C1-C4-alkyl, in particular hydrogen or C1-C4-alkyl.

[1110] An important group of compounds are those compounds in which R8 is a C3-C6-cycloalkyl group, in particular if A is S, SO or SO2.

[1111] Among the pyrazolyl derivatives of the formula I mentioned as being preferred, preference is in turn given to those compounds in which Pz in formula I is a group of the formula IIa. Amongst these, in turn, particular preference is given to compounds of the formula I in which the variables R7, R8 and R9 in formula IIa on their own and particularly preferably in combination with one another have the following meanings:

[1112] R7 is hydroxyl, halogen, OR10, SR10, SO2R11, OSO2R11, NR14R15, ONR14R15 or N-bonded heterocyclyl which may be partially or fully halogenated and/or may carry one, two or three of the following radicals: nitro, cyano, C1-C4-alkyl,

[1113] C1-C4-haloalkyl, C1-C4-alkoxy or C1-C4-haloalkoxy, in particular hydroxyl, OR10 and OSO2R11;

[1114] R8 is C1-C4-alkyl, C3-C6-cycloalkyl; in particular cyclopropyl;

[1115] R9 is hydrogen or C1-C4-alkyl.

[1116] Among the compounds of the formula I in which Pz is a pyrazolyl radical of the formula IIa, very particular preference is given to those compounds in which the variables R7, R8 and R9 together have the following meanings:

[1117] R7 is hydroxyl, C1-C4-alkyloxy, acetoxy, O—CH2-phenyl,

[1118] phenylcarbonyloxy, 2-, 3- or 4-fluorophenylcarbonyloxy,

[1119] cyclopropylcarbonyloxy, C1-C4-sulfonyloxy, phenylsulfonyloxy

[1120] and 2-, 3- or 4-methylphenylsulfonyloxy;

[1121] R8 is C1-C4-alkyl or cyclopropyl and

[1122] R9 is hydrogen or C1-C4-alkyl.

[1123] Examples of particularly preferred radicals of the formula IIa are the radicals IIa1 to IIa90 listed in Table 1.

TABLE 1
7
	IIa	R7	R8	R9
	IIa1	OH	CH3	H
	IIa2	OCH3	CH3	H
	IIa3	OCH2—C6H5	CH3	H
	IIa4	OC(O)CH3	CH3	H
	IIa5	OC(O)C6H5	CH3	H
	IIa6	OC(O)-(3-C6H4F)	CH3	H
	IIa7	OS(O)2CH3	CH3	H
	IIa8	OS(O)2-(4-C6H4CH3)	CH3	H
	IIa9	OH	C2H5	H
	IIa10	OCH3	C2H5	H
	IIa11	OCH2—C6H5	C2H5	H
	IIa12	OC(O)CH3	C2H5	H
	IIa13	OC(O)C6H5	C2H5	H
	IIa14	OC(O)-(3-C6H4F)	C2H5	H
	IIa15	OS(O)2CH3	C2H5	H
	IIa16	OS(O)2-(4-C6H4CH3)	C2H5	H
	IIa17	OH	i-C3H7	H
	IIa18	OCH3	i-C3H7	H
	IIa19	OCH2—C6H5	i-C3H7	H
	IIa20	OC(O)CH3	i-C3H7	H
	IIa21	OC(O)C6H5	i-C3H7	H
	IIa22	OC(O)-(3-C6H4F)	i-C3H7	H
	IIa23	OS(O)2CH3	i-C3H7	H
	IIa24	OS(O)2-(4-C6H4CH3)	i-C3H7	H
	IIa25	OH	t-C4H9	H
	IIa26	OCH3	t-C4H9	H
	IIa27	OCH2—C6H5	t-C4H9	H
	IIa28	OC(O)CH3	t-C4H9	H
	IIa29	OC(O)C6H5	t-C4H9	H
	IIa30	OC(O)-(3-C6H4F)	t-C4H9	H
	IIa31	OS(O)2CH3	t-C4H9	H
	IIa32	OS(O)2-(4-C6H4CH3)	t-C4H9	H
	IIa33	OH	CH3	CH3
	IIa34	OCH3	CH3	CH3
	IIa35	OCH2—C6H5	CH3	CH3
	IIa36	OC(O)CH3	CH3	CH3
	IIa37	OC(O)C6H5	CH3	CH3
	IIa38	OC(O)-(3-C6H4F)	CH3	CH3
	IIa39	OS(O)2CH3	CH3	CH3
	IIa40	OS(O)2-(4-C6H4CH3)	CH3	CH3
	IIa41	OH	C2H5	CH3
	IIa42	OCH3	C2H5	CH3
	IIa43	OCH2—C6H5	C2H5	CH3
	IIa44	OC(O)CH3	C2H5	CH3
	IIa45	OC(O)C6H5	C2H5	CH3
	IIa46	OC(O)-(3-C6H4F)	C2H5	CH3
	IIa47	OS(O)2CH3	C2H5	CH3
	IIa48	OS(O)2-(4-C6H4CH3)	C2H5	CH3
	IIa49	OH	i-C3H7	CH3
	IIa50	OCH3	i-C3H7	CH3
	IIa51	OCH2—C6H5	i-C3H7	CH3
	IIa52	OC(O)CH3	i-C3H7	CH3
	IIa53	OC(O)C6H5	i-C3H7	CH3
	IIa54	OC(O)-(3-C6H4F)	i-C3H7	CH3
	IIa55	OS(O)2CH3	i-C3H7	CH3
	IIa56	OS(O)2(4-C6H4CH3)	i-C3H7	CH3
	IIa57	OH	t-C4H9	CH3
	IIa58	OCH3	t-C4H9	CH3
	IIa59	OCH2—C6H5	t-C4H9	CH3
	IIa60	OC(O)CH3	t-C4H9	CH3
	IIa61	OC(O)C6H5	t-C4H9	CH3
	IIa62	OC(O)-(3-C6H4F)	t-C4H9	CH3
	IIa63	OS(O)2CH3	t-C4H9	CH3
	IIa64	OS(O)2-(4-C6H4CH3)	t-C4H9	CH3
	IIa65	OH	c-C3H5	CH3
	IIa66	OCH3	c-C3H5	CH3
	IIa67	OCH2—C6H5	c-C3H5	CH3
	IIa68	OC(O)CH3	c-C3H5	CH3
	IIa69	OC(O)C6H5	c-C3H5	CH3
	IIa70	OC(O)-(3-C6H4F)	c-C3H5	CH3
	IIa71	OS(O)2CH3	c-C3H5	CH3
	IIa72	OS(O)2-(4-C6H4CH3)	c-C3H5	CH3
	IIa73	OH	c-C3H5	H
	IIa74	OCH3	c-C3H5	H
	IIa75	OCH2—C6H5	c-C3H5	H
	IIa76	OC(O)CH3	c-C3H5	H
	IIa77	OC(O)C6H5	c-C3H5	H
	IIa78	OC(O)-(3-C6H4F)	c-C3H5	H
	IIa79	OS(O)2CH3	c-C3H5	H
	IIa80	OS(O)2-(4-C6H4CH3)	c-C3H5	H
	IIa81	OC(O)c-C3H5	CH3	H
	IIa82	OC(O)-c-C3H5	C2H5	H
	IIa83	OC(O)-c-C3H5	i-C3H7	H
	IIa84	OC(O)-c-C3H5	t-C4H9	H
	IIa85	OC(O)-c-C3H5	c-C3H5	H
	IIa86	OC(O)-c-C3H5	CH3	CH3
	IIa87	OC(O)-c-C3H5	C2H5	CH3
	IIa88	OC(O)-c-C3H5	i-C3H7	CH3
	IIa89	OC(O)-c-C3H5	t-C4H9	CH3
	IIa90	OC(O)-c-C3H5	c-C3H5	CH3
	i-C3H7: isopropyl
	c-C3H5: cyclopropyl
	t-C4H9: tertiary butyl
	C6H5: phenyl
	3-C6H4F: 3-fluorophenyl
	4-C6H4CH3: 4-methylphenyl

[1124] Examples of compounds of the formula I which are particularly preferred according to the invention are the benzazolonylcarbonylpyrazoles I listed in Tables 2 to 25 below, where R1, R2, R3 and A in each case have the meanings given in one row of Table A.

TABLE 2
Compounds I-1a.1 to I-1a.3960
8

[1125]

TABLE 3
Compounds I-1b.1 to I-1b.3960
9

[1126]

TABLE 4
Compounds I-1c.1 to I-1c.3960
10

[1127]

TABLE 5
Compounds I-1d.1 to I-1d.3960
11

[1128]

TABLE 6
Compounds I-1e.1 to I-1e.3960
12

[1129]

TABLE 7
Compounds I-1f.1 to I-1f.3960
13

[1130]

TABLE 8
Compounds I-1g.1 to I-1g.3960
14

[1131]

TABLE 9
Compounds I-1h.1 to I-1h.3960
15

[1132]

TABLE 10
Compounds I-1i.1 to I-1i.3960
16

[1133]

TABLE 11
Compounds I-1k.1 to I-1k.3960
I-1k
17

[1134]

TABLE 12
Compounds I-1l.1 to I-1l.3960
I-1l
18

[1135]

TABLE 13
Compounds I-1m.1 to I-1m.3960
I-1m
19

[1136]

TABLE 14
Compounds I-1n.1 to I-1n.3960
I-1n
20

[1137]

TABLE 15
Compounds I-1o.1 to I-1o.3960
I-1o
21

[1138]

TABLE 16
Compounds I-1p.1 to I-1p.3960
I-1p
22

[1139]

TABLE 17
Compounds I-1q.1 to I-1q.3960
I-1q
23

[1140]

TABLE 18
Compounds I-1r.1 to I-1r.3960
I-1r
24

[1141]

TABLE 19
Compounds I-1s.1 to I-1s.3960
I-1s
25

[1142]

TABLE 20
Compounds I-1t.1 to I-1t.3960
I-1t
26

[1143]

TABLE 21
Compounds I-1u.1 to I-1u.3960
27

[1144]

TABLE 22
Compounds I-1v.1 to I-1v.3960
28

[1145]

Table 23
Compounds I-1w.1 to I-1w.3960
29

[1146]

TABLE 24
Compounds I-1x.1 to I-1x.3960
30

[1147]

TABLE 25
Compounds I-1y.1 to I-1y.3960
31

[1148]

