Amide derivative, pest control agent containing the amide derivative, and use of the amide derivative

Abstract

An amide derivative represented by the following Formula (1) is provided as an amide derivative showing a significantly excellent effect for a pest control action.

Description

BACKGROUND OF THE INVENTION

Field of the Invention

The present invention relates to a pest control agent, an amide derivative contained in the pest control agent, and a method for using the amide derivative.

Description of the Related Art

Various amide derivatives are described in the pamphlets of International Publication WO 2005/21488, International Publication WO 2005/73165, International Publication WO 2006/137376, and International Publication WO 2006/137395.

SUMMARY OF THE INVENTION

In the production of, for example, agricultural and horticultural crops, due to causes such as currently-occurring large scale damage due to pests or the like and the propagation of pests having resistance to existing chemicals, there is a demand for a novel agricultural/horticultural pest control agent.

It is an object of the present invention to provide an amide derivative showing a pesticidal effect against a wide range of agricultural/horticultural pests, a pest control agent containing the amide derivative as an active ingredient, and a pest controlling method.

The present inventors have conducted intensive studies to develop a novle pest control agent, and as a result, they have found that the aromatic carboxamide derivative represented by Formula (1) of the present invention is a novel compound unknown in the literature, and it is also a pest control agent, particularly an agricultural/horticultural pest control agent, showing a particularly high efficiency, thereby completing the present invention.

Further, they have also discovered a novel preparation method and a useful intermediate for the preparation of the compound of the present invention. As a result, they have completed the present invention.

That is, the present invention is as follows.

<1> An amide derivative represented by the following Formula (1):

1. An amide derivative represented by the following Formula (1):

Wherein, in Formula (1), A represents a carbon atom, an oxygen atom, a nitrogen atom, an oxidized nitrogen atom, or a sulfur atom. K represents a non-metal atom group necessary for forming a cyclic linking group derived from benzene, pyridine, pyridine-N-oxide, pyrimidine, pyrazine, pyridazine, triazine, pyrrole, pyrazole, imidazole, oxazole, isoxazole, thiazole, isothiazole, furan, thiophene, oxadiazole, thiodiazole, or triazole, in combination with A and two carbon atoms to which A bonds.

X represents a hydrogen atom, a halogen atom, a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C3-C9 cycloalkyl group, a C3-C9 halocycloalkyl group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 haloalkynyl group, a C1-C6 alkoxy group, a C1-C6 haloalkoxy group, a C2-C6 alkenyloxy group, a C2-C6 haloalkenyloxy group, a C2-C6 alkynyloxy group, a C2-C6 haloalkynyloxy group, a C3-C9 cycloalkoxy group, a C3-C9 halocycloalkoxy group, a C1-C6 alkylthio group, a C1-C6 haloalkylthio group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a C1-C6 alkylsulfonyloxy group, a C1-C6 haloalkylsulfonyloxy group, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C3-C7 alkenylcarbonyl group, a C3-C7 haloalkenylcarbonyl group, a C3-C7 alkynylcarbonyl group, a C3-C7 haloalkynylcarbonyl group, a C4-C10 cycloalkylcarbonyl group, a C4-C10 halocycloalkylcarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, arylcarbonyloxy group, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a C4-C10 cycloalkyloxycarbonyl group, a C4-C10 halocycloalkyloxycarbonyl group, a C2-C7 alkylcarbonylamino group, a C2-C7 haloalkylcarbonylamino group, a C2-C7 alkoxycarbonylamino group, a C2-C7 haloalkoxycarbonylamino group, a C2-C7 alkoxycarbonyloxy group, a C2-C7 haloalkoxycarbonyloxy group, an arylcarbonylamino group, an amino group, a carbamoyl group, a cyano group, a hydroxy group, pentafluorosulfanyl group, a C1-C6 alkylamino group, a C1-C6 haloalkylamino group, a C2-C6 alkenylamino group, a C2-C6 haloalkenylamino group, a C2-C6 alkynylamino group, a C2-C6 haloalkynylamino group, a C3-C9 cycloalkylamino group, a C3-C9 halocycloalkylamino group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C3-C7 alkenylaminocarbonyl group, a C3-C7 haloalkenylaminocarbonyl group, a C3-C7 alkypylaminocarbonyl group, a C3-C7 haloalkynylaminocarbonyl group, a C4-C10 cycloalkylaminocarbonyl group, a C4-C10 halocycloalkylaminocarbonyl group, a phenyl group, or a heterocyclic group, and when there are plural X's, each X may be the same as or different from an other.

n represents an integer of from 0 to 4.

T represents —C(=G₁)-Q₁ or —C(=G₁)-G₂Q₂.

G₁ and G₂ each independently represent an oxygen atom or a sulfur atom,

Q₁ and Q₂ each represent a hydrogen atom, a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 haloalkynyl group, a C3-C9 cycloalkyl group, a C3-C9 halocycloalkyl group, a benzyl group, a phenyl group which may have a substituent, a naphthyl group, or a heterocyclic group which may have a substituent.

Y₁ and Y₅ each independently represent a halogen atom, a C1-C6 haloalkoxy group, or a C1-C3 haloalkyl group, Y₂ and Y₄ each independently represent a hydrogen atom, a halogen atom, or a C1-C4 alkyl group, Y₃ represents a C2-C5 haloalkyl group.

Wherein in Q₁ and Q₂, the substituent of a phenyl group which may have a substituent and a heterocyclic group which may have a substituent represents one or more substituent selected from a group consisting of a halogen atom, a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C3-C9 cycloalkyl group, a C3-C9 halocycloalkyl group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 haloalkynyl group, a C1-C6 alkoxy group, a C1-C6 haloalkoxy group, a C2-C6 alkenyloxy group, a C2-C6 haloalkenyloxy group, a C2-C6 alkynyloxy group, a C2-C6 haloalkynyloxy group, a C3-C9 cycloalkoxy group, a C3-C9 halocycloalkoxy group, a C1-C6 alkylthio group, a C1-C6 haloalkylthio group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C3-C7 alkenylcarbonyl group, a C3-C7 haloalkenylcarbonyl group, a C3-C7 alkynylcarbonyl group, a C3-C7 haloalkynylcarbonyl group, a C4-C10 cycloalkylcarbonyl group, a C4-C10 halocycloalkylcarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a C1-C6 alkylsulfonyloxy group, a C1-C6 haloalkylsulfonyloxy group, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a C4-C10 cycloalkyloxycarbonyl group, a C4-C10 halocycloalkyloxycarbonyl group, a C2-C7 alkylcarbonylamino group, a C2-C7 haloalkylcarbonylamino group, a C2-C7 alkoxycarbonylamino group, a C2-C7 haloalkoxycarbonylamino group, a C1-C6 alkylamino group, a C1-C6 haloalkylamino group, a C2-C6 alkenylamino group, a C2-C6 haloalkenylamino group, a C2-C6 alkynylamino group, a C2-C6 haloalkynylamino group, a C3-C9 cycloalkylamino group, a C3-C9 halocycloalkylamino group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C3-C7 alkenylaminocarbonyl group, a C3-C7 haloalkenylaminocarbonyl group, a C3-C7 alkynylaminocarbonyl group, a C3-C7 haloalkynylaminocarbonyl group, a C4-C10 cycloalkylaminocarbonyl group, a C4-C10 halocycloalkylaminocarbonyl group, an amino group, a carbamoyl group, a cyano group, a nitro group, a hydroxy group, pentafluorosulfanyl group, a phenyl group which may have a substituent, and a heterocyclic group which may have a substituent, and when there are two or more substituents, the substituents may be the same as or different from each other.

Wherein the heterocyclic group in X, Q₁, and Q₂ represent a pyridyl group, a pyridine-N-oxide group, a pyrimidinyl group, a pyrazinyl group, a pyridazyl group, a furyl group, a thienyl group, an oxazolyl group, an isoxazolyl group, an oxadiazolyl group, a thiazolyl group, an isothiazolyl group, a thiadiazolyl group, a pyrrolyl group, an imidazolyl group, a triazolyl group, a pyrazolyl group, or a tetrazolyl group.

G₃ represents an oxygen atom or a sulfur atom.

R₁ and R₂ each independently represent a hydrogen atom, an oxygen atom, a halogen atom, a hydroxy group, a nitro group, a nitroso group, a trimethylsilyl group, a t-butyldimethylsilyl group, a cyano group, an amino group, a C1-C6 alkyl group which may have a substituent, a C1-C6 haloalkyl group which may have a substituent, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C6 alkenyl group which may have a substituent, a C2-C6 haloalkenyl group which may have a substituent, a C2-C6 alkynyl group which may have a substituent, a C2-C6 haloalkynyl group which may have a substituent, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a phenoxycarbonyl group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a benzoyl group, a C1-C6 alkoxy group, a C1-C6 haloalkoxy group, a C1-C6 alkylthio group, a C1-C6 haloalkylthio group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a benzenesulfonyl group, a benzylsulfonyl group, a benzyl group, or —C(═O)C(═O)R₇, wherein R₇ represents a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C1-C6 alkoxy group, or a C1-C6 haloalkoxy group.

However the amide derivative represented by Formula (1) is not one of (A) to (I).

(A) A case where, in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyridine in combination with A and two carbon atoms to which A bonds, Y₁ represents a halogen atom, and Y₅ represents a C1-C6 haloalkoxy group, and T is —C(=G₁)-Q₁.

(B) A case where, in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyrrole, pyrazole, imidazole, oxazole, isoxazole, thiazole, isothiazole, furan, thiophene, oxadiazole, thiodiazole, or triazole, in combination with A and two carbon atoms to which A bonds, Y₁ and Y₅ represent each independently a halogen atom, and T is —C(=G₁)-G₂Q₂.

(C) A case where, in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyrrole, pyrazole, imidazole, oxazole, isoxazole, thiazole, isothiazole, furan, thiophene, oxadiazole, thiodiazole, or triazole, in combination with A and two carbon atoms to which A bonds, T represents —C(=G₁)-Q₁, Y₁ is a halogen atom, and Y₅ represents a halogen atom or a haloalkoxy group.

(D) A case where, the amide derivative is an amide compound represented by the following Formula (2):

Wherein in Formula (2), Y₂ to Y₄, Q₁, G₁, G₃, R₁, and R₂ have the same definitions as Y₂ to Y₄, Q₁, G₁, G₃, R₁, and R₂, respectively, in Formula (1), Y₁ represents a halogen atom, and Y₅ represents a C1-C2 haloalkoxy group.

(E) A case where, in Formula (2), Y₁ and Y₅ each independently represent a halogen atom, all X's represent hydrogen atoms, and Y₃ represents a C2-C3 haloalkyl group.

(F) A case where, the amide derivative is an amide derivative represented by the following Formula (3)

Wherein in Formula (3), Y₁ and Y₅ each independently represent a halogen atom, X₁ and X₃ each independently represent a hydrogen atom or a fluorine atom, Q₁ has the same definition as Q₁ in Formula (1), R₁ represents a hydrogen atom or a methyl group, and Y₃ represents a C3-C4 perfluoroalkyl group.

(G) A case where the amide derivative is an amide derivative represented by the following Formula (4):

Wherein in Formula (4), X₁ represents a fluorine atom, X₂, X₃, and X₄ represent hydrogen atoms, Y₁ and Y₅ are different from each other and represent a bromine atom or a trifluoromethoxy group, Y₂ and Y₄ represent hydrogen atoms, Y₃ represents a heptafluoroisopropyl group, Q₁ represents a phenyl group or a 2-chloropyridin-3-yl group, and R₁ and R₂ are different from each other, and each represent a hydrogen atom or a methyl group.

Alternatively, X₁ represents a fluorine atom, X₂, X₃, and X₄ represent hydrogen atoms, Y₁ and Y₅ represent bromine atoms, Y₂ and Y₄ represent hydrogen atoms, Y₃ represents a pentafluoroethyl group, Q₁ represents a 2-fluorophenyl group, and R₁ and R₂ each independently represent a hydrogen atom or a methyl group}.

(H) A case where, the amide derivative is an amide derivative represented by the following Formula (5):

Wherein, in Formula (5), Y₁ and Y₅ each independently represent a halogen atom, X₁ represents a hydrogen atom or a fluorine atom, Q₂ represents a 2,2,2-trichloroethyl group or a 3,3,3-trifluoro-n-propyl group, and Y₃ represents a C2-C4 haloalkyl group.

(I) A case where the amide derivative is an amide derivative represented by the following Formula (6):

Wherein, in Formula (6), Y₁ and Y₅ each independently represent a halogen atom, Q₂ has the same definition as Q₂ in Formula (1), R₁ represents a hydrogen atom or a methyl group, and Y₃ represents a C3-C4 haloalkyl group.

<2> The amide compound according to <1>, which is represented by the following Formula (7):

Wherein, in Formula (7), n represents 4, and X, Y₁ to Y₅, Q₁, G₁, G₃, R₁, and R₂ have the same definitions as X, Y₁ to Y₅, Q₁, G₁, G₃, R₁, and R₂, respectively, in Formula (1).

<3> The amide derivative according to <2>, which is represented by the following Formula (8):

Wherein, in Formula (8), Q₁ represents a phenyl group which may have a substituent or a pyridyl group which may have a substituent.

X₁, X₂, X₃, and X₄ each independently represent a hydrogen atom or a fluorine atom.

R₁ and R₂ each independently represent a hydrogen atom or a C1-C3 alkyl group.

Y₁ and Y₅ each independently represent a halogen atom, a C1-C3 haloalkoxy group, or a C1-C3 haloalkyl group, Y₂ and Y₄ each independently represent a hydrogen atom, a halogen atom, or a C1-C4 alkyl group, and Y₃ represents a C3-C4 haloalkyl group.

In a case where Y₁ and Y₅ represent halogen atoms simultaneously, at least one of X₁ and X₂ represents a fluorine atom. Further, in a case where Y₁ or Y₅ represents a C1-C3 haloalkoxy group, X₂ represents a fluorine atom.

<4> The amide derivative according to <3>, wherein in Formula (8), Y₃ represents a C3-C4 perfluoroalkyl group.

<5> The amide derivative according to <4>, wherein in Formula (8), Y₁ and Y₅ each independently represent a chlorine atom, a bromine atom, an iodine atom, a trifluoromethoxy group, a trifluoromethyl group, or a pentafluoroethyl group, and Y₂ and Y₄ represent hydrogen atoms.

<6> The amide derivative according to <5>, wherein in Formula (8), X₁ and X₂ each independently represent a hydrogen atom or a fluorine atom, and X₃ and X₄ represent hydrogen atoms.

<7> The amide derivative according to <6>, wherein in Formula (8), R₁ and R₂ each independently represent a hydrogen atom or a methyl group.

<8> The amide derivative according to claim 7, wherein in Formula (8), Q₁ represents a phenyl group or a pyridyl group which may have a substituent selected from a group consisting of a halogen atom, a C1 haloalkyl group, a nitro group, and a cyano group.

<9> The amide derivative according to claim 8, wherein in Formula (8), the number of the substituents in Q₁ is 1 or 2.

<10> The amide derivative according to <9>, wherein in Formula (8), Q₁ represents a phenyl group, a 2-fluorophenyl group, a 3-fluorophenyl group, a 4-fluorophenyl group, a 2-chlorophenyl group, a 3-chlorophenyl group, a 4-chlorophenyl group, a 2-bromophenyl group, a 3-bromophenyl group, a 4-bromophenyl group, a 2-iodophenyl group, a 3-iodophenyl group, a 4-iodophenyl group, a (2-triofluoromethyl)phenyl group, a (3-triofluoromethyl)phenyl group, a (4-triofluoromethyl)phenyl group, a 2-nitrophenyl group, a 3-nitrophenyl group, a 4-nitrophenyl group, a 2-cyanophenyl group, a 3-cyanophenyl group, a 4-cyanophenyl group, a 2,6-difluorophenyl group, a 3,4-dichlorophenyl group, a 2,4-dichlorophenyl group, a 2-chloro-4-fluorophenyl group, a 2-chloro-4, 5-difluorophenyl group, a 4-bromo-2-chlorophenyl group, a 2-bromo-4-chlorophenyl group, a 2-bromo-4-fluorophenyl group, a 2-chloro-4-nitrophenyl group, a 3, 5-dicyanophenyl group, a 4-cyano-2-fluorophenyl group, a 2-chloro-4-cyanophenyl group, a pyridin-3-yl group, a 2-fluoropyridin-3-yl group, a 2-chloropyridin-3-yl group, a 2-bromopyridin-3-yl group, a 2-iodopyridin-3-yl group, a 2-(trifluoromethyl)pyridin-3-yl group, a 2-nitropyridin-3-yl group, a 2-cyanopyridin-3-yl group, a 6-fluoropyridin-3-yl group, a 6-chloropyridin-3-yl group, a 6-bromopyridin-3-yl group, a 6-iodopyridin-3-yl group, a 6-(trifluoromethyl)pyridin-3-yl group, a 6-nitropyridin-3-yl group, a 6-cyanopyridin-3-yl group, a 5-fluoropyridin-3-yl group, a 5-chloropyridin-3-yl group, a 5-bromopyridin-3-yl group, a 5-iodopyridin-3-yl group, a 5-(trifluoromethyl)pyridin-3-yl group, a 5-nitropyridin-3-yl group, a 5-cyanopyridin-3-yl group, a 4-fluoropyridin-3-yl group, a 4-chloropyridin-3-yl group, a 4-bromopyridin-3-yl group, a 4-iodopyridin-3-yl group, a 4-(trifluoromethyl)pyridin-3-yl group, a 4-nitropyridin-3-yl group, a 4-cyanopyridin-3-yl group, a 2,6-dichloropyridin-3-yl group, a pyridin-3-yl N-oxide group, a pyridin-4-yl group, a 2-chloropyridin-4-yl group, a 3-bromopyridin-4-yl group, a 3,5-dichloropyridin-4-yl group, a 3-(trifluoromethyl)pyridine-4-yl group, a 2,6-dicyanopyridin-4-yl group, a pyridin-4-yl N-oxide group, a pyridin-2-yl group, a 3-chloropyridin-2-yl group, a 4-bromopyridin-2-yl group, a 5-iodopyridin-2-yl group, a 6-chloropyridin-2-yl group, or a 4-cyanopyridin-2-yl group,

<11> The amide derivative according to <10>, wherein the compound represented by Formula (8) is 3-benzamido-N-(2-bromo-6-chloro-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, 2-chloro-N-(3-(2,6-dibromo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)nicotinamide, 3-(4-cyano-N-methylbenzamiido)-N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, 2-chloro-N-(3-(2,6-dibromo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-N-methylnicotinamide, 3-benzamido-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, 3-benzamido-N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamido)benzamide, 6-chloro-N-(3-(2,6-dibromo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-N-methylnicotinamide, 3-(3-cyano-N-methylbenzamido)-N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, N-(2,6-dichloro-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamido)benzamide, 3-(4-cyano-N-methylbenzamido)-N-(2,6-dichloro-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, 2-chloro-N-(3-(2,6-dichloro-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-N-methylnicotinamide, N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamiido)benzamide, 3-(4-cyano-N-methylbenzamido)-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, 3-benzamido-N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide, N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(2-fluorobenzamido)benzamide, N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(4-fluorobenzamido)benzamide, 3-(2,6-difluorobenzamido)-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, N-(2-bromo-6-iodo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamido)benzamide, N-(3-(2-bromo-6-iodo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2-chloro-N-methylnicotinamide,

3-(4-cyanobenzamido)-N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide, 3-(3-cyanobenzamido)-N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide, N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamido)benzamide, 3-(4-cyano-N-methylbenzamido)-N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide, 3-(3-cyano-N-methylbenzamido)-N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide, 6-chloro-N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-N-methylnicotinamide, 3-benzamido-N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide, 3-(3-cyanobenzamido)-N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide, 3-(4-cyanobenzamido)-N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide, N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamido)benzamide, 3-(3-cyano-N-methylbenzamido)-N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide, 3-(4-cyano-N-methylbenzamiido)-N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide, 3-benzamido-N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)benzamide, 2-chloro-N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)nicotinamide, 6-chloro-N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)nicotinamide, 3-cyano-N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)benzamide, 3-(4-cyanobenzamido)-N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)benzamide, N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-2-fluorobenzamide, N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-3-(3-fluorobenzamido)benzamide, N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-3-(4-fluorobenzamido)benzamide,

N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-2,6-difluorobenzamide, N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 2-chloro-N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, 6-chloro-N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, 3-cyano-N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 4-cyano-N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-N-methylbenzamide, N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-2-fluoro-N-methylbenzamide, N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-3-fluoro-N-methylbenzamide, N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-4-fluoro-N-methylbenzamide, N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-2,6-difluoro-N-methylbenzamide, 2-chloro-N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)nicotinamide, 6-chloro-N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)nicotinamide, N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(2-fluorobenzamido)benzamide, N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(3-fluorobenzamido)benzamide, N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(4-fluorobenzamido)benzamide, 3-(2,6-difluorobenzamido)-N-(2,6-d iodo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide, 3-benzamido-N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)benzamide, 6-chloro-N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)nicotinamide, N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-2-fluorobenzamide, 2-chloro-N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)nicotinamide,

N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-3-(3-fluorobenzamido)benzamide, N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-3-(4-fluorobenzamido)benzamide, N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-2,6-difluorobenzamide, 3-cyano-N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)benzamide, 3-(4-cyanobenzamido)-N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)benzamide, 2-chloro-N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-N-methylnicotinamide, 6-chloro-N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-N-methylnicotinamide, N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2-fluoro-N-methylbenzamide, N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(3-fluoro-N-methylbenzamido)benzamide, N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(4-fluoro-N-methylbenzamido)benzamide, N-(3-(2,6-diiodo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2,6-difluoro-N-methylbenzamide, N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 2-chloro-N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, 6-chloro-N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, 3-cyano-N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 4-cyano-N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-N-methylbenzamide, N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-2-fluoro-N-methylbenzamide, N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-3-fluoro-N-methylbenzamide, N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-4-fluoro-N-methylbenzamide, N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)phenyl)-2,6-difluoro-N-methylbenzamide,

2-chloro-N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)nicotinamide, 6-chloro-N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)nicotinamide, N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(2-fluorobenzamido)benzamide, N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(3-fluorobenzamido)benzamide, N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(4-fluorobenzamido)benzamide, N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-3-(2,6-difluorobenzamido)-2-fluorobenzamide, 2-chloro-N-(3-(2,6-diiodo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)nicotinamide, 6-chloro-N-(3-(2,6-diiodo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)nicotinamide, 3-(3-cyanobenzamido)-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, 3-(4-cyanobenzamido)-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(3-fluorobenzamido)benzamide, 2-chloro-N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-N-methylnicotinamide, N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2-fluoro-N-methylbenzamide, N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(3-fluoro-N-methylbenzamido)benzamide, N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(4-fluoro-N-methylbenzamido)benzamide, N-(3-(2,6-dibromo-4-(perfluorobutan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2,6-difluoro-N-methylbenzamide, 3-(3-cyano-N-methylbenzamido)-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, N-(3-(2,6-diiodo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2-fluoro-N-methylbenzamide, N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(3-fluoro-N-methylbenzamido)benzamide, 6-chloro-N-(3-(2,6-diiodo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-N-methylnicotinamide,

N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(4-fluoro-N-methylbenzamido)benzamide, N-(3-(2,6-diiodo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2,6-difluoro-N-methylbenzamide, N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(2-fluorobenzamido)benzamide, N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(3-fluorobenzamido)benzamide, N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(4-fluorobenzamido)benzamide, N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-3-(2,6-difluorobenzamido)-2-fluorobenzamide, 6-chloro-N-3-(2,6-dibromo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)nicotinamide, 3-(3-cyanobenzamido)-N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, 3-(4-cyanobenzamido)-N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, 2-chloro-N-(3-(2,6-diiodo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-N-methylnicotinamide, N-(3-(2,6-dibromo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2-fluoro-N-methylbenzamide, N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(3-fluoro-N-methylbenzamido)benzamide, N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-(4-fluoro-N-methylbenzamido)benzamide, N-(3-(2,6-dibromo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2,6-difluoro-N-methylbenzamide, 3-benzamido-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)phenyl)-2-fluorobenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)phenylcarbamoyl)-2-fluorophenyl)-2-chloronicotinamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)phenyl)-3-(4-cyanobenzamido)-2-fluorobenzamide, 3-benzamido-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-chloronicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-trifluoromethyl)phenylcarbamoyl)phenyl)-2-chloro-N-methylnicotinamide, 3-benzamido-N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-chloro-N-(3-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(3-cyanobenzamido)benzamide,

N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-cyanobenzamido)benzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-3-cyano-N-methylbenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-4-cyano-N-methylbenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-fluoro-N-methylnicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methyl-4-nitrobenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-6-chloro-N-methylnicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-6-cyano-N-methylnicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methyl-3-nitrobenzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-N-methyl-3-(N-methylbenzamido)benzamide, N-(3-((2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)(methyl)carbamoyl)phenyl)-2-chloro-N-methylnicotinamide, 2-bromo-N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, 2-chloro-N-(3-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, N-(3-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-4 cyano-N-methylbenzamide, 3-benzamido-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-fluorobenzamide, N-(5-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-2-chloronicotinamide, N-(3-((2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)(methyl)carbamoyl)phenyl)-2-chloronicotinamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-fluoro-3-(N-methylbenzamiido)benzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-cyano-N-methylbenzamido)-4-fluorobenzamide, N-(5-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-2-chloro-N-methylnicotinamide, 3-benzamido-N-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)benzamide,

2-chloro-N-(3-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, N-methyl-N-(3-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 2-chloro-N-methyl-N-(3-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, 3-benzamido-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-N-methylbenzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(3-cyanobenzamido)-N-methylbenzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-cyanobenzamido)-N-methylbenzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(3-cyano-N-methylbenzamido)-N-methylbenzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-cyano-N-methylbenzamido)-N-methylbenzamide, 2-bromo-N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, 3-benzamido-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluorobenzamide, 2-bromo-N-(3-((2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)(methyl)carbamoyl)phenyl)nicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-2-chloronicotinamide, 3-benzamido-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-chloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-4-cyano-2-fluoro-N-methylbenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-4-cyano-2-fluorobenzamide, 3-cyano-N-(3-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 3-(4-cyanobenzamido)-N-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)benzamide, 3-cyano-N-methyl-N-(3-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 4-cyano-N-methyl-N-(3-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide,

N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-cyanobenzamido)-2-fluorobenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-2-chloro-N-methylnicotinamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-cyano-N-methylbenzamido)-2-fluorobenzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(N-methylbenzamido)benzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(3-cyano-N-methylbenzamido)-2-fluorobenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-chloro-4-cyano-N-methylbenzamide, 3-benzamido-N-methyl-N-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)benzamide, 2-chloro-N-(3-(methyl(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)carbamoyl)phenyl)nicotinamide, 3-(3-cyanobenzamido)-N-methyl-N-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)benzamide, 2-bromo-N-(3-(methyl(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)carbamoyl)phenyl)nicotinamide, 2-bromo-N-(3-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, 2-bromo-N-methyl-N-(3-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, 3-(4-cyanobenzamido)-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 3-cyano-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 2-bromo-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, 4-cyano-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 2-chloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-iodonicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-N-methylnicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-6-fluoro-N-methylnicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-4-cyano-2-fluoro-N-methylbenzamide,

N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-6-chloro-N-methylnicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-3,5-dicyano-N-methylbenzamide, 3-benzamido-2-fluoro-N-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)benzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-3,5-dicyano-N-methylbenzamide, 3-benzamido-2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, 3-benzamido-N-(2-bromo-6-(perfluoroethyl)-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, 3-benzamido-N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluorobenzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-2-chloronicotinamide, N-(2-bromo-6-(perfluoroethyl)-4-(per-fluoropropan-2-yl)phenyl)-3-(4-cyanobenzamido)-2-fluorobenzamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(N-methylbenzamido)benzamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(3-cyano-N-methylbenzamido)-2-fluorobenzamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-cyano-N-methylbenzamido)-2-fluorobenzamide, 2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(N-methylbenzamiido)benzamide, 3-(4-cyano-N-methylbenzamido)-2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 3-benzamido-N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 3-benzamido-2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(N-methylbenzamido)benzamide, 3-(4-cyano-N-methylbenzamido)-2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide,

3-(3-cyano-N-methylbenzamido)-2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 2-fluoro-3-(3-fluoro-N-methylbenzamido)-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-3-(4-fluoro-N-methylbenzamiido)-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2,6-difluoro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 6-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, 3-(3-cyanobenzamido)-2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 3-(4-cyanobenzamido)-2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-3-(2-fluorobenzamido)-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-3-(3-fluorobenzamido)-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-2-fluoro-N-methylbenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-2,6-difluoro-N-methylbenzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(3-fluoro-N-methylbenzamido)benzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(4-fluoro-N-methylbenzamido)benzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-2-chloronicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-6-chloronicotinamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(3-cyanobenzamido)-2-fluorobenzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(2-fluorobenzamido)benzamide, N-(2-bromo--(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(3-fluorobenzamido)benzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(4-fluorobenzamido)benzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-N-methylnicotinamide, 2-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylnicotinamide,

2-fluoro-3-(4-fluorobenzamido)-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 3-(2,6-difluorobenzamido)-2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 6-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropan-2-yl)-6-(rifluoromethyl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-6-chloronicotinamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-fluorobenzamide, N-(2-bromo-4-(perfluowopropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(3-fluorobenzamido)benzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-fluorobenzamido)benzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2,6-difluorobenzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(2,6-difluorobenzamido)-2-fluorobenzamide, 3-fluoro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 3-(4-fluorobenzamido)-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 2,6-difluoro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 6-chloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, 6-chloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, 3-cyano-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 2-fluoro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 3-fluoro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 4-fluoro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-fluoro-N-methylbenzamide,

N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-3-fluoro-N-methylbenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-4-fluoro-N-methylbenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2,6-difluoro-N-methylbenzamide, 2,4-dichloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 3-(2,4-dichlorobenzamido)-2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2,6-difluoro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 3-(2-chloro-4-fluorobenzamido)-2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 3-benzamido-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-cloro-N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, 6-chloro-N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, 3-cyano-N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 3-(4-cyanobenzamido)-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 3-fluoro-N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 3-(4-fluorobenzamido)-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2,6-difluoro-N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 2-chloro-N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, 3-cyano-N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 4-cyano-N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide,

3-fluoro-N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 4-fluoro-N-(3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-N-methylisonicotinamide, 3-((3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)(methyl)carbamoyl)pyridine 1-oxide, 4-((3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)(methyl)carbamoyl)pyridine 1-oxide, 2-chloro-4-fluoro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-chloronicotinamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(3-cyanobenzamido)benzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-fluorobenzamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(3-fluorobenzamido)benzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-6-chloronicotinamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-cyanobenzamido)benzamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-fluorobenzamido)benzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2,6-difluorobenzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-chloro-N-methylnicotinamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-3-cyano-N-methylbenzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-fluoro-N-methylbenzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-3-fluoro-N-methylbenzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-6-chloro-N-methylnicotinamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-4-cyano-N-methylbenzamide,

N-(3-(2-bromo--(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-4-fluoro-N-methylbenzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2,6-difluoro-N-methylbenzamide, 6-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide, 3-(3-cyanobenzamido)-2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 3-(4 cyanobenzamido)-2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-3-(2-fluorobenzamido)-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-3-(3-fluorobenzamido)-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-3-(4-fluorobenzamido)-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 3-(2,6-difluorobenzamido)-2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, N-(3-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-6-chloronicotinamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(3-cyanobenzamido)-2-fluorobenzamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-cyanobenzamido)-2-fluorobenzamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(2-fluorobenzamido)benzamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(3-fluorobenzamido)benzamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(4-fluorobenzamido)benzamide, N-(2-bromo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(2,6-difluorobenzamido)-2-fluorobenzamide, 2-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, 6-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, 3-(3-cyano-N-methylbenzamido)-2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-N-(2-fluoro-3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide,

2-fluoro-3-(3-fluoro-N-methylbenzamido)-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-3-(4-fluoro-N-methylbenzamido)-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-chloro-4,5-difluoro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 2-chloro-4-fluoro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-chloro-4-fluorobenzamide, 2-chloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 3-(2-chlorobenzamido)-2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-chloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-2-chlorobenzamide, 2-chloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-4-nitrobenzamide, N-(2-fluoro-3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylnicotinamide, 3-((2-fluoro-3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)(methyl)carbamoyl)pyridine 1-oxide, 4-bromo-2-chloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 2-bromo-4-chloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoro methyl)phenylcarbamoyl)phenyl)benzamide, 2-bromo-4-fluoro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)benzamide, 2-fluoro-3-(3-fluoro-N-methylbenzamido)-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-N-methylbenzamide, N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-N-methy 1-3-(N-methylbenzamido)benzamide, or N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(N-methylbenzamido)benzamide.

<12> The amide derivative according to <2>, wherein in Formula (7), at least one of X represents a chlorine atom, a bromine atom, an iodine atom, a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C3-C9 cycloalkyl group, a C3-C9 halocycloalkyl group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 haloalkynyl group, a C1-C6 alkoxy group, a C1-C6 haloalkoxy group, a C2-C6 alkenyloxy group, a C2-C6 haloalkenyloxy group, a C2-C6 alkynyloxy group, a C2-C6 haloalkynyloxy group, a C3-C9 cycloalkoxy group, a C3-C9 halocycloalkoxy group, a C1-C6 alkylthio group, a C1-C6 haloalkylthio group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a C1-C6 alkylsulfonyloxy group, a C1-C6 haloalkylsulfonyloxy group, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C3-C7 alkenylcarbonyl group, a C3-C7 haloalkenylcarbonyl group, a C3-C7 alkynylcarbonyl group, a C3-C7 haloalkynylcarbonyl group, a C4-C10 cycloalkylcarbonyl group, a C4-C10 halocycloalkylcarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, arylcarbonyloxy group, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a C4-C10 cycloalkyloxycarbonyl group, a C4-C10 halocycloalkyloxycarbonyl group, a C2-C7 alkylcarbonylamino group, a C2-C7 haloalkylcarbonylamino group, a C2-C7 alkoxycarbonylamino group, a C2-C7 haloalkoxycarbonylamino group, a C2-C7 alkoxycarbonyloxy group, a C2-C7 haloalkoxycarbonyloxy group, an arylcarbonylamino group, an amino group, a carbamoyl group, a cyano group, a hydroxy group, pentafluorosulfanyl group, a C1-C6 alkylamino group, a C1-C6 haloalkylamino group, a C2-C6 alkenylamino group, a C2-C6 haloalkenylamino group, a C2-C6 alkynylamino group, a C2-C6 haloalkynylamino group, a C3-C9 cycloalkylamino group, a C3-C9 halocycloalkylamino group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C3-C7 alkenylaminocarbonyl group, a C3-C7 haloalkenylaminocarbonyl group, a C3-C7 alkynylaminocarbonyl group, a C3-C7 haloalkynylaminocarbonyl group, a C4-C10 cycloalkylaminocarbonyl group, a C4-C10 halocycloalkylaminocarbonyl group, a phenyl group, or a heterocyclic group, and when there are plural X's, each X may be the same as or different from an other. Y₁ represents a halogen atom, a C1-C6 haloalkoxy group, or a C1-C3 haloalkyl group. Y₅ represents a C1-C6 haloalkoxy group, or C1-C3 haloalkyl group.

<13> The amide derivative according to <12>, wherein in Formula (7), Y₃ represents a C2-C4 perfluoroalkyl group.

<14> The amide derivative according to <13>, wherein in Formula (7), Y₁ represents a halogen atom or a C1-C3 haloalkyl group, and Y₅ represents a C1-C3 haloalkyl group.

<15> The amide derivative according to <14>, wherein in Formula (7), Y₂ and Y₄ represent a hydrogen atom.

<16> The amide derivative according to <15>, wherein in Formula (7), X₁ to X₄ each independently represents a hydrogen atom, a halogen atom, or a cyano group.

<17> The amide derivative according to <1>, which is represented by the following Formula (9):

Wherein, in Formula (9), n represents 4, and X, Y₁ to Y₅, Q₂, G₁ to G₃, R₁, and R₂ have the same definitions as X, Y₁ to Y₅, Q₂, G₁ to G₃, R₁, and R₂, respectively, in Formula (1).

<18> The amide derivative according to <17>, wherein in Formula (9), Y₁ represents a halogen atom, a C1-C6 haloalkoxy group, or a C1-C3 haloalkyl group, and Y₅ is a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group.

<19> The amide derivative according to <18>, wherein in Formula (9), Y₃ represents a C2-C4 perfluoroalkyl group.

<20> The amide derivative according to <19>, wherein in Formula (9), Y₁ and Y₅ represent halogen atoms or C1-C3 haloalkyl groups, and either Y₁ or Y₅ represent a C1-C3 haloalkyl group.

<21> The amide derivative according to <20>, wherein in Formula (9), Y₂ and Y₄ represent hydrogen atoms.

<22> The amide derivative according to <21>, wherein in Formula (9), X₁ to X₄ each independently represents a hydrogen atom, a halogen atom, or a cyano group.

<23> The amide derivative according to <1>, wherein in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyridine, pyridine-N-oxide, pyrimidine, pyrazine, pyridazine, triazine, pyrrole, pyrazole, imidazole, oxazole, isoxazole, thiazole, isothiazole, furan, thiophene, oxadiazole, thiodiazole, or triazole, in combination with A and two carbon atoms to which A bonds.

<24> The amide derivative according to <23>, wherein in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyridine, in combination with A and two carbon atoms to which A bonds, and when T is —C(=G₁)-Q₁, Y₁ and Y₅ each independently represents a halogen atom or a C1-C3 haloalkyl group.

<25> The amide derivative according to <23>, wherein in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyrrole, pyrazole, imidazole, oxazole, isoxazole, thiazole, isothiazole, furan, thiophene, oxadiazole, thiodiazole, or trizole, in combination with A and two carbon atoms to which A bonds, and in a case where T represents —C(=G₁)-Q₁, R₁ represents an oxygen atom, a halogen atom, a hydroxy group, a nitro group, a nitroso group, a trimethylsilyl group, a t-butyldimethylsilyl group, a cyano group, an amino group, a C1-C6 alkyl group which may have a substituent, a C1-C6 haloalkyl group which may have a substituent, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C6 alkenyl group which may have a substituent, a C2-C6 haloalkenyl group which may have a substituent, a C2-C6 alkynyl group which may have a substituent, a C2-C6 haloalkynyl group which may have a substituent, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a phenoxycarbonyl group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a benzoyl group, a C1-C6 alkoxy group, a C1-C6 haloalkoxy group, a C1-C6 alkylthio group, a C1-C6 haloalkylthio group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a benzenesulfonyl group, a benzylsulfonyl group, a benzyl group, or —C(═O)C(═O)R₇ (wherein R₇ represents a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C1-C6 alkoxy group, or a C1-C6 haloalkoxy group).

<26> The amide derivative according to <23>, wherein in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyrrole, pyrazole, imidazole, oxazole, isoxazole, thiazole, isothiazole, furan, thiophene, oxadiazole, thiodiazole, or trizole, in combination with A and two carbon atoms to which A bonds, and in a case where T represents —C(=G₁)-Q₁, R₂ represents an oxygen atom, a halogen atom, a hydroxy group, a nitro group, a nitroso group, a trimethylsilyl group, a t-butyldimethylsilyl group, a cyano group, an amino group, a C1-C6 alkyl group which may have a substituent, a C1-C6 haloalkyl group which may have a substituent, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C6 alkenyl group which may have a substituent, a C2-C6 haloalkenyl group which may have a substituent, a C2-C6 alkynyl group which may have a substituent, a C2-C6 haloalkynyl group which may have a substituent, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a phenoxycarbonyl group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a benzoyl group, a C1-C6 alkoxy group, a C1-C6 haloalkoxy group, a C1-C6 alkylthio group, a C1-C6 haloalkylthio group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a benzenesulfonyl group, a benzylsulfonyl group, a benzyl group, or —C(═O)C(═O)R₇ (wherein R₇ represents a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C1-C6 alkoxy group, or a C1-C6 haloalkoxy group).

<27> The amide derivative according to any one of <23> to <26>, wherein in Formula (1), Y₃ represents a C2-C4 perfluoroalkyl group.

<28> The amide derivative according to <27>, wherein in Formula (1), Y₁ and Y₅ each independently represent a halogen atom or a C1-C3 haloalkyl group, and either Y₁ or Y₅ represent a C1-C3 haloalkyl group.

<29> The amide derivative according to <28>, wherein in Formula (1), Y₂ and Y₄ represent hydrogen atoms.

<30> The amide derivative according to <29>, wherein in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyridine, pyridine-N-oxide, pyrrole, thiazole, furan, or thiophene, in combination with A and two carbon atoms to which A bonds.

<31> The amide derivative according to <29>, wherein in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyridine, pyridine-N-oxide, or thiazole, in combination with A and two carbon atoms to which A bonds.

<32> The amide derivative according to <16>, wherein in Formula (7), G₁ and G₃ represent oxygen atoms.

<33> The amide derivative according to <22>, wherein in Formula (9), G₁, G₂, and G₃ represent oxygen atoms.

<34> The amide derivative according to <31>, wherein in Formula (1), G₁, G₂, and G₃ represent oxygen atoms.

<35> A pest control agent comprising at least one amide derivative according to any one of <1> to <34> as an active ingredient.

<36> An agricultural chemical comprising at least one amide derivative according to any one of <1> to <34> as an active ingredient.

<37> A pesticide comprising at least one amide derivative according to any one of <1> to <34> as an active ingredient.

<38> A pest controlling method, comprising applying a chemical agent according to any one of <35> to <37>.

<39> A compound represented by the following Formula (56):

Wherein, wherein Y₅ represents a C1-C3 haloalkyl group, and Y₂, Y₃, and Y₄ represent the same definitions as Y₂, Y₃, and Y₄, respectively, in <1>.

<40> A compound represented by the following Formula (57):

Wherein Y₅ represents a C1-C3 haloalkyl group, and Y₁, Y₂, Y₃, and Y₄ represent the same definitions as Y₁, Y₂, Y₃, and Y₄, respectively, in <1>.

<41> The compound according to <40>, wherein in Formula (57), Y₁ represents a halogen atom.

<42> A method for producing a compound represented by the following Formula (57a) according to <41>, including reacting a compound represented by Formula (56) according to <39> with a halogenating agent:

Wherein Y₅ represents a C1-C3 haloalkyl group, Y₂, Y₃, and Y₄ represent the same definitions as Y₂, Y₃, and Y₄, respectively, in <1>, and Y₁ represents a halogen atom.

<43> A compound represented by the following Formula (60a):

Wherein A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>. In a case where K forms a benzene ring together with A and two carbon atoms to which A bonds and all X's represent hydrogen atoms, Y₅ represents a C1-C3 haloalkyl group. Further, when K forms a benzene ring together with A and two carbon atoms to which A bonds and X's are cyano groups, Y₅ represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group.

<44> A method for producing a compound represented by the following Formula (60a) according to <43>, comprising reacting a compound represented by the following Formula (59) with a compound represented by the following Formula (57b):

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and A, K, X, n, and G₃ have the same definitions as A, K, X, n, and G₃, respectively, in <1>.

Wherein Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

Wherein A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>. In a case where K forms a benzene ring together with A and two carbon atoms to which A bonds and X's represent all hydrogen atoms, Y₅ represents a C1-C3 haloalkyl group. Further, in a case where K forms a benzene ring together with A and two carbon atoms to which A bonds and X represents a cyano group, Y₅ represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group.

<45> A compound represented by the following Formula (61a):

Wherein A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ represent the same definitions as A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>. In a case where K forms a benzene ring together with A and two carbon atoms to which A bonds and all X's represent hydrogen atoms, Y₅ represents a C1-C3 haloalkyl group. Further, when K forms a benzene ring together with A and two carbon atoms to which A bonds and X represents a cyano group, Y₅ represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group.

<46> A method for producing a compound represented by the following Formula (61a) according to <45>, including reacting a compound represented by Formula (60a) according to <43> with a reducing agent:

Wherein A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>. In a case where K forms a benzene ring together with A and two carbon atoms to which A bonds and all X's represent hydrogen atoms, Y₅ represents a C1-C3 haloalkyl group. Further, when K forms a benzene ring together with A and two carbon atoms to which A bonds and X represents a cyano group, Y₅ represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group.

<47> A compound represented by the following Formula (69):

Wherein T, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y have the same definitions as T, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<48> A method for producing a compound represented by the following Formula (69) according to <47>, including reacting a compound represented by the following Formula (61b) with a compound represented by the following Formula (62):

Wherein A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.T-LG  Formula (62)

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, and the like, and T represents the same definition as T in <1>.

Wherein T, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ represent the same definitions as T, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ respectively, in <1>.

<49> A compound represented by the following Formula (51a):

Wherein T, R₁, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as T, R₁, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<50> A method for producing a compound represented by the following Formula (51b), including reacting a compound represented by the following Formula (69) according to <47> with a compound represented by the following Formula (64):

Wherein T, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as T, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.R₁-LG  Formula (64)

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, R₁ represents a trimethylsilyl group, a t-butyldimethylsilyl group, a cyano group, a C1-C6 alkyl group which may have a substituent, a C1-C6 haloalkyl group which may have a substituent, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C6 alkenyl group which may have a substituent, a C2-C6 haloalkenyl group which may have a substituent, a C2-C6 alkynyl group which may have a substituent, a C2-C6 haloalkynyl group which may have a substituent, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a phenoxycarbonyl group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a benzoyl group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a benzenesulfonyl group, a benzylsulfonyl group, a benzyl group, or —C(═O)C(═O)R₇ (wherein R₇ represents a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C1-C6 alkoxy group, or a C1-C6 haloalkoxy group.

Wherein R₁ represents the same definition as R₁ in Formula (64), and T, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as T, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<51> A compound represented by the following Formula (57c):

Wherein Y₅ represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group, R₂ represents an oxygen atom, a halogen atom, a hydroxy group, a nitro group, a nitroso group, a trimethylsilyl group, a t-butyldimethylsilyl group, a cyano group, an amino group, a C1-C6 alkyl group which may have a substituent, a C1-C6 haloalkyl group which may have a substituent, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C6 alkenyl group which may have a substituent, a C2-C6 haloalkenyl group which may have a substituent, a C2-C6 alkynyl group which may have a substituent, a C2-C6 haloalkynyl group which may have a substituent, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a phenoxycarbonyl group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a benzoyl group, a C1-C6 alkoxy group, a C1-C6 haloalkoxy group, a C1-C6 alkylthio group, a C1-C6 haloalkylthio group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a benzenesulfonyl group, a benzylsulfonyl group, a benzyl group, or —C(═O)C(═O)R₇ (wherein R₇ represents a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C1-C6 alkoxy group, or a C1-C6 haloalkoxy group), and Y₁, Y₂, Y₃, and Y₄ have the same definitions as Y₁, Y₂, Y₃, and Y₄, respectively, in <1>.

<52> A method for producing a compound represented by the following Formula (57m), including reacting a compound represented by the following Formula (57k) with a compound represented by the following Formula (66):

Wherein Y₅ represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group, and Y₁, Y₂, Y₃, and Y₄ have the same definitions as Y₁, Y₂, Y₃, and Y₄, respectively, in <1>.R₂-LG  Formula (66)

Wherein, LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, R₂ represents a trimethylsilyl group, a t-butyldimethylsilyl group, a cyano group, a C1-C6 alkyl group which may have a substituent, a C1-C6 haloalkyl group which may have a substituent, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C6 alkenyl group which may have a substituent, a C2-C6 haloalkenyl group which may have a substituent, a C2-C6 alkynyl group which may have a substituent, a C2-C6 haloalkynyl group which may have a substituent, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a phenoxycarbonyl group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a benzoyl group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a benzenesulfonyl group, a benzylsulfonyl group, a benzyl group, or —C(═O)C(═O)R₇, wherein R₇ represents a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C1-C6 alkoxy group, or a C1-C6 haloalkoxy group.

Wherein Y₅ represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group, R₂ represents the same definition as R₂ in Formula (66), and Y₁, Y₂, Y₃, and Y₄ have the same definitions as Y₁, Y₂, Y₃, and Y₄, respectively, in <1>.

<53> A method for producing a compound represented by the following Formula (57n), including reacting a compound represented by the following Formula (57k) according to <52> with an aldehyde:

Wherein Y₅ represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group, and Y₁, Y₂, Y₃, and Y₄ have the same definitions as Y₁, Y₂, Y₃, and Y₄, respectively, in <1>.

Wherein Y₅ represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group, R₂ represents a C1-C6 alkyl group which may have a substituent, a C1-C6 haloalkyl group which may have a substituent, or a benzyl group, and Y₁, Y₂, Y₃, and Y₄ have the same definitions as Y₁, Y₂, Y₃, and Y₄, respectively, in <1>.

<54> A compound represented by the following Formula (60):

Wherein R₂ represents the same definition as R₂ in <51>, and A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<55> A method for producing a compound represented by the following Formula (60e), including reacting a compound represented by the following Formula (60f) with a compound represented by the following Formula (66) according to <52>:

Wherein A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.R₂-LG  Formula (66)

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, R₂ represents a trimethylsilyl group, a t-butyldimethylsilyl group, a cyano group, a C1-C6 alkyl group which may have a substituent, a C1-C6 haloalkyl group which may have a substituent, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C6 alkenyl group which may have a substituent, a C2-C6 haloalkenyl group which may have a substituent, a C2-C6 alkynyl group which may have a substituent, a C2-C6 haloalkynyl group which may have a substituent, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a phenoxycarbonyl group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a benzoyl group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a benzenesulfonyl group, a benzylsulfonyl group, a benzyl group, or —C(═O)C(═O)R₇ (wherein R₇ represents a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C1-C6 alkoxy group, or a C1-C6 haloalkoxy group.

Wherein R₂ has the same definition as R₂ in Formula (66), and A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<56> A method for producing a compound represented by the following Formula (60) according to <54>, including reacting a compound represented by the following Formula (57d) with a compound represented by the following Formula (59) according to <44>:

Wherein R₂ has the same definition as R₂ in <51>, and Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Y₁, Y₂, Y₃, Y₄, and Y₅ respectively, in <1>.

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and A, K, X, n, and G₃ have the same definitions as A, K, X, n, and G₃, respectively, in <1>.

Wherein R₂ has the same definition as R₂ in <51>, and A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<57> A compound represented by the following Formula (61):

Wherein R₂ has the same definition as R₂ in <51>, and A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<58> A method for producing a compound represented by the following Formula (61) according to <57>, including the compound represented by Formula (60) according to <54> in the presence of a reducing agent:

Wherein R₂ has the same definition as R₂ in <51>, and A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<59> A compound represented by the following Formula (63):

Wherein T, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as T, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<60> A method for producing a compound represented by the following Formula (63) according to <59>, including reacting a compound represented by the following Formula (61e) with a compound represented by the following Formula (62) according to <48>:

Wherein R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.T-LG  Formula (62)

(wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and T has the same definition as T in <1>.

Wherein T, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ represent the same definitions as T, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<61> A method for producing a compound represented by the following Formula (1b), including reacting a compound represented by the following Formula (63) according to <59> with a compound represented by the following Formula (64) according to <50>:

Wherein T, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as T, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.R₁-LG  Formula ((64)

Wherein, LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, R₁ represents a trimethylsilyl group, a t-butyldimethylsilyl group, a cyano group, a C1-C6 alkyl group which may have a substituent, a C1-C6 haloalkyl group which may have a substituent, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C6 alkenyl group which may have a substituent, a C2-C6 haloalkenyl group which may have a substituent, a C2-C6 alkynyl group which may have a substituent, a C2-C6 haloalkynyl group which may have a substituent, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a phenoxycarbonyl group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a benzoyl group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a benzenesulfonyl group, a benzylsulfonyl group, a benzyl group, or —C(═O)C(═O)R₇, wherein R₇ represents a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C1-C6 alkoxy group, or a C1-C6 haloalkoxy group.