TABLE A
Particularly preferred combinations of R1, R2, R3 and A
No.	R1	R2	R3	A
1	CH3	H	H	O
2	CH3	CH3	H	O
3	CH3	C2H5	H	O
4	CH3	n-C3H7	H	O
5	CH3	i-C3H7	H	O
6	CH3	n-C4H9	H	O
7	CH3	i-C4H9	H	O
8	CH3	s-C4H9	H	O
9	CH3	t-C4H9	H	O
10	CH3	CH2OCH3	H	O
11	CH3	CF3	H	O
12	CH3	CF2H	H	O
13	CH3	CN	H	O
14	CH3	OH	H	O
15	CH3	OCH3	H	O
16	CH3	NH2	H	O
17	CH3	NHCH3	H	O
18	CH3	N(CH3)2	H	O
19	CH3	CO2CH3	H	O
20	CH3	CO2C2H5	H	O
21	CH3	C(O)CH3	H	O
22	CH3	C(O)CF3	H	O
23	CH3	C(═NOCH3)CH3	H	O
24	CH3	SO2CH3	H	O
25	CH3	SO2CF3	H	O
26	CH3	CH2CO2H	H	O
27	CH3	CH2COOCH3	H	O
28	CH3	CH2COOC2H5	H	O
29	CH3	prop-1-en-3-yl	H	O
30	CH3	trans-but-2-en-1-yl	H	O
31	CH3	cis-but-2-en-1-yl	H	O
32	CH3	cis-3-methyl-	H	O
		but-2-en-1-yl
33	CH3	cyclopropyl	H	O
34	CH3	cyclopentyl	H	O
35	CH3	cyclohexyl	H	O
36	CH3	4,5-dihydroisoxazol-	H	O
		3-yl
37	CH3	4-methyl-4,5-dihydroisoxazol-	H	O
		3-yl
38	CH3	isoxazol-3-yl	H	O
39	CH3	4-methylisoxazol-3-yl	H	O
40	CH3	4,5-dihydroisoxazol-	H	O
		4-yl
41	CH3	3-methyl-4,5-dihydroisoxazol-	H	O
		4-yl
42	CH3	isoxazol-4-yl	H	O
43	CH3	3-methylisoxazol-4-yl	H	O
44	CH3	phenyl	H	O
45	CH3	benzyl	H	O
46	CH3	benzoyl	H	O
47	CH3	2-pyridyl	H	O
48	CH3	H	CH3	O
49	CH3	CH3	CH3	O
50	CH3	C2H5	CH3	O
51	CH3	n-C3H7	CH3	O
52	CH3	i-C3H7	CH3	O
53	CH3	n-C4H9	CH3	O
54	CH3	i-C4H9	CH3	O
55	CH3	s-C4H9	CH3	O
56	CH3	t-C4H9	CH3	O
57	CH3	CH2OCH3	CH3	O
58	CH3	CF3	CH3	O
59	CH3	CF2H	CH3	O
60	CH3	CN	CH3	O
61	CH3	OH	CH3	O
62	CH3	OCH3	CH3	O
63	CH3	NH2	CH3	O
64	CH3	NHCH3	CH3	O
65	CH3	N(CH3)2	CH3	O
66	CH3	CO2CH3	CH3	O
67	CH3	CO2C2H5	CH3	O
68	CH3	C(O)CH3	CH3	O
69	CH3	C(O)CF3	CH3	O
70	CH3	C(═NOCH3)CH3	CH3	O
71	CH3	SO2CH3	CH3	O
72	CH3	SO2CF3	CH3	O
73	CH3	CH2CO2H	CH3	O
74	CH3	CH2COOCH3	CH3	O
75	CH3	CH2COOC2H5	CH3	O
76	CH3	prop-1-en-3-yl	CH3	O
77	CH3	trans-but-2-en-1-yl	CH3	O
78	CH3	cis-but-2-en-1-yl	CH3	O
79	CH3	cis-3-methyl-	CH3	O
		but-2-en-1-yl
80	CH3	cyclopropyl	CH3	O
81	CH3	cyclopentyl	CH3	O
82	CH3	cyclohexyl	CH3	O
83	CH3	4,5-dihydroisoxazol-	CH3	O
		3-yl
84	CH3	4-methyl-4,5-dihydroisoxazol-	CH3	O
		3-yl
85	CH3	isoxazol-3-yl	CH3	O
86	CH3	4-methylisoxazol-3-yl	CH3	O
87	CH3	4,5-dihydroisoxazol-	CH3	O
		4-yl
88	CH3	3-methyl-4,5-dihydroisoxazol-	CH3	O
		4-yl
89	CH3	isoxazol-4-yl	CH3	O
90	CH3	3-methylisoxazol-4-yl	CH3	O
91	CH3	phenyl	CH3	O
92	CH3	benzyl	CH3	O
93	CH3	benzoyl	CH3	O
94	CH3	2-pyridyl	CH3	O
95	CH3	H	Cl	O
96	CH3	CH3	Cl	O
97	CH3	C2H5	Cl	O
98	CH3	n-C3H7	Cl	O
99	CH3	i-C3H7	Cl	O
100	CH3	n-C4H9	Cl	O
101	CH3	i-C4H9	Cl	O
102	CH3	s-C4H9	Cl	O
103	CH3	t-C4H9	Cl	O
104	CH3	CH2OCH3	Cl	O
105	CH3	CF3	Cl	O
106	CH3	CF2H	Cl	O
107	CH3	CN	Cl	O
108	CH3	OH	Cl	O
109	CH3	OCH3	Cl	O
110	CH3	NH2	Cl	O
111	CH3	NHCH3	Cl	O
112	CH3	N(CH3)2	Cl	O
113	CH3	CO2CH3	Cl	O
114	CH3	CO2C2H5	Cl	O
115	CH3	C(O)CH3	Cl	O
116	CH3	C(O)CF3	Cl	O
117	CH3	C(═NOCH3)CH3	Cl	O
118	CH3	SO2CH3	Cl	O
119	CH3	SO2CF3	Cl	O
120	CH3	CH2CO2H	Cl	O
121	CH3	CH2COOCH3	Cl	O
122	CH3	CH2COOC2H5	Cl	O
123	CH3	prop-1-en-3-yl	Cl	O
124	CH3	trans-but-2-en-1-yl	Cl	O
125	CH3	cis-but-2-en-1-yl	Cl	O
126	CH3	cis-3-methyl-	Cl	O
		but-2-en-1-yl
127	CH3	cyclopropyl	Cl	O
128	CH3	cyclopentyl	Cl	O
129	CH3	cyclohexyl	Cl	O
130	CH3	4,5-dihydroisoxazol-	Cl	O
		3-yl
131	CH3	4-methyl-4,5-dihydroisoxazol-	Cl	O
		3-yl
132	CH3	isoxazol-3-yl	Cl	O
133	CH3	4-methylisoxazol-3-yl	Cl	O
134	CH3	4,5-dihydroisoxazol-	Cl	O
		4-yl
135	CH3	3-methyl-4,5-dihydroisoxazol-	Cl	O
		4-yl
136	CH3	isoxazol-4-yl	Cl	O
137	CH3	3-methylisoxazol-4-yl	Cl	O
138	CH3	phenyl	Cl	O
139	CH3	benzyl	Cl	O
140	CH3	benzoyl	Cl	O
141	CH3	2-pyridyl	Cl	O
142	Cl	H	H	O
143	Cl	CH3	H	O
144	Cl	C2H5	H	O
145	Cl	n-C3H7	H	O
146	Cl	i-C3H7	H	O
147	Cl	n-C4H9	H	O
148	Cl	i-C4H9	H	O
149	Cl	s-C4H9	H	O
150	Cl	t-C4H9	H	O
151	Cl	CH2OCH3	H	O
152	Cl	CF3	H	O
153	Cl	CF2H	H	O
154	Cl	CN	H	O
155	Cl	OH	H	O
156	Cl	OCH3	H	O
157	Cl	NH2	H	O
158	Cl	NHCH3	H	O
159	Cl	N(CH3)2	H	O
160	Cl	CO2CH3	H	O
161	Cl	CO2C2H5	H	O
162	Cl	C(O)CH3	H	O
163	Cl	C(O)CF3	H	O
164	Cl	C(═NOCH3)CH3	H	O
165	Cl	SO2CH3	H	O
166	Cl	SO2CF3	H	O
167	Cl	CH2CO2H	H	O
168	Cl	CH2COOCH3	H	O
169	Cl	CH2COOC2H5	H	O
170	Cl	prop-1-en-3-yl	H	O
171	Cl	trans-but-2-en-1-yl	H	O
172	Cl	cis-but-2-en-1-yl	H	O
173	Cl	cis-3-methyl-	H	O
		but-2-en-1-yl
174	Cl	cyclopropyl	H	O
175	Cl	cyclopentyl	H	O
176	Cl	cyclohexyl	H	O
177	Cl	4,5-dihydroisoxazol-	H	O
		3-yl
178	Cl	4-methyl-4,5-dihydroisoxazol-	H	O
		3-yl
179	Cl	isoxazol-3-yl	H	O
180	Cl	4-methylisoxazol-3-yl	H	O
181	Cl	4,5-dihydroisoxazol-	H	O
		4-yl
182	Cl	3-methyl-4,5-dihydroisoxazol-	H	O
		4-yl
183	Cl	isoxazol-4-yl	H	O
184	Cl	3-methylisoxazol-4-yl	H	O
185	Cl	phenyl	H	O
186	Cl	benzyl	H	O
187	Cl	benzoyl	H	O
188	Cl	2-pyridyl	H	O
189	Cl	H	CH3	O
190	Cl	CH3	CH3	O
191	Cl	C2H5	CH3	O
192	Cl	n-C3H7	CH3	O
193	Cl	i-C3H7	CH3	O
194	Cl	n-C4H9	CH3	O
195	Cl	i-C4H9	CH3	O
196	Cl	s-C4H9	CH3	O
197	Cl	t-C4H9	CH3	O
198	Cl	CH2OCH3	CH3	O
199	Cl	CF3	CH3	O
200	Cl	CF2H	CH3	O
201	Cl	CN	CH3	O
202	Cl	OH	CH3	O
203	Cl	OCH3	CH3	O
204	Cl	NH2	CH3	O
205	Cl	NHCH3	CH3	O
206	Cl	N(CH3)2	CH3	O
207	Cl	CO2CH3	CH3	O
208	Cl	CO2C2H5	CH3	O
209	Cl	C(O)CH3	CH3	O
210	Cl	C(O)CF3	CH3	O
211	Cl	C(═NOCH3)CH3	CH3	O
212	Cl	SO2CH3	CH3	O
213	Cl	SO2CF3	CH3	O
214	Cl	CH2CO2H	CH3	O
215	Cl	CH2COOCH3	CH3	O
216	Cl	CH2COOC2H5	CH3	O
217	Cl	prop-1-en-3-yl	CH3	O
218	Cl	trans-but-2-en-1-yl	CH3	O
219	Cl	cis-but-2-en-1-yl	CH3	O
220	Cl	cis-3-methyl-	CH3	O
		but-2-en-1-yl
221	Cl	cyclopropyl	CH3	O
222	Cl	cyclopentyl	CH3	O
223	Cl	cyclohexyl	CH3	O
224	Cl	4,5-dihydroisoxazol-	CH3	O
		3-yl
225	Cl	4-methyl-4,5-dihydroisoxazol-	CH3	O
		3-yl
226	Cl	isoxazol-3-yl	CH3	O
227	Cl	4-methylisoxazol-3-yl	CH3	O
228	Cl	4,5-dihydroisoxazol-	CH3	O
		4-yl
229	Cl	3-methyl-4,5-dihydroisoxazol-	CH3	O
		4-yl
230	Cl	isoxazol-4-yl	CH3	O
231	Cl	3-methylisoxazol-4-yl	CH3	O
232	Cl	phenyl	CH3	O
233	Cl	benzyl	CH3	O
234	Cl	benzoyl	CH3	O
235	Cl	2-pyridyl	CH3	O
236	Cl	H	Cl	O
237	Cl	CH3	Cl	O
238	Cl	C2H5	Cl	O
239	Cl	n-C3H7	Cl	O
240	Cl	i-C3H7	Cl	O
241	Cl	n-C4H9	Cl	O
242	Cl	i-C4H9	Cl	O
243	Cl	s-C4H9	Cl	O
244	Cl	t-C4H9	Cl	O
245	Cl	CH2OCH3	Cl	O
246	Cl	CF3	Cl	O
247	Cl	CF2H	Cl	O
248	Cl	CN	Cl	O
249	Cl	OH	Cl	O
250	Cl	OCH3	Cl	O
251	Cl	NH2	Cl	O
252	Cl	NHCH3	Cl	O
253	Cl	N(CH3)2	Cl	O
254	Cl	CO2CH3	Cl	O
255	Cl	CO2C2H5	Cl	O
256	Cl	C(O)CH3	Cl	O
257	Cl	C(O)CF3	Cl	O
258	Cl	C(═NOCH3)CH3	Cl	O
259	Cl	SO2CH3	Cl	O
260	Cl	SO2CF3	Cl	O
261	Cl	CH2CO2H	Cl	O
262	Cl	CH2COOCH3	Cl	O
263	Cl	CH2COOC2H5	Cl	O
264	Cl	prop-1-en-3-yl	Cl	O
265	Cl	trans-but-2-en-1-yl	Cl	O
266	Cl	cis-but-2-en-1-yl	Cl	O
267	Cl	cis-3-methyl-	Cl	O
		but-2-en-1-yl
268	Cl	cyclopropyl	Cl	O
269	Cl	cyclopentyl	Cl	O
270	Cl	cyclohexyl	Cl	O
271	Cl	4,5-dihydroisoxazol-	Cl	O
		3-yl
272	Cl	4-methyl-4,5-dihydroisoxazol-	Cl	O
		3-yl
273	Cl	isoxazol-3-yl	Cl	O
274	Cl	4-methylisoxazol-3-yl	Cl	O
275	Cl	4,5-dihydroisoxazol-	Cl	O
		4-yl
276	Cl	3-methyl-4,5-dihydroisoxazol-	Cl	O
		4-yl
277	Cl	isoxazol-4-yl	Cl	O
278	Cl	3-methylisoxazol-4-yl	Cl	O
279	Cl	phenyl	Cl	O
280	Cl	benzyl	Cl	O
281	Cl	benzoyl	Cl	O
282	Cl	2-pyridyl	Cl	O
283	OCH3	H	H	O
284	OCH3	CH3	H	O
285	OCH3	C2H5	H	O
286	OCH3	n-C3H7	H	O
287	OCH3	i-C3H7	H	O
288	OCH3	n-C4H9	H	O
289	OCH3	i-C4H9	H	O
290	OCH3	s-C4H9	H	O
291	OCH3	t-C4H9	H	O
292	OCH3	CH2OCH3	H	O
293	OCH3	CF3	H	O
294	OCH3	CF2H	H	O
295	OCH3	CN	H	O
296	OCH3	OH	H	O
297	OCH3	OCH3	H	O
298	OCH3	NH2	H	O
299	OCH3	NHCH3	H	O
300	OCH3	N(CH3)2	H	O
301	OCH3	CO2CH3	H	O
302	OCH3	CO2C2H5	H	O
303	OCH3	C(O)CH3	H	O
304	OCH3	C(O)CF3	H	O
305	OCH3	C(═NOCH3)CH3	H	O
306	OCH3	SO2CH3	H	O
307	OCH3	SO2CF3	H	O
308	OCH3	CH2CO2H	H	O
309	OCH3	CH2COOCH3	H	O
310	OCH3	CH2COOC2H5	H	O
311	OCH3	prop-1-en-3-yl	H	O
312	OCH3	trans-but-2-en-1-yl	H	O
313	OCH3	cis-but-2-en-1-yl	H	O
314	OCH3	cis-3-methyl-	H	O
		but-2-en-1-yl
315	OCH3	cyclopropyl	H	O
316	OCH3	cyclopentyl	H	O
317	OCH3	cyclohexyl	H	O
318	OCH3	4,5-dihydroisoxazol-	H	O
		3-yl
319	OCH3	4-methyl-4,5-dihydroisoxazol-	H	O
		3-yl
320	OCH3	isoxazol-3-yl	H	O
321	OCH3	4-methylisoxazol-3-yl	H	O
322	OCH3	4,5-dihydroisoxazol-	H	O
		4-yl
323	OCH3	3-methyl-4,5-dihydroisoxazol-	H	O
		4-yl
324	OCH3	isoxazol-4-yl	H	O
325	OCH3	3-methylisoxazol-4-yl	H	O
326	OCH3	phenyl	H	O
327	OCH3	benzyl	H	O
328	OCH3	benzoyl	H	O
329	OCH3	2-pyridyl	H	O
330	OCH3	H	CH3	O
331	OCH3	CH3	CH3	O
332	OCH3	C2H5	CH3	O
333	OCH3	n-C3H7	CH3	O
334	OCH3	i-C3H7	CH3	O
335	OCH3	n-C4H9	CH3	O
336	OCH3	i-C4H9	CH3	O
337	OCH3	s-C4H9	CH3	O
338	OCH3	t-C4H9	CH3	O
339	OCH3	CH2OCH3	CH3	O
340	OCH3	CF3	CH3	O
341	OCH3	CF2H	CH3	O
342	OCH3	CN	CH3	O
343	OCH3	OH	CH3	O
344	OCH3	OCH3	CH3	O
345	OCH3	NH2	CH3	O
346	OCH3	NHCH3	CH3	O
347	OCH3	N(CH3)2	CH3	O
348	OCH3	CO2CH3	CH3	O
349	OCH3	CO2C2H5	CH3	O
350	OCH3	C(O)CH3	CH3	O
351	OCH3	C(O)CF3	CH3	O
352	OCH3	C(═NOCH3)CH3	CH3	O
353	OCH3	SO2CH3	CH3	O
354	OCH3	SO2CF3	CH3	O
355	OCH3	CH2CO2H	CH3	O
356	OCH3	CH2COOCH3	CH3	O
357	OCH3	CH2COOC2H5	CH3	O
358	OCH3	prop-1-en-3-yl	CH3	O
359	OCH3	trans-but-2-en-1-yl	CH3	O
360	OCH3	cis-but-2-en-1-yl	CH3	O
361	OCH3	cis-3-methyl-	CH3	O
		but-2-en-1-yl
362	OCH3	cyclopropyl	CH3	O
363	OCH3	cyclopentyl	CH3	O
364	OCH3	cyclohexyl	CH3	O
365	OCH3	4,5-dihydroisoxazol-	CH3	O
		3-yl
366	OCH3	4-methyl-4,5-dihydroisoxazol-	CH3	O
		3-yl
367	OCH3	isoxazol-3-yl	CH3	O
368	OCH3	4-methylisoxazol-3-yl	CH3	O
369	OCH3	4,5-dihydroisoxazol-	CH3	O
		4-yl
370	OCH3	3-methyl-4,5-dihydroisoxazol-	CH3	O
		4-yl
371	OCH3	isoxazol-4-yl	CH3	O
372	OCH3	3-methylisoxazol-4-yl	CH3	O
373	OCH3	phenyl	CH3	O
374	OCH3	benzyl	CH3	O
375	OCH3	benzoyl	CH3	O
376	OCH3	2-pyridyl	CH3	O
377	OCH3	H	Cl	O
378	OCH3	CH3	Cl	O
379	OCH3	C2H5	Cl	O
380	OCH3	n-C3H7	Cl	O
381	OCH3	i-C3H7	Cl	O
382	OCH3	n-C4H9	Cl	O
383	OCH3	i-C4H9	Cl	O
384	OCH3	s-C4H9	Cl	O
385	OCH3	t-C4H9	Cl	O
386	OCH3	CH2OCH3	Cl	O
387	OCH3	CF3	Cl	O
388	OCH3	CF2H	Cl	O
389	OCH3	CN	Cl	O
390	OCH3	OH	Cl	O
391	OCH3	OCH3	Cl	O
392	OCH3	NH2	Cl	O
393	OCH3	NHCH3	Cl	O
394	OCH3	N(CH3)2	Cl	O
395	OCH3	CO2CH3	Cl	O
396	OCH3	CO2C2H5	Cl	O
397	OCH3	C(O)CH3	Cl	O
398	OCH3	C(O)CF3	Cl	O
399	OCH3	C(═NOCH3)CH3	Cl	O
400	OCH3	SO2CH3	Cl	O
401	OCH3	SO2CF3	Cl	O
402	OCH3	CH2CO2H	Cl	O
403	OCH3	CH2COOCH3	Cl	O
404	OCH3	CH2COOC2H5	Cl	O
405	OCH3	prop-1-en-3-yl	Cl	O
406	OCH3	trans-but-2-en-1-yl	Cl	O
407	OCH3	cis-but-2-en-1-yl	Cl	O
408	OCH3	cis-3-methyl-	Cl	O
		but-2-en-1-yl
409	OCH3	cyclopropyl	Cl	O
410	OCH3	cyclopentyl	Cl	O
411	OCH3	cyclohexyl	Cl	O
412	OCH3	4,5-dihydroisoxazol-	Cl	O
		3-yl
413	OCH3	4-methyl-4,5-dihydroisoxazol-	Cl	O
		3-yl
414	OCH3	isoxazol-3-yl	Cl	O
415	OCH3	4-methylisoxazol-3-yl	Cl	O
416	OCH3	4,5-dihydroisoxazol-	Cl	O
		4-yl
417	OCH3	3-methyl-4,5-dihydroisoxazol-	Cl	O
		4-yl
418	OCH3	isoxazol-4-yl	Cl	O
419	OCH3	3-methylisoxazol-4-yl	Cl	O
420	OCH3	phenyl	Cl	O
421	OCH3	benzyl	Cl	O
422	OCH3	benzoyl	Cl	O
423	OCH3	2-pyridyl	Cl	O
424	OCF3	H	H	O
425	OCF3	CH3	H	O
426	OCF3	C2H5	H	O
427	OCF3	n-C3H7	H	O
428	OCF3	i-C3H7	H	O
429	OCF3	n-C4H9	H	O
430	OCF3	i-C4H9	H	O
431	OCF3	s-C4H9	H	O
432	OCF3	t-C4H9	H	O
433	OCF3	CH2OCH3	H	O
434	OCF3	CF3	H	O
435	OCF3	CF2H	H	O
436	OCF3	CN	H	O
437	OCF3	OH	H	O
438	OCF3	OCH3	H	O
439	OCF3	NH2	H	O
440	OCF3	NHCH3	H	O
441	OCF3	N(CH3)2	H	O
442	OCF3	CO2CH3	H	O
443	OCF3	CO2C2H5	H	O
444	OCF3	C(O)CH3	H	O
445	OCF3	C(O)CF3	H	O
446	OCF3	C(═NOCH3)CH3	H	O
447	OCF3	SO2CH3	H	O
448	OCF3	SO2CF3	H	O
449	OCF3	CH2CO2H	H	O
450	OCF3	CH2COOCH3	H	O
451	OCF3	CH2COOC2H5	H	O
452	OCF3	prop-1-en-3-yl	H	O
453	OCF3	trans-but-2-en-1-yl	H	O
454	OCF3	cis-but-2-en-1-yl	H	O
455	OCF3	cis-3-methyl-	H	O
		but-2-en-1-yl
456	OCF3	cyclopropyl	H	O
457	OCF3	cyclopentyl	H	O
458	OCF3	cyclohexyl	H	O
459	OCF3	4,5-dihydroisoxazol-	H	O
		3-yl
460	OCF3	4-methyl-4,5-dihydroisoxazol-	H	O
		3-yl
461	OCF3	isoxazol-3-yl	H	O
462	OCF3	4-methylisoxazol-3-yl	H	O
463	OCF3	4,5-dihydroisoxazol-	H	O
		4-yl
464	OCF3	3-methyl-4,5-dihydroisoxazol-	H	O
		4-yl
465	OCF3	isoxazol-4-yl	H	O
466	OCF3	3-methylisoxazol-4-yl	H	O
467	OCF3	phenyl	H	O
468	OCF3	benzyl	H	O
469	OCF3	benzoyl	H	O
470	OCF3	2-pyridyl	H	O
471	OCF3	H	CH3	O
472	OCF3	CH3	CH3	O
473	OCF3	C2H5	CH3	O
474	OCF3	n-C3H7	CH3	O
475	OCF3	i-C3H7	CH3	O
476	OCF3	n-C4H9	CH3	O
477	OCF3	i-C4H9	CH3	O
478	OCF3	s-C4H9	CH3	O
479	OCF3	t-C4H9	CH3	O
480	OCF3	CH2OCH3	CH3	O
481	OCF3	CF3	CH3	O
482	OCF3	CF2H	CH3	O
483	OCF3	CN	CH3	O
484	OCF3	OH	CH3	O
485	OCF3	OCH3	CH3	O
486	OCF3	NH2	CH3	O
487	OCF3	NHCH3	CH3	O
488	OCF3	N(CH3)2	CH3	O
489	OCF3	CO2CH3	CH3	O
490	OCF3	CO2C2H5	CH3	O
491	OCF3	C(O)CH3	CH3	O
492	OCF3	C(O)CF3	CH3	O
493	OCF3	C(═NOCH3)CH3	CH3	O
494	OCF3	SO2CH3	CH3	O
495	OCF3	SO2CF3	CH3	O
496	OCF3	CH2CO2H	CH3	O
497	OCF3	CH2COOCH3	CH3	O
498	OCF3	CH2COOC2H5	CH3	O
499	OCF3	prop-1-en-3-yl	CH3	O
500	OCF3	trans-but-2-en-1-yl	CH3	O
501	OCF3	cis-but-2-en-1-yl	CH3	O
502	OCF3	cis-3-methyl-	CH3	O
		but-2-en-1-yl
503	OCF3	cyclopropyl	CH3	O
504	OCF3	cyclopentyl	CH3	O
505	OCF3	cyclohexyl	CH3	O
506	OCF3	4,5-dihydroisoxazol-	CH3	O
		3-yl
507	OCF3	4-methyl-4,5-dihydroisoxazol-	CH3	O
		3-yl
508	OCF3	isoxazol-3-yl	CH3	O
509	OCF3	4-methylisoxazol-3-yl	CH3	O
510	OCF3	4,5-dihydroisoxazol-	CH3	O
		4-yl
511	OCF3	3-methyl-4,5-dihydroisoxazol-	CH3	O
		4-yl
512	OCF3	isoxazol-4-yl	CH3	O
513	OCF3	3-methylisoxazol-4-yl	CH3	O
514	OCF3	phenyl	CH3	O
515	OCF3	benzyl	CH3	O
516	OCF3	benzoyl	CH3	O
517	OCF3	2-pyridyl	CH3	O
518	OCF3	H	Cl	O
519	OCF3	CH3	Cl	O
520	OCF3	C2H5	Cl	O
521	OCF3	n-C3H7	Cl	O
522	OCF3	i-C3H7	Cl	O
523	OCF3	n-C4H9	Cl	O
524	OCF3	i-C4H9	Cl	O
525	OCF3	s-C4H9	Cl	O
526	OCF3	t-C4H9	Cl	O
527	OCF3	CH2OCH3	Cl	O
528	OCF3	CF3	Cl	O
529	OCF3	CF2H	Cl	O
530	OCF3	CN	Cl	O
531	OCF3	OH	Cl	O
532	OCF3	OCH3	Cl	O
533	OCF3	NH2	Cl	O
534	OCF3	NHCH3	Cl	O
535	OCF3	N(CH3)2	Cl	O
536	OCF3	CO2CH3	Cl	O
537	OCF3	CO2C2H5	Cl	O
538	OCF3	C(O)CH3	Cl	O
539	OCF3	C(O)CF3	Cl	O
540	OCF3	C(═NOCH3)CH3	Cl	O
541	OCF3	SO2CH3	Cl	O
542	OCF3	SO2CF3	Cl	O
543	OCF3	CH2CO2H	Cl	O
544	OCF3	CH2COOCH3	Cl	O
545	OCF3	CH2COOC2H5	Cl	O
546	OCF3	prop-1-en-3-yl	Cl	O
547	OCF3	trans-but-2-en-1-yl	Cl	O
548	OCF3	cis-but-2-en-1-yl	Cl	O
549	OCF3	cis-3-methyl-	Cl	O
		but-2-en-1-yl
550	OCF3	cyclopropyl	Cl	O
551	OCF3	cyclopentyl	Cl	O
552	OCF3	cyclohexyl	Cl	O
553	OCF3	4,5-dihydroisoxazol-	Cl	O
		3-yl
554	OCF3	4-methyl-4,5-dihydroisoxazol-	Cl	O
		3-yl
555	OCF3	isoxazol-3-yl	Cl	O
556	OCF3	4-methylisoxazol-3-yl	Cl	O
557	OCF3	4,5-dihydroisoxazol-	Cl	O
		4-yl
558	OCF3	3-methyl-4,5-dihydroisoxazol-	Cl	O
		4-yl
559	OCF3	isoxazol-4-yl	Cl	O
560	OCF3	3-methylisoxazol-4-yl	Cl	O
561	OCF3	phenyl	Cl	O
562	OCF3	benzyl	Cl	O
563	OCF3	benzoyl	Cl	O
564	OCF3	2-pyridyl	Cl	O
565	SCH3	H	H	O
566	SCH3	CH3	H	O
567	SCH3	C2H5	H	O
568	SCH3	n-C3H7	H	O
569	SCH3	i-C3H7	H	O
570	SCH3	n-C4H9	H	O
571	SCH3	i-C4H9	H	O
572	SCH3	s-C4H9	H	O
573	SCH3	t-C4H9	H	O
574	SCH3	CH2OCH3	H	O
575	SCH3	CF3	H	O
576	SCH3	CF2H	H	O
577	SCH3	CN	H	O
578	SCH3	OH	H	O
579	SCH3	OCH3	H	O
580	SCH3	NH2	H	O
581	SCH3	NHCH3	H	O
582	SCH3	N(CH3)2	H	O
583	SCH3	CO2CH3	H	O
584	SCH3	CO2C2H5	H	O
585	SCH3	C(O)CH3	H	O
586	SCH3	C(O)CF3	H	O
587	SCH3	C(═NOCH3)CH3	H	O
588	SCH3	SO2CH3	H	O
589	SCH3	SO2CF3	H	O
590	SCH3	CH2CO2H	H	O
591	SCH3	CH2COOCH3	H	O
592	SCH3	CH2COOC2H5	H	O
593	SCH3	prop-1-en-3-yl	H	O
594	SCH3	trans-but-2-en-1-yl	H	O
595	SCH3	cis-but-2-en-1-yl	H	O
596	SCH3	cis-3-methyl-	H	O
		but-2-en-1-yl
597	SCH3	cyclopropyl	H	O
598	SCH3	cyclopentyl	H	O
599	SCH3	cyclohexyl	H	O
600	SCH3	4,5-dihydroisoxazol-	H	O
		3-yl
601	SCH3	4-methyl-4,5-dihydroisoxazol-	H	O
		3-yl
602	SCH3	isoxazol-3-yl	H	O
603	SCH3	4-methylisoxazol-3-yl	H	O
604	SCH3	4,5-dihydroisoxazol-	H	O
		4-y1
605	SCH3	3-methyl-4,5-dihydroisoxazol-	H	O
		4-yl
606	SCH3	isoxazol-4-yl	H	O
607	SCH3	3-methylisoxazol-4-yl	H	O
608	SCH3	phenyl	H	O
609	SCH3	benzyl	H	O
610	SCH3	benzoyl	H	O
611	SCH3	2-pyridyl	H	O
612	SCH3	H	CH3	O
613	SCH3	CH3	CH3	O
614	SCH3	C2H5	CH3	O
615	SCH3	n-C3H7	CH3	O
616	SCH3	i-C3H7	CH3	O
617	SCH3	n-C4H9	CH3	O
618	SCH3	i-C4H9	CH3	O
619	SCH3	s-C4H9	CH3	O
620	SCH3	t-C4H9	CH3	O
621	SCH3	CH2OCH3	CH3	O
622	SCH3	CF3	CH3	O
623	SCH3	CF2H	CH3	O
624	SCH3	CN	CH3	O
625	SCH3	OH	CH3	O
626	SCH3	OCH3	CH3	O
627	SCH3	NH2	CH3	O
628	SCH3	NHCH3	CH3	O
629	SCH3	N(CH3)2	CH3	O
630	SCH3	CO2CH3	CH3	O
631	SCH3	CO2C2H5	CH3	O
632	SCH3	C(O)CH3	CH3	O
633	SCH3	C(O)CF3	CH3	O
634	SCH3	C(═NOCH3)CH3	CH3	O
635	SCH3	SO2CH3	CH3	O
636	SCH3	SO2CF3	CH3	O
637	SCH3	CH2CO2H	CH3	O
638	SCH3	CH2COOCH3	CH3	O
639	SCH3	CH2COOC2H5	CH3	O
640	SCH3	prop-1-en-3-yl	CH3	O
641	SCH3	trans-but-2-en-1-yl	CH3	O
642	SCH3	cis-but-2-en-1-yl	CH3	O
643	SCH3	cis-3-methyl-	CH3	O
		but-2-en-1-yl
644	SCH3	cyclopropyl	CH3	O
645	SCH3	cyclopentyl	CH3	O
646	SCH3	cyclohexyl	CH3	O
647	SCH3	4,5-dihydroisoxazol-	CH3	O
		3-yl
648	SCH3	4-methyl-4,5-dihydroisoxazol-	CH3	O
		3-yl
649	SCH3	isoxazol-3-yl	CH3	O
650	SCH3	4-methylisoxazol-3-yl	CH3	O
651	SCH3	4,5-dihydroisoxazol-	CH3	O
		4-yl
652	SCH3	3-methyl-4,5-dihydroisoxazol-	CH3	O
		4-yl
653	SCH3	isoxazol-4-yl	CH3	O
654	SCH3	3-methylisoxazol-4-yl	CH3	O
655	SCH3	phenyl	CH3	O
656	SCH3	benzyl	CH3	O
657	SCH3	benzoyl	CH3	O
658	SCH3	2-pyridyl	CH3	O
659	SCH3	H	Cl	O
660	SCH3	CH3	Cl	O
661	SCH3	C2H5	Cl	O
662	SCH3	n-C3H7	Cl	O
663	SCH3	i-C3H7	Cl	O
664	SCH3	n-C4H9	Cl	O
665	SCH3	i-C4H9	Cl	O
666	SCH3	s-C4H9	Cl	O
667	SCH3	t-C4H9	Cl	O
668	SCH3	CH2OCH3	Cl	O
669	SCH3	CF3	Cl	O
670	SCH3	CF2H	Cl	O
671	SCH3	CN	Cl	O
672	SCH3	OH	Cl	O
673	SCH3	OCH3	Cl	O
674	SCH3	NH2	Cl	O
675	SCH3	NHCH3	Cl	O
676	SCH3	N(CH3)2	Cl	O
677	SCH3	CO2CH3	Cl	O
678	SCH3	CO2C2H5	Cl	O
679	SCH3	C(O)CH3	Cl	O
680	SCH3	C(O)CF3	Cl	O
681	SCH3	C(═NOCH3)CH3	Cl	O
682	SCH3	SO2CH3	Cl	O
683	SCH3	SO2CF3	Cl	O
684	SCH3	CH2CO2H	Cl	O
685	SCH3	CH2COOCH3	Cl	O
686	SCH3	CH2COOC2H5	Cl	O
687	SCH3	prop-1-en-3-yl	Cl	O
688	SCH3	trans-but-2-en-1-yl	Cl	O
689	SCH3	cis-but-2-en-1-yl	Cl	O
690	SCH3	cis-3-methyl-	Cl	O
		but-2-en-1-yl
691	SCH3	cyclopropyl	Cl	O
692	SCH3	cyclopentyl	Cl	O
693	SCH3	cyclohexyl	Cl	O
694	SCH3	4,5-dihydroisoxazol-	Cl	O
		3-yl
695	SCH3	4-methyl-4,5-dihydroisoxazol-	Cl	O
		3-yl
696	SCH3	isoxazol-3-yl	Cl	O
697	SCH3	4-methylisoxazol-3-yl	Cl	O
698	SCH3	4,5-dihydroisoxazol-	Cl	O
		4-yl
699	SCH3	3-methyl-4,5-dihydroisoxazol-	Cl	O
		4-yl
700	SCH3	isoxazol-4-yl	Cl	O
701	SCH3	3-methylisoxazol-4-yl	Cl	O
702	SCH3	phenyl	Cl	O
703	SCH3	benzyl	Cl	O
704	SCH3	benzoyl	Cl	O
705	SCH3	2-pyridyl	Cl	O
706	SO2CH3	H	H	O
707	SO2CH3	CH3	H	O
708	SO2CH3	C2H5	H	O
709	SO2CH3	n-C3H7	H	O
710	SO2CH3	i-C3H7	H	O
711	SO2CH3	n-C4H9	H	O
712	SO2CH3	i-C4H9	H	O
713	SO2CH3	s-C4H9	H	O
714	SO2CH3	t-C4H9	H	O
715	SO2CH3	CH2OCH3	H	O
716	SO2CH3	CF3	H	O
717	SO2CH3	CF2H	H	O
718	SO2CH3	CN	H	O
719	SO2CH3	OH	H	O
720	SO2CH3	OCH3	H	O
721	SO2CH3	NH2	H	O
722	SO2CH3	NHCH3	H	O
723	SO2CH3	N(CH3)2	H	O
724	SO2CH3	CO2CH3	H	O
725	SO2CH3	CO2C2H5	H	O
726	SO2CH3	C(O)CH3	H	O
727	SO2CH3	C(O)CF3	H	O
728	SO2CH3	C(═NOCH3)CH3	H	O
729	SO2CH3	SO2CH3	H	O
730	SO2CH3	SO2CF3	H	O
731	SO2CH3	CH2CO2H	H	O
732	SO2CH3	CH2COOCH3	H	O
733	SO2CH3	CH2COOC2H5	H	O
734	SO2CH3	prop-1-en-3-yl	H	O
735	SO2CH3	trans-but-2-en-1-yl	H	O
736	SO2CH3	cis-but-2-en-1-yl	H	O
737	SO2CH3	cis-3-methyl-	H	O
		but-2-en-1-yl
738	SO2CH3	cyclopropyl	H	O
739	SO2CH3	cyclopentyl	H	O
740	SO2CH3	cyclohexyl	H	O
741	SO2CH3	4,5-dihydroisoxazol-	H	O
		3-yl
742	SO2CH3	4-methyl-4,5-dihydroisoxazol-	H	O
		3-yl
743	SO2CH3	isoxazol-3-yl	H	O
744	SO2CH3	4-methylisoxazol-3-yl	H	O
745	SO2CH3	4,5-dihydroisoxazol-	H	O
		4-yl
746	SO2CH3	3-methyl-4,5-dihydroisoxazol-	H	O
		4-yl
747	SO2CH3	isoxazol-4-yl	H	O
748	SO2CH3	3-methylisoxazol-4-yl	H	O
749	SO2CH3	phenyl	H	O
750	SO2CH3	benzyl	H	O
751	SO2CH3	benzoyl	H	O
752	SO2CH3	2-pyridyl	H	O
753	SO2CH3	H	CH3	O
754	SO2CH3	CH3	CH3	O
755	SO2CH3	C2H5	CH3	O
756	SO2CH3	n-C3H7	CH3	O
757	SO2CH3	i-C3H7	CH3	O
758	SO2CH3	n-C4H9	CH3	O
759	SO2CH3	i-C4H9	CH3	O
760	SO2CH3	s-C4H9	CH3	O
761	SO2CH3	t-C4H9	CH3	O
762	SO2CH3	CH2OCH3	CH3	O
763	SO2CH3	CF3	CH3	O
764	SO2CH3	CF2H	CH3	O
765	SO2CH3	CN	CH3	O
766	SO2CH3	OH	CH3	O
767	SO2CH3	OCH3	CH3	O
768	SO2CH3	NH2	CH3	O
769	SO2CH3	NHCH3	CH3	O
770	SO2CH3	N(CH3)2	CH3	O
771	SO2CH3	CO2CH3	CH3	O
772	SO2CH3	CO2C2H5	CH3	O
773	SO2CH3	C(O)CH3	CH3	O
774	SO2CH3	C(O)CF3	CH3	O
775	SO2CH3	C(═NOCH3)CH3	CH3	O
776	SO2CH3	SO2CH3	CH3	O
777	SO2CH3	SO2CF3	CH3	O
778	SO2CH3	CH2CO2H	CH3	O
779	SO2CH3	CH2COOCH3	CH3	O
780	SO2CH3	CH2COOC2H5	CH3	O
781	SO2CH3	prop-1-en-3-yl	CH3	O
782	SO2CH3	trans-but-2-en-1-yl	CH3	O
783	SO2CH3	cis-but-2-en-1-yl	CH3	O
784	SO2CH3	cis-3-methyl-	CH3	O
		but-2-en-1-yl
785	SO2CH3	cyclopropyl	CH3	O
786	SO2CH3	cyclopentyl	CH3	O
787	SO2CH3	cyclohexyl	CH3	O
788	SO2CH3	4,5-dihydroisoxazol-	CH3	O
		3-yl
789	SO2CH3	4-methyl-4,5-dihydroisoxazol-	CH3	O
		3-yl
790	SO2CH3	isoxazol-3-yl	CH3	O
791	SO2CH3	4-methylisoxazol-3-yl	CH3	O
792	SO2CH3	4,5-dihydroisoxazol-	CH3	O
		4-yl
793	SO2CH3	3-methyl-4,5-dihydroisoxazol-	CH3	O
		4-yl
794	SO2CH3	isoxazol-4-yl	CH3	O
795	SO2CH3	3-methylisoxazol-4-yl	CH3	O
796	SO2CH3	phenyl	CH3	O
797	SO2CH3	benzyl	CH3	O
798	SO2CH3	benzoyl	CH3	O
799	SO2CH3	2-pyridyl	CH3	O
800	SO2CH3	H	Cl	O
801	SO2CH3	CH3	Cl	O
802	SO2CH3	C2H5	Cl	O
803	SO2CH3	n-C3H7	Cl	O
804	SO2CH3	i-C3H7	Cl	O
805	SO2CH3	n-C4H9	Cl	O
806	SO2CH3	i-C4H9	Cl	O
807	SO2CH3	s-C4H9	Cl	O
808	SO2CH3	t-C4H9	Cl	O
809	SO2CH3	CH2OCH3	Cl	O
810	SO2CH3	CF3	Cl	O
811	SO2CH3	CF2H	Cl	O
812	SO2CH3	CN	Cl	O
813	SO2CH3	OH	Cl	O
814	SO2CH3	OCH3	Cl	O
815	SO2CH3	NH2	Cl	O
816	SO2CH3	NHCH3	Cl	O
817	SO2CH3	N(CH3)2	Cl	O
818	SO2CH3	CO2CH3	Cl	O
819	SO2CH3	CO2C2H5	Cl	O
820	SO2CH3	C(O)CH3	Cl	O
821	SO2CH3	C(O)CF3	Cl	O
822	SO2CH3	C(═NOCH3)CH3	Cl	O
823	SO2CH3	SO2CH3	Cl	O
824	SO2CH3	SO2CF3	Cl	O
825	SO2CH3	CH2CO2H	Cl	O
826	SO2CH3	CH2COOCH3	Cl	O
827	SO2CH3	CH2COOC2H5	Cl	O
828	SO2CH3	prop-1-en-3-yl	Cl	O
829	SO2CH3	trans-but-2-en-1-yl	Cl	O
830	SO2CH3	cis-but-2-en-1-yl	Cl	O
831	SO2CH3	cis-3-methyl-	Cl	O
		but-2-en-1-yl
832	SO2CH3	cyclopropyl	Cl	O
833	SO2CH3	cyclopentyl	Cl	O
834	SO2CH3	cyclohexyl	Cl	O
835	SO2CH3	4,5-dihydroisoxazol-	Cl	O
		3-yl
836	SO2CH3	4-methyl-4,5-dihydroisoxazol-	Cl	O
		3-yl
837	SO2CH3	isoxazol-3-yl	Cl	O
838	SO2CH3	4-methylisoxazol-3-yl	Cl	O
839	SO2CH3	4,5-dihydroisoxazol-	Cl	O
		4-yl
840	SO2CH3	3-methyl-4,5-dihydroisoxazol-	Cl	O
		4-yl
841	SO2CH3	isoxazol-4-yl	Cl	O
842	SO2CH3	3-methylisoxazol-4-yl	Cl	O
843	SO2CH3	phenyl	Cl	O
844	SO2CH3	benzyl	Cl	O
845	SO2CH3	benzoyl	Cl	O
846	SO2CH3	2-pyridyl	Cl	O
847	CF3	H	H	O
848	CF3	CH3	H	O
849	CF3	C2H5	H	O
850	CF3	n-C3H7	H	O
851	CF3	i-C3H7	H	O
852	CF3	n-C4H9	H	O
853	CF3	i-C4H9	H	O
854	CF3	s-C4H9	H	O
855	CF3	t-C4H9	H	O
856	CF3	CH2OCH3	H	O
857	CF3	CF3	H	O
858	CF3	CF2H	H	O
859	CF3	CN	H	O
860	CF3	OH	H	O
861	CF3	OCH3	H	O
862	CF3	NH2	H	O
863	CF3	NHCH3	H	O
864	CF3	N(CH3)2	H	O
865	CF3	CO2CH3	H	O
866	CF3	CO2C2H5	H	O
867	CF3	C(O)CH3	H	O
868	CF3	C(O)CF3	H	O
869	CF3	C(═NOCH3)CH3	H	O
870	CF3	SO2CH3	H	O
871	CF3	SO2CF3	H	O
872	CF3	CH2CO2H	H	O
873	CF3	CH2COOCH3	H	O
874	CF3	CH2COOC2H5	H	O
875	CF3	prop-1-en-3-yl	H	O
876	CF3	trans-but-2-en-1-yl	H	O
877	CF3	cis-but-2-en-1-yl	H	O
878	CF3	cis-3-methyl-	H	O
		but-2-en-1-yl
879	CF3	cyclopropyl	H	O
880	CF3	cyclopentyl	H	O
881	CF3	cyclohexyl	H	O
882	CF3	4,5-dihydroisoxazol-	H	O
		3-yl
883	CF3	4-methyl-4,5-dihydroisoxazol-	H	O
		3-yl
884	CF3	isoxazol-3-yl	H	O
885	CF3	4-methylisoxazol-3-yl	H	O
886	CF3	4,5-dihydroisoxazol-	H	O
		4-yl
887	CF3	3-methyl-4,5-dihydroisoxazol-	H	O
		4-yl
888	CF3	isoxazol-4-yl	H	O
889	CF3	3-methylisoxazol-4-yl	H	O
890	CF3	phenyl	H	O
891	CF3	benzyl	H	O
892	CF3	benzoyl	H	O
893	CF3	2-pyridyl	H	O
894	CF3	H	CH3	O
895	CF3	CH3	CH3	O
896	CF3	C2H5	CH3	O
897	CF3	n-C3H7	CH3	O
898	CF3	i-C3H7	CH3	O
899	CF3	n-C4H9	CH3	O
900	CF3	i-C4H9	CH3	O
901	CF3	s-C4H9	CH3	O
902	CF3	t-C4H9	CH3	O
903	CF3	CH2OCH3	CH3	O
904	CF3	CF3	CH3	O
905	CF3	CF2H	CH3	O
906	CF3	CN	CH3	O
907	CF3	OH	CH3	O
908	CF3	OCH3	CH3	O
909	CF3	NH2	CH3	O
910	CF3	NHCH3	CH3	O
911	CF3	N(CH3)2	CH3	O
912	CF3	CO2CH3	CH3	O
913	CF3	CO2C2H5	CH3	O
914	CF3	C(O)CH3	CH3	O
915	CF3	C(O)CF3	CH3	O
916	CF3	C(═NOCH3)CH3	CH3	O
917	CF3	SO2CH3	CH3	O
918	CF3	SO2CF3	CH3	O
919	CF3	CH2CO2H	CH3	O
920	CF3	CH2COOCH3	CH3	O
921	CF3	CH2COOC2H5	CH3	O
922	CF3	prop-1-en-3-yl	CH3	O
923	CF3	trans-but-2-en-1-yl	CH3	O
924	CF3	cis-but-2-en-1-yl	CH3	O
925	CF3	cis-3-methyl-	CH3	O
		but-2-en-1-yl
926	CF3	cyclopropyl	CH3	O
927	CF3	cyclopentyl	CH3	O
928	CF3	cyclohexyl	CH3	O
929	CF3	4,5-dihydroisoxazol-	CH3	O
		3-yl
930	CF3	4-methyl-4,5-dihydroisoxazol-	CH3	O
		3-yl
931	CF3	isoxazol-3-yl	CH3	O
932	CF3	4-methylisoxazol-3-yl	CH3	O
933	CF3	4,5-dihydroisoxazol-	CH3	O
		4-yl
934	CF3	3-methyl-4,5-dihydroisoxazol-	CH3	O
		4-yl
935	CF3	isoxazol-4-yl	CH3	O
936	CF3	3-methylisoxazol-4-yl	CH3	O
937	CF3	phenyl	CH3	O
938	CF3	benzyl	CH3	O
939	CF3	benzoyl	CH3	O
940	CF3	2-pyridyl	CH3	O
941	CF3	H	Cl	O
942	CF3	CH3	Cl	O
943	CF3	C2H5	Cl	O
944	CF3	n-C3H7	Cl	O
945	CF3	i-C3H7	Cl	O
946	CF3	n-C4H9	Cl	O
947	CF3	i-C4H9	Cl	O
948	CF3	s-C4H9	Cl	O
949	CF3	t-C4H9	Cl	O
950	CF3	CH2OCH3	Cl	O
951	CF3	CF3	Cl	O
952	CF3	CF2H	Cl	O
953	CF3	CN	Cl	O
954	CF3	OH	Cl	O
955	CF3	OCH3	Cl	O
956	CF3	NH2	Cl	O
957	CF3	NHCH3	Cl	O
958	CF3	N(CH3)2	Cl	O
959	CF3	CO2CH3	Cl	O
960	CF3	CO2C2H5	Cl	O
961	CF3	C(O)CH3	Cl	O
962	CF3	C(O)CF3	Cl	O
963	CF3	C(═NOCH3)CH3	Cl	O
964	CF3	SO2CH3	Cl	O
965	CF3	SO2CF3	Cl	O
966	CF3	CH2CO2H	Cl	O
967	CF3	CH2COOCH3	Cl	O
968	CF3	CH2COOC2H5	Cl	O
969	CF3	prop-1-en-3-yl	Cl	O
970	CF3	trans-but-2-en-1-yl	Cl	O
971	CF3	cis-but-2-en-1-yl	Cl	O
972	CF3	cis-3-methyl-	Cl	O
		but-2-en-1-yl
973	CF3	cyclopropyl	Cl	O
974	CF3	cyclopentyl	Cl	O
975	CF3	cyclohexyl	Cl	O
976	CF3	4,5-dihydroisoxazol-	Cl	O
		3-yl
977	CF3	4-methyl-4,5-dihydroisoxazol-	Cl	O
		3-yl
978	CF3	isoxazol-3-yl	Cl	O
979	CF3	4-methylisoxazol-3-yl	Cl	O
980	CF3	4,5-dihydroisoxazol-	Cl	O
		4-yl
981	CF3	3-methyl-4,5-dihydroisoxazol-	Cl	O
		4-yl
982	CF3	isoxazol-4-yl	Cl	O
983	CF3	3-methylisoxazol-4-yl	Cl	O
984	CF3	phenyl	Cl	O
985	CF3	benzyl	Cl	O
986	CF3	benzoyl	Cl	O
987	CF3	2-pyridyl	Cl	O
988	C2H5	H	H	O
989	C2H5	CH3	H	O
990	C2H5	C2H5	H	O
991	C2H5	n-C3H7	H	O
992	C2H5	i-C3H7	H	O
993	C2H5	n-C4H9	H	O
994	C2H5	i-C4H9	H	O
995	C2H5	s-C4H9	H	O
996	C2H5	t-C4H9	H	O
997	C2H5	CH2OCH3	H	O
998	C2H5	CF3	H	O
999	C2H5	CF2H	H	O
1000	C2H5	CN	H	O
1001	C2H5	OH	H	O
1002	C2H5	OCH3	H	O
1003	C2H5	NH2	H	O
1004	C2H5	NHCH3	H	O
1005	C2H5	N(CH3)2	H	O
1006	C2H5	CO2CH3	H	O
1007	C2H5	CO2C2H5	H	O
1008	C2H5	C(O)CH3	H	O
1009	C2H5	C(O)CF3	H	O
1010	C2H5	C(═NOCH3)CH3	H	O
1011	C2H5	SO2CH3	H	O
1012	C2H5	SO2CF3	H	O
1013	C2H5	CH2CO2H	H	O
1014	C2H5	CH2COOCH3	H	O
1015	C2H5	CH2COOC2H5	H	O
1016	C2H5	prop-1-en-3-yl	H	O
1017	C2H5	trans-but-2-en-1-yl	H	O
1018	C2H5	cis-but-2-en-1-yl	H	O
1019	C2H5	cis-3-methyl-	H	O
		but-2-en-1-yl
1020	C2H5	cyclopropyl	H	O
1021	C2H5	cyclopentyl	H	O
1022	C2H5	cyclohexyl	H	O
1023	C2H5	4,5-dihydroisoxazol-	H	O
		3-yl
1024	C2H5	4-methyl-4,5-dihydroisoxazol-	H	O
		3-yl
1025	C2H5	isoxazol-3-yl	H	O
1026	C2H5	4-methylisoxazol-3-yl	H	O
1027	C2H5	4,5-dihydroisoxazol-	H	O
		4-yl
1028	C2H5	3-methyl-4,5-dihydroisoxazol-	H	O
		4-yl
1029	C2H5	isoxazol-4-yl	H	O
1030	C2H5	3-methylisoxazol-4-yl	H	O
1031	C2H5	phenyl	H	O
1032	C2H5	benzyl	H	O
1033	C2H5	benzoyl	H	O
1034	C2H5	2-pyridyl	H	O
1035	C2H5	H	CH3	O
1036	C2H5	CH3	CH3	O
1037	C2H5	C2H5	CH3	O
1038	C2H5	n-C3H7	CH3	O
1039	C2H5	i-C3H7	CH3	O
1040	C2H5	n-C4H9	CH3	O
1041	C2H5	i-C4H9	CH3	O
1042	C2H5	s-C4H9	CH3	O
1043	C2H5	t-C4H9	CH3	O
1044	C2H5	CH2OCH3	CH3	O
1045	C2H5	CF3	CH3	O
1046	C2H5	CF2H	CH3	O
1047	C2H5	CN	CH3	O
1048	C2H5	OH	CH3	O
1049	C2H5	OCH3	CH3	O
1050	C2H5	NH2	CH3	O
1051	C2H5	NHCH3	CH3	O
1052	C2H5	N(CH3)2	CH3	O
1053	C2H5	CO2CH3	CH3	O
1054	C2H5	CO2C2H5	CH3	O
1055	C2H5	C(O)CH3	CH3	O
1056	C2H5	C(O)CF3	CH3	O
1057	C2H5	C(═NOCH3)CH3	CH3	O
1058	C2H5	SO2CH3	CH3	O
1059	C2H5	SO2CF3	CH3	O
1060	C2H5	CH2CO2H	CH3	O
1061	C2H5	CH2COOCH3	CH3	O
1062	C2H5	CH2COOC2H5	CH3	O
1063	C2H5	prop-1-en-3-yl	CH3	O
1064	C2H5	trans-but-2-en-1-yl	CH3	O
1065	C2H5	cis-but-2-en-1-yl	CH3	O
1066	C2H5	cis-3-methyl-	CH3	O
		but-2-en-1-yl
1067	C2H5	cyclopropyl	CH3	O
1068	C2H5	cyclopentyl	CH3	O
1069	C2H5	cyclohexyl	CH3	O
1070	C2H5	4,5-dihydroisoxazol-	CH3	O
		3-yl
1071	C2H5	4-nethyl-4,5-dihydroisoxazol-	CH3	O
		3-yl
1072	C2H5	isoxazol-3-yl	CH3	O
1073	C2H5	4-methylisoxazol-3-yl	CH3	O
1074	C2H5	4,5-dihydroisoxazol-	CH3	O
		4-yl
1075	C2H5	3-methyl-4,5-dihydroisoxazol-	CH3	O
		4-yl
1076	C2H5	isoxazol-4-yl	CH3	O
1077	C2H5	3-methylisoxazol-4-yl	CH3	O
1078	C2H5	phenyl	CH3	O
1079	C2H5	benzyl	CH3	O
1080	C2H5	benzoyl	CH3	O
1081	C2H5	2-pyridyl	CH3	O
1082	C2H5	H	Cl	O
1083	C2H5	CH3	Cl	O
1084	C2H5	C2H5	Cl	O
1085	C2H5	n-C3H7	Cl	O
1086	C2H5	i-C3H7	Cl	O
1087	C2H5	n-C4H9	Cl	O
1088	C2H5	i-C4H9	Cl	O
1089	C2H5	s-C4H9	Cl	O
1090	C2H5	t-C4H9	Cl	O
1091	C2H5	CH2OCH3	Cl	O
1092	C2H5	CF3	Cl	O
1093	C2H5	CF2H	Cl	O
1094	C2H5	CN	Cl	O
1095	C2H5	OH	Cl	O
1096	C2H5	OCH3	Cl	O
1097	C2H5	NH2	Cl	O
1098	C2H5	NHCH3	Cl	O
1099	C2H5	N(CH3)2	Cl	O
1100	C2H5	CO2CH3	Cl	O
1101	C2H5	CO2C2H5	Cl	O
1102	C2H5	C(O)CH3	Cl	O
1103	C2H5	C(O)CF3	Cl	O
1104	C2H5	C(═NOCH3)CH3	Cl	O
1105	C2H5	SO2CH3	Cl	O
1106	C2H5	SO2CF3	Cl	O
1107	C2H5	CH2CO2H	Cl	O
1108	C2H5	CH2COOCH3	Cl	O
1109	C2H5	CH2COOC2H5	Cl	O
1110	C2H5	prop-1-en-3-yl	Cl	O
1111	C2H5	trans-but-2-en-1-yl	Cl	O
1112	C2H5	cis-but-2-en-1-yl	Cl	O
1113	C2H5	cis-3-methyl-	Cl	O
		but-2-en-1-yl
1114	C2H5	cyclopropyl	Cl	O
1115	C2H5	cyclopentyl	Cl	O
1116	C2H5	cyclohexyl	Cl	O
1117	C2H5	4,5-dihydroisoxazol-	Cl	O
		3-yl
1118	C2H5	4-methyl-4,5-dihydroisoxazol-	Cl	O
		3-yl
1119	C2H5	isoxazol-3-yl	Cl	O
1120	C2H5	4-methylisoxazol-3-yl	Cl	O
1121	C2H5	4,5-dihydroisoxazol-	Cl	O
		4-yl
1122	C2H5	3-methyl-4,5-dihydroisoxazol-	Cl	O
		4-yl
1123	C2H5	isoxazol-4-yl	Cl	O
1124	C2H5	3-methylisoxazol-4-yl	Cl	O
1125	C2H5	phenyl	Cl	O
1126	C2H5	benzyl	Cl	O
1127	C2H5	benzoyl	Cl	O
1128	C2H5	2-pyridyl	Cl	O
1129	CH3	CH3	H	S
1130	CH3	H	H	S
1131	CH3	C2H5	H	S
1132	CH3	n-C3H7	H	S
1133	CH3	i-C3H7	H	S
1134	CH3	n-C4H9	H	S
1135	CH3	i-C4H9	H	S
1136	CH3	s-C4H9	H	S
1137	CH3	t-C4H9	H	S
1138	CH3	CH2OCH3	H	S
1139	CH3	CF3	H	S
1140	CH3	CF2H	H	S
1141	CH3	CN	H	S
1142	CH3	OH	H	S
1143	CH3	OCH3	H	S
1144	CH3	NH2	H	S
1145	CH3	NHCH3	H	S
1146	CH3	N(CH3)2	H	S
1147	CH3	CO2CH3	H	S
1148	CH3	CO2C2H5	H	S
1149	CH3	C(O)CH3	H	S
1150	CH3	C(O)CF3	H	S
1151	CH3	C(═NOCH3)CH3	H	S
1152	CH3	SO2CH3	H	S
1153	CH3	SO2CF3	H	S
1154	CH3	CH2CO2H	H	S
1155	CH3	CH2COOCH3	H	S
1156	CH3	CH2COOC2H5	H	S
1157	CH3	prop-1-en-3-yl	H	S
1158	CH3	trans-but-2-en-1-yl	H	S
1159	CH3	cis-but-2-en-1-yl	H	S
1160	CH3	cis-3-methyl-	H	S
		but-2-en-1-yl
1161	CH3	cyclopropyl	H	S
1162	CH3	cyclopentyl	H	S
1163	CH3	cyclohexyl	H	S
1164	CH3	4,5-dihydroisoxazol-	H	S
		3-yl
1165	CH3	4-methyl-4,5-dihydroisoxazol-	H	S
		3-yl
1166	CH3	isoxazol-3-yl	H	S
1167	CH3	4-methylisoxazol-3-yl	H	S
1168	CH3	4,5-dihydroisoxazol-	H	S
		4-y1
1169	CH3	3-methyl-4,5-dihydroisoxazol-	H	S
		4-yl
1170	CH3	isoxazol-4-yl	H	S
1171	CH3	3-methylisoxazol-4-yl	H	S
1172	CH3	phenyl	H	S
1173	CH3	benzyl	H	S
1174	CH3	benzoyl	H	S
1175	CH3	2-pyridyl	H	S
1176	CH3	H	CH3	S
1177	CH3	CH3	CH3	S
1178	CH3	C2H5	CH3	S
1179	CH3	n-C3H7	CH3	S
1180	CH3	i-C3H7	CH3	S
1181	CH3	n-C4H9	CH3	S
1182	CH3	i-C4H9	CH3	S
1183	CH3	s-C4H9	CH3	S
1184	CH3	t-C4H9	CH3	S
1185	CH3	CH2OCH3	CH3	S
1186	CH3	CF3	CH3	S
1187	CH3	CF2H	CH3	S
1188	CH3	CN	CH3	S
1189	CH3	OH	CH3	S
1190	CH3	OCH3	CH3	S
1191	CH3	NH2	CH3	S
1192	CH3	NHCH3	CH3	S
1193	CH3	N(CH3)2	CH3	S
1194	CH3	CO2CH3	CH3	S
1195	CH3	CO2C2H5	CH3	S
1196	CH3	C(O)CH3	CH3	S
1197	CH3	C(O)CF3	CH3	S
1198	CH3	C(═NOCH3)CH3	CH3	S
1199	CH3	SO2CH3	CH3	S
1200	CH3	SO2CF3	CH3	S
1201	CH3	CH2CO2H	CH3	S
1202	CH3	CH2COOCH3	CH3	S
1203	CH3	CH2COOC2H5	CH3	S
1204	CH3	prop-1-en-3-yl	CH3	S
1205	CH3	trans-but-2-en-1-yl	CH3	S
1206	CH3	cis-but-2-en-1-yl	CH3	S
1207	CH3	cis-3-methyl-	CH3	S
		but-2-en-1-yl
1208	CH3	cyclopropyl	CH3	S
1209	CH3	cyclopentyl	CH3	S
1210	CH3	cyclohexyl	CH3	S
1211	CH3	4,5-dihydroisoxazol-	CH3	S
		3-yl
1212	CH3	4-methyl-4,5-dihydroisoxazol-	CH3	S
		3-yl
1213	CH3	isoxazol-3-yl	CH3	S
1214	CH3	4-methylisoxazol-3-yl	CH3	S
1215	CH3	4,5-dihydroisoxazol-	CH3	S
		4-yl
1216	CH3	3-methyl-4,5-dihydroisoxazol-	CH3	S
		4-yl
1217	CH3	isoxazol-4-yl	CH3	S
1218	CH3	3-methylisoxazol-4-yl	CH3	S
1219	CH3	phenyl	CH3	S
1220	CH3	benzyl	CH3	S
1221	CH3	benzoyl	CH3	S
1222	CH3	2-pyridyl	CH3	S
1223	CH3	H	Cl	S
1224	CH3	CH3	Cl	S
1225	CH3	C2H5	Cl	S
1226	CH3	n-C3H7	Cl	S
1227	CH3	i-C3H7	Cl	S
1228	CH3	n-C4H9	Cl	S
1229	CH3	i-C4H9	Cl	S
1230	CH3	s-C4H9	Cl	S
1231	CH3	t-C4H9	Cl	S
1232	CH3	CH2OCH3	Cl	S
1233	CH3	CF3	Cl	S
1234	CH3	CF2H	Cl	S
1235	CH3	CN	Cl	S
1236	CH3	OH	Cl	S
1237	CH3	OCH3	Cl	S
1238	CH3	NH2	Cl	S
1239	CH3	NHCH3	Cl	S
1240	CH3	N(CH3)2	Cl	S
1241	CH3	CO2CH3	Cl	S
1242	CH3	CO2C2H5	Cl	S
1243	CH3	C(O)CH3	Cl	S
1244	CH3	C(O)CF3	Cl	S
1245	CH3	C(═NOCH3)CH3	Cl	S
1246	CH3	SO2CH3	Cl	S
1247	CH3	SO2CF3	Cl	S
1248	CH3	CH2CO2H	Cl	S
1249	CH3	CH2COOCH3	Cl	S
1250	CH3	CH2COOC2H5	Cl	S
1251	CH3	prop-1-en-3-yl	Cl	S
1252	CH3	trans-but-2-en-1-yl	Cl	S
1253	CH3	cis-but-2-en-1-yl	Cl	S
1254	CH3	cis-3-methyl-	Cl	S
		but-2-en-1-yl
1255	CH3	cyclopropyl	Cl	S
1256	CH3	cyclopentyl	Cl	S
1257	CH3	cyclohexyl	Cl	S
1258	CH3	4,5-dihydroisoxazol-	Cl	S
		3-yl
1259	CH3	4-methyl-4,5-dihydroisoxazol-	Cl	S
		3-yl
1260	CH3	isoxazol-3-yl	Cl	S
1261	CH3	4-methylisoxazol-3-yl	Cl	S
1262	CH3	4,5-dihydroisoxazol-	Cl	S
		4-yl
1263	CH3	3-methyl-4,5-dihydroisoxazol-	Cl	S
		4-yl
1264	CH3	isoxazol-4-yl	Cl	S
1265	CH3	3-methylisoxazol-4-yl	Cl	S
1266	CH3	phenyl	Cl	S
1267	CH3	benzyl	Cl	S
1268	CH3	benzoyl	Cl	S
1269	CH3	2-pyridyl	Cl	S
1270	Cl	H	H	S
1271	Cl	CH3	H	S
1272	Cl	C2H5	H	S
1273	Cl	n-C3H7	H	S
1274	Cl	i-C3H7	H	S
1275	Cl	n-C4H9	H	S
1276	Cl	i-C4H9	H	S
1277	Cl	s-C4H9	H	S
1278	Cl	t-C4H9	H	S
1279	Cl	CH2OCH3	H	S
1280	Cl	CF3	H	S
1281	Cl	CF2H	H	S
1282	Cl	CN	H	S
1283	Cl	OH	H	S
1284	Cl	OCH3	H	S
1285	Cl	NH2	H	S
1286	Cl	NHCH3	H	S
1287	Cl	N(CH3)2	H	S
1288	Cl	CO2CH3	H	S
1289	Cl	CO2C2H5	H	S
1290	Cl	C(O)CH3	H	S
1291	Cl	C(O)CF3	H	S
1292	Cl	C(═NOCH3)CH3	H	5
1293	Cl	SO2CH3	H	S
1294	Cl	SO2CF3	H	S
1295	Cl	CH2CO2H	H	S
1296	Cl	CH2COOCH3	H	S
1297	Cl	CH2COOC2H5	H	S
1298	Cl	Prop-1-en-3-yl	H	S
1299	Cl	trans-but-2-en-1-yl	H	S
1300	Cl	cis-but-2-en-1-yl	H	S
1301	Cl	cis-3-methyl-	H	S
		but-2-en-1-yl
1302	Cl	cyclopropyl	H	S
1303	Cl	cyclopentyl	H	S
1304	Cl	cyclohexyl	H	S
1305	Cl	4,5-dihydroisoxazol-	H	S
		3-yl
1306	Cl	4-methyl-4,5-dihydroisoxazol-	H	S
		3-yl
1307	Cl	isoxazol-3-yl	H	S
1308	Cl	4-methylisoxazol-3-yl	H	S
1309	Cl	4,5-dihydroisoxazol-	H	S
		4-yl
1310	Cl	3-methyl-4,5-dihydroisoxazol-	H	S
		4-yl
1311	Cl	isoxazol-4-yl	H	S
1312	Cl	3-methylisoxazol-4-yl	H	S
1313	Cl	phenyl	H	S
1314	Cl	benzyl	H	S
1315	Cl	benzoyl	H	S
1316	Cl	2-pyridyl	H	S
1317	Cl	H	CH3	S
1318	Cl	CH3	CH3	S
1319	Cl	C2H5	CH3	S
1320	Cl	n-C3H7	CH3	S
1321	Cl	i-C3H7	CH3	S
1322	Cl	n-C4H9	CH3	S
1323	Cl	i-C4H9	CH3	S
1324	Cl	s-C4H9	CH3	S
1325	Cl	t-C4H9	CH3	S
1326	Cl	CH2OCH3	CH3	S
1327	Cl	CF3	CH3	S
1328	Cl	CF2H	CH3	S
1329	Cl	CN	CH3	S
1330	Cl	OH	CH3	S
1331	Cl	OCH3	CH3	S
1332	Cl	NH2	CH3	S
1333	Cl	NHCH3	CH3	S
1334	Cl	N(CH3)2	CH3	S
1335	Cl	CO2CH3	CH3	S
1336	Cl	CO2C2H5	CH3	S
1337	Cl	C(O)CH3	CH3	S
1338	Cl	C(O)CF3	CH3	S
1339	Cl	C(═NOCH3)CH3	CH3	S
1340	Cl	SO2CH3	CH3	S
1341	Cl	SO2CF3	CH3	S
1342	Cl	CH2CO2H	CH3	S
1343	Cl	CH2COOCH3	CH3	S
1344	Cl	CH2COOC2H5	CH3	S
1345	Cl	prop-1-en-3-yl	CH3	S
1346	Cl	trans-but-2-en-1-yl	CH3	S
1347	Cl	cis-but-2-en-1-yl	CH3	S
1348	Cl	cis-3-methyl-	CH3	S
		but-2-en-1-yl
1349	Cl	cyclopropyl	CH3	S
1350	Cl	cyclopentyl	CH3	S
1351	Cl	cyclohexyl	CH3	S
1352	Cl	4,5-dihydroisoxazol-	CH3	S
		3-yl
1353	Cl	4-methyl-4,5-dihydroisoxazol-	CH3	S
		3-yl
1354	Cl	isoxazol-3-yl	CH3	S
1355	Cl	4-methylisoxazol-3-yl	CH3	S
1356	Cl	4,5-dihydroisoxazol-	CH3	S
		4-yl
1357	Cl	3-methyl-4,5-dihydroisoxazol-	CH3	S
		4-yl
1358	Cl	isoxazol-4-yl	CH3	S
1359	Cl	3-methylisoxazol-4-yl	CH3	S
1360	Cl	phenyl	CH3	S
1361	Cl	benzyl	CH3	S
1362	Cl	benzoyl	CH3	S
1363	Cl	2-pyridyl	CH3	S
1364	Cl	H	Cl	S
1365	Cl	CH3	Cl	S
1366	Cl	C2H5	Cl	S
1367	Cl	n-C3H7	Cl	S
1368	Cl	i-C3H7	Cl	S
1369	Cl	n-C4H9	Cl	S
1370	Cl	i-C4H9	Cl	S
1371	Cl	s-C4H9	Cl	S
1372	Cl	t-C4H9	Cl	S
1373	Cl	CH2OCH3	Cl	S
1374	Cl	CF3	Cl	S
1375	Cl	CF2H	Cl	S
1376	Cl	CN	Cl	S
1377	Cl	OH	Cl	S
1378	Cl	OCH3	Cl	S
1379	Cl	NH2	Cl	S
1380	Cl	NHCH3	Cl	s
1381	Cl	N(CH3)2	Cl	S
1382	Cl	CO2CH3	Cl	S
1383	Cl	CO2C2H5	Cl	S
1384	Cl	C(O)CH3	Cl	S
1385	Cl	C(O)CF3	Cl	S
1386	Cl	C(═NOCH3)CH3	Cl	S
1387	Cl	SO2CH3	Cl	S
1388	Cl	SO2CF3	Cl	S
1389	Cl	CH2CO2H	Cl	S
1390	Cl	CH2COOCH3	Cl	S
1391	Cl	CH2COOC2H5	Cl	S
1392	Cl	prop-1-en-3-yl	Cl	S
1393	Cl	trans-but-2-en-1-yl	Cl	S
1394	Cl	cis-but-2-en-1-yl	Cl	S
1395	Cl	cis-3-methyl-	Cl	S
		but-2-en-1-yl
1396	Cl	cyclopropyl	Cl	S
1397	Cl	cyclopentyl	Cl	S
1398	Cl	cyclohexyl	Cl	S
1399	Cl	4,5-dihydroisoxazol-	Cl	S
		3-yl
1400	Cl	4-methyl-4,5-dihydroisoxazol-	Cl	S
		3-yl
1401	Cl	isoxazol-3-yl	Cl	S
1402	Cl	4-methylisoxazol-3-yl	Cl	S
1403	Cl	4,5-dihydroisoxazol-	Cl	S
		4-yl
1404	Cl	3-methyl-4,5-dihydroisoxazol-	Cl	S
		4-yl
1405	Cl	isoxazol-4-yl	Cl	S
1406	Cl	3-methylisoxazol-4-yl	Cl	S
1407	Cl	phenyl	Cl	S
1408	Cl	benzyl	Cl	S
1409	Cl	benzoyl	Cl	S
1410	Cl	2-pyridyl	Cl	S
1411	OCH3	H	H	S
1412	OCH3	CH3	H	S
1413	OCH3	C2H5	H	S
1414	OCH3	n-C3H7	H	S
1415	OCH3	i-C3H7	H	S
1416	OCH3	n-C4H9	H	S
1417	OCH3	i-C4H9	H	S
1418	OCH3	s-C4H9	H	S
1419	OCH3	t-C4H9	H	S
1420	OCH3	CH2OCH3	H	S
1421	OCH3	CF3	H	S
1422	OCH3	CF2H	H	S
1423	OCH3	CN	H	S
1424	OCH3	OH	H	S
1425	OCH3	OCH3	H	S
1426	OCH3	NH2	H	S
1427	OCH3	NHCH3	H	S
1428	OCH3	N(CH3)2	H	S
1429	OCH3	CO2CH3	H	S
1430	OCH3	CO2C2H5	H	5
1431	OCH3	C(O)CH3	H	S
1432	OCH3	C(O)CF3	H	S
1433	OCH3	C(═NOCH3)CH3	H	S
1434	OCH3	SO2CH3	H	S
1435	OCH3	SO2CF3	H	S
1436	OCH3	CH2CO2H	H	S
1437	OCH3	CH2COOCH3	H	S
1438	OCH3	CH2COOC2H5	H	S
1439	OCH3	prop-1-en-3-yl	H	S
1440	OCH3	trans-but-2-en-1-yl	H	S
1441	OCH3	cis-but-2-en-1-yl	H	S
1442	OCH3	cis-3-methyl-	H	S
		but-2-en-1-yl
1443	OCH3	cyclopropyl	H	S
1444	OCH3	cyclopentyl	H	S
1445	OCH3	cyclohexyl	H	S
1446	OCH3	4,5-dihydroisoxazol-	H	S
		3-yl
1447	OCH3	4-methyl-4,5-dihydroisoxazol-	H	S
		3-yl
1448	OCH3	isoxazol-3-yl	H	S
1449	OCH3	4-methylisoxazol-3-yl	H	S
1450	OCH3	4,5-dihydroisoxazol-	H	S
		4-yl
1451	OCH3	3-methyl-4,5-dihydroisoxazol-	H	S
		4 -yl
1452	OCH3	isoxazol-4-yl	H	S
1453	OCH3	3-methylisoxazol-4-yl	H	S
1454	OCH3	phenyl	H	S
1455	OCH3	benzyl	H	S
1456	OCH3	benzoyl	H	S
1457	OCH3	2-pyridyl	H	S
1458	OCH3	H	CH3	S
1459	OCH3	CH3	CH3	S
1460	OCH3	C2H5	CH3	S
1461	OCH3	n-C3H7	CH3	S
1462	OCH3	i-C3H7	CH3	S
1463	OCH3	n-C4H9	CH3	S
1464	OCH3	i-C4H9	CH3	S
1465	OCH3	s-C4H9	CH3	S
1466	OCH3	t-C4H9	CH3	S
1467	OCH3	CH2OCH3	CH3	S
1468	OCH3	CF3	CH3	S
1469	OCH3	CF2H	CH3	S
1470	OCH3	CN	CH3	S
1471	OCH3	OH	CH3	S
1472	OCH3	OCH3	CH3	S
1473	OCH3	NH2	CH3	S
1474	OCH3	NHCH3	CH3	S
1475	OCH3	N(CH3)2	CH3	S
1476	OCH3	CO2CH3	CH3	S
1477	OCH3	CO2C2H5	CH3	S
1478	OCH3	C(O)CH3	CH3	S
1479	OCH3	C(O)CF3	CH3	S
1480	OCH3	C(═NOCH3)CH3	CH3	S
1481	OCH3	SO2CH3	CH3	S
1482	OCH3	SO2CF3	CH3	S
1483	OCH3	CH2CO2H	CH3	S
1484	OCH3	CH2COOCH3	CH3	S
1485	OCH3	CH2COOC2H5	CH3	S
1486	OCH3	prop-1-en-3-yl	CH3	S
1487	OCH3	trans-but-2-en-1-yl	CH3	S
1488	OCH3	cis-but-2-en-1-yl	CH3	S
1489	OCH3	cis-3-methyl-	CH3	S
		but-2-en-1-yl
1490	OCH3	cyclopropyl	CH3	S
1491	OCH3	cyclopentyl	CH3	S
1492	OCH3	cyclohexyl	CH3	S
1493	OCH3	4,5-dihydroisoxazol-	CH3	S
		3-yl
1494	OCH3	4-methyl-4,5-dihydroisoxazol-	CH3	S
		3-yl
1495	OCH3	isoxazol-3-yl	CH3	S
1496	OCH3	4-methylisoxazol-3-yl	CH3	S
1497	OCH3	4,5-dihydroisoxazol- CH3	S
		4-yl
1498	OCH3	3-methyl-4,5-dihydroisoxazol-	CH3	S
		4-yl
1499	OCH3	isoxazol-4-yl	CH3	S
1500	OCH3	3-methylisoxazol-4-yl	CH3	S
1501	OCH3	phenyl	CH3	S
1502	OCH3	benzyl	CH3	S
1503	OCH3	benzoyl	CH3	S
1504	OCH3	2-pyridyl	CH3	S
1505	OCH3	H	Cl	S
1506	OCH3	CH3	Cl	S
1507	OCH3	C2H5	Cl	S
1508	OCH3	n-C3H7	Cl	S
1509	OCH3	i-C3H7	Cl	S
1510	OCH3	n-C4H9	Cl	S
1511	OCH3	i-C4H9	Cl	S
1512	OCH3	s-C4H9	Cl	S
1513	OCH3	t-C4H9	Cl	S
1514	OCH3	CH2OCH3	Cl	S
1515	OCH3	CF3	Cl	S
1516	OCH3	CF2H	Cl	S
1517	OCH3	CN	Cl	S
1518	OCH3	OH	Cl	S
1519	OCH3	OCH3	Cl	S
1520	OCH3	NH2	Cl	S
1521	OCH3	NHCH3	Cl	S
1522	OCH3	N(CH3)2	Cl	S
1523	OCH3	CO2CH3	Cl	S
1524	OCH3	CO2C2H5	Cl	S
1525	OCH3	C(O)CH3	Cl	S
1526	OCH3	C(O)CF3	Cl	S
1527	OCH3	C(═NOCH3)CH3	Cl	S
1528	OCH3	SO2CH3	Cl	S
1529	OCH3	SO2CF3	Cl	S
1530	OCH3	CH2CO2H	Cl	S
1531	OCH3	CH2COOCH3	Cl	S
1532	OCH3	CH2COOC2H5	Cl	S
1533	OCH3	prop-1-en-3-yl	Cl	S
1534	OCH3	trans-but-2-en-1-yl	Cl	S
1535	OCH3	cis-but-2-en-1-yl	Cl	S
1536	OCH3	cis-3-methyl-	Cl	S
		but-2-en-1-yl
1537	OCH3	cyclopropyl	Cl	S
1538	OCH3	cyclopentyl	Cl	S
1539	OCH3	cyclohexyl	Cl	S
1540	OCH3	4,5-dihydroisoxazol-	Cl	S
		3-yl
1541	OCH3	4-methyl-4,5-dihydroisoxazol-	Cl	S
		3-yl
1542	OCH3	isoxazol-3-yl	Cl	S
1543	OCH3	4-methylisoxazol-3-yl	Cl	S
1544	OCH3	4,5-dihydroisoxazol-	Cl	S
		4-yl
1545	OCH3	3-methyl-4,5-dihydroisoxazol-	Cl	S
		4-yl
1546	OCH3	isoxazol-4-yl	Cl	S
1547	OCH3	3-methylisoxazol-4-yl	Cl	S
1548	OCH3	phenyl	Cl	S
1549	OCH3	benzyl	Cl	S
1550	OCH3	benzoyl	Cl	S
1551	OCH3	2-pyridyl	Cl	S
1552	OCF3	H	H	S
1553	OCF3	CH3	H	S
1554	OCF3	C2H5	H	S
1555	OCF3	n-C3H7	H	S
1556	OCF3	i-C3H7	H	S
1557	OCF3	n-C4H9	H	S
1558	OCF3	i-C4H9	H	S
1559	OCF3	s-C4H9	H	S
1560	OCF3	t-C4H9	H	S
1561	OCF3	CH2OCH3	H	S
1562	OCF3	CF3	H	S
1563	OCF3	CF2H	H	S
1564	OCF3	CN	H	S
1565	OCF3	OH	H	S
1566	OCF3	OCH3	H	S
1567	OCF3	NH2	H	S
1568	OCF3	NHCH3	H	S
1569	OCF3	N(CH3)2	H	S
1570	OCF3	CO2CH3	H	S
1571	OCF3	CO2C2H5	H	S
1572	OCF3	C(O)CH3	H	S
1573	OCF3	C(O)CF3	H	S
1574	OCF3	C(═NOCH3)CH3	H	S
1575	OCF3	SO2CH3	H	S
1576	OCF3	SO2CF3	H	S
1577	OCF3	CH2CO2H	H	S
1578	OCF3	CH2COOCH3	H	S
1579	OCF3	CH2COOC2H5	H	S
1580	OCF3	prop-1-en-3-yl	H	S
1581	OCF3	trans-but-2-en-1-yl	H	S
1582	OCF3	cis-but-2-en-1-yl	H	S
1583	OCF3	cis-3-methyl-	H	S
		but-2-en-1-yl
1584	OCF3	cyclopropyl	H	S
1585	OCF3	cyclopentyl	H	S
1586	OCF3	cyclohexyl	H	S
1587	OCF3	4,5-dihydroisoxazol-	H	S
		3-yl
1588	OCF3	4-methyl-4,5-dihydroisoxazol-	H	S
		3-yl
1589	OCF3	isoxazol-3-yl	H	S
1590	OCF3	4-methylisoxazol-3-yl	H	S
1591	OCF3	4,5-dihydroisoxazol-	H	S
		4-yl
1592	OCF3	3-methyl-4,5-dihydroisoxazol-	H	S
		4-yl
1593	OCF3	isoxazol-4-yl	H	S
1594	OCF3	3-methylisoxazol-4-yl	H	S
1595	OCF3	phenyl	H	S
1596	OCF3	benzyl	H	S
1597	OCF3	benzoyl	H	S
1598	OCF3	2-pyridyl	H	S
1599	OCF3	H	CH3	S
1600	OCF3	CH3	CH3	S
1601	OCF3	C2H5	CH3	S
1602	OCF3	n-C3H7	CH3	S
1603	OCF3	i-C3H7	CH3	S
1604	OCF3	n-C4H9	CH3	S
1605	OCF3	i-C4H9	CH3	S
1606	OCF3	s-C4H9	CH3	S
1607	OCF3	t-C4H9	CH3	S
1608	OCF3	CH2OCH3	CH3	S
1609	OCF3	CF3	CH3	S
1610	OCF3	CF2H	CH3	S
1611	OCF3	CN	CH3	S
1612	OCF3	OH	CH3	S
1613	OCF3	OCH3	CH3	S
1614	OCF3	NH2	CH3	S
1615	OCF3	NHCH3	CH3	S
1616	OCF3	N(CH3)2	CH3	S
1617	OCF3	CO2CH3	CH3	S
1618	OCF3	CO2C2H5	CH3	S
1619	OCF3	C(O)CH3	CH3	S
1620	OCF3	C(O)CF3	CH3	S
1621	OCF3	C(═NOCH3)CH3	CH3	S
1622	OCF3	SO2CH3	CH3	S
1623	OCF3	SO2CF3	CH3	S
1624	OCF3	CH2CO2H	CH3	S
1625	OCF3	CH2COOCH3	CH3	S
1626	OCF3	CH2COOC2H5	CH3	S
1627	OCF3	prop-1-en-3-yl	CH3	S
1628	OCF3	trans-but-2-en-1-yl	CH3	S
1629	OCF3	cis-but-2-en-1-yl	CH3	S
1630	OCF3	cis-3-methyl-	CH3	S
		but-2-en-1-yl
1631	OCF3	cyclopropyl	CH3	S
1632	OCF3	cyclopentyl	CH3	S
1633	OCF3	cyclohexyl	CH3	S
1634	OCF3	4,5-dihydroisoxazol-	CH3	S
		3-yl
1635	OCF3	4-methyl-4,5-dihydroisoxazol-	CH3	S
		3-yl
1636	OCF3	isoxazol-3-yl	CH3	S
1637	OCF3	4-methylisoxazol-3-yl	CH3	S
1638	OCF3	4,5-dihydroisoxazol-	CH3	S
		4-yl
1639	OCF3	3-methyl-4,5-dihydroisoxazol-	CH3	S
		4-yl
1640	OCF3	isoxazol-4-yl	CH3	S
1641	OCF3	3-methylisoxazol-4-yl	CH3	S
1642	OCF3	phenyl	CH3	S
1643	OCF3	benzyl	CH3	S
1644	OCF3	benzoyl	CH3	S
1645	OCF3	2-pyridyl	CH3	S
1646	OCF3	H	Cl	S
1647	OCF3	CH3	Cl	S
1648	OCF3	C2H5	Cl	S
1649	OCF3	n-C3H7	Cl	S
1650	OCF3	i-C3H7	Cl	S
1651	OCF3	n-C4H9	Cl	S
1652	OCF3	i-C4H9	Cl	S
1653	OCF3	s-C4H9	Cl	S
1654	OCF3	t-C4H9	Cl	S
1655	OCF3	CH2OCH3	Cl	S
1656	OCF3	CF3	Cl	S
1657	OCF3	CF2H	Cl	S
1658	OCF3	CN	Cl	S
1659	OCF3	OH	Cl	S
1660	OCF3	OCH3	Cl	S
1661	OCF3	NH2	Cl	S
1662	OCF3	NHCH3	Cl	S
1663	OCF3	N(CH3)2	Cl	S
1664	OCF3	CO2CH3	Cl	S
1665	OCF3	CO2C2H5	Cl	S
1666	OCF3	C(O)CH3	Cl	S
1667	OCF3	C(O)CF3	Cl	S
1668	OCF3	C(═NOCH3)CH3	Cl	S
1669	OCF3	SO2CH3	Cl	S
1670	OCF3	SO2CF3	Cl	S
1671	OCF3	CH2CO2H	Cl	S
1672	OCF3	CH2COOCH3	Cl	S
1673	OCF3	CH2COOC2H5	Cl	S
1674	OCF3	prop-1-en-3-yl	Cl	S
1675	OCF3	trans-but-2-en-1-yl	Cl	S
1676	OCF3	cis-but-2-en-1-yl	Cl	S
1677	OCF3	cis-3-methyl-	Cl	S
		but-2-en-1-yl
1678	OCF3	cyclopropyl	Cl	S
1679	OCF3	cyclopentyl	Cl	S
1680	OCF3	cyclohexyl	Cl	S
1681	OCF3	4,5-dihydroisoxazol-	Cl	S
		3-yl
1682	OCF3	4-methyl-4,5-dihydroisoxazol-	Cl	S
		3-yl
1683	OCF3	isoxazol-3-yl	Cl	S
1684	OCF3	4-methylisoxazol-3-yl	Cl	S
1685	OCF3	4,5-dihydroisoxazol-	Cl	S
		4-yl
1686	OCF3	3-methyl-4,5-dihydroisoxazol-	Cl	S
		4-yl
1687	OCF3	isoxazol-4-yl	Cl	S
1688	OCF3	3-methylisoxazol-4-yl	Cl	S
1689	OCF3	phenyl	Cl	S
1690	OCF3	benzyl	Cl	S
1691	OCF3	benzoyl	Cl	S
1692	OCF3	2-pyridyl	Cl	S
1693	SCH3	H	H	S
1694	SCH3	CH3	H	S
1695	SCH3	C2H5	H	S
1696	SCH3	n-C3H7	H	S
1697	SCH3	i-C3H7	H	S
1698	SCH3	n-C4H9	H	S
1699	SCH3	i-C4H9	H	S
1700	SCH3	s-C4H9	H	S
1701	SCH3	t-C4H9	H	S
1702	SCH3	CH2OCH3	H	S
1703	SCH3	CF3	H	S
1704	SCH3	CF2H	H	S
1705	SCH3	CN	H	S
1706	SCH3	OH	H	S
1707	SCH3	OCH3	H	S
1708	SCH3	NH2	H	S
1709	SCH3	NHCH3	H	S
1710	SCH3	N(CH3)2	H	S
1711	SCH3	CO2CH3	H	S
1712	SCH3	CO2C2H5	H	S
1713	SCH3	C(O)CH3	H	S
1714	SCH3	C(O)CF3	H	S
1715	SCH3	C(═NOCH3)CH3	H	S
1716	SCH3	SO2CH3	H	S
1717	SCH3	SO2CF3	H	S
1718	SCH3	CH2CO2H	H	S
1719	SCH3	CH2COOCH3	H	S
1720	SCH3	CH2COOC2H5	H	S
1721	SCH3	prop-1-en-3-yl	H	S
1722	SCH3	trans-but-2-en-1-yl	H	S
1723	SCH3	cis-but-2-en-1-yl	H	S
1724	SCH3	cis-3-methyl-	H	S
		but-2-en-1-yl
1725	SCH3	cyclopropyl	H	S
1726	SCH3	cyclopentyl	H	S
1727	SCH3	cyclohexyl	H	S
1728	SCH3	4,5-dihydroisoxazol-	H	S
		3-yl
1729	SCH3	4-methyl-4,5-dihydroisoxazol-	H	S
		3-yl
1730	SCH3	isoxazol-3-yl	H	S
1731	SCH3	4-methylisoxazol-3-yl	H	S
1732	SCH3	4,5-dihydroisoxazol-	H	S
		4-yl
1733	SCH3	3-methyl-4,5-dihydroisoxazol-	H	S
		4-yl
1734	SCH3	isoxazol-4-yl	H	S
1735	SCH3	3-methylisoxazol-4-yl	H	S
1736	SCH3	phenyl	H	S
1737	SCH3	benzyl	H	S
1738	SCH3	benzoyl	H	S
1739	SCH3	2-pyridyl	H	S
1740	SCH3	H	CH3	S
1741	SCH3	CH3	CH3	S
1742	SCH3	C2H5	CH3	S
1743	SCH3	n-C3H7	CH3	S
1744	SCH3	i-C3H7	CH3	S
1745	SCH3	n-C4H9	CH3	S
1746	SCH3	i-C4H9	CH3	S
1747	SCH3	s-C4H9	CH3	S
1748	SCH3	t-C4H9	CH3	S
1749	SCH3	CH2OCH3	CH3	S
1750	SCH3	CF3	CH3	S
1751	SCH3	CF2H	CH3	S
1752	SCH3	CN	CH3	S
1753	SCH3	OH	CH3	S
1754	SCH3	OCH3	CH3	S
1755	SCH3	NH2	CH3	S
1756	SCH3	NHCH3	CH3	S
1757	SCH3	N(CH3)2	CH3	S
1758	SCH3	CO2CH3	CH3	S
1759	SCH3	CO2C2H5	CH3	S
1760	SCH3	C(O)CH3	CH3	S
1761	SCH3	C(O)CF3	CH3	S
1762	SCH3	C(═NOCH3)CH3	CH3	S
1763	SCH3	SO2CH3	CH3	S
1764	SCH3	SO2CF3	CH3	S
1765	SCH3	CH2CO2H	CH3	S
1766	SCH3	CH2COOCH3	CH3	S
1767	SCH3	CH2COOC2H5	CH3	S
1768	SCH3	prop-1-en-3-yl	CH3	S
1769	SCH3	trans-but-2-en-1-yl	CH3	S
1770	SCH3	cis-but-2-en-1-yl	CH3	S
1771	SCH3	cis-3-methyl-	CH3	S
		but-2-en-1-yl
1772	SCH3	cyclopropyl	CH3	S
1773	SCH3	cyclopentyl	CH3	S
1774	SCH3	cyclohexyl	CH3	S
1775	SCH3	4,5-dihydroisoxazol-	CH3	S
		3-yl
1776	SCH3	4-methyl-4,5-dihydroisoxazol-	CH3	S
		3-yl
1777	SCH3	isoxazol-3-yl	CH3	S
1778	SCH3	4-methylisoxazol-3-yl	CH3	S
1779	SCH3	4,5-dihydroisoxazol-	CH3	S
		4-yl
1780	SCH3	3-methyl-4,5-dihydroisoxazol-	CH3	S
		4-yl
1781	SCH3	isoxazol-4-yl	CH3	S
1782	SCH3	3-methylisoxazol-4-yl	CH3	S
1783	SCH3	phenyl	CH3	S
1784	SCH3	benzyl	CH3	S
1785	SCH3	benzoyl	CH3	S
1786	SCH3	2-pyridyl	CH3	S
1787	SCH3	H	Cl	S