Wherein R₁ has the same definition as R₁ in Formula (64), and R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<62> A compound represented by the following Formula (65a):

Wherein R₁, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₁, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>. In a case where K forms a benzene ring together with A and two carbon atoms to which A bonds, all X's represent hydrogen atoms, and R₂ represents a hydrogen atom, Y₅ is a C1-C3 haloalkyl group. Further, in a case where K forms a benzene ring together with A and two carbon atoms to which A bonds, X represents a cyano group, and R₁ and R₂ represent hydrogen atoms, and Y₅ represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group.

<63> A method for producing a compound represented by the following Formula (65c), including reacting a compound represented by the following Formula (61e) according to <60> with an aldehyde:

Wherein R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

Wherein R₁ represents a C1-C6 alkyl group which may have a substituent, a C1-C6 haloalkyl group which may have a substituent, or a benzyl group, and R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ represent the same definitions as R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>. In a case where K forms a benzene ring together with A and two carbon atoms to which A bonds, all X's represent hydrogen atoms, and R₂ represents a hydrogen atom, Y₅ represents a C1-C3 haloalkyl group.

<64> A method for producing a compound represented by the following Formula (1), including reacting a compound represented by the following Formula (65b) with a compound represented by the following Formula (62) according to <48>:

Wherein R₁, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₁, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.T-LG  Formula (62)

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and T has the same definition as T in <1>.

<65> A compound represented by the following Formula (68):

Wherein Xa represents a chlorine atom, a bromine atom, or an iodine atom, and R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y have the same definitions as R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <23>.

<66> A method for producing a compound represented by the following Formula (68) according to <65>, including reacting a compound represented by the following Formula (57j) with a compound represented by the following Formula (67):

Wherein R₂, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, Xa represents a chlorine atom, a bromine atom, or an iodine atom, and A, K, X, n, and G₃ have the same definitions as A, K, X, n, and G₃, respectively, in <23>.

Wherein Xa represents a chlorine atom, a bromine atom, or an iodine atom, and R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <23>.

<67> A method for producing a compound represented by the following Formula (65d), including reacting a compound represented by the following Formula (68) according to <65> with an aminating agent:

Wherein Xa represents a chlorine atom, a bromine atom, or an iodine atom, and R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <23>.

Wherein R₁, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₁, R₂, A, K, X, n, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <23>.

<68> A compound represented by the following Formula (70):

Wherein Xb represents a chlorine atom, a bromine atom, or an iodine atom, and R₂, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definition as, respectively, in <1>.

<69> A compound represented by the following Formula (72):

Wherein R₂, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<70> A method for producing a compound represented by the following Formula (72) according to <69>, including reacting a compound represented by Formula (70) according to <68> with a fluorinating agent:

Wherein R₂, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<71> A compound represented by the following Formula (73):

Wherein Xc represents a halogen atom, and R₂, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <1>.

<72> A compound represented by the following Formula (75):

Wherein Y represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group, and R₂, G₃, Y₁, Y₂, Y₃, and Y₄ have the same definitions as R₂, G₃, Y₁, Y₂, Y₃, and Y₄, respectively, in <1>.

<73> A method for producing a compound represented by the following Formula (75) according to <72>, including reacting a compound represented by Formula (73) according to <71>, in which Y₅ is a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group, with a cyanating agent:

Wherein Y₅ represents a C1-C6 haloalkoxy group or a C1-C3 haloalkyl group, R₂, G₃, Y₁, Y₂, Y₃, and Y₄ have the same definitions as R₂, G₃, Y₁, Y₂, Y₃, and Y₄, respectively, in <1>.

<74> A compound represented by the following Formula (56a):

Wherein Y₅ represents a C1-C3 haloalkyl group, and Y₂, Y₃, and Y₄ have the same definitions as Y₂, Y₃, and Y₄, respectively, in <3>.

<75> A compound represented by the following Formula (57e):

Wherein Y₅ represents a C1-C3 haloalkyl group, and Y₁, Y₂, Y₃, and Y₄ have the same definitions as Y₁, Y₂, Y₃, and Y₄ according to <3>.

<76> The compound according to <75>, wherein in Formula (57e), Y₁ is a halogen atom.

<77> A method for producing a compound represented by the following Formula (57f) according to <76>, including reacting a compound represented by Formula (56a) according to <74> with a halogenating agent:

Wherein Y₅ represents a C1-C3 haloalkyl group, Y₂, Y₃, and Y₄ represent the same definitions as Y₂, Y₃, and Y₄, respectively, in <3>, and Y₁ represents a halogen atom.

<78> A compound represented by the following Formula (60b):

Wherein X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>. In a case where X₁, X₂, X₃, and X₄ represent all hydrogen atoms, Y₅ represents a C1-C3 haloalkyl group, and in a case where X₂ represents a cyano group, and X₁, X₃, and X₄ represent hydrogen atoms, Y₅ represents a C1-C3 haloalkoxy group or a C1-C3 haloalkyl group.

<79> A method for producing a compound represented by the following Formula (60b) according to <78>, including reacting a compound represented by the following Formula (59a) with a compound represented by the following Formula (57g):

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and X₁, X₂, X₃, and X₄ have the same definitions as X₁, X₂, X₃, and X₄ in <3>.

Wherein Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

Wherein X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>. In a case where X₁, X₂, X₃, and X₄ represent all hydrogen atoms, Y₅ represents a C1-C3 haloalkyl group, and in a case where X₂ represents a cyano group, and X₁, X₃, and X₄ represent hydrogen atoms, Y₅ represents a C1-C3 haloalkoxy group or a C1-C3 haloalkyl group.

<80> A compound represented by the following Formula (61f):

Wherein X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>. In a case where X₁, X₂, X₃, and X₄ represent all hydrogen atoms, Y₅ represents a C1-C3 haloalkyl group, and in a case where X₂ represents a cyano group, and X₁, X₃, and X₄ represent hydrogen atoms, Y₅ represents a C1-C3 haloalkoxy group or a C1-C3 haloalkyl group.

<81> A method for producing a compound represented by the following Formula (61 f) according to <80>, including reacting a compound represented by a compound represented by Formula (60b) according to <78> in the presence of a reducing agent:

Wherein X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>. In a case where X₁, X₂, X₃, and X₄ represent all hydrogen atoms, Y₅ represents a C1-C3 haloalkyl group, and in a case where X₂ represents a cyano group, and X₁, X₃, and X₄ represent hydrogen atoms, Y represents a C1-C3 haloalkoxy group or a C1-C3 haloalkyl group.

<82> A compound represented by the following Formula (69a):

Wherein Q₁, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Q₁, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<83> A method for producing a compound represented by the following Formula (69a) according to <82>, including reacting a compound represented by the following Formula (61c) with a compound represented by the following Formula (62a):

Wherein X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ represent the same definitions as X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and Q₁ represents the same definition as Q₁ in <3>.

Wherein Q₁, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ represent the same definitions as Q₁, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<84> A compound represented by the following Formula (53a):

Wherein Q₁, R₁, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Q₁, R₁, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<85> A method for producing a compound represented by the following Formula (53b), including reacting a compound represented by the following Formula (69a) according to <82> with a compound represented by the following Formula (64a):

Wherein Q₁, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Q₁, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.R₁-LG  Formula (64a)

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and R₁ represents a C1-C3 alkyl group.

Wherein R₁ has the same definition as R₁ in Formula (64a), and Q₁, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Q₁, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<86> A compound represented by the following Formula (57h):

Wherein Y₅ represents a C1-C3 haloalkoxy group or a C1-C3 haloalkyl group, R₂ represents a C1-C3 alkyl group, and Y₁, Y₂, Y₃, and Y₄ have the same definitions as Y₁, Y₂, Y₃, and Y₄, respectively, in <3>.

<87> A method for producing a compound represented by the following Formula (57h) according to <86>, including reacting a compound represented by the following Formula (57l) with a compound represented by the following Formula (66a):

Wherein Y₅ represents a C1-C3 haloalkoxy group or a C1-C3 haloalkyl group, and Y₁, Y₂, Y₃, and Y₄ have the same definitions as Y₁, Y₂, Y₃, and Y₄, respectively, in <3>.R₂-LG  Formula (66a)

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and R₂ represents a C1-C3 alkyl group.

Wherein Y₅ represents a C1-C3 haloalkoxy group or a C1-C3 haloalkyl group, R₂ represents a C1-C3 alkyl group, and Y₁, Y₂, Y₃, and Y₄ have the same definitions as Y₁, Y₂, Y₃, and Y₄, respectively, in <3>.

<88> A method for producing a compound represented by the following Formula (57h) according to <86>, including reacting a compound represented by the following Formula (57l) according to <87> with an aldehyde:

Wherein Y₅ represents a C1-C3 haloalkoxy group or a C1-C3 haloalkyl group, and Y₁, Y₂, Y₃, and Y₄ have the same definitions as Y₁, Y₂, Y₃, and Y₄, respectively, in <3>.

Wherein Y₅ represents a C1-C3 haloalkoxy group or a C1-C3 haloalkyl group, R₂ represents a C1-C3 alkyl group, and Y₁, Y₂, Y₃, and Y₄ have the same definitions as Y₁, Y₂, Y₃, and Y₄, respectively, in <3>.

<89> A compound represented by the following Formula (60c):

Wherein R₂ represents a C1-C3 alkyl group, and X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<90> A method for producing a compound represented by the following Formula (60c) according to <89>, including reacting a compound represented by the following Formula (60d) with a compound represented by the following Formula (66a) according to <87>:

Wherein X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.R₂-LG  Formula (66a)

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and R₂ represents a C1-C3 alkyl group.

(Wherein R₂ represents a C1-C3 alkyl group, and X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<91> A method for producing a compound represented by the following Formula (60c) according to <89>, including reacting a compound represented by the following Formula (57i) with a compound represented by the following Formula (59a) according to <79>:

Wherein R₂ represents a C1-C3 alkyl group, and Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, X₁, X₂, X₃, and X₄ have the same definitions as X₁, X₂, X₃, and X₄ in <3>.

Wherein R₂ represents a C1-C3 alkyl group, and X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<92> A compound represented by the following Formula (61g):

Wherein R₂ represents a C1-C3 alkyl group, and X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<93> A method for producing a compound represented by the following Formula (61g) according to <92>, including reacting a compound represented by Formula (60c) according to <89> in the presence of a reducing agent:

Wherein R₂ represents a C1-C3 alkyl group, and X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<94> A compound represented by the following Formula (63c):

Wherein Q₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Q₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<95> A method for producing a compound represented by the following Formula (63c) according to <94>, including reacting a compound represented by the following Formula (61d) with a compound represented by the following Formula (62a) according to <83>:

Wherein R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and Q₁ has the same definition as Q₁ in <3>.

Wherein Q₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Q₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<96> A method for producing a compound represented by the following Formula (3a), including reacting a compound represented by the following Formula (63c) according to <94> with a compound represented by the following Formula (64a) according to <85>:

Wherein Q₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Q₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.R₁-LG  Formula (64a)

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and R₁ represents a C1-C3 alkyl group.

Wherein R₁ has the same definition as R₁ in Formula (64a), and Q₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as Q₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<97> A compound represented by the following Formula (65e):

Wherein R₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>. In a case where X₁, X₂, X₃, and X₄, represent all hydrogen atoms, and R₂ represents a hydrogen atom, Y₅ represents a C1-C3 haloalkyl group, and in a case where X₂ represents a cyano group, X₁, X₃, and X₄ represent hydrogen atoms, and R₁ and R₂ represent hydrogen atoms, Y₅ represents a C1-C3 haloalkoxy group or a C1-C3 haloalkyl group.

<98> A method for producing a compound represented by the following Formula (65f), including reacting a compound represented by the following Formula (61d) with an aldehyde:

Wherein R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

Wherein R₁ represents a C1-C3 alkyl group, and R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>. In a case where X₁, X₂, X₃, and X₄ represent all hydrogen atoms, and R₂ represents a hydrogen atom, Y₅ represents a C1-C3 haloalkyl group.

<99> A method for producing a compound represented by the following Formula (3) according to <3>, including reacting a compound represented by the following Formula (65g) with a compound represented by the following Formula (62a) according to <83>:

Wherein R₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₁, R₂, X₁, X₂, X₃, X₄, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

Wherein LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, and Q₁ has the same definition as Q₁ in <3>.

<100> A compound represented by the following Formula (70a):

Wherein Xb represents a chlorine atom, a bromine atom, or an iodine atom, and R₂, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<101> A compound represented by the following Formula (72a):

Wherein R₂, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<102> A method for producing a compound represented by the following Formula (72a) according to <101>, including reacting a compound represented by Formula (70a) according to <100> with a fluorinating agent:

Wherein R₂, Y₁, Y₂, Y₃, Y₄, and Y₅ have the same definitions as R₂, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in <3>.

<103> A composition for controlling a pest comprising as an active ingredient at least one amide derivative represented by the following Formula (A1):

Wherein, in Formula (A1), Q₁ represents a phenyl group or a phenyl group substituted with a halogen atom; X₁ represents a fluorine atom; X₂, X₃, and X₄ are each a hydrogen atom; R₁ represents a hydrogen atom or a C1-C3 alkyl group; R₂ is a hydrogen atom; Y₁ and Y₅ each independently represent a halogen atom or a C1-C3 haloalkyl group; Y₂ and Y₄ each represent a hydrogen atom; and Y₃ represents a heptafluoroisopropyl group.

<104> The composition according to <103>, wherein the pest is an animal parasite.

<105> The composition according to <104>, wherein in Formula (A1), Q₁ represents a phenyl group or a phenyl group substituted with a single fluorine atom; R₁ represents a hydrogen atom or a methyl group; and Y₁ and Y₅ each independently represent a bromine or iodine atom or a trifluoromethyl group.

<106> The composition according to <105>, wherein the amide derivative represented by Formula (A1) is 2-fluoro-3-(N-methylbenzamide)-N-(2-bromo-6-trifluoromethyl-4-(heptafluoropropan-2-yl)phenyl)benzamide, 2-fluoro-3-(4-fluoro-N-methylbenzamide)-N-(2-iodo-6-trifluoromethyl-4-(heptafluoropropan-2-yl)phenyl)benzamide, 2-fluoro-3-(3-fluoro-N-methylbenzamide)-N-(2-iodo-6-trifluoromethyl-4-(heptafluoropropan-2-yl)phenyl)benzamide, 2-fluoro-3-(4-fluorobenzamide)-N-(2-iodo-6-trifluoromethyl-4-(heptafluoropropan-2-yl)phenyl)benzamide, or 2-fluoro-3-(N-methylbenzamide)-N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)benzamide.

<107> A method for exterminating animal parasites, comprising administering to an animal the composition according to <104> to <106>.

<108> The method according to <107>, wherein the animal parasite is an ectoparasite.

<109> The method according to <108>, wherein the ectoparasite is Siphonaptera pests.

<110> The method according to <108>, wherein the ectoparasite is Acarina pests.

According to the present invention, an amide derivative showing a pesticidal effect against a wide range of agricultural/horticultural pests, a pest control agent containing the amide derivative as an active ingredient, and a pest controlling method are provided.

DETAILED DESCRIPTION OF THE INVENTION

An amide compound according to the present invention is represented by the following Formula (1).

In Formula (1), A represents a carbon atom, an oxygen atom, a nitrogen atom, an oxidized nitrogen atom, or a sulfur atom. K represents a non-metal atom group necessary for forming a cyclic linking group derived from benzene, pyridine, pyridine-N-oxide, pyrimidine, pyrazine, pyridazine, triazine, pyrrole, pyrazole, imidazole, oxazole, isoxazole, thiazole, isothiazole, furan, thiophene, oxadiazole, thiodiazole, or triazole, in combination with A and two carbon atoms to which A bonds.

X represents a hydrogen atom, a halogen atom, a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C3-C9 cycloalkyl group, a C3-C9 halocycloalkyl group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 haloalkynyl group, a C1-C6 alkoxy group, a C1-C6 haloalkoxy group, a C1-C6 alkylthio group, a C1-C6 haloalkylthio group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a C1-C6 alkylsulfonyloxy group, a C1-C6 haloalkylsulfonyloxy group, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, arylcarbonyloxy group, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C2-C7 alkylcarbonylamino group, a C2-C7 haloalkylcarbonylamino group, a C2-C7 alkoxycarbonylamino group, a C2-C7 haloalkoxycarbonylamino group, a C2-C7 alkoxycarbonyloxy group, a C2-C7 haloalkoxycarbonyloxy group, an arylcarbonylamino group, an amino group, a carbamoyl group, a cyano group, a hydroxy group, pentafluorosulfanyl group, a C1-C6 alkylamino group, a C1-C6 haloalkylamino group, a C2-C6 alkenylamino group, a C2-C6 haloalkenylamino group, a C2-C6 alkynylamino group, a C2-C6 haloalkynylamino group, a C3-C9 cycloalkylamino group, a C3-C9 halocycloalkylamino group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C3-C7 alkenylaminocarbonyl group, a C3-C7 haloalkenylaminocarbonyl group, a C3-C7 alkynylaminocarbonyl group, a C3-C7 haloalkynylaminocarbonyl group, a C4-C10 cycloalkylaminocarbonyl group, a C4-C10 halocycloalkylaminocarbonyl group, a phenyl group, or a heterocyclic group, and when there are plural X's, each X may be the same as or different from an other.

n represents an integer of from 0 to 4. T represents —C(=G₁)-Q₁ or —C(=G₁)-G₂Q₂. G₁ and G₂ each independently represent an oxygen atom or a sulfur atom, and Q₁ and Q₂ represent a hydrogen atom, a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 haloalkynyl group, a C3-C9 cycloalkyl group, a C3-C9 halocycloalkyl group, a benzyl group, a phenyl group which may have a substituent, a naphthyl group, or a heterocyclic group which may have a substituent.

Y₁ and Y₅ each independently represent a halogen atom, a C1-C6 haloalkoxy group, or a C1-C3 haloalkyl group, Y₂ and Y₄ each independently represent a hydrogen atom, a halogen atom, or a C1-C4 alkyl group, Y₃ represents a C2-C5 haloalkyl group.

Further, in Q₁ and Q₂, the substituent of a phenyl group which may have a substituent and a heterocyclic group which may have a substituent represents one or more substituent selected from a group consisting of a halogen atom, a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C3-C9 cycloalkyl group, a C3-C9 halocycloalkyl group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 haloalkynyl group, a C1-C6 alkoxy group, a C1-C6 haloalkoxy group, a C1-C6 alkylthio group, a C1-C6 haloalkylthio group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a C1-C6 alkylsulfonyloxy group, a C1-C6 haloalkylsulfonyloxy group, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C2-C7 alkylcarbonylamino group, a C2-C7 haloalkylcarbonylamino group, a C2-C7 alkoxycarbonylamino group, a C2-C7 haloalkoxycarbonylamino group, a C1-C6 alkylamino group, a C1-C6 haloalkylamino group, a C2-C6 alkenylamino group, a C2-C6 haloalkenylamino group, a C2-C6 alkynylamino group, a C2-C6 haloalkynylamino group, a C3-C9 cycloalkylamino group, a C3-C9 halocycloalkylamino group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C3-C7 alkenylaminocarbonyl group, a C3-C7 haloalkenylaminocarbonyl group, a C3-C7 alkynylaminocarbonyl group, a C3-C7 haloalkynylaminocarbonyl group, a C4-C10 cycloalkylaminocarbonyl group, a C4-C10 halocycloalkylaminocarbonyl group, an amino group, a carbamoyl group, a cyano group, a nitro group, a hydroxy group, pentafluorosulfanyl group, a phenyl group which may have a substituent, and a heterocyclic group which may have a substituent, and when there are two or more substituents, each substituent may be the same as or different from each other.

Moreover, the heterocyclic group in X, Q₁, and Q₂ represent a pyridyl group, a pyridine-N-oxide group, a pyrimidinyl group, a pyrazinyl group, a pyridazyl group, furyl group, thienyl group, an oxazolyl group, an isoxazolyl group, an oxadiazolyl group, a thiazolyl group, an isothiazolyl group, a thiadiazolyl group, a pyrrolyl group, an imidazolyl group, a triazolyl group, a pyrazolyl group, or a tetrazolyl group.

G₃ represents an oxygen atom or a sulfur atom.

R₁ and R₂ each independently represent a hydrogen atom, an oxygen atom, a halogen atom, a hydroxy group, a nitro group, a nitroso group, a trimethylsilyl group, a t-butyldimethylsilyl group, a cyano group, an amino group, a C1-C6 alkyl group which may have a substituent, a C1-C6 haloalkyl group which may have a substituent, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C6 alkenyl group which may have a substituent, a C2-C6 haloalkenyl group which may have a substituent, a C2-C6 alkynyl group which may have a substituent, a C2-C6 haloalkynyl group which may have a substituent, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C3-C7 alkenyloxycarbonyl group, a C3-C7 haloalkenyloxycarbonyl group, a C3-C7 alkynyloxycarbonyl group, a C3-C7 haloalkynyloxycarbonyl group, a phenoxycarbonyl group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a benzoyl group, a C1-C6 alkoxy group, a C1-C6 haloalkoxy group, a C1-C6 alkylthio group, a C1-C6 haloalkylthio group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a benzenesulfonyl group, a benzylsulfonyl group, a benzyl group, or —C(═O)C(═O)R₇ (wherein R₇ represents a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C1-C6 alkoxy group, or a C1-C6 haloalkoxy group).

However the amide derivative represented by Formula (1) is not one of (A) to (I):

(A) A case where in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyridine in combination with A and two carbon atoms to which A bonds, Y₁ represents a halogen atom, and Y₅ represents a C1-C6 haloalkoxy group, and T is —C(=G₁)-Q₁.

(B) A case where in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyrrole, pyrazole, imidazole, oxazole, isoxazole, thiazole, isothiazole, furan, thiophene, oxadiazole, thiodiazole, or triazole, in combination with A and two carbon atoms to which A bonds, Y₁ and Y₅ represent each independently a halogen atom, and T is —C(=G₁)-G₂Q₂.

(C) A case where in Formula (1), K represents a non-metal atom group necessary for forming a cyclic linking group derived from pyrrole, pyrazole, imidazole, oxazole, isoxazole, thiazole, isothiazole, furan, thiophene, oxadiazole, thiodiazole, or triazole, in combination with A and two carbon atoms to which A bonds, T represents —C(=G₁)-Q₁, Y₁ is a halogen atom, and Y₅ represents a halogen atom or a haloalkoxy group.

(D) A case where the amide derivative is an amide compound represented by the following Formula (2):

In Formula (2), Y₂ to Y₄, Q₁, G₁, G₃, R₁, and R₂ have the same definitions as Y₂ to Y₄, Q₁, G₁, G₃, R₁, and R₂, respectively, in Formula (1), Y₁ represents a halogen atom, and Y₅ represents a C1-C2 haloalkoxy group.

(E) A case where in Formula (2), Y₁ and Y₅ represent halogen atoms, all X's represent hydrogen atoms, and Y₃ represents a C2-C3 haloalkyl group.

(F) A case where the amide derivative is an amide derivative represented by the following Formula (3)

In Formula (3), Y₁ and Y₅ each independently represent a halogen atom, X₁ and X₃ each independently represent a hydrogen atom or a fluorine atom, Q₁ has the same definition as Q₁ in Formula (1), R₁ represents a hydrogen atom or a methyl group, and Y₃ represents a C3-C4 perfluoroalkyl group.

(G) A case where the amide derivative is an amide derivative represented by the following Formula (4):

In Formula (4), X₁ represents a fluorine atom, X₂, X₃, and X₄ represent hydrogen atoms, Y₁ and Y₅ are different from each other and represent a bromine atom or a trifluoromethoxy group, Y₂ and Y₄ represent hydrogen atoms, Y₃ represents a heptafluoroisopropyl group, Q₁ represents a phenyl group or a 2-chloropyridin-3-yl group, and R₁ and R₂ are different from each other, and represent a hydrogen atom or a methyl group.

Alternatively, X₁ represents a fluorine atom, X₂, X₃, and X₄ represent hydrogen atoms, Y₁ and Y₅ represent bromine atoms, Y₂ and Y₄ represent hydrogen atoms, Y₃ represents a pentafluoroethyl group, Q₁ represents a 2-fluorophenyl group, and R₁ and R₂ each independently represent a hydrogen atom or a methyl group.

(H) A case where the amide derivative is an amide derivative represented by the following Formula (5):

In Formula (5), Y₁ and Y₅ each independently represent a halogen atom, X₁ represents a hydrogen atom or a fluorine atom, Q₂ represents a 2,2,2-trichloroethyl group or a 3,3,3-trifluoro-n-propyl group, and Y₃ represents a C2-C4 haloalkyl group.

(I) A case where the amide derivative is an amide derivative represented by the following Formula (6)

In Formula (6), Y₁ and Y₅ each independently represent a halogen atom, Q₂ has the same definition as Q₂ in Formula (1), R₁ represents a hydrogen atom or a methyl group, and Y₃ represents a C3-C4 haloalkyl group

In the aspect of a pest control activity, the amide derivative preferably represented by the following Formula (7), and more preferably represented by the following Formula (8).

In Formula (7), X, n is 4, Y₁ to Y₅, Q₁, G₁, G₃, R₁, and R₂ have the same definitions as X, Y₁ to Y₅, Q₁, G₁, G₃, R₁, and R₂, respectively, in Formula (1).

In Formula (8), Q₁ represents a phenyl group which may have a substituent or a pyridyl group which may have a substituent. X₁, X₂, X₃ and X₄ each independently represent hydrogen atoms or fluorine atoms. R₁ and R₂ each independently represent hydrogen atoms or C1-C3 alkyl groups.

Y₁ and Y₅ each independently represent halogen atoms, C1-C3 haloalkoxyl groups, or C1-C3 haloalkyl groups, Y₂ and Y₄ each independently represent hydrogen atoms, halogen atoms, C1-C4 alkyl groups, and Y₃ represents a C3-C4 haloalkyl group.

In a case where Y₁ and Y₅ represent halogen atoms simultaneously, at least one of X₁ and X₂ represents a fluorine atom. Further, in a case where Y₁ or Y₅ represents a C1-C3 haloalkoxy group, X₂ represents a fluorine atom.

The terms used in the formulae including the Formula (1) and the like according to the present invention, have the same meanings as described below in the definitions.

The “halogen atom” represents a fluorine atom, a chlorine atom, a bromine atom, or an iodine atom.

The expression “Ca-Cb (wherein a and b represent an integer of 1 or more)”, for example, “C1-C3” means the number of carbon atoms of from 1 to 3, the “C2-C6” means the number of carbon atoms of from 2 to 6, and the “C1-C4” means the number of carbon atoms of from 1 to 4.

“n-” means normal, “i-” means iso, “s-” means secondary, and “t-” means tertiary.

The “C1-C3 alkyl group” in the present invention represents, for example, a linear or branched alkyl group having from 1 to 3 carbon atoms such as methyl, ethyl, n-propyl, i-propyl, and the like.

The “C1-C3 haloalkyl group” represents, for example, a linear or branched alkyl group having from 1 to 3 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethyl, pentafluoroethyl, heptafluoro-n-propyl, heptafluoro-i-propyl, 2,2-difluoroethyl, 2,2-dichloroethyl, 2,2,2-trifluoroethyl, 2-fluoroethyl, 2-chloroethyl, 2-bromoethyl, 2-iodoethyl, 2,2,2-trichloroethyl, 2,2,2-tribromoethyl, 1,3-difluoro-2-propyl, 1,3-dichloro-2-propyl, 1-chloro-3-fluoro-2-propyl, 1,1,1-trifluoro-2-propyl, 2,3,3,3-trifluoro-n-propyl, 1,1,1,3,3,3-hexafluoro-2-propyl, 1,1,1,3,3,3-hexafluoro-2-chloro-2-propyl, 1,1,1,3,3,3-hexafluoro-2-bromo-2-propyl, 1,1,2,3,3,3-hexafluoro-2-chloro-n-propyl, 1,1,2,3,3,3-hexafluoro-2-bromo-n-propyl, 1,1,2,3,3,3-hexafluoro-1-bromo-2-propyl, 2,2,3,3,3-pentafluoro-n-propyl, 3-fluoro-n-propyl, 3-chloro-n-propyl, 3-bromo-n-propyl, and the like.

The “C1-C4 alkyl group” represents, for example, a linear or branched alkyl group having from 1 to 4 carbon atoms such as methyl, ethyl, n-propyl, i-propyl, n-butyl, s-butyl, t-butyl, and the like.

The “C1-C3 haloalkoxy group” represents, for example, a linear or branched alkoxy group having from 1 to 3 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethoxy, pentafluoroethoxy, heptafluoro-n-propyloxy, heptafluoro-i-propyloxy, 2,2-difluoroethoxy, 2,2-dichloroethoxy, 2,2,2-trifluoroethoxy, 2-fluoroethoxy, 2-chloroethoxy, 2-bromoethoxy, 2-iodoethoxy, 2,2,2-trichloroethoxy, 2,2,2-tribromoethoxy, 1,3-difluoro-2-propyloxy, 1,3-dichloro-2-propyloxy, 1-chloro-3-fluoro-2-propyloxy, 1,1,1-trifluoro-2-propyloxy, 2,3,3,3-trifluoro-n-propyloxy, 1,1,1,3,3,3-hexafluoro-2-propyloxy, 1,1,1,3,3,3-hexafluoro-2-chloro-2-propyloxy, 1,1,1,3,3,3-hexafluoro-2-bromo-2-propyloxy, 1,1,2,3,3,3-hexafluoro-2-chloro-n-propyloxy, 1,1,2,3,3,3-hexafluoro-2-bromo-n-propyloxy, 1,1,2,3,3,3-hexafluoro-1-bromo-2-propyloxy, 2,2,3,3,3-pentafluoro-n-propyloxy, 3-fluoro-n-propyloxy, 3-chloro-n-propyloxy, 3-bromo-n-propyloxy, and the like.

The “C3-C4 perfluoroalkyl group” represents, for example, a linear or branched alkyl group having from 3 to 4 carbon atoms, that all hydrogen atoms is substituted with fluorine atoms such as perfluoro-n-propyl, perfluoro-i-propyl, perfluoro-n-butyl, perfluoro-i-butyl, perfluoro-s-butyl, perfluoro-t-butyl, and the like.

The “C1 haloalkyl group” represents, for example, a methyl group that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethyl, 1,1-difluoro-1-bromomethyl, and the like.

The “C1-C6 alkyl group” in the present invention represents, for example, a linear or branched alkyl group having from 1 to 6 carbon atoms such as methyl, ethyl, n-propyl, i-propyl, n-butyl, s-butyl, t-butyl, n-pentyl, 2-pentyl, neopentyl, 4-methyl-2-pentyl, n-hexyl, 3-methyl-n-pentyl, and the like.

The “C1-C6 haloalkyl group” represents, for example, a linear or branched alkyl group having from 1 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethyl, pentafluoroethyl, heptafluoro-n-propyl, heptafluoro-i-propyl, 2,2-difluoroethyl, 2,2-dichloroethyl, 2,2,2-trifluoroethyl, 2-fluoroethyl, 2-chloroethyl, 2-bromoethyl, 2-iodoethyl, 2,2,2-trichloroethyl, 2,2,2-tribromoethyl, 1,3-difluoro-2-propyl, 1,3-dichloro-2-propyl, 1-chloro-3-fluoro-2-propyl, 1,1,1-trifluoro-2-propyl, 2,3,3,3-trifluoro-n-propyl, 4,4,4-trifluoro-n-butyl, 1,1,1,3,3,3-hexafluoro-2-propyl, 1,1,1,3,3,3-hexafluoro-2-chloro-2-propyl, 1,1,1,3,3,3-hexafluoro-2-bromo-2-propyl, 1,1,2,3,3,3-hexafluoro-2-chloro-n-propyl, 1,1,2,3,3,3-hexafluoro-2-bromo-n-propyl, 1,1,2,3,3,3-hexafluoro-1-bromo-2-propyl, 2,2,3,3,3-pentafluoro-n-propyl, 3-fluoro-n-propyl, 3-chloro-n-propyl, 3-bromo-n-propyl, 3,3,4,4,4-pentafluoro-2-butyl, nonafluoro-n-butyl, nonafluoro-2-butyl, 5,5,5-trifluoro-n-pentyl, 4,4,5,5,5-pentafluoro-2-pentyl, 3-chloro-n-pentyl, 4-bromo-2-pentyl, and the like.

The “C3-C9 cycloalkyl group” represents, for example, a cycloalkyl group having from 3 to 9 carbon atoms, that has a cyclic structure, such as cyclopropyl, cyclobutyl, cyclopentyl, 2-methylcyclopentyl, 3-methylcyclopentyl, cyclohexyl, 2-methylcyclohexyl, 3-methylcyclohexyl, 4-methylcyclohexyl, and the like.

The “C3-C9 halocycloalkyl group” represents, for example, a cycloalkyl group having 3 to 9 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a cyclic structure, such as, 2,2,3,3-tetrafluorocyclobutyl, 2-chlorocyclohexyl, 4-chlorocyclohexyl, and the like.

The “C2-C6 alkenyl group” represents, for example, an alkenyl group having from 2 to 6 carbon atoms, that has a double bond in the carbon chain, such as vinyl, allyl, 2-butenyl, 3-butenyl, and the like.

The “C2-C6 haloalkenyl group” represents, for example, a linear or branched alkenyl group having from 2 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a double bond in the carbon chain, such as 3,3-difluoro-2-propenyl, 3,3-dichloro-2-propenyl, 3,3-dibromo-2-propenyl, 2,3-dibromo-2-propenyl, 4,4-difluoro-3-butenyl, 3,4,4-tribromo-3-butenyl, and the like.

The “C2-C6 alkynyl group” represents, for example, an alkynyl group having from 2 to 6 carbon atoms, that has a triple bond in the carbon chain, such as propargyl, 1-butyn-3-yl, 1-butyn-3-methyl-3-yl, and the like.

The “C2-C6 haloalkynyl group” represents, for example, a linear or branched alkynyl group having from 2 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a triple bond in the carbon chain, such as fluoroethynyl, chloroethynyl, bromoethynyl, 3,3,3-trifluoro-1-propynyl, 3,3,3-trichloro-1-propynyl, 3,3,3-tribromo-1-propynyl, 4,4,4-trifluoro-1-butynyl, 4,4,4-trichloro-1-butynyl, 4,4,4-tribromo-1-butynyl, and the like.

The “C1-C6 alkoxy group” represents, for example, a linear, branched, or cyclic alkoxy group having from 1 to 6 carbon atoms, such as methoxy, ethoxy, n-propyloxy, i-propyloxy, cyclopropoxy, n-butoxy, s-butoxy, i-butoxy, t-butoxy, n-pentyloxy, i-pentyloxy, n-hexyloxy, cyclohexyloxy, and the like.

The “C1-C6 haloalkoxy group” represents, for example, a linear, branched, or cyclic alkoxy group having from 1 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethoxy, pentafluoroethoxy, 2-chloroethoxy, 2,2,2-trifluoroethoxy, heptafluoro-n-propoxy, heptafluoro-i-propoxy, 1,1,1,3,3,3-hexafluoro-2-propoxy, 3-fluoro-n-propoxy, 1-chlorocyclopropoxy, 2-bromocyclopropoxy, 3,3,4,4,4-pentafluoro-2-butoxy, nonafluoro-n-butoxy, nonafluoro-2-butoxy, 5,5,5-trifluoro-n-pentyloxy, 4,4,5,5,5-pentafluoro-2-pentyloxy, 3-chloro-n-pentyloxy, 4-bromo-2-pentyloxy, 4-chlorobutyloxy, 2-iodo-n-propyloxy, and the like.

The “C1-C6 alkylthio group” represents, for example, a linear, branched, or cyclic alkylthio group having from 1 to 6 carbon atoms, such as methylthio, ethylthio, n-propylthio, i-propylthio, cyclopropylthio, n-butylthio, s-butylthio, i-butylthio, t-butylthio, n-pentylthio, i-pentylthio, n-hexylthio, cyclohexylthio, and the like.

The “C1-C6 haloalkylthio group” represents, for example, a linear, branched, or cyclic alkylthio group having from 1 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethylthio, pentafluoroethylthio, 2-chloroethylthio, 2,2,2-trifluoroethylthio, heptafluoro-n-propylthio, heptafluoro-i-propylthio, 1,1,1,3,3,3-hexafluoro-2-propylthio, 3-fluoro-n-propylthio, 1-chlorocyclopropylthio, 2-bromocyclopropylthio, 3,3,4,4,4-pentafluoro-2-butylthio, nonafluoro-n-butylthio, nonafluoro-2-butylthio, 5,5,5-trifluoro-n-pentylthio, 4,4,5,5,5-pentafluoro-2-pentylthio, 3-chloro-n-pentylthio, 4-bromo-2-pentylthio, 4-chlorobutylthio, 2-iodo-n-propylthio, and the like.

The “C1-C6 alcylsulfinyl group” represents, for example, a linear, branched, or cyclic alkylsulfinyl group having from 1 to 6 carbon atoms, such as methylsulfinyl, ethylsulfinyl, n-propylsulfinyl, i-propylsulfinyl, cyclopropylsulfinyl, n-butylsulfinyl, s-butylsulfinyl, i-butylsulfinyl, t-butylsulfinyl, n-pentylsulfinyl, i-pentylsulfinyl, n-hexylsulfinyl, cyclohexylsulfinyl, and the like.

The “C1-C6 haloalkylsulfinyl group” represents, for example, a linear, branched, or cyclic alkylsulfinyl group having from 1 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethylsulfinyl, pentafluoroethylsulfinyl, 2-chloroethylsulfnyl, 2,2,2-trifluoroethylsulfinyl, heptafluoro-n-propylsulfinyl, heptafluoro-i-propylsulfinyl, 1,1,1,3,3,3-hexafluoro-2-propylsulfinyl, 3-fluoro-n-propylsulfinyl, 1-chlorocyclopropylsulfinyl, 2-bromocyclopropylsulfinyl, 3,3,4,4,4-pentafluoro-2-butylsulfinyl, nonafluoro-n-butylsulfinyl, nonafluoro-2-butylsulfinyl, 5,5,5-trifluoro-n-pentylsulfinyl, 4,4,5,5,5-pentafluoro-2-pentylsulfinyl, 3-chloro-n-pentylsulfinyl, 4-bromo-2-pentylsulfinyl, 4-chlorobutylsulfinyl, 2-iodo-n-propylsulfinyl, and the like.

The “C1-C6 alkylsulfonyl group” represents, for example, a linear, branched, or cyclic alkylsulfonyl group having from 1 to 6 carbon atoms, such as methylsulfonyl, ethylsulfonyl, n-propylsulfonyl, i-propylsulfonyl, cyclopropylsulfonyl, n-butylsulfonyl, s-butylsulfonyl, i-butylsulfonyl, t-butylsulfonyl, n-pentylsulfonyl, i-pentylsulfonyl, n-hexylsulfonyl, cyclohexylsulfonyl, and the like.

The “C1-C6 haloalkylsulfonyl group” represents, for example, a linear, branched, or cyclic alkylsulfonyl group having from 1 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethylsulfonyl, pentafluoroethylsulfonyl, 2-chloroethylsulfonyl, 2,2,2-trifluoroethylsulfonyl, heptafluoro-n-propylsulfonyl, heptafluoro-i-propylsulfonyl, 1,1,1,3,3,3-hexafluoro-2-propylsulfonyl, 3-fluoro-n-propylsulfonyl, 1-chlorocyclopropylsulfonyl, 2-bromocyclopropylsulfonyl, 3,3,4,4,4-pentafluoro-2-butylsulfonyl, nonafluoro-n-butylsulfonyl, nonafluoro-2-butylsulfonyl, 5,5,5-trifluoro-n-pentylsulfonyl, 4,4,5,5,5-pentafluoro-2-pentylsulfonyl, 3-chloro-n-pentylsulfonyl, 4-bromo-2-pentylsulfonyl, 4-chlorobutylsulfonyl, 2-iodo-n-propylsulfonyl, and the like.

The “C1-C6 alkylsulfonyloxy group” represents, for example, a linear, branched, or cyclic alkylsulfonyloxy group having from 1 to 6 carbon atoms, such as methanesulfonyloxy, ethanesulfonyloxy, n-propanesulfonyloxy, i-propanesulfonyloxy, cyclopropanesulfonyloxy, n-butanesulfonyloxy, s-butanesulfonyloxy, i-butanesulfonyloxy, t-butanesulfonyloxy, n-pentanesulfonyloxy, i-pentanesulfonyloxy, n-hexanesulfonyloxy, cyclohexanesulfonyloxy, and the like.

The “C1-C6 haloalkylsulfonyloxy group” represents, for example, a linear, branched, or cyclic alkylsulfonyloxy group having from 1 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethanesulfonyloxy, pentafluoropropanesulfonyloxy, 2-chloropropanesulfonyloxy, 2,2,2-trifluoropropanesulfonyloxy, heptafluoro-n-propanesulfonyloxy, heptafluoro-i-propanesulfonyloxy, 1,1,1,3,3,3-hexafluoro-2-propanesulfonyloxy, 3-fluoro-n-propanesulfonyloxy, 1-chlorocyclopropanesulfonyloxy, 2-bromocyclopropanesulfonyloxy, 3,3,4,4,4-pentafluoro-2-butanesulfonyloxy, nonafluoro-n-butanesulfonyloxy, nonafluoro-2-butanesulfonyloxy, 5,5,5-trifluoro-n-pentanesulfonyloxy, 4,4,5,5,5-pentafluoro-2-pentanesulfonyloxy, 3-chloro-n-pentanesulfonyloxy, 4-bromo-2-pentanesulfonyloxy, 4-chlorobutanesulfonyloxy, 2-iodo-n-propanesulfonyloxy, and the like.

The “C2-C7 alkylcarbonyl group” represents, for example, a linear, branched, or cyclic alkylcarbonyl group having from 2 to 7 carbon atoms, such as acetyl, propionyl, i-propylcarbonyl, cyclopropylcarbonyl, n-butylcarbonyl, s-butylcarbonyl, t-butylcarbonyl, n-pentylcarbonyl, 2-pentylcarbonyl, neopentylcarbonyl, cyclopentylcarbonyl, and the like.

The “C2-C7 haloalkylcarbonyl group” represents, for example, a linear, branched, or cyclic alkylcarbonyl group having from 2 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoroacetyl, pentafluoropropionyl, 2-chloropropionyl, 2,2,2-trifluoropropionyl, heptafluoro-n-propylcarbonyl, heptafluoro-i-propylcarbonyl, 1,1,1,3,3,3-hexafluoro-2-propylcarbonyl, 3-fluoro-n-propylcarbonyl, 1-chlorocyclopropylcarbonyl, 2-bromocyclopropylcarbonyl, 3,3,4,4,4-pentafluoro-2-butylcarbonyl, nonafluoro-n-butylcarbonyl, nonafluoro-2-butylcarbonyl, 5,5,5-trifluoro-n-pentylcarbonyl, 4,4,5,5,5-pentafluoro-2-pentylcarbonyl, 3-chloro-n-pentylcarbonyl, 4-bromo-2-pentylcarbonyl, 4-chlorobutylcarbonyl, 2-iodo-n-propylcarbonyl, and the like.

The “C2-C7 alkylcarbonyloxy group” represents, for example, a linear, branched, or cyclic alkylcarbonyloxy group having from 2 to 7 carbon atoms, such as acetyloxy, propionyloxy, i-propylcarbonyloxy, cyclopropylcarbonyloxy, n-butylcarbonyloxy, s-butylcarbonyloxy, t-butylcarbonyloxy, n-pentylcarbonyloxy, 2-pentylcarbonyloxy, neopentylcarbonyloxy, cyclopentylcarbonyloxy, and the like.

The “C2-C7 haloalkylcarbonyloxy group” represents, for example, a linear, branched, or cyclic alkylcarbonyloxy group having from 2 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoroacetyloxy, pentafluoropropionyloxy, 2-chloropropionyloxy, 2,2,2-trifluoropropionyloxy, heptafluoro-n-propylcarbonyloxy, heptafluoro-i-propylcarbonyloxy, 1,1,1,3,3,3-hexafluoro-2-propylcarbonyloxy, 3-fluoro-n-propylcarbonyloxy, 1-chlorocyclopropylcarbonyloxy, 2-bromocyclopropylcarbonyloxy, 3,3,4,4,4-pentafluoro-2-butylcarbonyloxy, nonafluoro-n-butylcarbonyloxy, nonafluoro-2-butylcarbonyloxy, 5,5,5-trifluoro-n-pentylcarbonyloxy, 4,4,5,5,5-pentafluoro-2-pentylcarbonyloxy, 3-chloro-n-pentylcarbonyloxy, 4-bromo-2-pentylcarbonyloxy, 4-chlorobutylcarbonyloxy, 2-iodo-n-propylcarbonyloxy, and the like.

The “C2-C7 alkoxycarbonyl group” represents, for example, a linear, branched, or cyclic alkoxycarbonyl group having from 2 to 7 carbon atoms, such as methoxycarbonyl, ethoxycarbonyl, isopropoxycarbonyl, cyclopropoxycarbonyl, n-butoxycarbonyl, s-butoxycarbonyl, t-butoxycarbonyl, n-pentyloxycarbonyl, 2-pentyloxycarbonyl, neopentyloxycarbonyl, cyclopentyloxycarbonyl, and the like.

The “C2-C7 haloalkoxycarbonyl group” represents, for example, a linear, branched, or cyclic alkoxycarbonyl group having from 2 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethoxycarbonyl, pentafluoroethoxycarbonyl, 2-chloroethoxycarbonyl, 2,2,2-trifluoroethoxycarbonyl, heptafluoro-n-propoxycarbonyl, heptafluoro-i-propoxycarbonyl, 1,1,1,3,3,3-hexafluoro-2-propoxycarbonyl, 3-fluoro-n-propoxycarbonyl, 1-chlorocyclopropoxycarbonyl, 2-bromocyclopropoxycarbonyl, 3,3,4,4,4-pentafluoro-2-butoxycarbonyl, nonafluoro-n-butoxycarbonyl, nonafluoro-2-butoxycarbonyl, 5,5,5-trifluoro-n-pentyloxycarbonyl, 4,4,5,5,5-pentafluoro-2-pentyloxycarbonyl, 3-chloro-n-pentyloxycarbonyl, 4-bromo-2-pentyloxycarbonyl, 4-chlorobutyloxycarbonyl, 2-iodo-n-propyloxycarbonyl, and the like.

The “C2-C7 alkylcarbonylamino group” represents, for example, a linear, branched, or cyclic alkylcarbonylamino group having from 2 to 7 carbon atoms, such as acetylamino, propionylamino, n-propylcarbonylamino, i-propylcarbonylamino, cyclopropylcarbonylamino, n-butylcarbonylamino, s-butylcarbonylamino, i-butylcarbonylamino, t-butylcarbonylamino, n-pentylcarbonylamino, i-pentylcarbonylamino, n-hexylcarbonylamino, cyclohexylcarbonylamino, and the like.

The “C2-C7 haloalkylcarbonylamino group” represents, for example, a linear, branched, or cyclic alkylcarbonylamino group having from 2 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoroacetylamino, pentafluoropropionylamino, 2-chloropropionylamino, 2,2,2-trifluoropropionylamino, heptafluoro-n-propylcarbonylamino, heptafluoro-i-propylcarbonylamino, 1,1,1,3,3,3-hexafluoro-2-propylcarbonylamino, 3-fluoro-n-propylcarbonylamino, 1-chlorocyclopropylcarbonylamino, 2-bromocyclopropylcarbonylamino, 3,3,4,4,4-pentafluoro-2-butylcarbonylamino, nonafluoro-n-butylcarbonylamino, nonafluoro-2-butylcarbonylamino, 5,5,5-trifluoro-n-pentylcarbonylamino, 4,4,5,5,5-pentafluoro-2-pentylcarbonylamino, 3-chloro-n-pentylcarbonylamino, 4-bromo-2-pentylcarbonylamino, 4-chlorobutylcarbonylamino, 2-iodo-n-propylcarbonylamino, and the like.

The “C2-C7 alkoxycarbonylamino group” represents, for example, a linear, branched, or cyclic alkoxycarbonylamino group having from 2 to 7 carbon atoms, such as methoxycarbonylamino, ethoxycarbonylamino, n-propyloxycarbonylamino, i-propyloxycarbonylamino, cyclopropoxycarbonylamino, n-butoxycarbonylamino, s-butoxycarbonylamino, i-butoxycarbonylamino, t-butoxycarbonylamino, n-pentyloxycarbonylamino, i-pentyloxycarbonylamino, n-hexyloxycarbonylamino, cyclohexyloxycarbonylamino, and the like.

The “C2-C7 haloalkoxycarbonylamino group” represents, for example, a linear, branched, or cyclic alkoxycarbonylamino group having from 2 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethoxycarbonylamino, pentafluoroethoxycarbonylamino, 2-chloroethoxycarbonylamino, 2,2,2-trifluoroethoxycarbonylamino, heptafluoro-n-propoxycarbonylamino, heptafluoro-i-propoxycarbonylamino, 1,1,1,3,3,3-hexafluoro-2-propoxycarbonylamino, 3-fluoro-n-propoxycarbonylamino, 1-chlorocyclopropoxycarbonylamino, 2-bromocyclopropoxycarbonylamino, 3,3,4,4,4-pentafluoro-2-butoxycarbonylamino, nonafluoro-n-butoxycarbonylamino, nonafluoro-2-butoxycarbonylamino, 5,5,5-trifluoro-n-pentyloxycarbonylamino, 4,4,5,5,5-pentafluoro-2-pentyloxycarbonylamino, 3-chloro-n-pentyloxycarbonylamino, 4-bromo-2-pentyloxycarbonylamino, 4-chlorobutyloxycarbonylamino, 2-iodo-n-propyloxycarbonylamino, and the like.

The “C2-C7 alkoxycarbonyloxy group” represents, for example, a linear, branched, or cyclic alkoxycarbonyloxy group having from 2 to 7 carbon atoms, such as methoxycarbonyloxy, ethoxycarbonyloxy, n-propyloxycarbonyloxy, i-propyloxycarbonyloxy, cyclopropoxycarbonyloxy, n-butoxycarbonyloxy, s-butoxycarbonyloxy, i-butoxycarbonyloxy, t-butoxycarbonyloxy, n-pentyloxycarbonyloxy, i-pentyloxycarbonyloxy, n-hexyloxycarbonyloxy, cyclohexyloxycarbonyloxy, and the like.

The “C2-C7 haloalkoxycarbonyloxy group” represents, for example, a linear, branched, or cyclic alkoxycarbonyloxy group having from 2 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethoxycarbonyloxy, pentafluoroethoxycarbonyloxy, 2-chloroethoxycarbonyloxy, 2,2,2-trifluoroethoxycarbonyloxy, heptafluoro-n-propoxycarbonyloxy, heptafluoro-i-propoxycarbonyloxy, 1,1,1,3,3,3-hexafluoro-2-propoxycarbonyloxy, 3-fluoro-n-propoxycarbonyloxy, 1-chlorocyclopropoxycarbonyloxy, 2-bromocyclopropoxycarbonyloxy, 3,3,4,4,4-pentafluoro-2-butoxycarbonyloxy, nonafluoro-n-butoxycarbonyloxy, nonafluoro-2-butoxycarbonyloxy, 5,5,5-trifluoro-n-pentyloxycarbonyloxy, 4,4,5,5,5-pentafluoro-2-pentyloxycarbonyloxy, 3-chloro-n-pentyloxycarbonyloxy, 4-bromo-2-pentyloxycarbonyloxy, 4-chlorobutyloxycarbonyloxy, 2-iodo-n-propyloxycarbonyloxy, and the like.