1788	SCH3	CH3	Cl	S
1789	SCH3	C2H5	Cl	S
1790	SCH3	n-C3H7	Cl	S
1791	SCH3	i-C3H7	Cl	S
1792	SCH3	n-C4H9	Cl	S
1793	SCH3	i-C4H9	Cl	S
1794	SCH3	s-C4H9	Cl	S
1795	SCH3	t-C4H9	Cl	S
1796	SCH3	CH2OCH3	Cl	S
1797	SCH3	CF3	Cl	S
1798	SCH3	CF2H	Cl	S
1799	SCH3	CN	Cl	S
1800	SCH3	OH	Cl	S
1801	SCH3	OCH3	Cl	S
1802	SCH3	NH2	Cl	S
1803	SCH3	NHCH3	Cl	S
1804	SCH3	N(CH3)2	Cl	S
1805	SCH3	CO2CH3	Cl	S
1806	SCH3	CO2C2H5	Cl	S
1807	SCH3	C(O)CH3	Cl	S
1808	SCH3	C(O)CF3	Cl	S
1809	SCH3	C(═NOCH3)CH3	Cl	S
1810	SCH3	SO2CH3	Cl	S
1811	SCH3	SO2CF3	Cl	S
1812	SCH3	CH2CO2H	Cl	S
1813	SCH3	CH2COOCH3	Cl	S
1814	SCH3	CH2COOC2H5	Cl	S
1815	SCH3	prop-1-en-3-yl	Cl	S
1816	SCH3	trans-but-2-en-1-yl	Cl	S
1817	SCH3	cis-but-2-en-1-yl	Cl	S
1818	SCH3	cis-3-methyl-	Cl	S
		but-2-en-1-yl
1819	SCH3	cyclopropyl	Cl	S
1820	SCH3	cyclopentyl	Cl	S
1821	SCH3	cyclohexyl	Cl	S
1822	SCH3	4,5-dihydroisoxazol-	Cl	S
		3-yl
1823	SCH3	4-methyl-4,5-dihydroisoxazol-	Cl	S
		3-yl
1824	SCH3	isoxazol-3-yl	Cl	S
1825	SCH3	4-methylisoxazol-3-yl	Cl	S
1826	SCH3	4,5-dihydroisoxazol-	Cl	S
		4-yl
1827	SCH3	3-methyl-4,5-dihydroisoxazol-	Cl	S
		4-yl
1828	SCH3	isoxazol-4-yl	Cl	S
1829	SCH3	3-methylisoxazol-4-yl	Cl	S
1830	SCH3	phenyl	Cl	S
1831	SCH3	benzyl	Cl	S
1832	SCH3	benzoyl	Cl	S
1833	SCH3	2-pyridyl	Cl	S
1834	SO2CH3	H	H	S
1835	SO2CH3	CH3	H	S
1836	SO2CH3	C2H5	H	S
1837	SO2CH3	n-C3H7	H	S
1838	SO2CH3	i-C3H7	H	S
1839	SO2CH3	n-C4H9	H	S
1840	SO2CH3	i-C4H9	H	S
1841	SO2CH3	s-C4H9	H	S
1842	SO2CH3	t-C4H9	H	S
1843	SO2CH3	CH2OCH3	H	S
1844	SO2CH3	CF3	H	S
1845	SO2CH3	CF2H	H	S
1846	SO2CH3	CN	H	S
1847	SO2CH3	OH	H	S
1848	SO2CH3	OCH3	H	S
1849	SO2CH3	NH2	H	S
1850	SO2CH3	NHCH3	H	S
1851	SO2CH3	N(CH3)2	H	S
1852	SO2CH3	CO2CH3	H	S
1853	SO2CH3	CO2C2H5	H	S
1854	SO2CH3	C(O)CH3	H	S
1855	SO2CH3	C(O)CF3	H	S
1856	SO2CH3	C(═NOCH3)CH3	H	S
1857	SO2CH3	SO2CH3	H	S
1858	SO2CH3	SO2CF3	H	S
1859	SO2CH3	CH2CO2H	H	S
1860	SO2CH3	CH2COOCH3	H	S
1861	SO2CH3	CH2COOC2H5	H	S
1862	SO2CH3	prop-1-en-3-yl	H	S
1863	SO2CH3	trans-but-2-en-1-yl	H	S
1864	SO2CH3	cis-but-2-en-1-yl	H	S
1865	SO2CH3	cis-3-methyl-	H	S
		but-2-en-1-yl
1866	SO2CH3	cyclopropyl	H	S
1867	SO2CH3	cyclopentyl	H	S
1868	SO2CH3	cyclohexyl	H	S
1869	SO2CH3	4,5-dihydroisoxazol-	H	S
		3-yl
1870	SO2CH3	4-methyl-4,5-dihydroisoxazol-	H	S
		3-yl
1871	SO2CH3	isoxazol-3-yl	H	S
1872	SO2CH3	4-methylisoxazol-3-yl	H	S
1873	SO2CH3	4,5-dihydroisoxazol-	H	S
		4-yl
1874	SO2CH3	3-methyl-4,5-dihydroisoxazol-	H	S
		4-yl
1875	SO2CH3	isoxazol-4-yl	H	S
1876	SO2CH3	3-methylisoxazol-4-yl	H	S
1877	SO2CH3	phenyl	H	S
1878	SO2CH3	benzyl	H	S
1879	SO2CH3	benzoyl	H	S
1880	SO2CH3	2-pyridyl	H	S
1881	SO2CH3	H	CH3	S
1882	SO2CH3	CH3	CH3	S
1883	SO2CH3	C2H5	CH3	S
1884	SO2CH3	n-C3H7	CH3	S
1885	SO2CH3	i-C3H7	CH3	S
1886	SO2CH3	n-C4H9	CH3	S
1887	SO2CH3	i-C4H9	CH3	S
1888	SO2CH3	s-C4H9	CH3	S
1889	SO2CH3	t-C4H9	CH3	S
1890	SO2CH3	CH2OCH3	CH3	S
1891	SO2CH3	CF3	CH3	S
1892	SO2CH3	CF2H	CH3	S
1893	SO2CH3	CN	CH3	S
1894	SO2CH3	OH	CH3	S
1895	SO2CH3	OCH3	CH3	S
1896	SO2CH3	NH2	CH3	S
1897	SO2CH3	NHCH3	CH3	S
1898	SO2CH3	N(CH3)2	CH3	S
1899	SO2CH3	CO2CH3	CH3	S
1900	SO2CH3	CO2C2H5	CH3	S
1901	SO2CH3	C(O)CH3	CH3	S
1902	SO2CH3	C(O)CF3	CH3	S
1903	SO2CH3	C(═NOCH3)CH3	CH3	S
1904	SO2CH3	SO2CH3	CH3	S
1905	SO2CH3	SO2CF3	CH3	S
1906	SO2CH3	CH2CO2H	CH3	S
1907	SO2CH3	CH2COOCH3	CH3	S
1908	SO2CH3	CH2COOC2H5	CH3	S
1909	SO2CH3	prop-1-en-3-yl	CH3	S
1910	SO2CH3	trans-but-2-en-1-yl	CH3	S
1911	SO2CH3	cis-but-2-en-1-yl	CH3	S
1912	SO2CH3	cis-3-methyl-	CH3	S
		but-2-en-1-yl
1913	SO2CH3	cyclopropyl	CH3	S
1914	SO2CH3	cyclopentyl	CH3	S
1915	SO2CH3	cyclohexyl	CH3	S
1916	SO2CH3	4,5-dihydroisoxazol-	CH3	S
		3-yl
1917	SO2CH3	4-methyl-4,5-dihydroisoxazol-	CH3	S
		3-yl
1918	SO2CH3	isoxazol-3-yl	CH3	S
1919	SO2CH3	4-methylisoxazol-3-yl	CH3	S
1920	SO2CH3	4,5-dihydroisoxazol-	CH3	S
		4-yl
1921	SO2CH3	3-methyl-4,5-dihydroisoxazol-	CH3	S
		4-yl
1922	SO2CH3	isoxazol-4-yl	CH3	S
1923	SO2CH3	3-methylisoxazol-4-yl	CH3	S
1924	SO2CH3	phenyl	CH3	S
1925	SO2CH3	benzyl	CH3	S
1926	SO2CH3	benzoyl	CH3	S
1927	SO2CH3	2-pyridyl	CH3	S
1928	SO2CH3	H	Cl	S
1929	SO2CH3	CH3	Cl	S
1930	SO2CH3	C2H5	Cl	S
1931	SO2CH3	n-C3H7	Cl	S
1932	SO2CH3	i-C3H7	Cl	S
1933	SO2CH3	n-C4H9	Cl	S
1934	SO2CH3	i-C4H9	Cl	S
1935	SO2CH3	s-C4H9	Cl	S
1936	SO2CH3	t-C4H9	Cl	S
1937	SO2CH3	CH2OCH3	Cl	S
1938	SO2CH3	CF3	Cl	S
1939	SO2CH3	CF2H	Cl	S
1940	SO2CH3	CN	Cl	S
1941	SO2CH3	OH	Cl	S
1942	SO2CH3	OCH3	Cl	S
1943	SO2CH3	NH2	Cl	S
1944	SO2CH3	NHCH3	Cl	S
1945	SO2CH3	N(CH3)2	Cl	S
1946	SO2CH3	CO2CH3	Cl	S
1947	SO2CH3	CO2C2H5	Cl	S
1948	SO2CH3	C(O)CH3	Cl	S
1949	SO2CH3	C(O)CF3	Cl	S
1950	SO2CH3	C(═NOCH3)CH3	Cl	S
1951	SO2CH3	SO2CH3	Cl	S
1952	SO2CH3	SO2CF3	Cl	S
1953	SO2CH3	CH2CO2H	Cl	S
1954	SO2CH3	CH2COOCH3	Cl	S
1955	SO2CH3	CH2COOC2H5	Cl	S
1956	SO2CH3	prop-1-en-3-yl	Cl	S
1957	SO2CH3	trans-but-2-en-1-yl	Cl	S
1958	SO2CH3	cis-but-2-en-1-yl	Cl	S
1959	SO2CH3	cis-3-methyl-	Cl	S
		but-2-en-1-yl
1960	SO2CH3	cyclopropyl	Cl	S
1961	SO2CH3	cyclopentyl	Cl	S
1962	SO2CH3	cyclohexyl	Cl	S
1963	SO2CH3	4,5-dihydroisoxazol-	Cl	S
		3-yl
1964	SO2CH3	4-methyl-4,5-dihydroisoxazol-	Cl	S
		3-yl
1965	SO2CH3	isoxazol-3-yl	Cl	S
1966	SO2CH3	4-methylisoxazol-3-yl	Cl	S
1967	SO2CH3	4,5-dihydroisoxazol-	Cl	S
		4-yl
1968	SO2CH3	3-methyl-4,5-dihydroisoxazol-	Cl	S
		4-yl
1969	SO2CH3	isoxazol-4-yl	Cl	S
1970	SO2CH3	3-methylisoxazol-4-yl	Cl	S
1971	SO2CH3	phenyl	Cl	S
1972	SO2CH3	benzyl	Cl	S
1973	SO2CH3	benzoyl	Cl	S
1974	SO2CH3	2-pyridyl	Cl	S
1975	CF3	H	H	S
1976	CF3	CH3	H	S
1977	CF3	C2H5	H	S
1978	CF3	n-C3H7	H	S
1979	CF3	i-C3H7	H	S
1980	CF3	n-C4H9	H	S
1981	CF3	i-C4H9	H	S
1982	CF3	s-C4H9	H	S
1983	CF3	t-C4H9	H	S
1984	CF3	CH2OCH3	H	S
1985	CF3	CF3	H	S
1986	CF3	CF2H	H	S
1987	CF3	CN	H	S
1988	CF3	OH	H	S
1989	CF3	OCH3	H	S
1990	CF3	NH2	H	S
1991	CF3	NHCH3	H	S
1992	CF3	N(CH3)2	H	S
1993	CF3	CO2CH3	H	S
1994	CF3	CO2C2H5	H	S
1995	CF3	C(O)CH3	H	S
1996	CF3	C(O)CF3	H	S
1997	CF3	C(═NOCH3)CH3	H	S
1998	CF3	SO2CH3	H	S
1999	CF3	SO2CF3	H	S
2000	CF3	CH2CO2H	H	S
2001	CF3	CH2COOCH3	H	S
2002	CF3	CH2COOC2H5	H	S
2003	CF3	prop-1-en-3-yl	H	S
2004	CF3	trans-but-2-en-1-yl	H	S
2005	CF3	cis-but-2-en-1-yl	H	S
2006	CF3	cis-3-methyl-	H	S
		but-2-en-1-yl
2007	CF3	cyclopropyl	H	S
2008	CF3	cyclopentyl	H	S
2009	CF3	cyclohexyl	H	S
2010	CF3	4,5-dihydroisoxazol-	H	S
		3-yl
2011	CF3	4-methyl-4,5-dihydroisoxazol-	H	S
		3-yl
2012	CF3	isoxazol-3-yl	H	S
2013	CF3	4-methylisoxazol-3-yl	H	S
2014	CF3	4,5-dihydroisoxazol-	H	S
		4-yl
2015	CF3	3-methyl-4,5-dihydroisoxazol-	H	S
		4-yl
2016	CF3	isoxazol-4-yl	H	S
2017	CF3	3-methylisoxazol-4-yl	H	S
2018	CF3	phenyl	H	S
2019	CF3	benzyl	H	S
2020	CF3	benzoyl	H	S
2021	CF3	2-pyridyl	H	S
2022	CF3	H	CH3	S
2023	CF3	CH3	CH3	S
2024	CF3	C2H5	CH3	S
2025	CF3	n-C3H7	CH3	S
2026	CF3	i-C3H7	CH3	S
2027	CF3	n-C4H9	CH3	S
2028	CF3	i-C4H9	CH3	S
2029	CF3	s-C4H9	CH3	S
2030	CF3	t-C4H9	CH3	S
2031	CF3	CH2OCH3	CH3	S
2032	CF3	CF3	CH3	S
2033	CF3	CF2H	CH3	S
2034	CF3	CN	CH3	S
2035	CF3	OH	CH3	S
2036	CF3	OCH3	CH3	S
2037	CF3	NH2	CH3	S
2038	CF3	NHCH3	CH3	S
2039	CF3	N(CH3)2	CH3	S
2040	CF3	CO2CH3	CH3	S
2041	CF3	CO2C2H5	CH3	S
2042	CF3	C(O)CH3	CH3	S
2043	CF3	C(O)CF3	CH3	S
2044	CF3	C(═NOCH3)CH3	CH3	S
2045	CF3	SO2CH3	CH3	S
2046	CF3	SO2CF3	CH3	S
2047	CF3	CH2CO2H	CH3	S
2048	CF3	CH2COOCH3	CH3	S
2049	CF3	CH2COOC2H5	CH3	S
2050	CF3	prop-1-en-3-yl	CH3	S
2051	CF3	trans-but-2-en-1-yl	CH3	S
2052	CF3	cis-but-2-en-1-yl	CH3	S
2053	CF3	cis-3-methyl-	CH3	S
		but-2-en-1-yl
2054	CF3	cyclopropyl	CH3	S
2055	CF3	cyclopentyl	CH3	S
2056	CF3	cyclohexyl	CH3	S
2057	CF3	4,5-dihydroisoxazol-	CH3	S
		3-yl
2058	CF3	4-methyl-4,5-dihydroisoxazol-	CH3	S
		3-yl
2059	CF3	isoxazol-3-yl	CH3	S
2060	CF3	4-methylisoxazol-3-yl	CH3	S
2061	CF3	4,5-dihydroisoxazol-	CH3	S
		4-yl
2062	CF3	3-methyl-4,5-dihydroisoxazol-	CH3	S
		4-yl
2063	CF3	isoxazol-4-yl	CH3	S
2064	CF3	3-methylisoxazol-4-yl	CH3	S
2065	CF3	phenyl	CH3	S
2066	CF3	benzyl	CH3	S
2067	CF3	benzoyl	CH3	S
2068	CF3	2-pyridyl	CH3	S
2069	CF3	H	Cl	S
2070	CF3	CH3	Cl	S
2071	CF3	C2H5	Cl	S
2072	CF3	n-C3H7	Cl	S
2073	CF3	i-C3H7	Cl	S
2074	CF3	n-C4H9	Cl	S
2075	CF3	i-C4H9	Cl	S
2076	CF3	s-C4H9	Cl	S
2077	CF3	t-C4H9	Cl	S
2078	CF3	CH2OCH3	Cl	S
2079	CF3	CF3	Cl	S
2080	CF3	CF2H	Cl	S
2081	CF3	CN	Cl	S
2082	CF3	OH	Cl	S
2083	CF3	OCH3	Cl	S
2084	CF3	NH2	Cl	S
2085	CF3	NHCH3	Cl	S
2086	CF3	N(CH3)2	Cl	S
2087	CF3	CO2CH3	Cl	S
2088	CF3	CO2C2H5	Cl	S
2089	CF3	C(O)CH3	Cl	S
2090	CF3	C(O)CF3	Cl	S
2091	CF3	C(═NOCH3)CH3	Cl	S
2092	CF3	SO2CH3	Cl	S
2093	CF3	SO2CF3	Cl	S
2094	CF3	CH2CO2H	Cl	S
2095	CF3	CH2COOCH3	Cl	S
2096	CF3	CH2COOC2H5	Cl	S
2097	CF3	prop-1-en-3-yl	Cl	S
2098	CF3	trans-but-2-en-1-yl	Cl	S
2099	CF3	cis-but-2-en-1-yl	Cl	S
2100	CF3	cis-3-methyl-	Cl	S
		but-2-en-1-yl
2101	CF3	cyclopropyl	Cl	S
2102	CF3	cyclopentyl	Cl	S
2103	CF3	cyclohexyl	Cl	S
2104	CF3	4,5-dihydroisoxazol-	Cl	S
		3-yl
2105	CF3	4-methyl-4,5-dihydroisoxazol-	Cl	S
		3-yl
2106	CF3	isoxazol-3-yl	Cl	S
2107	CF3	4-methylisoxazol-3-yl	Cl	S
2108	CF3	4,5-dihydroisoxazol-	Cl	S
		4-yl
2109	CF3	3-methyl-4,5-dihydroisoxazol-	Cl	S
		4-yl
2110	CF3	isoxazol-4-yl	Cl	S
2111	CF3	3-methylisoxazol-4-yl	Cl	S
2112	CF3	phenyl	Cl	S
2113	CF3	benzyl	Cl	S
2114	CF3	benzoyl	Cl	S
2115	CF3	2-pyridyl	Cl	S
2116	C2H5	H	H	S
2117	C2H5	CH3	H	S
2118	C2H5	C2H5	H	S
2119	C2H5	n-C3H7	H	S
2120	C2H5	i-C3H7	H	S
2121	C2H5	n-C4H9	H	S
2122	C2H5	i-C4H9	H	S
2123	C2H5	s-C4H9	H	S
2124	C2H5	t-C4H9	H	S
2125	C2H5	CH2OCH3	H	S
2126	C2H5	CF3	H	S
2127	C2H5	CF2H	H	S
2128	C2H5	CN	H	S
2129	C2H5	OH	H	S
2130	C2H5	OCH3	H	S
2131	C2H5	NH2	H	S
2132	C2H5	NHCH3	H	S
2133	C2H5	N(CH3)2	H	S
2134	C2H5	CO2CH3	H	S
2135	C2H5	CO2C2H5	H	S
2136	C2H5	C(O)CH3	H	S
2137	C2H5	C(O)CF3	H	S
2138	C2H5	C(═NOCH3)CH3	H	S
2139	C2H5	SO2CH3	H	S
2140	C2H5	SO2CF3	H	S
2141	C2H5	CH2CO2H	H	S
2142	C2H5	CH2COOCH3	H	S
2143	C2H5	CH2COOC2H5	H	S
2144	C2H5	prop-1-en-3-yl	H	S
2145	C2H5	trans-but-2-en-1-yl	H	S
2146	C2H5	cis-but-2-en-1-yl	H	S
2147	C2H5	cis-3-methyl-	H	S
		but-2-en-1-yl
2148	C2H5	cyclopropyl	H	S
2149	C2H5	cyclopentyl	H	S
2150	C2H5	cyclohexyl	H	S
2151	C2H5	4,5-dihydroisoxazol-	H	S
		3-yl
2152	C2H5	4-methyl-4,5-dihydroisoxazol-	H	S
		3-yl
2153	C2H5	isoxazol-3-yl	H	S
2154	C2H5	4-methylisoxazol-3-yl	H	S
2155	C2H5	4,5-dihydroisoxazol-	H	S
		4-yl
2156	C2H5	3-methyl-4,5-dihydroisoxazol-	H	S
		4-yl
2157	C2H5	isoxazol-4-yl	H	S
2158	C2H5	3-methylisoxazol-4-yl	H	S
2159	C2H5	phenyl	H	S
2160	C2H5	benzyl	H	S
2161	C2H5	benzoyl	H	S
2162	C2H5	2-pyridyl	H	S
2163	C2H5	H	CH3	S
2164	C2H5	CH3	CH3	S
2165	C2H5	C2H5	CH3	S
2166	C2H5	n-C3H7	CH3	S
2167	C2H5	i-C3H7	CH3	S
2168	C2H5	n-C4H9	CH3	S
2169	C2H5	i-C4H9	CH3	S
2170	C2H5	s-C4H9	CH3	S
2171	C2H5	t-C4H9	CH3	S
2172	C2H5	CH2OCH3	CH3	S
2173	C2H5	CF3	CH3	S
2174	C2H5	CF2H	CH3	S
2175	C2H5	CN	CH3	S
2176	C2H5	OH	CH3	S
2177	C2H5	OCH3	CH3	S
2178	C2H5	NH2	CH3	S
2179	C2H5	NHCH3	CH3	S
2180	C2H5	N(CH3)2	CH3	S
2181	C2H5	CO2CH3	CH3	S
2182	C2H5	CO2C2H5	CH3	S
2183	C2H5	C(O)CH3	CH3	S
2184	C2H5	C(O)CF3	CH3	S
2185	C2H5	C(═NOCH3)CH3	CH3	S
2186	C2H5	SO2CH3	CH3	S
2187	C2H5	SO2CF3	CH3	S
2188	C2H5	CH2CO2H	CH3	S
2189	C2H5	CH2COOCH3	CH3	S
2190	C2H5	CH2COOC2H5	CH3	S
2191	C2H5	prop-1-en-3-yl	CH3	S
2192	C2H5	trans-but-2-en-1-yl	CH3	S
2193	C2H5	cis-but-2-en-1-yl	CH3	S
2194	C2H5	cis-3-methyl-	CH3	S
		but-2-en-1-yl
2195	C2H5	cyclopropyl	CH3	S
2196	C2H5	cyclopentyl	CH3	S
2197	C2H5	cyclohexyl	CH3	S
2198	C2H5	4,5-dihydroisoxazol-	CH3	S
		3-yl
2199	C2H5	4-methyl-4,5-dihydroisoxazol-	CH3	S
		3-yl
2200	C2H5	isoxazol-3-yl	CH3	S
2201	C2H5	4-methylisoxazol-3-yl	CH3	S
2202	C2H5	4,5-dihydroisoxazol-	CH3	S
		4-yl
2203	C2H5	3-methyl-4,5-dihydroisoxazol-	CH3	S
		4-yl
2204	C2H5	isoxazol-4-yl	CH3	S
2205	C2H5	3-methylisoxazol-4-yl	CH3	S
2206	C2H5	phenyl	CH3	S
2207	C2H5	benzyl	CH3	S
2208	C2H5	benzoyl	CH3	S
2209	C2H5	2-pyridyl	CH3	S
2210	C2H5	H	Cl	S
2211	C2H5	CH3	Cl	S
2212	C2H5	C2H5	Cl	S
2213	C2H5	n-C3H7	Cl	S
2214	C2H5	i-C3H7	Cl	S
2215	C2H5	n-C4H9	Cl	S
2216	C2H5	i-C4H9	Cl	S
2217	C2H5	s-C4H9	Cl	S
2218	C2H5	t-C4H9	Cl	S
2219	C2H5	CH2OCH3	Cl	S
2220	C2H5	CF3	Cl	S
2221	C2H5	CF2H	Cl	S
2222	C2H5	CN	Cl	S
2223	C2H5	OH	Cl	S
2224	C2H5	OCH3	Cl	S
2225	C2H5	NH2	Cl	S
2226	C2H5	NHCH3	Cl	S
2227	C2H5	N(CH3)2	Cl	S
2228	C2H5	CO2CH3	Cl	S
2229	C2H5	CO2C2H5	Cl	S
2230	C2H5	C(O)CH3	Cl	S
2231	C2H5	C(O)CF3	Cl	S
2232	C2H5	C(═NOCH3)CH3	Cl	S
2233	C2H5	SO2CH3	Cl	S
2234	C2H5	SO2CF3	Cl	S
2235	C2H5	CH2CO2H	Cl	S
2236	C2H5	CH2COOCH3	Cl	S
2237	C2H5	CH2COOC2H5	Cl	S
2238	C2H5	prop-1-en-3-yl	Cl	S
2239	C2H5	trans-but-2-en-1-yl	Cl	S
2240	C2H5	cis-but-2-en-1-yl	Cl	S
2241	C2H5	cis-3-methyl-	Cl	S
		but-2-en-1-yl
2242	C2H5	cyclopropyl	Cl	S
2243	C2H5	cyclopentyl	Cl	S
2244	C2H5	cyclohexyl	Cl	S
2245	C2H5	4,5-dihydroisoxazol-	Cl	S
		3-yl
2246	C2H5	4-methyl-4,5-dihydroisoxazol-	Cl	S
		3-yl
2247	C2H5	isoxazol-3-yl	Cl	S
2248	C2H5	4-methylisoxazol-3-yl	Cl	S
2249	C2H5	4,5-dihydroisoxazol-	Cl	S
		4-yl
2250	C2H5	3-methyl-4,5-dihydroisoxazol-	Cl	S
		4-yl
2251	C2H5	isoxazol-4-yl	Cl	S
2252	C2H5	3-methylisoxazol-4-yl	Cl	S
2253	C2H5	phenyl	Cl	S
2254	C2H5	benzyl	Cl	S
2255	C2H5	benzoyl	Cl	S
2256	C2H5	2-pyridyl	Cl	S
2257	CH3	H	H	NCH3
2258	CH3	CH3	H	NCH3
2259	CH3	C2H5	H	NCH3
2260	CH3	n-C3H7	H	NCH3
2261	CH3	i-C3H7	H	NCH3
2262	CH3	n-C4H9	H	NCH3
2263	CH3	i-C4H9	H	NCH3
2264	CH3	s-C4H9	H	NCH3
2265	CH3	t-C4H9	H	NCH3
2266	CH3	CH2OCH3	H	NCH3
2267	CH3	CF3	H	NCH3
2268	CH3	CF2H	H	NCH3
2269	CH3	CN	H	NCH3
2270	CH3	OH	H	NCH3
2271	CH3	OCH3	H	NCH3
2272	CH3	NH2	H	NCH3
2273	CH3	NHCH3	H	NCH3
2274	CH3	N(CH3)2	H	NCH3
2275	CH3	CO2CH3	H	NCH3
2276	CH3	CO2C2H5	H	NCH3
2277	CH3	C(O)CH3	H	NCH3
2278	CH3	C(O)CF3	H	NCH3
2279	CH3	C(═NOCH3)CH3	H	NCH3
2280	CH3	SO2CH3	H	NCH3
2281	CH3	SO2CF3	H	NCH3
2282	CH3	CH2CO2H	H	NCH3
2283	CH3	CH2COOCH3	H	NCH3
2284	CH3	CH2COOC2H5	H	NCH3
2285	CH3	prop-1-en-3-yl	H	NCH3
2286	CH3	trans-but-2-en-1-yl	H	NCH3
2287	CH3	cis-but-2-en-1-yl	H	NCH3
2288	CH3	cis-3-methyl-	H	NCH3
		but-2-en-1-yl
2289	CH3	cyclopropyl	H	NCH3
2290	CH3	cyclopentyl	H	NCH3
2291	CH3	cyclohexyl	H	NCH3
2292	CH3	4,5-dihydroisoxazol-	H	NCH3
		3-yl
2293	CH3	4-methyl-4,5-dihydroisoxazol-	H	NCH3
		3-yl
2294	CH3	isoxazol-3-yl	H	NCH3
2295	CH3	4-methylisoxazol-3-yl	H	NCH3
2296	CH3	4,5-dihydroisoxazol-	H	NCH3
		4-y1
2297	CH3	3-methyl-4,5-dihydroisoxazol-	H	NCH3
		4-yl
2298	CH3	isoxazol-4-yl	H	NCH3
2299	CH3	3-methylisoxazol-4-yl	H	NCH3
2300	CH3	phenyl	H	NCH3
2301	CH3	benzyl	H	NCH3
2302	CH3	benzoyl	H	NCH3
2303	CH3	2-pyridyl	H	NCH3
2304	CH3	H	CH3	NCH3
2305	CH3	CH3	CH3	NCH3
2306	CH3	C2H5	CH3	NCH3
2307	CH3	n-C3H7	CH3	NCH3
2308	CH3	i-C3H7	CH3	NCH3
2309	CH3	n-C4H9	CH3	NCH3
2310	CH3	i-C4H9	CH3	NCH3
2311	CH3	s-C4H9	CH3	NCH3
2312	CH3	t-C4H9	CH3	NCH3
2313	CH3	CH2OCH3	CH3	NCH3
2314	CH3	CF3	CH3	NCH3
2315	CH3	CF2H	CH3	NCH3
2316	CH3	CN	CH3	NCH3
2317	CH3	OH	CH3	NCH3
2318	CH3	OCH3	CH3	NCH3
2319	CH3	NH2	CH3	NCH3
2320	CH3	NHCH3	CH3	NCH3
2321	CH3	N(CH3)2	CH3	NCH3
2322	CH3	CO2CH3	CH3	NCH3
2323	CH3	CO2C2H5	CH3	NCH3
2324	CH3	C(O)CH3	CH3	NCH3
2325	CH3	C(O)CF3	CH3	NCH3
2326	CH3	C(═NOCH3)CH3	CH3	NCH3
2327	CH3	SO2CH3	CH3	NCH3
2328	CH3	SO2CF3	CH3	NCH3
2329	CH3	CH2CO2H	CH3	NCH3
2330	CH3	CH2COOCH3	CH3	NCH3
2331	CH3	CH2COOC2H5	CH3	NCH3
2332	CH3	prop-1-en-3-yl	CH3	NCH3
2333	CH3	trans-but-2-en-1-yl	CH3	NCH3
2334	CH3	cis-but-2-en-1-yl	CH3	NCH3
2335	CH3	cis-3-methyl-	CH3	NCH3
		but-2-en-1-yl
2336	CH3	cyclopropyl	CH3	NCH3
2337	CH3	cyclopentyl	CH3	NCH3
2338	CH3	cyclohexyl	CH3	NCH3
2339	CH3	4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
2340	CH3	4-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
2341	CH3	isoxazol-3-yl	CH3	NCH3
2342	CH3	4-methylisoxazol-3-yl	CH3	NCH3
2343	CH3	4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
2344	CH3	3-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
2345	CH3	isoxazol-4-yl	CH3	NCH3
2346	CH3	3-methylisoxazol-4-yl	CH3	NCH3
2347	CH3	phenyl	CH3	NCH3
2348	CH3	benzyl	CH3	NCH3
2349	CH3	benzoyl	CH3	NCH3
2350	CH3	2-pyridyl	CH3	NCH3
2351	CH3	H	Cl	NCH3
2352	CH3	CH3	Cl	NCH3
2353	CH3	C2H5	Cl	NCH3
2354	CH3	n-C3H7	Cl	NCH3
2355	CH3	i-C3H7	Cl	NCH3
2356	CH3	n-C4H9	Cl	NCH3
2357	CH3	i-C4H9	Cl	NCH3
2358	CH3	s-C4H9	Cl	NCH3
2359	CH3	t-C4H9	Cl	NCH3
2360	CH3	CH2OCH3	Cl	NCH3
2361	CH3	CF3	Cl	NCH3
2362	CH3	CF2H	Cl	NCH3
2363	CH3	CN	Cl	NCH3
2364	CH3	OH	Cl	NCH3
2365	CH3	OCH3	Cl	NCH3
2366	CH3	NH2	Cl	NCH3
2367	CH3	NHCH3	Cl	NCH3
2368	CH3	N(CH3)2	Cl	NCH3
2369	CH3	CO2CH3	Cl	NCH3
2370	CH3	CO2C2H5	Cl	NCH3
2371	CH3	C(O)CH3	Cl	NCH3
2372	CH3	C(O)CF3	Cl	NCH3
2373	CH3	C(═NOCH3)CH3	Cl	NCH3
2374	CH3	SO2CH3	Cl	NCH3
2375	CH3	SO2CF3	Cl	NCH3
2376	CH3	CH2CO2H	Cl	NCH3
2377	CH3	CH2COOCH3	Cl	NCH3
2378	CH3	CH2COOC2H5	Cl	NCH3
2379	CH3	prop-1-en-3-yl	Cl	NCH3
2380	CH3	trans-but-2-en-1-yl	Cl	NCH3
2381	CH3	cis-but-2-en-1-yl	Cl	NCH3
2382	CH3	cis-3-methyl-	Cl	NCH3
		but-2-en-1-yl
2383	CH3	cyclopropyl	Cl	NCH3
2384	CH3	cyclopentyl	Cl	NCH3
2385	CH3	cyclohexyl	Cl	NCH3
2386	CH3	4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
2387	CH3	4-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
2388	CH3	isoxazol-3-yl	Cl	NCH3
2389	CH3	4-methylisoxazol-3-yl	Cl	NCH3
2390	CH3	4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
2391	CH3	3-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
2392	CH3	isoxazol-4-yl	Cl	NCH3
2393	CH3	3-methylisoxazol-4-yl	Cl	NCH3
2394	CH3	phenyl	Cl	NCH3
2395	CH3	benzyl	Cl	NCH3
2396	CH3	benzoyl	Cl	NCH3
2397	CH3	2-pyridyl	Cl	NCH3
2398	Cl	H	H	NCH3
2399	Cl	CH3	H	NCH3
2400	Cl	C2H5	H	NCH3
2401	Cl	n-C3H7	H	NCH3
2402	Cl	i-C3H7	H	NCH3
2403	Cl	n-C4H9	H	NCH3
2404	Cl	i-C4H9	H	NCH3
2405	Cl	s-C4H9	H	NCH3
2406	Cl	t-C4H9	H	NCH3
2407	Cl	CH2OCH3	H	NCH3
2408	Cl	CF3	H	NCH3
2409	Cl	CF2H	H	NCH3
2410	Cl	CN	H	NCH3
2411	Cl	OH	H	NCH3
2412	Cl	OCH3	H	NCH3
2413	Cl	NH2	H	NCH3
2414	Cl	NHCH3	H	NCH3
2415	Cl	N(CH3)2	H	NCH3
2416	Cl	CO2CH3	H	NCH3
2417	Cl	CO2C2H5	H	NCH3
2418	Cl	C(O)CH3	H	NCH3
2419	Cl	C(O)CF3	H	NCH3
2420	Cl	C(═NOCH3)CH3	H	NCH3
2421	Cl	SO2CH3	H	NCH3
2422	Cl	SO2CF3	H	NCH3
2423	Cl	CH2CO2H	H	NCH3
2424	Cl	CH2COOCH3	H	NCH3
2425	Cl	CH2COOC2H5	H	NCH3
2426	Cl	prop-1-en-3-yl	H	NCH3
2427	Cl	trans-but-2-en-1-yl	H	NCH3
2428	Cl	cis-but-2-en-1-yl	H	NCH3
2429	Cl	cis-3-methyl-	H	NCH3
		but-2-en-1-yl
2430	Cl	cyclopropyl	H	NCH3
2431	Cl	cyclopentyl	H	NCH3
2432	Cl	cyclohexyl	H	NCH3
2433	Cl	4,5-dihydroisoxazol-	H	NCH3
		3-yl
2434	Cl	4-methyl-4,5-dihydroisoxazol-	H	NCH3
		3-yl
2435	Cl	isoxazol-3-yl	H	NCH3
2436	Cl	4-methylisoxazol-3-yl	H	NCH3
2437	Cl	4,5-dihydroisoxazol-	H	NCH3
		4-yl
2438	Cl	3-methyl-4,5-dihydroisoxazol-	H	NCH3
		4-yl
2439	Cl	isoxazol-4-yl	H	NCH3
2440	Cl	3-methylisoxazol-4-yl	H	NCH3
2441	Cl	phenyl	H	NCH3
2442	Cl	benzyl	H	NCH3
2443	Cl	benzoyl	H	NCH3
2444	Cl	2-pyridyl	H	NCH3
2445	Cl	H	CH3	NCH3
2446	Cl	CH3	CH3	NCH3
2447	Cl	C2H5	CH3	NCH3
2448	Cl	n-C3H7	CH3	NCH3
2449	Cl	i-C3H7	CH3	NCH3
2450	Cl	n-C4H9	CH3	NCH3
2451	Cl	i-C4H9	CH3	NCH3
2452	Cl	s-C4H9	CH3	NCH3
2453	Cl	t-C4H9	CH3	NCH3
2454	Cl	CH2OCH3	CH3	NCH3
2455	Cl	CF3	CH3	NCH3
2456	Cl	CF2H	CH3	NCH3
2457	Cl	CN	CH3	NCH3
2458	Cl	OH	CH3	NCH3
2459	Cl	OCH3	CH3	NCH3
2460	Cl	NH2	CH3	NCH3
2461	Cl	NHCH3	CH3	NCH3
2462	Cl	N(CH3)2	CH3	NCH3
2463	Cl	CO2CH3	CH3	NCH3
2464	Cl	CO2C2H5	CH3	NCH3
2465	Cl	C(O)CH3	CH3	NCH3
2466	Cl	C(O)CF3	CH3	NCH3
2467	Cl	C(═NOCH3)CH3	CH3	NCH3
2468	Cl	SO2CH3	CH3	NCH3
2469	Cl	SO2CF3	CH3	NCH3
2470	Cl	CH2CO2H	CH3	NCH3
2471	Cl	CH2COOCH3	CH3	NCH3
2472	Cl	CH2COOC2H5	CH3	NCH3
2473	Cl	prop-1-en-3-yl	CH3	NCH3
2474	Cl	trans-but-2-en-1-yl	CH3	NCH3
2475	Cl	cis-but-2-en-1-yl	CH3	NCH3
2476	Cl	cis-3-methyl-	CH3	NCH3
		but-2-en-1-yl
2477	Cl	cyclopropyl	CH3	NCH3
2478	Cl	cyclopentyl	CH3	NCH3
2479	Cl	cyclohexyl	CH3	NCH3
2480	Cl	4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
2481	Cl	4-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
2482	Cl	isoxazol-3-yl	CH3	NCH3
2483	Cl	4-methylisoxazol-3-yl	CH3	NCH3
2484	Cl	4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
2485	Cl	3-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
2486	Cl	isoxazol-4-yl	CH3	NCH3
2487	Cl	3-methylisoxazol-4-yl	CH3	NCH3
2488	Cl	phenyl	CH3	NCH3
2489	Cl	benzyl	CH3	NCH3
2490	Cl	benzoyl	CH3	NCH3
2491	Cl	2-pyridyl	CH3	NCH3
2492	Cl	H	Cl	NCH3
2493	Cl	CH3	Cl	NCH3
2494	Cl	C2H5	Cl	NCH3
2495	Cl	n-C3H7	Cl	NCH3
2496	Cl	i-C3H7	Cl	NCH3
2497	Cl	n-C4H9	Cl	NCH3
2498	Cl	i-C4H9	Cl	NCH3
2499	Cl	s-C4H9	Cl	NCH3
2500	Cl	t-C4H9	Cl	NCH3
2501	Cl	CH2OCH3	Cl	NCH3
2502	Cl	CF3	Cl	NCH3
2503	Cl	CF2H	Cl	NCH3
2504	Cl	CN	Cl	NCH3
2505	Cl	OH	Cl	NCH3
2506	Cl	OCH3	Cl	NCH3
2507	Cl	NH2	Cl	NCH3
2508	Cl	NHCH3	Cl	NCH3
2509	Cl	N(CH3)2	Cl	NCH3
2510	Cl	CO2CH3	Cl	NCH3
2511	Cl	CO2C2H5	Cl	NCH3
2512	Cl	C(O)CH3	Cl	NCH3
2513	Cl	C(O)CF3	Cl	NCH3
2514	Cl	C(═NOCH3)CH3	Cl	NCH3
2515	Cl	SO2CH3	Cl	NCH3
2516	Cl	SO2CF3	Cl	NCH3
2517	Cl	CH2CO2H	Cl	NCH3
2518	Cl	CH2COOCH3	Cl	NCH3
2519	Cl	CH2COOC2H5	Cl	NCH3
2520	Cl	prop-1-en-3-yl	Cl	NCH3
2521	Cl	trans-but-2-en-1-yl	Cl	NCH3
2522	Cl	cis-but-2-en-1-yl	Cl	NCH3
2523	Cl	cis-3-methyl-	Cl	NCH3
		but-2-en-1-yl
2524	Cl	cyclopropyl	Cl	NCH3
2525	Cl	cyclopentyl	Cl	NCH3
2526	Cl	cyclohexyl	Cl	NCH3
2527	Cl	4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
2528	Cl	4-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
2529	Cl	isoxazol-3-yl	Cl	NCH3
2530	Cl	4-methylisoxazol-3-yl	Cl	NCH3
2531	Cl	4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
2532	Cl	3-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
2533	Cl	isoxazol-4-yl	Cl	NCH3
2534	Cl	3-methylisoxazol-4-yl	Cl	NCH3
2535	Cl	phenyl	Cl	NCH3
2536	Cl	benzyl	Cl	NCH3
2537	Cl	benzoyl	Cl	NCH3
2538	Cl	2-pyridyl	Cl	NCH3
2539	OCH3	H	H	NCH3
2540	OCH3	CH3	H	NCH3
2541	OCH3	C2H5	H	NCH3
2542	OCH3	n-C3H7	H	NCH3
2543	OCH3	i-C3H7	H	NCH3
2544	OCH3	n-C4H9	H	NCH3
2545	OCH3	i-C4H9	H	NCH3
2546	OCH3	s-C4H9	H	NCH3
2547	OCH3	t-C4H9	H	NCH3
2548	OCH3	CH2OCH3	H	NCH3
2549	OCH3	CF3	H	NCH3
2550	OCH3	CF2H	H	NCH3
2551	OCH3	CN	H	NCH3
2552	OCH3	OH	H	NCH3
2553	OCH3	OCH3	H	NCH3
2554	OCH3	NH2	H	NCH3
2555	OCH3	NHCH3	H	NCH3
2556	OCH3	N(CH3)2	H	NCH3
2557	OCH3	CO2CH3	H	NCH3
2558	OCH3	CO2C2H5	H	NCH3
2559	OCH3	C(O)CH3	H	NCH3
2560	OCH3	C(O)CF3	H	NCH3
2561	OCH3	C(═NOCH3)CH3	H	NCH3
2562	OCH3	SO2CH3	H	NCH3
2563	OCH3	SO2CF3	H	NCH3
2564	OCH3	CH2CO2H	H	NCH3
2565	OCH3	CH2COOCH3	H	NCH3
2566	OCH3	CH2COOC2H5	H	NCH3
2567	OCH3	prop-1-en-3-yl	H	NCH3
2568	OCH3	trans-but-2-en-1-yl	H	NCH3
2569	OCH3	cis-but-2-en-1-yl	H	NCH3
2570	OCH3	cis-3-methyl-	H	NCH3
		but-2-en-1-yl
2571	OCH3	cyclopropyl	H	NCH3
2572	OCH3	cyclopentyl	H	NCH3
2573	OCH3	cyclohexyl	H	NCH3
2574	OCH3	4,5-dihydroisoxazol-	H	NCH3
		3-yl
2575	OCH3	4-methyl-4,5-dihydroisoxazol-	H	NCH3
		3-yl
2576	OCH3	isoxazol-3-yl	H	NCH3
2577	OCH3	4-methylisoxazol-3-yl	H	NCH3
2578	OCH3	4,5-dihydroisoxazol-	H	NCH3
		4-yl
2579	OCH3	3-methyl-4,5-dihydroisoxazol-	H	NCH3
		4-yl
2580	OCH3	isoxazol-4-yl	H	NCH3
2581	OCH3	3-methylisoxazol-4-yl	H	NCH3
2582	OCH3	phenyl	H	NCH3
2583	OCH3	benzyl	H	NCH3
2584	OCH3	benzoyl	H	NCH3
2585	OCH3	2-pyridyl	H	NCH3
2586	OCH3	H	CH3	NCH3
2587	OCH3	CH3	CH3	NCH3
2588	OCH3	C2H5	CH3	NCH3
2589	OCH3	n-C3H7	CH3	NCH3
2590	OCH3	i-C3H7	CH3	NCH3
2591	OCH3	n-C4H9	CH3	NCH3
2592	OCH3	i-C4H9	CH3	NCH3
2593	OCH3	s-C4H9	CH3	NCH3
2594	OCH3	t-C4H9	CH3	NCH3
2595	OCH3	CH2OCH3	CH3	NCH3
2596	OCH3	CF3	CH3	NCH3
2597	OCH3	CF2H	CH3	NCH3
2598	OCH3	CN	CH3	NCH3
2599	OCH3	OH	CH3	NCH3
2600	OCH3	OCH3	CH3	NCH3
2601	OCH3	NH2	CH3	NCH3
2602	OCH3	NHCH3	CH3	NCH3
2603	OCH3	N(CH3)2	CH3	NCH3
2604	OCH3	CO2CH3	CH3	NCH3
2605	OCH3	CO2C2H5	CH3	NCH3
2606	OCH3	C(O)CH3	CH3	NCH3
2607	OCH3	C(O)CF3	CH3	NCH3
2608	OCH3	C(═NOCH3)CH3	CH3	NCH3
2609	OCH3	SO2CH3	CH3	NCH3
2610	OCH3	SO2CF3	CH3	NCH3
2611	OCH3	CH2CO2H	CH3	NCH3
2612	OCH3	CH2COOCH3	CH3	NCH3
2613	OCH3	CH2COOC2H5	CH3	NCH3
2614	OCH3	prop-1-en-3-yl	CH3	NCH3