The “C1-C6 alkylamino group” represents, for example, a linear, branched, or cyclic alkylamino group having from 1 to 6 carbon atoms, such as methylamino, dimethylamino, ethylamino, diethylamino, n-propylamino, i-propylamino, cyclopropylamino, n-butylamino, s-butylamino, i-butylamino, t-butylamino, n-pentylamino, i-pentylamino, n-hexylamino, cyclohexylamino, and the like.

The “C1-C6 haloalkylamino group” represents, for example, a linear, branched, or cyclic alkylamino group having from 1 to 6 carbon atoms substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethylamino, ditrifluoromethylamino, pentafluoroethylamino, dipentafluoroethylamino, 2-chloroethylamino, 2,2,2-trifluoroethylamino, heptafluoro-n-propylamino, heptafluoro-i-propylamino, 1,1,1,3,3,3-hexafluoro-2-propylamino, 3-fluoro-n-propylamino, 1-chlorocyclopropylamino, 2-bromocyclopropylamino, 3,3,4,4,4-pentafluoro-2-butylamino, nonafluoro-n-butylamino, nonafluoro-2-butylamino, 5,5,5-trifluoro-n-pentylamino, 4,4,5,5,5-pentafluoro-2-pentylamino, 3-chloro-n-pentylamino, 4-bromo-2-pentylamino, 4-chlorobutylamino, 2-iodo-n-propylamino, and the like.

The “C2-C6 alkenyloxy group” represents, for example, an alkenyloxy group having from 2 to 6 carbon atoms, that has a double bond in the carbon chain, such as vinyloxy, allyloxy, 2-butenyloxy, 3-butenyloxy, and the like.

The “C2-C6 haloalkenyloxy group” represents, for example, a linear or branched alkenyloxy group having from 2 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a double bond in the carbon chain, such as 3,3-difluoro-2-propenyloxy, 3,3-dichloro-2-propenyloxy, 3,3-dibromo-2-propenyloxy, 2,3-dibromo-2-propenyloxy, 4,4-difluoro-3-butenyloxy, 3,4,4-tribromo-3-butenyloxy, and the like.

The “C2-C6 alkynyloxy group” represents, for example, an alkynyloxy group having from 2 to 6 carbon atoms, that has a triple bond in the carbon chain, such as propargyloxy, 1-butyn-3-yloxy, 1-butyn-3-methyl-3-yloxy, and the like.

The “C2-C6 haloalkynyloxy group” represents, for example, a linear or branched alkynyloxy group having from 2 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a triple bond in the carbon chain, such as fluoroethynyloxy, chloroethynyloxy, bromoethynyloxy, 3,3,3-trifluoro-1-propynyloxy, 3,3,3-trichloro-1-propynyloxy, 3,3,3-tribromo-1-propynyloxy, 4,4,4-trifluoro-1-butynyloxy, 4,4,4-trichloro-1-butynyloxy, 4,4,4-tribromo-1-butynyloxy, and the like.

The “C3-C9 cycloalkoxy group” represents, for example, a cycloalkyloxy group having from 3 to 9 carbon atoms, that has a cyclic structure, such as cyclopropyloxy, cyclobutyloxy, cyclopentyloxy, 2-methylcyclopentyloxy, 3-methylcyclopentyloxy, cyclohexyloxy, 2-methylcyclohexyloxy, 3-methylcyclohexyloxy, 4-methylcyclohexyloxy, and the like.

The “C3-C9 halocycloalkoxy group” represents, for example, a cycloalkyloxy group having from 3 to 9 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a cyclic structure, such as 2,2,3,3-tetrafluorocyclobutyloxy, 2-chlorocyclohexyloxy, 4-chlorocyclohexyloxy, and the like.

The “C3-C7 alkenylcarbonyl group” represents, for example, an alkenylcarbonyl group having from 3 to 7 carbon atoms, that has a double bond in the carbon chain, such as vinylcarbonyl, allylcarbonyl, 2-butenylcarbonyl, 3-butenylcarbonyl, and the like.

The “C3-C7 haloalkenylcarbonyl group” represents an alkenylcarbonyl group having from 3 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a double bond in the carbon chain, such as 3,3-difluoro-2-propenylcarbonyl, 3,3-dichloro-2-propenylcarbonyl, 3,3-dibromo-2-propenylcarbonyl, 2,3-dibromo-2-propenylcarbonyl, 4,4-difluoro-3-butenylcarbonyl, 3,4,4-tribromo-3-butenylcarbonyl, and the like.

The “C3-C7 alkynylcarbonyl group” represents an alkynylcarbonyl group having from 3 to 7 carbon atoms and has a triple bond in the carbon chain, such as propargylcarbonyl, 1-butyn-3-ylcarbonyl, 1-butyn-3-methyl-3-ylcarbonyl, and the like.

The “C3-C7 haloalkynylcarbonyl group” represents, for example, a linear or branched alkynylcarbonyl group having from 3 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a triple bond in the carbon chain, such as fluoroethynylcarbonyl, chloroethynylcarbonyl, bromoethynylcarbonyl, 3,3,3-trifluoro-1-propynylcarbonyl, 3,3,3-trichloro-1-propynylcarbonyl, 3,3,3-tribromo-1-propynylcarbonyl, 4,4,4-trifluoro-1-butynylcarbonyl, 4,4,4-trichloro-1-butynylcarbonyl, 4,4,4-tribromo-1-butynylcarbonyl, and the like.

The “C4-C10 cycloalkylcarbonyl group” represents, for example, a cycloalkylcarbonyl group having from 4 to 10 carbon atoms, that has a cyclic structure, such as cyclopropylcarbonyl, cyclobutylcarbonyl, cyclopentylcarbonyl, 2-methylcyclopentylcarbonyl, 3-methylcyclopentylcarbonyl, cyclohexylcarbonyl, 2-methylcyclohexylcarbonyl, 3-methylcyclohexylcarbonyl, 4-methylcyclohexylcarbonyl, and the like.

The “C4-C10 halocycloalkylcarbonyl group” represents, for example, a cycloalkylcarbonyl group having from 4 to 10 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a cyclic structure, such as 2,2,3,3-tetrafluorocyclobutylcarbonyl, 2-chlorocyclohexylcarbonyl, 4-chlorocyclohexylcarbonyl, and the like.

The “C3-C7 alkenyloxycarbonyl group” represents an alkenyloxycarbonyl group having 3 to 7 carbon atoms, that has a double bond in the carbon chain, such as vinyloxycarbonyl, allyloxycarbonyl, 2-butenyloxycarbonyl, 3-butenyloxycarbonyl, and the like.

The “C3-C7 haloalkenyloxycarbonyl group” represents, for example, a linear or branched alkenyloxycarbonyl group having from 3 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a double bond in the carbon chain, such as 3,3-difluoro-2-propenyloxycarbonyl, 3,3-dichloro-2-propenyloxycarbonyl, 3,3-dibromo-2-propenyloxycarbonyl, 2,3-dibromo-2-propenyloxycarbonyl, 4,4-difluoro-3-butenyloxycarbonyl, 3,4,4-tribromo-3-butenyloxycarbonyl, and the like.

The “C3-C7 alkynyloxycarbonyl group” represents, for example, an alkynyloxycarbonyl group having from 3 to 7 carbon atoms, that has a triple bond in the carbon chain, such as propargyloxycarbonyl, 1-butyn-3-yloxycarbonyl, 1-butyn-3-methyl-3-yloxycarbonyl, and the like.

The “C3-C7 haloalkynyloxycarbonyl group” represents, for example, a linear or branched alkynyloxycarbonyl group having from 3 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a triple bond in the carbon chain, such as fluoroethynyloxycarbonyl, chloroethynyloxycarbonyl, bromoethynyloxycarbonyl, 3,3,3-trifluoro-1-propynyloxycarbonyl, 3,3,3-trichloro-1-propynyloxycarbonyl, 3,3,3-tribromo-1-propynyloxycarbonyl, 4,4,4-trifluoro-1-butynyloxycarbonyl, 4,4,4-trichloro-1-butynyloxycarbonyl, 4,4,4-tribromo-1-butynyloxycarbonyl, and the like.

The “C4-C10 cycloalkyloxycarbonyl group” represents, for example, a cycloalkyloxycarbonyl group having from 4 to 10 carbon atoms, that has a cyclic structure, such as cyclopropyloxycarbonyl, cyclobutyloxycarbonyl, cyclopentyloxycarbonyl, 2-methylcyclopentyloxycarbonyl, 3-methylcyclopentyloxycarbonyl, cyclohexyloxycarbonyl, 2-methylcyclohexyloxycarbonyl, 3-methylcyclohexyloxycarbonyl, 4-methylcyclohexyloxycarbonyl, and the like.

The “C4-C10 halocycloalkyloxycarbonyl group” represents, for example, a cycloalkyloxycarbonyl group having from 4 to 10 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a cyclic structure, such as 2,2,3,3-tetrafluorocyclobutyloxycarbonyl, 2-chlorocyclohexyloxycarbonyl, 4-chlorocyclohexyloxycarbonyl, and the like.

The “C2-C6 alkenylamino group” represents, for example, an alkenylamino group having 2 to 6 carbon atoms, that has a double bond in the carbon chain, such as vinylamino, allylamino, 2-butenylamino, 3-butenylamino, and the like.

The “C2-C6 haloalkenylamino group” represents a linear or branched alkenylamino group having from 2 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a double bond in the carbon chain, such as 3,3-difluoro-2-propenylamino, 3,3-dichloro-2-propenylamino, 3,3-dibromo-2-propenylamino, 2,3-dibromo-2-propenylamino, 4,4-difluoro-3-butenylamino, 3,4,4-tribromo-3-butenylamino, and the like.

The “C2-C6 alkynylamino group” represents, for example, an alkynylamino group having from 2 to 6 carbon atoms, that has a triple bond in the carbon chain, such as propargylamino, 1-butyn-3-ylamino, 1-butyn-3-methyl-3-ylamino, and the like.

The “C2-C6 haloalkynylamino group” represents, for example, a linear or branched alkynylamino group having from 2 to 6 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a triple bond in the carbon chain, such as fluoroethynylamino, chloroethynylamino, bromoethynylamino, 3,3,3-trifluoro-1-propynylamino, 3,3,3-trichloro-1-propynylamino, 3,3,3-tribromo-1-propynylamino, 4,4,4-trifluoro-1-butynylamino, 4,4,4-trichloro-1-butynylamino, 4,4,4-tribromo-1-butynylamino, and the like.

The “C3-C9 cycloalkylamino group” represents, for example, a cycloalkyl group amino having from 3 to 9 carbon atoms, that has a cyclic structure, such as cyclopropylamino, cyclobutylamino, cyclopentylamino, 2-methylcyclopentylamino, 3-methylcyclopentylamino, cyclohexylamino, 2-methylcyclohexylamino, 3-methylcyclohexylamino, 4-methylcyclohexylamino, and the like.

The “C3-C9 halocycloalkylamino group” represents, for example, a cycloalkylamino group having from 3 to 9 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a cyclic structure, such as 2,2,3,3-tetrafluorocyclobutylamino, 2-chlorocyclohexylamino, 4-chlorocyclohexylamino, and the like.

The “C2-C7 alkylaminocarbonyl group” represents, for example, a linear or branched alkylaminocarbonyl group having from 2 to 7 carbon atoms, such as methylaminocarbonyl, ethylaminocarbonyl, n-propylaminocarbonyl, i-propylaminocarbonyl, n-butylaminocarbonyl, s-butylaminocarbonyl, t-butylaminocarbonyl, n-pentylaminocarbonyl, 2-pentylaminocarbonyl, neopentylaminocarbonyl, 4-methyl-2-pentylaminocarbonyl, n-hexylaminocarbonyl, 3-methyl-n-pentylaminocarbonyl, and the like.

The “C2-C7 haloalkylaminocarbonyl group” represents, for example, a linear or branched alkylaminocarbonyl group having from 2 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethylaminocarbonyl, pentafluoroethylaminocarbonyl, heptafluoro-n-propylaminocarbonyl, heptafluoro-i-propylaminocarbonyl, 2,2-difluoroethylaminocarbonyl, 2,2-dichloroethylaminocarbonyl, 2,2,2-trifluoroethylaminocarbonyl, 2-fluoroethylaminocarbonyl, 2-chloroethylaminocarbonyl, 2-bromoethylaminocarbonyl, 2-iodoethylaminocarbonyl, 2,2,2-trichloroethylaminocarbonyl, 2,2,2-tribromoethylaminocarbonyl, 1,3-difluoro-2-propylaminocarbonyl, 1,3-dichloro-2-propylaminocarbonyl, 1-chloro-3-fluoro-2-propylaminocarbonyl, 1,1,1-trifluoro-2-propylaminocarbonyl, 2,3,3,3-trifluoro-n-propylaminocarbonyl, 4,4,4-trifluoro-n-butylaminocarbonyl, 1,1,1,3,3,3-hexafluoro-2-propylaminocarbonyl, 1,1,1,3,3,3-hexafluoro-2-chloro-2-propylaminocarbonyl, 1,1,1,3,3,3-hexafluoro-2-bromo-2-propylaminocarbonyl, 1,1,2,3,3,3-hexafluoro-2-chloro-n-propylaminocarbonyl, 1,1,2,3,3,3-hexafluoro-2-bromo-n-propylaminocarbonyl, 1,1,2,3,3,3-hexafluoro-1-bromo-2-propylaminocarbonyl, 2,2,3,3,3-pentafluoro-n-propylaminocarbonyl, 3-fluoro-n-propylaminocarbonyl, 3-chloro-n-propylaminocarbonyl, 3-bromo-n-propylaminocarbonyl, 3,3,4,4,4-pentafluoro-2-butylaminocarbonyl, nonafluoro-n-butylaminocarbonyl, nonafluoro-2-butylaminocarbonyl, 5,5,5-trifluoro-n-pentylaminocarbonyl, 4,4,5,5,5-pentafluoro-2-pentylaminocarbonyl, 3-chloro-n-pentylaminocarbonyl, 4-bromo-2-pentylaminocarbonyl, and the like.

The “C3-C7 alkenylaminocarbonyl group” represents, for example, an alkenylaminocarbonyl group having from 3 to 7 carbon atoms, that has a double bond in the carbon chain, such as vinylaminocarbonyl, allylaminocarbonyl, 2-butenylaminocarbonyl, 3-butenylaminocarbonyl, and the like.

The “C3-C7 haloalkenylaminocarbonyl group” represents, for example, a linear or branched alkenylaminocarbonyl group having from 3 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a double bond in the carbon chain, such as 3,3-difluoro-2-propenylaminocarbonyl, 3,3-dichloro-2-propenylaminocarbonyl, 3,3-dibromo-2-propenylaminocarbonyl, 2,3-dibromo-2-propenylaminocarbonyl, 4,4-difluoro-3-butenylaminocarbonyl, 3,4,4-tribromo-3-butenylaminocarbonyl, and the like.

The “C3-C7 alkynylaminocarbonyl group” represents, for example, an alkynylaminocarbonyl group having from 3 to 7 carbon atoms, that has a triple bond in the carbon chain, such as propargylaminocarbonyl, 1-butyn-3-ylaminocarbonyl, 1-butyn-3-methyl-3-ylaminocarbonyl, and the like.

The “C3-C7 haloalkynylaminocarbonyl group” represents, for example, a linear or branched alkynylaminocarbonyl group having from 3 to 7 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other and has a triple bond in the carbon chain, such as fluoroethynylaminocarbonyl, chloroethynylaminocarbonyl, bromoethynylaminocarbonyl, 3,3,3-trifluoro-1-propynylaminocarbonyl, 3,3,3-trichloro-1-propynylaminocarbonyl, 3,3,3-tribromo-1-propynylaminocarbonyl, 4,4,4-trifluoro-1-butynylaminocarbonyl, 4,4,4-trichloro-1-butynylaminocarbonyl, 4,4,4-tribromo-1-butynylaminocarbonyl, and the like.

The “C4-C10 cycloalkylaminocarbonyl group” represents, for example, a cycloalkylaminocarbonyl group having from 4 to 10 carbon atoms, that has a cyclic structure, such as cyclopropylaminocarbonyl, cyclobutylaminocarbonyl, cyclopentylaminocarbonyl, 2-methylcyclopentylaminocarbonyl, 3-methylcyclopentylaminocarbonyl, cyclohexylaminocarbonyl, 2-methylcyclohexylaminocarbonyl, 3-methylcyclohexylaminocarbonyl, 4-methylcyclohexylaminocarbonyl, and the like.

The “C4-C10 halocycloalkylaminocarbonyl group” represents, for example, a cycloalkylaminocarbonyl group having from 4 to 10 carbon atoms that is substituted with one or more halogen atoms which may be the same as or different from each other and has a cyclic structure, such as 2,3,3-tetrafluorocyclobutylaminocarbonyl, 2-chlorocyclohexylaminocarbonyl, 4-chlorocyclohexylaminocarbonyl, and the like.

The “aryl group” represents, for example, a monocyclic and polycyclic aromatic hydrocarbon, such as phenyl group, naphtyl group, and the like.

The “arylcarbonyloxy group” represents, for example, a arylcarbonyloxy group, such as phenylcarbonyloxy group, naphtylcarbonyloxy group, and the like.

The “arylcarbonylamino group” represents, for example, a arylcarbonylamino group, such as phenylcarbonylamino group, naphtylcarbonylamino group, and the like.

The “C1-C6 alkyl group which may have a substituent” in R₁ and R₂ represents an unsubstituted linear, branched, or cyclic alkyl group having 1 to 6 carbon atoms, or a linear, branched, or cyclic alkyl group having from 1 to 6 carbon atoms, which is substituted only with at least one of a nitro group, a phenyl group which may have a substituent, and an unsaturated heterocyclic group which may have a substituent. Further, when there are two or more substituents, these substituents may be the same as or different from each other.

The “C1-C6 haloalkyl group which may have a substituent” in R₁ and R₂ represents a linear, branched, or cyclic alkyl group having from 1 to 6 carbon atoms, which is substituted with one or more halogen atoms, or a linear, branched, or cyclic alkyl group having 1 to 6 carbon atoms, which is substituted with at least one of a nitro group, a phenyl group which may have a substituent, and an unsaturated heterocyclic group which may have a substituent, in addition to one or more halogen atoms.

The “C2-C6 alkenyl group which may have a substituent” in R₁ and R₂ represents an unsubstituted linear, branched, or cyclic alkenyl group having from 2 to 6 carbon atoms, or a linear, branched, or cyclic alkenyl group having 2 to 6 carbon atoms, which is substituted with at least one of a nitro group, a phenyl group which may have a substituent, and an unsaturated heterocyclic group which may have a substituent. Further, when there are two or more substituents, these substituents may be the same as or different from each other.

The “C2-C6 haloalkenyl group which may have a substituent” in R₁ and R₂ represents a linear, branched, or cyclic alkenyl group having from 2 to 6 carbon atoms, which is substituted only with one or more halogen atoms, or a linear, branched, or cyclic alkenyl group having 2 to 6 carbon atoms, which is substituted with at least one of a nitro group, a phenyl group which may have a substituent, and an unsaturated heterocyclic group which may have a substituent, in addition to one or more halogen atoms.

The “C2-C6 alkynyl group which may have a substituent” in R₁ and R₂ represents an unsubstituted linear, branched, or cyclic alkynyl group having from 2 to 6 carbon atoms, or a linear, branched, or cyclic alkynyl group having 2 to 6 carbon atoms, which is substituted with at least one of a nitro group, a phenyl group which may have a substituent, and an unsaturated heterocyclic group which may have a substituent. Further, when there are two or more substituents, these substituents may be the same as or different from each other.

The “C2-C6 haloalkynyl group which may have a substituent” in R₁ and R₂ represents a linear, branched, or cyclic alkynyl group having from 2 to 6 carbon atoms, which is substituted only with one or more halogen atoms, or a linear, branched, or cyclic alkynyl group having 2 to 6 carbon atoms, which is substituted with at least one of a nitro group, a phenyl group which may have a substituent, and an unsaturated heterocyclic group which may have a substituent, in addition to one or more halogen atoms.

Further, each of the substituents in the present invention may further have a substituent, and examples of the substituent include the following:

one or more substituents selected from a group consisting of a halogen atom, a C1-C6 alkyl group, a C1-C6 haloalkyl group, a C3-C9 cycloalkyl group, a C3-C9 halocycloalkyl group, a C2-C6 alkenyl group, a C2-C6 haloalkenyl group, a C2-C6 alkynyl group, a C2-C6 haloalkynyl group, a C1-C6 alkoxy group, a C1-C6 haloalkoxy group, a C1-C6 alkylthio group, a C1-C6 haloalkylthio group, a C1-C6 alkylsulfinyl group, a C1-C6 haloalkylsulfinyl group, a C1-C6 alkylsulfonyl group, a C1-C6 haloalkylsulfonyl group, a C2-C7 alkylcarbonyl group, a C2-C7 haloalkylcarbonyl group, a C2-C7 alkylcarbonyloxy group, a C2-C7 haloalkylcarbonyloxy group, a C1-C6 alkylsulfonyloxy group, a C1-C6 haloalkylsulfonyloxy group, a C2-C7 alkoxycarbonyl group, a C2-C7 haloalkoxycarbonyl group, a C2-C7 alkylcarbonylamino group, a C2-C7 haloalkylcarbonylamino group, a C2-C7 alkoxycarbonylamino group, a C2-C7 haloalkoxycarbonylamino group, a C2-C7 alkylaminocarbonyl group, a C2-C7 haloalkylaminocarbonyl group, a C1-C6 alkylamino group, a C1-C6 haloalkylamino group, a C2-C6 alkenylamino group, a C2-C6 haloalkenylamino group, a C2-C6 alkynylamino group, a C2-C6 haloalkynylamino group, a C3-C9 cycloalkylamino group, a C3-C9 halocycloalkylamino group, a C3-C7 alkenylaminocarbonyl group, a C3-C7 haloalkenylaminocarbonyl group, a C3-C7 alkynylaminocarbonyl group, a C3-C7 haloalkynylaminocarbonyl group, a C4-C10 cycloalkylaminocarbonyl group, a C4-C10 halocycloalkylaminocarbonyl group, an amino group, a carbamoyl group, a sulfamoyl group, a cyano group, a nitro group, a hydroxyl group, a carboxylic group, a pentafluorosulfanyl group, a phenyl group which may have a substituent, a heterocyclic group which may have a substituent, a benzyl group which may have a substituent, a phenylcarbonyl group which may have a substituent, and a phenylamino group which may have a substituent, and when there are two or more substituents, each substituent may be the same as or different from each other.

The compounds represented by Formula (1), Formula (7), Formula (8), and the like of the present invention may include one or plural chiral carbon atoms or chiral centers in their structural Formulae, and thus two or more optical isomers may exist. However, the present invention includes each of the optical isomers and a mixture thereof at any proportions. Further, the compounds represented by Formula (1), Formula (7), Formula (8), and the like of the present invention may include two or more kinds of geometrical isomers derived from carbon-carbon double bonds in the structural Formulae. However, the present invention includes each of the geometrical isomers and a mixture thereof at any proportions.

The combinations of the substituents or atoms preferred as the substituents or the like for the amide derivative represented by Formula (1) of the present invention are as follows.

T is preferably —C(=G₁)-Q₁, G₁ is preferably an oxygen atom, Q₁ is preferably a phenyl group which may have a substituent, or a pyridyl group which may have a substituent, and Q₁ is more preferably a phenyl group or a pyridyl group which has one or more substituents selected from a group consisting of a halogen atom, a C1 haloalkyl group, a nitro group, and a cyano group, and when there are two or more substituents, each substituent may be the same as or different from each other.

G₃ is preferably an oxygen atom.

R₁ is preferably a hydrogen atom or a C1-C3 alkyl group.

R₂ is preferably a hydrogen atom.

A is preferably a carbon atom, and K is preferably a non-metal atom group which is combined with A and two carbon atoms to which A bonds to form a benzene ring.

X is preferably a hydrogen atom, a halogen atom, or a cyano group, and more preferably a hydrogen atom, a fluorine atom, or a cyano group.

When X is a substituent other than a hydrogen atom, n is preferably 0, 1, or 2.

Y₁ is preferably a halogen atom or a C1-C3 haloalkyl group.

Y₅ is preferably a C1-C3 haloalkyl group.

Y₂ and Y₄ are preferably hydrogen atoms, halogen atoms, or C1-C4 alkyl groups, and more preferably hydrogen atoms.

Y₃ is preferably a C2-C5 haloalkyl group, and more preferably a C2-C4 perfluoroalkyl group.

Furthermore, the combinations of the substituent or atom preferred as the substituent and the like for the amide derivative represented by Formula (8) are as follows.

Q₁ is preferably a phenyl group or a pyridyl group which has one or more substituents selected from a group consisting of a halogen atom, a C1 haloalkyl group, a nitro group, and a cyano group, and when there are two or more substituents, each substituent may be the same as or different from each other.

R₁ is preferably a hydrogen atom or a C1-C3 alkyl group.

R₂ is preferably a hydrogen atom.

X₁ and X₂ are preferably hydrogen atoms or fluorine atoms, and X3 and X4 are preferably hydrogen atoms.

Y₁ and Y₅ are preferably halogen atoms or C1-C3 haloalkyl groups. Y₂ and Y₄ are preferably hydrogen atoms. Y₃ is preferably a C3-C4 perfluoroalkyl group.

The representative methods for producing the compound of the present invention are shown below, and the method for producing the amide derivative of the present invention is not limited to the preparation methods below.

In Formula shown in the following preparation method, A, K, X, n, R₁, R₂, T, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅ represent the same definitions as A, K, X, n, R₁, R₂, T, G₃, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in Formula (1). LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, Hal represents a chlorine atom or a bromine atom, and Xa, Xb, and Xc represent chlorine atoms, bromine atoms, or iodine atoms.

<Preparation Method 1>

1-(i)-: Formula (21)+Formula (22)→Formula (23)

Formula (21)+Formula (22)→Formula (28)

A nitro aromatic carboxamide derivative represented by Formula (23) or Formula (28) can be prepared by reacting a nitro aromatic carboxylic acid derivative having a leaving group represented by Formula (21) with an aromatic amine derivative represented by Formula (22) in a suitable solvent or without a solvent. In the present step, a suitable base can be used.

The solvent may be any of those which do not inhibit the present reaction significantly. Examples thereof may include water and aromatic hydrocarbons such as benzene, toluene, xylene, and the like, halogenated hydrocarbons such as dichloromethane, chloroform, carbon tetrachloride, and the like, chained or cyclic ethers such as diethyl ether, dioxane, tetrahydrofuran, 1,2-dimethoxy ethane, and the like, esters such as ethyl acetate, butyl acetate, and the like, alcohols such as methanol, ethanol, and the like, ketones such as acetone, methyl isobutyl ketone, cyclohexanone, and the like, amides such as dimethyl formamide, dimethylacetamide, and the like, nitriles such as acetonitrile and the like, and inert solvents such as 1,3-dimethyl-2-imidazolidinone and the like. These solvents may be used alone or as a mixture of two or more kinds thereof.

Furthermore, examples of the base may include organic bases such as triethylamine, tri-n-butyl amine, pyridine, 4-dimethylamino pyridine, and the like, alkali metal hydroxides such as sodium hydroxide, potassium hydroxide, and the like, carbonates such as sodium hydrogen carbonate, potassium carbonate, and the like, phosphates such as dipotassium monohydrogen phosphate, trisodium phosphate, and the like, alkali metal hydride salts such as sodium hydride and the like, alkali metal alkoxides such as sodium methoxide, sodium ethoxide, and the like, and lithium amides such as lithium diisopropyl amide, and the like.

These bases may be appropriately used in an amount in the range from 0.01-fold molar equivalent to 5-fold molar equivalents with respect to the compound represented by Formula (21).

The reaction temperature may be appropriately selected from −20° to the reflux temperature of the solvent used. Further, the reaction time may be appropriately selected within the range from several minutes to 96 hours.

Among the compounds represented by Formula (21), the aromatic carbonyl halide derivative can be prepared easily by a general method using a halogenating agent from an aromatic carboxylic acid. Examples of the halogenating agent include thionyl chloride, thionyl bromide, phosphorus oxychloride, oxalyl chloride, phosphorus trichloride, and the like.

Meanwhile, it is possible to prepare the compound represented by Formula (23) or Formula (28) from the nitro aromatic carboxylic acid derivative and the compound represented by Formula (22) without using a halogenating agent. Examples of the method may include a method described in, for example, Chem. Ber. p. 788 (1970), in which a condensing agent such as N,N′-dicyclohexylcarbodiimide and the like is appropriately used, suitably with the use of an additive such as 1-hydroxybenzotriazole and the like. Other condensing agents that can be used in this case may include 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide, 1,1′-carbonylbis-1H-imidazole, and the like.

Furthermore, examples of other methods for producing the compound represented by Formula (23) or Formula (28) may include a mixed anhydride method using chloroformic acid esters, and examples thereof include a method described in J. Am. Chem. Soc., p. 5012 (1967), whereby the compound represented by Formula (23) or Formula (28) can be prepared. Examples of the chloroformic acid esters used in this case may include isobutyl chloroformate, isopropyl chloroformate and the like. In addition to chloroformic acid esters, diethylacetyl chloride, trimethylacetyl chloride and the like may also be included.

Both the method using a condensing agent and the mixed anhydride method are not limited by the solvent, the reaction temperature, and the reaction time according to the literature above. An inert solvent may be used which does not inhibit the progress of the appropriate reaction significantly, and the reaction temperature and the reaction time may also be selected appropriately according to the progress of the reaction.

1-(ii): Formula (23)→Formula (24)

Formula (28)→Formula (29)

An aromatic carboxamide derivative having an amino group represented by Formula (24) or Formula (29) can be derived from the aromatic carboxamide derivative having a nitro group represented by Formula (23) or Formula (28) by means of a reduction reaction. Examples of such reduction include a method using a hydrogenation reaction and a method using a metal compound (for example, stannous chloride (anhydride), iron powder, zinc powder, and the like).

The reaction of the former method can be carried out in a suitable solvent in the presence of a catalyst at normal pressure or a higher pressure under a hydrogen atmosphere. Examples of the catalyst may include palladium catalysts such as palladium-carbon and the like, nickel catalysts such as Raney-nickel and the like, cobalt catalysts, ruthenium catalysts, rhodium catalysts, platinum catalysts, and the like, and examples of the solvent may include water, alcohols such as methanol, ethanol, and the like; aromatic hydrocarbons such as benzene, toluene, and the like; chained or cyclic ethers such as ether, dioxane, tetrahydrofuran, and the like; and esters such as ethyl acetate and the like. The pressure may be appropriately selected within a range of 0.1 MPa to 10 MPa, the reaction temperature may be appropriately selected within a range of −20° C. to the reflux temperature of the solvent used, and the reaction time may be appropriately selected within a range of several minutes to 96 hours, whereby the compound of Formula (24) or Formula (29) can be efficiently prepared.

Examples of the latter method include a method using stannous chloride (anhydride) as a metal compound under the conditions described in “Organic Syntheses” Coll. Vol. III, P. 453.

1-(iii): Formula (24)+Formula (26)→Formula (25)

An aromatic carboxamide or carbamate derivative represented by Formula (25) can be prepared by reacting the aromatic amine derivative represented by Formula (24) with the carboxylic acid derivative or the carbonate ester derivative having a leaving group represented by Formula (26) in a suitable solvent. In the present step, a suitable base or solvent can be used, and as the base or solvent, those exemplified in 1-(i) can be used. Examples of the reaction temperature, the reaction time, and the like may include those exemplified in 1-(i).

In Formula (26), the carbonyl chloride derivative can be prepared easily from a carboxylic acid derivative by a general method using a halogenating agent. The halogenating agent may include those exemplified in 1-(i).

There may be a method for producing a compound represented by Formula (25) from the carboxylic acid derivative (26) and the compound represented by Formula (24) without the use of a halogenating agent, and the preparation can be conducted according to the method exemplified in 1-(i).

1-(iv): Formula (25)+Formula (27)→Formula (1)

The compound represented by Formula (1) of the present invention can be prepared by reacting the amide compound represented by Formula (25) with the compound having a leaving group such as halogen and the like, represented by Formula (27) in a solvent or without a solvent. In the present step, a suitable base or solvent can be used, and as the base or solvent, those exemplified in 1-(i) can be used. Examples of the reaction temperature, the reaction time, and the like may include those exemplified in 1-(i).

1-(v): Formula (28)+Formula (30)→Formula (23)

A compound represented by Formula (23) can be prepared by reacting the amide compound represented by Formula (28) with the compound having a leaving group such as halogen and the like, represented by Formula (30) in a solvent or without a solvent. In the present step, a suitable base or solvent can be used, and as the base or solvent, those exemplified in 1-(i) can be used. Examples of the reaction temperature, the reaction time, and the like may include those exemplified in 1-(i).

1-(vi): Formula (29)→Formula (31)

(Method A)

A compound represented by Formula (31) can be prepared by reacting the compound represented by Formula (29) with an aldehyde or a ketone in a solvent, and reacting them under a hydrogen atmosphere with the addition of a catalyst.

The solvent may be any of those which do not inhibit the progress of the reaction significantly, and examples thereof may include aliphatic hydrocarbons such as hexane, cyclohexane, methylcyclohexane, and the like, aromatic hydrocarbons such as benzene, xylene, toluene, and the like, halogenated hydrocarbons such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, and the like, ethers such as diethyl ether, dioxane, tetrahydrofuran, 1,2-dimethoxy ethane, and the like, amides such as dimethyl formamide, dimethylacetamide, and the like, nitriles such as acetonitrile, propionitrile, and the like, ketones such as acetone, methyl isobutyl ketone, cyclohexanone, methyl ethyl ketone, and the like, esters such as ethyl acetate, butyl acetate, and the like, alcohols such as 1,3-dimethyl-2-imidazolidinone, sulfolane, dimethylsulfoxide, methanol, ethanol, and the like, and water. These solvents may be used alone or as a mixture of two or more kinds thereof.

Examples of the catalyst may include palladium catalysts such as palladium-carbon, palladium hydroxide-carbon, and the like, nickel catalysts such as Raney-nickel and the like, cobalt catalysts, platinum catalysts, ruthenium catalysts, rhodium catalysts, and the like. Examples of the aldehydes may include formaldehyde, acetaldehyde, propionaldehyde, trifluoroacetaldehyde, difluoroacetaldehyde, fluoroacetaldehyde, chloroacetaldehyde, dichloroacetaldehyde, trichloroacetaldehyde, bromoacetaldehyde, and the like.

Examples of the ketones may include acetone, perfluoroacetone, methyl ethyl ketone, and the like.

The reaction pressure may be appropriately selected within the range of 1 atm to 100 atm. The reaction temperature may be appropriately selected within the range from −20° C. to the reflux temperature of the solvent used. Further, the reaction time may be appropriately selected within the range from several minutes to 96 hours.

(Method B)

A compound represented by Formula (31) can be prepared by reacting the compound represented by Formula (29) with an aldehyde or a ketone in a solvent, and treating the product with a reducing agent.

The solvent may be any of those which do not inhibit the progress of the reaction significantly, and examples thereof may include aliphatic hydrocarbons such as hexane, cyclohexane, methylcyclohexane, and the like, aromatic hydrocarbons such as benzene, xylene, toluene, and the like, halogenated hydrocarbons such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, and the like, ethers such as diethyl ether, dioxane, tetrahydrofuran, 1,2-dimethoxy ethane, and the like, amides such as dimethyl formamide, dimethylacetamide, and the like, nitriles such as acetonitrile, propionitrile, and the like, ketones such as acetone, methyl isobutyl ketone, cyclohexanone, methyl ethyl ketone, and the like, esters such as ethyl acetate, butyl acetate, and the like, alcohols such as 1,3-dimethyl-2-imidazolidinone, sulfolane, dimethylsulfoxide, methanol, ethanol, and the like, water, and the like. These solvents may be used alone or as a mixture of two or more kinds thereof.

Examples of the reducing agent may include, for example, borohydrides such as sodium borohydride, sodium cyanoborohydride, sodium triacetate borohydride, and the like.

Examples of the aldehydes may include formaldehyde, acetaldehyde, propionaldehyde, trifluoroacetaldehyde, difluoroacetaldehyde, fluoroacetaldehyde, chloroacetaldehyde, dichloroacetaldehyde, trichloroacetaldehyde, bromoacetaldehyde, and the like.

Examples of the ketones may include acetone, perfluoroacetone, methyl ethyl ketone, and the like.

The reaction temperature may be appropriately selected within the range from −20° C. to the reflux temperature of the solvent used. Further, the reaction time may be appropriately selected within the range from several minutes to 96 hours.

(Method C)

A compound of Formula (31) can be prepared by reacting the compound represented by Formula (29) with an aldehyde in a solvent or without a solvent.

The solvent may be any of those which do not inhibit the progress of the reaction significantly, and examples thereof may include aliphatic hydrocarbons such as hexane, cyclohexane, methylcyclohexane, and the like, aromatic hydrocarbons such as benzene, xylene, toluene, and the like, halogenated hydrocarbons such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, and the like, ethers such as diethyl ether, dioxane, tetrahydrofuran, 1,2-dimethoxy ethane, and the like, amides such as dimethyl formamide, dimethylacetamide, and the like, nitriles such as acetonitrile, propionitrile, and the like, ketones such as acetone, methyl isobutyl ketone, cyclohexanone, methyl ethyl ketone, and the like, esters such as ethyl acetate, butyl acetate, and the like, alcohols such as 1,3-dimethyl-2-imidazolidinone, sulfolane, dimethylsulfoxide, methanol, ethanol, and the like, inorganic acids such as sulfuric acid, hydrochloric acid, and the like, organic acids such as formic acid, acetic acid, and the like, water, and the like. These solvents may be used alone or as a mixture of two or more kinds thereof.

Examples of the aldehydes may include formaldehyde, acetaldehyde, propionaldehyde, and the like.

The reaction temperature may be appropriately selected within the range from −20° C. to the reflux temperature of the solvent used, and the reaction time may be appropriately selected within the range from several minutes to 96 hours.

1-(vii): Formula (31)+Formula (26)→General Formula (32)

An aromatic carboxamide or carbamate derivative represented by Formula (32) can be prepared by reacting the aromatic amine derivative represented by Formula (31) with the carboxylic acid derivative or the carbonate ester derivative having a leaving group represented by Formula (26) in a suitable solvent. In the present step, a suitable base or solvent can be used, and as the base or solvent, those exemplified in 1-(i) can be used. Examples of the reaction temperature, the reaction time, and the like may include those exemplified in 1-(i).

In Formula (26), the carbonyl chloride derivative can be prepared easily from a carboxylic acid derivative by a general method using a halogenating agent. The halogenating agent may include those exemplified in 1-(i).

There may be exemplified a method for producing a compound represented by Formula (32) from the carboxylic acid derivative (26) and the compound represented by Formula (31) without the use of a halogenating agent, and the preparation can be conducted according to the method exemplified in 1-(i).

1-(viii): Formula (32)+Formula (30)→Formula (1)

The compound represented by Formula (1) of the present invention can be prepared by reacting the amide compound represented by Formula (32) with the compound having a leaving group such as a halogen and the like, represented by Formula (30) in a solvent or without a solvent. In the present step, a suitable base or solvent can be used, and as the base or solvent, those exemplified in 1-(i) can be used. Examples of the reaction temperature, the reaction time, and the like may include those exemplified in 1-(i).

<Preparation Method 2>

2-(i): Formula (33)+Formula (22)→Formula (34)

A compound represented by Formula (34) can be prepared by reacting the compound represented by Formula (33) with a compound represented by Formula (22) under the condition described in l-(i).

2-(ii): Formula (34)→Formula (36)

A compound represented by Formula (36) can be prepared by carrying out an amination reaction using an amination agent such as ammonia and the like according to the conditions described, for example, in J. Org. Chem. p. 280 (1958). However, the conditions such as a reaction solvent and the like are not restricted to those described in the literature, and an inert solvent which does not inhibit the proper progress of the reaction significantly may be used. The reaction temperature and reaction time may be suitably selected as the reaction proceeds. Further, examples of the amination agent include methylamine, ethylamine or the like, in addition to ammonia.

2-(iii): Formula (36)+Formula (26)→Formula (1)

The compound represented by Formula (1) can be prepared by reacting the compound represented by Formula (36) with a compound represented by Formula (26) according to the conditions described in 1-(i).

<Preparation Method 3>

3-(i): Formula (29)+Formula (26)→Formula (35)

An aromatic carboxamide or carbamate derivative represented by Formula (35) can be prepared by reacting the aromatic amine derivative represented by Formula (29) with the carboxylic acid derivative or the carbonate ester derivative having a leaving group represented by Formula (26) in a suitable solvent. In the present step, a suitable base or solvent can be used, and as the base or solvent, those exemplified in 1-(i) can be used. Examples of the reaction temperature, the reaction time, and the like may include those exemplified in 1-(i).

In Formula (26), the carbonyl chloride derivative can be prepared easily from a carboxylic acid derivative by a general method using a halogenating agent. The halogenating agent may include those exemplified in 1-(i).

There may be exemplified a method for producing a compound represented by Formula (35) from the carboxylic acid derivative (26) and the compound represented by Formula (29) without the use of a halogenating agent, and the preparation can be conducted according to the method exemplified in 1-(i).

3-(ii): Formula (35)+Formula (27)→Formula (1a)

The compound represented by Formula (1a) of the present invention can be prepared by reacting the amide compound represented by Formula (35) with the compound having a leaving group such as halogen and the like, represented by Formula (27) in a solvent or without a solvent. In the present step, a suitable base or solvent can be used, and as the base or solvent, those exemplified in 1-(i) can be used. Examples of the reaction temperature, the reaction time, and the like may include those exemplified in 1-(i).

<Preparation Method 4>

4-(i): Formula (24)→Formula (36)

A compound represented by Formula (36) can be prepared by reacting the compound represented by Formula (24) as a starting material according to the conditions of (Method A), (Method B), or (Method C) described in 1-(vi).

4-(i′): Formula (24)+Formula (27)→Formula (36)

An aromatic carboxamide represented by Formula (36) can be prepared by reacting the aromatic amine derivative represented by Formula (24) with the carboxylic acid derivative or the carbonate ester derivative having a leaving group represented by Formula (27) in a suitable solvent. In the present step, a suitable base or solvent can be used, and as the base or solvent, those exemplified in 1-(i) can be used. Examples of the reaction temperature, the reaction time, and the like may include those exemplified in 1-(i).

In Formula (27), the carbonyl chloride derivative can be prepared easily from a carboxylic acid derivative by a general method using a halogenating agent. The halogenating agent may include those exemplified in 1-(i).

There may be exemplified a method for producing a compound represented by Formula (36) from the carboxylic acid derivative (27) and the compound represented by Formula (24) without the use of a halogenating agent, and the preparation can be conducted according to the method exemplified in 1-(i).

4-(ii): Formula (36)+Formula (26)→Formula (1)

A compound represented by Formula (1) can be prepared by reacting the compound represented by Formula (36) and the compound represented by Formula (26) as starting materials according to the conditions described in 1-(i).

<Preparation Method 5>

5-(i): Formula (37)+Formula (22)→Formula (38)

A compound represented by Formula (38) can be prepared by reacting the compound represented by Formula (37) and the compound represented by Formula (22) according to the conditions described in 1-(i).

5-(ii): Formula (38)→Formula (39)

A compound represented by Formula (39) can be prepared by reacting the nitro aromatic carboxamide derivative represented by Formula (38) with a suitable fluorinating agent in a suitable solvent or without a solvent.

The solvent may be any of those which do not inhibit the progress of the reaction significantly, and examples thereof may include aliphatic hydrocarbons such as hexane, cyclohexane, methylcyclohexane, and the like, aromatic hydrocarbons such as benzene, toluene, xylene, and the like, halogenated hydrocarbons such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, and the like, chained or cyclic ethers such as diethyl ether, dioxane, tetrahydrofuran, 1,2-dimethoxy ethane, and the like, esters such as ethyl acetate, butyl acetate, and the like, ketones such as acetone, methyl isobutyl ketone, cyclohexanone, methyl ethyl ketone, and the like, nitriles such as acetonitrile, propionitrile, and the like, and aprotic polar solvents such as 1,3-dimethyl-2-imidazolidinone, sulfolane, dimethylsulfoxide, N,N-dimethyl formamide, N-methyl pyrrolidone, N,N-dimethylacetamide, and the like. These solvents may be used alone or as a mixture of two or more kinds thereof.

Examples of the fluorinating agent may include 1,1,2,2-tetrafluoroethyl diethylamine, 2-chloro-1,1,2-trifluoroethyl diethylamine, trifluorodiphenylphospholane, difluorotriphenylphospholane, fluoroformic acid esters, sulfur tetrafluoride, potassium fluoride, potassium hydrogen fluoride, cesium fluoride, rubidium fluoride, sodium fluoride, lithium fluoride, antimony (III) fluoride, antimony (V) fluoride, zinc fluoride, cobalt fluoride, lead fluoride, copper fluoride, mercury (II) fluoride, silver fluoride, silver fluoroborate, thallium (I) fluoride, molybdenum (VI) fluoride, arsenic (III) fluoride, bromine fluoride, selenium tetrafluoride, tris(dimethylamino)sulfonium difluorotrimethylsilicate, sodium hexafluorosilicate, quaternary ammonium fluorides, (2-chloroethyl) diethylamine, diethylaminosulfur trifluoride, morpholinosulfur trifluoride, silicon tetrafluoride, hydrogen fluoride, hydrofluoric acid, hydrogen fluoride-pyridine complex, hydrogen fluoride-triethylamine complex, hydrogen fluoride salts, bis(2-methoxyethyl)amino sulfurtrifluoride, 2,2-difluoro-1,3-dimethyl-2-imidazolidinone, iodine pentafluoride, tris(diethylamino)phosphonium 2,2,3,3,4,4-hexafluorocyclobutanilide, triethylammonium hexafluorocylcobutanilide, hexafluoropropene, and the like. These fluorinating agents may be used alone or as a mixture of two or more kinds thereof.

The fluorinating agent may be appropriately selected and used as a solvent, in the range of 1-fold molar equivalent to 10-fold molar equivalents with respect to the nitro aromatic carboxamide derivative represented by Formula (38).

Additives may be used, and examples thereof may include crown ethers such as 18-crown-6 and the like, phase transfer catalysts such as a tetraphenylphosphonium salt and the like, inorganic salts such as calcium fluoride, calcium chloride, and the like, metal oxides such as mercury oxide and the like, ion exchange resins, and the like. These additives may not only be added to the reaction system but also used as a pretreating agent for the fluorinating agent.

The reaction temperature may be appropriately selected within the range from −80° C. to the reflux temperature of the solvent used, and the reaction time may be appropriately selected within the range from several minutes to 96 hours.

<Preparation Method 6>

6-(i): Formula (40)+Formula (22)→Formula (41)

A compound represented by Formula (41) can be prepared by reacting the compound represented by Formula (40) with a compound represented by Formula (22) according to the conditions described in 1-(i).

6-(ii): Formula (41)→Formula (42)

A compound represented by Formula (42) can be prepared by reacting the halogen aromatic carboxamide derivative represented by Formula (41) with a suitable cyanating agent in a suitable solvent or without a solvent.

The solvent may be any of those which do not inhibit the progress of the present reaction significantly. Examples thereof may include aliphatic hydrocarbons such as hexane, cyclohexane, methylcyclohexane, and the like, aromatic hydrocarbons such as benzene, toluene, xylene, and the like, halogenated hydrocarbons such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, and the like, chained or cyclic ethers such as diethyl ether, dioxane, tetrahydrofuran, 1,2-dimethoxy ethane, and the like, esters such as ethyl acetate, butyl acetate, and the like, ketones such as acetone, methyl isobutyl ketone, cyclohexanone, methyl ethyl ketone, and the like, nitriles such as acetonitrile, propionitrile, and the like, and aprotic polar solvents such as 1,3-dimethyl-2-imidazolidinone, sulfolane, dimethylsulfoxide, N,N-dimethyl formamide, N-methyl pyrrolidone, N,N-dimethylacetamide, and the like. These solvents may be used alone or as a mixture of two or more kinds thereof.

Examples of the cyanating agent include cyanide salts such as sodium cyanide, potassium cyanide, sodium cyanoborohydride, and the like, metal cyanides such as copper cyanide, silver cyanide, lithium cyanide, and the like, hydrogen cyanide, tetraehtylammonium cyanide, and the like.

These cyanating agents may be appropriately selected and used in the range of 1-fold molar equivalent to 10-fold molar equivalents with respect to the halogen aromatic carboxamide derivative represented by Formula (41).

Additives may be used, and examples thereof may include crown ethers such as 18-crown-6 and the like, phase transfer catalysts such as a tetraphenylphosphonium salt and the like, inorganic salts such as sodium iodide and the like.

The reaction temperature may be appropriately selected within the range from −20° C. to the reflux temperature of the solvent used. Further, the reaction time may be appropriately selected within the range from several minutes to 96 hours.

<Preparation Method 7>

7-(i): Formula (43)→Formula (44)

A compound represented by Formula (44) can be prepared by reacting the compound represented by Formula (43) with a Lawesson's reagent according to the known conditions described in Synthesis p. 463 (1993), Synthesis p. 829 (1984) and the like. The conditions such as a solvent, reaction temperature and the like are not restricted to those described in the literature.

2-(ii): Formula (44)+Formula (26)→Formula (45)

A compound represented by Formula (45) can be prepared by reacting the compound represented by Formula (44) with a compound represented by Formula (26) according to the conditions described in 1-(i).

<Preparation Method 8>

8: Formula (46)→Formula (47)+Formula (48)

The compounds represented by Formula (47) and Formula (48) can be prepared from a compound represented by Formula (46) according to the conditions described in 7-(i). The conditions such as a solvent, a reaction temperature, and the like are not restricted to those described in the literature. These two compounds can be easily separated and purified by a known separation and purification technique such as silica gel column chromatography and the like.

<Preparation Method 9>

9-(i): Formula (49)+Formula (26)→Formula (50)

Carboxylic acids having an acylamino group represented by Formula (50) can be prepared by reacting a carboxylic acid having an amino group represented by Formula (49) as a starting material with a compound represented by Formula (26) according to the conditions described in 1-(i).

9-(ii): Formula (50)→Formula (51)

A compound represented by Formula (51) can be prepared by a known general method including reacting the compound represented by Formula (50) with thionyl chloride, oxalyl chloride, phosgene, phosphorus oxychloride, phosphorus pentachloride, phosphorus trichloride, thionyl bromide, phosphorus tribromide, diethylaminosulfur trifluoride, or the like.

9-(iii): Formula (51)+Formula (22)→Formula (1)

The compound represented by Formula (1) can be prepared by reacting a compound represented by Formula (51) with a compound represented by Formula (22) according to the conditions described in 1-(i).

9-(iv): Formula (50)+Formula (22)→Formula (1)

The compound represented by Formula (1) can be prepared by reacting the compound represented by Formula (50) with a compound represented by Formula (22) according to the condition using a condensing agent or the condition using a mixed anhydride method according to 1-(i).

In all of the preparation methods as described above, a desired product may be isolated from the reaction system after the reaction is completed according to a general method, but if required, purification can be carried out by operations such as recrystallization, column chromatography, distillation, and the like. In addition, the desired product can be also provided to the subsequent reaction process without being separated from the reaction system.

Hereinbelow, examples of the representative compounds of the amide derivative represented by Formula (1), Formula (7), or Formula (8) as an active ingredient for the pest control agent of the present invention will be given in Table 1 to Table 51 below, but the present invention is not limited thereto.

In addition, in the tables, “n-” represents normal, “i-” represents iso, “s-” represents secondary, “t-” represents tertiary, “Me” represents a methyl group, “Et” represents an ethyl group, “n-Pr” represents a normal propyl group, “i-Pr” represents an isopropyl group, “n-Bu” represents a normal butyl group, “i-Bu” represents an isobutyl group, “s-Bu” represents a secondary butyl group, “t-Bu” represents a tertiary butyl group, “CF3” represents a trifluoromethyl group, “C2F5” represents a pentafluoroethyl group, “n-C3F7” represents a heptafluoronormal propyl group, “i-C3F7” represents a heptafluoroisopropyl group, “OCF3” represents a trifluoromethoxy group, “OC2F5” represents a pentafluoroethoxy group, “H” represents a hydrogen atom, “F” represents a fluorine atom, “Cl” represents a chlorine atom, “Br” represents a bromine atom, “I” represents an iodine atom, “O” represents an oxygen atom, “C(O)” represents a carbonyl group, “CN” represents a cyano group, “Py” represents a pyridyl group, “Ph” represents a phenyl group, and “S(O)2” represents a sulfonyl group, respectively.

TABLE 1

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

1-1

phenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-13

4-iodophenyl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

OCF3

1-16

(4-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OC2F5

1-17

2-nitrophenyl

H

H

H

CN

H

H

F

H

heptafluoroisopropyl

H

OCF3

1-20

2-cyanophenyl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

OC2F5

1-21

3-cyanophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-22

4-cyanophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-28

4-bromo-2-chlorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OC2F5

1-36

2-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

OCF3

1-37

2-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-44

6-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OC2F5

1-50

5-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OC2F5

1-55

5-nitropyridin-3-yl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

OCF3

1-57

4-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

OCF3

1-59

4-bromopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OC2F5

1-60

4-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OC2F5

1-79

phenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-95

2-nitrophenyl

H

H

H

CN

H

H

F

H

nonafluoro-2-butyl

H

OCF3

1-99

3-cyanophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-100

4-cyanophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-105

2-chloro-4,5-difluorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OC2F5

1-115

2-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-121

6-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OC2F5

1-130

5-bromopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OC2F5

1-131

5-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OC2F5

1-139

4-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OC2F5

1-140

4-nitropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OC2F5

1-157

phenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

1-177

3-cyanophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

1-178

4-cyanophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

1-193

2-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

1-200

6-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

1-222

pyridin-4-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

1-235

phenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-255

3-cyanophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-256

4-cyanophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-271

2-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-313

phenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

1-314

2-fluorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

1-333

3-cyanophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

1-334

4-cyanophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

1-349

2-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

1-356

6-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

1-391

phenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

1-411

3-cyanophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

1-412

4-cyanophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

1-427

2-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

1-434

6-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

1-469

phenyl

H

H

H

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

1-470

phenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-471

2-fluorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-472

3-fluorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-473

4-fluorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-474

2-chlorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-475

3-chlorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-476

4-chlorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-477

2-bromophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-478

3-bromophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-479

4-bromophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-480

2-iodophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-481

3-iodophenyl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

1-482

4-iodophenyl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

1-483

(2-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-484

(3-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-485

(4-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-486

2-nitrophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-487

3-nitrophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-488

4-nitrophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-489

2-cyanophenyl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

C2F5

1-490

3-cyanophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-491

4-cyanophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-492

2,6-difluorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-493

3,4-dichlorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-494

2,4-dichlorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

1-495

2-chloro-4-fluorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-496

2-chloro-4,5-difluorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-497

4-bromo-2-chlorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-498

2-bromo-4-chlorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

1-499

2-bromo-4-fluorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-500

2-chloro-4-nitrophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-501

3,5-dicyanophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-502

4-cyano-2-fluorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-503

2-chloro-4-cyanophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-504

pyrdin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-505

2-fuoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

1-506

2-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-507

2-bromopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-508

2-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-509

2-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-510

2-nitropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-511

2-cyanopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-512

6-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-513

6-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-514

6-bromopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-515

6-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-516

6-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-517

6-nitropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-518

6-cyanopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-519

5-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

1-520

5-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-521

5-bromopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

1-522

5-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

1-523

5-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-524

5-nitropyridin-3-yl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

1-525

5-cyanopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-526

4-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

1-527

4-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-528

4-bromopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-529

4-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-530

4-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-531

4-nitropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-532

4-cyanopyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-533

2,6-dichloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-534

pyridin-3-yl N-oxide

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-535

pyridin-4-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-536

2-chloropyridin-4-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-537

3-bromopyridin-4-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-538

3,5-dichloropyridin-4-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-539

3-(trifluoromethyl) pyridin-4-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-540

2,6-dichloropyridin-4-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-541

pyridin-4-yl N-oxide

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-542

pyridin-2-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-543

3-chloropyridin-2-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-544

4-bromopyridin-2-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-545

5-iodopyridin-2-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-546

6-chloropyridin-2-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-547

4-cyanopyridin-2-yl

H

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

1-548

phenyl

H

H

H

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

1-549

phenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-550

2-fluorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-551

3-fluorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-552

4-fluorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-553

2-chlorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-554

3-chlorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-555

4-chlorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-556

2-bromophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-557

3-bromophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-558

4-bromophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-559

2-iodophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-560

3-iodophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-561

4-iodophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

1-562

(2-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-563

(3-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-564

(4-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-565

2-nitrophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-566

3-nitrophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-567

4-nitrophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-568

2-cyanophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-569

3-cyanophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-570

4-cyanophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-571

2,6-difluorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-572

3,4-dichlorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-573

2,4-dichlorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-574

2-chloro-4-fluorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-575

2-chloro-4,5-difluorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-576

4-bromo-2-chlorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-577

2-bromo-4-chlorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-578

2-bromo-4-fluorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-579

2-chloro-4-nitrophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

1-580

3,5-dicyanophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-581

4-cyano-2-fluorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-582

2-chloro-4-cyanophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-583

pyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-584

2-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-585

2-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-586

2-bromopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-587

2-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-588

2-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-589

2-nitropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-590

2-cyanopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-591

6-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-592

6-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-593

6-bromopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-594

6-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-595

6-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-596

6-nitropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-597

6-cyanopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-598

5-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

1-599

5-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-600

5-bromopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

1-601

5-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

1-602

5-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-603

5-nitropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-604

5-cyanopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-605

4-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

1-606

4-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-607

4-bromopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-608

4-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-609

4-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

1-610

4-nitropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

1-611

4-cyanopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-612

2,6-dichloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-613

pyridin-3-yl N-oxide

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-614

pyridin-4-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-615

2-chloropyridin-4-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-616

3-bromopyridin-4-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-617

3,5-dichloropyridin-4-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-618

3-(trifluoromethyl) pyridin-4-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-619

2,6-dicyanopyridin-4-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-620

pyridin-4-yl N-oxide

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-621

pyridin-2-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-622

3-chloropyridin-2-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-623

4-bromopyridin-2-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-624

5-iodopyridin-2-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-625

6-chloropyridin-2-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-626

4-cyanopyridin-2-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

1-627

phenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-628

2-fluorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-629

3-fluorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-630

4-fluorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-631

2-chlorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-632

3-chlorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-633

4-chlorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-634

2-bromophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-635

3-bromophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-636

4-bromophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-637

2-iodophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-638

3-iodophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-639

4-iodophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-640

(2-trifluoromethyl) phenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-641

(3-trifluoromethyl) phenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-642

(4-trifluoromethyl) phenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-643

2-nitrophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-644

3-nitrophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-645

4-nitrophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-646

2-cyanophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-647

3-cyanophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-648

4-cyanophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-649

2,6-difluorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-650

3,4-dichlorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-651

2,4-dichlorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-652

2-chloro-4-fluorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-653

2-chloro-4,5-difluorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-654

4-bromo-2-chlorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-655

2-bromo-4-chlorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-656

2-bromo-2-fluorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-657

2-chloro-4-nitrophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-658

3,5-dicyanophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-659

4-cyano-2-fluorophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-660

2-chloro-4-cyanophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-661

pyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-662

2-fluoropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-663

2-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-664

2-bromopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-665

2-iodopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-666

2-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-667

2-nitropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-668

2-cyanopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-669

6-fluoropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-670

6-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-671

6-bromopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-672

6-iodopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-673

6-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-674

6-nitropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-675

6-cyanopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-676

5-fluoropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-677

5-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-678

5-bromopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-679

5-iodopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-680

5-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-681

5-nitropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-682

5-cyanopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-683

4-fluoropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-684

4-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-685

4-bromopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-686

4-iodopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-687

4-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-688

4-nitropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-689

4-cyanopyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-690

2,6-dichloropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-691

pyridin-3-yl N-oxide

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-692

pyridin-4-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-693

2-chloropyridin-4-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-694

3-bromopyridin-4-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-695

3,5-dichloropyridin-4-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-696

3-(trifluoromethyl) pyridin-4-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-697

2,6-dicyanopyridin-4-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-698

pyridin-4-yl N-oxide

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-699

pyridin-2-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-700

3-chloropyridin-2-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-701

4-bromopyridin-2-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-702

5-iodopyridin-2-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-703

6-chloropyridin-2-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-704

4-cyanopyridin-2-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-705

phenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-706

2-fluorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-707

3-fluorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-708

4-fluorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-709

2-chlorephenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-710

3-chlorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-711

4-chlorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-712

2-bromophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-713

3-bromophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-714

4-bromophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-715

2-iodophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-716

3-iodophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-717

4-iodophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-718

(2-trifluoromethyl) phenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-719

(3-trifluoromethyl) phenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-720

(4-trifluoromethyl) phenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-721

2-nitrophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-722

3-nitrophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-723

4-nitrophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-724

2-cyanophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-725

3-cyanophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-726

4-cyanophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-727

2,6-diflurophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-728

3,4-dichlorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-729

2,4-dichlorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-730

2-chloro-4-flurorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-731

2-chloro-4,5-diflurorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-732

4-bromo-2-chlorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-733

2-bromo-4-chlorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-734

2-bromo-4-chlorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-735

2-chloro-4-nitrophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-736

3,5-dicyanophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-737

4-cyano-2-fluorophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-738

2-chloro-4-cyanophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-739

pyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-740

2-fluoropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-741

2-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-742

2-bromopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-743

2-iodopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-744

2-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-745

2-nitropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-746

2-cyanopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-747

6-fluoropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-748

6-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-749

6-bromopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-750

6-iodopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-751

6-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-752

6-nitropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-753

6-cyanopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-754

5-fluoropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-755

5-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-756

5-bromopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-757

5-iodopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-758

5-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-759

5-nitropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-760

5-cyanopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-761

4-fluoropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-762

4-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-763

4-bromopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-764

4-iodopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-765

4-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-766

4-nitropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-767

4-cyanopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-768

2,6-dichloropyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-769

pyridin-3-yl N-oxide

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-770

pyridin-4-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-771

2-chloropyridin-4-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-772

3-bromopyridin-4-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-773

3,5-dichloropyridin-4-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-774

3-(trifluoromethyl) pyridin-4-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-775

2,6-dicyanopyridin-3-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-776

pyridin-4-yl N-oxide

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-777

pyridin-2-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-778

3-chloropyridin-2-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-779

4-bromopyridin-2-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-780

5-iodopyridin-2-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-781

6-chloropyridin-2-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-782

4-cyanopyridin-2-yl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-783

phenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-784

2-flourophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-785

3-flourophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-786

4-flourophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-787

2-chlorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-788

3-chlorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-789

4-chlorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-790

2-bromophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-791

3-bromophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-792

4-bromophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-793

2-iodophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-794

3-iodophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-795

4-iodophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-796

(2-trifluoromethyl) phenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-797

(3-trifluoromethyl) phenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-798

(4-trifluoromethyl) phenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-799

2-nitrophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-800

3-nitrophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-801

4-nitrophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-802

2-cyanophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-803

3-cyanophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-804

4-cyanophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-805

2,6-difluorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-806

3,4-dichlorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-807

2,4-dichlorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-808

2-chloro-4-fluorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-809

2-chloro-4,5-difluorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-810

4-bromo-2-chlorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-811

2-bromo-4-chlorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-812

2-bromo-4-fluorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-813

2-chloro-4-nitrophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-814

3,5-dicyanophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-815

4-cyano-2-fluorophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-816

2-chloro-4-cyanophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-817

pyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-818

2-fluoropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-819

2-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-820

2-bromopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-821

2-iodopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-822

2-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-823

2-nitropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-824

2-cyanopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-825

6-fluoropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-826

6-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-827

6-bromopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-828

6-iodopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-829

6-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-830

6-nitropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-831

6-cyanopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-832

5-fluoropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-833

5-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-834

5-bromopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-835

5-iodopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-836

5-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-837

5-nitropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-838

5-cyanopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-839

4-fluoropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-840

4-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-841

4-bromopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-842

4-iodopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-843

4-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-844

4-nitropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-845

4-cyanopyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-846

2,6-dichloropyridin-3-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-847

pyridin-3-yl N-oxide

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-848

pyridin-4-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-849

2-chloropyridin-4-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-850

3-bromopyridin-4-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-851

3,5-dichloropyridin-4-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-852

3-(trifluoromethyl) pyridin-4-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-853

2,6-dicyanopyridin-4-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-854

pyridin-4-yl N-oxide

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-855

pyridin-2-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-856

3-chloropyridin-2-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-857

4-bromopyridin-2-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-858

5-iodopyridin-2-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-859

6-chloropyridin-2-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-860

4-cyanopyridin-2-yl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-861

phenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-862

2-flourophenyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-863

3-fluorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-864

4-fluorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-865

2-chlorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-866

3-chlorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-867

4-chlorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-868

2-bromophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-869

3-bromophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-870

4-bromophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-871

2-iodophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-872

3-iodophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-873

4-iodophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-874

(2-trifluoromethyl) phenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-875

(3-trifluoromethyl) phenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-876

(4-trifluoromethyl) phenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-877

2-nitrophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-878

3-nitrophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-879

4-nitrophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-880

2-cyanophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-881

3-cyanophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-882

4-cyanophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-883

2,6-difluorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-884

3,4-dichlorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-885

2,4-dichlorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-886

2-chloro-4-fluorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-887

2-chloro-4,5-difluorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-888

4-bromo-2-chlorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-889

2-bromo-4-chlorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-890

2-bromo-4-fluorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-891

2-chloro-4-nitrophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-892

3,5-dicyanophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-893

4-cyano-2-fluorophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-894

2-chloro-4-cyanophenyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-895

pyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-896

2-fluoropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-897

2-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-9utyl

H

CF3

1-898

2-bromopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-899

2-iodopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-900

(2-trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-901

2-nitropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-902

2-cyanopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-903

6-fluoropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-904

6-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-905

6-bromopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-906

6-iodopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-907

6-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-908

6-nitropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-909

6-cyanopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-910

5-fluoropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-911

5-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-912

5-bromopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-913

5-iodopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-914

5-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-915

5-nitropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-916

5-cyanopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-917

4-fluoropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-918

4-chloropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-919

4-bromopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-920

4-iodopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-921

4-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-922

4-nitropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-923

4-cyanopyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-924

2,6-dichloropyridin-3-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-9utyl

H

CF3

1-925

pyridin-3-yl N-oxide

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-926

pyridin-4-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-927

2-chloropyridin-4-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-928

3-bromopyridin-4-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-929

3,5-dichloropyridin-4-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-930

3-(trifluoromethyl) pyridin-4-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-931

2,6-dicyanopyridin-4-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-932

pyridin-4-yl N-oxide

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-933

pyridin-2-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-934

3-chloropyridin-2-yl

H

H

H

CN

H

F1

I

H

nonafluoro-2-butyl

H

CF3

1-935

4-bromopyridin-2-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

C F3

1-936

5-iodopyridin-2-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-937

6-chloropyridin-2-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-938

4-cyanopyridin-2-yl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-939

phenyl

H

H

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-954

3-cyanophenyl

H

H

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-955

4-cyanophenyl

H

H

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-970

2-chloropyridin-3-yl

H

H

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-995

phenyl

H

H

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-1010

3-cyanophenyl

H

H

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-1011

4-cyanophenyl

H

H

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-1026

2-chloropyridin-3-yl

H

H

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-1051

phenyl

H

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-1066

3-cyanophenyl

H

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-1067

4-cyanophenyl

H

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-1082

2-chloropyridin-3-yl

H

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-1107

phenyl

H

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-1122

3-cyanophenyl

H

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-1123

4-cyanophenyl

H

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-1138

2-chloropyridin-3-yl

H

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-1163

phenyl

H

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

1-1175

4-iodophenyl

H

H

H

CN

H

H

CF3

H

pentafluoroethyl

H

CF3

1-1177

(3-trifluoromethyl) phenyl

H

H

H

CN

H

H

C2F5

H

heptafluoroisopropyl

H

CF3

1-1183

3-cyanophenyl

H

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

1-1184

4-cyanophenyl

H

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

1-1190

4-bromo-2-chlorophenyl

H

H

H

CN

H

H

n-C3F7

H

heptafluoroisopropyl

H

CF3

1-1195

4-cyano-2-fluorophenyl

H

H

H

CN

H

H

i-C3F7

H

heptafluoroisopropyl

H

CF3

1-1199

2-chloropyridin-3-yl

H

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

1-1200

2-bromopyridin-3-yl

H

H

H

CN

H

H

C2F5

H

heptafluoroisopropyl

H

C2F5

1-1211

6-cyanopyridin-3-yl

H

H

H

CN

H

H

C2F5

H

heptafluoroisopropyl

H

n-C3F7

1-1215

4-cyanopyridin-3-yl

H

H

H

CN

H

H

C2F5

H

heptafluoroisopropyl

H

i-C3F7

1-1231

phenyl

H

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

1-1243

4-iodophenyl

H

H

H

CN

H

H

C2F5

H

nonafluoro-2-butyl

H

CF3

1-1251

3-cyanophenyl

H

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

1-1252

4-cyanophenyl

H

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

1-1258

4-bromo-2-chlorophenyl

H

H

H

CN

H

H

n-C3F7

H

nonafluoro-2-butyl

H

CF3

1-1263

4-cyano-2-fluorophenyl

H

H

H

CN

H

H

i-C3F7

H

nonafluoro-2-butyl

H

CF3

1-1267

2-chloropyridin-3-yl

H

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

1-1268

2-bromopyridin-3-yl

H

H

H

CN

H

H

C2F5

H

nonafluoro-2-butyl

H

C2F5

1-1279

6-cyanopyridin-3-yl

H

H

H

CN

H

H

C2F5

H

nonafluoro-2-butyl

H

n-C3F7

1-1283

4-cyanopyridin-3-yl

H

H

H

CN

H

H

C2F5

H

nonafluoro-2-butyl

H

i-C3F7

1-1299

phenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-1319

3-cyanophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-1320

4-cyanophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-1335

2-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-1377

phenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-1384

3-bromophenyl

H

H

H

CN

H

H

F

H

nonafluoro-2-butyl

H

OCF3

1-1397

3-cyanophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-1398

4-cyanophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-1413

2-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-1455

phenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

1-1475

3-cyanophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

1-1476

4-cyanophenyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

1-1491

2-chloropyridin-3-yl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

1-1533

phenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-1553

3-cyanophenyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-1554

4-cyanophenyl

H

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-1569

2-chloropyridin-3-yl

H

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-1611

phenyl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

1-1631

3-cyanophenyl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

1-1632

4-cyanophenyl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

1-1647

2-chloropyridin-3-yl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

1-1689

phenyl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

1-1709

3-cyanophenyl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

1-1710

4-cyanophenyl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

1-1725

2-chloropyridin-3-yl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

1-1767

phenyl

H

H

F

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

1-1768

phenyl

H

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-1788

3-cyanophenyl

H

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-1789

4-cyanophenyl

H

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-1804

2-ehloropyridin-3-yl

H

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

1-1846

phenyl

H

H

F

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

1-1847

phenyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-1867

3-cyanophenyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-1868

4-cyanophenyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-1883

2-chloropyridin-3-yl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-1925

phenyl

H

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-1945

3-cyanophenyl

H

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-1946

4-cyanophenyl

H

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-1961

2-chloropyridin-3-yl

H

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-1968

6-chloropyridin-3-yl

H

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

1-2003

phenyl

H

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-2023

3-cyanophenyl

H

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-2024

4-cyanophenyl

H

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-2039

2-chloropyridin-3-yl

H

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

1-2081

phenyl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-2101

3-cyanophenyl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-2102

4-cyanophenyl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-2117

2-chloropyridin-3-yl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

1-2159

phenyl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-2179

3-cyanophenyl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-2180

4-cyanophenyl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-2195

2-chloropyridin-3-yl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

1-2237

phenyl

H

H

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-2252

3-cyanophenyl

H

H

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-2253

4-cyanophenyl

H

H

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-2268

2-chloropyridin-3-yl

H

H

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-2293

phenyl

H

H

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-2308

3-cyanophenyl

H

H

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-2309

4-cyanophenyl

H

H

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-2324

2-chloropyridin-3-yl

H

H

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-2325

2-bromopyridin-3-yl

H

H

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-2349

phenyl

H

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-2364

3-cyanophenyl

H

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-2365

4-cyanophenyl

H

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-2380

2-chloropyridin-3-yl

H

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-2405

phenyl

H

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-2420

3-cyanophenyl

H

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-2421

4-cyanophenyl

H

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-2436

2-chloropyridin-3-yl

H

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-2461

phenyl

H

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

1-2481

3-cyanophenyl

H

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

1-2482

4-cyanophenyl

H

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

1-2497

2-chloropyridin-3-yl

H

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

1-2529

phenyl

H

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

1-2549

3-cyanophenyl

H

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

1-2550

4-cyanophenyl

H

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

1-2565

2-chloropyridin-3-yl

H

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

1-2597

phenyl

H

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-2617

3-cyanophenyl

H

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-2618

4-cyanophenyl

H

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-2633

2-chloropyridin-3-yl

H

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

1-2675

phenyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-2695

3-cyanophenyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-2696

4-cyanophenyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-2711

2-chloropyridin-3-yl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

1-2753

phenyl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

1-2773

3-cyanophenyl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

1-2774

4-cyanophenyl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

1-2789

2-chloropyridin-3-yl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

1-2831

phenyl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-2851

3-cyanophenyl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-2852

4-cyanophenyl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-2867

2-chloropyridin-3-yl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

1-2909

phenyl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

1-2929

3-cyanophenyl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

1-2930

4-cyanophenyl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

1-2945

2-chloropyridin-3-yl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

1-2987

phenyl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

1-3007

3-cyanophenyl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

1-3008

4-cyanophenyl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

1-3023

2-chloropyridin-3-yl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

1-3065

phenyl

H

H

F

CN

F

H

F

H

heptafluoroisopropyl

H

CF3

1-3066

phenyl

H

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

1-3086

3-cyanophenyl

H

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

1-3087

4-cyanophenyl

H

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

1-3102

2-chloropyridin-3-yl

H

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

1-3144

phenyl

H

H

F

CN

F

H

F

H

nonafluoro-2-butyl

H

CF3

1-3145

phenyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-3165

3-cyanophenyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-3166

4-cyanophenyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-3181

2-chloropyridin-3-yl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

1-3223

phenyl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

1-3243

3-cyanophenyl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

1-3244

4-cyanophenyl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

1-3259

2-chloropyridin-3-yl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

1-3301

phenyl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

1-3321

3-cyanophenyl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

1-3322

4-cyanophenyl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

1-3337

2-chloropyridin-3-yl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

1-3379

phenyl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

1-3399

3-cyanophenyl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

1-3400

4-cyanophenyl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

1-3415

2-chloropyridin-3-yl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

1-3457

phenyl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

1-3477

3-cyanophenyl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

1-3478

4-cyanophenyl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

1-3493

2-chloropyridin-3-yl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

1-3535

phenyl

H

H

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-3550

3-cyanophenyl

H

H

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-3551

4-cyanophenyl

H

H

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-3566

2-chloropyridin-3-yl

H

H

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

1-3591

phenyl

H

H

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-3606

3-cyanophenyl

H

H

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-3607

4-cyanophenyl

H

H

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-3622

2-chloropyridin-3-yl

H

H

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

1-3647

phenyl

H

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-3662

3-cyanophenyl

H

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-3663

4-cyanophenyl

H

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-3678

2-chloropyridin-3-yl

H

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

1-3703

phenyl

H

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-3718

3-cyanophenyl

H

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-3719

4-cyanophenyl

H

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-3734

2-chloropyridin-3-yl

H

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

1-3759

phenyl

H

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

1-3779

3-cyanophenyl

H

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

1-3780

4-cyanophenyl

H

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

1-3795

2-chloropyridin-3-yl

H

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

1-3827

phenyl

H

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

1-3847

3-cyanophenyl

H

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

1-3848

4-cyanophenyl

H

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

1-3863

2-chloropyridin-3-yl

H

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 2

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

2-1

phenyl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-21

3-cyanophenyl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-22

4-cyanophenyl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-37

2-chloropyridin-3-yl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-79

phenyl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-99

3-cyanophenyl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-100

4-cyanophenyl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-115

2-chloropyridin-3-yl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-157

phenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

2-177

3-cyanophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

2-178

4-cyanophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

2-193

2-chloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

2-235

phenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-255

3-cyanophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-256

4-cyanophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-271

2-chloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-313

phenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

2-333

3-cyanophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

2-334

4-cyanophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

2-349

2-chloropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

2-391

phenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

2-411

3-cyanophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

2-412

4-cyanophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

2-427

2-chloropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

2-469

phenyl

Me

H

H

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

2-470

phenyl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-481

3-iodophenyl

Me

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

2-482

4-iodophenyl

Me

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

2-484

(3-trifluoromethyl) phenyl

Et

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-489

2-cyanophenyl

Me

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

C2F5

2-490

3-cyanophenyl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-491

4-cyanophenyl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-494

2,4-dichlorophenyl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

2-495

2-chloro-4-fluorophenyl

n-Pr

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-498

2-bromo-4-chlorophenyl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

2-505

2-fluoropyridin-3-yl

Me

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

2-506

2-chloropyridin-3-yl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-512

6-fluoropydin-3-yl

i-Pr

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-513

6-chloropyridin-3-yl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-518

6-cyanopyridin-3-yl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-519

5-fluoropyridin-3-yl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

2-521

5-bromopyridin-3-yl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

2-522

5-iodopyridin-3-yl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

2-524

5-nitropyridin-3-yl

Me

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

2-526

4-fluoropyridin-3-yl

Me

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

2-528

4-bromopyridin-3-yl

CH2CH═CH2

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

2-529

4-iodopyridin-3-yl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

2-535

pyridin-4-yl

CN

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-547

4-cyanopyridin-2-yl

Me

H

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

2-548

phenyl

Me

H

H

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

2-549

phenyl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-556

2-bromophenyl

CH2C═CH

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-562

(2-triflouromethyl) phenyl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

2-563

(3-triflouromethyl) phenyl

NH2

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-569

3-cyanophenyl

Me

H

H

CN

H

H

Cl

H

nona5uoro-2-butyl

H

CF3

2-570

4-cyanophenyl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-576

4-bromo-2-chlorophenyl

C(O)OMe

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-579

2-chloro-4-nitrophenyl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

2-585

2-chloropyridin-3-yl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-596

6-nitropyridin-3-y'

C(O)OEt

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-598

5-fluoropyridin-3-yl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

2-600

5-bromopyridin-3-yl

Me

H

H

CN

H

H

Cl

H

nona5uoro-2-butyl

H

n-C3F7

2-601

5-iodopydin-3-yl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

2-605

4-fluoropyridin-3-yl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

2-607

4-bromopyridin-3-yl

C(O)C(O)Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-609

4-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

Cl

H

nona9uoro-2-butyl

H

n-C3F7

2-610

4-nitropyridin-3-yl

C(O)O(O)Et

H

H

CN

H

H

Cl

H

nona5uoro-2-butyl

H

i-C3F7

2-623

4-bromopyridin-2-yl

C(O)Me

H

H

CN

H

H

Cl

H

nona5uoro-2-butyl

H

CF3

2-625

6-chloropyridin-2-yl

C(O)Et

H

H

CN

H

H

Cl

H

nona5uoro-2-butyl

H

CF3

2-626

4-cyanopyridin-2-yl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

2-627

phenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-628

2-fluorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-629

3-fluorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-630

4-fluorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-631

2-chlorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-632

3-chlorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-633

4-chlorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-634

2-bromophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-635

3-bromophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-636

4-bromophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-637

2-iodophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-638

3-iodophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-639

4-iodophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-640

(2-trifluoromethyl) phenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-641

(3-trifluoromethyl) phenyl

S(O)2Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-642

(4-trifluoromethyl) phenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-643

2-nitrophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-644

3-nitropheeyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-645

4-nitrophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-646

2-cyanophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-647

3-cyanophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-648

4-cyanophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-649

2,6-difluorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-650

3,4-dichlorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-651

2,4-dichlorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-652

2-chloro-4-fluorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-653

2-chloro-4,5-difluorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-654

4-bromo-4-chlorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-655

2-bromo-4-chlorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-656

2-bromo-4-fluorophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-657

2-chloro-4-nitrophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-658

3,5-dicyanophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-659

4-cyano-2-fluorophenyl

S(O)2Et

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-660

2-chloro-4-cyanophenyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-661

pyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-662

2-fluoropyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-663

2-chloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-664

2-bromopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-665

2-iodopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-666

2-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-667

2-nitropyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-668

2-cyanopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-669

6-fluoropyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-670

6-chloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-671

6-bromopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-672

6-iodopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-673

6-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-674

6-nitropyridin-3-yl

CH2Ph

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-675

6-cyanopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-676

5-fluoropyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-677

5-chloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-678

5-bromopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-679

5-iodopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-680

5-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-681

5-nitropyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-682

5-cyanopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-683

4-fluoropyri4in-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-684

4-chloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-685

4-bromopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-686

4-iodopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-687

4-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-688

4-nitropyridin-3-yl

CH2(3-Py)

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-689

4-cyanopyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-690

2,6-dichloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-691

pyridin-3-yl N-oxide

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-692

pyridin-4-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-693

2-chloropyridin-4-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-694

3-bromopyridin-4-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-695

3,5-dichloropyridin-4-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-696

3-(trifluoromethyl) pyridin-4-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-697

2,6-dicyanopyridin-4-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-698

pyridin-4-yl N-oxide

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-699

pyridin-2-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-700

3-chloropyridin-2-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-701

4-bromopyridin-2-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-702

5-iodopyridin-2-yl

CH2(3-Py-N-

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-703

6-chloropyridin-2-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-704

4-cyanopyridin-2-yl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-705

phenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-706

2-fluorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-707

3-fluorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-708

4-fluorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-709

2-chlorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-710

3-chlorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-711

4-chlorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-712

2-bromophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-713

3-bromophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-714

4-bromophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-715

2-iodophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-716

3-iodophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-717

4-iodophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-718

(2-trifluoromethyl) phenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-719

(3-trifluoromethyl) phenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-720

(4-trifluoromethyl) phenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-721

2-nitrophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-722

3-nitrophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-723

4-nitrophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-724

2-cyanophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-725

3-cyanophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-726

4-cyanophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-727

2,6-difluorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-728

3,4-dichlorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-729

2,4-dichlorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-730

2-chloro-4-fluorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-731

2-chloro-4,5-difluorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-732

4-bromo-2-chlorophenyl

Et

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-733

2-bromo-4-chlorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-734

4-bromo-4-fluorophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-735

2-chloro-4-nitrophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-736

3,5-dicyanophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-737

4-cyano-2-flurophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-738

2-chloro-4-cyanophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-739

pyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-740

2-fluoropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-741

2-chloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-742

2-bromopyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-743

2-iodopyndin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-744

2-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-745

2-nitropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-746

2-cyanopyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-747

6-fluoropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-748

6-chloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-749

6-bromopyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-750

6-iodopyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-751

6-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-752

6-nitropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-753

6-cyanopyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-754

5-fluoropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-755

5-chloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-756

5-bromopyridin-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-757

5-iodopyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-758

5-(trifluoromethyl) pyridin-3-yl

CN

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-759

5-nitropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-760

5-cyanopyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-761

4-fluoropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-762

4-chloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-763

4-bromopyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-764

4-iodopyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-765

4-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-766

4-nitropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-767

4-cyanopyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-768

2,6-dichloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-769

pyridin-3-yl N-oxide

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-770

pyridin-4-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-771

2-chloropyridin-4-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-772

3-bromopyridin-4-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-773

3,5-dichloropyridin-4-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-774

3-(trifluoromethyl) pyridin-4-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-775

2,6-dicyanopyridin-4-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-776

pyridin-4-yl N-oxide

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-777

pyridin-2-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-778

3-chloropyridin-2-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-779

4-bromopyridin-2-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-780

5-iodopyridin-2-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-781

6-chloropyridin-2-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-782

4-cyanopyridin-2-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-783

phenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-784

2-flurophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-785

3-flurophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-786

4-flurophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-787

2-chlorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-788

3-chlorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-789

4-chlorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-790

2-bromophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-791

3-bromophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-792

4-bromophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-793

2-iodophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-794

3-iodophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-795

4-iodophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-796

(2-trifluoromethyl) phenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-797

(3-trifluoromethyl) phenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-798

(4-trifluoromethyl) phenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-799

2-nitrophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-800

3-nitrophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-801

4-nitrophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-802

2-cyanophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-803

3-cyanophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-804

4-cyanophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-805

2,6-difluorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-806

3,4-dichlorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-807

2,4-dichlorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-808

2-chloro-4-fluorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-809

2-chloro-4,5-difluorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-810

4-bromo-2-chlorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-811

2-bromo-4-chlorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-812

2-bromo-4-fluorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-813

2-chloro-4-nitrophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-814

3,5-dicyanophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-815

4-cyano-2-fluorophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-816

2-chloro-4-cyanophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-817

pyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-818

2-fluoropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-819

2-chloropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-820

2-bromopyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-821

2-iodopyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-822

2-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-823

2-nitropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-824

2-cyanopyridin-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-825

6-fluoropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-826

6-chloropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-827

6-bromopyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-828

6-iodopyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-829

6-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-830

6-nitropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-831

6-cyanopyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-832

5-fluoropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-833

5-chloropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-834

5-bromopyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-835

5-iodopyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-836

5-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-837

5-nitropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-838

5-cyanopyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-839

4-fluoropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-840

4-chloropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-841

4-bromopyridin-3-yl

C(O)Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-842

4-iodopyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-843

4-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-844

4-nitropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-845

4-cyanopyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-846

2,6-dichloropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-847

pyridin-3-yl N-oxide

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-848

pyridin-4-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-849

2-chloropyridin-4-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-850

3-bromopyridin-4-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-851

3,6-dichloropyridin-4-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-852

3-(trifluoromethyl) pyridin-4-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-853

2,6-dichloropyridin-4-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-854

pyridin-4-yl N-oxide

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-855

pyridin-2-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-856

3-chloropyridin-2-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-857

4-bromopyridin-2-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-858

5-iodopyridin-2-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-859

6-chloropyridin-2-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-860

4-cyanopyridin-2-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-861

phenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-862

2-fluorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-863

3-fluorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-864

4-fluorophenyl

Me

H

H

CH

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-865

2-chlorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-866

3-chlorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-867

4-chlorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-868

2-bromophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-869

3-bromophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-870

4-bromophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-871

2-iodophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-872

3-iodophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-873

4-iodophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-874

(2-trifluoromethyl) phenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-875

(3-trifluoromethyl) phenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-876

(4-trifluoromethyl) phenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-877

2-nitrophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-878

3-nitrophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-879

4-nrtrophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-880

2-cyanophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-881

3-cyanophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-882

4-cyanophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-883

2,6-difluorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-884

3,4-dichlorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-885

2,4-dichlorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-886

2-chloro-4-fluorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-887

2-chloro-4,5-difluorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-888

4-bromo-2-chlorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-889

2-bromo-4-chlorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-890

2-bromo-4-fluorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-891

2-chloro-4-nitrophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-892

3,5-dicyanophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-893

4-cyano-2-fluorophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-894

2-chloro-4-cyanophenyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-895

pyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-896

2-fluoropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-897

2-chloropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-898

2-bromopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-899

2-iodopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-900

2-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-901

2-nitropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-902

2-cyanopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-903

6-fluoropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-904

6-chloropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-905

6-bromopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-906

6-iodopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-907

6-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-908

6-nitropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-909

6-cyanopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-910

5-fluoropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-911

5-chloropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-912

5-bromopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-913

5-iodopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-914

5-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-915

5-nitropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-916

5-cyanopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-917

4-fluoropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-918

4-chloropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-919

4-bromopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-920

4-iodopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-921

4-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-922

4-nitropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-923

4-cyanopyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-924

2,6-dichloropyridin-3-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-925

pyridin-3-yl N-oxide

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-926

pyridin-4-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-927

2-chloropyridin-4-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-928

3-bromopyridin-4-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-929

3,5-dichloropyridin-4-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-930

3-(trifluoromethyl) pyridin-4-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-931

2,6-dicyanopyridin-4-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-932

pyridin-4-yl N-oxide

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-933

pyridin-2-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-934

3-chloropyridin-2-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-935

4-bromopyridin-2-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-936

5-iodopyridin-2-yl

Me

H

H

CN

H

H

I

H

nona8uoro-2-butyl

H

CF3

2-937

6-chloropyridin-2-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-938

4-cyanopyridin-2-yl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-939

phenyl

Me

H

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

2-970

2-chloropyridin-3-yl

Me

H

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

2-995

phenyl

Me

H

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

2-1026

2-chloropyridin-3-yl

Me

H

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

2-1051

phenyl

Me

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

2-1082

2-chloropyridin-3-yl

Me

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

2-1107

phenyl

Me

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

2-1138

2-chloropyridin-3-yl

Me

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

2-1163

phenyl

Me

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

2-1183

3-cyanophenyl

Me

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

2-1184

4-cyanophenyl

Me

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

2-1199

2-chloropyridin-3-yl

Me

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

2-1231

phenyl

Me

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

2-1251

3-cyanophenyl

Me

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

2-1252

4-cyanophenyl

Me

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

2-1267

2-chloropyridin-3-yl

Me

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

2-1299

phenyl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-1319

3-cyanophenyl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-1320

4-cyanophenyl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-1335

2-chloropyridin-3-yl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-1377

phenyl

Me

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-1397

3-cyanophenyl

Me

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-1398

4-cyanophenyl

Me

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-1413

2-chloropyridin-3-yl

Me

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-1455

phenyl

Me

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

2-1475

3-cyanophenyl

Me

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

2-1476

4-cyanophenyl

Me

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

2-1491

2-chloropyridin-3-yl

Me

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

2-1533

phenyl

Me

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-1553

3-cyanophenyl

Me

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-1554

4-cyanophenyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-1569

2-chloropyridin-3-yl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-1611

phenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

2-1631

3-cyanophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

2-1632

4-cyanophenyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

2-1647

2-chloropyridin-3-yl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

2-1689

phenyl

Me

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

2-1709

3-cyanophenyl

Me

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

2-1710

4-cyanophenyl

Me

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

2-1725

2-chloropyridin-3-yl

Me

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

2-1767

phenyl

Me

H

F

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

2-1768

phenyl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-1788

3-cyanophenyl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-1789

4-cyanophenyl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-1804

2-chloropyridin-3-yl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

2-1846

phenyl

Me

H

F

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

2-1847

phenyl

Me

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-1867

3-cyanophenyl

Me

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-1868

4-cyanophenyl

Me

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-1883

2-chloropyridin-3-yl

Me

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-1925

phenyl

Me

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-1945

3-cyanophenyl

Me

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-1946

4-cyanophenyl

Me

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-1961

2-chloropyridin-3-yl

Me

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

2-2003

phenyl

Me

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-2023

3-cyanophenyl

Me

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-2024

4-cyanophenyl

Me

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-2039

2-chloropyridin-3-yl

Me

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

2-2081

phenyl

Me

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-2101

3-cyanophenyl

Me

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-2102

4-cyanophenyl

Me

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-2117

2-chloropyridin-3-yl

Me

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

2-2159

phenyl

Me

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-2179

3-cyanophenyl

Me

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-2180

4-cyanophenyl

Me

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-2195

2-chloropyridin-3-yl

Me

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

2-2237

phenyl

Me

H

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

2-2268

2-chloropyridin-3-yl

Me

H

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

2-2293

phenyl

Me

H

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

2-2324

2-chloropyridin-3-yl

Me

H

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

2-2349

phenyl

Me

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

2-2380

2-chloropyridin-3-yl

Me

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

2-2405

phenyl

Me

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

2-2436

2-chloropyridin-3-yl

Me

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

2-2461

phenyl

Me

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

2-2481

3-cyanophenyl

Me

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

2-2482

4-cyanophenyl

Me

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

2-2497

2-chloropyridin-3-yl

Me

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

2-2529

phenyl

Me

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

2-2549

3-cyanophenyl

Me

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

2-2550

4-cyanophenyl

Me

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

2-2565

2-chloropyridin-3-yl

Me

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

2-2597

phenyl

Me

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-2617

3-cyanophenyl

Me

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-2618

4-cyanophenyl

Me

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-2633

2-chloropyridin-3-yl

Me

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

2-2675

phenyl

Me

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-2695

3-cyanophenyl

Me

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-2696

4-cyanophenyl

Me

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-2711

2-chloropyridin-3-yl

Me

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

2-2753

phenyl

Me

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

2-2773

3-cyanophenyl

Me

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

2-2774

4-cyanophenyl

Me

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

2-2789

2-chloropyridin-3-yl

Me

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

2-2831

phenyl

Me

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-2851

3-cyanophenyl

Me

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-2852

4-cyanophenyl

Me

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-2867

2-chloropyridin-3-yl

Me

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

2-2909

phenyl

Me

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

2-2929

3-cyanophenyl

Me

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

2-2930

4-cyanophenyl

Me

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

2-2945

2-chloropyridin-3-yl

Me

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

2-2987

phenyl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

2-3007

3-cyanophenyl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

2-3008

4-cyanophenyl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

2-3023

2-chloropyridin-3-yl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

2-3065

phenyl

Me

H

F

CN

F

H

F

H

heptafluoroisopropyl

H

CF3

2-3066

phenyl

Me

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

2-3086

3-cyanophenyl

Me

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

2-3087

4-cyanophenyl

Me

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

2-3102

2-chloropyridin-3-yl

Me

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

2-3144

phenyl

Me

H

F

CN

F

H

F

H

nonafluoro-2-butyl

H

CF3

2-3165

3-cyanophenyl

Me

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-3166

4-cyanophenyl

Me

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-3181

2-chloropyridin-3-yl

Me

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

2-3223

phenyl

Me

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

2-3243

3-cyanophenyl

Me

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

2-3244

4-cyanophenyl

Me

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

2-3259

2-chloropyridin-3-yl

Me

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

2-3301

phenyl

Me

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

2-3321

3-cyanophenyl

Me

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

2-3322

4-cyanophenyl

Me

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

2-3337

2-chloropyridin-3-yl

Me

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

2-3379

phenyl

Me

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

2-3399

3-cyanophenyl

Me

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

2-3400

4-cyanophenyl

Me

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

2-3415

2-chloropyridin-3-yl

Me

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

2-3457

phenyl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

2-3477

3-cyanophenyl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

2-3478

4-cyanophenyl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

2-3493

2-chloropyridin-3-yl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

2-3494

2-bromopyridin-3-yl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

2-3535

phenyl

Me

H

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

2-3566

2-chloropyridin-3-yl

Me

H

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

2-3591

phenyl

Me

H

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

2-3622

2-chloropyridin-3-yl

Me

H

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

2-3647

phenyl

Me

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

2-3678

2-chloropyridin-3-yl

Me

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

2-3703

phenyl

Me

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

2-3734

2-chloropyridin-3-yl

Me

H

F

Cil

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

2-3759

phenyl

Me

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

2-3779

3-cyanophenyl

Me

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

2-3780

4-cyanophenyl

Me

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

2-3795

2-chloropyridin-3-yl

Me

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

2-3827

phenyl

Me

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

2-3847

3-cyanophenyl

Me

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

2-3848

4-cyanophenyl

Me

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

2-3863

2-chloropyridin-3-yl

Me

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 3

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

3-1

phenyl

H

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-21

3-cyanophenyl

H

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-22

4-cyanophenyl

H

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-37

2-chloropyridin-3-yl

H

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-79

phenyl

H

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-99

3-cyanophenyl

H

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-100

4-cyanophenyl

H

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-115

2-chloropyridin-3-yl

H

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-157

phenyl

H

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

3-177

3-cyanophenyl

H

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

3-178

4-cyanophenyl

H

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

3-193

2-chloropyridin-3-yl

H

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

3-235

phenyl

H

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-255

3-cyanophenyl

H

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-256

4-cyanophenyl

H

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-271

2-chloropyridin-3-yl

H

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-313

phenyl

H

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

3-333

3-cyanophenyl

H

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

3-334

4-cyanophenyl

H

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

OC2F5

3-349

2-chloropyridin-3-yl

H

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

3-391

phenyl

H

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

3-411

3-cyanophenyl

H

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

3-412

4-cyanophenyl

H

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

3-427

2-chloropyridin-3-yl

H

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

3-469

phenyl

H

Me

H

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

3-470

phenyl

H

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

3-484

(3-trifluoromethyl) phenyl

H

Et

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

3-490

3-cyanophenyl

H

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

3-491

4-cyanophenyl

H

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

3-495

2-chloro-4-fluorophenyl

H

n-Pr

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

3-506

2-chloropyridin-3-yl

H

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

3-512

6-fluoropyridin-3-yl

H

i-Pr

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

3-528

4-bromopyridin-3-yl

H

CH2CH═CH2

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

3-535

pyridin-4-yl

H

CN

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

3-548

phenyl

H

Me

H

CN

H

H

F

H

nonafiuoro-2-butyl

H

CF3

3-549

phenyl

H

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-556

2-bromophenyl

H

CH2C≡CH

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-563

(3-trifluoromethyl) phenyl

H

NH2

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-569

3-cyanophenyl

H

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-570

4-cyanophenyl

H

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-576

4-bromo-2-chlorophenyl

H

C(O)OMe

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-585

2-chloropyridin-3-yl

H

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-596

6-nitropyridin-3-yl

H

C(O)OEt

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-607

4-bromopyridin-3-yl

H

C(O)C(O)Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-610

4-nitropyridin-3-yl

H

C(O)C(O)Et

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

3-623

4-bromopyridin-2-yl

H

C(O)Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-625

6-chloropyridin-2-yl

H

C(O)Et

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-627

phenyl

H

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-641

(3-trifluoromethyl) phenyl

H

S(O)2Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-647

3-cyanophenyl

H

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-648

4-cyanophenyl

H

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-659

4-cyano-2-fluorophenyl

H

S(O)2Et

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-663

2-chloropyridin-3-yl

H

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-674

6-nitropyridin-3-yl

H

CH2Ph

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-688

4-nitropyridin-3-yl

H

CH2(3-Py)