2615	OCH3	trans-but-2-en-1-yl	CH3	NCH3
2616	OCH3	cis-but-2-en-1-yl	CH3	NCH3
2617	OCH3	cis-3-methyl-	CH3	NCH3
		but-2-en-1-yl
2618	OCH3	cyclopropyl	CH3	NCH3
2619	OCH3	cyclopentyl	CH3	NCH3
2620	OCH3	cyclohexyl	CH3	NCH3
2621	OCH3	4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
2622	OCH3	4-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
2623	OCH3	isoxazol-3-yl	CH3	NCH3
2624	OCH3	4-methylisoxazol-3-yl	CH3	NCH3
2625	OCH3	4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
2626	OCH3	3-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
2627	OCH3	isoxazol-4-yl	CH3	NCH3
2628	OCH3	3-methylisoxazol-4-yl	CH3	NCH3
2629	OCH3	phenyl	CH3	NCH3
2630	OCH3	benzyl	CH3	NCH3
2631	OCH3	benzoyl	CH3	NCH3
2632	OCH3	2-pyridyl	CH3	NCH3
2633	OCH3	H	Cl	NCH3
2634	OCH3	CH3	Cl	NCH3
2635	OCH3	C2H5	Cl	NCH3
2636	OCH3	n-C3H7	Cl	NCH3
2637	OCH3	i-C3H7	Cl	NCH3
2638	OCH3	n-C4H9	Cl	NCH3
2639	OCH3	i-C4H9	Cl	NCH3
2640	OCH3	s-C4H9	Cl	NCH3
2641	OCH3	t-C4H9	Cl	NCH3
2642	OCH3	CH2OCH3	Cl	NCH3
2643	OCH3	CF3	Cl	NCH3
2644	OCH3	CF2H	Cl	NCH3
2645	OCH3	CN	Cl	NCH3
2646	OCH3	OH	Cl	NCH3
2647	OCH3	OCH3	Cl	NCH3
2648	OCH3	NH2	Cl	NCH3
2649	OCH3	NHCH3	Cl	NCH3
2650	OCH3	N(CH3)2	Cl	NCH3
2651	OCH3	CO2CH3	Cl	NCH3
2652	OCH3	CO2C2H5	Cl	NCH3
2653	OCH3	C(O)CH3	Cl	NCH3
2654	OCH3	C(O)CF3	Cl	NCH3
2655	OCH3	C(═NOCH3)CH3	Cl	NCH3
2656	OCH3	SO2CH3	Cl	NCH3
2657	OCH3	SO2CF3	Cl	NCH3
2658	OCH3	CH2CO2H	Cl	NCH3
2659	OCH3	CH2COOCH3	Cl	NCH3
2660	OCH3	CH2COOC2H5	Cl	NCH3
2661	OCH3	prop-1-en-3-yl	Cl	NCH3
2662	OCH3	trans-but-2-en-1-yl	Cl	NCH3
2663	OCH3	cis-but-2-en-1-yl	Cl	NCH3
2664	OCH3	cis-3-methyl-	Cl	NCH3
		but-2-en-1-yl
2665	OCH3	cyclopropyl	Cl	NCH3
2666	OCH3	cyclopentyl	Cl	NCH3
2667	OCH3	cyclohexyl	Cl	NCH3
2668	OCH3	4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
2669	OCH3	4-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
2670	OCH3	isoxazol-3-yl	Cl	NCH3
2671	OCH3	4-methylisoxazol-3-yl	Cl	NCH3
2672	OCH3	4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
2673	OCH3	3-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
2674	OCH3	isoxazol-4-yl	Cl	NCH3
2675	OCH3	3-methylisoxazol-4-yl	Cl	NCH3
2676	OCH3	phenyl	Cl	NCH3
2677	OCH3	benzyl	Cl	NCH3
2678	OCH3	benzoyl	Cl	NCH3
2679	OCH3	2-pyridyl	Cl	NCH3
2680	OCF3	H	H	NCH3
2681	OCF3	CH3	H	NCH3
2682	OCF3	C2H5	H	NCH3
2683	OCF3	n-C3H7	H	NCH3
2684	OCF3	i-C3H7	H	NCH3
2685	OCF3	n-C4H9	H	NCH3
2686	OCF3	i-C4H9	H	NCH3
2687	OCF3	s-C4H9	H	NCH3
2688	OCF3	t-C4H9	H	NCH3
2689	OCF3	CH2OCH3	H	NCH3
2690	OCF3	CF3	H	NCH3
2691	OCF3	CF2H	H	NCH3
2692	OCF3	CN	H	NCH3
2693	OCF3	OH	H	NCH3
2694	OCF3	OCH3	H	NCH3
2695	OCF3	NH2	H	NCH3
2696	OCF3	NHCH3	H	NCH3
2697	OCF3	N(CH3)2	H	NCH3
2698	OCF3	CO2CH3	H	NCH3
2699	OCF3	CO2C2H5	H	NCH3
2700	OCF3	C(O)CH3	H	NCH3
2701	OCF3	C(O)CF3	H	NCH3
2702	OCF3	C(═NOCH3)CH3	H	NCH3
2703	OCF3	SO2CH3	H	NCH3
2704	OCF3	SO2CF3	H	NCH3
2705	OCF3	CH2CO2H	H	NCH3
2706	OCF3	CH2COOCH3	H	NCH3
2707	OCF3	CH2COOC2H5	H	NCH3
2708	OCF3	prop-1-en-3-yl	H	NCH3
2709	OCF3	trans-but-2-en-1-yl	H	NCH3
2710	OCF3	cis-but-2-en-1-yl	H	NCH3
2711	OCF3	cis-3-methyl-	H	NCH3
		but-2-en-1-yl
2712	OCF3	cyclopropyl	H	NCH3
2713	OCF3	cyclopentyl	H	NCH3
2714	OCF3	cyclohexyl	H	NCH3
2715	OCF3	4,5-dihydroisoxazol-	H	NCH3
		3-yl
2716	OCF3	4-methyl-4,5-dihydroisoxazol-	H	NCH3
		3-yl
2717	OCF3	isoxazol-3-yl	H	NCH3
2718	OCF3	4-methylisoxazol-3-yl	H	NCH3
2719	OCF3	4,5-dihydroisoxazol-	H	NCH3
		4-yl
2720	OCF3	3-methyl-4,5-dihydroisoxazol-	H	NCH3
		4-yl
2721	OCF3	isoxazol-4-yl	H	NCH3
2722	OCF3	3-methylisoxazol-4-yl	H	NCH3
2723	OCF3	phenyl	H	NCH3
2724	OCF3	benzyl	H	NCH3
2725	OCF3	benzoyl	H	NCH3
2726	OCF3	2-pyridyl	H	NCH3
2727	OCF3	H	CH3	NCH3
2728	OCF3	CH3	CH3	NCH3
2729	OCF3	C2H5	CH3	NCH3
2730	OCF3	n-C3H7	CH3	NCH3
2731	OCF3	i-C3H7	CH3	NCH3
2732	OCF3	n-C4H9	CH3	NCH3
2733	OCF3	i-C4H9	CH3	NCH3
2734	OCF3	s-C4H9	CH3	NCH3
2735	OCF3	t-C4H9	CH3	NCH3
2736	OCF3	CH2OCH3	CH3	NCH3
2737	OCF3	CF3	CH3	NCH3
2738	OCF3	CF2H	CH3	NCH3
2739	OCF3	CN	CH3	NCH3
2740	OCF3	OH	CH3	NCH3
2741	OCF3	OCH3	CH3	NCH3
2742	OCF3	NH2	CH3	NCH3
2743	OCF3	NHCH3	CH3	NCH3
2744	OCF3	N(CH3)2	CH3	NCH3
2745	OCF3	CO2CH3	CH3	NCH3
2746	OCF3	CO2C2H5	CH3	NCH3
2747	OCF3	C(O)CH3	CH3	NCH3
2748	OCF3	C(O)CF3	CH3	NCH3
2749	OCF3	C(═NOCH3)CH3	CH3	NCH3
2750	OCF3	SO2CH3	CH3	NCH3
2751	OCF3	SO2CF3	CH3	NCH3
2752	OCF3	CH2CO2H	CH3	NCH3
2753	OCF3	CH2COOCH3	CH3	NCH3
2754	OCF3	CH2COOC2H5	CH3	NCH3
2755	OCF3	prop-1-en-3-yl	CH3	NCH3
2756	OCF3	trans-but-2-en-1-yl	CH3	NCH3
2757	OCF3	cis-but-2-en-1-yl	CH3	NCH3
2758	OCF3	cis-3-methyl-	CH3	NCH3
		but-2-en-l-yl
2759	OCF3	cyclopropyl	CH3	NCH3
2760	OCF3	cyclopentyl	CH3	NCH3
2761	OCF3	cyclohexyl	CH3	NCH3
2762	OCF3	4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
2763	OCF3	4-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
2764	OCF3	isoxazol-3-yl	CH3	NCH3
2765	OCF3	4-methylisoxazol-3-yl	CH3	NCH3
2766	OCF3	4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
2767	OCF3	3-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
2768	OCF3	isoxazol-4-yl	CH3	NCH3
2769	OCF3	3-methylisoxazol-4-yl	CH3	NCH3
2770	OCF3	phenyl	CH3	NCH3
2771	OCF3	benzyl	CH3	NCH3
2772	OCF3	benzoyl	CH3	NCH3
2773	OCF3	2-pyridyl	CH3	NCH3
2774	OCF3	H	Cl	NCH3
2775	OCF3	CH3	Cl	NCH3
2776	OCF3	C2H5	Cl	NCH3
2777	OCF3	n-C3H7	Cl	NCH3
2778	OCF3	i-C3H7	Cl	NCH3
2779	OCF3	n-C4H9	Cl	NCH3
2780	OCF3	i-C4H9	Cl	NCH3
2781	OCF3	s-C4H9	Cl	NCH3
2782	OCF3	t-C4H9	Cl	NCH3
2783	OCF3	CH2OCH3	Cl	NCH3
2784	OCF3	CF3	Cl	NCH3
2785	OCF3	CF2H	Cl	NCH3
2786	OCF3	CN	Cl	NCH3
2787	OCF3	OH	Cl	NCH3
2788	OCF3	OCH3	Cl	NCH3
2789	OCF3	NH2	Cl	NCH3
2790	OCF3	NHCH3	Cl	NCH3
2791	OCF3	N(CH3)2	Cl	NCH3
2792	OCF3	CO2CH3	Cl	NCH3
2793	OCF3	CO2C2H5	Cl	NCH3
2794	OCF3	C(O)CH3	Cl	NCH3
2795	OCF3	C(O)CF3	Cl	NCH3
2796	OCF3	C(═NOCH3)CH3	Cl	NCH3
2797	OCF3	SO2CH3	Cl	NCH3
2798	OCF3	SO2CF3	Cl	NCH3
2799	OCF3	CH2CO2H	Cl	NCH3
2800	OCF3	CH2COOCH3	Cl	NCH3
2801	OCF3	CH2COOC2H5	Cl	NCH3
2802	OCF3	prop-1-en-3-yl	Cl	NCH3
2803	OCF3	trans-but-2-en-1-yl	Cl	NCH3
2804	OCF3	cis-but-2-en-1-yl	Cl	NCH3
2805	OCF3	cis-3-methyl-	Cl	NCH3
		but-2-en-1-yl
2806	OCF3	cyclopropyl	Cl	NCH3
2807	OCF3	cyclopentyl	Cl	NCH3
2808	OCF3	cyclohexyl	Cl	NCH3
2809	OCF3	4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
2810	OCF3	4-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
2811	OCF3	isoxazol-3-yl	Cl	NCH3
2812	OCF3	4-methylisoxazol-3-yl	Cl	NCH3
2813	OCF3	4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
2814	OCF3	3-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
2815	OCF3	isoxazol-4-yl	Cl	NCH3
2816	OCF3	3-methylisoxazol-4-yl	Cl	NCH3
2817	OCF3	phenyl	Cl	NCH3
2818	OCF3	benzyl	Cl	NCH3
2819	OCF3	benzoyl	Cl	NCH3
2820	OCF3	2-pyridyl	Cl	NCH3
2821	SCH3	H	H	NCH3
2822	SCH3	CH3	H	NCH3
2823	SCH3	C2H5	H	NCH3
2824	SCH3	n-C3H7	H	NCH3
2825	SCH3	i-C3H7	H	NCH3
2826	SCH3	n-C4H9	H	NCH3
2827	SCH3	i-C4H9	H	NCH3
2828	SCH3	s-C4H9	H	NCH3
2829	SCH3	t-C4H9	H	NCH3
2830	SCH3	CH2OCH3	H	NCH3
2831	SCH3	CF3	H	NCH3
2832	SCH3	CF2H	H	NCH3
2833	SCH3	CN	H	NCH3
2834	SCH3	OH	H	NCH3
2835	SCH3	OCH3	H	NCH3
2836	SCH3	NH2	H	NCH3
2837	SCH3	NHCH3	H	NCH3
2838	SCH3	N(CH3)2	H	NCH3
2839	SCH3	CO2CH3	H	NCH3
2840	SCH3	CO2C2H5	H	NCH3
2841	SCH3	C(O)CH3	H	NCH3
2842	SCH3	C(O)CF3	H	NCH3
2843	SCH3	C(═NOCH3)CH3	H	NCH3
2844	SCH3	SO2CH3	H	NCH3
2845	SCH3	SO2CF3	H	NCH3
2846	SCH3	CH2CO2H	H	NCH3
2847	SCH3	CH2COOCH3	H	NCH3
2848	SCH3	CH2COOC2H5	H	NCH3
2849	SCH3	prop-1-en-3-yl	H	NCH3
2850	SCH3	trans-but-2-en-1-yl	H	NCH3
2851	SCH3	cis-but-2-en-1-yl	H	NCH3
2852	SCH3	cis-3-methyl-	H	NCH3
		but-2-en-1-yl
2853	SCH3	cyclopropyl	H	NCH3
2854	SCH3	cyclopentyl	H	NCH3
2855	SCH3	cyclohexyl	H	NCH3
2856	SCH3	4,5-dihydroisoxazol-	H	NCH3
		3-yl
2857	SCH3	4-methyl-4,5-dihydroisoxazol-	H	NCH3
		3-yl
2858	SCH3	isoxazol-3-yl	H	NCH3
2859	SCH3	4-methylisoxazol-3-yl	H	NCH3
2860	SCH3	4,5-dihydroisoxazol-	H	NCH3
		4-yl
2861	SCH3	3-methyl-4,5-dihydroisoxazol-	H	NCH3
		4-yl
2862	SCH3	isoxazol-4-yl	H	NCH3
2863	SCH3	3-methylisoxazol-4-yl	H	NCH3
2864	SCH3	phenyl	H	NCH3
2865	SCH3	benzyl	H	NCH3
2866	SCH3	benzoyl	H	NCH3
2867	SCH3	2-pyridyl	H	NCH3
2868	SCH3	H	CH3	NCH3
2869	SCH3	CH3	CH3	NCH3
2870	SCH3	C2H5	CH3	NCH3
2871	SCH3	n-C3H7	CH3	NCH3
2872	SCH3	i-C3H7	CH3	NCH3
2873	SCH3	n-C4H9	CH3	NCH3
2874	SCH3	i-C4H9	CH3	NCH3
2875	SCH3	s-C4H9	CH3	NCH3
2876	SCH3	t-C4H9	CH3	NCH3
2877	SCH3	CH2OCH3	CH3	NCH3
2878	SCH3	CF3	CH3	NCH3
2879	SCH3	CF2H	CH3	NCH3
2880	SCH3	CN	CH3	NCH3
2881	SCH3	OH	CH3	NCH3
2882	SCH3	OCH3	CH3	NCH3
2883	SCH3	NH2	CH3	NCH3
2884	SCH3	NHCH3	CH3	NCH3
2885	SCH3	N(CH3)2	CH3	NCH3
2886	SCH3	CO2CH3	CH3	NCH3
2887	SCH3	CO2C2H5	CH3	NCH3
2888	SCH3	C(O)CH3	CH3	NCH3
2889	SCH3	C(O)CF3	CH3	NCH3
2890	SCH3	C(═NOCH3)CH3	CH3	NCH3
2891	SCH3	SO2CH3	CH3	NCH3
2892	SCH3	SO2CF3	CH3	NCH3
2893	SCH3	CH2CO2H	CH3	NCH3
2894	SCH3	CH2COOCH3	CH3	NCH3
2895	SCH3	CH2COOC2H5	CH3	NCH3
2896	SCH3	prop-1-en-3-yl	CH3	NCH3
2897	SCH3	trans-but-2-en-1-yl	CH3	NCH3
2898	SCH3	cis-but-2-en-1-yl	CH3	NCH3
2899	SCH3	cis-3-methyl-	CH3	NCH3
		but-2-en-1-yl
2900	SCH3	cyclopropyl	CH3	NCH3
2901	SCH3	cyclopentyl	CH3	NCH3
2902	SCH3	cyclohexyl	CH3	NCH3
2903	SCH3	4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
2904	SCH3	4-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
2905	SCH3	isoxazol-3-yl	CH3	NCH3
2906	SCH3	4-methylisoxazol-3-yl	CH3	NCH3
2907	SCH3	4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
2908	SCH3	3-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
2909	SCH3	isoxazol-4-yl	CH3	NCH3
2910	SCH3	3-methylisoxazol-4-yl	CH3	NCH3
2911	SCH3	phenyl	CH3	NCH3
2912	SCH3	benzyl	CH3	NCH3
2913	SCH3	benzoyl	CH3	NCH3
2914	SCH3	2-pyridyl	CH3	NCH3
2915	SCH3	H	Cl	NCH3
2916	SCH3	CH3	Cl	NCH3
2917	SCH3	C2H5	Cl	NCH3
2918	SCH3	n-C3H7	Cl	NCH3
2919	SCH3	i-C3H7	Cl	NCH3
2920	SCH3	n-C4H9	Cl	NCH3
2921	SCH3	i-C4H9	Cl	NCH3
2922	SCH3	s-C4H9	Cl	NCH3
2923	SCH3	t-C4H9	Cl	NCH3
2924	SCH3	CH2OCH3	Cl	NCH3
2925	SCH3	CF3	Cl	NCH3
2926	SCH3	CF2H	Cl	NCH3
2927	SCH3	CN	Cl	NCH3
2928	SCH3	OH	Cl	NCH3
2929	SCH3	OCH3	Cl	NCH3
2930	SCH3	NH2	Cl	NCH3
2931	SCH3	NHCH3	Cl	NCH3
2932	SCH3	N(CH3)2	Cl	NCH3
2933	SCH3	CO2CH3	Cl	NCH3
2934	SCH3	CO2C2H5	Cl	NCH3
2935	SCH3	C(O)CH3	Cl	NCH3
2936	SCH3	C(O)CF3	Cl	NCH3
2937	SCH3	C(═NOCH3) CH3	Cl	NCH3
2938	SCH3	SO2CH3	Cl	NCH3
2939	SCH3	SO2CF3	Cl	NCH3
2940	SCH3	CH2CO2H	Cl	NCH3
2941	SCH3	CH2COOCH3	Cl	NCH3
2942	SCH3	CH2COOC2H5	Cl	NCH3
2943	SCH3	prop-1-en-3-yl	Cl	NCH3
2944	SCH3	trans-but-2-en-1-yl	Cl	NCH3
2945	SCH3	cis-but-2-en-1-yl	Cl	NCH3
2946	SCH3	cis-3-methyl-	Cl	NCH3
		but-2-en-1-yl
2947	SCH3	cyclopropyl	Cl	NCH3
2948	SCH3	cyclopentyl	Cl	NCH3
2949	SCH3	cyclohexyl	Cl	NCH3
2950	SCH3	4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
2951	SCH3	4-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
2952	SCH3	isoxazol-3-yl	Cl	NCH3
2953	SCH3	4-methylisoxazol-3-yl	Cl	NCH3
2954	SCH3	4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
2955	SCH3	3-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
2956	SCH3	isoxazol-4-yl	Cl	NCH3
2957	SCH3	3-methylisoxazol-4-yl	Cl	NCH3
2958	SCH3	phenyl	Cl	NCH3
2959	SCH3	benzyl	Cl	NCH3
2960	SCH3	benzoyl	Cl	NCH3
2961	SCH3	2-pyridyl	Cl	NCH3
2962	SO2CH3	H	H	NCH3
2963	SO2CH3	CH3	H	NCH3
2964	SO2CH3	C2H5	H	NCH3
2965	SO2CH3	n-C3H7	H	NCH3
2966	SO2CH3	i-C3H7	H	NCH3
2967	SO2CH3	n-C4H9	H	NCH3
2968	SO2CH3	i-C4H9	H	NCH3
2969	SO2CH3	s-C4H9	H	NCH3
2970	SO2CH3	t-C4H9	H	NCH3
2971	SO2CH3	CH2OCH3	H	NCH3
2972	SO2CH3	CF3	H	NCH3
2973	SO2CH3	CF2H	H	NCH3
2974	SO2CH3	CN	H	NCH3
2975	SO2CH3	OH	H	NCH3
2976	SO2CH3	OCH3	H	NCH3
2977	SO2CH3	NH2	H	NCH3
2978	SO2CH3	NHCH3	H	NCH3
2979	SO2CH3	N(CH3)2	H	NCH3
2980	SO2CH3	CO2CH3	H	NCH3
2981	SO2CH3	CO2C2H5	H	NCH3
2982	SO2CH3	C(O)CH3	H	NCH3
2983	SO2CH3	C(O)CF3	H	NCH3
2984	SO2CH3	C(═NOCH3)CH3	H	NCH3
2985	SO2CH3	SO2CH3	H	NCH3
2986	SO2CH3	SO2CF3	H	NCH3
2987	SO2CH3	CH2CO2H	H	NCH3
2988	SO2CH3	CH2COOCH3	H	NCH3
2989	SO2CH3	CH2COOC2H5	H	NCH3
2990	SO2CH3	prop-1-en-3-yl	H	NCH3
2991	SO2CH3	trans-but-2-en-1-yl	H	NCH3
2992	SO2CH3	cis-but-2-en-1-yl	H	NCH3
2993	SO2CH3	cis-3-methyl-	H	NCH3
		but-2-en-1-yl
2994	SO2CH3	cyclopropyl	H	NCH3
2995	SO2CH3	cyclopentyl	H	NCH3
2996	SO2CH3	cyclohexyl	H	NCH3
2997	SO2CH3	4,5-dihydroisoxazol-	H	NCH3
		3-yl
2998	SO2CH3	4-methyl-4,5-dihydroisoxazol-	H	NCH3
		3-yl
2999	SO2CH3	isoxazol-3-yl	H	NCH3
3000	SO2CH3	4-methylisoxazol-3-yl	H	NCH3
3001	SO2CH3	4,5-dihydroisoxazol-	H	NCH3
		4-yl
3002	SO2CH3	3-methyl-4,5-dihydroisoxazol-	H	NCH3
		4-yl
3003	SO2CH3	isoxazol-4-yl	H	NCH3
3004	SO2CH3	3-methylisoxazol-4-yl	H	NCH3
3005	SO2CH3	phenyl	H	NCH3
3006	SO2CH3	benzyl	H	NCH3
3007	SO2CH3	benzoyl	H	NCH3
3008	SO2CH3	2-pyridyl	H	NCH3
3009	SO2CH3	H	CH3	NCH3
3010	SO2CH3	CH3	CH3	NCH3
3011	SO2CH3	C2H5	CH3	NCH3
3012	SO2CH3	n-C3H7	CH3	NCH3
3013	SO2CH3	i-C3H7	CH3	NCH3
3014	SO2CH3	n-C4H9	CH3	NCH3
3015	SO2CH3	i-C4H9	CH3	NCH3
3016	SO2CH3	s-C4H9	CH3	NCH3
3017	SO2CH3	t-C4H9	CH3	NCH3
3018	SO2CH3	CH2OCH3	CH3	NCH3
3019	SO2CH3	CF3	CH3	NCH3
3020	SO2CH3	CF2H	CH3	NCH3
3021	SO2CH3	CN	CH3	NCH3
3022	SO2CH3	OH	CH3	NCH3
3023	SO2CH3	OCH3	CH3	NCH3
3024	SO2CH3	NH2	CH3	NCH3
3025	SO2CH3	NHCH3	CH3	NCH3
3026	SO2CH3	N(CH3)2	CH3	NCH3
3027	SO2CH3	CO2CH3	CH3	NCH3
3028	SO2CH3	CO2C2H5	CH3	NCH3
3029	SO2CH3	C(O)CH3	CH3	NCH3
3030	SO2CH3	C(O)CF3	CH3	NCH3
3031	SO2CH3	C(═NOCH3)CH3	CH3	NCH3
3032	SO2CH3	SO2CH3	CH3	NCH3
3033	SO2CH3	SO2CF3	CH3	NCH3
3034	SO2CH3	CH2CO2H	CH3	NCH3
3035	SO2CH3	CH2COOCH3	CH3	NCH3
3036	SO2CH3	CH2COOC2H5	CH3	NCH3
3037	SO2CH3	prop-1-en-3-yl	CH3	NCH3
3038	SO2CH3	trans-but-2-en-1-yl	CH3	NCH3
3039	SO2CH3	cis-but-2-en-1-yl	CH3	NCH3
3040	SO2CH3	cis-3-methyl-	CH3	NCH3
		but-2-en-1-yl
3041	SO2CH3	cyclopropyl	CH3	NCH3
3042	SO2CH3	cyclopentyl	CH3	NCH3
3043	SO2CH3	cyclohexyl	CH3	NCH3
3044	SO2CH3	4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
3045	SO2CH3	4-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
3046	SO2CH3	isoxazol-3-yl	CH3	NCH3
3047	SO2CH3	4-methylisoxazol-3-yl	CH3	NCH3
3048	SO2CH3	4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
3049	SO2CH3	3-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
3050	SO2CH3	isoxazol-4-yl	CH3	NCH3
3051	SO2CH3	3-methylisoxazol-4-yl	CH3	NCH3
3052	SO2CH3	phenyl	CH3	NCH3
3053	SO2CH3	benzyl	CH3	NCH3
3054	SO2CH3	benzoyl	CH3	NCH3
3055	SO2CH3	2-pyridyl	CH3	NCH3
3056	SO2CH3	H	Cl	NCH3
3057	SO2CH3	CH3	Cl	NCH3
3058	SO2CH3	C2H5	Cl	NCH3
3059	SO2CH3	n-C3H7	Cl	NCH3
3060	SO2CH3	i-C3H7	Cl	NCH3
3061	SO2CH3	n-C4H9	Cl	NCH3
3062	SO2CH3	i-C4H9	Cl	NCH3
3063	SO2CH3	s-C4H9	Cl	NCH3
3064	SO2CH3	t-C4H9	Cl	NCH3
3065	SO2CH3	CH2OCH3	Cl	NCH3
3066	SO2CH3	CF3	Cl	NCH3
3067	SO2CH3	CF2H	Cl	NCH3
3068	SO2CH3	CN	Cl	NCH3
3069	SO2CH3	OH	Cl	NCH3
3070	SO2CH3	OCH3	Cl	NCH3
3071	SO2CH3	NH2	Cl	NCH3
3072	SO2CH3	NHCH3	Cl	NCH3
3073	SO2CH3	N(CH3)2	Cl	NCH3
3074	SO2CH3	CO2CH3	Cl	NCH3
3075	SO2CH3	CO2C2H5	Cl	NCH3
3076	SO2CH3	C(O)CH3	Cl	NCH3
3077	SO2CH3	C(O)CF3	Cl	NCH3
3078	SO2CH3	C(═NOCH3)CH3	Cl	NCH3
3079	SO2CH3	SO2CH3	Cl	NCH3
3080	SO2CH3	SO2CF3	Cl	NCH3
3081	SO2CH3	CH2CO2H	Cl	NCH3
3082	SO2CH3	CH2COOCH3	Cl	NCH3
3083	SO2CH3	CH2COOC2H5	Cl	NCH3
3084	SO2CH3	prop-1-en-3-yl	Cl	NCH3
3085	SO2CH3	trans-but-2-en-1-yl	Cl	NCH3
3086	SO2CH3	cis-but-2-en-1-yl	Cl	NCH3
3087	SO2CH3	cis-3-methyl-	Cl	NCH3
		but-2-en-1-yl
3088	SO2CH3	cyclopropyl	Cl	NCH3
3089	SO2CH3	cyclopentyl	Cl	NCH3
3090	SO2CH3	cyclohexyl	Cl	NCH3
3091	SO2CH3	4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
3092	SO2CH3	4-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
3093	SO2CH3	isoxazol-3-yl	Cl	NCH3
3094	SO2CH3	4-methylisoxazol-3-yl	Cl	NCH3
3095	SO2CH3	4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
3096	SO2CH3	3-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
3097	SO2CH3	isoxazol-4-yl	Cl	NCH3
3098	SO2CH3	3-methylisoxazol-4-yl	Cl	NCH3
3099	SO2CH3	phenyl	Cl	NCH3
3100	SO2CH3	benzyl	Cl	NCH3
3101	SO2CH3	benzoyl	Cl	NCH3
3102	SO2CH3	2-pyridyl	Cl	NCH3
3103	CF3	H	H	NCH3
3104	CF3	CH3	H	NCH3
3105	CF3	C2H5	H	NCH3
3106	CF3	n-C3H7	H	NCH3
3107	CF3	i-C3H7	H	NCH3
3108	CF3	n-C4H9	H	NCH3
3109	CF3	i-C4H9	H	NCH3
3110	CF3	s-C4H9	H	NCH3
3111	CF3	t-C4H9	H	NCH3
3112	CF3	CH2OCH3	H	NCH3
3113	CF3	CF3	H	NCH3
3114	CF3	CF2H	H	NCH3
3115	CF3	CN	H	NCH3
3116	CF3	OH	H	NCH3
3117	CF3	OCH3	H	NCH3
3118	CF3	NH2	H	NCH3
3119	CF3	NHCH3	H	NCH3
3120	CF3	N(CH3)2	H	NCH3
3121	CF3	CO2CH3	H	NCH3
3122	CF3	CO2C2H5	H	NCH3
3123	CF3	C(O)CH3	H	NCH3
3124	CF3	C(O)CF3	H	NCH3
3125	CF3	C(═NOCH3)CH3	H	NCH3
3126	CF3	SO2CH3	H	NCH3
3127	CF3	SO2CF3	H	NCH3
3128	CF3	CH2CO2H	H	NCH3
3129	CF3	CH2COOCH3	H	NCH3
3130	CF3	CH2COOC2H5	H	NCH3
3131	CF3	prop-1-en-3-yl	H	NCH3
3132	CF3	trans-but-2-en-1-yl	H	NCH3
3133	CF3	cis-but-2-en-1-yl	H	NCH3
3134	CF3	cis-3-methyl-	H	NCH3
		but-2-en-1-yl
3135	CF3	cyclopropyl	H	NCH3
3136	CF3	cyclopentyl	H	NCH3
3137	CF3	cyclohexyl	H	NCH3
3138	CF3	4,5-dihydroisoxazol-	H	NCH3
		3-yl
3139	CF3	4-methyl-4,5-dihydroisoxazol-	H	NCH3
		3-yl
3140	CF3	isoxazol-3-yl	H	NCH3
3141	CF3	4-methylisoxazol-3-yl	H	NCH3
3142	CF3	4,5-dihydroisoxazol-	H	NCH3
		4-yl
3143	CF3	3-methyl-4,5-dihydroisoxazol-	H	NCH3
		4-yl
3144	CF3	isoxazol-4-yl	H	NCH3
3145	CF3	3-methylisoxazol-4-yl	H	NCH3
3146	CF3	phenyl	H	NCH3
3147	CF3	benzyl	H	NCH3
3148	CF3	benzoyl	H	NCH3
3149	CF3	2-pyridyl	H	NCH3
3150	CF3	H	CH3	NCH3
3151	CF3	CH3	CH3	NCH3
3152	CF3	C2H5	CH3	NCH3
3153	CF3	n-C3H7	CH3	NCH3
3154	CF3	i-C3H7	CH3	NCH3
3155	CF3	n-C4H9	CH3	NCH3
3156	CF3	i-C4H9	CH3	NCH3
3157	CF3	s-C4H9	CH3	NCH3
3158	CF3	t-C4H9	CH3	NCH3
3159	CF3	CH2OCH3	CH3	NCH3
3160	CF3	CF3	CH3	NCH3
3161	CF3	CF2H	CH3	NCH3
3162	CF3	CN	CH3	NCH3
3163	CF3	OH	CH3	NCH3
3164	CF3	OCH3	CH3	NCH3
3165	CF3	NH2	CH3	NCH3
3166	CF3	NHCH3	CH3	NCH3
3167	CF3	N(CH3)2	CH3	NCH3
3168	CF3	CO2CH3	CH3	NCH3
3169	CF3	CO2C2H5	CH3	NCH3
3170	CF3	C(O)CH3	CH3	NCH3
3171	CF3	C(O)CF3	CH3	NCH3
3172	CF3	C(═NOCH3)CH3	CH3	NCH3
3173	CF3	SO2CH3	CH3	NCH3
3174	CF3	SO2CF3	CH3	NCH3
3175	CF3	CH2CO2H	CH3	NCH3
3176	CF3	CH2COOCH3	CH3	NCH3
3177	CF3	CH2COOC2H5	CH3	NCH3
3178	CF3	prop-1-en-3-yl	CH3	NCH3
3179	CF3	trans-but-2-en-1-yl	CH3	NCH3
3180	CF3	cis-but-2-en-1-yl	CH3	NCH3
3181	CF3	cis-3-methyl-	CH3	NCH3
		but-2-en-1-yl
3182	CF3	cyclopropyl	CH3	NCH3
3183	CF3	cyclopentyl	CH3	NCH3
3184	CF3	cyclohexyl	CH3	NCH3
3185	CF3	4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
3186	CF3	4-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
3187	CF3	isoxazol-3-yl	CH3	NCH3
3188	CF3	4-methylisoxazol-3-yl	CH3	NCH3
3189	CF3	4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
3190	CF3	3-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
3191	CF3	isoxazol-4-yl	CH3	NCH3
3192	CF3	3-methylisoxazol-4-yl	CH3	NCH3
3193	CF3	phenyl	CH3	NCH3
3194	CF3	benzyl	CH3	NCH3
3195	CF3	benzoyl	CH3	NCH3
3196	CF3	2-pyridyl	CH3	NCH3
3197	CF3	H	Cl	NCH3
3198	CF3	CH3	Cl	NCH3
3199	CF3	C2H5	Cl	NCH3
3200	CF3	n-C3H7	Cl	NCH3
3201	CF3	i-C3H7	Cl	NCH3
3202	CF3	n-C4H9	Cl	NCH3
3203	CF3	i-C4H9	Cl	NCH3
3204	CF3	s-C4H9	Cl	NCH3
3205	CF3	t-C4H9	Cl	NCH3
3206	CF3	CH2OCH3	Cl	NCH3
3207	CF3	CF3	Cl	NCH3
3208	CF3	CF2H	Cl	NCH3
3209	CF3	CN	Cl	NCH3
3210	CF3	OH	Cl	NCH3
3211	CF3	OCH3	Cl	NCH3
3212	CF3	NH2	Cl	NCH3
3213	CF3	NHCH3	Cl	NCH3
3214	CF3	N(CH3)2	Cl	NCH3
3215	CF3	CO2CH3	Cl	NCH3
3216	CF3	CO2C2H5	Cl	NCH3
3217	CF3	C(O)CH3	Cl	NCH3
3218	CF3	C(O)CF3	Cl	NCH3
3219	CF3	C(═NOCH3)CH3	Cl	NCH3
3220	CF3	SO2CH3	Cl	NCH3
3221	CF3	SO2CF3	Cl	NCH3
3222	CF3	CH2CO2H	Cl	NCH3
3223	CF3	CH2COOCH3	Cl	NCH3
3224	CF3	CH2COOC2H5	Cl	NCH3
3225	CF3	prop-1-en-3-yl	Cl	NCH3
3226	CF3	trans-but-2-en-1-yl	Cl	NCH3
3227	CF3	cis-but-2-en-1-yl	Cl	NCH3
3228	CF3	cis-3-methyl-	Cl	NCH3
		but-2-en-1-yl
3229	CF3	cyclopropyl	Cl	NCH3
3230	CF3	cyclopentyl	Cl	NCH3
3231	CF3	cyclohexyl	Cl	NCH3
3232	CF3	4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
3233	CF3	4-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
3234	CF3	isoxazol-3-yl	Cl	NCH3
3235	CF3	4-methylisoxazol-3-yl	Cl	NCH3
3236	CF3	4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
3237	CF3	3-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
3238	CF3	isoxazol-4-yl	Cl	NCH3
3239	CF3	3-methylisoxazol-4-yl	Cl	NCH3
3240	CF3	phenyl	Cl	NCH3
3241	CF3	benzyl	Cl	NCH3
3242	CF3	benzoyl	Cl	NCH3
3243	CF3	2-pyridyl	Cl	NCH3
3244	C2H5	H	H	NCH3
3245	C2H5	CH3	H	NCH3
3246	C2H5	C2H5	H	NCH3
3247	C2H5	n-C3H7	H	NCH3
3248	C2H5	i-C3H7	H	NCH3
3249	C2H5	n-C4H9	H	NCH3
3250	C2H5	i-C4H9	H	NCH3
3251	C2H5	s-C4H9	H	NCH3
3252	C2H5	t-C4H9	H	NCH3
3253	C2H5	CH2OCH3	H	NCH3
3254	C2H5	CF3	H	NCH3
3255	C2H5	CF2H	H	NCH3
3256	C2H5	CN	H	NCH3
3257	C2H5	OH	H	NCH3
3258	C2H5	OCH3	H	NCH3
3259	C2H5	NH2	H	NCH3
3260	C2H5	NHCH3	H	NCH3
3261	C2H5	N(CH3)2	H	NCH3
3262	C2H5	CO2CH3	H	NCH3
3263	C2H5	CO2C2H5	H	NCH3
3264	C2H5	C(O)CH3	H	NCH3
3265	C2H5	C(O)CF3	H	NCH3
3266	C2H5	C(═NOCH3)CH3	H	NCH3
3267	C2H5	SO2CH3	H	NCH3
3268	C2H5	SO2CF3	H	NCH3
3269	C2H5	CH2CO2H	H	NCH3
3270	C2H5	CH2COOCH3	H	NCH3
3271	C2H5	CH2COOC2H5	H	NCH3
3272	C2H5	prop-1-en-3-yl	H	NCH3
3273	C2H5	trans-but-2-en-1-yl	H	NCH3
3274	C2H5	cis-but-2-en-1-yl	H	NCH3
3275	C2H5	cis-3-methyl-	H	NCH3
		but-2-en-1-yl
3276	C2H5	cyclopropyl	H	NCH3
3277	C2H5	cyclopentyl	H	NCH3
3278	C2H5	cyclohexyl	H	NCH3
3279	C2H5	4,5-dihydroisoxazol-	H	NCH3
		3-yl
3280	C2H5	4-methyl-4,5-dihydroisoxazol-	H	NCH3
		3-yl
3281	C2H5	isoxazol-3-yl	H	NCH3
3282	C2H5	4-methylisoxazol-3-yl	H	NCH3
3283	C2H5	4,5-dihydroisoxazol-	H	NCH3
		4-yl
3284	C2H5	3-methyl-4,5-dihydroisoxazol-	H	NCH3
		4-yl
3285	C2H5	isoxazol-4-yl	H	NCH3
3286	C2H5	3-methylisoxazol-4-yl	H	NCH3
3287	C2H5	phenyl	H	NCH3
3288	C2H5	benzyl	H	NCH3
3289	C2H5	benzoyl	H	NCH3
3290	C2H5	2-pyridyl	H	NCH3
3291	C2H5	H	CH3	NCH3
3292	C2H5	CH3	CH3	NCH3
3293	C2H5	C2H5	CH3	NCH3
3294	C2H5	n-C3H7	CH3	NCH3
3295	C2H5	i-C3H7	CH3	NCH3
3296	C2H5	n-C4H9	CH3	NCH3
3297	C2H5	i-C4H9	CH3	NCH3
3298	C2H5	s-C4H9	CH3	NCH3
3299	C2H5	t-C4H9	CH3	NCH3
3300	C2H5	CH2OCH3	CH3	NCH3
3301	C2H5	CF3	CH3	NCH3
3302	C2H5	CF2H	CH3	NCH3
3303	C2H5	CN	CH3	NCH3
3304	C2H5	OH	CH3	NCH3
3305	C2H5	OCH3	CH3	NCH3
3306	C2H5	NH2	CH3	NCH3
3307	C2H5	NHCH3	CH3	NCH3
3308	C2H5	N(CH3)2	CH3	NCH3
3309	C2H5	CO2CH3	CH3	NCH3
3310	C2H5	CO2C2H5	CH3	NCH3
3311	C2H5	C(O)CH3	CH3	NCH3
3312	C2H5	C(O)CF3	CH3	NCH3
3313	C2H5	C(═NOCH3)CH3	CH3	NCH3
3314	C2H5	SO2CH3	CH3	NCH3
3315	C2H5	SO2CF3	CH3	NCH3
3316	C2H5	CH2CO2H	CH3	NCH3
3317	C2H5	CH2COOCH3	CH3	NCH3
3318	C2H5	CH2COOC2H5	CH3	NCH3
3319	C2H5	prop-1-en-3-yl	CH3	NCH3
3320	C2H5	trans-but-2-en-1-yl	CH3	NCH3
3321	C2H5	cis-but-2-en-1-yl	CH3	NCH3
3322	C2H5	cis-3-methyl-	CH3	NCH3
		but-2-en-1-yl
3323	C2H5	cyclopropyl	CH3	NCH3
3324	C2H5	cyclopentyl	CH3	NCH3
3325	C2H5	cyclohexyl	CH3	NCH3
3326	C2H5	4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
3327	C2H5	4-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		3-yl
3328	C2H5	isoxazol-3-yl	CH3	NCH3
3329	C2H5	4-methylisoxazol-3-yl	CH3	NCH3
3330	C2H5	4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
3331	C2H5	3-methyl-4,5-dihydroisoxazol-	CH3	NCH3
		4-yl
3332	C2H5	isoxazol-4-yl	CH3	NCH3
3333	C2H5	3-methylisoxazol-4-yl	CH3	NCH3
3334	C2H5	phenyl	CH3	NCH3
3335	C2H5	benzyl	CH3	NCH3
3336	C2H5	benzoyl	CH3	NCH3
3337	C2H5	2-pyridyl	CH3	NCH3
3338	C2H5	H	Cl	NCH3
3339	C2H5	CH3	Cl	NCH3
3340	C2H5	C2H5	Cl	NCH3
3341	C2H5	n-C3H7	Cl	NCH3
3342	C2H5	i-C3H7	Cl	NCH3
3343	C2H5	n-C4H9	Cl	NCH3
3344	C2H5	i-C4H9	Cl	NCH3
3345	C2H5	s-C4H9	Cl	NCH3
3346	C2H5	t-C4H9	Cl	NCH3
3347	C2H5	CH2OCH3	Cl	NCH3
3348	C2H5	CF3	Cl	NCH3
3349	C2H5	CF2H	Cl	NCH3
3350	C2H5	CN	Cl	NCH3
3351	C2H5	OH	Cl	NCH3
3352	C2H5	OCH3	Cl	NCH3
3353	C2H5	NH2	Cl	NCH3
3354	C2H5	NHCH3	Cl	NCH3
3355	C2H5	N(CH3)2	Cl	NCH3
3356	C2H5	CO2CH3	Cl	NCH3
3357	C2H5	CO2C2H5	Cl	NCH3
3358	C2H5	C(O)CH3	Cl	NCH3
3359	C2H5	C(O)CF3	Cl	NCH3