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-702

5-iodopyridin-2-yl

H

CH2(3-Py—N-

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

3-705

phenyl

H

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

3-725

3-cyanophenyl

H

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

3-726

4-cyanophenyl

H

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

3-732

4-bromo-2-chlorophenyl

H

Et

H

CN

H

H

Br

H

nonafluoro-2-buty1

H

CF3

3-741

2-chloropyridin-3-yl

H

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

3-758

5-(trifluoromethyl) pyridin-3-yl

H

CN

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

3-783

phenyl

H

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

3-803

3-cyanophenyl

H

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

3-804

4-cyanophenyl

H

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

3-819

2-chloropyridin-3-yl

H

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

3-841

4-bromopyridin-3-yl

H

C(O)Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

3-861

phenyl

H

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

3-881

3-cyanophenyl

H

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

3-882

4-cyanophenyl

H

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

3-897

2-chloropyridin-3-yl

H

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

3-939

phenyl

H

Me

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

3-970

2-chloropyridin-3-yl

H

Me

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

3-995

phenyl

H

Me

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

3-1026

2-chloropyridin-3-yl

H

Me

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

3-1051

phenyl

H

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

3-1082

2-chloropyridin-3-yl

H

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

3-1107

phenyl

H

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

3-1138

2-chloropyridin-3-yl

H

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

3-1163

phenyl

H

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

3-1183

3-cyanophenyl

H

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

3-1184

4-cyanophenyl

H

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

3-1199

2-chloropyridin-3-yl

H

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

3-1231

phenyl

H

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

3-1251

3-cyanophenyl

H

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

C2F5

3-1252

4-cyanophenyl

H

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

3-1267

2-chloropyridin-3-yl

H

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

3-1299

phenyl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-1319

3-cyanophenyl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-1320

4-cyanophenyl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-1335

2-chloropyridin-3-yl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-1377

phenyl

H

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-1397

3-cyanophenyl

H

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-1398

4-cyanophenyl

H

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-1413

2-chloropyridin-3-yl

H

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-1455

phenyl

H

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

3-1491

2-chloropyridin-3-yl

H

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

3-1533

phenyl

H

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-1553

3-cyanophenyl

H

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-1554

4-cyanophenyl

H

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-1569

2-chloropyridin-3-yl

H

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-1611

phenyl

H

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

3-1631

3-cyanophenyl

H

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

3-1632

4-cyanophenyl

H

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

3-1647

2-chloropyridin-3-yl

H

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

3-1689

phenyl

H

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

3-1709

3-cyanophenyl

H

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

3-1710

4-cyanophenyl

H

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

3-1725

2-chloropyridin-3-yl

H

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

3-1767

phenyl

H

Me

F

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

3-1768

phenyl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

3-1788

3-cyanophenyl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

3-1789

4-cyanophenyl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

3-1804

2-chloropyridin-3-yl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

3-1846

phenyl

H

Me

F

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

3-1847

phenyl

H

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-1867

3-cyanophenyl

H

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-1868

4-cyanophenyl

H

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-1883

2-chloropyridin-3-yl

H

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-1925

phenyl

H

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-1945

3-cyanophenyl

H

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-1946

4-cyanophenyl

H

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-1961

2-chloropyridin-3-yl

H

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

3-2003

phenyl

H

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

3-2023

3-cyanophenyl

H

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

3-2024

4-cyanophenyl

H

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

3-2039

2-chloropyridin-3-yl

H

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

3-2081

phenyl

H

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

3-2101

3-cyanophenyl

H

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

3-2102

4-cyanophenyl

H

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

3-2117

2-chloropyridin-3-yl

H

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

3-2159

phenyl

H

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

3-2179

3-cyanophenyl

H

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

3-2180

4-cyanophenyl

H

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

3-2195

2-chloropyridin-3-yl

H

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

3-2237

phenyl

H

Me

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

3-2268

2-chloropyridin-3-yl

H

Me

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

3-2293

phenyl

H

Me

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

3-2324

2-chloropyridin-3-yl

H

Me

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

3-2349

phenyl

H

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

3-2380

2-chloropyridin-3-yl

H

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

3-2405

phenyl

H

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

3-2436

2-chloropyridin-3-yl

H

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

3-2461

phenyl

H

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

3-2481

3-cyanophenyl

H

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

3-2482

4-cyanophenyl

H

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

3-2497

2-chloropyridin-3-yl

H

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

3-2529

phenyl

H

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

3-2549

3-cyanophenyl

H

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

3-2550

4-cyanophenyl

H

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

3-2565

2-chloropyridin-3-yl

H

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

3-2597

phenyl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-2617

3-cyanophenyl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-2618

4-cyanophenyl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-2633

2-chloropyridin-3-yl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

3-2675

phenyl

H

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-2695

3-cyanophenyl

H

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-2696

4-cyanophenyl

H

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-2711

2-chloropyridin-3-yl

H

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

3-2753

phenyl

H

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

3-2773

3-cyanophenyl

H

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

3-2774

4-cyanophenyl

H

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

3-2789

2-chloropyridin-3-yl

H

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

3-2831

phenyl

H

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-2851

3-cyanophenyl

H

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-2852

4-cyanophenyl

H

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-2867

2-chloropyridin-3-yl

H

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

3-2909

phenyl

H

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

3-2929

3-cyanophenyl

H

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

3-2930

4-cyanophenyl

H

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

3-2945

2-chloropyridin-3-yl

H

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

3-2987

phenyl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

3-2988

2-flurophenyl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

3-3007

3-cyanophenyl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

3-3008

4-cyanophenyl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

3-3023

2-chloropyridin-3-yl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

3-3065

phenyl

H

Me

F

CN

F

H

F

H

heptafluoroisopropyl

H

CF3

3-3066

phenyl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

3-3086

3-cyanophenyl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

3-3087

4-cyanophenyl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

3-3102

2-chloropyridin-3-yl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

3-3144

phenyl

H

Me

F

CN

F

H

F

H

nonafluoro-2-butyl

H

CF3

3-3145

phenyl

H

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-3165

3-cyanophenyl

H

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-3166

4-cyanophenyl

H

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-3181

2-chloropyridin-3-yl

H

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

3-3223

phenyl

H

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

3-3243

3-cyanophenyl

H

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

3-3244

4-cyanophenyl

H

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

3-3259

2-chloropyridin-3-yl

H

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

3-3301

phenyl

H

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

3-3321

3-cyanophenyl

H

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

3-3322

4-cyanophenyl

H

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

3-3337

2-chloropyridin-3-yl

H

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

3-3379

phenyl

H

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

3-3399

3-cyanophenyl

H

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

3-3400

4-cyanophenyl

H

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

3-3415

2-chloropyridin-3-yl

H

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

3-3457

phenyl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

3-3477

3-cyanophenyl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

3-3478

4-cyanophenyl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

3-3493

2-chloropyridin-3-yl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

3-3535

phenyl

H

Me

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

3-3566

2-chloropyridin-3-yl

H

Me

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

3-3591

phenyl

H

Me

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

3-3622

2-chloropyridin-3-yl

H

Me

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

3-3647

phenyl

H

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

3-3678

2-chloropyridin-3-yl

H

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

3-3703

phenyl

H

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

3-3734

2-chloropyridin-3-yl

H

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

3-3759

phenyl

H

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

3-3779

3-cyanophenyl

H

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

3-3780

4-cyanophenyl

H

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

3-3795

2-chloropyridin-3-yl

H

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

TABLE 4

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

4-1

phenyl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

4-21

3-cyanophenyl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

4-22

4-cyanophenyl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

4-37

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

4-79

phenyl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

4-99

3-cyanophenyl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

4-100

4-cyanophenyl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

4-115

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

4-157

phenyl

Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

4-177

3-cyanophenyl

Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

4-178

4-cyanophenyl

Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

4-193

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

4-235

phenyl

Me

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

4-255

3-cyanophenyl

Me

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

4-256

4-cyanophenyl

Me

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

4-271

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

4-313

phenyl

Me

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

4-314

2-fluorophenyl

Me

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

OOF3

4-333

3-cyanophenyl

Me

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

4-334

4-cyanophenyl

Me

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

4-349

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

I

H

heptaftuoroisopropyl

H

OCF3

4-391

phenyl

Me

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

4-392

2-fluorophenyl

Me

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

4-411

3-cyanophenyl

Me

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

4-412

4-cyanophenyl

Me

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

4-427

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

4-665

phenyl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-666

(3-trifluoromethyl) phenyl

Et

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-667

(4-trifluoromethyl) phenyl

Me

Et

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-671

2-cyanophenyl

Me

Me

H

CN

H

H

Cl

H

pentafluoroethyl

H

C2F5

4-672

3-cyanophenyl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-673

4-cyanophenyl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-676

2,4-dichlorophenyl

Me

Me

H

CN

H

H

Cl

H

heptafluorosopropyl

H

C2F5

4-677

2-chloro-4-fluorophenyl

n-Pr

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-680

2-bromo-4-chlorophenyl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

4-681

2-bromo-4-fluorophenyl

Me

n-Pr

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-687

2-fluoropyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

4-688

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-692

2-nitropyridin-3-yl

Me

i-Pr

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-694

6-fluoropyridin-3-yl

i-Pr

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-701

5-fluoropyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

4-703

5-bromopyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

4-704

5-iodopyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

4-706

5-nitropyridin-3-yl

Me

CH2CH═CH2

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

4-708

5-fluoropyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

4-710

4-bromopyridin-3-yl

CH2CH═CH2

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

4-711

4-iodopyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

4-717

pyridin-4-yl

CN

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-724

pyridin-2-yl

Me

CN

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-729

4-cyanopyridin-2-yl

Me

Me

H

CN

H

H

Cl

H

pentafluoroethyl

H

CF3

4-730

phenyl

Me

Me

H

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

4-731

phenyl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-732

2-fluorophenyl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-739

3-bromophenyl

CH2C≡CH

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-744

(2-trifluoromethyl) phenyl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

4-745

(3-trifluoromethyl) phenyl

Me

CH2C≡CH

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-746

(4-trifluoromethyl) phenyl

NH2

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-750

2-cyanophenyl

Me

NH2

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-751

3-cyanophenyl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-752

4-cyanophenyl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-759

2-bromo-4-chlorophenyl

C(O)OMe

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-761

2-chloro-4-nitrophenyl

Me

C(O)OMe

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

4-767

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-773

6-fluoropyridin-3-yl

Me

C(O)OEt

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-780

5-fluoropyridin-3-yl

C(O)OEt

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

4-781

5-chloropyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-782

5-bromopyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

4-783

5-iodopyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

i-C357

4-785

5-nitropyridin-3-yl

Me

C(O)C(O)Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-787

4-fluoropyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

4-789

4-bromopyridin-3-yl

C(O)C(O)Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-790

4-iodopyridin-3-yl

Me

C(O)C(O)Et

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-791

4-(trifluoromethyl) pyridin-3-yl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

4-792

4-nitropyridin-3-yl

C(O)C(O)Et

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

4-803

pyridin-2-yl

Me

C(O)Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-805

4-bromopyridin-2-yl

Me

C(O)Et

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-806

5-iodopyridin-2-yl

C(O)Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-808

4-cyanopyridin-2-yl

C(O)Et

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

4-809

phenyl

Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-823

(3-trifluoromethyl) phenyl

S(O)2Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-828

2-cyanophenyl

Me

S(O)2Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-829

3-cyanophenyl

Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-830

4-cyanophenyl

Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-839

2-chloro-4-nitrophenyl

Me

S(O)2Et

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-841

4-cyano-2-fluorophenyl

S(O)2Et

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-845

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-853

6-bromopyridin-3-yl

Me

CH2Ph

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-855

6-(trifluoromethyl) pyridin-3-yl

Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-856

6-nitropyridin-3-yl

CH2Ph

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-863

5-nitropyridin-3-yl

Me

CH2(3-Py)

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-865

4-fluoropyridin-3-yl

CH2(3-Py)

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-883

4-bromopyridin-2-yl

Me

CH2(3-Py—N-

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

4-886

4-cyanopyridin-2-yl

CH2(3-Py—N-

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

4-887

phenyl

Me

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

4-907

3-cyanophenyl

Me

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

4-908

4-cyanophenyl

Me

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

4-923

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

4-965

phenyl

Me

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

4-985

3-cyanophenyl

Me

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

4-986

4-cyanophenyl

Me

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

4-1001

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

4-1043

phenyl

Me

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1063

3-cyanophenyl

Me

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1064

4-cyanophenyl

Me

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1079

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1121

phenyl

Et

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1122

phenyl

Et

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1123

phenyl

Et

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1124

phenyl

Et

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1125

phenyl

Et

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1126

phenyl

Et

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1127

phenyl

Et

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1128

phenyl

Et

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1129

phenyl

Et

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1130

phenyl

Et

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1131

phenyl

Et

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1132

phenyl

Et

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1133

phenyl

Et

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1134

phenyl

Et

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1135

phenyl

n-Pr

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1136

phenyl

n-Pr

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1137

phenyl

n-Pr

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1138

phenyl

n-Pr

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1139

phenyl

n-Pr

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1140

phenyl

n-Pr

CH2C≡OH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1141

phenyl

n-Pr

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1142

phenyl

n-Pr

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1143

phenyl

n-Pr

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1144

phenyl

n-Pr

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1145

phenyl

n-Pr

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1146

phenyl

n-Pr

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1147

phenyl

n-Pr

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1148

phenyl

n-Pr

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1149

phenyl

i-Pr

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1150

phenyl

i-Pr

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1151

phenyl

i-Pr

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1152

phenyl

i-Pr

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1153

phenyl

i-Pr

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1154

phenyl

i-Pr

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1155

phenyl

i-Pr

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1156

phenyl

i-Pr

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1157

phenyl

i-Pr

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1158

phenyl

i-Pr

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1159

phenyl

i-Pr

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1160

phenyl

i-Pr

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1161

phenyl

i-Pr

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1162

phenyl

i-Pr

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1163

phenyl

CH2CH═CH2

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1164

phenyl

CH2CH═CH2

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1165

phenyl

CH2CH═CH2

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1166

phenyl

CH2CH═CH2

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1167

phenyl

CH2CH═CH2

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1168

phenyl

CH2CH═CH2

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1169

phenyl

CH2CH═CH2

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1170

phenyl

CH2CH═CH2

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1171

phenyl

CH2CH═CH2

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1172

phenyl

CH2CH═CH2

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1173

phenyl

CH2CH═CH2

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1174

phenyl

CH2CH═CH2

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1175

phenyl

CH2CH═CH2

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1176

phenyl

CH2CH═CH2

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1177

phenyl

CN

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1178

phenyl

CN

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1179

phenyl

CN

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1180

phenyl

CN

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1181

phenyl

CN

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1182

phenyl

CN

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1183

phenyl

CN

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1184

phenyl

CN

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1185

phenyl

CN

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1186

phenyl

CN

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1187

phenyl

CN

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1188

phenyl

CN

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1189

phenyl

CN

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1190

phenyl

CN

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1191

phenyl

CH2C≡CH

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1192

phenyl

CH2C≡CH

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1193

phenyl

CH2C≡CH

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1194

phenyl

CH2C≡CH

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1195

phenyl

CH2C≡CH

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1196

phenyl

CH2C≡CH

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1197

phenyl

CH2C≡CH

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1198

phenyl

CH2C≡CH

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1199

phenyl

CH2C≡CH

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1200

phenyl

CH2C≡CH

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1201

phenyl

CH2C≡CH

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1202

phenyl

CH2C≡CH

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1203

phenyl

CH2C≡CH

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1204

phenyl

CH2C≡CH

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1205

phenyl

NH2

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1206

phenyl

NH2

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1207

phenyl

NH2

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1208

phenyl

NH2

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1209

phenyl

NH2

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1210

phenyl

NH2

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1211

phenyl

NH2

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1212

phenyl

NH2

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1213

phenyl

NH2

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1214

phenyl

NH2

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1215

phenyl

NH2

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1216

phenyl

NH2

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1217

phenyl

NH2

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1218

phenyl

NH2

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1219

phenyl

C(O)OMe

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1220

phenyl

C(O)OMe

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1221

phenyl

C(O)OMe

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1222

phenyl

C(O)OMe

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1223

phenyl

C(O)OMe

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1224

phenyl

C(O)OMe

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1225

phenyl

C(O)OMe

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1226

phenyl

C(O)OMe

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1227

phenyl

C(O)OMe

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1228

phenyl

C(O)OMe

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1229

phenyl

C(O)OMe

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1230

phenyl

C(O)OMe

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1231

phenyl

C(O)OMe

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1232

phenyl

C(O)OMe

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1233

phenyl

C(O)C(O)OMe

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1234

phenyl

C(O)C(O)OMe

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1235

phenyl

C(O)C(O)OMe

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1236

phenyl

C(O)C(O)OMe

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1237

phenyl

C(O)C(O)OMe

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1238

phenyl

C(O)C(O)OMe

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1239

phenyl

C(O)C(O)OMe

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1240

phenyl

C(O)C(O)OMe

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1241

phenyl

C(O)C(O)OMe

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1242

phenyl

C(O)C(O)OMe

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1243

phenyl

C(O)C(O)OMe

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1244

phenyl

C(O)C(O)OMe

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1245

phenyl

C(O)C(O)OMe

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1246

phenyl

C(O)C(O)OMe

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1247

phenyl

C(O)Me

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1248

phenyl

C(O)Me

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1249

phenyl

C(O)Me

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1250

phenyl

C(O)Me

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1251

phenyl

C(O)Me

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1252

phenyl

C(O)Me

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1253

phenyl

C(O)Me

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1254

phenyl

C(O)Me

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1255

phenyl

C(O)Me

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1256

phenyl

C(O)Me

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1257

phenyl

C(O)Me

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1258

phenyl

C(O)Me

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1259

phenyl

C(O)Me

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1260

phenyl

C(O)Me

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1261

phenyl

S(O)2Me

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1262

phenyl

S(O)2Me

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1263

phenyl

S(O)2Me

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1264

phenyl

S(O)2Me

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1265

phenyl

S(O)2Me

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1266

phenyl

S(O)2Me

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1267

phenyl

S(O)2Me

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1268

phenyl

S(O)2Me

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1269

phenyl

S(O)2Me

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1270

phenyl

S(O)2Me

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1271

phenyl

S(O)2Me

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1272

phenyl

S(O)2Me

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1273

phenyl

S(O)2Me

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1274

phenyl

S(O)2Me

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1275

phenyl

CH2Ph

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1276

phenyl

CH2Ph

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1277

phenyl

CH2Ph

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1278

phenyl

CH2Ph

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1279

phenyl

CH2Ph

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1280

phenyl

CH2Ph

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1281

phenyl

CH2Ph

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1282

phenyl

CH2Ph

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1283

phenyl

CH2Ph

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1284

phenyl

CH2Ph

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1285

phenyl

CH2Ph

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1286

phenyl

CH2Ph

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1287

phenyl

CH2Ph

CH2(3-Py)

H

CN

H

H

I

H

nonaftuoro-2-butyl

H

CF3

4-1288

phenyl

CH2Ph

CH2(3-Py—N

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1289

phenyl

CH2(3-Py)

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1290

phenyl

CH2(3-Py)

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1291

phenyl

CH2(3-Py)

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1292

phenyl

CH2(3-Py)

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1293

phenyl

CH2(3-Py)

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1294

phenyl

CH2(3-Py)

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1295

phenyl

CH2(3-Py)

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1296

phenyl

CH2(3-Py)

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1297

phenyl

CH2(3-Py)

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1298

phenyl

CH2(3-Py)

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1299

phenyl

CH2(3-Py)

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1300

phenyl

CH2(3-Py)

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1301

phenyl

CH2(3-Py)

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-1302

phenyl

CH2(3-Py)

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1303

phenyl

CH2(3-Py—N-

Et

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1304

phenyl

CH2(3-Py—N-

n-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1305

phenyl

CH2(3-Py—N-

i-Pr

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1306

phenyl

CH2(3-Py—N-

CH2CH═CH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1307

phenyl

CH2(3-Py—N-

CN

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1308

phenyl

CH2(3-Py—N-

CH2C≡CH

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1309

phenyl

CH2(3-Py—N-

NH2

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1310

phenyl

CH2(3-Py—N-

C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1311

phenyl

CH2(3-Py—N-

C(O)C(O)OMe

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1312

phenyl

CH2(3-Py—N-

C(O)Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1313

phenyl

CH2(3-Py—N-

S(O)2Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1314

phenyl

CH2(3-Py—N-

CH2Ph

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1315

phenyl

CH2(3-Py—N-

CH2(3-Py)

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

4-1316

phenyl

CH2(3-Py—N-

CH2(3-Py—N-

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

oxide)

4-1317

phenyl

Me

Me

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

4-1348

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

4-1373

phenyl

Me

Me

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

4-1404

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

4-1429

phenyl

Me

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

4-1460

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

4-1485

phenyl

Me

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

4-1516

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

4-1541

phenyl

Me

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

4-1561

3-cyanophenyl

Me

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

4-1562

4-cyanophenyl

Me

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

4-1577

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

4-1609

phenyl

Me

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

4-1629

3-cyanophenyl

Me

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

4-1630

4-cyanophenyl

Me

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

4-1645

2-chloropyridin-3-yl

Me

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

4-1873

phenyl

Me

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

4-1893

3-cyanophenyl

Me

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

4-1909

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

4-1951

phenyl

Me

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

4-1971

3-cyanophenyl

Me

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

4-1972

4-cyanophenyl

Me

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

4-1987

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

4-2029

phenyl

Me

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

4-2049

3-cyanophenyl

Me

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

4-2050

4-cyanophenyl

Me

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

4-2065

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

4-2107

phenyl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

4-2127

3-cyanophenyl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

4-2128

4-cyanophenyl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-buty1

H

OCF3

4-2143

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

4-2185

phenyl

Me

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

4-2205

3-cyanophenyl

Me

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

4-2206

4-cyanophenyl

Me

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

4-2221

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

4-2263

phenyl

Me

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

4-2283

3-cyanophenyl

Me

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

4-2284

4-cyanophenyl

Me

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

4-2299

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

4-2537

phenyl

Me

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-2538

phenyl

Et

Me

F

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

4-2544

3-cyanophenyl

Me

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-2545

4-cyanophenyl

Me

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-2560

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

4-2602

phenyl

Me

Me

F

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

4-2603

phenyl

Me

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-2623

3-cyanophenyl

Me

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-2624

4-cyanophenyl

Me

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-2639

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-2681

phenyl

Me

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-2701

3-cyanophenyl

Me

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-2702

4-cyanophenyl

Me

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-2717

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

4-2759

phenyl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

4-2779

3-cyanophenyl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

4-2780

4-cyanophenyl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

4-2795

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

4-2837

phenyl

Me

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

4-2857

3-cyanophenyl

Me

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

4-2858

4-cyanophenyl

Me

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

4-2873

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

4-2915

phenyl

Me

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-2935

3-cyanophenyl

Me

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-2936

4-cyanophenyl

Me

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-2951

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

4-3189

phenyl

Me

Me

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

4-3220

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

4-3245

phenyl

Me

Me

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

4-3276

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

4-3301

phenyl

Me

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

4-3332

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

4-3357

phenyl

Me

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

4-3388

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

4-3413

phenyl

Me

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

4-3433

3-cyanophenyl

Me

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

4-3434

4-cyanophenyl

Me

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

4-3449

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

4-3481

phenyl

Me

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

4-3493

4-iodophenyl

Me

Me

F

CN

H

H

C2F5

H

nonafluoro-2-butyl

H

CF3

4-3501

3-cyanophenyl

Me

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

4-3502

4-cyanophenyl

Me

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

4-3517

2-chloropyridin-3-yl

Me

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

4-3745

phenyl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

4-3765

3-cyanophenyl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

4-3766

4-cyanophenyl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

4-3781

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

4-3823

phenyl

Me

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

4-3843

3-cyanophenyl

Me

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

FI

OCF3

4-3844

4-cyanophenyl

Me

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

4-3859

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

4-3901

phenyl

Me

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

4-3921

3-cyanophenyl

Me

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

4-3922

4-cyanophenyl

Me

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

4-3937

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

4-3979

phenyl

Me

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

4-3999

3-cyanophenyl

Me

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

4-4000

4-cyanophenyl

Me

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

4-4015

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

4-4057

phenyl

Me

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

4-4077

3-cyanophenyl

Me

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

4-4078

4-cyanophenyl

Me

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

4-4093

2-chloropyridin-3-y1

Me

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

4-4135

phenyl

Me

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

4-4155

3-cyanophenyl

Me

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

4-4156

4-cyanophenyl

Me

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

4-4171

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

4-4409

phenyl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

4-4410

phenyl

Et

Me

F

CN

F

H

F

H

heptafluoroisopropyl

H

CF3

4-4416

3-cyanophenyl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

4-4417

4-cyanophenyl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

4-4432

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

4-4474

phenyl

Me

Me

F

CN

F

H

F

H

nonafluoro-2-butyl

H

CF3

4-4475

phenyl

Me

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-4495

3-cyanophenyl

Me

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-4496

4-cyanophenyl

Me

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-4511

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

4-4553

phenyl

Me

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

4-4573

3-cyanophenyl

Me

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

4-4574

4-cyanophenyl

Me

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

4-4589

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

4-4631

phenyl

Me

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

4-4651

3-cyanophenyl

Me

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

4-4652

4-cyanophenyl

Me

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

4-4667

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

4-4709

phenyl

Me

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

4-4729

3-cyanophenyl

Me

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

4-4730

4-cyanophenyl

Me

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

4-4745

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

4-4787

phenyl

Me

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

4-4807

3-cyanophenyl

Me

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

4-4808

4-cyanophenyl

Me

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

4-4823

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

4-5061

phenyl

Me

Me

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

4-5092

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

4-5117

phenyl

Me

Me

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

4-5148

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

4-5173

phenyl

Me

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

4-5204

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

4-5229

phenyl

Me

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

4-5260

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

4-5285

phenyl

Me

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

4-5305

3-cyanophenyl

Me

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

4-5306

4-cyanophenyl

Me

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

4-5321

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

4-5353

phenyl

Me

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

4-5373

3-cyanophenyl

Me

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

4-5374

4-cyanophenyl

Me

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

4-5389

2-chloropyridin-3-yl

Me

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 5

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

5-9

3-bromophenyl

H

Et

H

CN

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

5-39

2-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

5-144

phenyl

H

H

H

CN

H

H

Cl

F

heptafluoroisopropyl

H

CF3

5-145

2-fluorophenyl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

F

CF3

5-146

3-fluorophenyl

H

Me

H

CN

H

H

Cl

Cl

heptafluoroisopropyl

H

CF3

5-147

4-fluorophenyl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

Cl

CF3

5-148

2-chlorophenyl

H

H

H

CN

H

H

F

Br

heptafluoroisopropyl

H

CF3

5-149

3-chlorophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

Br

CF3

5-150

4-chlorophenyl

Et

H

H

CN

H

H

Cl

I

heptafluorolsopropyl

H

C2F5

5-151

2-bromophenyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

I

CF3

5-152

3-bromophenyl

H

Et

H

CN

H

H

Cl

F

heptafluoroisopropyl

F

CF3

5-153

4-bromophenyl

H

H

H

CN

H

H

Cl

F

heptafluoroisopropyl

Cl

CF3

5-154

2-iodophenyl

H

H

H

CN

H

H

Cl

F

heptafluoroisopropyl

Br

CF3

5-155

3-iodophenyl

Et

Et

H

CN

H

H

Cl

F

pentafluoroethyl

I

C2F5

5-156

4-iodophenyl

H

H

H

CN

H

H

Cl

Cl

pentafluoroethyl

F

CF3

5-157

(2-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

Cl

heptafluoroisopropyl

Cl

CF3

5-158

(3-fluoromethyl) phenyl

n-Pr

H

H

CN

H

H

Cl

Cl

heptafluoroisopropyl

Br

CF3

6-159

(4-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

Cl

heptafluoroisopropyl

I

n-C3F7

5-160

2-nitrophenyl

H

n-Pr

H

CN

H

H

Cl

Br

heptafluoroisopropyl

F

CF3

5-161

3-nitrophenyl

H

H

H

CN

H

H

Cl

Br

heptafluoroisopropyl

Cl

CF3

5-162

4-nitrophenyl

H

H

H

CN

H

H

Cl

Br

heptafluoroisopropyl

Br

CF3

5-163

2-cyanophenyl

n-Pr

n-Pr

H

CN

H

H

Cl

Br

pentafluoroethyl

I

CF3

5-164

3-cyanophenyl

H

H

H

CN

H

H

F

I

nonefluoro-2-butyl

F

CF3

5-165

4-cyanophenyl

H

H

H

CN

H

H

Cl

I

nonafluoro-2-butyl

Cl

CF3

6-166

2,6-difluorophenyl

H

H

H

CN

H

H

Cl

I

nonafluoro-2-butyl

Br

CF3

5-167

3,4-dichlorophenyl

H

H

H

CN

H

H

Cl

I

nonafluoro-2-butyl

I

CF3

5-168

2,4-dichlorophenyl

H

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

5-169

2-chloro-4-fluorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

5-170

2-chloro-4,5-difluorophenyl

i-Pr

H

H

CN

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

5-171

4-bromo-2-chlorophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

5-172

2-bromo-4-chlorophenyl

H

H

H

CN

H

H

Cl

n-Pr

nonafluoro-2-butyl

H

CF3

5-173

2-bromo-4-fluorophenyl

H

i-Pr

H

CN

H

H

Cl

H

nonafluoro-2-butyl

n-Pr

CF3

5-174

2-chloro-4-nitrophened

i-Pr

i-Pr

H

CN

H

H

Cl

1-Pr

nonafluoro-2-butyl

H

CF3

5-175

3,5-dicyanophenyl

H

H

H

CN

H

H

Cl

H

nonefluoro-2-butyl

i-Pr

CF3

5-176

4-cyano-2-fluorophenyl

H

H

H

CN

H

H

Cl

n-Bu

nonafluoro-2-butyl

H

CF3

5-177

2-chloro-4-cyanophenyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

n-Bu

CF3

5-178

pyridin-3-yl

H

H

H

CN

H

H

Cl

i-Bu

nonafluoro-2-butyl

H

CF3

5-179

2-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

i-Bu

CF3

5-180

2-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

s-Bu

nonafluoro-2-butyl

H

C2F5

5-181

2-bromopyridin-3-yl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

s-Bu

CF3

5-182

2-iodopyridin-3-yl

H

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

5-183

2-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

5-184

2-nitropyridin-3-yl

C(O)Me

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

n-Pr

CF3

5-185

2-cyanopyridin-3-yl

H

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

i-Pr

CF3

5-186

6-fluoropyridin-3-yl

H

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

n-Bu

CF3

5-187

6-chloropyridin-3-yl

H

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

i-Bu

CF3

5-188

6-bromopyridin-3-yl

H

C(O)Me

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

s-Bu

CF3

5-189

6-iodopyridin-3-yl

H

H

H

CN

H

H

Br

Et

nonafluoro-2-butyl

Me

n-C3F7

5-190

6-(trifluoromethyl)pyridin-3-yl

H

H

H

CN

H

H

Br

Et

nonafluoro-2-butyl

Et

i-C3F7

5-191

6-nitropyridin-3-yl

C(O)Me

C(O)Me

H

CN

H

H

Br

Et

nonafluoro-2-butyl

n-Pr

CF3

5-192

6-cyanopyridin-3-yl

H

H

H

CN

H

H

Br

Et

nonafluoro-2-butyl

i-Pr

CF3

5-193

phenyl

H

H

H

CN

H

H

Br

Et

heptafluoroisopropyl

n-Bu

CF3

5-194

5-fluoropyridin-3-yl

H

H

H

CN

H

H

Br

Et

heptafluoroisopropyl

i-Bu

CF3

5-195

5-chloropyridin-3-yl

H

H

H

CN

H

H

Br

Et

heptafluoroisopropyl

s-Bu

CF3

5-196

5-bromopyridin-3-yl

H

H

H

CN

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

5-197

5-iodopyridin-3-yl

H

H

H

CN

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

5-198

5-(trifluoromethyl) pyridin-3-yl

Me

Et

H

CN

H

H

Br

n-Pr

pentafluoroethyl

n-Pr

CF3

5-199

5-nitropyridin-3-yl

H

H

H

CN

H

H

Br

n-Pr

heptafluoroisopropyl

i-Pr

CF3

5-200

5-cyanopyridin-3-yl

H

H

H

CN

H

H

Br

n-Pr

pentafluoroethyl

n-Bu

CF3

5-201

4-fluoropyridin-3-yl

H

H

H

CN

H

H

Br

n-Pr

heptafluoroisopropyl

i-Bu

CF3

5-202

4-chloropyridin-3-yl

H

H

H

CN

H

H

Br

n-Pr

heptafluoroisopropyl

s-Bu

CF3

5-203

4-bromopyridin-3-yl

Me

n-Pr

H

CN

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

5-204

4-iodopyridin-3-yl

H

H

H

CN

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

5-205

4-(fluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

i-Pr

heptafluoroisopropyl

n-Pr

CF3

5-206

4-nitropyridin-3-yl

H

H

H

CN

H

H

Br

1-Pr

heptafluoroisopropyl

i-Pr

CF3

5-207

4-cyanopyridin-3-yl

H

H

H

CN

H

H

Br

i-Pr

heptafluoroisopropyl

n-Bu

CF3

5-208

2,6-dichloropyridin-3-yl

H

H

H

CN

H

H

Br

i-Pr

heptafluoroisopropyl

i-Bu

CF3

5-209

pyridin-3-yl N-oxide

Me

i-Pr

H

CN

H

H

Br

i-Pr

heptafluoroisopropyl

s-Bu

CF3

5-210

pyridin-4-yl

H

H

H

CN

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

5-211

2-chloropyridin-4-yl

H

H

H

CN

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

5-212

3-bromopyridin-4-yl

H

H

H

CN

H

H

Br

n-Bu

heptafluoroisopropyl

n-Pr

CF3

5-213

3,5-dichloropyridin-4-yl

H

H

H

CN

H

H

Br

n-Bu

nonafluoro-2-butyl

i-Pr

CF3

5-214

3-(trifluoromethyl) pyridin-4-yl

H

H

H

CN

H

H

Br

n-Bu

nonafluoro-2-butyl

n-Bu

CF3

5-215

2,6-dicyanopyridin-4-yl

H

H

H

CN

H

H

Br

n-Bu

nonafluoro-2-butyl

i-Bu

CF3

5-216

pyridin-4-yl N-oxide

Me

C(O)Me

H

CN

H

H

Br

n-Bu

nonafluoro-2-butyl

s-Bu

CF3

5-217

pyridin-2-yl

H

H

H

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

5-218

3-chloropyridin-2-yl

H

H

H

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

5-219

4-bromopyridin-2-yl

H

H

H

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

i-Pr

CF3

5-220

5-iodopyridin-2-yl

H

H

H

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

i-Pr

CF3

5-221

6-chloropyridin-2-yl

H

H

H

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

n-Bu

CF3

5-222

4-cyanopyridin-2-yl

H

H

H

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

i-Bu

CF3

5-223

phenyl

H

H

H

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

s-Bu

C2F5

5-224

2-fluorophenyl

H

H

H

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

5-225

3-fluorophenyl

H

H

H

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

5-226

4-fluorophenyl

H

H

H

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

n-Pr

CF3

5-227

2-ohlorophenyl

H

H

H

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

i-Pr

CF3

5-228

3-chlorophenyl

H

H

H

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

n-Bu

CF3

5-229

4-chlorophenyl

H

H

H

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

i-Bu

CF3

5-230

2-bromophenyl

Et

Me

H

CN

H

H

Sr

s-Bu

nonafluoro-2-butyl

s-Bu

CF3

5-231

3-bromophenyl

H

H

H

CN

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

5-232

4-bromophenyl

H

H

H

CN

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

5-233

2-iodophenyl

H

H

H

CN

H

H

Br

F

nonafluoro-2-butyl

n-Pr

CF3

5-234

3-iodophenyl

H

H

H

CN

H

H

Br

F

nonafluoro-2-butyl

i-Pr

CF3

5-235

4-iodophenyl

H

H

H

CN

H

H

Br

F

nonafluoro-2-butyl

n-Bu

CF3

5-236

(2-trifluoromethyl) phenyl

H

H

H

CN

H

H

Br

F

nonafluoro-2-butyl

i-Bu

CF3

5-237

(3-trifluoromethyl) phenyl

Et

n-Pr

H

CN

H

H

Br

F

nonafluoro-2-butyl

s-Bu

CF3

5-238

(4-trifluoromethyl) phenyl

Et

i-Pr

H

CN

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

5-239

2-nitrophenyl

H

H

H

CN

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

5-240

phenyl

H

H

H

CN

H

H

I

Cl

pentafluoroethyl

n-Pr

i-C3F7

5-241

3-nitrophenyl

H

H

H

CN

H

H

I

Cl

heptafluoroisopropyl

i-Pr

CF3

5-242

4-nitrophenyl

H

H

H

CN

H

H

I

Cl

heptafluoroisopropyl

n-Bu

CF3

5-243

2-cyanophenyl

Et

C(O)Me

H

CN

H

H

I

Cl

heptafluoroisopropyl

i-Bu

CF3

5-244

3-cyanophenyl

H

H

H

CN

H

H

I

Cl

heptafluoroisopropyl

s-Bu

CF3

5-245

4-cyanophenyl

H

H

H

CN

H

H

I

Br

heptafluoroisopropyl

Me

CF3

5-246

2,6-difluorophenyl

H

H

H

CN

H

H

I

Br

heptafluoroisopropyl

Et

CF3

5-247

3,4-dichlorophenyl

H

H

H

CN

H

H

I

Br

pentafluoroethyl

n-Pr

CF3

5-248

2,4-dichlorophenyl

H

H

H

CN

H

H

I

Br

heptafluoroisopropyl

i-Pr

CF3

5-249

2-chloro-4-fluorophenyl

H

H

H

CN

H

H

I

Br

heptafluoroisopropyl

n-Bu

CF3

5-250

2-chloro-4,5-difluorophenyl

H

H

H

CN

H

H

I

Br

heptafluoroisopropyl

i-Bu

CF3

5-251

4-bromo-2-chlorophenyl

H

H

H

CN

H

H

I

Br

heptafluoroisopropyl

s-Bu

CF3

5-252

2-bromo-4-chlorophenyl

n-Pr

Me

H

CN

H

H

I

I

heptafluoroisopropyl

Me

CF3

5-253

2-bromo-4-fluorophenyl

H

H

H

CN

H

H

I

I

heptafluoroisopropyl

Et

CF3

5-254

2-chloro-4-nitrophenyl

n-Pr

Et

H

CN

H

H

I

I

heptafluoroisopropyl

n-Pr

CF3

5-255

3,5-dicyanophenyl

H

H

H

CN

H

H

I

I

heptafluoroisopropyl

i-Pr

CF3

5-256

4-cyano-2-fluorophenyl

H

H

H

CN

H

H

I

I

heptafluoroisopropyl

n-Bu

CF3

5-257

2-chloro-4-cyanophenyl

H

H

H

CN

H

H

I

I

heptafluoroisopropyl

i-Bu

CF3

5-258

pyridin-3-yl

H

H

H

CN

H

H

I

I

heptafluoroisopropyl

s-Bu

CF3

5-259

2-fluoropyridin-3-yl

H

H

H

CN

H

H

I

Me

heptafluoroisopropyl

F

C2F5

5-260

2-chloropyridin-3-yl

H

H

H

CN

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

5-261

2-bromopyridin-3-yl

H

H

H

CN

H

H

I

Me

nonafluoro-2-butyl

Br

n-C3F7

5-262

2-iodopyridin-3-yl

H

H

H

CN

H

H

I

Me

nonafluoro-2-butyl

I

i-C3F7

5-263

2-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

Et

nonafluoro-2-butyl

F

CF3

5-264

2-nitropyridin-3-yl

H

H

H

CN

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

5-265

2-cyanopyridin-3-yl

H

H

H

CN

H

H

I

Et

nonafluoro-2-butyl

Br

CF3

5-266

6-fluoropyridin-3-yl

n-Pr

i-Pr

H

CN

H

H

I

Et

nonafluoro-2-butyl

I

C2F5

5-267

6-chloropyridin-3-yl

H

H

H

CN

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

5-268

6-bromopyridin-3-yl

H

H

H

CN

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

5-269

6-iodopyridin-3-yl

H

H

H

CN

H

H

I

n-Pr

nonafluoro-2-butyl

Br

CF3

5-270

6-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

n-Pr

nonafluoro-2-butyl

I

n-C3F7

5-271

6-nitropyridin-3-yl

H

H

H

CN

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

5-272

6-cyanopyridin-3-yl

H

H

H

CN

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

5-273

5-fluoropyridin-3-yl

n-Pr

C(O)Me

H

CN

H

H

I

i-Pr

nonafluoro-2-butyl

Br

CF3

5-274

5-chloropyridin-yl

H

H

H

CN

H

H

I

i-Pr

nonafluoro-2-butyl

I

CF3

5-275

5-bromopyridin-3-yl

H

H

H

CN

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

5-276

5-iodopyridin-3-yl

H

H

H

CN

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

5-277

5-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

n-Bu

nonafluoro-2-butyl

Br

CF3

5-278

5-nitropyridin-3-yl

i-Pr

Me

H

CN

H

H

I

n-Bu

nonafluoro-2-butyl

I

CF3

5-279

5-cyanopyridin-3-yl

H

H

H

CN

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

5-280

4-fluoropyridin-3-yl

H

H

H

CN

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

5-281

4-chloropyridin-3-yl

H

H

H

CN

H

H

I

i-Bu

nonafluoro-2-butyl

Br

CF3

5-282

4-bromopyridin-3-yl

i-Pr

Et

H

CN

H

H

I

i-Bu

nonafluoro-2-butyl

I

CF3

5-283

4-iodopyridin-3-yl

i-Pr

n-Pr

H

CN

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

5-284

4-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

5-285

4-nitropyridin-3-yl

i-Pr

C(O)Me

H

CN

H

H

I

s-Bu

nonafluoro-2-butyl

Br

CF3

5-286

4-cyanopyridin-3-yl

H

H

H

CN

H

H

I

s-Bu

nonafluoro-2-butyl

I

CF3

5-295

3-bromophenyl

H

Et

H

CN

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

5-325

2-iodopyridin-3-yl

H

H

H

CN

H

H

OCF3

Me

nonefluoro-2-butyl

Me

OCF3

5-438

3-bromophenyl

H

Et

H

CN

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

5-468

2-iodopyridin-3-yl

H

H

H

CN

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OF3

5-581

3-bromophenyl

H

Et

H

CN

H

H

CF3

F

heptafluoroisopropyl

F

CF3

5-611

2-iodopyridin-3-yl

H

H

H

CN

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

5-724

3-bromophenyl

H

Et

F

CN

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

5-754

2-iodopyridin-3-yl

H

H

F

CN

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

5-863

2-chlorophenyl

H

H

F

CN

H

H

F

Br

heptafluoroisopropyl

H

CF3

5-869

2-iodophenyl

H

H

F

CN

H

H

Cl

F

heptafluoroisopropyl

Br

CF3

5-876

3-nitrophenyl

H

H

F

CN

H

H

Cl

Br

heptafluoroisopropyl

Cl

CF3

5-883

2,4-dichlorophenyl

H

H

F

CN

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

5-884

2-chloro-4-fluorophenyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

5-885

2-chloro-4,5-difluorophenyl

i-Pr

H

F

CN

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

5-886

4-bromo-2-chlorophenyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

5-897

2-iodopyridin-3-yl

H

H

F

CN

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

5-898

2-(trifluoromethyl) pyridin-3-yl

H

H

F

CN

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

5-904

6-iodopyridin-3-yl

H

H

F

CN

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

5-905

6-(trifluoromethyl) pyridin-3-yl

H

H

F

CN

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

5-911

5-bromopyridin-3-yl

H

H

F

CN

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

5-912

5-iodopyridin-3-yl

H

H

F

CN

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

5-918

4-bromopyridin-3yl

Me

n-Pr

F

CN

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

5-919

4-iodopyridin-3-yl

H

H

F

CN

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

5-925

pyridin-4-yl

H

H

F

CN

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

5-926

2-chloropyridin-4-yl

H

H

F

CN

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

5-932

pyridin-2-yl

H

H

F

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

5-933

3-chloropyridin-2-yl

H

H

F

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

5-939

2-fluorophenyl

H

H

F

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

5-940

3-fluorophenyl

H

H

F

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

5-946

3-bromophenyl

H

H

F

CN

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

5-947

4-bromophenyl

H

H

F

CN

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

5-953

(4-trifluoromethyl) phenyl

Et

i-Pr

F

CN

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

5-954

2-nitrophenyl

H

H

F

CN

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

5-960

4-cyanophenyl

H

H

F

CN

H

H

I

Br

heptafluoroisopropyl

Me

CF3

5-961

2,6-difluorophenyl

H

H

F

CN

H

H

I

Br

heptafluoroisopropyl

Et

CF3

5-967

2-bromo-4-chlorophenyl

n-Pr

Me

F

CN

H

H

I

I

heptafluoroisopropyl

Me

CF3

5-968

2-bromo-4-fluorophenyl

H

H

F

CN

H

H

I

I

heptafluoroisopropyl

Et

CF3

5-974

2-fluoropyridin-3-yl

H

H

F

CN

H

H

I

Me

heptafluoroisopropyl

F

C2F5

5-975

2-chloropyridin-3-yl

H

H

F

CN

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

5-978

2-(trifluoromethyl) pyridin-3-yl

H

H

F

CN

H

H

I

Et

nonafluoro-2-butyl

F

CF3

5-979

2-nitropyridin-3-yl

H

H

F

CN

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

5-982

6-chloropyridin-3-yl

H

H

F

CN

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

5-983

6-bromopyridin-3-yl

H

H

F

CN

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

5-986

6-nitropyridin-3-yl

H

H

F

CN

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

5-987

6-cyanopyridin-3-yl

H

H

F

CN

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

5-990

5-bromopyridin-3-yl

H

H

F

CN

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

5-991

5-iodopyridin-3-yl

H

H

F

CN

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

OF3

5-994

5-cyanopyridin-3-yl

H

H

F

CN

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

5-995

4-fluoropyridin-3-yl

H

H

F

CN

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

5-998

4-iodopyridin-3-yl

i-Pr

n-Pr

F

CN

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

5-999

4-(trifluoromethyl) pyridin-3-yl

H

H

F

CN

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

5-1010

3-bromophenyl

H

Et

F

CN

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

5-1040

2-iodopyridin-3-yl

H

H

F

CN

H

H

OCF3

Me

nonafluoro-2-butyl

Mn

OCF3

5-1153

3-bromophenyl

H

Et

F

CN

H

H

OCF3

F

heptatluoroisopropyl

F

CF3

5-1183

2-iodopyridin-3-yl

H

H

F

CN

H

H

OCF3

Mn

nonafluoro-2-butyl

Me

CF3

5-1296

3-bromophenyl

H

Et

F

CN

H

H

CF3

F

heptafluoroisopropyl

F

CF3

5-1326

2-iodopyridin-3-yl

H

H

F

CN

H

H

CF3

Mn

nonafluoro-2-butyl

Mn

CF3

5-1439

3-bromophenyl

H

Et

F

CN

F

H

Cl

F

heptafluoroisopropyl

F

OCF3

5-1469

2-iodopyridin-3-yl

H

H

F

CN

F

H

Cl

Mn

nonafluoro-2-butyl

Mn

OCF3

5-1576

3-fluorophenyl

H

Me

F

CN

F

H

Cl

Cl

heptafluoroisopropyl

H

CF3

5-1583

4-bromophenyl

H

H

F

CN

F

H

Cl

F

heptafluoroisopropyl

Cl

CF3

5-1591

3-nitrophenyl

H

H

F

CN

F

H

Cl

Br

heptafluoroisopropyl

Cl

CF3

5-1598

2,4-dichlorophonyl

H

H

F

CN

F

H

Cl

Me

nonafluoro-2-butyl

H

CF3

5-1599

2-chloro-4-fluorophenyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

Me

CF3

5-1600

2-chloro-4,5-difluorophenyl

i-Pr

H

F

CN

F

H

Cl

Et

nonafluoro-2-butyl

H

CF3

5-1601

4-bromo-2-chlorophenyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

Et

CF3

5-1612

2-iodopyridin-3-yl

H

H

F

CN

F

H

Cl

Mn

nonafluoro-2-butyl

Me

n-C3F7

5-1613

2-(trifluoromethyl) pyridin-3-yl

H

H

F

CN

F

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

5-1619

6-iodopyridin-3-yl

H

H

F

CN

F

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

5-1620

6-(trifluoromethyl) pyridin-3-yl

H

H

F

CN

F

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

5-1626

5-bromopyridin-3-yl

H

H

F

CN

F

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

5-1627

5-iodopyridin-3-yl

H

H

F

CN

F

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

5-1633

4-bromopyridin-3-yl

Me

n-Pr

F

CN

F

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

5-1634

4-iodopyridin-3-yl

H

H

F

CN

F

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

5-1640

pyridin-4-yl

H

H

F

CN

F

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

5-1641

2-chloropyridin-4-yl

H

H

F

CN

F

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

5-1647

pyridin-2-yl

H

H

F

CN

F

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

5-1648

3-chloropyridin-2-yl

H

H

F

CN

F

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

5-1654

2-fluorophenyl

H

H

F

CN

F

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

5-1655

3-fluorophenyl

H

H

F

CN

F

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

5-1661

3-bromophenyl

H

H

F

CN

F

H

Br

F

nonafluoro-2-butyl

Me

CF3

5-1662

4-bromophenyl

H

H

F

CN

F

H

Br

F

nonafluoro-2-butyl

Et

CF3

5-1668

(4-trifluoromethyl) phenyl

Et

i-Pr

F

CN

F

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

5-1669

2-nitrophenyl

H

H

F

CN

F

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

5-1675

4-cyanophenyl

H

H

F

CN

F

H

I

Br

heptafluoroisopropyl

Me

CF3

5-1676

2,6-difluorophenyl

H

H

F

CN

F

H

I

Br

heptafluoroisopropyl

Et

CF3

5-1682

2-bromo-4-chlorophenyl

n-Pr

Me

F

CN

F

H

I

I

heptafluoroisopropyl

Me

CF3

5-1683

2-bromo-4-fluorophenyl

H

H

F

CN

F

H

I

I

heptafluoroisopropyl

Et

CF3

5-1689

2-fluoropyridin-3-yl

H

H

F

CN

F

H

I

Me

heptafluoroisopropyl

F

C2F5

5-1690

2-chloropyridin-3-yl

H

H

F

CN

F

H

I

Me

nonafluoro-2-butyl

Cl

CF3

5-1693

2-(trifluoromethyl) pyridin-3-yl

H

H

F

CN

F

H

I

Et

nonafluoro-2-butyl

F

CF3

5-1694

2-nitropyridin-3-yl

H

H

F

CN

F

H

I

Et

nonafluoro-2-butyl

Cl

CF3

5-1697

6-chloropyridin-3-yl

H

H

F

CN

F

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

5-1698

6-bromopyridin-3-yl

H

H

F

CN

F

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

5-1701

6-nitropyridin-3-yl

H

H

F

CN

F

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

5-1702

6-cyanopyridin-3-yl

H

H

F

CN

F

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

5-1705

5-bromopyridin-3-yl

H

H

F

CN

F

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

5-1706

5-iodopyrdin-3-yl

H

H

F

CN

F

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

5-1709

5-cyanopyridin-3-yl

H

H

F

CN

F

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

5-1710

4-fluoropyridin-3-yl

H

H

F

CN

F

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

5-1713

4-iodopyridin-3-yl

i-Pr

N-Pr

F

CN

F

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

5-1714

4-(trifluoropmethyl) pyridin-3-yl

H

H

F

CN

F

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

5-1725

3-bromophenyl

H

Et

F

CN

F

H

OCF3

F

heptafluoroisopropyl

F

OCF3

5-1755

2-iodopyridin-3-yl

H

H

F

CN

F

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

5-1868

3-bromophenyl

H

Et

F

CN

F

H

OCF3

F

heptafluoroisopropyl

F

CF3

5-1898

2-iodopyridin-3-yl

H

H

F

CN

F

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

5-2011

3-bromophenyl

H

Et

F

CN

F

H

CF3

F

heptafluoroisopropyl

F

CF3

5-2041

2-iodopyridin-3-yl

H

H

F

CN

F

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

TABLE 6

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

6-1

phenyl

H

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

6-2

3-cyanophenyl

H

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

6-3

4-cyanophenyl

H

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

6-4

2-chloropyridin-3-yl

H

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

6-5

phenyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-12

3-cyanophenyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-13

4-cyanophenyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-24

2-chloropyridin-3-yl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-38

phenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-39

2-fluorophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-45

3-cyanophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-46

4-cyanophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-47

2,6-difluorophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-57

2-chloropyridin-3-yl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-60

6-chloropyridin-3-yl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-71

phenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-72

2-fluorophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-78

3-cyanophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-79

4-cyanophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-80

2,6-difluorophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-90

2-chloropyridin-3-yl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-93

6-chloropyridin-3-yl

H

H

H

H

H

H

1

H

nonafluoro-2-butyl

H

I

6-104

phenyl

H

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

Cl

6-105

phenyl

H

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

Br

6-106

phenyl

H

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

I

6-107

phenyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Br

6-108

phenyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

I

6-109

phenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

I

6-110

phenyl

H

H

H

H

H

H

F

H

heptafluoroisopropyl

H

CF3

6-111

phenyl

H

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-131

3-cyanophenyl

H

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-132

4-cyanophenyl

H

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-147

2-chloropyridin-3-yl

H

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-189

phenyl

H

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

6-190

phenyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-210

3-cyanophenyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-211

4-cyanophenyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-226

2-chloropyridin-3-yl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-268

phenyl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-269

2-fluorophenyl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-270

3-fluorophenyl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-271

4-fluorophenyl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-272

2-chlorophenyl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-288

3-cyanophenyl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-289

4-cyanophenyl

H

H

H

H

H

H

.Br

H

heptafluoroisopropyl

H

CF3

6-290

2,6-difluorophenyl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-293

2-chloro-4-fluorophenyl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-300

4-cyano-2-fluorophenyl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-304

2-chloropyridin-3-yl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-305

2-bromopyridin-3-yl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-306

2-iodopyridin-3-yl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-311

6-chloropyridin-3-yl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-346

phenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-347

2-fluorophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-348

3-fluorophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-349

4-fluorophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-366

3-cyanophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-367

4-cyanophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-368

2,6-difluorophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-382

2-chloropyridin-3-yl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-389

6-chloropyridin-3-yl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-424

phenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-425

2-fluorophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-426

3-fluorophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-427

4-fluorophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-428

2-chlorophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-444

3-cyanophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-445

4-cyanophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-446

2,6-difluorophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-448

2,4-dichlorophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-449

2-chloro-4-fluorophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-450

2-chloro-4,5-difluorophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-451

4-bromo-2-chlorophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-452

2-bromo-4-chlorophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-453

2-bromo-4-fluorophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-454

2-chloro-4-nitrophenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-460

2-chloropyridin-3-yl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-461

2-bromopyridin-3-yl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-467

6-chloropyridin-3-yl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-502

phenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-503

2-fluorophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-504

3-fluorophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-505

4-fluorophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-522

3-cyanophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-523

4-cyanophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-524

2,6-difluorophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-538

2-chloropyridin-3-yl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-545

6-chloropyridin-3-yl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-580

phenyl

H

H

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-595

3-cyanophenyl

H

H

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-596

4-cyanophenyl

H

H

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-611

2-chloropyridin-3-yl

H

H

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-636

phenyl

H

H

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-651

3-cyanophenyl

H

H

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-652

4-cyanophenyl

H

H

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-667

2-chloropyridin-3-yl

H

H

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-692

phenyl

H

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-707

3-cyanophenyl

H

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-708

4-cyanophenyl

H

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-723

2-chloropyridin-3-yl

H

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-748

phenyl

H

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-763

3-cyanophenyl

H

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-764

4-cyanophenyl

H

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-779

2-chloropyridin-3-yl

H

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-804

phenyl

H

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-824

3-cyanophenyl

H

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-825

4-cyanophenyl

H

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-840

2-chloropyridin-3-yl

H

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-841

2-bromopyridin-3-yl

H

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-872

phenyl

H

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-892

3-cyanophenyl

H

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-893

4-cyanophenyl

H

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-908

2-chloropyridin-3-yl

H

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-940

phenyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

6-941

3-cyanophenyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

6-942

4-cyanophenyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

6-943

2-chloropyridin-3-yl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

6-944

phenyl

H

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

6-945

3-cyanophenyl

H

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

6-946

4-cyanophenyl

H

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

6-947

2-chloropyridin-3-yl

H

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

6-948

phenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-952

2-chlorophenyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

Cl

6-956

3-bromophenyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

Br

6-961

(2-trifluoromethyl) phenyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

I

6-964

2-nitrophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Br

6-968

3-cyanophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-969

4-cyanophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-970

2,6-difluorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

I

6-982

pyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

I

6-984

2-chloropyridin-3-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-1026

phenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-1046

3-cyanophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-1047

4-cyanophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-1062

2-chloropyridin-3-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-1104

phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1105

2-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1106

3-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1107

4-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1124

3-cyanophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1125

4-cyanophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1126

2,6-difluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1140

2-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1147

6-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1182

phenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-1183

2-fluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-1184

3-fluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-1185

4-fluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-1202

3-cyanophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-1203

4-cyanophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-1204

2,6-difluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-1218

2-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-1225

6-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-1260

phenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1261

2-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1262

3-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1263

4-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1280

3-cyanophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1281

4-cyanophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1282

2,6-difluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1296

2-chloropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1303

6-chloropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1338

phenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-1339

2-fluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-1340

3-fluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-1341

4-fluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-1358

3-cyanophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-1359

4-cyanophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-1360

2,6-difluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-1374

2-chloropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-1381

6-chloropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-1416

phenyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

CF3

6-1417

phenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1418

2-fluorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1422

3-chlorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1426

4-bromophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1427

2-iodophenyl

H

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

6-1431

(3-trifluoromethyl) phenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1435

4-nitrophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1436

2-cyanophenyl

H

H

F

H

H

H

Cl

H

pentafluoroethyl

H

C2F5

6-1437

3-cyanophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1438

4-cyanophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1439

2,6-difluorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1440

3,4-dichlorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1441

2,4-dichlorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

6-1442

2-chloro-4-fluorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1445

2-bromo-4-chlorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

6-1446

2-bromo-4-fluorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1447

2-chloro-4-nitrophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1448

3,5-dicyanophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1449

4-cyano-2-fluorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1451

pyridin-3-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1452

2-fluoropyridin-3-yl

H

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

6-1453

2-chloropyridin-3-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1456

2-(fluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1457

2-nitropyridin-3-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

6-1460

6-chloropyridin-3-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

6-1467

5-chloropyridin-3-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1474

4-chloropyridin-3-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1480

2,6-dichloropyridin-3-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1481

pyridin-3-yl N-oxide

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1482

pyridin-4-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1483

2-chloropyridin-4-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1485

3,5-dichloropyridin-4-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1488

pyridin-4-yl N-oxide

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1489

pyridin-2-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1490

3-chloropyridin-2-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1493

6-chloropyridin-2-yl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1495

phenyl

H

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

6-1496

phenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1498

3-fluorophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1502

4-chlorophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1503

2-bromophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1507

3-iodophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1511

(4-trifluoromethyl) phenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1512

2-nitrophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1516

3-cyanophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1517

4-cyanophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1518

2,6-difluorophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1520

2,4-dichlorophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1521

2-chloro-4-fluorophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1524

2-bromo-4-chlorophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1525

2-bromo-4-fluorophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1526

2-chloro-4-nitrophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

6-1528

4-cyano-2-fluorophenyl

H

H

F

H

H

H

Cl

H

nonefluoro-2-butyl

H

CF3

6-1529

2-chloro-4-cyanophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1530

pyridin-3-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1532

2-chloropyridin-3-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1539

6-chloropyridin-3-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1545

5-fluoropyrdin-3-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

6-1552

4-fluoropyridin-3-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

6-1559

2,6-dichloropyridin-3-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1560

pyridin-3-yl N-oxide

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1561

pyridin-4-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1562

2-chloropyridin-4-yl

H

H

F

H

H

H

CI

H

nonafluoro-2-butyl

H

CF3

6-1567

pyridin-4-yl N-oxide

H

H

F

H

H

H

CI

H

nonafluoro-2-butyl

H

CF3

6-1568

pyridin-2-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1569

3-chloropyridin-2-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1572

6-chloropyridin-2-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-1574

phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1575

2-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1576

3-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1577

4-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1578

2-chlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1579

3-chlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1580

4-chlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1581

2-bromophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1582

3-bromophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1583

4-bromophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1584

2-iodophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1585

3-iodophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1586

4-iodophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1587

(2-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1588

(3-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1589

(4-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1590

2-nitrophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1591

3-nitrophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1592

4-nitrophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1593

2-cyanophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1594

3-cyanophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1595

4-cyanophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1596

2,6-difluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1597

3,4-dichlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1598

2,4-dichlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1599

2-chloro-4-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1600

2-chloro-4,5-difluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1601

4-bromo-2-chlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1602

2-bromo-4-chlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1603

2-bromo-4-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1604

2-chloro-4-nitrophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1605

3,5-dicyanophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1606

4-cyano-2-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1607

2-chloro-4-cyanophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1608

pyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1609

2-fluoropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1610

2-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1611

2-bromopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1612

2-iodopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1613

2-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1614

2-nitropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1615

2-cyanopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1616

6-fluoropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1617

6-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1618

6-bromopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1619

6-iodopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1620

6-(trifluoremethyl) pyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1621

6-nitropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1622

6-cyanopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1623

5-fluoropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1624

5-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1625

5-bromopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1626

5-iodopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1627

5-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1628

5-nitropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1629

5-cyanopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1630

4-fluoropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1631

4-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1632

4-bromopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1633

4-iodopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1634

4-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1635

4-nitropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1636

4-cyanopyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1637

2,6-dichloropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1638

pyridin-3-yl N-oxide

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1639

pyridin-4-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1640

2-chloropyridin-4-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1641

3-bromopyridin-4-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1642

3,5-dichloropyridin-4-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1643

3-(trifluoromethyl) pyridin-4-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1644

2,6-dicyanopyridin-4-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1645

pyridin-4-yl N-oxide

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1646

pyridin-2-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1647

3-chloropyridin-2-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1648

4-bromopyridin-2-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1649

5-iodopyridin-2-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1650

6-chloropyridin-2-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1651

4-cyanopyridin-2-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1652

phenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1653

2-fluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1654

3-fluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1655

4-fluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1656

2-chlorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1657

3-chlorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1658

4-chlorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1659

2-bromophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1660

3-bromophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1661

4-bromophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1662

2-iodophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1663

3-iodophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1664

4-iodophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1665

(2-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1666

(3-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1667

(4-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1668

2-nitrophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1669

3-nitrophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1670

4-nitrophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1671

2-cyanophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1672

3-cyanophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1673

4-cyanophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1674

2,6-difluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1675

3,4-dichlorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1676

2,4-dichlorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1677

2-chloro-4-fluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1678

2-chloro-4,5-difluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1679

4-bromo-2-chlorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1680

2-bromo-4-chlorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1681

2-bromo-4-fluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1682

2-chloro-4-nitrophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1683

3,5-dicyanophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1684

4-cyano-2-fluorophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1685

2-chloro-4-cyanophenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1686

pyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1687

2-fluoropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1688

2-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1689

2-bromopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1690

2-iodopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1691

2-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1692

2-nitropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1693

2-cyanopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1694

6-fluoropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1695

6-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1696

6-bromopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1697

6-iodopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1698

6-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1699

6-nitropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1700

6-cyanopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1701

5-fluoropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1702

5-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1703

5-bromopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1704

5-iodopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1705

5-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1706

5-nitropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1707

5-cyanopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1708

4-fluoropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1709

4-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1710

4-bromopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1711

4-iodopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1712

4-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1713

4-nitropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1714

4-cyanopyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1715

2,6-dichloropyridin-3-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1716

pyridin-3-yl N-oxide

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1717

pyridin-4-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1718

2-chloropyridin-4-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1719

3-bromopyridin-4-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1720

3,5-dichloropyridin-4-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1721

3-(trifluoromethyl) pyridin-4-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1722

2,6-dicyanopyridin-4-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1723

pyridin-4-yl N-oxide

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1724

pyridin-2-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1725

3-chloropyridin-2-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1726

4-bromopyridin-2-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1727

5-iodopyridin-2-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1728

6-chloropyridin-2-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1729

4-cyanopyridin-2-yl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-1730

phenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1731

2-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1732

3-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1733

4-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1734

2-chlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1735

3-chlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1736

4-chlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1737

2-bromophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1738

3-bromophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1739

4-bromophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1740

2-iodophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1741

3-iodophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1742

4-iodophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1743

(2-trifluoromethyl) phenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1744

(3-trifluoromethyl) phenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1745

(4-trifluoromethyl) phenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1746

2-nitrophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1747

3-nitrophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1748

4-nitrophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1749

2-cyanophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1750

3-cyanophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1751

4-cyanophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1752

2,6-difluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1753

3,4-dichlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1754

2,4-dichlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1755

2-chloro-4-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1756

2-chloro-4,5-difluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1757

4-bromo-2-chlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1758

2-bromo-4-chlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1759

2-bromo-4-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1760

2-chloro-4-nitrophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1761

3,5-dicyanophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1762

4-cyano-2-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1763

2-chloro-4-cyanophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1764

pyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1765

2-fluoropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1766

2-chloropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1767

2-bromopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1768

2-iodopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1769

2-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1770

2-nitropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1771

2-cyanopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1772

6-fluoropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1773

6-chloropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1774

6-bromopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1775

6-iodopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1776

6-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1777

6-nitropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1778

6-cyanopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1779

5-fluoropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1780

5-chloropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1781

5-bromopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1782

5-iodopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1783

5-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1784

5-nitropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1785

5-cyanopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1786

4-fluoropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1787

4-chloropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1788

4-bromopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1789

4-iodopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1790

4-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1791

4-nitropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1792

4-cyanopyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1793

2,6-dichloropyridin-3-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1794

pyridin-3-yl N-oxide

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1795

pyridin-4-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1796

2-chloropyridin-4-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1797

3-bromopyridin-4-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1798

3,5-dichloropyridin-4-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1799

3-(trifluoromethyl) pyridin-4-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1800

2,6-dicyanopyridin-4-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1801

pyridin-4-yl N-oxide

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1802

pyridin-2-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1803

3-chloropyridin-2-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1804

4-bromopyridin-2-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1805

5-iodopyridin-2-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1806

6-chloropyridin-2-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1807

4-cyanopyridin-2-yl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1808

phenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1809

2-fluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1810

3-fluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1811

4-fluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1812

2-chlorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1813

3-chlorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1814

4-chlorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1815

2-bromophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1816

3-bromophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1817

4-bromophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1818

2-iodophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1819

3-iodophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1820

4-iodophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1821

(2-trifluoromethyl) phenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1822

(3-trifluoromethyl) phenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1823

(4-trifluoromethyl) phenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1824

2-nitrophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1825

3-nitrophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1826

4-nitrophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1827

2-cyanophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1828

3-cyanophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1829

4-cyanophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1830

2,6-difluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1831

3,4-dichlorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1832

2,4-dichlorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1833

2-chloro-4-fluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1834

2-chloro-4,5-difluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1835

4-bromo-2-chlorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1836

2-bromo-4-chlorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1837

2-bromo-4-fluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1838

2-chloro-4-nitrophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1839

3,5-dicyanophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1840

4-cyano-2-fluorophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1841

2-chloro-4-cyanophenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1842

pyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1843

2-fluoropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1844

2-chloropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1845

2-bromopyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1846

2-iodopyrdin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1847

2-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1848

2-nitropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1849

2-cyanopyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1850

6-fluoropyrdin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1851

6-chloropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1852

6-bromopyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1853

6-iodopyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1854

6-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1855

6-nitropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1856

6-cyanopyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1857

5-fluoropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1858

5-chloropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1859

5-bromopyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1860

5-iodopyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1861

5-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1862

5-nitropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1863

5-cyanopyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1864

4-fluoropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1865

4-chloropyridin-3-yl

H

H

F

H

H

H

1

H

nonafluoro-2-butyl

H

CF3

6-1866

4-bromopyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1867

4-iodopyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1868

4-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1869

4-nitropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1870

4-cyanopyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1871

2,6-dichloropyridin-3-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1872

pyridin-3-yl N-oxide

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1873

pyridin-4-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1874

2-chloropyridin-4-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1875

3-bromopyridin-4-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1876

3,5-dichloropyridin-4-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1877

3-(trifluoromethyl) pyridin-4-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1878

2,6-dicyanopyridin-4-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1879

pyridin-4-yl N-oxide

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1880

pyridin-2-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1881

3-chloropyridin-2-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1882

4-bromopyridin-2-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1883

5-iodopyridin-2-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1884

6-chloropyridin-2-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1885

4-cyanopyridin-2-yl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-1886

phenyl

H

H

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-1901

3-cyanophenyl

H

H

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-1902

4-cyanophenyl

H

H

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-1917

2-chloropyridin-3-yl

H

H

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-1942

phenyl

H

H

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-1957

3-cyanophenyl

H

H

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-1958

4-cyanophenyl

H

H

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-1973

2-chloropyridin-3-yl

H

H

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-1998

phenyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-2013

3-cyanophenyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-2014

4-cyanophenyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-2029

2-chloropyridin-3-yl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-2054

phenyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-2069

3-cyanophenyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-2070

4-cyanophenyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-2085

2-chloropyridin-3-yl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-2110

phenyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-2130

3-cyanophenyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-2131

4-cyanophenyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-2146

2-chloropyridin-3-yl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-2178

phenyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-2198

3-cyanophenyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-2199

4-cyanophenyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-2214

2-chloropyridin-3-yl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-2246

phenyl

H

H

H

F

H

H

F

H

heptafluoroisopropyl

H

F

6-2247

3-cyanophenyl

H

H

H

F

H

H

F

H

heptafluoroisopropyl

H

F

6-2248

4-cyanophenyl

H

H

H

F

H

H

F

H

heptafluoroisopropyl

H

F

6-2249

2-chloropyridin-3-yl

H

H

H

F

H

H

F

H

heptafluoroisopropyl

H

F

6-2250

phenyl

H

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

6-2251

3-cyanophenyl

H

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

6-2252

4-cyanophenyl

H

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

6-2253

2-chloropyridin-3-yl

H

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

6-2254

phenyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-2274

3-cyanophenyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-2275

4-cyanophenyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-2290

2-chloropyridin-3-yl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-2332

phenyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-2352

3-cyanophenyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-2353

4-cyanophenyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-2368

2-chloropyridin-3-yl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-2410

phenyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

6-2430

3-cyanophenyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

6-2431

4-cyanophenyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

6-2446

2-chloropyridin-3-yl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

6-2488

phenyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-2508

3-cyanophenyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-2509

4-cyanophenyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-2524

2-chloropyridin-3-yl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-2566

phenyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

I

6-2586

3-cyanophenyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

I

6-2587

4-cyanophenyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

I

6-2602

2-chloropyridin-3-yl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

I

6-2644

phenyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

6-2664

3-cyanophenyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

6-2665

4-cyanophenyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

6-2680

2-chloropyridin-3-yl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

6-2722

phenyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

6-2742

3-cyanophenyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

6-2743

4-cyanophenyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

6-2758

2-chloropyridin-3-yl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

6-2800

phenyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

6-2820

3-cyanophenyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

6-2821

4-cyanophenyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

6-2836

2-chloropyridin-3-yl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

6-2878

phenyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

6-2898

3-cyanophenyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

6-2899

4-cyanophenyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

6-2914

2-chloropyridin-3-yl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

6-2956

phenyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

6-2976

3-cyanophenyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

6-2977

4-cyanophenyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

6-2992

2-chloropyriclin-3-yl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

6-3034

phenyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

6-3054

3-cyanophenyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

6-3055

4-cyanophenyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

6-3070

2-chloropyridin-3-yl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

6-3112

phenyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

6-3132

3-cyanophenyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

6-3133

4-cyanophenyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

6-3148

2-chloropyridin-3-yl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

6-3190

phenyl

H

H

H

F

H

H

F

H

heptafluoroisopropyl

H

CF3

6-3191

phenyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-3211

3-cyanophenyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-3212

4-cyanophenyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-3227

2-chloropyridin-3-yl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-3269

phenyl

H

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

6-3270

phenyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-3290

3-cyanophenyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-3291

4-cyanophenyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-3306

2-chloropyridin-3-yl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-3348

phenyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-3368

3-cyanophenyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-3369

4-cyanophenyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-3384

2-chloropyridin-3-yl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-3426

phenyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-3446

3-cyanophenyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-3447

4-cyanophenyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-3462

2-chloropyridin-3-yl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-3504

phenyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

6-3524

3-cyanophenyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

6-3525

4-cyanophenyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

6-3540

2-chloropyridin-3-yl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

6-3582

phenyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-3602

3-cyanophenyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-3603

4-cyanophenyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-3618

2-chloropyridin-3-yl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-3660

phenyl

H

H

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-3675

3-cyanophenyl

H

H

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-3676

4-cyanophenyl

H

H

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-3691

2-chloropyridin-3-yl

H

H

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-3716

phenyl

H

H

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-3731

3-cyanophenyl

H

H

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-3732

4-cyanophenyl

H

H

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-3747

2-chloropyridin-3-yl

H

H

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-3772

phenyl

H

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-3787

3-cyanophenyl

H

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-3788

4-cyanophenyl

H

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-3803

2-chloropyridin-3-yl

H

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-3828

phenyl

H

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-3843

3-cyanophenyl

H

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-3844

4-cyanophenyl

H

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-3859

2-chloropyridin-3-yl

H

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-3884

phenyl

H

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-3904

3-cyanophenyl

H

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-3905

4-cyanophenyl

H

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-3920

2-chloropyridin-3-yl

H

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-3952

phenyl

H

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-3972

3-cyanophenyl

H

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-3973

4-cyanophenyl

H

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-3988

2-chloropyridin-3-yl

H

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-4020

phenyl

H

H

F

F

H

H

F

H

heptafluoroisopropyl

H

F

6-4021

3-cyanophenyl

H

H

F

F

H

H

F

H

heptafluoroisopropyl

H

F

6-4022

4-cyanophenyl

H

H

F

F

H

H

F

H

heptafluoroisopropyl

H

F

6-4023

2-chloropyridin-3-yl

H

H

F

F

H

H

F

H

heptafluoroisopropyl

H

F

6-4024

phenyl

H

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

6-4025

3-cyanophenyl

H

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

6-4026

4-cyanophenyl

H

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

6-4027

2-chlorpyridin-3-yl

H

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

6-4028

phenyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-4048

3-cyanophenyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-4049

4-cyanophenyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-4064

2-chlorphenyl-3-yl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-4106

phenyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-4126

3-cyanophenyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-4127

4-cyanophenyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-4142

2-chloropyridin-3-yl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

6-4184

phenyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

6-4204

3-cyanophenyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

6-4205

4-cyanophenyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

6-4220

2-chloropyridin-3-yl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

6-4262

phenyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-4282

3-cyanophenyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-4283

4-cyanophenyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-4298

2-chloropyrid6-3-yl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-4340

phenyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

I

6-4360

3-cyanophenyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

I

6-4361

4-cyanophenyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

I

6-4376

2-chloropyridin-3-yl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

I

6-4418

phenyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

6-4438

3-cyanophenyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

6-4439

4-cyanophenyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

6-4454

2-chloropyridin-3-yl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

6-4496

phenyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

6-4516

3-cyanophenyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

6-4517

4-cyanophenyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

6-4532

2-chloropyridin-3-yl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

6-4574

phenyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

6-4594

3-cyanophenyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

6-4595

4-cyanophenyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

6-4610

2-chloropyridin-3-yl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

6-4652

phenyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

6-4672

3-cyanophenyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

6-4673

4-cyanophenyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

6-4688

2-chloropyridin-3-yl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

6-4730

phenyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

6-4750

3-cyanophenyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

6-4751

4-cyanophenyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

6-4766

2-chloropyridin-3-yl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

6-4808

phenyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

6-4828

3-cyanophenyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

6-4829

4-cyanophenyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

6-4844

2-chloropyridin-3-yl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

6-4886

phenyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

6-4906

3-cyanophenyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

6-4907

4-cyanophenyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

6-4922

2-chloropyridin-3-yl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

6-4964

phenyl

H

H

F

F

H

H

F

H

heptafluoroisopropyl

H

CF3

6-4965

phenyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-4985

3-cyanophenyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-4986

4-cyanophenyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-5001

2-chloropyridin-3-yl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-5043

phenyl

H

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

6-5044

phenyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-5064

3-cyanophenyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-5065

4-cyanophenyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-5080

2-chloropyridin-3-yl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

6-5122

phenyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-5142

3-cyanophenyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-5143

4-cyanophenyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-5158

2-chloropyridin-3-yl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-5200

phenyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-5220

3-cyanophenyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-5221

4-cyanophenyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-5236

2-chloropyridin-3-yl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

6-5278

phenyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

6-5298

3-cyanophenyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

6-5299

4-cyanophenyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

6-5314

2-chlorpyridin-3-yl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

6-5356

phenyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-5376

3-cyanophenyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-5377

4-cyanophenyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-5392

2-chloropyridin-3-yl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

6-5434

phenyl

H

H

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-5449

3-cyanophenyl

H

H

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-5450

4-cyanophenyl

H

H

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-5465

2-chloropyridin-3-yl

H

H

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

6-5490

phenyl

H

H

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-5505

3-cyanophenyl

H

H

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-5506

4-cyanophenyl

H

H

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-5521

2-chloropyridin-3-yl

H

H

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

6-5546

phenyl

H

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-5561

3-cyanophenyl

H

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-5562

4-cyanophenyl

H

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-5577

2-chloropyridin-3-yl

H

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

6-5602

phenyl

H

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-5617

3-cyanophenyl

H

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-5633

2-chloropyridin-3-yl

H

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

6-5658

phenyl

H

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-5678

3-cyanophenyl

H

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-5694

2-chloropyridin-3-yl

H

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-5726

phenyl

H

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-5746

3-cyanophenyl

H

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-5747

4-cyanophenyl

H

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-5762

2-chloropyridin-3-yl

H

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-5794

phenyl

H

H

F

F

F

H

Cl

H

pentafluoroethyl

H

Cl

6-5795

phenyl

H

H

F

F

F

H

Br

H

heptafluoroisopropyl

H

Br

6-5796

phenyl

H

H

F

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

6-5797

phenyl

H

H

F

F

F

H

I

H

heptafluoroisopropyl

H

CF3

6-5798

phenyl

H

H

F

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

6-5799

phenyl

H

H

F

F

F

H

I

H

nonafluoro-2-butyl

H

I

6-5800

phenyl

H

H

F

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

6-5801

phenyl

H

H

F

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

6-5802

phenyl

H

H

F

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-5803

phenyl

H

H

H

H

F

H

Cl

H

pentafluoroethyl

H

Cl

6-5804

phenyl

H

H

H

H

F

H

Br

H

heptafluoroisopropyl

H

Br

6-5805

phenyl

H

H

H

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

6-5806

phenyl

H

H

H

H

F

H

I

H

heptafluoroisopropyl

H

CF3

6-5807

phenyl

H

H

H

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

6-5808

phenyl

H

H

H

H

F

H

I

H

nonafluoro-2-butyl

H

I

6-5809

phenyl

H

H

H

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

6-5810

phenyl

H

H

H

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

6-5811

phenyl

H

H

H

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-5812

phenyl

H

H

H

H

H

F

Cl

H

pentafluoroethyl

H

Cl

6-5813

phenyl

H

H

H

H

H

F

Br

H

heptafluoroisopropyl

H

Br

6-5814

phenyl

H

H

H

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

6-5815

phenyl

H

H

H

H

H

F

I

H

heptafluoroisopropyl

H

CF3

6-5816

phenyl

H

H

H

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

6-5817

phenyl

H

H

H

H

H

F

I

H

nonafluoro-2-butyl

H

I

6-5818

phenyl

H

H

H

H

H

F

CI

H

nonafluoro-2-butyl

H

OCF3

6-5819

phenyl

H

H

H

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

6-5820

phenyl

H

H

H

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

6-5821

phenyl

H

H

F

H

F

H

Cl

H

pentafluoroethyl

H

CI

6-5822

phenyl

H

H

F

H

F

H

Br

H

heptafluoroisopropyl

H

Br

6-5823

phenyl

H

H

F

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

6-5824

phenyl

H

H

F

H

F

H

I

H

heptafluoroisopropyl

H

CF3

6-5825

phenyl

H

H

F

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

6-5826

phenyl

H

H

F

H

H

F

I

H

nonafluoro-2-butyl

H

I

6-5827

phenyl

H

H

F

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

6-5828

phenyl

H

H

F

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

6-5829

phenyl

H

H

F

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

6-5830

phenyl

H

H

F

H

H

F

Cl

H

pentafluoroethyl

H

Cl

6-5831

phenyl

H

H

F

H

H

F

Br

H

heptafluoroisopropyl

H

Br

6-5832

phenyl

H

H

F

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

6-5833

phenyl

H

H

F

H

H

F

I

H

heptafluoroisopropyl

H

CF3

6-5834

phenyl

H

H

F

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

6-5835

phenyl

H

H

F

H

H

F

I

H

nonafluoro-2-butyl

H

I

6-5836

phenyl

H

H

F

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

6-5837

phenyl

H

H

F

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

6-5838

phenyl

H

H

F

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

6-5839

phenyl

H

H

H

F

F

H

Cl

H

pentafluoroethyl

H

Cl

6-5840

phenyl

H

H

H

F

F

H

Br

H

heptafluoroisopropyl

H

Br

6-5841

phenyl

H

H

H

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

6-5842

phenyl

H

H

H

F

F

H

I

H

heptafluoroisopropyl

H

CF3

6-5843

phenyl

H

H

H

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

6-5844

phenyl

H

H

H

F

F

H

I

H

nonafluoro-2-butyl

H

I

6-5845

phenyl

H

H

H

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

6-5846

phenyl

H

H

H

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

6-5847

phenyl

H

H

H

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

6-5848

phenyl

H

H

H

F

H

F

Cl

H

pentafluoroethyl

H

Cl

6-5849

phenyl

H

H

H

F

H

F

Br

H

heptafluoroisopropyl

H

Br

6-5850

phenyl

H

H

H

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

6-5851

phenyl

H

H

H

F

H

F

I

H

heptafluoroisopropyl

H

CF3

6-5852

phenyl

H

H

H

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

6-5853

phenyl

H

H

H

F

H

F

I

H

nonafluoro-2-butyl

H

I

6-5854

phenyl

H

H

H

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

6-5855

phenyl

H

H

H

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

6-5856

phenyl

H

H

H

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

6-5857

phenyl

H

H

H

H

F

F

Cl

H

pentafluoroethyl

H

Cl

6-5858

phenyl

H

H

H

H

F

F

Br

H

heptafluoroisopropyl

H

Br

6-5859

phenyl

H

H

H

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

6-5860

phenyl

H

H

H

H

F

F

I

H

heptafluoroisopropyl

H

CF3

6-5861

phenyl

H

H

H

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

6-5862

phenyl

H

H

H

H

F

F

I

H

nonafluoro-2-butyl

H

I

6-5863

phenyl

H

H

H

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

6-5864

phenyl

H

H

H

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

6-5865

phenyl

H

H

H

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

6-5866

phenyl

H

H

F

F

H

F

Cl

H

pentafluoroethyl

H

Cl

6-5867

phenyl

H

H

F

F

H

F

Br

H

heptafluoroisopropyl

H

Br

6-5868

phenyl

H

H

F

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

6-5869

phenyl

H

H

F

F

H

F

I

H

heptafluoroisopropyl

H

CF3

6-5870

phenyl

H

H

F

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

6-5871

phenyl

H

H

F

F

H

F

I

H

nonafluoro-2-butyl

H

I

6-5872

phenyl

H

H

F

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

6-5873

phenyl

H

H

F

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

6-5874

phenyl

H

H

F

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

6-5875

phenyl

H

H

F

H

F

F

Cl

H

pentafluoroethyl

H

Cl

6-5876

phenyl

H

H

F

H

F

F

Br

H

heptafluoroisopropyl

H

Br

6-5877

phenyl

H

H

F

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

6-5878

phenyl

H

H

F

H

F

F

I

H

heptafluoroisopropyl

H

CF3

6-5879

phenyl

H

H

F

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

6-5880

phenyl

H

H

F

H

F

F

I

H

nonafluoro-2-butyl

H

I

6-5881

phenyl

H

H

F

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

6-5882

phenyl

H

H

F

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

6-5883

phenyl

H

H

F

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

6-5884

phenyl

H

H

H

F

F

F

Cl

H

pentafluoroethyl

H

Cl

6-5885

phenyl

H

H

H

F

F

F

Br

H

heptafluoroisopropyl

H

Br

6-5886

phenyl

H

H

H

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

6-5887

phenyl

H

H

H

F

F

F

I

H

heptafluoroisopropyl

H

CF3

6-5888

phenyl

H

H

H

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

6-5889

phenyl

H

H

H

F

F

F

I

H

nonafluoro-2-butyl

H

I

6-5890

phenyl

H

H

F

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

6-5891

phenyl

H

H

F

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

6-5892

phenyl

H

H

F

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

6-5893

phenyl

H

H

F

F

F

F

Cl

H

pentafluoroethyl

H

Cl

6-5894

phenyl

H

H

F

F

F

F

Br

H

heptafluoroisopropyl

H

Br

6-5895

phenyl

H

H

F

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

6-5896

phenyl

H

H

F

F

F

F

I

H

heptafluoroisopropyl

H

CF3

6-5897

phenyl

H

H

F

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

6-5898

phenyl

H

H

F

F

F

F

I

H

nonafluoro-2-butyl

H

I

6-5899

phenyl

H

H

F

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

6-5900

phenyl

H

H

F

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

6-5901

phenyl

H

H

F

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

6-5902

phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Cl

6-5903

3-fluorophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-5904

4-fluorophenyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

6-5905

3-fluorophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-5906

4-fluorophenyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

6-5907

phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

6-5908

2-chloropyridin-3-yl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

6-5909

4-cyanophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

6-5910

phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

C2F5

6-5911

4-cyanophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

C2F5

6-5912

2-chloro-4-(methylsulfonyl) phenyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-5913

phenyl

H

H

H

H

H

H

Br

H

pentafluoroethyl

H

CF3

6-5914

2-chloropyridin-3-yl

H

H

H

H

H

H

Br

H

pentafluoroethyl

H

CF3

TABLE 7

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

7-1

phenyl

Me

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

7-2

3-cyanophenyl

Me

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

7-3

4-cyanophenyl

Me

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

7-4

2-chloropyridin-3-yl

Me

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

7-5

phenyl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-12

3-cyanophenyl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-13

4-cyanophenyl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-24

2-chloropyridin-3-yl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-38

phenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-39

2-fluorophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-45

3-cyanophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-46

4-cyanophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-47

2,6-difluorophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-57

2-chloropyridin-3-yl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-60

6-chloropyridin-3-yl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-71

phenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-72

2-fluorophenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-78

3-cyanophenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-79

4-cyanophenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-80

2,6-difluorophenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-90

2-chloropyridin-3-yl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-93

6-chloropyridin-3-yl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-104

phenyl

Me

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

Cl

7-105

phenyl

Me

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

Br

7-106

phenyl

Me

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

I

7-107

phenyl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Br

7-108

phenyl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

I

7-109

phenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

I

7-110

phenyl

Me

H

H

H

H

H

F

H

heptafluoroisopropyl

H

CF3

7-111

phenyl

Me

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-131

3-cyanophenyl

Me

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-132

4-cyanophenyl

Me

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-147

2-chloropyridin-3-yl

Me

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-189

phenyl

Me

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

7-190

phenyl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-210

3-cyanophenyl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-211

4-cyanophenyl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-226

2-chloropyridin-3-yl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-268

phenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-269

2-fluorophenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-270

3-fluorophenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-271

4-fluorophenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-285

3-nitrophenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-286

4-nitrophenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-288

3-cyanophenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-289

4-cyanophenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-290

2,6-difluorophenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-299

3,5-dicyanophenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-300

4-cyano-2-fluorophenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-301

2-chloro-4-cyanophenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-303

2-fluoropyridin-3-yl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-304

2-chloropyridin-3-yl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-305

2-bromopyridin-3-yl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-311

6-chloropyridin-3-yl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-316

6-cyanopyridin-3-yl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-346

phenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-347

2-fluorophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-348

3-fluorophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-349

4-fluorophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-366

3-cyanophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-367

4-cyanophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-368

2,6-difluorophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-382

2-chloropyridin-3-yl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-389

6-chloropyridin-3-yl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-424

phenyl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-425

2-fluorophenyl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-426

3-fluorophenyl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-427

4-fluorophenyl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-428

2-chlorophenyl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-444

3-cyanophenyl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-445

4-cyanophenyl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-446

2,6-difluorophenyl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-449

2-chloro-4-fluorophenyl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-460

2-chloropyridin-3-yl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-467

6-chloropyridin-3-yl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-502

phenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-504

3-fluorophenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-505

4-fluorophenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-522

3-cyanophenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-523

4-cyanophenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-538

2-chloropyridin-3-yl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-580

phenyl

Me

H

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

7-611

2-chloropyridin-3-yl

Me

H

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

7-636

phenyl

Me

H

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

7-667

2-chloropyridin-3-yl

Me

H

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

7-692

phenyl

Me

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

7-723

2-chloropyridin-3-yl

Me

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

7-748

phenyl

Me

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

7-779

2-chloropyridin-3-yl

Me

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

7-804

phenyl

Me

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-824

3-cyanophenyl

Me

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-825

4-cyanophenyl

Me

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-840

2-chloropyridin-3-yl

Me

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-841

2-bromopyridin-3-yl

Me

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-872

phenyl

Me

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-892

3-cyanophenyl

Me

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-893

4-cyanophenyl

Me

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-908

2-chloropyridin-3-yl

Me

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-940

phenyl

Me

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

7-941

3-cyanophenyl

Me

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

7-942

4-cyanophenyl

Me

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

7-943

2-chloropyridin-3-yl

Me

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

7-944

phenyl

Me

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

7-945

3-cyanophenyl

Me

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

7-946

4-cyanophenyl

Me

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

7-947

2-chloropyridin-3-yl

Me

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

7-948

phenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-968

3-cyanophenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-969

4-cyanophenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-984

2-chloropyridin-3-yl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-1026

phenyl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-1046

3-cyanophenyl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-1047

4-cyanophenyl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-1062

2-chloropyridin-3-yl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-1104

phenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1105

2-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1106

3-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1107

4-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1124

3-cyanophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1125

4-cyanophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1126

2,6-difluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1140

2-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1147

6-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1182

phenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-1183

2-fluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-1184

3-fluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-1185

4-fluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-1202

3-cyanophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-1203

4-cyanophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-1204

2,6-difluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-1218

2-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-1225

6-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-1260

phenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1261

2-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1262

3-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1263

4-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1280

3-cyanophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1281

4-cyanophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1282

2,6-difluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1296

2-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1303

6-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1338

phenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-1339

2-fluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-1340

3-fluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-1341

4-fluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-1358

3-cyanophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-1359

4-cyanophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-1360

2,6-difluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-1374

2-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-1381

6-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-1416

phenyl

Me

H

F

H

H

H

F

H

heptafluoroisopropyl

H

CF3

7-1417

phenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-1428

3-iodophenyl

Me

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

7-1429

4-iodophenyl

Me

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

7-1431

(3-trifluoromethyl)phenyl

Et

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-1436

2-cyanophenyl

Me

H

F

H

H

H

Cl

H

pentafluoroethyl

H

C2F5

7-1437

3-cyanophenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-1438

4-cyanophenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-1441

2,4-dichlorophenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

7-1442

2-chloro-4-fluorophenyl

n-Pr

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-1445

2-bromo-4-chlorophenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

7-1452

2-fluoropyridin-3-yl

Me

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

7-1453

2-chloropyridin-3-yl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-1459

6-fluoropyridin-3-yl

i-Pr

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-1466

5-fluoropyridin-3-yl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

7-1468

5-bromopyridin-3-yl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

7-1469

5-iodopyridin-3-yl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

7-1471

5-nitropyridin-3-yl

Me

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

7-1473

4-fluoropyridin-3-yl

Me

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

7-1475

4-bromopyridin-3-yl

CH2CH═CH2

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

7-1476

4-iodopyridin-3-yl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

7-1482

pyridin-4-yl

CN

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-1494

4-cyanopyridin-2-yl

Me

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

7-1495

phenyl

Me

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

7-1496

phenyl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-1504

3-bromophenyl

CH2C≡CH

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-1509

(2-trifluoromethyl)phenyl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

7-1511

(4-trifluoromethyl)phenyl

NH2

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-1516

3-cyanophenyl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-1517

4-cyanophenyl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-1524

2-bromo-4-chlorophenyl

C(O)OMe

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-1526

2-chloro-4-nitrophenyl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

7-1532

2-chloropyridin-3-yl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-1545

5-fluoropyridin-3-yl

C(O)OEt

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

7-1547

5-bromopyridin-3-yl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

7-1548

5-iodopyridin-3-yl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

7-1552

4-fluoropyridin-3-yl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

7-1554

4-bromopyridin-3-yl

C(O)C(O)Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-1556

4-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

7-1557

4-nitropyridin-3-yl

C(O)C(O)Et

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

7-1571

5-iodopyridin-2-yl

C(O)Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-1573

4-cyanopyridin-2-yl

C(O)Et

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

7-1574

phenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1575

2-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1576

3-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1577

4-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1578

2-chlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1579

3-chlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1580

4-chlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1581

2-bromophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1582

3-bromophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1583

4-bromophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1584

2-iodophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1585

3-iodophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1586

4-iodophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1587

(2-trifluoromethyl)phenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1588

(3-trifluoromethyl)phenyl

S(O)2Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1589

(4-trifluoromethyl)phenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1590

2-nitrophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1591

3-nitrophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1592

4-nitrophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1593

2-cyanophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1594

3-cyanophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1595

4-cyanophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1596

2,6-difluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1597

3,4-dichlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1598

2,4-dichlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1599

2-chloro-4-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1600

2-chloro-4,5-difluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1601

4-bromo-2-chlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1602

2-bromo-4-chlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1603

2-bromo-4-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1604

2-chloro-4-nitrophenyl

S(O)2Et

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1605

3,5-dicyanophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1606

4-cyano-2-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1607

2-chloro-4-cyanophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1608

pyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1609

2-fluoropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1610

2-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1611

2-bromopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1612

2-iodopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1613

2-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1614

2-nitropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1615

2-cyanopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1616

6-fluoropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1617

6-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1618

6-bromopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1619

6-iodopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1620

6-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1621

6-nitropyridin-3-yl

CH2Ph

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1622

6-cyanopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1623

5-fluoropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1624

5-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1625

5-bromopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1626

5-iodopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1627

5-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1628

5-nitropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1629

5-cyanopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1630

4-fluoropyridin-3-yl

CH2(3-Py)

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1631

4-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1632

4-bromopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1633

4-iodopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1634

4-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1635

4-nitropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1636

4-cyanopyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1637

2,6-dichloropyridin-3-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1638

pyridin-3-yl N-oxide

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1639

pyridin-4-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1640

2-chloropyridin-4-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1641

3-bromopyridin-4-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1642

3,5-dichloropyridin-4-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1643

3-(trifluoromethyl)pyridin-4-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1644

2,6-dicyanopyridin-4-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1645

pyridin-4-yl N-oxide

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1646

pyridin-2-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1647

3-chloropyridin-2-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1648

4-bromopyridin-2-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1649

5-iodopyridin-2-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1650

6-chloropyridin-2-yl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1651

4-cyanopyridin-2-yl

CH2(3-Py—N-

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

7-1652

phenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1653

2-fluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1654

3-fluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1655

4-fluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1656

2-chlorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1657

3-chlorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1658

4-chlorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1659

2-bromophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1660

3-bromophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1661

4-bromophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1662

2-iodophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1663

3-iodophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1664

4-iodophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1665

(2-trifluoromethyl)phenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1666

(3-trifluoromethyl)phenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1667

(4-trifluoromethyl)phenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1668

2-nitrophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1669

3-nitrophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1670

4-nitrophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1671

2-cyanophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1672

3-cyanophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1673

4-cyanophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1674

2,6-difluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1675

3,4-dichlorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1676

2,4-dichlorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1677

2-chloro-4-fluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1678

2-chloro-4,5-difluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1679

4-bromo-2-chlorophenyl

Et

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1680

2-bromo-4-chlorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1681

2-bromo-4-fluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1682

2-chloro-4-nitrophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1683

3,5-dicyanophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1684

4-cyano-2-fluorophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1685

2-chloro-4-cyanophenyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1686

pyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1687

2-fluoropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1688

2-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1689

2-bromopyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1690

2-iodopyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1691

2-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1692

2-nitropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1693

2-cyanopyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1694

6-fluoropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1695

6-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1696

6-bromopyridin-3-yl

Me

H

F

H

H

H

Br

H

nanafluoro-2-butyl

H

CF3

7-1697

6-iodopyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1698

6-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1699

6-nitropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1700

6-cyanopyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1701

5-fluoropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1702

5-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1703

5-bromopyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1704

5-iodopyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1705

5-(trifluoromethyl)pyridin-3-yl

CN

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1706

5-nitropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1707

5-cyanopyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1708

4-fluoropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1709

4-chloropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1710

4-bromopyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1711

4-iodopyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1712

4-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1713

4-nitropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1714

4-cyanopyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1715

2,6-dichloropyridin-3-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1716

pyridin-3-yl N-oxide

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1717

pyridin-4-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1718

2-chloropyridin-4-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1719

3-bromopyridin-4-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1720

3,5-dichloropyridin-4-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1721

3-(trifluoromethyl)pyridin-4-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1722

2,6-dicyanopyridin-4-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1723

pyridin-4-yl N-oxide

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1724

pyridin-2-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1725

3-chloropyridin-2-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1726

4-bromopyridin-2-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1727

5-iodopyridin-2-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1728

6-chloropyridin-2-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1729

4-cyanopyridin-2-yl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-1730

phenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1731

2-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1732

3-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1733

4-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1734

2-chlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1735

3-chlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1736

4-chlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1737

2-bromophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1738

3-bromophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1739

4-bromophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1740

2-iodophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1741

3-iodophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1742

4-iodophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1743

(2-trifluoromethyl)phenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1744

(3-trifluoromethyl)phenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1745

(4-trifluoromethyl)phenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1746

2-nitrophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1747

3-nitrophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1748

4-nitrophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1749

2-cyanophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1750

3-cyanophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1751

4-cyanophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1752

2,6-difluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1753

3,4-dichlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1754

2,4-dichlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1755

2-chloro-4-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1756

2-chloro-4,5-difluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1757

4-bromo-2-chlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1758

2-bromo-4-chlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1759

2-bromo-4-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1760

2-chloro-4-nitrophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1761

3,5-dicyanophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1762

4-cyano-2-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1763

2-chloro-4-cyanophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1764

pyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1765

2-fluoropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1766

2-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1767

2-bromopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1768

2-iodopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1769

2-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1770

2-nitropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1771

2-cyanopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1772

6-fluoropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1773

6-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1774

6-bromopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1775

6-iodopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1776

6-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1777

6-nitropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1778

6-cyanopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1779

5-fluoropyridin-3-yl

C(O)Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1780

5-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1781

5-bromopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1782

5-iodopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1783

5-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1784

5-nitropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1785

5-cyanopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1786

4-fluoropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1787

4-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1788

4-bromopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1789

4-iodopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1790

4-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1791

4-nitropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1792

4-cyanopyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1793

2,6-dichloropyridin-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1794

pyridin-3-yl N-oxide

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1795

pyridin-4-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1796

2-chloropyridin-4-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1797

3-bromopyridin-4-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1798

3,5-dichloropyridin-4-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1799

3-(trifluoromethyl)pyridin-4-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1800

2,6-dicyanopyridin-4-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1801

pyridin-4-yl N-oxide

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1802

pyridin-2-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1803

3-chloropyridin-2-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1804

4-bromopyridin-2-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1805

5-iodopyridin-2-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1806

6-chloropyridin-2-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1807

4-cyanopyridin-2-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1808

phenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1809

2-fluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1810

3-fluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1811

4-fluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1812

2-chlorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1813

3-chlorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1814

4-chlorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1815

2-bromophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1816

3-bromophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1817

4-bromophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1818

2-iodophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1819

3-iodophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1820

4-iodophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1821

(2-trifluoromethyl)phenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1822

(3-trifluoromethyl)phenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1823

(4-trifluoromethyl)phenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1824

2-nitrophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1825

3-nitrophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1826

4-nitrophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1827

2-cyanophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1828

3-cyanophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1829

4-cyanophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1830

2,6-difluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1831

3,4-dichlorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1832

2,4-dichlorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1833

2-chloro-4-fluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1834

2-chloro-4,5-difluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1835

4-bromo-2-chlorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1836

2-bromo-4-chlorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1837

2-bromo-4-fluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1838

2-chloro-4-nitrophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1839

3,5-dicyanophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1840

4-cyano-2-fluorophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1841

2-chloro-4-cyanophenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1842

pyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1843

2-fluoropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1844

2-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1845

2-bromopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1846

2-iodopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1847

2-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1848

2-nitropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1849

2-cyanopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1850

6-fluoropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1851

6-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1852

6-bromopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1853

6-iodopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1854

6-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1855

6-nitropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1856

6-cyanopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1857

5-fluoropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1858

5-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1859

5-bromopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1860

5-iodopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1861

5-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1862

5-nitropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1863

5-cyanopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1864

4-fluoropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1865

4-chloropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1866

4-bromopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1867

4-iodopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1868

4-(trifluoromethyl)pyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1869

4-nitropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1870

4-cyanopyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1871

2,6-dichloropyridin-3-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1872

pyridin-3-yl N-oxide

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1873

pyridin-4-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1874

2-chloropyridin-4-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1875

3-bromopyridin-4-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1876

3,5-dichloropyridin-4-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1877

3-(trifluoromethyl)pyridin-4-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1878