3360	C2H5	C(═NOCH3)CH3	Cl	NCH3
3361	C2H5	SO2CH3	Cl	NCH3
3362	C2H5	SO2CF3	Cl	NCH3
3363	C2H5	CH2CO2H	Cl	NCH3
3364	C2H5	CH2COOCH3	Cl	NCH3
3365	C2H5	CH2COOC2H5	Cl	NCH3
3366	C2H5	prop-1-en-3-yl	Cl	NCH3
3367	C2H5	trans-but-2-en-1-yl	Cl	NCH3
3368	C2H5	cis-but-2-en-1-yl	Cl	NCH3
3369	C2H5	cis-3-methyl-	Cl	NCH3
		but-2-en-1-yl
3370	C2H5	cyclopropyl	Cl	NCH3
3371	C2H5	cyclopentyl	Cl	NCH3
3372	C2H5	cyclohexyl	Cl	NCH3
3373	C2H5	4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
3374	C2H5	4-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		3-yl
3375	C2H5	isoxazol-3-yl	Cl	NCH3
3376	C2H5	4-methylisoxazol-3-yl	Cl	NCH3
3377	C2H5	4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
3378	C2H5	3-methyl-4,5-dihydroisoxazol-	Cl	NCH3
		4-yl
3379	C2H5	isoxazol-4-yl	Cl	NCH3
3380	C2H5	3-methylisoxazol-4-yl	Cl	NCH3
3381	C2H5	phenyl	Cl	NCH3
3382	C2H5	benzyl	Cl	NCH3
3383	C2H5	benzoyl	Cl	NCH3
3384	C2H5	2-pyridyl	Cl	NCH3
3385	CH3	n-Pentyl	H	O
3386	CH3	CH2—C≡C—CH2—CH3	H	O
3387	CH3	CH2—CH2—CH═CH2	H	O
3388	CH3	CH2—CH2—CH2—CH═CH2	H	O
3389	CH3	CH2—[(3-OCH3)C6H4]	H	O
3390	CH3	CH2—C≡C—CH3	H	O
3391	CH3	CH2—CH2-(1,3-dioxolan-	H	O
		2-yl)
3392	CH3	CH2-(1,3-dioxolan-	H	O
		2-yl)
3393	CH3	n-Pentyl	CH3	O
3394	CH3	CH2—C≡C—CH2—CH3	CH3	O
3395	CH3	CH2—CH2—CH═CH2	CH3	O
3396	CH3	CH2—CH2—CH2—CH═CH2	CH3	O
3397	CH3	CH2—[(3-OCH3)C6H4]	CH3	O
3398	CH3	CH2—C≡C—CH3	CH3	O
3399	CH3	CH2—CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3400	CH3	CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3401	CH3	n-Pentyl	Cl	O
3402	CH3	CH2—C≡C—CH2—CH3	Cl	O
3403	CH3	CH2—CH2—CH═CH2	Cl	O
3404	CH3	CH2—CH2—CH2—CH═CH2	Cl	O
3405	CH3	CH2—[(3-OCH3)C6H4]	Cl	O
3406	CH3	CH2—C≡C—CH3	Cl	O
3407	CH3	CH2—CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3408	CH3	CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3409	Cl	n-Pentyl	H	O
3410	Cl	CH2—C≡C—CH2—CH3	H	O
3411	Cl	CH2—CH2—CH═CH2	H	O
3412	Cl	CH2—CH2—CH2—CH═CH2	H	O
3413	Cl	CH2—[(3-OCH3)C6H4]	H	O
3414	Cl	CH2—C≡C—CH3	H	O
3415	Cl	CH2—CH2-(1,3-dioxolan-	H	O
		2-yl)
3416	Cl	CH2-(1,3-dioxolan-	H	O
		2-yl)
3417	Cl	n-Pentyl	CH3	O
3418	Cl	CH2—C≡C—CH2—CH3	CH3	O
3419	Cl	CH2—CH2—CH═CH2	CH3	O
3420	Cl	CH2—CH2—CH2—CH═CH2	CH3	O
3421	Cl	CH2—[(3-OCH3)C6H4]	CH3	O
3422	Cl	CH2—C≡C—CH3	CH3	O
3423	Cl	CH2—CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3424	Cl	CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3425	Cl	n-Pentyl	Cl	O
3426	Cl	CH2—C≡C-CH2—CH3	Cl	O
3427	Cl	CH2—CH2—CH═CH2	Cl	O
3428	Cl	CH2—CH2—CH2—CH═CH2	Cl	O
3429	Cl	CH2—[(3-OCH3)C6H4]	Cl	O
3430	Cl	CH2—C≡C—CH3	Cl	O
3431	Cl	CH2—CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3432	Cl	CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3433	OCH3	n-Pentyl	H	O
3434	OCH3	CH2—C≡C—CH2—CH3	H	O
3435	OCH3	CH2—CH2—CH═CH2	H	O
3436	OCH3	CH2—CH2—CH2—CH═CH2	H	O
3437	OCH3	CH2—[(3-OCH3)C6H4]	H	O
3438	OCH3	CH2—C≡C—CH3	H	O
3439	OCH3	CH2—CH2-(1,3-dioxolan-	H	O
		2-yl)
3440	OCH3	CH2-(1,3-dioxolan-	H	O
		2-yl)
3441	OCH3	n-Pentyl	CH3	O
3442	OCH3	CH2—C≡C—CH2—CH3	CH3	O
3443	OCH3	CH2—CH2—CH═CH2	CH3	O
3444	OCH3	CH2—CH2—CH2—CH═CH2	CH3	O
3445	OCH3	CH2—[(3-OCH3)C6H4]	CH3	O
3446	OCH3	CH2—C≡C—CH3	CH3	O
3447	OCH3	CH2—CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3448	OCH3	CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3449	OCH3	n-Pentyl	Cl	O
3450	OCH3	CH2—C≡C—CH2—CH3	Cl	O
3451	OCH3	CH2—CH2—CH═CH2	Cl	O
3452	OCH3	CH2—CH2—CH2—CH═CH2	Cl	O
3453	OCH3	CH2—[(3-OCH3)C6H4]	Cl	O
3454	OCH3	CH2—C≡C—CH3	Cl	O
3455	OCH3	CH2—CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3456	OCH3	CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3457	OCF3	n-Pentyl	H	O
3458	OCF3	CH2—C≡C—CH2—CH3	H	O
3459	OCF3	CH2—CH2—CH═CH2	H	O
3460	OCF3	CH2—CH2—CH2—CH═CH2	H	O
3461	OCF3	CH2—[(3-OCH3)C6H4]	H	O
3462	OCF3	CH2—C≡C—CH3	H	O
3463	OCF3	CH2—CH2-(1,3-dioxolan-	H	O
		2-yl)
3464	OCF3	CH2-(1,3-dioxolan-	H	O
		2-yl)
3465	OCF3	n-Pentyl	CH3	O
3466	OCF3	CH2—C≡C—CH2—CH3	CH3	O
3467	OCF3	CH2—CH2—CH═CH2	CH3	O
3468	OCF3	CH2—CH2—CH2—CH═CH2	CH3	O
3469	OCF3	CH2—[(3-OCH3)C6H4]	CH3	O
3470	OCF3	CH2—C≡C—CH3	CH3	O
3471	OCF3	CH2—CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3472	OCF3	CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3473	OCF3	n-Pentyl	Cl	O
3474	OCF3	CH2—C≡C—CH2—CH3	Cl	O
3475	OCF3	CH2—CH2—CH═CH2	Cl	O
3476	OCF3	CH2—CH2—CH2—CH═CH2	Cl	O
3477	OCF3	CH2—[(3-OCH3)C6H4]	Cl	O
3478	OCF3	CH2—C≡C—CH3	Cl	O
3479	OCF3	CH2—CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3480	OCF3	CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3481	SCH3	n-Pentyl	H	O
3482	SCH3	CH2—C≡C—CH2—CH3	H	O
3483	SCH3	CH2—CH2—CH═CH2	H	O
3484	SCH3	CH2—CH2—CH2—CH═CH2	H	O
3485	SCH3	CH2—[(3-OCH3)C6H4]	H	O
3486	SCH3	CH2—C≡C—CH3	H	O
3487	SCH3	CH2—CH2-(1,3-dioxolan-	H	O
		2-yl)
3488	SCH3	CH2-(1,3-dioxolan-	H	O
		2-yl)
3489	SCH3	n-Pentyl	CH3	O
3490	SCH3	CH2—C≡C—CH2—CH3	CH3	O
3491	SCH3	CH2—CH2—CH═CH2	CH3	O
3492	SCH3	CH2—CH2—CH2—CH═CH2	CH3	O
3493	SCH3	CH2—[(3-OCH3)C6H4]	CH3	O
3494	SCH3	CH2—C≡C—CH3	CH3	O
3495	SCH3	CH2—CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3496	SCH3	CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3497	SCH3	n-Pentyl	Cl	O
3498	SCH3	CH2—C≡C—CH2—CH3	Cl	O
3499	SCH3	CH2—CH2—CH═CH2	Cl	O
3500	SCH3	CH2—CH2—CH2—CH═CH2	Cl	O
3501	SCH3	CH2—[(3-OCH3)C6H4]	Cl	O
3502	SCH3	CH2—C≡C—CH3	Cl	O
3503	SCH3	CH2—CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3504	SCH3	CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3505	SO2CH3	n-Pentyl	H	O
3506	SO2CH3	CH2—C≡C—CH2—CH3	H	O
3507	SO2CH3	CH2—CH2—CH═CH2	H	O
3508	SO2CH3	CH2—CH2—CH2—CH═CH2	H	O
3509	SO2CH3	CH2—[(3-OCH3)C6H4]	H	O
3510	SO2CH3	CH2—C≡C—CH3	H	O
3511	SO2CH3	CH2—CH2-(1,3-dioxolan-	H	O
		2-yl)
3512	SO2CH3	CH2-(1,3-dioxolan-	H	O
		2-yl)
3513	SO2CH3	n-Pentyl	CH3	O
3514	SO2CH3	CH2—C≡C—CH2—CH3	CH3	O
3515	SO2CH3	CH2—CH2—CH═CH2	CH3	O
3516	SO2CH3	CH2—CH2—CH2—CH═CH2	CH3	O
3517	SO2CH3	CH2—[(3-OCH3)C6H4]	CH3	O
3518	SO2CH3	CH2—C≡C—CH3	CH3	O
3519	SO2CH3	CH2—CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3520	SO2CH3	CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3521	SO2CH3	n-Pentyl	Cl	O
3522	SO2CH3	CH2—C≡C—CH2—CH3	Cl	O
3523	SO2CH3	CH2—CH2—CH═CH2	Cl	O
3524	SO2CH3	CH2—CH2—CH2—CH═CH2	Cl	O
3525	SO2CH3	CH2—[(3-OCH3)C6H4]	Cl	O
3526	SO2CH3	CH2—C≡C—CH3	Cl	O
3527	SO2CH3	CH2—CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3528	SO2CH3	CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3529	CF3	n-Pentyl	H	O
3530	CF3	CH2—C≡C—CH2—CH3	H	O
3531	CF3	CH2—CH2—CH═CH2	H	O
3532	CF3	CH2—CH2—CH2—CH═CH2	H	O
3533	CF3	CH2—[(3-OCH3)C6H4]	H	O
3534	CF3	CH2—C≡C—CH3	H	O
3535	CF3	CH2—CH2-(1,3-dioxolan-	H	O
		2-yl)
3536	CF3	CH2-(1,3-dioxolan-	H	O
		2-yl)
3537	CF3	n-Pentyl	CH3	O
3538	CF3	CH2—C≡C—CH2—CH3	CH3	O
3539	CF3	CH2—CH2—CH═CH2	CH3	O
3540	CF3	CH2—CH2—CH2—CH═CH2	CH3	O
3541	CF3	CH2—[(3-OCH3)C6H4]	CH3	O
3542	CF3	CH2—C≡C—CH3	CH3	O
3543	CF3	CH2—CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3544	CF3	CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3545	CF3	n-Pentyl	Cl	O
3546	CF3	CH2—C≡C—CH2—CH3	Cl	O
3547	CF3	CH2—CH2—CH═CH2	Cl	O
3548	CF3	CH2—CH2—CH2—CH═CH2	Cl	O
3549	CF3	CH2—[(3-OCH3)C6H4]	Cl	O
3550	CF3	CH2—C≡C—CH3	Cl	O
3551	CF3	CH2—CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3552	CF3	CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3553	C2H5	n-Pentyl	H	O
3554	C2H5	CH2—C≡C—CH2—CH3	H	O
3555	C2H5	CH2—CH2—CH═CH2	H	O
3556	C2H5	CH2—CH2—CH2—CH═CH2	H	O
3557	C2H5	CH2—[(3-OCH3)C6H4]	H	O
3558	C2H5	CH2—C≡C—CH3	H	O
3559	C2H5	CH2—CH2-(1,3-dioxolan-	H	O
		2-yl)
3560	C2H5	CH2-(1,3-dioxolan-	H	O
		2-yl)
3561	C2H5	n-Pentyl	CH3	O
3562	C2H5	CH2—C≡C—CH2—CH3	CH3	O
3563	C2H5	CH2—CH2—CH═CH2	CH3	O
3564	C2H5	CH2—CH2—CH2—CH═CH2	CH3	O
3565	C2H5	CH2—[(3-OCH3)C6H4]	CH3	O
3566	C2H5	CH2C≡C—CH3	CH3	O
3567	C2H5	CH2—CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3568	C2H5	CH2-(1,3-dioxolan-	CH3	O
		2-yl)
3569	C2H5	n-Pentyl	Cl	O
3570	C2H5	CH2—C≡C—CH2—CH3	Cl	O
3571	C2H5	CH2—CH2—CH═CH2	Cl	O
3572	C2H5	CH2—CH2—CH2—CH═CH2	Cl	O
3573	C2H5	CH2—[(3-OCH3)C6H4]	Cl	O
3574	C2H5	CH2—C≡C—CH3	Cl	O
3575	C2H5	CH2—CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3576	C2H5	CH2-(1,3-dioxolan-	Cl	O
		2-yl)
3577	CH3	n-Pentyl	H	S
3578	CH3	CH2—C≡C—CH2—CH3	H	S
3579	CH3	CH2—CH2—CH═CH2	H	S
3580	CH3	CH2—CH2—CH2—CH═CH2	H	S
3581	CH3	CH2—[(3-OCH3)C6H4]	H	S
3582	CH3	CH2—C≡C—CH3	H	S
3583	CH3	CH2—CH2-(1,3-dioxolan-	H	S
		2-yl)
3584	CH3	CH2-(1,3-dioxolan-	H	S
		2-yl)
3585	CH3	n-Pentyl	CH3	S
3586	CH3	CH2—C≡C—CH2—CH3	CH3	S
3587	CH3	CH2—CH2—CH═CH2	CH3	S
3588	CH3	CH2—CH2—CH2—CH═CH2	CH3	S
3589	CH3	CH2—[(3-OCH3)C6H4]	CH3	S
3590	CH3	CH2—C≡C—CH3	CH3	S
3591	CH3	CH2—CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3592	CH3	CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3593	CH3	n-Pentyl	Cl	S
3594	CH3	CH2—C≡C—CH2—CH3	Cl	S
3595	CH3	CH2—CH2—CH═CH2	Cl	S
3596	CH3	CH2—CH2—CH2—CH═CH2	Cl	S
3597	CH3	CH2—[(3-OCH3)C6H4]	Cl	S
3598	CH3	CH2—C≡C—CH3	Cl	S
3599	CH3	CH2—CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3600	CH3	CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3601	Cl	n-Pentyl	H	S
3602	Cl	CH2—C≡C—CH2—CH3	H	S
3603	Cl	CH2—CH2—CH═CH2	H	S
3604	Cl	CH2—CH2—CH2—CH═CH2	H	S
3605	Cl	CH2—[(3-OCH3)C6H4]	H	S
3606	Cl	CH2—C≡C—CH3	H	S
3607	Cl	CH2—CH2-(1,3-dioxolan-	H	S
		2-yl)
3608	Cl	CH2-(1,3-dioxolan-	H	S
		2-yl)
3609	Cl	n-Pentyl	CH3	S
3610	Cl	CH2—C≡C—CH2—CH3	CH3	S
3611	Cl	CH2—CH2—CH═CH2	CH3	S
3612	Cl	CH2—CH2—CH2—CH═CH2	CH3	S
3613	Cl	CH2—[(3-OCH3)C6H4]	CH3	S
3614	Cl	CH2—C≡C—CH3	CH3	S
3615	Cl	CH2—CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3616	Cl	CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3617	Cl	n-Pentyl	Cl	S
3618	Cl	CH2—C≡C—CH2—CH3	Cl	S
3619	Cl	CH2—CH2—CH═CH2	Cl	S
3620	Cl	CH2—CH2—CH2—CH═CH2	Cl	S
3621	Cl	CH2—[(3-OCH3)C6H4]	Cl	S
3622	Cl	CH2—C≡C—CH3	Cl	S
3623	Cl	CH2—CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3624	Cl	CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3625	OCH3	n-Pentyl	H	S
3626	OCH3	CH2—C≡C—CH2—CH3	H	S
3627	OCH3	CH2—CH2—CH═CH2	H	S
3628	OCH3	CH2—CH2—CH2—CH═CH2	H	S
3629	OCH3	CH2—[(3-OCH3)C6H4]	H	S
3630	OCH3	CH2—C≡C—CH3	H	S
3631	OCH3	CH2—CH2-(1,3-dioxolan-	H	S
		2-yl)
3632	OCH3	CH2-(1,3-dioxolan-	H	S
		2-yl)
3633	OCH3	n-Pentyl	CH3	S
3634	OCH3	CH2—C≡C—CH2—CH3	CH3	S
3635	OCH3	CH2—CH2—CH═CH2	CH3	S
3636	OCH3	CH2—CH2—CH2—CH═CH2	CH3	S
3637	OCH3	CH2—[(3-OCH3)C6H4]	CH3	S
3638	OCH3	CH2—C≡C—CH3	CH3	S
3639	OCH3	CH2—CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3640	OCH3	CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3641	OCH3	n-Pentyl	Cl	S
3642	OCH3	CH2—C≡C—CH2—CH3	Cl	S
3643	OCH3	CH2—CH2—CH═CH2	Cl	S
3644	OCH3	CH2—CH2—CH2—CH═CH2	Cl	S
3645	OCH3	CH2—[(3-OCH3)C6H4]	Cl	S
3646	OCH3	CH2—C≡C—CH3	Cl	S
3647	OCH3	CH2—CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3648	OCH3	CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3649	OCF3	n-Pentyl	H	S
3650	OCF3	CH2—C≡C—CH2—CH3	H	S
3651	OCF3	CH2—CH2—CH═CH2	H	S
3652	OCF3	CH2—CH2—CH2—CH═CH2	H	S
3653	OCF3	CH2—[(3-OCH3)C6H4]	H	S
3654	OCF3	CH2—C≡C—CH3	H	S
3655	OCF3	CH2—CH2-(1,3-dioxolan-	H	S
		2-yl)
3656	OCF3	CH2-(1,3-dioxolan-	H	S
		2-yl)
3657	OCF3	n-Pentyl	CH3	S
3658	OCF3	CH2—C≡C—CH2—CH3	CH3	S
3659	OCF3	CH2—CH2—CH═CH2	CH3	S
3660	OCF3	CH2—CH2—CH2—CH═CH2	CH3	S
3661	OCF3	CH2—[(3-OCH3)C6H4]	CH3	S
3662	OCF3	CH2—C≡C—CH3	CH3	S
3663	OCF3	CH2—CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3664	OCF3	CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3665	OCF3	n-Pentyl	Cl	S
3666	OCF3	CH2—C≡C—CH2—CH3	Cl	S
3667	OCF3	CH2—CH2—CH═CH2	Cl	S
3668	OCF3	CH2—CH2—CH2—CH═CH2	Cl	S
3669	OCF3	CH2—[(3-OCH3)C6H4]	Cl	S
3670	OCF3	CH2—C≡C—CH3	Cl	S
3671	OCF3	CH2—CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3672	OCF3	CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3673	SCH3	n-Pentyl	H	S
3674	SCH3	CH2—C≡C—CH2—CH3	H	S
3675	SCH3	CH2—CH2—CH═CH2	H	S
3676	SCH3	CH2—CH2—CH2—CH═CH2	H	S
3677	SCH3	CH2—[(3-OCH3)C6H4]	H	S
3678	SCH3	CH2—C≡C—CH3	H	S
3679	SCH3	CH2—CH2-(1,3-dioxolan-	H	S
		2-yl)
3680	SCH3	CH2-(1,3-dioxolan-	H	S
		2-yl)
3681	SCH3	n-Pentyl	CH3	S
3682	SCH3	CH2—C≡C—CH2—CH3	CH3	S
3683	SCH3	CH2—CH2—CH═CH2	CH3	S
3684	SCH3	CH2—CH2—CH2—CH═CH2	CH3	S
3685	SCH3	CH2—[(3-OCH3)C6H4]	CH3	S
3686	SCH3	CH2—C≡C—CH3	CH3	S
3687	SCH3	CH2—CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3688	SCH3	CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3689	SCH3	n-Pentyl	Cl	S
3690	SCH3	CH2—C≡C—CH2—CH3	Cl	S
3691	SCH3	CH2—CH2—CH═CH2	Cl	S
3692	SCH3	CH2—CH2—CH2—CH═CH2	Cl	S
3693	SCH3	CH2—[(3-OCH3)C6H4]	Cl	S
3694	SCH3	CH2—C≡C—CH3	Cl	S
3695	SCH3	CH2—CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3696	SCH3	CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3697	SO2CH3	n-Pentyl	H	S
3698	SO2CH3	CH2—C≡C—CH2—CH3	H	S
3699	SO2CH3	CH2—CH2—CH═CH2	H	S
3700	SO2CH3	CH2—CH2—CH2—CH═CH2	H	S
3701	SO2CH3	CH2—[(3-OCH3)C6H4]	H	S
3702	SO2CH3	CH2—C≡C—CH3	H	S
3703	SO2CH3	CH2—CH2-(1,3-dioxolan-	H	S
		2-yl)
3704	SO2CH3	CH2-(1,3-dioxolan-	H	S
		2-yl)
3705	SO2CH3	n-Pentyl	CH3	S
3706	SO2CH3	CH2—C≡C—CH2—CH3	CH3	S
3707	SO2CH3	CH2—CH2—CH═CH2	CH3	S
3708	SO2CH3	CH2—CH2—CH2—CH═CH2	CH3	S
3709	SO2CH3	CH2—[(3-OCH3)C6H4]	CH3	S
3710	SO2CH3	CH2—C≡C—CH3	CH3	S
3711	SO2CH3	CH2—CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3712	SO2CH3	CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3713	SO2CH3	n-Pentyl	Cl	S
3714	SO2CH3	CH2—C≡C—CH2—CH3	Cl	S
3715	SO2CH3	CH2—CH2—CH═CH2	Cl	S
3716	SO2CH3	CH2—CH2—CH2—CH═CH2	Cl	S
3717	SO2CH3	CH2—[(3-OCH3)C6H4]	Cl	S
3718	SO2CH3	CH2—C≡C—CH3	Cl	S
3719	SO2CH3	CH2—CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3720	SO2CH3	CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3721	CF3	n-Pentyl	H	S
3722	CF3	CH2—C≡C—CH2—CH3	H	S
3723	CF3	CH2—CH2—CH═CH2	H	S
3724	CF3	CH2—CH2—CH2—CH═CH2	H	S
3725	CF3	CH2—[(3-OCH3)C6H4]	H	S
3726	CF3	CH2—C≡C—CH3	H	S
3727	CF3	CH2—CH2-(1,3-dioxolan-	H	S
		2-yl)
3728	CF3	CH2-(1,3-dioxolan-	H	S
		2-yl)
3729	CF3	n-Pentyl	CH3	S
3730	CF3	CH2—C≡C—CH2—CH3	CH3	S
3731	CF3	CH2—CH2—CH═CH2	CH3	S
3732	CF3	CH2—CH2—CH2—CH═CH2	CH3	S
3733	CF3	CH2—[(3-OCH3)C6H4]	CH3	S
3734	CF3	CH2—C≡C—CH3	CH3	S
3735	CF3	CH2—CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3736	CF3	CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3737	CF3	n-Pentyl	Cl	S
3738	CF3	CH2—C≡C—CH2—CH3	Cl	S
3739	CF3	CH2—CH2—CH═CH2	Cl	S
3740	CF3	CH2—CH2—CH2—CH═CH2	Cl	S
3741	CF3	CH2—[(3-OCH3)C6H4]	Cl	S
3742	CF3	CH2—C≡C—CH3	Cl	S
3743	CF3	CH2—CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3744	CF3	CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3745	C2H5	n-Pentyl	H	S
3746	C2H5	CH2—C≡C—CH2—CH3	H	S
3747	C2H5	CH2—CH2—CH═CH2	H	S
3748	C2H5	CH2—CH2—CH2—CH═CH2	H	S
3749	C2H5	CH2—[(3-OCH3)C6H4]	H	S
3750	C2H5	CH2—C≡C—CH3	H	S
3751	C2H5	CH2—CH2-(1,3-dioxolan-	H	S
		2-yl)
3752	C2H5	CH2-(1,3-dioxolan-	H	S
		2-yl)
3753	C2H5	n-Pentyl	CH3	S
3754	C2H5	CH2—C≡C—CH2—CH3	CH3	S
3755	C2H5	CH2—CH2—CH═CH2	CH3	S
3756	C2H5	CH2—CH2—CH2—CH═CH2	CH3	S
3757	C2H5	CH2—[(3-OCH3)C6H4]	CH3	S
3758	C2H5	CH2—C≡C—CH3	CH3	S
3759	C2H5	CH2—CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3760	C2H5	CH2-(1,3-dioxolan-	CH3	S
		2-yl)
3761	C2H5	n-Pentyl	Cl	S
3762	C2H5	CH2—C≡C—CH2—CH3	Cl	S
3763	C2H5	CH2—CH2—CH═CH2	Cl	S
3764	C2H5	CH2—CH2—CH2—CH═CH2	Cl	S
3765	C2H5	CH2—[(3-OCH3)C6H4]	Cl	S
3766	C2H5	CH2—C≡C—CH3	Cl	S
3767	C2H5	CH2—CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3768	C2H5	CH2-(1,3-dioxolan-	Cl	S
		2-yl)
3769	CH3	n-Pentyl	H	NCH3
3770	CH3	CH2—C≡C—CH2—CH3	H	NCH3
3771	CH3	CH2—CH2—CH═CH2	H	NCH3
3772	CH3	CH2—CH2—CH2—CHC═CH2	H	NCH3
3773	CH3	CH2—[(3-OCH3)C6H4]	H	NCH3
3774	CH3	CH2—C≡C—CH3	H	NCH3
3775	CH3	CH2—CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3776	CH3	CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3777	CH3	n-Pentyl	CH3	NCH3
3778	CH3	CH2—C≡C—CH2—CH3	CH3	NCH3
3779	CH3	CH2—CH2—CH═CH2	CH3	NCH3
3780	CH3	CH2—CH2—CH2—CH═CH2	CH3	NCH3
3781	CH3	CH2—[(3-OCH3)C6H4]	CH3	NCH3
3782	CH3	CH2—C≡C—CH3	CH3	NCH3
3783	CH3	CH2—CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3784	CH3	CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3785	CH3	n-Pentyl	Cl	NCH3
3786	CH3	CH2—C≡C—CH2—CH3	Cl	NCH3
3787	CH3	CH2—CH2—CH═CH2	Cl	NCH3
3788	CH3	CH2—CH2—CH2—CH═CH2	Cl	NCH3
3789	CH3	CH2—[(3-OCH3)C6H4]	Cl	NCH3
3790	CH3	CH2—C≡C—CH3	Cl	NCH3
3791	CH3	CH2—CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3792	CH3	CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3793	Cl	n-Pentyl	H	NCH3
3794	Cl	CH2—C≡C—CH2—CH3	H	NCH3
3795	Cl	CH2—CH2—CH═CH2	H	NCH3
3796	Cl	CH2—CH2—CH2—CH═CH2	H	NCH3
3797	Cl	CH2—[(3-OCH3)C6H4]	H	NCH3
3798	Cl	CH2—C≡C—CH3	H	NCH3
3799	Cl	CH2—CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3800	Cl	CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3801	Cl	n-Pentyl	CH3	NCH3
3802	Cl	CH2—C≡C—CH2—CH3	CH3	NCH3
3803	Cl	CH2—CH2—CH═CH2	CH3	NCH3
3804	Cl	CH2—CH2—CH2—CH═CH2	CH3	NCH3
3805	Cl	CH2—[(3-OCH3)C6H4]	CH3	NCH3
3806	Cl	CH2—C≡C—CH3	CH3	NCH3
3807	Cl	CH2—CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3808	Cl	CH2(1,3-dioxolan-	CH3	NCH3
		2-yl)
3809	Cl	n-Pentyl	Cl	NCH3
3810	Cl	CH2—C≡C—CH2—CH3	Cl	NCH3
3811	Cl	CH2—CH2—CH═CH2	Cl	NCH3
3812	Cl	CH2—CH2—CH2—CH═CH2	Cl	NCH3
3813	Cl	CH2—[(3-OCH3)C6H4]	Cl	NCH3
3814	Cl	CH2—C≡C—CH3	Cl	NCH3
3815	Cl	CH2—CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3816	Cl	CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3817	OCH3	n-Pentyl	H	NCH3
3818	OCH3	CH2—C≡C—CH2—CH3	H	NCH3
3819	OCH3	CH2—CH2—CH═CH2	H	NCH3
3820	OCH3	CH2—CH2—CH2—CH═CH2	H	NCH3
3821	OCH3	CH2—[(3-OCH3)C6H4]	H	NCH3
3822	OCH3	CH2—C≡C—CH3	H	NCH3
3823	OCH3	CH2—CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3824	OCH3	CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3825	OCH3	n-Pentyl	CH3	NCH3
3826	OCH3	CH2—C≡C—CH2—CH3	CH3	NCH3
3827	OCH3	CH2—CH2—CH═CH2	CH3	NCH3
3828	OCH3	CH2—CH2—CH2—CH═CH2	CH3	NCH3
3829	OCH3	CH2—[(3-OCH3)C6H4]	CH3	NCH3
3830	OCH3	CH2—C≡C—CH3	CH3	NCH3
3831	OCH3	CH2—CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3832	OCH3	CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3833	OCH3	n-Pentyl	Cl	NCH3
3834	OCH3	CH2—C≡C—CH2—CH3	Cl	NCH3
3835	OCH3	CH2—CH2—CH═CH2	Cl	NCH3
3836	OCH3	CH2—CH2—CH2—CH═CH2	Cl	NCH3
3837	OCH3	CH2—[(3-OCH3)C6H4]	Cl	NCH3
3838	OCH3	CH2—C≡C—CH3	Cl	NCH3
3839	OCH3	CH2—CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3840	OCH3	CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3841	OCF3	n-Pentyl	H	NCH3
3842	OCF3	CH2—C≡C—CH2—CH3	H	NCH3
3843	OCF3	CH2—CH2—CH═CH2	H	NCH3
3844	OCF3	CH2—CH2—CH2—CH═CH2	H	NCH3
3845	OCF3	CH2—[(3-OCH3)C6H4]	H	NCH3
3846	OCF3	CH2—C≡C—CH3	H	NCH3
3847	OCF3	CH2—CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3848	OCF3	CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3849	OCF3	n-Pentyl	CH3	NCH3
3850	OCF3	CH2—C≡C—CH2—CH3	CH3	NCH3
3851	OCF3	CH2—CH2—CH═CH2	CH3	NCH3
3852	OCF3	CH2—CH2—CH2—CH═CH2	CH3	NCH3
3853	OCF3	CH2—[(3-OCH3)C6H4]	CH3	NCH3
3854	OCF3	CH2—C≡C—CH3	CH3	NCH3
3855	OCF3	CH2—CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3856	OCF3	CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3857	OCF3	n-Pentyl	Cl	NCH3
3858	OCF3	CH2—C≡C—CH2—CH3	Cl	NCH3
3859	OCF3	CH2—CH2—CH═CH2	Cl	NCH3
3860	OCF3	CH2—CH2—CH2—CH═CH2	Cl	NCH3
3861	OCF3	CH2—[(3-OCH3)C6H4]	Cl	NCH3
3862	OCF3	CH2—C≡C—CH3	Cl	NCH3
3863	OCF3	CH2—CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3864	OCF3	CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3865	SCH3	n-Pentyl	H	NCH3
3866	SCH3	CH2—C≡C—CH2—CH3	H	NCH3
3867	SCH3	CH2—CH2—CH═CH2	H	NCH3
3868	SCH3	CH2—CH2—CH2—CH═CH2	H	NCH3
3869	SCH3	CH2—[(3-OCH3)C6H4]	H	NCH3
3870	SCH3	CH2—C≡C—CH3	H	NCH3
3871	SCH3	CH2—CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3872	SCH3	CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3873	SCH3	n-Pentyl	CH3	NCH3
3874	SCH3	CH2—C≡C—CH2—CH3	CH3	NCH3
3875	SCH3	CH2—CH2—CH═CH2	CH3	NCH3
3876	SCH3	CH2—CH2—CH2—CH═CH2	CH3	NCH3
3877	SCH3	CH2—[(3-OCH3)C6H4]	CH3	NCH3
3878	SCH3	CH2—C≡C—CH3	CH3	NCH3
3879	SCH3	CH2—CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3880	SCH3	CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3881	SCH3	n-Pentyl	Cl	NCH3
3882	SCH3	CH2—C≡C—CH2—CH3	Cl	NCH3
3883	SCH3	CH2—CH2—CH═CH2	Cl	NCH3
3884	SCH3	CH2—CH2—CH2—CH═CH2	Cl	NCH3
3885	SCH3	CH2—[(3-OCH3)C6H4]	Cl	NCH3
3886	SCH3	CH2—C≡C—CH3	Cl	NCH3
3887	SCH3	CH2—CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3888	SCH3	CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3889	SO2CH3	n-Pentyl	H	NCH3
3890	SO2CH3	CH2—C≡C—CH2—CH3	H	NCH3
3891	SO2CH3	CH2—CH2—CH═CH2	H	NCH3
3892	SO2CH3	CH2—CH2—CH2—CH═CH2	H	NCH3
3893	SO2CH3	CH2—[(3-OCH3)C6H4]	H	NCH3
3894	SO2CH3	CH2—C≡C—CH3	H	NCH3
3895	SO2CH3	CH2—CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3896	SO2CH3	CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3897	SO2CH3	n-Pentyl	CH3	NCH3
3898	SO2CH3	CH2—C≡C—CH2—CH3	CH3	NCH3
3899	SO2CH3	CH2—CH2—CH═CH2	CH3	NCH3
3900	SO2CH3	CH2—CH2—CH2—CH═CH2	CH3	NCH3
3901	SO2CH3	CH2—[(3-OCH3)C6H4]	CH3	NCH3
3902	SO2CH3	CH2—C≡C—CH3	CH3	NCH3
3903	SO2CH3	CH2—CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3904	SO2CH3	CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3905	SO2CH3	n-Pentyl	Cl	NCH3
3906	SO2CH3	CH2—C≡C—CH2—CH3	Cl	NCH3
3907	SO2CH3	CH2—CH2—CH═CH2	Cl	NCH3
3908	SO2CH3	CH2—CH2—CH2—CH═CH2	Cl	NCH3
3909	SO2CH3	CH2—[(3-OCH3)C6H4]	Cl	NCH3
3910	SO2CH3	CH2—C≡C—CH3	Cl	NCH3
3911	SO2CH3	CH2—CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3912	SO2CH3	CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3913	CF3	n-Pentyl	H	NCH3
3914	CF3	CH2—C≡C—CH2—CH3	H	NCH3
3915	CF3	CH2—CH2—CH═CH2	H	NCH3
3916	CF3	CH2—CH2—CH2—CH═CH2	H	NCH3
3917	CF3	CH2—[(3-OCH3)C6H4]	H	NCH3
3918	CF3	CH2—C≡C—CH3	H	NCH3
3919	CF3	CH2—CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3920	CF3	CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3921	CF3	n-Pentyl	CH3	NCH3
3922	CF3	CH2—C≡C—CH2—CH3	CH3	NCH3
3923	CF3	CH2—CH2—CH═CH2	CH3	NCH3
3924	CF3	CH2—CH2—CH2—CH═CH2	CH3	NCH3
3925	CF3	CH2—[(3-OCH3)C6H4]	CH3	NCH3
3926	CF3	CH2—C≡C—CH3	CH3	NCH3
3927	CF3	CH2—CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3928	CF3	CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3929	CF3	n-Pentyl	Cl	NCH3
3930	CF3	CH2—C≡C—CH2—CH3	Cl	NCH3
3931	CF3	CH2—CH2—CH═CH2	Cl	NCH3
3932	CF3	CH2—CH2—CH2—CH═CH2	Cl	NCH3
3933	CF3	CH2—[(3-OCH3)C6H4]	Cl	NCH3
3934	CF3	CH2—C≡C—CH3	Cl	NCH3
3935	CF3	CH2—CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3936	CF3	CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3937	C2H5	n-Pentyl	H	NCH3
3938	C2H5	CH2—C≡C—CH2—CH3	H	NCH3
3939	C2H5	CH2—CH2—CH═CH2	H	NCH3
3940	C2H5	CH2—CH2—CH2—CH═CH2	H	NCH3
3941	C2H5	CH2—[(3-OCH3)C6H4]	H	NCH3
3942	C2H5	CH2—C≡C—CH3	H	NCH3
3943	C2H5	CH2—CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3944	C2H5	CH2-(1,3-dioxolan-	H	NCH3
		2-yl)
3945	C2H5	n-Pentyl	CH3	NCH3
3946	C2H5	CH2—C≡C—CH2—CH3	CH3	NCH3
3947	C2H5	CH2—CH2—CH═CH2	CH3	NCH3
3948	C2H5	CH2—CH2—CH2—CH═CH2	CH3	NCH3
3949	C2H5	CH2—[(3-OCH3)C6H4]	CH3	NCH3
3950	C2H5	CH2—C≡C—CH3	CH3	NCH3
3951	C2H5	CH2—CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3952	C2H5	CH2-(1,3-dioxolan-	CH3	NCH3
		2-yl)
3953	C2H5	n-Pentyl	Cl	NCH3
3954	C2H5	CH2—C≡C—CH2—CH3	Cl	NCH3
3955	C2H5	CH2—CH2—CH═CH2	Cl	NCH3
3956	C2H5	CH2—CH2—CH2—CH═CH2	Cl	NCH3
3957	C2H5	CH2—[(3-OCH3)C6H4]	Cl	NCH3
3958	C2H5	CH2—C≡C—CH3	Cl	NCH3
3959	C2H5	CH2—CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)
3960	C2H5	CH2-(1,3-dioxolan-	Cl	NCH3
		2-yl)

[1149] Compounds of the formula I where R7 is hydroxyl are prepared by reacting an activated carboxylic acid IVb or a carboxylic acid IVa, which is preferably activated in situ, with 5-hydroxypyrazole of the formula III to give the acylation product, followed by rearrangement. 32

[1150] L1 is a nucleophilically replaceable leaving group, such as halogen, for example bromine or chlorine, hetaryl, for example imidazolyl or pyridyl, carboxylate, for example acetate or trifluoroacetate, etc.

[1151] The activated carboxylic acid IVb can be employed directly, such as in the case of the benzoyl halides, or be generated in situ, for example using a carbodiimide, such as ethyl-(3′-dimethylaminopropyl)carbodiimide, dicyclohexylcarbodiimide, triphenylphosphine/azodicarboxylic ester, 2-pyridine disulfide/triphenylphosphine, carbonyldiimidazole, etc.

[1152] If appropriate, it may be advantageous to carry out the acylation reaction in the presence of a base. Here, the reactants and the auxiliary base are advantageously employed in equimolar amounts. In some cases, it may be advantageous to employ a slight excess of the auxiliary base, for example from 1.2 to 1.5 molar equivalents, based on IVa or IVb.

[1153] Suitable auxiliary bases are tertiary alkylamines, pyridine, 4-dimethylaminopyridine or alkali metal carbonates. Suitable solvents are, for example, chlorinated hydrocarbons, such as methylene chloride or 1,2-dichloroethane, aromatic hydrocarbons, such as toluene, xylene or chlorobenzene, ethers, such as diethyl ether, methyl tert-butyl ether, tetrahydrofuran or dioxane, polar aprotic solvents, such as acetonitrile, dimethylformamide or dimethyl sulfoxide, or esters, such as ethyl acetate, or mixtures of these.

[1154] If the activated carboxylic acid component used is a halide, it may be advantageous to cool the reaction mixture to 0-10° C. when adding this reactant. The mixture is subsequently stirred at 20-100° C., preferably at 25-50° C., until the reaction has gone to completion. Work-up is carried out in a customary manner, for example by pouring the reaction mixture into water and extracting the product of value. Solvents which are suitable for this purpose are, in particular, methylene chloride, diethyl ether and ethyl acetate. After the organic phase has been dried and the solvent has been removed, the crude ester can be employed for the rearrangement without further purification.

[1155] The rearrangement of the esters to give the compounds of the formula I is advantageously carried out at 20-100° C. in a solvent and in the presence of a base and, if appropriate, using a cyano compound as catalyst.

[1156] Suitable solvents are, for example, acetonitrile, methylene chloride, 1,2-dichloroethane, dioxane, ethyl acetate, toluene or mixtures of these. Preferred solvents are acetonitrile and dioxane.

[1157] Suitable bases are tertiary amines, such as triethylamine, aromatic amines, such as pyridine, or alkali metal carbonates, such as sodium carbonate or potassium carbonate, which are preferably employed in an equimolar amount or an up to 4-fold excess, based on the ester. Preference is given to using triethylamine or alkali metal carbonate, preferably in twice the equimolar amount, based on the ester.

[1158] Suitable cyano compounds are inorganic cyanides, such as sodium cyanide or potassium cyanide, and organic cyano compounds, such as acetonecyanohydrin or trimethylsilyl cyanide. They are employed in an amount of 1-50 mol percent, based on the ester. Preference is given to using acetonecyanohydrin or trimethylsilyl cyanide, for example in an amount of 5-15, preferably about 10, mol percent, based on the ester.

[1159] Work-up can be carried out in a manner known per se. The reaction mixture is, for example, acidified with dilute mineral acid, such as 5% strength hydrochloric acid or sulfuric acid, and extracted with an organic solvent, for example methylene chloride or ethyl acetate. The organic extract can be extracted with 5-10% strength alkali metal carbonate solution, for example sodium carbonate or potassium carbonate solution. The aqueous phase is acidified and the precipitate that is formed is filtered off with suction and/or extracted with methylene chloride or ethyl acetate, dried and concentrated.

[1160] B. Preparation of compounds of the formula I where R7=halogen is carried out by reacting pyrazole derivatives of the formula I (where R7=hydroxyl) with halogenating agents: 33

[1161] Here and below, “compound Ia” is a compound of the formula I where Pz is a pyrazolyl radical of the formula IIa and, correspondingly, compound Ib is a compound of the formula I where Pz is a radical IIb.

[1162] Suitable halogenating agents are, for example, phosgene, diphosgene, triphosgene, thionyl chloride, oxalyl chloride, phosphorus oxychloride, phosphorus pentachloride, mesyl chloride, chloromethylene-N,N-dimethylammonium chloride, oxalyl bromide, phosphorus oxybromide, etc.

[1163] C. Preparation of compounds of the formula I where R7=OR10, OSO2R11, OPOR12R13 or OPSR12R13 by reacting pyrazole derivatives of the formula I (where R7=hydroxyl) with alkylating, sulfonylating or phosphonylating agents Vα, Vβ, Vγ and Vδ, respectively. 34

[1164] L2 is a nucleophilically replaceable leaving group, such as halogen, for example chlorine or bromine, hetaryl, for example imidazolyl, carboxylate, for example acetate, or sulfonate, for example mesylate or triflate, etc.

[1165] When preparing compounds of the formula I where R7═OR10 from compounds of the formula I where R7═OH, the reaction is preferably carried out in the presence of a base.

[1166] The reactants and the base are expediently employed in equimolar amounts. A slight excess of base, for example 1.1-1.5 molar equivalents, based on I, may be advantageous in certain cases.

[1167] Suitable bases are tertiary amines, pyridines, alkali metal carbonates or alkali metal hydrides. Suitable solvents are, for example, chlorinated hydrocarbons, such as methylene chloride or 1,2-dichloroethane, aromatic hydrocarbons, such as toluene, xylene or chlorobenzene, ethers, such as diethyl ether, methyl tert-butyl ether, tetrahydrofuran, dioxane or dimethoxyethane, polar aprotic solvents, such as acetonitrile, dimethylformamide or dimethyl sulfoxide, or esters, such as ethyl acetate, and mixtures of these.

[1168] If, in place of the alcohol I (R7═OH) halides (R7=halogen) or activated alcohols, such as mesylates or tosylates (R7═OSO2CH3 or OSO2-tolyl) are used for the derivatization, it may be expedient to cool the reaction mixture to 0° C.-10° C. when adding the reaction partner. The mixture is then stirred at 20° C.-100° C., preferably at 20° C.-75° C., until the reaction has gone to completion.

[1169] Work-up is carried out in a customary manner; for example, the reaction mixture is poured into water and the product of value is extracted. Solvents which are suitable for this purpose are, in particular, solvents such as methylene chloride, ethyl acetate, methyl tert-butyl ether or diethyl ether. The organic phase is dried and the solvent is removed and the crude product can then, if required, be purified by silica gel column chromatography. Suitable mobile phases are solvents such as methylene chloride, ethyl acetate, cyclohexane, petroleum ether, methanol, acetone or chloroform, and mixtures of these.

[1170] Compounds of the formula Vα, Vβ, Vγ or Vδ can be employed directly, such as in the case of the carbonyl halides, or be generated in situ, for example activated carboxylic acids (using carboxylic acid and dicyclohexylcarbodiimide, etc.).

[1171] D. Compounds of the formula I where R7=OR10, SR10, POR12R13, NR14R15, ONR14R15 or N-bonded heterocyclyl are prepared by reacting compounds of the formula I where R7=halogen, OSO2R11 with compounds of the formula VIα, VIβ, VIγ, VIδ, VIε or VIη, if appropriate in the presence of a base or with prior formation of salt. 35

[1172] E. Compounds of the formula I where R7═SOR11, SO2R11 are prepared, for example, by reacting compounds of the formula I where R7═SR11 with an oxidizing agent. 36

[1173] Suitable oxidizing agents are, for example, m-chloro-perbenzoic acid, peroxyacetic acid, trifluoroperoxyacetic acid, hydrogen peroxide, if appropriate in the presence of a catalyst, such as tungstate.

[1174] For the reactions mentioned under points B to E, the following conditions apply:

[1175] The starting materials are generally employed in equimolar amounts. However, it may also be advantageous to employ an excess of one or the other component.

[1176] If appropriate, it may be advantageous to carry out the reactions in the presence of a base. Reactants and base are advantageously employed in equimolar amounts.

[1177] With respect to the processes C and D, it may, in certain cases, be advantageous to employ an excess of base, for example 1.5 to 3 molar equivalents, in each case based on the starting material.

[1178] Suitable bases are tertiary alkylamines, such as triethylamine, aromatic amines, such as pyridine, alkali metal carbonates, for example sodium carbonate or potassium carbonate, alkali metal bicarbonates, such as sodium bicarbonate and potassium bicarbonate, alkali metal alkoxides, such as sodium methoxide, sodium ethoxide, potassium tert-butoxide, or alkali metal hydrides, for example sodium hydride. Preference is given to using triethylamine or pyridine.

[1179] Suitable solvents are, for example, chlorinated hydrocarbons, such as methylene chloride or 1,2-dichloroethane, aromatic hydrocarbons, for example toluene, xylene or chlorobenzene, ethers, such as diethyl ether, methyl tert-butyl ether, tetrahydrofuran or dioxane, polar aprotic solvents, such as acetonitrile, dimethylformamide or dimethyl sulfoxide, or esters, such as ethyl acetate, or mixtures of these.

[1180] In general, the reaction temperature is in the range from 0° C. to the boiling point of the reaction mixture.

[1181] Work-up can be carried out in a manner known per se to give the product.

[1182] Depending on the reaction conditions, in the processes B to D the compounds Ia, Ib, or mixtures of these can be formed. The latter can be separated by classic separation methods, for example crystallization, chromatography, etc.

[1183] F. The preparation of compounds of the formula I where Pz is a group of the formula IIa can also be carried out by reacting a metallated pyrazole derivative of the formula VII with a carboxylic acid derivative of the formula IVb: 37

[1184] Here, M is a metal, in particular an alkali metal, such as lithium or sodium, an alkaline earth metal, such as magnesium, or a transition metal, such as palladium, nickel, etc., and L1 is a nucleophilically replaceable leaving group, such as halogen, for example chlorine or bromine, alkylsulfonate, such as mesylate, haloalkylsulfonate, such as triflate or cyanide. Preferably, R7 does not have any acidic hydrogen atoms.

[1185] The reaction is generally carried out at temperatures from −100° C. to the reflux temperature of the reaction mixture. Suitable solvents are inert aprotic solvents, such as ethers, for example diethyl ether, tetrahydrofuran. The compounds of the formula IVb are generally employed in excess; however, it may also be advantageous to employ them in equimolar amounts or in substoichiometric amounts. Work-up is carried out to afford the product.

[1186] The metallated pyrazole derivatives of the formula VII can be formed in a manner known per se by reacting pyrazoles which are halogenated in the 4 position with metals such as lithium, sodium, magnesium, etc., or with organometallic compounds, for example butyllithium. However, it is also possible to metallate pyrazoles which are linked in the 4 position to hydrogen directly, for example using the abovementioned metals or organometallic compounds. The reactions are generally carried out in an inert aprotic solvent, preferably in ethers, such as diethyl ether, tetrahydrofuran, etc. The reaction temperature is in the range from −100° C. to the boiling point of the reaction mixture. The compounds of the formula VII are preferably generated in situ and reacted directly.

[1187] The 5-hydroxypyrazoles of the formula III used as starting materials are known or can be prepared by processes known per se as described, for example, in EP-A 240 001, in J. Chem. Soc. 315, (1997), p. 383, J. Prakt. Chem. 315, (1973), p. 382 (see also the reviews in Advances Heterocycle. Chem. 48, (1990), pp. 223-299 and Katritzky, Rees (Eds.), Comprehensive Heterocyclic Chem. Vol. 5, Pergamon Press 1984, Oxford, pp. 167-343 and literature cited therein). Furthermore, 1,3-dimethyl-5-hydroxypyrazole is a compound which is commercially available.

[1188] The alkylating agents Vα, sulfonylating agents Vβ, phosphonylating agents Vγ and Vδ, and the compounds VIα, VIβ, VIγ, VIδ and VIε are likewise known, or they can be prepared by known processes.

[1189] The carboxylic acids of the formula IVa and their activated derivatives IVb are novel and also form part of the subject-matter of the present invention.

[1190] Scheme 1 shows a general route to compounds of the formula IVa in which A is oxygen or NR6. 38

[1191] According to scheme 1, benzazolonecarboxylic acids of the formula IVa (A=O or NR6) can be prepared from 2-nitroanilines or 2-nitrophenols of the formula VIII, which are substituted in position 3. In step a), the nitro compounds VIII are initially brominated in the position meta to the nitro group. Brominating agents which are customary for this purpose are bromine, N-bromosuccinimide, N-bromohydantoin or pyridinium perbromide which, if appropriate, are employed together with a Lewis acid such as FeBr3. The bromination is usually carried out in an inert solvent. Suitable solvents are aliphatic or cycloaliphatic hydrocarbons, for example n-hexane or cyclohexane, halogenated hydrocarbons, for example dichloromethane, trichloromethane, carbon tetrachloride, trichloroethane, trichloroethylene, heteroaromatic compounds, such as pyridine, or anhydrous inorganic or organic acids, such as acetic acid. Customary reaction temperatures are in the range from −15° C. to 150° C., preferably in the range from −15° C. to 100° C. Methods for brominating nitro compounds are known, for example from Organikum, 16th ed., 1986, p. 315.

[1192] Subsequently, in step b), the nitro group of the compound IX is reduced to the amino group. Suitable reducing agents are, for example, hydrazines, metal hydrides, such as aluminum hydride, and complex hydrides derived therefrom, such as lithium aluminum hydride, diisobutyl aluminum hydride, or boranes, and also nascent hydrogen, for example iron, zinc or tin the presence of acids, such as hydrochloric acid or carboxylic acids, such as acetic acid. A further suitable reducing agent is hydrogen in the presence of catalytic amounts of transition metals such as nickel, palladium, platinum, ruthenium or rhodium. The transition metals can be used as such or in supported form, for example on activated carbon, in the form of activated metals, for example Raney nickel, or in the form of soluble complex compounds. The reaction is preferably carried out in a solvent. Suitable solvents for the reduction are, depending on the solubility of the substrate to be hydrogenated and the chosen reducing agent, for example C1-C4-alcohols, such as methanol, ethanol, n-propanol, isopropanol or n-butanol, halogenated C1-C6-hydrocarbons, such as dichloromethane, trichloromethane, trichloroethane, trichloroethylene, aromatic hydrocarbons, such as benzene, toluene, xylenes, chlorobenzene, aqueous solutions of inorganic acids, such as aqueous hydrochloric acid, or organic acids, and mixtures thereof with water. The reduction is usually carried out at temperatures in the range from −15° C. to +100° C., preferably in the range from 0° C. to 40° C. The reduction with hydrogen is usually carried out at a hydrogen pressure in the range from 1 to 50 bar. Catalytic hydrogenations with hydrogen are preferably carried out in the range from 1 to 10 bar. For the catalytic hydrogenation of aromatic nitro groups, see, for example, Rylander in “Catalytic Hydrogenation over Platinum Metals”, Academic Press, New York, 1967, 168-202; Furst et al., Chem. Rev. 65 (1965), 52; Tepko et al., J. Org. Chem. 45 (1980), 4992.

[1193] The 3-bromoaniline X is then, in step c), condensed to the heterocycle by reacting the compound X with a carbonic acid equivalent, such as methyl chloroformate, phosgene or its synthesis equivalents, such as diphosgene or triphosgene, under conditions which are customary for phosgenation. In general, the cyclization is carried out under neutral to acidic reaction conditions at temperatures in the range from 0° C. to 150° C. and preferably in the range from 20° C. to 120° C. The phosgenation is usually carried out in a solvent. Suitable solvents are, in particular, aliphatic or cycloaliphatic hydrocarbons, such as n-hexane or cyclohexane, halogenated hydrocarbons, such as dichloromethane, chloroform, trichloroethane, trichloroethylene, aromatic hydrocarbons, such as benzene, aliphatic ethers, such as diethyl ether, methyl tert-butyl ether, or cyclic ethers, such as tetrahydrofuran or dioxane. Phosgenation methods are known, see, for example, Justus Liebigs Ann. Chem., (2), 1978 193-213; J. Med. Chem., 30 (N 7) (1987), 1166-1176, J. Heterocycl. Chem. 28 (8) (1991), 1937-1939; J. Nat. Prod. 58 (3) (1995), 456-458.

[1194] In step d), the substituent R2 is introduced, for example, by reacting the 5-bromobenzazol-2-one XI obtained in step c) with R2-L or its precursor, L being a nucleophilically displaceable leaving group. Suitable leaving groups are, for example, halogen, such as chlorine, bromine or iodine, carboxylate, such as acetate or trifluoroacetate, or sulfonates, such as tosylate, mesylate or triflate. The reaction is preferably carried out in the presence of an auxiliary base, for example alkali metal carbonates or alkaline earth metal carbonates, such as sodium carbonate, potassium carbonate, magnesium carbonate or calcium carbonate, alkali metal hydrides or alkaline earth metal hydrides, for example sodium hydride, tertiary alkylamines, for example triethylamine, aromatic amines, for example pyridine, DMPU. The reaction is generally carried out at temperatures in the range from −15° C. to 150° C. and preferably at from 0° C. to 100° C. The reaction is usually carried out in a solvent. Suitable solvents are, for example, the abovementioned inert hydrocarbons, the abovementioned halogenated hydrocarbons, aromatic hydrocarbons, such as benzene, toluene, xylene or chlorobenzene, the abovementioned acyclic or cyclic ethers, furthermore polar aprotic solvents, such as dimethylformamide, acetonitrile or dimethyl sulfoxide. Methods for introducing a substituent at a heterocylic amide nitrogen atom are known, see also Eur. J. Med. Chem. 30 (9) (1995), 715-719; Tetrahedron 54 (9) (1998), 1763-1772.

[1195] Successive reaction of XII with magnesium or alkylmagnesium halides to the corresponding Grignard reagent and subsequent reaction of the Grignard reagent with carbon dioxide gives the carboxylic acid IVa (step e)). Customary reaction temperatures are in the range from −15° C. to 150° C., preferably in the range from −15° C. to 100° C. Suitable solvents are anhydrous solvents, in particular the abovementioned inert cyclic or acyclic hydrocarbons, the abovementioned aromatic hydrocarbons or the abovementioned acyclic or cyclic ethers. The benzazolone-5-carboxylic acid IVa is obtained by introducing dry carbon dioxide into the resulting solution of the Grignard reagent corresponding to XII and subsequent aqueous work-up. The carbon dioxide pressure is usually from 1 to 6 bar.

[1196] Alternatively, XII can be converted into carboxylic acid IVa by halogen-metal exchange using an alkali metal alkyl, for example a lithium alkyl, such as methyllithium, n-butyllithium or tert-butyllithium, and subsequent reaction of the lithiated product with CO2. Customary reaction temperatures are in the range from −100° C. to 0° C., preferably in the range from −78° C. to −50° C. Suitable solvents are anhydrous solvents, in particular the abovementioned inert hydrocarbons, the abovementioned aromatic hydrocarbons or the abovementioned acyclic or cyclic ethers. Introduction of dry carbon dioxide into the solution of the lithiated product of XII gives the benzazolonecarboxylic acid IVa. The carbon dioxide pressure is usually from 1 to 6 bar.

[1197] Reaction step e) in scheme 1 can also be realized by reacting XII with carbon monoxide, a base and water, under elevated pressure in the presence of a palladium, nickel, cobalt or rhodium catalyst.

[1198] The catalysts nickel, cobalt, rhodium and in particular palladium can be present in metallic form or in the form of customary salts, such as in the form of halogen compounds, for example palladium(II) chloride, rhodium(III) chloride hydrate, acetates, for example palladium(II) acetate, cyanides, etc., in the known valence states. Metal complexes with tertiary phosphines, metal alkyl carbonyls, metal carbonyls, for example CO2(CO)8, Ni(CO)4, metal carbonyl complexes with tertiary phosphines, for example (PPh3)2Ni(CO)2, or transition metal salts complexed with tertiary phosphines can also be employed. The lastmentioned embodiment is preferred, in particular when the catalyst used is palladium. Here, the type of phosphine ligands is of minor importance. Suitable ligands are, for example, those of the formula: 39

[1199] where the radicals R24 to R26 are low-molecular-weight alkyl, for example C1-C6-alkyl, aryl, C1-C4-alkylaryl, for example benzyl, phenethyl, or aryloxy. Aryl is, for example naphthyl, anthryl and preferably unsubstituted or substituted phenyl, where, with respect to the substituents, attention has to be paid only to their inertness to the carboxylation reaction, otherwise they can be varied widely and include all inert organocarbon radicals, such as C1-C6-alkyl radicals, for example methyl, carboxyl radicals, such as COOH, COOM (M is, for example, an alkali metal, alkaline earth metal or ammonium salt), or organocarbon radicals attached via oxygen, such as C1-C6-alkoxy radicals. A is a divalent organic radical, for example C1-C4-alkylene, 1,2-cycloalkylene, α,α′-ferrocenediyl, α,α-biphenyl or similar bifunctional groups.

[1200] The phosphine complexes can be prepared in a manner known per se, for example as described in the documents mentioned at the outset. For example, customary commercially available metal salts such as palladium(II) chloride or palladium(II) acetate are used as starting materials and the phosphine, for example P(C6H5)3, P(n-C4H9)3, PCH3(C6H5)2, 1,2-bis(diphenylphosphino)ethane, is added.

[1201] The amount of phosphine, based on the transition metal, is usually from 0 to 20, in particular from 0.1 to 10, molar equivalents, particularly preferably from 1 to 5 molar equivalents.

[1202] The amount of transition metal is not critical. Of course, for reasons of cost, preference is given to using a relatively small amount, for example from 0.1 to 10 mol %, in particular from 1 to 5 mol %, based on the starting material IVa.

[1203] For preparing the benzazolonecarboxylic acid IVa, the reaction is carried out with carbon monoxide and at least equimolar amounts of water, based on the bromide obtained in step d). The reaction component water can simultaneously also serve as solvent, i.e. the maximum amount is not critical.

[1204] However, depending on the nature of the starting materials and the catalysts used, it may also be advantageous for the solvent used to be, instead of the reaction component, another inert solvent or the base which is used for the carboxylation.

[1205] Suitable inert solvents for carboxylation reactions are customary solvents such as hydrocarbons, for example toluene, xylene, hexane, pentane, cyclohexane, ethers, for example methyl tert-butyl ether, tetrahydrofuran, dioxane, dimethoxyethane, substituted amides, such as dimethylformamide, persubstituted ureas, such as tetra-C1-C4-alkylureas, or nitrites, such as benzonitrile or acetonitrile.

[1206] In a preferred embodiment of the process, one of the reaction components, in particular the base, is used in an excess, so that no additional solvent is necessary.

[1207] Bases which are suitable for the process are all inert bases which are able to bind hydrogen iodide or hydrogen bromide liberated during the reaction. Examples which may be mentioned here are tertiary amines, such as tert-alkylamines, trialkylamines, such as triethylamine, cyclic amines, such as N-methylpiperidine or N,N′-dimethylpiperazine, pyridine, alkali metal carbonates or bicarbonates, or tetraalkyl-substituted urea derivatives, such as tetra-C1-C4-alkylurea, for example tetramethylurea.

[1208] The amount of base is not critical: customarily from 1 to 10, in particular from 1 to 5, mol are used. When the base is simultaneously used as solvent, the amount is generally such that the reaction components are dissolved, unnecessarily high excesses being avoided for reasons of practicability in order to save costs, to be able to employ small reaction vessels and to ensure that the reaction components have maximum contact.

[1209] During the reaction, the carbon monoxide pressure is adjusted such that an excess of CO, based on the bromide, is always present. At room temperature, the carbon monoxide pressure is preferably from 1 to 250 bar, in particular from 5 to 150 bar, of CO.

[1210] The carbonylation is generally carried out continuously or batchwise at from 20 to 250° C., in particular from 30 to 150° C. In the case of batchwise operation, carbon monoxide is advantageously continuously injected onto the reaction mixture to maintain a constant pressure.

[1211] It is, of course, also possible to carry out reaction step e) first and then reaction step d).

[1212] The 2-nitroanilines or 2-nitrophenols of the formula VIII, which are substituted in the 3-position, used as starting materials for the synthesis of the benzazolonecarboxylic acids IVa are known and can be prepared by processes known per se. Alternatively, the compounds IX in which A is oxygen can be prepared in the manner shown below in scheme 7.

[1213] A further general route to the benzazolonecarboxylic acids of the formula IVa is shown in scheme 2. 40

[1214] Starting with the 2-nitroanilines or 2-nitrophenols of the formula VIII, which are substituted in the 3-position, the substituted acetophenone XIII can be prepared by Friedel-Crafts acylation in step f). The acetyl group can be introduced in a known manner by reacting the compound VIII with acetic acid or activated acetic acid, such as acetic anhydride or acetyl chloride, in the presence of a Lewis acid such as aluminum trichloride, boron trifluoride or trifluoroacetic acid, under anhydrous conditions. Usually, more than 1 mol of Lewis acid is required per mole of ketone formed, since the ketone formed binds the Lewis acid as a complex. After the reaction has ended, this complex is cleaved hydrolytically. Friedel-Crafts acylations are usually carried out in a solvent. Suitable solvents are the abovementioned cyclic and acyclic hydrocarbons, the abovementioned halogenated hydrocarbons, aromatic hydrocarbons, such as nitrobenzene, or the abovementioned ethers. The reaction temperatures are generally in the range from 0° C. to 150° C. and preferably in the range from 20° C. to 120° C. Methods for introducing acyl groups are known, see, for example, Organikum, 16th ed. 1986, p. 325.

[1215] In step g), the substituted acetophenone XIII is then reduced to the amino compound XIV. The reduction is carried out in the manner described in step b) in scheme 1. In step h), the aniline derivative XIV is then phosgenated in the manner described in step c) in scheme 1. The substituent R2 can be introduced similarly to step d) in scheme 1 (step i) in scheme 2).

[1216] The compound XVI obtained in step i) in scheme 2 is converted into the benzazolonecarboxylic acid IVa with the aid of the haloform reaction. To this end, a halogenating agent, such as hypohalite, for example hypochlorite, or chlorine in alkaline solution is allowed to act on the compound XVI. Initially, a trihalomethylcarbonyl derivative is formed, which, under the alkaline reaction conditions, is cleaved hydrolytically with formation of the desired benzazolonecarboxylic acid IVa. Suitable bases are, in particular, alkali metal hydroxides, such as sodium hydroxide or potassium hydroxide. The reaction is usually carried out in solution. Suitable solvents are in particular water, mixtures of water and organic solvents, such as C1-C4-alcohols, for example methanol, ethanol, propanol, butanol, or the abovementioned ethers. Customary reaction temperatures are in the range from 0° C. to 150° C., preferably in the range from 20° C. to 120° C. For the haloform reaction, see, for example, Organikum, 16th ed. 1986, p. 375.

[1217] If A in formula IVa is sulfur, the benzazolonecarboxylic acids of the general formula IVa can also be prepared in the manner shown in scheme 3. 41

[1218] According to scheme 3, the benzazolonecarboxylic acids of the formula IVa where A=sulfur can be prepared from the aminobenzothiazoles XVII. The 2-aminobenzothiazole XVII is converted into the 2-halobenzothiazole compound XVIII in a manner known per se under Sandmeyer conditions (step k)). In this manner, further functionalities can be introduced in the 2-position of the benzothiazole ring.

[1219] To this end, the 2-aminobenzothiazole XVII is initially reacted with inorganic or organic nitrite, such as sodium nitrite in the presence of acid, such as hydrochloric acid, or with tert-butyl nitrite. The resulting diazonium salt is then reacted with an inorganic halide, such as sodium chloride, with addition of copper or a Cu(I) halide, such as Cu(I) chloride. The reaction is generally carried out at temperatures in the range from 0° C. to 150° C. and preferably in the range from 20° C. to 100° C. Suitable solvents are in particular water or mixtures of water with organic solvents, such as the abovementioned alcohols or ethers. For preparing aromatic halides, in particular chlorides, according to Sandmeyer, see also Organikum, 16th ed. 1986, p. 545.

[1220] In step 1), the 2-halobenzothiazole compound XVIII can then be hydrolyzed under acidic or alkaline conditions to give the benzothiazolone. To this end, the compound XVIII is treated with a base, such as alkali metal hydroxide or alkaline earth metal hydroxide, for example sodium hydroxide, potassium hydroxide or magnesium hydroxide, or alkali metal alkoxide, such as sodium methoxide or potassium methoxide, or with an acid, such as hydrochloric acid. The hydrolysis is usually carried out in a solvent. Suitable solvents are, depending on the base used, polar aprotic solvents, such as dimethylformamide, dimethyl sulfoxide, N-methylpyrrolidone or acetonitrile, ethers, such as tetrahydrofuran or dioxane, water and mixtures of water with the abovementioned alcohols, ethers or polar aprotic solvents. The hydrolysis is generally carried out at from 0° C. to 150° C. and preferably at from 20° C. to 120° C. For the hydrolysis of haloheteroaromatic compounds to keto compounds see also J. Med. Chem. 20 (No. 6) (1977), 791-796.

[1221] In step m), the substituent R2 is introduced into the compound XIX as described in step d) in scheme 1. For the hydrolysis in step n), for example, the benzazolone methyl ester XX obtained in step m) is reacted with alkali metal hydroxide, for example lithium hydroxide, sodium hydroxide or potassium hydroxide, with alkaline earth metal hydroxide, such as magnesium hydroxide, or with alkali metal iodides, such as sodium iodide, in a suitable solvent, preferably in the absence of oxygen. Usual reaction temperatures are in the range from 0° C. to 200° C. and in particular in the range from 20° C. to 180° C. Suitable solvents are the abovementioned aliphatic or cycloaliphatic hydrocarbons, the halogenated hydrocarbons, the aromatic hydrocarbons, the abovementioned ethers and alcohols, aqueous monophasic systems, and also pyridine. For hydrolysis, see, for example, Organikum, 16th ed. 1986, p. 415, McMurry, Org. React. 24 (1976), 187; Taschner et al., Rocz. Chem. 30 (1956), 323; Houben-Weyl: “Methoden der organischen Chemie” [Methods of Organic Chemistry], volume E 8 b 1994; p. 1010 f.; J.Chem. Soc. Perkin Trans. 1, No. 12 (1976), 1291-1296; in particular A. R. Katritzky et al., J. Heterocycl. Chem., 30 (1) (1993) 135-139. The synthesis of the starting material XVII is described in PCT/EP 00/04042 and PCT/EP 00/04040.

[1222] A further route to the compounds of the formula IVa is shown in scheme 4. 42

[1223] In step o), the 2-chlorobenzothiazole compounds XXII can be prepared in a Sandmeyer reaction from the 2-aminobenzothiazoles of the formula XXI, which are known per se. The reaction conditions required correspond to those for step k) in scheme 3. The 2-chlorobenzothiazole XXII can be brominated in a manner similar to that of step a) in scheme 1, the bromine substituent being introduced selectively in the position ortho to R1 (step p)). The compound XXIII is then, under the conditions given for step 1) in scheme 3, subjected to basic hydrolysis (step q)). In step r), the substituent R2 can be introduced into XXIV under the conditions described for step d) in scheme 1. The carboxyl group is introduced (step s)) according to the reaction conditions described in step e) in scheme 1.

[1224] A variant for preparing the benzothiazolonecarboxylic acid IVa (A=S) is shown in scheme 5. 43

[1225] Again, the initial starting materials are substituted 2-aminobenzothiazoles XXI which are converted in the manner described above into the 2-chlorobenzothiazoles XXII (step o), see scheme 3). In step u), the 2-chlorobenzothiazoles XXII are then subjected to a Friedel-Crafts acylation under the conditions given in step f) in scheme 2, giving the compound XXVII. XXVII is hydrolyzed in a manner similar to that described for reaction step q) in scheme 4. In step w), the substituent R2 is introduced into XXVIII in a manner known per se, for example as described in step d) in scheme 1. The substituted acetophenone XXIX is then, in the concluding haloform reaction in step x), under the conditions given in step j) in scheme 2, converted into the desired benzazolonecarboxylic acid IVa, with loss of a carbon.

[1226] A further route to benzazolonecarboxylic acids of the formula IVa (A=sulfur) is shown in scheme 6. 44

[1227] The o-chloronitrobenzenes of the formula XXX, which are known per se, are initially converted with alkali metal salts of benzyl mercaptan into the corresponding thioethers XXXI (step 1)). The substitution is usually carried out in one of the abovementioned aliphatic or cycloaliphatic hydrocarbons, halogenated hydrocarbons, aromatic hydrocarbons, ethers, in dimethyl-formamide, NMP, sulfolane or dimethyl sulfoxide. Customary reaction temperatures are in the range from 0° C. to 250° C. and preferably in the range from 50° C. to 175° C. Methods for nucleophilic substitution are known, see also A. Bagno et al., J. Chem. Soc. Perkin Trans. II, 1991 (5), 651-655; J. R. Beck et al., J. Org. Chem. 43 (10), (1978), 2048-2052.

[1228] In step 2), the compound XXXI is then reduced to amino compound XXXII. The required reaction conditions correspond to those for step b) in scheme 1. The amino compound XXXII is then cyclized under the reaction conditions described in step c) in scheme 1 using carbonic acid equivalents, to give the benzothiazolone XXXIII (step 3)). The substituent R2 is subsequently introduced under the reaction conditions described in step d) in scheme 1 (step 4)). The acetyl group is introduced in the position ortho to substituent R1 by Friedel-Crafts acylation of the compound XXXIV (step 5)). The required reaction conditions correspond to those of step f) in scheme 2. The desired benzazolonecarboxylic acid IVa can be obtained from compound XXXV by haloform reaction (step 6)). The required reaction conditions correspond to those in step j) in scheme 2.

[1229] In a similar manner as in scheme 1, compounds of the formula IVa where A=sulfur can be obtained in a variant of this process starting with o-chloronitrobenzenes XXX by initially brominating the thioether XXXI obtained in step 1). The required reaction conditions correspond to those of step a) in scheme 1. The subsequent reduction of the nitro group to the amino group is carried out under the conditions mentioned in step b) in scheme 1. Condensation with carbonic acid equivalents gives the benzothiazolones. The required reaction conditions correspond to those of step c) in scheme 1. The substituent R2 is introduced in the customary manner, analogously to step d) in scheme 1. The carboxyl group is introduced by the procedure described in step e) in scheme 1.