2,6-dicyanopyridin-4-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1879

pyridin-4-yl N-oxide

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1880

pyridin-2-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1881

3-chloropyridin-2-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1882

4-bromopyridin-2-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1883

5-iodopyridin-2-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1884

6-chloropyridin-2-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1885

4-cyanopyridin-2-yl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-1886

phenyl

Me

H

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

7-1901

3-cyanophenyl

Me

H

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

7-1902

4-cyanophenyl

Me

H

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

7-1917

2-chloropyridin-3-yl

Me

H

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

7-1942

phenyl

Me

H

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

7-1957

3-cyanophenyl

Me

H

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

7-1958

4-cyanophenyl

Me

H

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

7-1973

2-chloropyridin-3-yl

Me

H

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

7-1998

phenyl

Me

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

7-2013

3-cyanophenyl

Me

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

7-2014

4-cyanophenyl

Me

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

7-2029

2-chloropyridin-3-yl

Me

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

7-2054

phenyl

Me

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

7-2069

3-cyanophenyl

Me

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

7-2070

4-cyanophenyl

Me

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

7-2085

2-chloropyridin-3-yl

Me

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

7-2110

phenyl

Me

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-2130

3-cyanophenyl

Me

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-2131

4-cyanophenyl

Me

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-2146

2-chloropyridin-3-yl

Me

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-2178

phenyl

Me

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-2198

3-cyanophenyl

Me

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-2199

4-cyanophenyl

Me

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-2214

2-chloropyridin-3-yl

Me

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-2246

phenyl

Me

H

H

F

H

H

F

H

heptafluoroisopropyl

H

F

7-2247

3-cyanophenyl

Me

H

H

F

H

H

F

H

heptafluoroisopropyl

H

F

7-2248

4-cyanophenyl

Me

H

H

F

H

H

F

H

heptafluoroisopropyl

H

F

7-2249

2-chloropyridin-3-yl

Me

H

H

F

H

H

F

H

heptafluoroisopropyl

H

F

7-2250

phenyl

Me

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

7-2251

3-cyanophenyl

Me

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

7-2252

4-cyanophenyl

Me

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

7-2253

2-chloropyridin-3-yl

Me

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

7-2254

phenyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-2274

3-cyanophenyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-2275

4-cyanophenyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-2290

2-chloropyridin-3-yl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-2332

phenyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-2352

3-cyanophenyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-2353

4-cyanophenyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-2368

2-chloropyridin-3-yl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-2410

phenyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

7-2430

3-cyanophenyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

7-2431

4-cyanophenyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

7-2446

2-chloropyridin-3-yl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

7-2488

phenyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-2508

3-cyanophenyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-2509

4-cyanophenyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-2524

2-chloropyridin-3-yl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-2566

phenyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

I

7-2586

3-cyanophenyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

I

7-2587

4-cyanophenyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

I

7-2602

2-chloropyridin-3-yl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

I

7-2644

phenyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

7-2664

3-cyanophenyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

7-2665

4-cyanophenyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

7-2680

2-chloropyridin-3-yl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

7-2722

phenyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

7-2742

3-cyanophenyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

7-2743

4-cyanophenyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

7-2758

2-chloropyridin-3-yl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

7-2800

phenyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-2820

3-cyanophenyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-2821

4-cyanophenyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-2836

2-chloropyridin-3-yl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-2878

phenyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

7-2898

3-cyanophenyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

7-2899

4-cyanophenyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

7-2914

2-chloropyridin-3-yl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

7-2956

phenyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

7-2976

3-cyanophenyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

7-2977

4-cyanophenyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

7-2992

2-chloropyridin-3-yl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

7-3034

phenyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

7-3054

3-cyanophenyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

7-3055

4-cyanophenyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

7-3070

2-chloropyridin-3-yl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

7-3112

phenyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

7-3132

3-cyanophenyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

7-3133

4-cyanophenyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

7-3148

2-chloropyridin-3-yl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

7-3190

phenyl

Me

H

H

F

H

H

F

H

heptafluoroisopropyl

H

CF3

7-3191

phenyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-3211

3-cyanophenyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-3212

4-cyanophenyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-3227

2-chloropyridin-3-yl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-3269

phenyl

Me

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

7-3270

phenyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-3290

3-cyanophenyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-3291

4-cyanophenyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-3306

2-chloropyridin-3-yl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-3348

phenyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-3368

3-cyanophenyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-3369

4-cyanophenyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-3384

2-chloropyridin-3-yl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-3426

phenyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-3446

3-cyanophenyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-3447

4-cyanophenyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-3462

2-chloropyridin-3-yl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-3504

phenyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

7-3524

3-cyanophenyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

7-3525

4-cyanophenyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

7-3582

phenyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-3602

3-cyanophenyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-3603

4-cyanophenyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-3618

2-chloropyridin-3-yl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-3660

phenyl

Me

H

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

7-3691

2-chloropyridin-3-yl

Me

H

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

7-3716

phenyl

Me

H

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

7-3747

2-chloropyrtdin-3-yl

Me

H

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

7-3772

phenyl

Me

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

7-3803

2-chloropyridin-3-yl

Me

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

7-3828

phenyl

Me

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

7-3859

2-chloropyridin-3-yl

Me

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

7-3884

phenyl

Me

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-3904

3-cyanophenyl

Me

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-3905

4-cyanophenyl

Me

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-3920

2-chloropyridin-3-yl

Me

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-3952

phenyl

Me

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-3972

3-cyanophenyl

Me

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-3973

4-cyanophenyl

Me

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-3988

2-chloropyridin-3-yl

Me

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-4020

phenyl

Me

H

F

F

H

H

F

H

heptafluoroisopropyl

H

F

7-4021

3-cyanophenyl

Me

H

F

F

H

H

F

H

heptafluoroisopropyl

H

F

7-4022

4-cyanophenyl

Me

H

F

F

H

H

F

H

heptafluoroisopropyl

H

F

7-4023

2-chloropyridin-3-yl

Me

H

F

F

H

H

F

H

heptafluoroisopropyl

H

F

7-4024

phenyl

Me

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

7-4025

3-cyanophenyl

Me

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

7-4026

4-cyanophenyl

Me

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

7-4027

2-chloropyridin-3-yl

Me

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

7-4028

phenyl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-4048

3-cyanophenyl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-4049

4-cyanophenyl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-4064

2-chloropyridin-3-yl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-4106

phenyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-4126

3-cyanophenyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-4127

4-cyanophenyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-4142

2-chloropyridin-3-yl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

7-4184

phenyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

7-4204

3-cyanophenyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

7-4205

4-cyanophenyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

7-4220

2-chloropyridin-3-yl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

7-4262

phenyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-4282

3-cyanophenyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-4283

4-cyanophenyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-4298

2-chloropyridin-3-yl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-4340

phenyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

I

7-4360

3-cyanophenyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

I

7-4361

4-cyanophenyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

I

7-4376

2-chloropyridin-3-yl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

I

7-4418

phenyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

7-4438

3-cyanophenyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

7-4439

4-cyanophenyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

7-4454

2-chloropyridin-3-yl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

7-4496

phenyl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

7-4516

3-cyanophenyl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

7-4517

4-cyanophenyl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

7-4532

2-chloropyridin-3-yl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

7-4574

phenyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-4594

3-cyanophenyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-4595

4-cyanophenyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-4610

2-chloropyridin-3-yl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-4652

phenyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

7-4672

3-cyanophenyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

7-4673

4-cyanophenyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

7-4688

2-chloropyridin-3-yl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

7-4730

phenyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

7-4750

3-cyanophenyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

7-4751

4-cyanophenyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

7-4766

2-chloropyridin-3-yl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

7-4808

phenyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

7-4828

3-cyanophenyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

7-4829

4-cyanophenyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

7-4844

2-chloropyridin-3-yl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

7-4886

phenyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

7-4906

3-cyanophenyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

7-4907

4-cyanophenyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

7-4922

2-chloropyridin-3-yl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

7-4964

phenyl

Me

H

F

F

H

H

F

H

heptafluoroisopropyl

H

CF3

7-4965

phenyl

Me

H

F

F

H

H

Cl

H

heptafluoroisoproplyl

H

CF3

7-4985

3-cyanophenyl

Me

H

F

F

H

H

Cl

H

heptafluoroisoprppyl

H

CF3

7-4986

4-cyanophenyl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-5001

2-chloropyridin-3-yl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-5043

phenyl

Me

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

7-5044

phenyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-5064

3-cyanophenyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-5065

4-cyanophenyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-5080

2-chloropyridin-3-yl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

7-5122

phenyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-5142

3-cyanophenyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-5143

4-cyanophenyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-5158

2-chloropyridin-3-yl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-5200

phenyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-5220

3-cyanophenyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-5221

4-cyanophenyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-5236

2-chloropyridin-3-yl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

7-5278

phenyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

7-5298

3-cyanophenyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

7-5299

4-cyanophenyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

7-5314

2-chloropyridin-3-yl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

7-5356

phenyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-5376

3-cyanophenyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-5377

4-cyanophenyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-5392

2-chloropyridin-3-yl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

7-5434

phenyl

Me

H

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

7-5465

2-chloropyridin-3-yl

Me

H

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

7-5490

phenyl

Me

H

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

7-5521

2-chloropyridin-3-yl

Me

H

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

7-5546

phenyl

Me

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

7-5577

2-chloropyridin-3-yl

Me

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

7-5602

phenyl

Me

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

7-5633

2-chloropyridin-3-yl

Me

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

7-5658

phenyl

Me

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-5678

3-cyanophenyl

Me

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-5679

4-cyanophenyl

Me

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-5694

2-chloropyridin-3-yl

Me

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-5726

phenyl

Me

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-5746

3-cyanophenyl

Me

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-5747

4-cyanophenyl

Me

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-5762

2-chloropyridin-3-yl

Me

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-5794

phenyl

Me

H

F

F

F

H

Cl

H

pentafluoroethyl

H

Cl

7-5795

phenyl

Me

H

F

F

F

H

Br

H

heptafluoroisopropyl

H

Br

7-5796

phenyl

Me

H

F

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

7-5797

phenyl

Me

H

F

F

F

H

I

H

heptafluoroisopropyl

H

CF3

7-5798

phenyl

Me

H

F

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

7-5799

phenyl

Me

H

F

F

F

H

I

H

nonafluoro-2-butyl

H

I

7-5800

phenyl

Me

H

F

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5801

phenyl

Me

H

F

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

7-5802

phenyl

Me

H

F

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-5803

phenyl

Me

H

H

H

F

H

Cl

H

pentafluoroethyl

H

Cl

7-5804

phenyl

Me

H

H

H

F

H

Br

H

heptafluoroisopropyl

H

Br

7-5805

phenyl

Me

H

H

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

7-5806

phenyl

Me

H

H

H

F

H

I

H

heptafluoroisopropyl

H

CF3

7-5807

phenyl

Me

H

H

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

7-5808

phenyl

Me

H

H

H

F

H

I

H

nonafluoro-2-butyl

H

I

7-5809

phenyl

Me

H

H

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5810

phenyl

Me

H

H

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

7-5811

phenyl

Me

H

H

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-5812

phenyl

Me

H

H

H

H

F

Cl

H

pentafluoroethyl

H

Cl

7-5813

phenyl

Me

H

H

H

H

F

Br

H

heptafluoroisopropyl

H

Br

7-5814

phenyl

Me

H

H

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

7-5815

phenyl

Me

H

H

H

H

F

I

H

heptafluoroisopropyl

H

CF3

7-5816

phenyl

Me

H

H

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

7-5817

phenyl

Me

H

H

H

H

F

I

H

nonafluoro-2-butyl

H

I

7-5818

phenyl

Me

H

H

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5819

phenyl

Me

H

H

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

7-5820

phenyl

Me

H

H

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

7-5821

phenyl

Me

H

F

H

F

H

Cl

H

pentafluoroethyl

H

Cl

7-5822

phenyl

Me

H

F

H

F

H

Br

H

heptafluoroisopropyl

H

Br

7-5823

phenyl

Me

H

F

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

7-5824

phenyl

Me

H

F

H

F

H

I

H

heptafluoroisopropyl

H

CF3

7-5825

phenyl

Me

H

F

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

7-5826

phenyl

Me

H

F

H

F

H

I

H

nonafluoro-2-butyl

H

I

7-5827

phenyl

Me

H

F

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5828

phenyl

Me

H

F

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

7-5829

phenyl

Me

H

F

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-5830

phenyl

Me

H

F

H

H

F

Cl

H

pentafluoroethyl

H

Cl

7-5831

phenyl

Me

H

F

H

H

F

Br

H

heptafluoroisopropyl

H

Br

7-5832

phenyl

Me

H

F

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

7-5833

phenyl

Me

H

F

H

H

F

I

H

heptafluoroisopropyl

H

CF3

7-5834

phenyl

Me

H

F

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

7-5835

phenyl

Me

H

F

H

H

F

I

H

nonafluoro-2-butyl

H

I

7-5836

phenyl

Me

H

F

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5837

phenyl

Me

H

F

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

7-5838

phenyl

Me

H

F

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

7-5839

phenyl

Me

H

H

F

F

H

Cl

H

pentafluoroethyl

H

Cl

7-5840

phenyl

Me

H

H

F

F

H

Br

H

heptafluoroisopropyl

H

Br

7-5841

phenyl

Me

H

H

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

7-5842

phenyl

Me

H

H

F

F

H

I

H

heptafluoroisopropyl

H

CF3

7-5843

phenyl

Me

H

H

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

7-5844

phenyl

Me

H

H

F

F

H

I

H

nonafluoro-2-butyl

H

I

7-5845

phenyl

Me

H

H

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5846

phenyl

Me

H

H

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

7-5847

phenyl

Me

H

H

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

7-5848

phenyl

Me

H

H

F

H

F

Cl

H

pentafluoroethyl

H

Cl

7-5849

phenyl

Me

H

H

F

H

F

Br

H

heptafluoroisopropyl

H

Br

7-5850

phenyl

Me

H

H

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

7-5851

phenyl

Me

H

H

F

H

F

I

H

heptafluoroisopropyl

H

CF3

7-5852

phenyl

Me

H

H

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

7-5853

phenyl

Me

H

H

F

H

F

I

H

nonafluoro-2-butyl

H

I

7-5854

phenyl

Me

H

H

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5855

phenyl

Me

H

H

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

7-5856

phenyl

Me

H

H

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

7-5857

phenyl

Me

H

H

H

F

F

Cl

H

pentafluoroethyl

H

Cl

7-5858

phenyl

Me

H

H

H

F

F

Br

H

heptafluoroisopropyl

H

Br

7-5859

phenyl

Me

H

H

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

7-5860

phenyl

Me

H

H

H

F

F

I

H

heptafluoroisopropyl

H

CF3

7-5861

phenyl

Me

H

H

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

7-5862

phenyl

Me

H

H

H

F

F

I

H

nonafluoro-2-butyl

H

I

7-5863

phenyl

Me

H

H

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5864

phenyl

Me

H

H

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

7-5865

phenyl

Me

H

H

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

7-5866

phenyl

Me

H

F

F

H

F

Cl

H

pentafluoroethyl

H

Cl

7-5867

phenyl

Me

H

F

F

H

F

Br

H

heptafluoroisopropyl

H

Br

7-5868

phenyl

Me

H

F

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

7-5869

phenyl

Me

H

F

F

H

F

I

H

heptafluoroisopropyl

H

CF3

7-5870

phenyl

Me

H

F

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

7-5871

phenyl

Me

H

F

F

H

F

I

H

nonafluoro-2-butyl

H

I

7-5872

phenyl

Me

H

F

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5873

phenyl

Me

H

F

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

7-5874

phenyl

Me

H

F

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

7-5875

phenyl

Me

H

F

H

F

F

Cl

H

pentafluoroethyl

H

Cl

7-5876

phenyl

Me

H

F

H

F

F

Br

H

heptafluoroisopropyl

H

Br

7-5877

phenyl

Me

H

F

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

7-5878

phenyl

Me

H

F

H

F

F

I

H

heptafluoroisopropyl

H

CF3

7-5879

phenyl

Me

H

F

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

7-5880

phenyl

Me

H

F

H

F

F

I

H

nonafluoro-2-butyl

H

I

7-5881

phenyl

Me

H

F

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5882

phenyl

Me

H

F

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

7-5883

phenyl

Me

H

F

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

7-5884

phenyl

Me

H

H

F

F

F

Cl

H

pentafluoroethyl

H

Cl

7-5885

phenyl

Me

H

H

F

F

F

Br

H

heptafluoroisopropyl

H

Br

7-5886

phenyl

Me

H

H

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

7-5887

phenyl

Me

H

H

F

F

F

I

H

heptafluoroisopropyl

H

CF3

7-5888

phenyl

Me

H

H

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

7-5889

phenyl

Me

H

H

F

F

F

I

H

nonafluoro-2-butyl

H

I

7-5890

phenyl

Me

H

H

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5891

phenyl

Me

H

H

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

7-5892

phenyl

Me

H

H

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

7-5893

phenyl

Me

H

F

F

F

F

Cl

H

pentafluoroethyl

H

Cl

7-5894

phenyl

Me

H

F

F

F

F

Br

H

heptafluoroisopropyl

H

Br

7-5895

phenyl

Me

H

F

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

7-5896

phenyl

Me

H

F

F

F

F

I

H

heptafluoroisopropyl

H

CF3

7-5897

phenyl

Me

H

F

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

7-5898

phenyl

Me

H

F

F

F

F

I

H

nonafluoro-2-butyl

H

I

7-5899

phenyl

Me

H

F

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

7-5900

phenyl

Me

H

F

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

7-5901

phenyl

Me

H

F

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

7-5902

phenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

Br

7-5903

2-chloropyridine-3-yl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

Br

7-5904

3-fluorophenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-5905

4-fluorophenyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

7-5906

3-fluorophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-5907

4-fluorophenyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

7-5908

4-(methylsulfonyl)phenyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-5909

pyrimidine-5-yl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-5910

3-cyano-5-(methoxycarbonyl)phenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-5911

phenyl

Me

H

H

H

H

H

Br

H

pentafluoroethyl

H

CF3

7-5912

2-chloropyridine-3-yl

Me

H

H

H

H

H

Br

H

pentafluoroethyl

H

CF3

TABLE 8

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

8-1

phenyl

H

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

8-2

3-cyanophenyl

H

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

8-3

4-cyanophenyl

H

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

8-4

2-chloropyridin-3-yl

H

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

8-5

phenyl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-12

3-cyanophenyl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-13

4-cyanophenyl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-24

2-chloropyridin-3-yl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-38

phenyl

H

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-45

3-cyanophenyl

H

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-46

4-cyanophenyl

H

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-57

2-chloropyridin-3-yl

H

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-71

phenyl

H

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

8-78

3-cyanophenyl

H

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

8-79

4-cyanophenyl

H

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

8-90

2-chloropyridin-3-yl

H

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

8-104

phenyl

H

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

Cl

8-105

phenyl

H

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

Br

8-106

phenyl

H

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

I

8-107

phenyl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Br

8-108

phenyl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

I

8-109

phenyl

H

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

I

8-110

phenyl

H

Me

H

H

H

H

F

H

heptafluoroisopropyl

H

CF3

8-111

phenyl

H

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-131

3-cyanophenyl

H

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-132

4-cyanophenyl

H

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-147

2-chloropyridin-3-yl

H

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-189

phenyl

H

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

8-190

phenyl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-210

3-cyanophenyl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-211

4-cyanophenyl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-226

2-chloropyridin-3-yl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-268

phenyl

H

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-288

3-cyanophenyl

H

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-289

4-cyanophenyl

H

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-304

2-chloropyridin-3-yl

H

Me

H

H

H

H

Br

H

heptafluorpisopropyl

H

CF3

8-305

2-bromopyridin-3-yl

H

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-346

phenyl

H

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-366

3-cyanophenyl

H

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-367

4-cyanophenyl

H

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-382

2-chloropyridin-3-yl

H

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-424

phenyl

H

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

8-444

3-cyanophenyl

H

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

8-445

4-cyanophenyl

H

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

8-460

2-chloropyridin-3-yl

H

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

8-502

phenyl

H

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-522

3-cyanophenyl

H

Me

H

H

H

H

I

H

npnafluoro-2-butyl

H

CF3

8-523

4-cyanophenyl

H

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-538

2-chloropyridin-3-yl

H

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-580

phenyl

H

Me

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

8-611

2-chloropyridin-3-yl

H

Me

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

8-636

phenyl

H

Me

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

8-667

2-chloropyridin-3-yl

H

Me

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

8-692

phenyl

H

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

8-723

2-chloropyridin-3-yl

H

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

8-748

phenyl

H

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

8-779

2-chloropyridin-3-yl

H

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

8-804

phenyl

H

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-824

3-cyanophenyl

H

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-825

4-cyanophenyl

H

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-840

2-chloropyridin-3-yl

H

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-841

2-bromopyridin-3-yl

H

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-872

phenyl

H

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-892

3-cyanophenyl

H

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-893

4-cyanophenyl

H

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-908

2-chloropyridin-3-yl

H

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-940

phenyl

H

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

F

8-941

3-cyanophenyl

H

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

F

8-942

4-cyanophenyl

H

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

F

8-943

2-chloropyridin-3-yl

H

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

F

8-944

phenyl

H

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

8-945

3-cyanophenyl

H

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

8-946

4-cyanophenyl

H

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

8-947

2-chloropyridin-3-yl

H

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

8-948

phenyl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-952

2-chlorophenyl

H

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

Cl

8-956

3-bromophenyl

H

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

Br

8-961

(2-trifluoromethyl)phenyl

H

i-Pr

F

H

H

H

F

H

heptafluoroisopropyl

H

I

8-964

2-nitrophenyl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Br

8-968

3-cyanophenyl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-969

4-cyanophenyl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-970

2,6-difluorophenyl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

I

8-982

pyridin-3-yl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

I

8-984

2-chloropyridin-3-yl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-1026

phenyl

H

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-1046

3-cyanophenyl

H

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-1047

4-cyanophenyl

H

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-1062

2-chloropyridin-3-yl

H

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-1104

phenyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

8-1124

3-cyanophenyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

8-1125

4-cyanophenyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

8-1140

2-chloropyridin-3-yl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

8-1182

phenyl

H

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-1202

3-cyanophenyl

H

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-1203

4-cyanophenyl

H

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-1218

2-chloropyridin-3-yl

H

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-1260

phenyl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

I

8-1280

3-cyanophenyl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

I

8-1281

4-cyanophenyl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

I

8-1296

2-chloropyridin-3-yl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

I

8-1338

phenyl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

8-1358

3-cyanophenyl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

8-1359

4-cyanophenyl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

8-1374

2-chloropyridin-3-yl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

8-1416

phenyl

H

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

CF3

8-1417

phenyl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-1431

(3-trifluoromethyl)phenyl

H

Et

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-1437

3-cyanophenyl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-1438

4-cyanophenyl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-1442

2-chloro-4-fluorophenyl

H

n-Pr

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-1453

2-chloropyridin-3-yl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-1459

6-fluoropyridin-3-yl

H

i-Pr

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-1475

4-bromopyridin-3-yl

H

CH2CH═CH2

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

8-1482

pyridin-4-yl

H

CN

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-1495

phenyl

H

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

8-1496

phenyl

H

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-1504

3-bromophenyl

H

CH2C≡CH

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-1511

(4-trifluoromethyl)phenyl

H

NH2

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-1516

3-cyanophenyl

H

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-1517

4-cyanophenyl

H

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-1524

2-bromo-4-chlorophenyl

H

C(O)OMe

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-1532

2-chloropyridin-3-yl

H

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-1545

5-fluoropyridin-3-yl

H

C(O)OEt

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

8-1554

4-bromopyridin-3-yl

H

C(O)C(O)Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-1557

4-nitropyridin-3-yl

H

C(O)C(O)Et

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

8-1571

5-iodopyridin-2-yl

H

C(O)Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-1573

4-cyanopyridin-2-yl

H

C(O)Et

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

8-1574

phenyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-1588

(3-trifluoromethyl)phenyl

H

S(O)2Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-1594

3-cyanophenyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-1595

4-cyanophenyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-1606

4-cyano-2-fluorophenyl

H

S(O)2Et

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-1610

2-chloropyridin-3-yl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-1621

6-nitropyridin-3-yl

H

CH2Ph

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-1630

4-fluoropyridin-3-yl

H

CH2(3-Py)

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-1651

4-cyanopyridin-2-yl

H

CH2(3-Py—N-

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

8-1652

phenyl

H

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-1672

3-cyanophenyl

H

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-1673

4-cyanophenyl

H

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-1679

4-bromo-2-chlorophenyl

H

Et

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-1688

2-chloropyridin-3-yl

H

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-1705

5-(trifluoromethyl)pyridin-3-yl

H

CN

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-1730

phenyl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

8-1750

3-cyanophenyl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

8-1751

4-cyanophenyl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

8-1766

2-chloropyridin-3-yl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

8-1779

5-fluoropyridin-3-yl

H

C(O)Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

8-1808

phenyl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-1828

3-cyanophenyl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-1829

4-cyanophenyl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-1844

2-chloropyridin-3-yl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-1886

phenyl

H

Me

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

8-1901

3-cyanophenyl

H

Me

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

8-1902

4-cyanophenyl

H

Me

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

8-1917

2-chloropyridin-3-yl

H

Me

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

8-1942

phenyl

H

Me

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

8-1957

3-cyanophenyl

H

Me

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

8-1958

4-cyanophenyl

H

Me

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

8-1973

2-chloropyridin-3-yl

H

Me

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

8-1998

phenyl

H

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

8-2013

3-cyanophenyl

H

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

8-2014

4-cyanophenyl

H

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

8-2029

2-chloropyridin-3-yl

H

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

8-2054

phenyl

H

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

8-2069

3-cyanophenyl

H

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

8-2070

4-cyanophenyl

H

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

8-2085

2-chloropyridin-3-yl

H

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

8-2110

phenyl

H

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-2130

3-cyanophenyl

H

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-2131

4-cyanophenyl

H

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-2146

2-chloropyridin-3-yl

H

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-2178

phenyl

H

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-2198

3-cyanophenyl

H

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-2199

4-cyanophenyl

H

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-2214

2-chloropyridin-3-yl

H

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-2246

phenyl

H

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

F

8-2247

3-cyanophenyl

H

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

F

8-2248

4-cyanophenyl

H

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

F

8-2249

2-chloropyridin-3-yl

H

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

F

8-2250

phenyl

H

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

8-2251

3-cyanophenyl

H

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

8-2252

4-cyanophenyl

H

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

8-2253

2-chloropyridin-3-yl

H

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

8-2254

phenyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-2274

3-cyanophenyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-2275

4-cyanophenyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-2290

2-chloropyridin-3-yl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-2332

phenyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-2352

3-cyanophenyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-2353

4-cyanophenyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-2368

2-chloropyridin-3-yl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-2410

phenyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

8-2430

3-cyanophenyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

8-2431

4-cyanophenyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

8-2446

2-chloropyridin-3-yl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

8-2488

phenyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-2508

3-cyanophenyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-2509

4-cyanophenyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-2524

2-chloropyridin-3-yl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-2566

phenyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

I

8-2586

3-cyanophenyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

I

8-2587

4-cyanophenyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

I

8-2602

2-chloropyridin-3-yl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

I

8-2644

phenyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

8-2664

3-cyanophenyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

8-2665

4-cyanophenyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

8-2680

2-chloropyridin-3-yl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

8-2722

phenyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

8-2742

3-cyanophenyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

8-2743

4-cyanophenyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

8-2758

2-chloropyridin-3-yl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

8-2800

phenyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-2820

3-cyanophenyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-2821

4-cyanophenyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-2836

2-chloropyridin-3-yl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-2878

phenyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

8-2898

3-cyanophenyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

8-2899

4-cyanophenyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

8-2914

2-chloropyridin-3-yl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

8-2956

phenyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

8-2976

3-cyanophenyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

8-2977

4-cyanophenyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

8-2992

2-chloropyridin-3-yl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

8-3034

phenyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

8-3054

3-cyanophenyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

8-3055

4-cyanophenyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

8-3070

2-chloropyridin-3-yl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

8-3112

phenyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

8-3132

3-cyanophenyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

8-3133

4-cyanophenyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

8-3148

2-chloropyridin-3-yl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

8-3190

phenyl

H

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

CF3

8-3191

phenyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-3211

3-cyanophenyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-3212

4-cyanophenyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-3227

2-chloropyridin-3-yl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-3269

phenyl

H

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

8-3270

phenyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-3290

3-cyanophenyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-3291

4-cyanophenyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-3306

2-chloropyridin-3-yl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-3348

phenyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-3368

3-cyanophenyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-3369

4-cyanophenyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-3384

2-chloropyridin-3-yl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-3426

phenyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-3446

3-cyanophenyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-3447

4-cyanophenyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-3462

2-chloropyridin-3-yl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-3504

phenyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

8-3524

3-cyanophenyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

8-3525

4-cyanophenyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

8-3540

2-chloropyridin-3-yl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

8-3582

phenyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-3602

3-cyanophenyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-3603

4-cyanophenyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-3618

2-chloropyridin-3-yl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-3660

phenyl

H

Me

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

8-3691

2-chloropyridin-3-yl

H

Me

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

8-3716

phenyl

H

Me

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

8-3747

2-chloropyridin-3-yl

H

Me

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

8-3772

phenyl

H

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

8-3803

2-chloropyridin-3-yl

H

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

8-3828

phenyl

H

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

8-3859

2-chloropyridin-3-yl

H

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

8-3884

phenyl

H

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-3904

3-cyanophenyl

H

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-3905

4-cyanophenyl

H

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-3920

2-chloropyridin-3-yl

H

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-3952

phenyl

H

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-3972

3-cyanophenyl

H

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-3973

4-cyanophenyl

H

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-3988

2-chloropyridin-3-yl

H

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-4020

phenyl

H

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

F

8-4021

3-cyanophenyl

H

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

F

8-4022

4-cyanophenyl

H

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

F

8-4023

2-chloropyridin-3-yl

H

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

F

8-4024

phenyl

H

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

8-4025

3-cyanophenyl

H

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

8-4026

4-cyanophenyl

H

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

8-4027

2-chloropyridin-3-yl

H

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

8-4028

phenyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-4048

3-cyanophenyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-4049

4-cyanophenyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-4064

2-chloropyridin-3-yl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

8-4106

phenyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-4126

3-cyanophenyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-4127

4-cyanophenyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-4142

2-chloropyridin-3-yl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

8-4184

phenyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

8-4204

3-cyanophenyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

8-4205

4-cyanophenyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

8-4220

2-chloropyridin-3-yl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

8-4262

phenyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-4282

3-cyanophenyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-4283

4-cyanophenyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-4298

2-chloropyridin-3-yl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

8-4340

phenyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

I

8-4360

3-cyanophenyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

I

8-4361

4-cyanophenyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

I

8-4376

2-chloropyridin-3-yl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

I

8-4418

phenyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

8-4438

3-cyanophenyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

8-4439

4-cyanophenyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

8-4454

2-chloropyridin-3-yl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

8-4496

phenyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

8-4516

3-cyanophenyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

8-4517

4-cyanophenyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

8-4532

2-chloropyridin-3-yl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

8-4574

phenyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-4594

3-cyanophenyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-4595

4-cyanophenyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-4610

2-chloropyridin-3-yl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-4652

phenyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

8-4672

3-cyanophenyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

8-4673

4-cyanophenyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

8-4688

2-chloropyridin-3-yl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

8-4730

phenyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

8-4750

3-cyanophenyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

8-4751

4-cyanophenyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

8-4808

phenyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

8-4828

3-cyanophenyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

8-4829

4-cyanophenyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

8-4844

2-chloropyridin-3-yl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

8-4886

phenyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

8-4906

3-cyanophenyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

8-4907

4-cyanophenyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

8-4922

2-chloropyridin-3-yl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

8-4964

phenyl

H

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

CF3

8-4965

phenyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-4985

3-cyanophenyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-4986

4-cyanophenyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-5001

2-chloropyridin-3-yl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

8-5043

phenyl

H

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

8-5044

phenyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-5064

3-cyanophenyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-5065

4-cyanophenyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-5080

2-chloropyridin-3-yl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

8-5122

phenyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-5142

3-cyanophenyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-5143

4-cyanophenyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-5158

2-chloropyridin-3-yl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

8-5200

phenyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-5220

3-cyanophenyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-5221

4-cyanophenyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-5236

2-chloropyridin-3-yl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

8-5278

phenyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

8-5298

3-cyanophenyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

8-5299

4-cyanophenyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

8-5314

2-chloropyridin-3-yl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

8-5356

phenyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-5376

3-cyanophenyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-5377

4-cyanophenyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-5392

2-chloropyridin-3-yl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

8-5434

phenyl

H

Me

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

8-5465

2-chloropyridin-3-yl

H

Me

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

8-5490

phenyl

H

Me

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

8-5521

2-chloropyridin-3-yl

H

Me

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

8-5546

phenyl

H

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

8-5577

2-chloropyridin-3-yl

H

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

8-5602

phenyl

H

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

8-5633

2-chloropyridin-3-yl

H

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

8-5678

3-cyanophenyl

H

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-5679

4-cyanophenyl

H

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-5694

2-chloropyridin-3-yl

H

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

8-5726

phenyl

H

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-5746

3-cyanophenyl

H

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-5747

4-cyanophenyl

H

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-5762

2-chloropyridin-3-yl

H

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-5794

phenyl

H

Me

F

F

F

H

Cl

H

pentafluoroethyl

H

Cl

8-5795

phenyl

H

Me

F

F

F

H

Br

H

heptafluoroisopropyl

H

Br

8-5796

phenyl

H

Me

F

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

8-5797

phenyl

H

Me

F

F

F

H

I

H

heptafluoroisopropyl

H

CF3

8-5798

phenyl

H

Me

F

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

8-5799

phenyl

H

Me

F

F

F

H

I

H

nonafluoro-2-butyl

H

I

8-5800

phenyl

H

Me

F

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5801

phenyl

H

Me

F

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

8-5802

phenyl

H

Me

F

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-5803

phenyl

H

Me

H

H

F

H

Cl

H

pentafluoroethyl

H

Cl

8-5804

phenyl

H

Me

H

H

F

H

Br

H

heptafluoroisopropyl

H

Br

8-5805

phenyl

H

Me

H

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

8-5806

phenyl

H

Me

H

H

F

H

I

H

heptafluoroisopropyl

H

CF3

8-5807

phenyl

H

Me

H

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

8-5808

phenyl

H

Me

H

H

F

H

I

H

nonafluoro-2-butyl

H

I

8-5809

phenyl

H

Me

H

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5810

phenyl

H

Me

H

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

8-5811

phenyl

H

Me

H

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-5812

phenyl

H

Me

H

H

H

F

Cl

H

pentafluoroethyl

H

Cl

8-5813

phenyl

H

Me

H

H

H

F

Br

H

heptafluoroisopropyl

H

Br

8-5814

phenyl

H

Me

H

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

8-5815

phenyl

H

Me

H

H

H

F

I

H

heptafluoroisopropyl

H

CF3

8-5816

phenyl

H

Me

H

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

8-5817

phenyl

H

Me

H

H

H

F

I

H

nonafluoro-2-butyl

H

I

8-5818

phenyl

H

Me

H

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5819

phenyl

H

Me

H

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

8-5820

phenyl

H

Me

H

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

8-5821

phenyl

H

Me

F

H

F

H

Cl

H

pentafluoroethyl

H

Cl

8-5822

phenyl

H

Me

F

H

F

H

Br

H

heptafluoroisopropyl

H

Br

8-5823

phenyl

H

Me

F

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

8-5824

phenyl

H

Me

F

H

F

H

I

H

heptafluoroisopropyl

H

CF3

8-5825

phenyl

H

Me

F

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

8-5826

phenyl

H

Me

F

H

F

H

I

H

nonafluoro-2-butyl

H

I

8-5827

phenyl

H

Me

F

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5828

phenyl

H

Me

F

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

8-5829

phenyl

H

Me

F

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-5830

phenyl

H

Me

F

H

H

F

Cl

H

pentafluoroethyl

H

Cl

8-5831

phenyl

H

Me

F

H

H

F

Br

H

heptafluoroisopropyl

H

Br

8-5832

phenyl

H

Me

F

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

8-5833

phenyl

H

Me

F

H

H

F

I

H

heptafluoroisopropyl

H

CF3

8-5834

phenyl

H

Me

F

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

8-5835

phenyl

H

Me

F

H

H

F

I

H

nonafluoro-2-butyl

H

I

8-5836

phenyl

H

Me

F

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5837

phenyl

H

Me

F

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

8-5838

phenyl

H

Me

F

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

8-5839

phenyl

H

Me

H

F

F

H

Cl

H

pentafluoroethyl

H

Cl

8-5840

phenyl

H

Me

H

F

F

H

Br

H

heptafluoroisopropyl

H

Br

8-5841

phenyl

H

Me

H

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

8-5842

phenyl

H

Me

H

F

F

H

I

H

heptafluoroisopropyl

H

CF3

8-5843

phenyl

H

Me

H

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

8-5844

phenyl

H

Me

H

F

F

H

I

H

nonafluoro-2-butyl

H

I

8-5845

phenyl

H

Me

H

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5846

phenyl

H

Me

H

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

8-5847

phenyl

H

Me

H

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

8-5848

phenyl

H

Me

H

F

H

F

Cl

H

pentafluoroethyl

H

Cl

8-5849

phenyl

H

Me

H

F

H

F

Br

H

heptafluoroisopropyl

H

Br

8-5850

phenyl

H

Me

H

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

8-5851

phenyl

H

Me

H

F

H

F

I

H

heptafluoroisopropyl

H

CF3

8-5852

phenyl

H

Me

H

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

8-5853

phenyl

H

Me

H

F

H

F

I

H

nonafluoro-2-butyl

H

I

8-5854

phenyl

H

Me

H

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5855

phenyl

H

Me

H

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

8-5856

phenyl

H

Me

H

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

8-5857

phenyl

H

Me

H

H

F

F

Cl

H

pentafluoroethyl

H

Cl

8-5858

phenyl

H

Me

H

H

F

F

Br

H

heptafluoroisopropyl

H

Br

8-5859

phenyl

H

Me

H

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

8-5860

phenyl

H

Me

H

H

F

F

I

H

heptafluoroisopropyl

H

CF3

8-5861

phenyl

H

Me

H

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

8-5862

phenyl

H

Me

H

H

F

F

I

H

nonafluoro-2-butyl

H

I

8-5863

phenyl

H

Me

H

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5864

phenyl

H

Me

H

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

8-5865

phenyl

H

Me

H

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

8-5866

phenyl

H

Me

F

F

H

F

Cl

H

pentafluoroethyl

H

Cl

8-5867

phenyl

H

Me

F

F

H

F

Br

H

heptafluoroisopropyl

H

Br

8-5868

phenyl

H

Me

F

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

8-5869

phenyl

H

Me

F

F

H

F

I

H

heptafluoroisopropyl

H

CF3

8-5870

phenyl

H

Me

F

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

8-5871

phenyl

H

Me

F

F

H

F

I

H

nonafluoro-2-butyl

H

I

8-5872

phenyl

H

Me

F

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5873

phenyl

H

Me

F

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

8-5874

phenyl

H

Me

F

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

8-5875

phenyl

H

Me

F

H

F

F

Cl

H

pentafluoroethyl

H

Cl

8-5876

phenyl

H

Me

F

H

F

F

Br

H

heptafluoroisopropyl

H

Br

8-5877

phenyl

H

Me

F

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

8-5878

phenyl

H

Me

F

H

F

F

I

H

heptafluoroisopropyl

H

CF3

8-5879

phenyl

H

Me

F

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

8-5880

phenyl

H

Me

F

H

F

F

I

H

nonafluoro-2-butyl

H

I

8-5881

phenyl

H

Me

F

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5882

phenyl

H

Me

F

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

8-5883

phenyl

H

Me

F

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

8-5884

phenyl

H

Me

H

F

F

F

Cl

H

pentafluoroethyl

H

Cl

8-5885

phenyl

H

Me

H

F

F

F

Br

H

heptafluoroisopropyl

H

Br

8-5886

phenyl

H

Me

H

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

8-5887

phenyl

H

Me

H

F

F

F

I

H

heptafluoroisopropyl

H

CF3

8-5888

phenyl

H

Me

H

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

8-5889

phenyl

H

Me

H

F

F

F

I

H

nonafluoro-2-butyl

H

I

8-5890

phenyl

H

Me

H

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5891

phenyl

H

Me

H

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

8-5892

phenyl

H

Me

H

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

8-5893

phenyl

H

Me

F

F

F

F

Cl

H

pentafluoroethyl

H

Cl

8-5894

phenyl

H

Me

F

F

F

F

Br

H

heptafluoroisopropyl

H

Br

8-5895

phenyl

H

Me

F

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

8-5896

phenyl

H

Me

F

F

F

F

I

H

heptafluoroisopropyl

H

CF3

8-5897

phenyl

H

Me

F

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

8-5898

phenyl

H

Me

F

F

F

F

I

H

nonafluoro-2-butyl

H

I

8-5899

phenyl

H

Me

F

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

8-5900

phenyl

H

Me

F

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

8-5901

phenyl

H

Me

F

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 9

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

9-1

phenyl

Me

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

9-2

3-cyanophenyl

Me

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

9-3

4-cyanophenyl

Me

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

9-4

2-chloropyridin-3-yl

Me

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

F

9-5

phenyl

Me

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-12

3-cyanophenyl

Me

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-13

4-cyanophenyl

Me

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-24

2-chloropyridin-3-yl

Me

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-38

phenyl

Me

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-45

3-cyanophenyl

Me

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-46

4-cyanophenyl

Me

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-57

2-chloropyridin-3-yl

Me

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-71

phenyl

Me

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

9-78

3-cyanophenyl

Me

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

9-79

4-cyanophenyl

Me

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

9-90

2-chloropyridin-3-yl

Me

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

I

9-109

phenyl

Me

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

Br

9-112

phenyl

Me

Me

H

H

H

H

F

H

heptafluoroisopropyl

H

CF3

9-113

phenyl

Me

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-133

3-cyanophenyl

Me

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-134

4-cyanophenyl

Me

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-149

2-chloropyridin-3-yl

Me

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-191

phenyl

Me

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

9-192

phenyl

Me

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-212

3-cyanophenyl

Me

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-213

4-cyanophenyl

Me

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-228

2-chloropyridin-3-yl

Me

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-270

phenyl

Me

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-290

3-cyanophenyl

Me

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-291

4-cyanophenyl

Me

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-306

2-chloropyridin-3-yl

Me

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-348

phenyl

Me

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-368

3-cyanophenyl

Me

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-369

4-cyanophenyl

Me

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-384

2-chloropyridin-3-yl

Me

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-426

phenyl

Me

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

9-446

3-cyanophenyl

Me

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

9-447

4-cyanophenyl

Me

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

9-462

2-chloropyridin-3-yl

Me

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

9-504

phenyl

Me

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-524

3-cyanophenyl

Me

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-525

4-cyanophenyl

Me

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-540

2-chloropyridin-3-yl

Me

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-778

phenyl

Me

Me

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

9-809

2-chloropyridin-3-yl

Me

Me

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

9-834

phenyl

Me

Me

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

9-865

2-chloropyridin-3-yl

Me

Me

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

9-890

phenyl

Me

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

9-921

2-chloropyridin-3-yl

Me

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

9-946

phenyl

Me

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

9-977

2-chloropyridin-3-yl

Me

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

9-1002

phenyl

Me

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-1022

3-cyanophenyl

Me

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-1023

4-cyanophenyl

Me

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-1038

2-chloropyridin-3-yl

Me

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-1070

phenyl

Me

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-1090

3-cyanophenyl

Me

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-1091

4-cyanophenyl

Me

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-1106

2-chloropyridin-3-yl

Me

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-1334

phenyl

Me

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

F

9-1335

3-cyanophenyl

Me

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

F

9-1336

4-cyanophenyl

Me

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

F

9-1337

2-chloropyridin-3-yl

Me

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

F

9-1338

phenyl

Me

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

9-1339

3-cyanophenyl

Me

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

9-1340

4-cyanophenyl

Me

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

9-1341

2-chloropyridin-3-yl

Me

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

F

9-1342

phenyl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-1362

3-cyanophenyl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-1363

4-cyanophenyl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-1378

2-chloropyridin-3-yl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-1420

phenyl

Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-1440

3-cyanophenyl

Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-1441

4-cyanophenyl

Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-1456

2-chloropyridin-3-yl

Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-1498

phenyl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

9-1518

3-cyanophenyl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

9-1519

4-cyanophenyl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

9-1534

2-chloropyridin-3-yl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

9-1576

phenyl

Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-1596

3-cyanophenyl

Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-1597

4-cyanophenyl

Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-1612

2-chloropyridin-3-yl

Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-1654

phenyl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

I

9-1674

3-cyanophenyl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

I

9-1675

4-cyanophenyl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

I

9-1690

2-chloropyridin-3-yl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

I

9-1732

phenyl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

9-1752

3-cyanophenyl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

9-1753

4-cyanophenyl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

9-1768

2-chloropyridin-3-yl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

I

9-2006

phenyl

Me

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

CF3

9-2007

phenyl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-2019

4-iodophenyl

Me

Et

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

9-2021

(3-trifluoromethyl) phenyl

Et

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

9-2027

3-cyanophenyl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-2028

4-cyanophenyl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-2030

3,4-dichlorophenyl

Me

n-Pr

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-2032

2-chloro-4-fluorophenyl

n-Pr

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-2043

2-chloropyridin-3-yl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-2047

2-nitropyridin-3-yl

Me

i-Pr

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-2049

6-fluoropyridin-3-yl

i-Pr

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-2063

4-fluoropyridin-3-yl

Me

CH2CH═CH2

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

9-2065

4-bromopyridin-3-yl

CH2CH═CH2

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

9-2070

2,6-dichloropyridin-3-yl

Me

CN

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-2072

pyridin-4-yl

CN

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-2085

phenyl

Me

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

9-2086

phenyl

Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2092

4-chlorophenyl

Me

CH2C≡CH

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2094

3-bromophenyl

CH2C≡CH

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2099

(2-trifluoromethyl) phenyl

Me

NH2

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

9-2101

(4-trifluoromethyl) phenyl

NH2

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2106

3-cyanophenyl

Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2107

4-cyanophenyl

Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2112

2-chloro-4,5-difluorophenyl

Me

C(O)OMe

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2114

2-bromo-4-chlorophenyl

C(O)OMe

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2122

2-chloropyridin-3-yl

Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2133

6-nitropyridin-3-yl

Me

C(O)OEt

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2135

5-fluoropyridin-3-yl

C(O)OEt

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

9-2142

4-fluoropyridin-3-yl

Me

C(O)C(O)Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

9-2144

4-bromopyridin-3-yl

C(O)C(O)Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2145

4-iodopyridin-3-yl

Me

C(O)C(O)Et

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2147

4-nitropyridin-3-yl

C(O)C(O)Et

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

9-2156

2,6-dicyanopyridin-4-yl

Me

C(O)Et

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2159

3-chloropyridin-2-yl

Me

C(O)Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2161

5-iodopyridin-2-yl

C(O)Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-2163

4-cyanopyridin-2-yl

C(O)Et

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

9-2164

phenyl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2176

4-iodophenyl

Me

S(O)2Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2178

(3-trifluoromethyl) phenyl

S(O)2Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2184

3-cyanophenyl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2185

4-cyanophenyl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2194

2-chloro-4-nitrophenyl

Me

S(O)2Et

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2196

4-cyano-2-fluorophenyl

S(O)2Et

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2200

2-chloropyridin-3-yl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2209

6-iodopyridin-3-yl

Me

CH2Ph

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2211

6-nitropyridin-3-yl

CH2Ph

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2218

5-nitropyridin-3-yl

Me

CH2(3-Py)

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2220

4-fluoropyridin-3-yl

CH2(3-Py)

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-2239

5-iodopyridin-2-yl

Me

CH2(3-Py—N-

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

9-2241

4-cyanopyridin-2-yl

CH2(3-Py—N-

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

9-2242

phenyl

Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-2262

3-cyanophenyl

Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-2263

4-cyanophenyl

Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-2267

2-chloro-4-fluorophenyl

Me

Et

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-2269

4-bromo-2-chlorophenyl

Et

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-2278

2-chloropyridin-3-yl

Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-2293

5-bromopyridin-3-yl

Me

CN

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-2295

5-(fluoromethyl) pyridin-3-yl

CN

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-2320

phenyl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

9-2322

3-fluorophenyl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

9-2340

3-cyanophenyl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

9-2341

4-cyanophenyl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

9-2356

2-chloropyridin-3-yl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

9-2367

6-nitropyridin-3-yl

Me

C(O)Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

9-2369

5-fluoropyridin-3-yl

C(O)Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

9-2398

phenyl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2418

3-cyanophenyl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2419

4-cyanophenyl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2434

2-chloropyridin-3-yl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2476

phenyl

Et

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2477

phenyl

Et

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2478

phenyl

Et

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2479

phenyl

Et

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2480

phenyl

Et

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2481

phenyl

Et

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2482

phenyl

Et

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2483

phenyl

Et

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2484

phenyl

Et

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2485

phenyl

Et

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2486

phenyl

Et

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2487

phenyl

Et

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2488

phenyl

Et

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2489

phenyl

Et

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2490

phenyl

n-Pr

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2491

phenyl

n-Pr

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2492

phenyl

n-Pr

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2493

phenyl

n-Pr

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2494

phenyl

n-Pr

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2495

phenyl

n-Pr

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2496

phenyl

n-Pr

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2497

phenyl

n-Pr

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2498

phenyl

n-Pr

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2499

phenyl

n-Pr

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2500

phenyl

n-Pr

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2501

phenyl

n-Pr

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2502

phenyl

n-Pr

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2503

phenyl

n-Pr

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2504

phenyl

i-Pr

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2505

phenyl

i-Pr

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2506

phenyl

i-Pr

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2507

phenyl

i-Pr

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2508

phenyl

i-Pr

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2509

phenyl

i-Pr

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2510

phenyl

i-Pr

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2511

phenyl

i-Pr

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2512

phenyl

i-Pr

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2513

phenyl

i-Pr

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2514

phenyl

i-Pr

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2515

phenyl

i-Pr

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2516

phenyl

i-Pr

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2517

phenyl

i-Pr

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2518

phenyl

CH2CH═CH2

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2519

phenyl

CH2CH═CH2

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2520

phenyl

CH2CH═CH2

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2521

phenyl

CH2CH═CH2

CH2CH=CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2522

phenyl

CH2CH═CH2

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2523

phenyl

CH2CH═CH2

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2524

phenyl

CH2CH═CH2

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2525

phenyl

CH2CH═CH2

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2526

phenyl

CH2CH═CH2

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2527

phenyl

CH2CH═CH2

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2528

phenyl

CH2CH═CH2

C(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2529

phenyl

CH2CH═CH2

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2530

phenyl

CH2CH═CH2

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2531

phenyl

CH2CH═CH2

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2532

phenyl

CN

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2533

phenyl

CN

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2534

phenyl

CN

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2535

phenyl

CN

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2536

phenyl

CN

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2537

phenyl

CN

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2538

phenyl

CN

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2539

phenyl

CN

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2540

phenyl

CN

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2541

phenyl

CN

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2542

phenyl

CN

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2543

phenyl

CN

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2544

phenyl

CN

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2545

phenyl

CN

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2546

phenyl

CH2C≡CH

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2547

phenyl

CH2C≡CH

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2548

phenyl

CH2C≡CH

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2549

phenyl

CH2C≡CH

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2550

phenyl

CH2C≡CH

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2551

phenyl

CH2C≡CH

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2552

phenyl

CH2C≡CH

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2553

phenyl

CH2C≡CH

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2554

phenyl

CH2C≡CH

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2555

phenyl

CH2C≡CH

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2556

phenyl

CH2C≡CH

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2557

phenyl

CH2C≡CH

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2558

phenyl

CH2C≡CH

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2559

phenyl

CH2C≡CH

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2560

phenyl

NH2

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2561

phenyl

NH2

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2562

phenyl

NH2

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2563

phenyl

NH2

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2564

phenyl

NH2

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2565

phenyl

NH2

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2566

phenyl

NH2

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2567

phenyl

NH2

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2568

phenyl

NH2

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2569

phenyl

NH2

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2570

phenyl

NH2

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

FI

CF3

9-2571

phenyl

NH2

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2572

phenyl

NH2

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2573

phenyl

NH2

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2574

phenyl

C(O)OMe

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2575

phenyl

C(O)OMe

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2576

phenyl

C(O)OMe

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2577

phenyl

C(O)OMe

CH2CH=CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2578

phenyl

C(O)OMe

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2579

phenyl

C(O)OMe

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2580

phenyl

C(O)OMe

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2581

phenyl

C(O)OMe

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2582

phenyl

C(O)OMe

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2583

phenyl

C(O)OMe

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2584

phenyl

C(O)OMe

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2585

phenyl

C(O)OMe

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2586

phenyl

C(O)OMe

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2587

phenyl

C(O)OMe

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2588

phenyl

C(O)C(O)OMe

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2589

phenyl

C(O)C(O)OMe

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2590

phenyl

C(O)C(O)OMe

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2591

phenyl

C(O)C(O)OMe

CH2CH=CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2592

phenyl

C(O)C(O)OMe

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2593

phenyl

C(O)C(O)OMe

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2594

phenyl

C(O)C(O)OMe

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2595

phenyl

C(O)C(O)OMe

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2596

phenyl

C(O)C(O)OMe

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2597

phenyl

C(O)C(O)OMe

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2598

phenyl

C(O)C(O)OMe

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2599

phenyl

C(O)C(O)OMe

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2600

phenyl

C(O)C(O)OMe

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2601

phenyl

C(O)C(O)OMe

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2602

phenyl

C(O)Me

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2603

phenyl

C(O)Me

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2604

phenyl

C(O)Me

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2605

phenyl

C(O)Me

CH2CH=CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2606

phenyl

C(O)Me

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2607

phenyl

C(O)Me

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2608

phenyl

C(O)Me

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2609

phenyl

C(O)Me

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2610

phenyl

C(O)Me

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2611

phenyl

C(O)Me

C(O)Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-2612

phenyl

C(O)Me

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2613

phenyl

C(O)Me

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2614

phenyl

C(O)Me

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2615

phenyl

C(O)Me

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2616

phenyl

S(O)2Me

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2617

phenyl

S(O)2Me

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2618

phenyl

S(O)2Me

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2619

phenyl

S(O)2Me

CH2CH=CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2620

phenyl

S(O)2Me

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2621

phenyl

S(O)2Me

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2622

phenyl

S(O)2Me

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2623

phenyl

S(O)2Me

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2624

phenyl

S(O)2Me

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2625

phenyl

S(O)2Me

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2626

phenyl

S(O)2Me

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2627

phenyl

S(O)2Me

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2628

phenyl

S(O)2Me

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2629

phenyl

S(O)2Me

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2630

phenyl

CH2Ph

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2631

phenyl

CH2Ph

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2632

phenyl

CH2Ph

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2633

phenyl

CH2Ph

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2634

phenyl

CH2Ph

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2635

phenyl

CH2Ph

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2636

phenyl

CH2Ph

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2637

phenyl

CH2Ph

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2638

phenyl

CH2Ph

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2639

phenyl

CH2Ph

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2640

phenyl

CH2Ph

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2641

phenyl

CH2Ph

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2642

phenyl

CH2P8

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2643

phenyl

CH2Ph

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2644

phenyl

CH2(3-Py)

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2645

phenyl

CH2(3-Py)

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2646

phenyl

CH2(3-Py)

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2647

phenyl

CH2(3-Py)

CH2CH=CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2648

phenyl

CH2(3-Py)

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2649

phenyl

CH2(3-Py)

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2650

phenyl

CH2(3-Py)

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2651

phenyl

CH2(3-Py)

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2652

phenyl

CH2(3-Py)

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2653

phenyl

CH2(3-Py)