[1230] A further route to benzazolonecarboxylic acids where A=oxygen is shown in scheme 7. 45

[1231] According to scheme 7, for example, o-chloronitrobenzenes of the formula XXX can be converted with alkali metal salts of alkoxides into the corresponding o-nitroethers XXXVI (step 7)). This nucleophilic substitution on the aromatic ring is generally carried out with exclusion of water, usually in a solvent. Suitable solvents are, in particular, the abovementioned aliphatic or cycloaliphatic hydrocarbons, halogenated hydrocarbons, aromatic hydrocarbons, ethers, DMF, NMP, sulfolane or dimethyl sulfoxide. The required reaction temperatures are generally in the range from 0° C. to 250° C. and preferably from 50° C. to 175° C. Methods for preparing aromatic ethers from o-nitrochloro compounds are known, see also A. Bagno et al., J.Chem. Soc. Perkin Trans. II, 1991 (5), 651-655; J. R. Beck et al., J. Org. Chem. 43 (10) (1978), 2048-2052.

[1232] The resulting o-nitroanisole XXXVI is brominated under the reaction conditions given in step a) in scheme 1, the bromine atom being introduced selectively in position para to the methoxy group (step 8)).

[1233] In step 9), the hydroxyl group is then exposed by ether cleavage under acidic reaction conditions in the presence of a Lewis acid, such as aluminum trichloride, aluminum tribromide or hydrohalic acids, such as hydriodic acid or hydrobromic acid, giving 4-bromo-2-nitrophenols of the formula IX. The ether cleavage is usually carried out in a solvent. Suitable solvents are the abovementioned acyclic and cyclic hydrocarbons, halogenated hydrocarbons, aromatic hydrocarbons or acids, such as acetic acid. The ether cleavage is generally carried out at temperatures in the range from −15° C. to 150° C., preferably in the range from 0° C. to 100° C. For the cleavage of phenol ethers, see also Organikum, 16th ed. 1986, p. 192.

[1234] The further reaction steps 10) to 13) in scheme 7 correspond to reaction steps b) to e) in scheme 1.

[1235] The examples below serve to illustrate the invention.

EXAMPLE 1

[1236] Preparation of 3,4-dimethyl-5-(5′-hydroxy-1′-methyl-pyrazol-4-yl)carbonyl benzothiazol-2-one (compound I-1a.1129) 46

[1237] 1.1 Methyl 2-chloro-4-methylbenzothiazole-5-carboxylate

[1238] A solution of 5 g (22.5 mmol) of methyl 2-amino-4-methylbenzothiazole-5-carboxylate in 2 1 of acetonitrile was admixed with 10 ml of water, 4.5 g (44.8 mmol) of copper(I) chloride, 6.6 g of sodium chloride (110 mmol) and 2 ml of 15-crown-5. A solution of 3 g (29 mmol) of tert-butyl nitrite was then added dropwise with stirring, the solution was heated at reflux for 15 h, the resulting precipitate was filtered off and the solution was concentrated under reduced pressure. The residue was then extracted three times with in each case 500 ml of ethyl acetate. To this end, the solvent was heated to boiling point and the solution was filtered whilst hot. The extracts were concentrated under reduced pressure. The residue was purified by trituration with n-hexane/diethyl ether. This gave 4.2 g (17.4 mmol, 77% yield) of methyl 2-chloro-4-methylbenzothiazole-5-carboxylate of m.p. 112° C.

[1239] 1 H-NMR (CDCl3): δ (ppm)=2.98 (s, 3H), 3.94 (s, 3H), 7.64 (d, 1H), 7.95 (d, 1H).

[1240] 1.2 Methyl 4-methylbenzothiazol-2-one-5-carboxylate

[1241] A solution of 22.5 g (93 mmol) of methyl 2-chloro-4-methylbenzothiazole-5-carboxylate in 360 ml of N-methylpyrrolidone was admixed with 13.6 g (186 mmol) of potassium methoxide and heated at 100° C. for 5 hours. After cooling, the resulting precipitate was filtered off with suction and the filtrate was admixed with water. The pH of the reaction solution was then adjusted to pH 1, the aqueous solution was extracted three times with ethyl acetate and the combined organic phases were washed and dried. The solvent was removed under reduced pressure and the residue was purified by trituration with methylene chloride/n-hexane. This gave, in a yield of 55%, 11.38 g (51 mmol) of methyl 4-methylbenzothiazol-2-one-5-carboxylate of m.p. 262° C.-266° C.

[1242] 1 H-NMR (CDCl3): δ (ppm)=2.64 (s, 3H), 3.91 (s, 3H), 7.28 (d, 1H), 7.74 (d, 1H), 9.94 (br s, 1 H, NH).

[1243] 1.3 Methyl 3,4-dimethylbenzothiazol-2-one-5-carboxylate

[1244] A solution of 11.38 g (51 mmol) of methyl 4-methylbenzothiazol-2-one-5-carboxylate in 400 ml of acetone was admixed with 14.18 g of potassium carbonate. 5.1 ml (54 mmol) of dimethyl sulfate were then added dropwise with stirring, and the mixture was stirred at 23° C. for 78 hours. The precipitated solid was filtered off and the solvent was removed under reduced pressure. Recrystallization from ether gave, in a yield of 84%, 10.15 g (43 mmol) of methyl 3,4-dimethylbenzothiazol-2-one-5-carboxylate of m.p. 97° C.-100° C.

[1245] 1 H-NMR (CDCl3): δ (ppm)=2.78 (s, 3H), 3.77 (s, 3H), 3.92 (s, 3H), 7.28 (d, 1H), 7.36 (d, 1H).

[1246] 1.4 Methyl 3,4-dimethylbenzothiazol-2-one-5-carboxylic acid

[1247] A solution of 10.15 g (43 mmol) of methyl 3,4-dimethylbenzothiazol-2-one-5-carboxylate in 100 ml of tetrahydrofuran and 100 ml of water was admixed with 2.06 g (86 mmol) of lithium hydroxide. The solution was then heated at reflux for 2 hours. After cooling, the tetrahydrofuran was removed under reduced pressure, the remaining aqueous solution was acidified and the precipitated solid was filtered off with suction and dried. More product was obtained by extracting the mother liquor with ethyl acetate. This gave a total of 8 g (36 mmol, 83% yield) of 3,4-dimethylbenzothiazol-2-one5-carboxylic acid of m.p. 235° C.-239° C.

[1248] 1 H-NMR (DMSO-D6): δ (ppm)=2.77 (s, 3H), 3.66 (s, 3H), 7.42 (d, 1H), 7.56 (d, 1H).

[1249] 1.5 1-Methylpyrazol-5-yl 3,4-dimethylbenzothiazol-2-one5-carboxylate 0.94 g (4 mmol) of 3,4-dimethylbenzothiazol-2-one5-carboxylic acid, 0.43 g of 5-hydroxy-1-methylpyrazole and 0.81 g of ethyl(3′-dimethylaminopropyl)carbodiimide were dissolved in 40 ml of acetonitrile, and the solution was stirred at 23° C. for 10 hours. After the reaction had ended, the precipitate was filtered off and the solution was concentrated under reduced pressure. The residue was taken up in water and extracted with methylene chloride. The organic phase was washed and dried and the solvent was then removed. This gave 0.72 g (2.4 mmol, 56% yield) of 1-methyl-pyrazol-5-yl 3,4-dimethylbenzothiazol-2-one-5-carboxylate of m.p. 168° C.-174° C.

[1250] 1 H-NMR (CDCl3): δ (ppm)=2.88 (s, 3H), 3.80 (s, 3H), 3.82 (s, 3H), 6.23 (s, 1H), 7.39 (d, 1H), 7.47 (s, 1H), 7.82 (d, 1H).

[1251] 1.6 3,4-Dimethyl-5-(5′-hydroxy-1′-methylpyrazol-4-yl)carbonylbenzothiazol-2-one

[1252] With stirring, 1.41 g of potassium carbonate were added to a solution of 0.61 g (2 mmol) of 1-methylpyrazol-5-yl 3,4-dimethylbenzothiazol-2-one-5-carboxylate in 40 ml of dimethoxyethane. The reaction mixture was heated at reflux for 72 hours. The solvent was removed under reduced pressure and the residue was then taken up in water. The aqueous phase was extracted with methylene chloride, initially at pH 10.8 and then 7.0. The product could to be obtained after acidification to pH 1 by extraction with methylene chloride. Removal of the solvent gave 0.52 g (1.7 mmol, 87% yield) of the title compound of m.p. 192° C.-195° C.

[1253] 1 H-NMR (CDCl3): δ (ppm)=2.66 (s, 3H), 3.73 (s, 3H), 3.79 (s, 3H), 4.60 (m, 1H), 7.26 (d, 1H), 7.36 (d, 1H), 7.38 (s, 1H).

EXAMPLE 2

[1254] Preparation of 3,4-dimethyl-5-(5′-hydroxy-1′-ethylpyrazol-4-yl)carbonylbenzothiazol-2-one (compound I-1b.1129) 47

[1255] 2.1 1-Ethylpyrazol-5-yl 3,4-dimethylbenzothiazol-2-one-5-carboxylate

[1256] The reaction was carried out analogously to the procedure described in Example 1.5, but using 1.1 g (5 mmol) of 3,4-dimethylbenzothiazol-2-one-5-carboxylic acid, 0.58 g of hydroxy-1-ethylpyrazole and 0.94 g of ethyl-(3′-dimethylaminopropyl)carbodiimide.

[1257] This gave 0.55 g (1.7 mmol, 34% yield) of 1-ethylpyrazol-5-yl 3,4-dimethylbenzothiazol-2-one-5-carboxylate of m.p. 122° C.-124° C.

[1258] 1 H-NMR (CDCl3): δ (ppm)=1.42 (t, 3H), 2.88 (s, 3H), 3.90 (s, 3H), 4.12 (q, 2H), 6.23 (s, 1H), 7.39 (d, 1H), 7.50 (s, 1H), 7.79 (d, 1H).

[1259] 2.2 3,4-Dimethyl-5-(5′-hydroxy-1′-ethylpyrazol-4-yl)carbonyl-benzothiazol-2-one

[1260] The reaction was carried out analogously to the procedure described in Example 1.6, but using, in place of 0.62 g (2 mmol) of 1-methylpyrazol-5-yl 3,4-dimethylbenzothiazol-2-one-5-carboxylate, 0.53 g (1.7 mmol) of 1-ethylpyrazol-5-yl 3,4-dimethylbenzothiazol-2-one-5-carboxylate.

[1261] The title compound was purified by triturating the resulting crude product with ether. This gave 0.17 g (0.5 mmol, 32% yield) of product of m.p. 147° C.-149° C.

[1262] 1 H-NMR (CDCl3): δ (ppm)=1.44 (t, 3H), 2.66 (s, 3H), 3.79 (s, 3H), 4.09 (q, 2H), 7.26 (d, 1H), 7.36 (d, 1H), 7.38 (s, 1H).

EXAMPLE 3

[1263] Preparation of 3,4-dimethyl-5-(5′-hydroxy-1′-isopropylpyrazol-4-yl)carbonylbenzothiazol-2-one (compound I-1c.1129) 48

[1264] 3.1 1-Isopropylpyrazol-5-yl 3,4-dimethylbenzothiazol-2-one-5-carboxylate

[1265] The reaction was carried out analogously to the procedure described in Example 1.5.

[1266] Starting with 1.1 g (5 mmol) of 3,4-dimethylbenzothiazol-2-one-5-carboxylic acid, 0.65 g of 5-hydroxy-1-isopropyl-pyrazole and 0.94 g of ethyl-(3′-dimethylaminopropyl)carbodiimide, 0.65 g (2 mmol, 40% yield) of 1-isopropyl-pyrazol-5-yl 3,4-dimethylbenzothiazol-2-one-5-carboxylate of m.p. 137° C.-140° C. were isolated.

[1267] 1 H-NMR (CDCl3): δ (ppm)=1.48 (d, 6H), 2.88 (s, 3H), 3.90 (s, 3H), 4.52 (m, 1H), 6.21 (s, 1H), 7.40 (d, 1H), 7.51 (s, 1H), 7.80 (d, 1H).

[1268] 3.2 3,4-Dimethyl-5-(5′-hydroxy-1′-isopropylpyrazol-4-yl)-carbonylbenzothiazol-2-one

[1269] The reaction was carried out analogously to the procedure in Example 1.6, but using, in place of 1-methylpyrazol-5-yl 3,4-dimethylbenzothiazol-2-one-5-carboxylate, 0.63 g (1.9 mmol) of 1-isopropylpyrazol-5-yl 3,4-dimethylbenzo-thiazol-2-one-5-carboxylate.

[1270] This gave 0.39 g (1.2 mmol, 65% yield) of the title compound of m.p. 175° C.-177° C.

[1271] 1 H-NMR (CDCl3): δ (ppm)=1.68 (d, 6H), 2.66 (s, 3H), 3.79 (s, 3H), 4.60 (m, 1H), 7.26 (d, 1H), 7.36 (d, 1H), 7.38 (s, 1H).

[1272] The compounds I of Examples 4 to 47 were obtained in a similar manner by reacting the respective carboxylic acid IVa with the 5-hydroxypyrazole III and optionally followed by derivatization of the thus obtained compound I.

		m.p. or 13C-NMR or 1H-NMR
Ex.	Structure/Compound No.	(CDCl3)
1	49	m.p. 192° C. to 195° C.
2	50	m.p. 147° C. to 149° C.
3	51	m.p. 175° C. to 177° C.
4	52	m.p. 155° C. to 158° C.
5	53	δ (ppm) = 193.08 (C═O), 170.49 (C═O), 16.14 (CH3)
6	54	m.p. 200° C. to 203° C.
7	55	m.p. 127° C. to 129° C.
8	56	m.p. 156° C. to 157° C.
9	57	m.p. 165° C. to 167° C.
10	58	m.p. 181° C. to 182° C.
11	59	m.p. 122° C. to 123° C.
12	60	m.p. 108° C. to 110° C.
13	61	m.p. 144° C. to 147° C.
14	62	δ (ppm) = 1.35 (t, 3H), 2.55 (s, 3H), 3.55 (s, 3H), 4.30 (m, 2H), 5.55 (s, 2H), 7.10 (d, 1H), 7.30-7.40 (m, 7H)
15	63	m.p. 135° C. to 137° C.
16	64	m.p. 65° C. to 71° C.
17	65	m.p. 142° C. to 144° C.
18	66	m.p. 153° C. to 156° C.
19	67	δ (ppm) = 0.95 (t, 3H), 1.50 (d, 6H), 1.75 (m, 2H), 2.65 (s, 3H), 4.20 (t, 2H), 4.60 (m, 1H), 7.20-7.35 (m, 3H), 8.6 (s, 1H)
20	68	m.p. 140° C. to 147° C.
21	69	m.p. 54° C. to 60° C.
22	70	δ (ppm) = 1.50 (d, 6H), 2.15 (m, 2H), 2.70 (s, 3H), 3.80 (m, 2H), 3.90 (m, 2H), 4.40 (m, 2H), 4.60 (m, 1H), 4.95 (m, 1H), 7.20-7.25 (m, 3H), 7.40 (d, 1H)
23	71	m.p. 54° C. to 58° C.
24	72	m.p. 133° C. to 134° C.
25	73	m.p. 117° C. to 121° C.
26	74	m.p. 150° C. to 151° C.
27	75	m.p. 104° C. to 105° C.
28	76	m.p. 56° C. to 61° C.
29	77	δ (ppm) = 1.70 (s, 3H), 1.75 (s, 3H), 2.70 (s, 3H), 3.65 (s, 3H), 4.90 (s, 2H), 7.00 (d, 1H), 7.35 (d, 1H)
30	78	δ (ppm) = 0.95 (t, 3H), 1.40 (m, 4H), 1.75, (m, 2H), 2.55 (s, 3H), 3.55 (s, 3H), 4.05 (m, 2H), 5.55 (s, 2H), 7.10 (d, 1H), 7.15 (d, 1H), 7.35 (m, 6H)
31	79	δ (ppm) = 0.95 (t, 3H), 1.25 (d, 6H), 1.40 (m, 4H), 1.80 (m, 2H), 2.55 (s, 3H), 3.55 (s, 3H), 4.05 (m, 2H), 5.55 (s, 2H), 7.10 (d, 1H), 7.15 (d, 1H), 7.35 (m, 6H)
32	80	δ (ppm) = 1.75 (s, 3H), 2.75 (s, 3H), 3.55 (s, 3H), 4.90 (s, 3H), 5.05 (s, 2H), 7.10 (d, 1H), 7.30-7.40 (m, 7H)
33	81	δ (ppm) = 1.25 (d, 6H), 1.80 (s, 3H), 2.75 (s, 3H), 4.50 (m, 1H), 4.90 (s, 2H), 5.05 (s, 2H), 7.10 (d, 1H), 7.30-7.40 (m, 7H)
34	82	δ (ppm) = 0.95 (t, 3H), 1.75 (m, 2H), 2.55 (s, 3H), 3.60 (s, 3H), 4.20 (m, 2H), 5.50 (s, 2H), 7.10 (d, 1H), 7.25-7.40 (m, 7H)
35	83	m.p. 150° C. to 151° C.
36	84	δ (ppm) = 1.25 (d, 6H), 2.35 (s, 3H), 4.45 (m, 1H), 5.45 (m, 4H), 7.10-7.35 (m, 11H)
37	85	δ (ppm) = 0.95 (t, 3H), 1.65 (m, 2H), 2.05 (s, 3H), 2.55 (s, 3H), 3.50 (s, 3H), 4.15 (m, 2H), 4.95 (s, 2H), 7.05-7.35 (m, 7H)
38	86	δ (ppm) = 0.95 (t, 3H), 1.25 (d, 6H), 1.75 (m, 2H), 2.60 (s, 3H), 4.20 (m, 2H), 4.50 (m, 1H), 5.55 (s, 2H), 7.15 (d, 1H), 7.30-7.40 (m, 7H)
39	87	m.p. 105° C. to 107° C.
40	88	δ (ppm) = 1.10 (t, 3H), 1.50 (d, 6H), 2.20 (m, 2H), 2.80 (s, 3H), 4.60 (m, 1H), 4.95 (s, 2H), 7.25-7.45 (m, 3H)
41	89	δ (ppm) = 0.90 (t, 3H), 1.35 (m, 4H), 1.75 (m, 2H), 2.55 (s, 3H), 3.55 (s, 3H), 4.20 (m, 2H), 5.55 (s, 2H), 7.10 (d, 1H), 7.30-7.40 (m, 7H)
42	90	δ (ppm) = 1.50 (d, 6H), 1.75 (s, 3H), 1.80 (s, 3H), 2.60 (s, 3H), 4.60 (m, 1H), 4.70 (m, 2H), 5.25 (m, 1H), 7.15 (d, 1H), 7.30 (d, 1H), 7.40 (d, 1H), 9.5 (s, 1H)
43	91	δ (ppm) = 2.50 (m, 2H), 2.65 (s, 3H), 3.75 (s, 3H), 4.30 (m, 2H), 5.05 (m, 2H), 5.80 (m, 1H), 7.25 (d, 1H), 7.40 (d, 1H), 8.9 (s, 1H)
44	92	m.p. 71° C. to 74° C.
45	93	m.p. 79° C. to 89° C.
46	94	δ (ppm) = 1.35 (t, 3H), 1.65 (s, 9H) 2.60 (s, 3H), 4.30 (q, 2H), 5.55 (s, 2H), 7.10-7.55 (m, 8H)
47	95	δ (ppm) = 1.25 (t, 3H), 1.40 (t, 3H), 2.60 (s, 3H), 3.95 (q, 2H), 4.30 (q, 2H), 5.55 (s, 2H), 7.10 (d, 1H), 7.25-7.40 (m, 7H)

[1273] The compounds I and their agriculturally useful salts are suitable, both as isomer mixtures and in the form of the pure isomers, for use as herbicides. The herbicidal compositions comprising compounds I effect very good control of vegetation on non-crop areas, especially at high application rates. In crops such as wheat, rice, maize, soybeans and cotton, they act against broad-leaved weeds and grass weeds without causing any significant damage to the crop plants. This effect is observed in particular at low application rates.

[1274] Depending on the application method in question, the compounds I or the herbicidal compositions comprising them can additionally be employed in a further number of crop plants for eliminating undesirable plants. Suitable crops are, for example, the following:

[1275] Allium cepa, Ananas comosus, Arachis hypogaea, Asparagus officinalis, Beta vulgaris spec. altissima, Beta vulgaris spec. rapa, Brassica napus var. napus, Brassica napus var. napobrassica, Brassica rapa var. silvestris, Camellia sinensis, Carthamus tinctorius, Carya illinoinensis, Citrus limon, Citrus sinensis, Coffea arabica (Coffea canephora, Coffea liberica), Cucumis sativus, Cynodon dactylon, Daucus carota, Elaeis guineensis, Fragaria vesca, Glycine max, Gossypium hirsutum, (Gossypium arboreum, Gossypium herbaceum, Gossypium vitifolium), Helianthus annuus, Hevea brasiliensis, Hordeum vulgare, Humulus lupulus, Ipomoea batatas, Juglans regia, Lens culinaris, Linum usitatissimum, Lycopersicon lycopersicum, Malus spec., Manihot esculenta, Medicago sativa, Musa spec., Nicotiana tabacum (N.rustica), Olea europaea, Oryza sativa, Phaseolus lunatus, Phaseolus vulgaris, Picea abies, Pinus spec., Pisum sativum, Prunus avium, Prunus persica, Pyrus communis, Ribes sylvestre, Ricinus communis, Saccharum officinarum, Secale cereale, Solanum tuberosum, Sorghum bicolor (s. vulgare), Theobroma cacao, Trifolium pratense, Triticum aestivum, Triticum durum, Vicia faba, Vitis vinifera and Zea mays.

[1276] In addition, the compounds I can also be used in crops which tolerate the action of herbicides due to breeding, including genetic engineering methods.

[1277] The compounds I, or the compositions comprising them, can be applied, for example, in the form of directly sprayable aqueous solutions, powders, suspensions, including highly-concentrated aqueous, oily or other suspensions or dispersions, emulsions, oil ispersions, pastes, dusts, materials for broadcasting or granules, by means of spraying, atomizing, dusting, broadcasting, pouring or seed dressing or mixing with the seed. The use forms depend on the intended purposes; in each case, they should ensure the finest possible distribution of the active compounds according to the invention. The herbicidal compositions comprise a herbicidally effective amount of at least one compound of the formula I or an agriculturally useful salt of I and auxiliaries which are customarily used for formulating crop protection agents.

[1278] Suitable inert additives are essentially:

[1279] Mineral oil fractions of medium to high boiling point, such as kerosene and diesel oil, furthermore coal tar oils and oils of vegetable or animal origin, aliphatic, cyclic and aromatic hydrocarbons, for example paraffin, tetrahydro-naphthalene, alkylated naphthalenes and their derivatives, alkylated benzenes and their derivatives, alcohols such as methanol, ethanol, propanol, butanol and cyclohexanol, ketones such as cyclohexanone, strongly polar solvents, for example amines such as N-methylpyrrolidone, and water.

[1280] Aqueous use forms can be prepared from emulsion concentrates, suspensions, pastes, wettable powders or water-dispersible granules by adding water. To prepare emulsions, pastes or oil dispersions, the compounds of the formula I, as such or dissolved in an oil or solvent, can be homogenized in water by means of wetting agent, tackifier, dispersant or emulsifier. Alternatively, it is possible to prepare concentrates from active substance, wetting agent, tackifier, dispersant or emulsifier and, if desired, solvent or oil, and these concentrates are suitable for dilution with water.

[1281] Suitable surfactants are the alkali metal salts, alkaline earth metal salts and ammonium salts of aromatic sulfonic acids, for example ligno-, phenol-, naphthalene- and dibutylnaphthalene-sulfonic acid, and of fatty acids, of alkyl- and alkylaryl-sulfonates, of alkyl sulfates, lauryl ether sulfates and fatty alcohol sulfates, and the salts of sulfated hexa-, hepta- and octadecanols and of fatty alcohol glycol ethers, condensates of sulfonated naphthalene and its derivatives with formaldehyde, condensates of naphthalene or of the naphthalenesulfonic acids with phenol and formaldehyde, polyoxyethylene octylphenol ether, ethoxylated isooctyl-, octyl- or nonylphenol, alkylphenyl polyglycol ethers, tributylphenyl polyglycol ether, alkylaryl polyether alcohols, isotridecyl alcohol, fatty alcohol/ethylene oxide condensates,-ethoxylated castor oil, polyoxyethylene alkyl ethers or polyoxypropylene alkyl ethers, lauryl alcohol polyglycol ether acetate, sorbitol esters, lignin-sulfite waste liquors or methylcellulose.

[1282] Powders, materials for spreading and dusts can be prepared by mixing or concomitant grinding of the active substances with a solid carrier.

[1283] Granules, e.g. coated granules, impregnated granules and homogeneous granules, can be prepared by binding the active compounds to solid carriers. Solid carriers are mineral earths such as silicas, silica gels, silicates, talc, kaolin, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate, magnesium sulfate, magnesium oxide, ground synthetic materials, fertilizers such as ammonium sulfate, ammonium phosphate, ammonium nitrate, ureas, and products of vegetable origin such as cereal meal, tree bark meal, wood meal and nutshell meal, cellulose powders, or other solid carriers.

[1284] The concentrations of the active compounds I in the ready-to-use products can be varied within wide ranges. In general, the formulations comprise from 0.001 to 98% by weight, preferably 0.01 to 95% by weight, of at least one active compound. The active compounds are employed in a purity of from 90% to 100%, preferably 95% to 100% (according to NMR spectrum).

[1285] The compounds I according to the invention can be formulated, for example, as follows:

[1286] I. 20 parts by weight of the compound of the formula I are dissolved in a mixture composed of 80 parts by weight of alkylated benzene, 10 parts by weight of the adduct of 8 to 10 mol of ethylene oxide to 1 mol of oleic acid N-monoethanolamide, 5 parts by weight of calcium dodecylbenzenesulfonate and 5 parts by weight of the adduct of 40 mol of ethylene oxide and 1 mol of castor oil. Pouring the solution into 100,000 parts by weight of water and finely distributing it therein gives an aqueous dispersion which comprises 0.02% by weight of the active compound.

[1287] II. 20 parts by weight of the compound of the formula I are dissolved in a mixture composed of 40 parts by weight of cyclohexanone, 30 parts by weight of isobutanol, 20 parts by weight of the adduct of 7 mol of ethylene oxide to 1 mol of isooctylphenol and 10 parts by weight of the adduct of 40 mol of ethylene oxide to 1 mol of castor oil. Pouring the solution into 100,000 parts by weight of water and finely distributing it therein gives an aqueous dispersion which comprises 0.02% by weight of the active compound.

[1288] III. 20 parts by weight of the active compound of the formula I are dissolved in a mixture composed of 25 parts by weight of cyclohexanone, 65 parts by weight of a mineral oil fraction of boiling point 210 to 280° C. and 10 parts by weight of the adduct of 40 mol of ethylene oxide and 1 mol of castor oil. Pouring the solution into 100,000 parts by weight of water and finely distributing it therein gives an aqueous dispersion which comprises 0.02% by weight of the active compound.

[1289] IV. 20 parts by weight of the active compound of the formula I are mixed thoroughly with 3 parts by weight of sodium diisobutylnaphthalenesulfonate, 17 parts by weight of the sodium salt of a lignosulfonic acid from a sulfite waste liquor and 60 parts by weight of pulverulent silica gel, and the mixture is ground in a hammer mill. Finely distributing the mixture in 20,000 parts by weight of water gives a spray mixture which comprises 0.1% by weight of the active compound.

[1290] V. 3 parts by weight of the active compound of the formula I are mixed with 97 parts by weight of finely divided kaolin. This gives a dust which comprises 3% by weight of the active compound.

[1291] VI. 20 parts by weight of the active compound of the formula I are mixed intimately with 2 parts by weight of calcium dodecylbenzenesulfonate, 8 parts by weight of fatty alcohol polyglycol ether, 2 parts by weight of the sodium salt of a phenol/urea/formaldehyde condensate and 68 parts by weight of a paraffinic mineral oil. This gives a stable oily dispersion.

[1292] VII. 1 part by weight of the compound of the formula I is dissolved in a mixture composed of 70 parts by weight of cyclohexanone, 20 parts by weight of ethoxylated isooctylphenol and 10 parts by weight of ethoxylated castor oil. This gives a stable emulsion concentrate.

[1293] VIII. 1 part by weight of the compound of the formula I is dissolved in a mixture composed of 80 parts by weight of cyclohexanone and 20 parts by weight of Wettol® EM 31 (=non-ionic emulsifier based on ethoxylated castor oil). This gives a stable emulsion concentrate.

[1294] The herbicidal compositions or the active compounds can be applied pre- or post-emergence or together in the seed of a crop plant. It is also possible to apply the herbicidal compositions or active compounds by applying crop plant seed pretreated with the herbicidal compositions or active compounds. If the active compounds are less-well tolerated by certain crop plants, it is possible to use application techniques in which the herbicidal compositions are sprayed, with the aid of the spraying equipment, in such a way that they come into as little contact as possible, if any, with the leaves of the sensitive crop plants while the active compounds reach the leaves of undesirable plants which grow underneath, or the bare soil surface (post-directed, lay-by).

[1295] Depending on the intended aim, the season, the target plants and the growth stage, the rates of application of the active compound I are from 0.001 to 3.0, preferably 0.01 to 1.0, kg of active substance (a.s.)/ha.

[1296] To widen the spectrum of action and to achieve synergistic effects, the compounds I may be mixed, and applied jointly, with a large number of representatives of other groups of herbicidally or growth-regulating active compounds. Suitable examples of components in mixtures are 1,2,4-thiadiazoles, 1,3,4-thiadiazoles, amides, aminophosphoric acid and its derivatives, aminotriazoles, anilides, (het)aryloxyalkanoic acids and their derivatives, benzoic acid and its derivatives, benzothiadiazinones, 2-aroyl-1,3-cyclohexanediones, 2-hetaroyl-1,3-cyclohexanedione, hetaryl aryl ketones, benzylisoxazolidinones, meta-CF3-phenyl derivatives, carbamates, quinolinecarboxylic acid and its derivatives, chloroacetanilides, cyclohexenone oxime ether derivatives, diazines, dichloropropionic acid and its derivatives, dihydrobenzofurans, dihydrofuran-3-ones, dinitroanilines, dinitrophenols, diphenyl ethers, dipyridyls, halocarboxylic acids and their derivatives, ureas, 3-phenyluracils, imidazoles, imidazolinones, N-phenyl-3,4,5,6-tetrahydrophthalimides, oxadiazoles, oxiranes, phenols, aryloxy- and hetaryloxyphenoxypropionic esters, phenylacetic acid and its derivatives, phenylpropionic acid and its derivatives, pyrazoles, phenylpyrazoles, pyridazines, pyridinecarboxylic acid and its derivatives, pyrimidyl ethers, sulfonamides, sulfonylureas, triazines, triazinones, triazolinones, triazolecarboxamides and uracils.

[1297] Moreover, it may be advantageous to apply the compounds I alone or in combination with other herbicides, even in the form of a mixture together with further crop protection agents, for example with pesticides or agents for controlling phytopathogenic fungi or bacteria. Also of interest is the miscibility with mineral salt solutions which are employed for treating nutritional and trace element deficiencies. Nonphytotoxic oils and oil concentrates may also be added.

[1298] Use Examples

[1299] The herbicidal activity of the benzazolones of the formula I was demonstrated by the following greenhouse experiments:

[1300] The culture containers used were plastic pots containing loamy sand with approximately 3.0% of humus as substrate. The seeds of the test plants were sown separately for each species.

[1301] For the pre-emergence treatment, the active compounds, suspended or emulsified in water, were applied directly after sowing by means of finely distributing nozzles. The containers were irrigated gently to promote germination and growth and subsequently covered with translucent plastic hoods until the plants had rooted. This cover caused uniform germination of the test plants unless this was adversely affected by the active compounds.

[1302] For the post-emergence treatment, the test plants were first grown to a plant height of from 3 to 15 cm, depending on the plant habit, and only then treated with the active compounds which had been suspended or emulsified in water. To this end, the test plants were either sown directly and grown in the same containers, or they were first grown separately as seedlings and transplanted into the test containers a few days prior to treatment. The rate of application for the post-emergence treatment was 31.3, 62.5, 125 and/or 250 g of a.s. (active substance) /ha.

[1303] Depending on the species, the plants were kept at from 10 to 25° C., or 20-35° C., respectively. The test period extended over 2 to 4 weeks. During this time, the plants were tended, and their response to the individual treatments was evaluated.

[1304] Evaluation was carried out using a scale of from 0 to 100. 100 means no emergence of the plants, or complete destruction of at least the aerial parts, and 0 means no damage, or normal course of growth. A damage of at least 95% corresponds to very good herbicidal action.

[1305] The plants used in the greenhouse experiments were of the following species:

Bayercode Common Name
AMARE     redroot pigweed
BIDPI     hairy beggarticks
BRAPL     marmelade grass
CHEAL     lambsquarters (goo-
          sefoot)
ECHCG     barnyardgrass
LAMAM     henbit
PAPRH     cornpoppy
PHBPU     morningglory, com-
          mon
POLPE     ladysthumb
SETFA     giant foxtail
STEME     chickweed
THLAR     pennycress

[1306] The following results were obtained by the post-emergence method.

[1307] At application rates of 31.3 or 62.5 g/ha (a.s.), the compound I-1a.1129 from Example 1, used by the post-emergence method, showed very good herbicidal action against CHEAL, SETFA, STEME and THLAR.

[1308] At application rates of 31.3 or 62.5 g/ha (a.s.), the compound I-1b.1129 from Example 2, used by the post-emergence method, showed very good herbicidal action against CHEAL, ECHCG, PARPH, STEME and THLAR.

[1309] At application rates of 31.3 or 62.5 g/ha (a.s.), the compound I-1c.1129 from Example 3, used by the post-emergence method, showed very good herbicidal action against AMARE, CHEAL, ECHCG and POLPE.

[1310] At application rates of 125 or 250 g/ha (a.s.), the compound I-1a.1131 from Example 10, used by the post-emergence method, showed very good herbicidal action against BRAPL. AMARE, CHEAL, ECHCG and SETFA.

[1311] At application rates of 125 or 250 g/ha (a.s.), the compound I-1b.1131 from Example 11, used by the post-emergence method, showed very good herbicidal action against BRAPL. AMARE, CHEAL, ECHCG and SETFA.

[1312] At application rates of 125 or 250 g/ha (a.s.), the compound I-1c.1131 from Example 12, used by the post-emergence method, showed very good herbicidal action against BRAPL. AMARE, CHEAL, ECHCG and SETFA.

[1313] At application rates of 125 or 250 g/ha (a.s.), the compound I-1d.1131 from Example 13, used by the post-emergence method, showed very good herbicidal action against BRAPL. AMARE, CHEAL, ECHCG and SETFA.

[1314] At application rates of 125 or 250 g/ha (a.s.), the compound I-1h.1131 from Example 47, used by the post-emergence method, showed very good herbicidal action against BRAPL. AMARE, CHEAL, ECHCG and SETFA.

[1315] At application rates of 125 or 250 g/ha (a.s.), the compound I-1y.1131 from Example 46, used by the post-emergence method, showed very good herbicidal action against BRAPL. PHBPU, CHEAL, ECHCG and SETFA.

[1316] At application rates of 125 or 250 g/ha (a.s.), the compound I-1g.1131 from Example 14, used by the post-emergence method, showed very good-herbicidal action against BRAPL. AMARE, CHEAL, ECHCG and SETFA.

[1317] At application rates of 125 or 62.5 g/ha (a.s.), the compound I-1a.4 from Example 25, used by the post-emergence method, showed very good herbicidal action against BRAPL. AMARE, CHEAL, ECHCG and SETFA.

[1318] At application rates of 125 or 250 g/ha (a.s.), the compound I-1a.6 from Example 9, used by the post-emergence method, showed very good herbicidal action against BIDPI, CHEAL, POLPE and SETFA.

Claims

1. A pyrazolylbenzazolone of the formula I

2. A benzazolone as claimed in claim 1 where A in the formula I is oxygen or NR6.

3. A benzazolone as claimed in claim 1 where A in the formula I is sulfur or SO2.

4. A benzazolone as claimed in any of the preceding claims where R1 in the formula I is selected from the group consisting of C1-C4-alkyl, halogen and C1-C4-alkoxy.

5. A benzazolone as claimed in any of the preceding claims where R2 is different from hydrogen.

6. A benzazolone as claimed in any of the preceding claims where R2 in the formula I is a heterocycle selected from the group consisting of 4,5-dihydroisoxazol-3-yl, 4,5-dihydroisoxazol-4-yl, isoxazol-3-yl, isoxazol-4-yl, 1,3-dioxolan-2-yl, 1,3-dithiolan-2-yl, 1,3-dioxan-2-yl, 1,3-dithian-2-yl, oxazolin-2-yl and oxazolidin-2-yl, where the abovementioned heterocycles may be mono-, di- or trisubstituted by C1-C4-alkyl.

7. A benzazolone as claimed in any of claims 1 to 5, where R2 in the formula I is cyano, C1-C4-alkyl, C3-C6-alkenyl, C1-C4-(halo)alkylcarbonyl, C1-C4-alkoxycarbonyl-C1-C4-alkyl or C1-C4-alkoxycarbonyl.

8. A benzazolone as claimed in any of the preceding claims where R3 in the formula I is hydrogen, C1-C4-alkyl or halogen.

9. A benzazolone as claimed in any of the preceding claims where Pz in the formula I is a radical of the formula IIa where R7 is selected from the group consisting of hydroxyl, OR10 and OSO2R11, where R10 and R11 are as defined in claim 1, R8 and R9 being as defined in claim 1.

10. A benzazolone as claimed in claim 9 where in the formula IIa R7 is hydroxyl, C1-C4-alkyloxy, acetoxy, O—CH2-phenyl, phenylcarbonyloxy, 2-, 3- or 4-fluorophenyl-carbonyloxy, cyclopropylcarbonyloxy, C1-C4-sulfonyloxy, phenylsulfonyloxy or 2-, 3- or 4-methylphenylsulfonyloxy;. R8 is C1-C4-alkyl or cyclopropyl and R9 is hydrogen or C1-C4-alkyl.

11. A benzazolonecarboxylic acid of the formula IVa

12. A composition, comprising at least one pyrazole derivative of the formula I or an agriculturally useful salt of I as claimed in any of claims 1 to 10, and customary auxiliaries.

13. A method for controlling undesirable vegetation, which comprises allowing a herbicidally effective amount of at least one pyrazole derivative of-the formula I or an agriculturally useful salt of I as claimed in any of claims 1 to 10 to act on plants, their habitat and/or on seed.

14. The use of pyrazole derivatives of the formula I or their agriculturally useful salts as claimed in any of claims 1 to 10 as herbicides.