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2654

phenyl

CH2(3-Py)

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2655

phenyl

CH2(3-Py)

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2656

phenyl

CH2(3-Py)

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-2657

phenyl

CH2(3-Py)

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2658

phenyl

CH2(3-Py—N-

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2659

phenyl

CH2(3-Py—N-

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2660

phenyl

CH2(3-Py—N-

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2661

phenyl

CH2(3-Py—N-

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2662

phenyl

CH2(3-Py—N-

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2663

phenyl

CH2(3-Py—N-

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2664

phenyl

CH2(3-Py—N-

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2665

phenyl

CH2(3-Py—N-

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2666

phenyl

CH2(3-Py—N-

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2667

phenyl

CH2(3-Py—N-

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2668

phenyl

CH2(3-Py—N-

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2669

phenyl

CH2(3-Py—N-

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2670

phenyl

CH2(3-Py—N-

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

9-2671

phenyl

CH2(3-Py—N-

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

oxide)

9-2672

phenyl

Me

Me

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

9-2687

3-cyanophenyl

Me

Me

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

9-2688

4-cyanophenyl

Me

Me

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

9-2703

2-chloropyridin-3-yl

Me

Me

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

9-2728

phenyl

Me

Me

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

9-2743

3-cyanophenyl

Me

Me

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

9-2744

4-cyanophenyl

Me

Me

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

9-2759

2-chloropyridin-3-yl

Me

Me

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

9-2784

phenyl

Me

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

9-2799

3-cyanophenyl

Me

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

9-2800

4-cyanophenyl

Me

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

9-2815

2-chloropyridin-3-yl

Me

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

9-2840

phenyl

Me

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

9-2855

3-cyanophenyl

Me

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

9-2856

4-cyanophenyl

Me

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

9-2871

2-chloropyridin-3-yl

Me

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

9-2896

phenyl

Me

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-2916

3-cyanophenyl

Me

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-2917

4-cyanophenyl

Me

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-2932

2-chloropyridin-3-yl

Me

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-2964

phenyl

Me

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-2984

3-cyanophenyl

Me

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-2985

4-cyanophenyl

Me

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-3000

2-chloropyridin-3-yl

Me

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-3228

phenyl

Me

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

F

9-3229

3-cyanophenyl

Me

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

F

9-3230

4-cyanophenyl

Me

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

F

9-3231

2-chloropyridin-3-yl

Me

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

F

9-3232

phenyl

Me

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

9-3233

3-cyanophenyl

Me

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

9-3234

4-cyanophenyl

Me

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

9-3235

2-chloropyridin-3-yl

Me

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

9-3236

phenyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-3256

3-cyanophenyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-3257

4-cyanophenyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-3272

2-chloropyridin-3-yl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-3314

phenyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-3334

3-cyanophenyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-3335

4-cyanophenyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-3350

2-chloropyridin-3-yl

Me

Me

H

F

F

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-3392

phenyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

9-3412

3-cyanophenyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

9-3413

4-cyanophenyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

9-3428

2-chloropyridin-3-yl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

9-3470

phenyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-3490

3-cyanophenyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-3491

4-cyanophenyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-3506

2-chloropyridin-3-yl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-3548

phenyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

I

9-3568

3-cyanophenyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

I

9-3569

4-cyanophenyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

I

9-3584

2-chloropyridin-3-yl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

I

9-3626

phenyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

9-3646

3-cyanophenyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

9-3647

4-cyanophenyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

9-3662

2-chloropyridin-3-yl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

9-3900

phenyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

9-3920

3-cyanophenyl

Me

Me

H

F

H

H

Cl

Cl

heptafluoroisopropyl

H

OCF3

9-3921

4-cyanophenyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

9-3936

2-chloropyridin-3-yl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

9-3978

phenyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

9-3998

3-cyanophenyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

9-3999

4-cyanophenyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

9-4014

2-chloropyridin-3-yl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

9-4056

phenyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

9-4076

3-cyanophenyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

9-4077

4-cyanophenyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

9-4092

2-chloropyridin-3-yl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

9-4134

phenyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

9-4154

3-cyanophenyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

9-4155

4-cyanophenyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

9-4170

2-chloropyridin-3-yl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

9-4212

phenyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

9-4232

3-cyanophenyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

9-4233

4-cyanophenyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

9-4248

2-chloropyridin-3-yl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

9-4290

phenyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

9-4310

3-cyanophenyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

9-4311

4-cyanophenyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

9-4326

2-chloropyridin-3-yl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

9-4564

phenyl

Me

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

CF3

9-4565

phenyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-4585

3-cyanophenyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-4586

4-cyanophenyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-4601

2-chloropyridin-3-yl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-4643

phenyl

Me

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

9-4644

phenyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-4664

3-cyanophenyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-4665

4-cyanophenyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-4680

2-chloropyridin-3-yl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-4722

phenyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-4742

3-cyanophenyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-4743

4-cyanophenyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-4758

2-chloropyridin-3-yl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-4800

phenyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-4820

3-cyanophenyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

FI

CF3

9-4821

4-cyanophenyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-4836

2-chloropyridin-3-yl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-4878

phenyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

9-4898

3-cyanophenyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

9-4899

4-cyanophenyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

9-4914

2-chloropyridin-3-yl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

9-4956

phenyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-4976

3-cyanophenyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-4977

4-cyanophenyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-4992

2-chloropyridin-3-yl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-5230

phenyl

Me

Me

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

9-5261

2-chloropyridin-3-yl

Me

Me

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

9-5286

phenyl

Me

Me

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

9-5317

2-chloropyridin-3-yl

Me

Me

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

9-5342

phenyl

Me

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

9-5373

2-chloropyridin-3-yl

Me

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

9-5398

phenyl

Me

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

9-5429

2-chloropyridin-3-yl

Me

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

9-5454

phenyl

Me

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-5474

3-cyanophenyl

Me

Me

H

F

H

H

CF3

H

heotafluoroisopropyl

H

CF3

9-5475

4-cyanophenyl

Me

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-5490

2-chloropyridin-3-yl

Me

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-5522

phenyl

Me

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-5542

3-cyanophenyl

Me

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-5543

4-cyanophenyl

Me

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-5558

2-chloropyridin-3-yl

Me

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-5786

phenyl

Me

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

F

9-5787

3-cyanophenyl

Me

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

F

9-5788

4-cyanophenyl

Me

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

F

9-5789

2-chloropyridin-3-yl

Me

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

F

9-5790

phenyl

Me

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

9-5791

3-cyanophenyl

Me

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

9-5792

4-cyanophenyl

Me

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

9-5793

2-chloropyridin-3-yl

Me

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

9-5794

phenyl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-5814

3-cyanophenyl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-5815

4-cyanophenyl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-5830

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

9-5872

phenyl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-5892

3-cyanophenyl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-5893

4-cyanophenyl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-5908

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

9-5950

phenyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

9-5970

3-cyanophenyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

9-5971

4-cyanophenyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

9-5986

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

9-6028

phenyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-6048

3-cyanophenyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-6049

4-cyanophenyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-6064

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

9-6106

phenyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

I

9-6126

3-cyanophenyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

I

9-6127

4-cyanophenyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

I

9-6142

2-chloropyridin-3-yl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

I

9-6184

phenyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

9-6204

3-cyanophenyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

9-6205

4-cyanophenyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

9-6220

2-chloropyridin-3-yl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

9-6458

phenyl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

9-6478

3-cyanophenyl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

9-6479

4-cyanephenyl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

9-6494

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

9-6536

phenyl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

9-6556

3-cyanophenyl

Me

Me

F

F

H

H

Cl

Cl

nonafluoro-2-butyl

H

OCF3

9-6557

4-cyanophenyl

Me

Me

F

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

9-6572

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

9-6614

phenyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

9-6634

3-cyanophenyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

9-6635

4-cyanophenyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

9-6650

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

9-6692

phenyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

9-6712

3-cyanophenyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

9-6713

4-cyanophenyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

9-6728

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

9-6770

phenyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

9-6790

3-cyanophenyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

9-6791

4-cyanophenyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

9-6806

2-chloropyridin-3-yl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

9-6848

phenyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

9-6868

3-cyanophenyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

9-6869

4-cyanophenyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

9-6884

2-chloropyridin-3-yl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

If

OCF3

9-7122

phenyl

Me

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

CF3

9-7123

phenyl

Me

Me

F

F

H

H

Cl

Cl

heptafluoroisopropyl

H

CF3

9-7143

3-cyanophenyl

Me

Me

F

F

H

H

Cl

Cl

heptafluoroisopropyl

H

CF3

9-7144

4-cyanophenyl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-7159

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

9-7201

phenyl

Me

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

9-7202

phenyl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-7222

3-cyanophenyl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-7223

4-cyanophenyl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-7238

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

9-7280

phenyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-7300

3-cyanophenyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-7301

4-cyanophenyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-7316

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

9-7358

phenyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-7378

3-cyanophenyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-7379

4-cyanophenyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-7394

2-chloropyridin-3-yl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

9-7436

phenyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

9-7456

3-cyanophenyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

9-7457

4-cyanophenyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

9-7472

2-chloropyridin-3-yl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

9-7514

phenyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-7534

3-cyanophenyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-7535

4-cyanophenyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-7550

2-chloropyridin-3-yl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

9-7788

phenyl

Me

Me

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

9-7819

2-chloropyridin-3-yl

Me

Me

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

9-7844

phenyl

Me

Me

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

9-7875

2-chloropyridin-3-yl

Me

Me

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

9-7900

phenyl

Me

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

9-7931

2-chloropyridin-3-yl

Me

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

9-7956

phenyl

Me

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

9-7987

2-chloropyridin-3-yl

Me

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

9-8012

phenyl

Me

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-8032

3-cyanophenyl

Me

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-8033

4-cyanophenyl

Me

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-8048

2-chloropyridin-3-yl

Me

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

9-8080

phenyl

Me

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-8100

3-cyanophenyl

Me

Me

F

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

9-8101

4-cyanophenyl

Me

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-8116

2-chloropyridin-3-yl

Me

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-8344

phenyl

Me

Me

F

F

F

H

Cl

H

pentafluoroethyl

H

Cl

9-8345

phenyl

Me

Me

F

F

F

H

Br

H

heptafluoroisopropyl

H

Br

9-8346

phenyl

Me

Me

F

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

9-8347

phenyl

Me

Me

F

F

F

H

I

H

heptafluoroisopropyl

H

CF3

9-8348

phenyl

Me

Me

F

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

9-8349

phenyl

Me

Me

F

F

F

H

I

H

nonafluoro-2-butyl

H

I

9-8350

phenyl

Me

Me

F

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8351

phenyl

Me

Me

F

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

9-8352

phenyl

Me

Me

F

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-8353

phenyl

Me

Me

H

H

F

H

Cl

H

pentafluoroethyl

H

Cl

9-8354

phenyl

Me

Me

H

H

F

H

Br

H

heptafluoroisopropyl

H

Br

9-8355

phenyl

Me

Me

H

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

9-8356

phenyl

Me

Me

H

H

F

H

I

H

heptafluoroisopropyl

H

CF3

9-8357

phenyl

Me

Me

H

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

9-8358

phenyl

Me

Me

H

H

F

H

I

H

nonafluoro-2-butyl

H

I

9-8359

phenyl

Me

Me

H

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8360

phenyl

Me

Me

H

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

9-8361

phenyl

Me

Me

H

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-8362

phenyl

Me

Me

H

H

H

F

Cl

H

pentafluoroethyl

H

Cl

9-8363

phenyl

Me

Me

H

H

H

F

Br

H

heptafluoroisopropyl

H

Br

9-8364

phenyl

Me

Me

H

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

9-8365

phenyl

Me

Me

H

H

H

F

I

H

heptafluoroisopropyl

H

CF3

9-8366

phenyl

Me

Me

H

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

9-8367

phenyl

Me

Me

H

H

H

F

I

H

nonafluoro-2-butyl

H

I

9-8368

phenyl

Me

Me

H

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8369

phenyl

Me

Me

H

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

9-8370

phenyl

Me

Me

H

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

9-8371

phenyl

Me

Me

F

H

F

H

Cl

H

pentafluoroethyl

H

Cl

9-8372

phenyl

Me

Me

F

H

F

H

Br

H

heptafluoroisopropyl

H

Br

9-8373

phenyl

Me

Me

F

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

9-8374

phenyl

Me

Me

F

H

F

H

I

H

heptafluoroisopropyl

H

CF3

9-8375

phenyl

Me

Me

F

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

9-8376

phenyl

Me

Me

F

H

F

H

I

H

nonafluoro-2-butyl

H

I

9-8377

phenyl

Me

Me

F

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8378

phenyl

Me

Me

F

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

9-8379

phenyl

Me

Me

F

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

9-8380

phenyl

Me

Me

F

H

H

F

Cl

H

pentafluoroethyl

H

Cl

9-8381

phenyl

Me

Me

F

H

H

F

Br

H

heptafluoroisopropyl

H

Br

9-8382

phenyl

Me

Me

F

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

9-8383

phenyl

Me

Me

H

F

H

F

I

H

heptafluoroisopropyl

H

CF3

9-8384

phenyl

Me

Me

H

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

9-8385

phenyl

Me

Me

H

F

H

F

I

H

nonafluoro-2-butyl

H

I

9-8386

phenyl

Me

Me

H

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8387

phenyl

Me

Me

H

F

H

F

Br

H

nonafluoro-2-butyl

H

Cf3

9-8388

phenyl

Me

Me

H

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

9-8389

phenyl

Me

Me

H

F

H

F

Cl

H

pentafluoroethyl

H

Cl

9-8390

phenyl

Me

Me

H

F

H

F

Br

H

heptafluoroisopropyl

H

Br

9-8391

phenyl

Me

Me

H

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

9-8392

phenyl

Me

Me

H

F

H

F

I

H

heptafluoroisopropyl

H

CF3

9-8393

phenyl

Me

Me

H

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

9-8394

phenyl

Me

Me

H

F

H

F

I

H

nonafluoro-2-butyl

H

I

9-8395

phenyl

Me

Me

H

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8396

phenyl

Me

Me

H

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

9-8397

phenyl

Me

Me

H

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

9-8398

phenyl

Me

Me

H

F

H

F

Cl

H

pentafluoroethyl

H

Cl

9-8399

phenyl

Me

Me

H

F

H

F

Br

H

heptafluoroisopropyl

H

Br

9-8400

phenyl

Me

Me

H

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

9-8401

phenyl

Me

Me

H

F

H

F

I

H

heptafluoroisopropyl

H

CF3

9-8402

phenyl

Me

Me

H

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

9-8403

phenyl

Me

Me

H

F

H

F

I

H

nonafluoro-2-butyl

H

I

9-8404

phenyl

Me

Me

H

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8405

phenyl

Me

Me

H

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

9-8406

phenyl

Me

Me

H

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

9-8407

phenyl

Me

Me

H

H

F

F

Cl

H

pentafluoroethyl

H

Cl

9-8408

phenyl

Me

Me

H

H

F

F

Br

H

heptafluoroisopropyl

H

Br

9-8409

phenyl

Me

Me

H

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

9-8410

phenyl

Me

Me

H

H

F

F

I

H

heptafluoroisopropyl

H

CF3

9-8411

phenyl

Me

Me

H

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

9-8412

phenyl

Me

Me

H

H

F

F

I

H

nonafluoro-2-butyl

H

I

9-8413

phenyl

Me

Me

H

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8414

phenyl

Me

Me

H

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

9-8415

phenyl

Me

Me

H

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

9-8416

phenyl

Me

Me

F

F

H

F

Cl

H

pentafluoroethyl

H

Cl

9-8417

phenyl

Me

Me

F

F

H

F

Br

H

heptafluoroisopropyl

H

Br

9-8418

phenyl

Me

Me

F

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

9-8419

phenyl

Me

Me

F

F

H

F

I

H

heptafluoroisopropyl

H

CF3

9-8420

phenyl

Me

Me

F

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

9-8421

phenyl

Me

Me

F

F

H

F

I

H

nonafluoro-2-butyl

H

I

9-8422

phenyl

Me

Me

F

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8423

phenyl

Me

Me

F

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

9-8424

phenyl

Me

Me

F

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

9-8425

phenyl

Me

Me

F

H

F

F

Cl

H

pentafluoroethyl

H

Cl

9-8426

phenyl

Me

Me

F

H

F

F

Br

H

heptafluoroisopropyl

H

Br

9-8427

phenyl

Me

Me

F

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

9-8428

phenyl

Me

Me

F

H

F

F

I

H

heptafluoroisopropyl

H

CF3

9-8429

phenyl

Me

Me

F

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

9-8430

phenyl

Me

Me

F

H

F

F

I

H

nonafluoro-2-butyl

H

I

9-8431

phenyl

Me

Me

F

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8432

phenyl

Me

Me

F

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

9-8433

phenyl

Me

Me

F

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

9-8434

phenyl

Me

Me

H

F

F

F

Cl

H

pentafluoroethyl

H

Cl

9-8435

phenyl

Me

Me

H

F

F

F

Br

H

heptafluoroisopropyl

H

Br

9-8436

phenyl

Me

Me

H

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

9-8437

phenyl

Me

Me

H

F

F

F

I

H

heptafluoroisopropyl

H

CF3

9-8438

phenyl

Me

Me

H

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

9-8439

phenyl

Me

Me

H

F

F

F

I

H

nonafluoro-2-butyl

H

I

9-8440

phenyl

Me

Me

H

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8441

phenyl

Me

Me

H

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

9-8442

phenyl

Me

Me

H

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

9-8443

phenyl

Me

Me

F

F

F

F

Cl

H

pentafluoroethyl

H

Cl

9-8444

phenyl

Me

Me

F

F

F

F

Br

H

heptafluoroisopropyl

H

Br

9-8445

phenyl

Me

Me

F

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

9-8446

phenyl

Me

Me

F

F

F

F

I

H

heptafluoroisopropyl

H

CF3

9-8447

phenyl

Me

Me

F

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

9-8448

phenyl

Me

Me

F

F

F

F

I

H

nonafluoro-2-butyl

H

I

9-8449

phenyl

Me

Me

F

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

9-8450

phenyl

Me

Me

F

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

9-8451

phenyl

Me

Me

F

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 10

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

10-9

3-bromophenyl

H

Et

H

H

H

H

Cl

F

nonafluoro-2-butyl

F

Cl

10-39

2-iodopyridin-3-yl

H

H

H

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

I

10-148

2-chlorophenyl

H

H

H

H

H

H

F

Br

heptafluoroisopropyl

H

CF3

10-153

4-bromophenyl

H

H

H

H

H

H

Cl

F

heptafluoroisopropyl

Cl

CF3

10-167

3,4-dichlorophenyl

H

H

H

H

H

H

Cl

I

nonafluoro-2-butyl

I

CF3

10-168

2,4-dichlorophenyl

H

H

H

H

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

10-169

2-chloro-4-fluorophenyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

10-170

2-chloro-4,5-difluorophenyl

i-Pr

H

H

H

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

10-171

4-bromo-2-chlorophenyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

10-182

2-iodopyridin-3-yl

H

H

H

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

10-183

2-(trifluoromethyl) pyridin-3-yl

H

H

H

H

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

10-189

6-iodopyridin-3-yl

H

H

H

H

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

10-190

6-(trifluoromethyl) pyridin-3-yl

H

H

H

H

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

10-196

5-bromopyridin-3-yl

H

H

H

H

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

10-197

5-iodopyridin-3-yl

H

H

H

H

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

10-203

4-bromopyridin-3-yl

Me

n-Pr

H

H

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

10-204

4-iodopyridin-3-yl

H

H

H

H

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

10-210

pyridin-4-yl

H

H

H

Fl

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

10-211

2-chloropyridin-4-yl

H

H

H

H

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

10-217

pyridin-2-yl

H

H

H

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

10-218

3-chloropyridin-2-yl

H

H

H

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

10-224

2-fluorophenyl

H

H

H

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

10-225

3-fluorophenyl

H

H

H

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

10-231

3-bromophenyl

H

H

H

H

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

10-232

4-bromophenyl

H

H

H

H

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

10-238

(4-trifluoromethyl) phenyl

Et

i-Pr

H

H

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

10-239

2-nitrophenyl

H

H

H

H

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

10-245

4-cyanophenyl

H

H

H

H

H

H

I

Br

heptafluoroisopropyl

Me

CF3

10-246

2,6-difluorophenyl

H

H

H

H

H

H

I

Br

heptafluoroisopropyl

Et

CF3

10-252

2-bromo-4-chlorophenyl

n-Pr

Me

H

H

H

H

I

I

heptafluoroisopropyl

Me

CF3

10-253

2-bromo-4-fluorophenyl

H

H

H

H

H

H

I

I

heptafluoroisopropyl

Et

CF3

10-259

2-fluoropyridin-3-yl

H

H

H

H

H

H

I

Me

heptafluoroisopropyl

F

C2F5

10-260

2-chloropyridin-3-yl

H

H

H

H

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

10-263

2-(triluoromethyl) pyridin-3-yl

H

H

H

H

H

H

I

Et

nonafluoro-2-butyl

F

CF3

10-264

2-nitropyridin-3-yl

H

H

H

H

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

10-267

6-chloropyridin-3-yl

H

H

H

H

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

10-268

6-bromopyridin-3-yl

H

H

H

H

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

10-271

6-nitropyridin-3-yl

H

H

H

H

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

10-272

6-cyanopyridin-3-yl

H

H

H

H

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

10-275

5-bromopyridin-3-yl

H

H

H

H

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

10-276

5-iodopyridin-3-yl

H

H

H

H

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

10-279

5-cyanopyr4in-3-yl

H

H

H

H

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

10-280

4-fluoropyridin-3-yl

H

H

H

H

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

10-283

4-iodopyridin-3-yl

i-Pr

n-Pr

H

H

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

10-284

4-(trifluoromethyl) pyridin-3-yl

H

H

H

H

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

10-295

3-bromophenyl

H

Et

H

H

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

10-325

2-iodopyridin-3-yl

H

H

H

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

10-438

3-bromophenyl

H

Et

H

H

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

10-468

2-iodopyridin-3-yl

H

H

H

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

10-581

3-bromophenyl

H

Et

H

H

H

H

CF3

F

heptafluoroisopropyl

F

CF3

10-611

2-iodopyridin-3-yl

H

H

H

H

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

10-724

3-bromophenyl

H

Et

F

H

H

H

Cl

F

heptafluoroisopropyl

F

Cl

10-754

2-iodopyridin-3-yl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

I

10-859

phenyl

H

H

F

H

H

H

Cl

F

heptafluoroisopropyl

H

CF3

10-860

2-fluorophenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

F

CF3

10-861

3-fluorophenyl

H

Me

F

H

H

H

Cl

Cl

heptafluoroisopropyl

H

CF3

10-862

4-fluorophenyl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

Cl

CF3

10-863

2-chlorophenyl

H

H

F

H

H

H

F

Br

heptafluoroisopropyl

H

CF3

10-864

3-chlorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

Br

CF3

10-865

4-chlorophenyl

Et

H

F

H

H

H

Cl

I

heptafluoroisopropyl

H

C2F5

10-866

2-bromophenyl

H

H

F

H

H

H

Cl

H

heptafluorolsopropyl

I

CF3

10-867

3-bromophenyl

H

Et

F

H

H

H

Cl

F

heptafluoroisopropyl

F

CF3

10-868

4-bromophenyl

H

H

F

H

H

H

Cl

F

heptafluoroisopropyl

Cl

CF3

10-869

2-iodophenyl

H

H

F

H

H

H

Cl

F

heptafluoroisopropyl

Br

CF3

10-870

3-iodophenyl

Et

Et

F

H

H

H

Cl

F

pentafluoroethyl

I

C2F5

10-871

4-iodophenyl

H

H

F

H

H

H

Cl

Cl

pentafluoroethyl

F

CF3

10-872

(2-trifluoromethyl) phenyl

H

H

F

H

H

H

Cl

Cl

heptafluoroisopropyl

Cl

CF3

10-873

(3-trifluoromethyl) phenyl

n-Pr

H

F

H

H

H

Cl

Cl

heptafluoroisopropyl

Br

CF3

10-874

(4-trifluoromethyl) phenyl

H

H

F

H

H

H

Cl

Cl

heptafluoroisopropyl

I

n-C3F7

10-875

2-nitrophenyl

H

n-Pr

F

H

H

H

Cl

Br

heptafluoroisopropyl

F

CF3

10-876

3-nitrophenyl

H

H

F

H

H

H

Cl

Br

heptafluoroisopropyl

Cl

CF3

10-877

4-nitrophenyl

H

H

F

H

H

H

Cl

Br

heptafluoroisopropyl

Br

CF3

10-878

2-cyanophenyl

n-Pr

n-Pr

F

H

H

H

Cl

Br

pentafluoroethyl

I

CF3

10-879

3-cyanophenyl

H

H

F

H

H

H

F

I

nonafluoro-2-butyl

F

CF3

10-880

4-cyanophenyl

H

H

F

H

H

H

Cl

I

nonafluoro-2-butyl

Cl

CF3

10-881

2,6-difluorophenyl

H

H

F

H

H

H

Cl

I

nonafluoro-2-butyl

Br

CF3

10-882

3,4-dichlorophenyl

H

H

F

H

H

H

Cl

I

nonafluoro-2-butyl

I

CF3

10-883

2,4-dichlorophenyl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

10-884

2-chloro-4-fluorophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

10-885

2-chloro-4,5-difluorophenyl

i-Pr

H

F

H

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

10-886

4-bromo-2-chlorophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

10-887

2-bromo-4-chlorophenyl

H

H

F

H

H

H

Cl

n-Pr

nonafluoro-2-butyl

H

CF3

10-888

2-bromo-4-fluorophenyl

H

i-Pr

F

H

H

H

Cl

H

nonafluoro-2-butyl

n-Pr

CF3

10-889

2-chloro-4-nitrophenyl

i-Pr

i-Pr

F

H

H

H

Cl

i-Pr

nonafluoro-2-butyl

H

CF3

10-890

3,5-dicyanophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

i-Pr

CF3

10-891

4-cyano-2-fluorophenyl

H

H

F

H

H

H

Cl

n-Bu

nonafluoro-2-butyl

H

CF3

10-892

2-chloro-4-cyanophenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

n-Bu

CF3

10-893

pyridin-3-yl

H

H

F

H

H

H

Cl

i-Bu

nonafluoro-2-butyl

H

CF3

10-894

2-fluoropyridin-3-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

i-Bu

CF3

10-895

2-chloropyridin-3-yl

H

H

F

H

H

H

Cl

s-Bu

nonafluoro-2-butyl

H

C2F5

10-896

2-bromopyridin-3-yl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

s-Bu

CF3

10-897

2-iodopyridin-3-yl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

10-898

2-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

10-899

2-nitropyridin-3-yl

C(O)Me

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

n-Pr

CF3

10-900

2-cyanopyridin-3-yl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

i-Pr

CF3

10-901

6-fluoropyridin-3-yl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

n-Bu

CF3

10-902

6-chloropyridin-3-yl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

i-Bu

CF3

10-903

6-bromopyridin-3-yl

H

C(O)Me

F

H

H

H

Cl

Me

nonafluoro-2-butyl

s-Bu

CF3

10-904

6-iodopyridin-3-yl

H

H

F

H

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

10-905

6-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

10-906

6-nitropyridin-3-yl

C(O)Me

C(O)Me

F

H

H

H

Cl

Et

nonafluoro-2-butyl

n-Pr

CF3

10-907

6-cyanopyridin-3-yl

H

H

F

H

H

H

Cl

Et

nonafluoro-2-butyl

i-Pr

CF3

10-908

phenyl

H

H

F

H

H

H

Br

Et

nonafluoro-2-butyl

n-Bu

CF3

10-909

5-fluoropyridin-3-yl

H

H

F

H

H

H

Br

Et

heptafluoroisopropyl

i-Bu

CF3

10-910

5-chloropyridin-3yl

H

H

F

H

H

H

Br

Et

heptafluoroisopropyl

s-Bu

CF3

10-911

5-bromopyridin-3-yl

H

H

F

H

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

10-912

5-iodopyridin-3-yl

H

H

F

H

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

10-913

5-(trifluoromethyl) pyridin-3-yl

Me

Et

F

H

H

H

Br

n-Pr

pentafluoroethyl

n-Pr

CF3

10-914

5-nitropyridin-3-yl

H

H

F

H

H

H

Br

n-Pr

heptafluoroisopropyl

i-Pr

CF3

10-915

5-cyanopyridin-3-yl

H

H

F

H

H

H

Br

n-Pr

pentafluoroethyl

n-Bu

CF3

10-916

4-fluoropyridin-3-yl

H

H

F

H

H

H

Br

n-Pr

heptafluoroisopropyl

i-Bu

CF3

10-917

4-chloropyridin-3-yl

H

H

F

H

H

H

Br

n-Pr

heptafluoroisopropyl

s-Bu

CF3

10-918

4-bromopyridin-3-yl

Me

n-Pr

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

10-919

4-iodopyridin-3-yl

H

H

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

10-920

4-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

n-Pr

CF3

10-921

4-nitropyridin-3-yl

H

H

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

i-Pr

CF3

10-922

4-cyanopyridin-3-yl

H

H

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

n-Bu

CF3

10-923

2,6-dichloropyridin-3-yl

H

H

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

i-Bu

CF3

10-924

pyridin-3-yl N-oxide

Me

i-Pr

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

s-Bu

CF3

10-925

pyridin-4-yl

H

H

F

H

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

10-926

2-chloropyridin-4-yl

H

H

F

H

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

10-927

3-bromopyridin-4-yl

H

H

F

H

H

H

Br

n-Bu

heptafluoroisopropyl

n-Pr

CF3

10-928

3,5-dichloropyridin-4-yl

H

H

F

H

H

H

Br

n-Bu

nonafluoro-2-butyl

i-Pr

CF3

10-929

3-(trifluoromethyl) pyridin-4-yl

H

H

F

H

H

H

Br

n-Bu

nonafluoro-2-butyl

n-Bu

CF3

10-930

2,5-dicyanopyridin-4-yl

H

H

F

H

H

H

Br

n-Bu

nonafluoro-2-butyl

i-Bu

CF3

10-931

pyridin-4-yl N-oxide

Me

C(O)Me

F

H

H

H

Br

n-Bu

nonafluoro-2-butyl

s-Bu

CF3

10-932

pyridin-2-yl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

10-933

3-chloropyridin-2-yl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

10-934

4-bromopyridin-2-yl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

n-Pr

CF3

10-935

5-iodopyridin-2-yl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

i-Pr

CF3

10-936

6-chloropyridin-2-yl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

n-Bu

CF3

10-937

4-cyanopyridin-2-yl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

i-Bu

CF3

10-938

phenyl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

s-Bu

C2F5

10-939

2-fluorophenyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

10-940

3-fluorophenyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

10-941

4-fluorophenyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

n-Pr

CF3

10-942

2-chlorophenyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

i-Pr

CF3

10-943

3-chlorophenyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

n-Bu

CF3

10-944

4-chlorophenyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

i-Bu

CF3

10-945

2-bromophenyl

Et

Me

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

s-Bu

CF3

10-946

3-bromophenyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

10-947

4-bromophenyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

10-948

2-iodophenyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

n-Pr

CF3

10-949

3-iodophenyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

i-Pr

CF3

10-950

4-iodophenyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

n-Bu

CF3

10-951

(2-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

i-Bu

CF3

10-952

(3-trifluoromethyl) phenyl

Et

n-Pr

F

H

H

H

Br

F

nonafluoro-2-butyl

s-Bu

CF3

10-953

(4-trifluoromethyl) phenyl

Et

i-Pr

F

H

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

10-954

2-nitrophenyl

H

H

F

H

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

10-955

phenyl

H

H

F

H

H

H

I

Cl

pentafluoroethyl

n-Pr

i-C3F7

10-956

3-ntrophenyl

H

H

F

H

H

H

I

Cl

heptafluoroisopropyl

i-Pr

CF3

10-957

4-nitrophenyl

H

H

F

H

H

H

I

Cl

heptafluoroisopropyl

n-Bu

CF3

10-958

2-cyanophenyl

Et

C(O)Me

F

H

H

H

I

Cl

heptafluoroisopropyl

i-Bu

CF3

10-959

3-cyanophenyl

H

H

F

H

H

H

I

Cl

heptafluoroisopropyl

s-Bu

CF3

10-960

4-cyanophenyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

Me

CF3

10-961

2,6-difluorophenyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

Et

CF3

10-962

3,4-dichlorophenyl

H

H

F

H

H

H

I

Br

pentafluoroethyl

n-Pr

CF3

10-963

2,4-dichlorophenyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

i-Pr

CF3

10-964

2-chloro-4-fluorophenyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

n-Bu

CF3

10-955

2-chloro-4,5-difluorophenyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

i-Bu

CF3

10-966

4-bromo-2-chlorophenyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

s-Bu

CF3

10-967

2-bromo-4-chlorophenyl

n-Pr

Me

F

H

H

H

I

I

heptafluoroisopropyl

Me

CF3

10-968

2-bromo-4-fluorophenyl

H

H

F

H

H

H

I

I

heptafluoroisopropyl

Et

CF3

10-969

2-chloro-4-nitrophenyl

n-Pr

Et

F

H

H

H

I

I

heptafluoroisopropyl

n-Pr

CF3

10-970

3,5-dicyanophenyl

H

H

F

H

H

H

I

I

heptafluoroisopropyl

i-Pr

CF3

10-971

4-cyano-2-fluorophenyl

H

H

F

H

H

H

I

I

heptafluoroisopropyl

n-Bu

CF3

10-972

2-chloro-4-cyanophenyl

H

H

F

H

H

H

I

I

heptafluoroisopropyl

i-Bu

CF3

10-973

pyridin-3-yl

H

H

F

H

H

H

I

I

heptafluoroisopropyl

s-Bu

CF3

10-974

2-fluoropyridin-3-yl

H

H

F

H

H

H

I

Me

heptafluoroisopropyl

F

C2F5

10-975

2-chloropyridin-3-yl

H

H

F

H

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

10-976

2-bromopyridin-3-yl

H

H

F

H

H

H

I

Me

nonafluoro-2-butyl

Br

n-C3F7

10-977

2-iodopyridin-3-yl

H

H

F

H

H

H

I

Me

nonafluoro-2-butyl

I

i-C3F7

10-978

2-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

Et

nonafluoro-2-butyl

F

CF3

10-979

2-nitropyridin-3-yl

H

H

F

H

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

10-980

2-cyanopyridin-3-yl

H

H

F

H

H

H

I

Et

nonafluoro-2-butyl

Br

CF3

10-981

6-fluoropyridin-3-yl

n-Pr

i-Pr

F

H

H

H

I

Et

nonafluoro-2-butyl

I

C2F5

10-982

6-chloropyridin-3-yl

H

H

F

H

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

10-983

6-bromopyridin-3-yl

H

H

F

H

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

10-984

6-iodopyridin-3-yl

H

H

F

H

H

H

I

n-Pr

nonafluoro-2-butyl

Br

CF3

10-985

6-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

n-Pr

nonafluoro-2-butyl

I

n-C3F7

10-986

6-nitropyridin-3-yl

H

H

F

H

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

10-987

6-cyanopyridin-3-yl

H

H

F

H

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

10-988

5-fluoropyridin-3-yl

n-Pr

C(O)Me

F

H

H

H

I

i-Pr

nonafluoro-2-butyl

Br

CF3

10-989

5-chloropyridin-3-yl

H

H

F

H

H

H

I

i-Pr

nonafluoro-2-butyl

I

CF3

10-990

5-bromopyridin-3-yl

H

H

F

H

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

10-991

5-iodopyridin-3-yl

H

H

F

H

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

10-992

5-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

n-Bu

nonafluoro-2-butyl

Br

CF3

10-993

5-nitropyridin-3-yl

i-Pr

Me

F

H

H

H

I

n-Bu

nonafluoro-2-butyl

I

CF3

10-994

5-cyanopyridin-3-yl

H

H

F

H

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

10-995

4-fluoropyrdin-3-yl

H

H

F

H

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

10-996

4-chloropyridin-3-yl

H

H

F

H

H

H

I

i-Bu

nonafluoro-2-butyl

Br

CF3

10-997

4-bromopyridin-3-yl

i-Pr

Et

F

H

H

H

I

i-Bu

nonafluoro-2-butyl

I

CF3

10-998

4-iodopyridin-3-yl

i-Pr

n-Pr

F

H

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

10-999

4-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

10-1000

4-nitropyridin-3-yl

i-Pr

C(O)Me

F

H

H

H

I

s-Bu

nonafluoro-2-butyl

Br

CF3

10-1001

4-cyanopyridin-3-yl

H

H

F

H

H

H

I

s-Bu

nonafluoro-2-butyl

I

CF3

10-1010

3-bromophenyl

H

Et

F

H

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

10-1040

2-iodopyridin-3-yl

H

H

F

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

10-1153

3-bromophenyl

H

Et

F

H

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

10-1183

2-iodopyridin-3-yl

H

H

F

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

10-1296

3-bromophenyl

H

Et

F

H

H

H

CF3

F

heptafluoroisopropyl

F

CF3

10-1326

2-iodopyridin-3-yl

H

H

F

H

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

10-1439

3-bromophenyl

H

Et

H

F

H

H

Cl

F

heptafluoroisopropyl

F

Cl

10-1469

2-iodopyridin-3-yl

H

H

H

F

H

H

Cl

Me

nonafluoro-2-butyl

Me

I

10-1582

3-bromophenyl

H

Et

H

F

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

10-1612

2-iodopyridin-3-yl

H

H

H

F

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

10-1726

4-bromophenyl

H

H

H

F

H

H

Cl

F

heptafluaroisopropyl

Cl

CF3

10-1733

2-nitrophenyl

H

n-Pr

H

F

H

H

Cl

Br

heptafluoroisopropyl

F

CF3

10-1741

2,4-dichlorophenyl

H

H

H

F

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

10-1742

2-chloro-4-fluorophenyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

10-1743

2-chloro-4,5-difluorophenyl

i-Pr

H

H

F

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

10-1744

4-bromo-2-chlorophenyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

10-1755

2-iodopyridin-3-yl

H

H

H

F

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

10-1756

2-(trifluoromethyl) pyridin-3-yl

H

H

H

F

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

10-1762

6-iodopyridin-3-yl

H

H

H

F

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

10-1763

6-(trifluoromethyl) pyridin-3-yl

H

H

H

F

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

10-1769

5-bromopyridin-3-yl

H

H

H

F

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

10-1770

5-iodopyridin-3-yl

H

H

H

F

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

10-1776

4-bromopyridin-3-yl

Me

n-Pr

H

F

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

10-1777

4-iodopyridin-3-yl

H

H

H

F

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

10-1783

pyridin-4-yl

H

H

H

F

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

10-1784

2-chloropyridin-4-yl

H

H

H

F

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

10-1790

pyridin-2-yl

H

H

H

F

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

10-1791

3-chloropyridin-2-yl

H

H

H

F

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

10-1797

2-fluorophenyl

H

H

H

F

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

10-1798

3-fluorophenyl

H

H

H

F

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

10-1804

3-bromophenyl

H

H

H

F

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

10-1805

4-bromophenyl

H

H

H

F

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

10-1811

(4-trifluoromethyl) phenyl

Et

i-Pr

H

F

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

10-1812

2-nitrophenyl

H

H

H

F

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

10-1818

4-cyanophenyl

H

H

H

F

H

H

I

Br

heptafluoroisopropyl

Me

CF3

10-1819

2,6-difluorophenyl

H

H

H

F

H

H

I

Br

heptafluoroisopropyl

Et

CF3

10-1825

2-bromo-4-chlorophenyl

n-Pr

Me

H

F

H

H

I

I

heptafluoroisopropyl

Me

CF3

10-1826

2-bromo-4-fluorophenyl

H

H

H

F

H

H

I

I

heptafluoroisopropyl

Et

CF3

10-1832

2-fluoropyridin-3-yl

H

H

H

F

H

H

I

Me

heptafluoroisopropyl

F

C2F5

10-1833

2-chloropyridin-3-yl

H

H

H

F

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

10-1834

2-bromopyridin-3-yl

H

H

H

F

H

H

I

Me

nonafluoro-2-butyl

Br

n-C3F7

10-1837

2-nitropyridin-3-yl

H

H

H

F

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

10-1838

2-cyanopyridin-3-yl

H

H

H

F

H

H

I

Et

nonafluoro-2-butyl

Br

CF3

10-1841

6-bromopyridin-3-yl

H

H

H

F

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

10-1842

6-iodopyridin-3-yl

H

H

H

F

H

H

I

n-Pr

nonafluoro-2-butyl

Br

CF3

10-1845

6-cyanopyridin-3-yl

H

H

H

F

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

10-1846

5-fluoropyridin-3-yl

n-Pr

C(O)Me

H

F

H

H

I

i-Pr

nonafluoro-2-butyl

Br

CF3

10-1849

5-iodopyridin-3-yl

H

H

H

F

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

10-1850

5-(trifluoromethyl) pyridin-3-yl

H

H

H

F

H

H

I

n-Bu

nonafluoro-2-butyl

Br

CF3

10-1853

4-fluoropyridin-3-yl

H

H

H

F

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

10-1854

4-chloropyridin-3-yl

H

H

H

F

H

H

I

i-Bu

nonafluoro-2-butyl

Br

CF3

10-1857

4-(trifluoromethyl) pyridin-3-yl

H

H

H

F

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

10-1858

4-nitropyridin-3-yl

i-Pr

C(O)Me

H

F

H

H

I

s-Bu

nonafluoro-2-butyl

Br

CF3

10-1898

2-iodopyridin-3-yl

H

H

H

F

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

10-2011

3-bromophenyl

H

Et

H

F

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

10-2041

2-iodopyridin-3-yl

H

H

H

F

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

10-2154

3-bromophenyl

H

Et

H

F

H

H

CF3

F

heptafluoroisopropyl

F

CF3

10-2184

2-iodopyridin-3-yl

H

H

H

F

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

10-2297

3-bromophenyl

H

Et

H

F

H

H

Cl

F

heptafluoroisopropyl

F

Cl

10-2327

2-iodopyridin-3-yl

H

H

H

F

H

H

Cl

Me

nonafluoro-2-butyl

Me

I

10-2440

3-bromophenyl

H

Et

H

F

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

10-2470

2-iodopyridin-3-yl

H

H

F

F

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

10-2584

4-bromophenyl

H

H

F

F

H

H

Cl

F

heptafluoroisopropyl

Cl

OF3

10-2594

2-cyanophenyl

n-Pr

n-Pr

F

F

H

H

Cl

Br

pentafluoroethyl

I

CF3

10-2599

2,4-dichlorophenyl

H

H

F

F

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

10-2600

2-chloro-4-fluorophenyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

10-2613

2-iodopyridin-3-yl

H

H

F

F

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

10-2614

2-(trifluoromethyl) pyridin-3-yl

H

H

F

F

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

10-2620

6-iodopyridin-3-yl

H

H

F

F

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

10-2621

6-(trifluoromethyl) pyridin-3-yl

H

H

F

F

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

10-2627

5-bromopyridin-3-yl

H

H

F

F

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

10-2628

5-iodopyridin-3-yl

H

H

F

F

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

10-2634

4-bromopyridin-3-yl

Me

n-Pr

F

F

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

10-2635

4-iodopyridin-3-yl

H

H

F

F

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

10-2641

pyridin-4-yl

H

H

F

F

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

10-2642

2-chloropyridin-4-yl

H

H

F

F

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

10-2648

pyridin-2-yl

H

H

F

F

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

10-2649

3-chloropyridin-2-yl

H

H

F

F

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

10-2655

2-fluorophenyl

H

H

F

F

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

10-2656

3-fluorophenyl

H

H

F

F

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

10-2662

3-bromophenyl

H

H

F

F

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

10-2663

4-bromophenyl

H

H

F

F

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

10-2669

(4-fluoromethyl) phenyl

Et

i-Pr

F

F

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

10-2670

2-nitrophenyl

H

H

F

F

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

10-2676

4-cyanophenyl

H

H

F

F

H

H

I

Br

heptafluoroisopropyl

Me

CF3

10-2677

2,6-difluorophenyl

H

H

F

F

H

H

I

Br

heptafluoroisopropyl

Et

CF3

10-2683

2-bromo-4-chlorophenyl

n-Pr

Me

F

F

H

H

I

I

heptafluoroisopropyl

Me

CF3

10-2684

2-bromo-4-fluorophenyl

H

H

F

F

H

H

I

I

heptafluoroisopropyl

Et

CF3

10-2690

2-fluoropyridin-3-yl

H

H

F

F

H

H

I

Me

heptafluoroisopropyl

F

C2F5

10-2691

2-chloropyridin-3-yl

H

H

F

F

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

10-2694

2-(trifluoromethyl) pyridin-3-yl

H

H

F

F

H

H

I

Et

nonafluoro-2-butyl

F

CF3

10-2695

2-nitropyridin-3-yl

H

H

F

F

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

10-2698

6-chloropyridin-3-yl

H

H

F

F

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

10-2699

6-bromopyridin-3-yl

H

H

F

F

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

10-2702

6-nitropyridin-3-yl

H

H

F

F

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

10-2703

6-cyanopyridin-3-yl

H

H

F

F

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

10-2706

5-bromopyridin-3-yl

H

H

F

F

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

10-2707

5-iodopyridin-3-yl

H

H

F

F

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

10-2710

5-cyanopyridin-3-yl

H

H

F

F

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

10-2711

4-fluoropyridin-3-yl

H

H

F

F

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

10-2714

4-iodopyridin-3-yl

i-Pr

n-Pr

F

F

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

10-2715

4-(fluoromethyl) pyridin-3-yl

H

H

F

F

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

10-2726

3-bromophenyl

H

Et

F

F

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

10-2756

2-iodopyridin-3-yl

H

H

F

F

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

10-2869

3-bromophenyl

H

H

F

F

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

10-2899

2-iodopyridin-3-yl

H

H

F

F

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

10-3012

3-bromophenyl

H

H

F

F

H

H

CF3

F

heptafluoroisopropyl

F

CF3

10-3042

2-iodopyridin-3-yl

H

H

F

F

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

10-3147

phenyl

H

H

F

F

F

H

Cl

F

pentafluoroethyl

H

Cl

10-3168

phenyl

H

H

H

H

F

H

Cl

I

pentafluoroethyl

Cl

Cl

10-3189

phenyl

H

H

H

H

H

F

Cl

Me

pentafluoroethyl

n-Bu

Cl

10-3198

phenyl

H

H

F

H

F

H

Cl

Et

pentafluoroethyl

s-Bu

Cl

10-3218

phenyl

H

H

F

H

H

F

Cl

n-Bu

pentafluoroethyl

i-Bu

Cl

10-3227

phenyl

H

H

H

F

F

H

Cl

s-Bu

pentafluoroethyl

Me

Cl

10-3236

phenyl

H

H

H

F

H

F

Cl

F

pentafluoroethyl

N-pr

Cl

10-3245

phenyl

H

H

H

H

F

F

Cl

Cl

pentafluoroethyl

n-Bu

Cl

10-3254

phenyl

H

H

F

F

H

F

Cl

Br

pentafluoroethyl

s-Bu

Cl

10-3263

phenyl

H

H

F

H

F

F

Cl

Me

pentafluoroethyl

Cl

Cl

10-3272

phenyl

H

H

H

F

F

F

Cl

n-Pr

pentafluoroethyl

Br

Cl

10-3281

phenyl

i-Pr

Me

F

F

F

F

Cl

n-Bu

pentafluoroethyl

I

Cl

TABLE 11

compound

number

Q2

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

11-1

2,2,2-trichloroethyl

H

H

H

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

11-2

2,2,2-trichloroethyl

H

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

11-13

2,2,2-trichloroethyl

H

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

11-42

2,2,2-trichloroethyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

11-71

2,2,2-trichloroethyl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-100

2,2,2-trichloroethyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-129

2,2,2-trichloroethyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-158

2,2,2-trichloroethyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-189

2,2,2-trichloroethyl

H

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-218

2,2,2-trichloroethyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-247

2,2,2-trichloroethyl

H

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-260

4,4,4-trifluoro-n-butyl

H

H

H

H

H

H

Br

H

pentafluoroethyl

H

CF3

11-276

2,2,2-trichloroethyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-289

4,4,4-trifluoro-n-butyl

H

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-305

2,2,2-trichloroethyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-318

4,4,4-trifluoro-n-butyl

H

H

H

H

H

H

I

H

heptafluoroisopropyl

H

C2F5

11-334

2,2,2-trichloroethyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-347

4,4,4-trifluoro-n-butyl

H

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-363

2,2,2-trichloroethyl

H

H

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

11-392

2,2,2-tnchloroethyl

H

H

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

11-421

2,2,2-trichloroethyl

H

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

11-450

2,2,2-trichloroethyl

H

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

11-479

2,2,2-trichloroethyl

H

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-508

2,2,2-trichloroethyl

H

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-527

2,2,2-trichloroethyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

11-528

2,2,2-trichloroethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

11-529

2,2,2-trichloroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

11-530

2,2,2-trichloroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

11-531

2,2,2-trichloroethyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

11-532

2,2,2-trichloroethyl

H

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

11-543

2,2,2-trichloroethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

11-556

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

11-572

2,2,2-trichloroethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

11-585

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

Cl

H

pentafluoroethyl

H

OCF3

11-591

methyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-592

ethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-593

2-fluoroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-594

2-chloroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-595

2-bromoethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-596

2-iodoethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OC2F5

11-597

2-cyanoethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-598

2,2-difluoroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-599

2,2-dichloroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-600

2,2,2-trifluoroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-601

2,2,2-trichloroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-602

2,2,2-tribromoethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-603

n-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-604

3-fluoro-n-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-605

3-chloro-n-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-606

3-bromo-n-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-607

i-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-608

1,2-difluoro-2-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-609

1,3-difluoro-2-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-610

1,3-dichloro-2-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-611

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-612

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-613

n-butyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-614

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-615

i-butyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-616

s-butyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-617

vinyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-618

benzyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-619

phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-620

methyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-621

ethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-622

2-fluoroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-623

2-chloroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-624

2-bromoethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-625

2-iodoethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-626

2-cyanoethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-627

2,2-difluoroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-628

2,2-dichloroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-629

2,2,2-trifluoroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-630

2,2,2-trichloroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-631

2,2,2-tribromoethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-632

n-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OC2F5

11-633

3-fluoro-n-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-634

3-chloro-n-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-635

3-bromo-n-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-636

i-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-637

1,2-difluoro-2-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-638

1,3-difluoro-2-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-639

1,3-dichloro-2-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-640

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-641

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-642

n-butyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-643

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-644

i-butyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-645

s-butyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-646

vinyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-647

benzyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-648

phenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-649

methyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-650

ethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-651

2-fluoroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-652

2-chloroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-653

2-bromoethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-654

2-iodoethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-655

2-cyanoethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-656

2,2-difluoroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-657

2,2-dichloroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-658

2,2,2-trifluoroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-659

2,2,2-trichloroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-660

2,2,2-tribromoethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-661

n-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-662

3-fluoro-n-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-663

3-chloro-n-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OC2F5

11-664

3-bromo-n-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-665

i-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-666

1,2-difluoro-2-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-667

1,3-difluoro-2-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-668

1,3-dichloro-2-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-669

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-670

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-671

n-butyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-672

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-673

i-butyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-674

s-butyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-675

vinyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-676

benzyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-677

phenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-678

methyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-679

ethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-680

2-fluoroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-681

2-chloroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-682

2-bromoethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-683

2-iodoethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-684

2-cyanoethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-685

2,2-difluoroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-686

2,2-dichloroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-687

2,2,2-trifluoroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-688

2,2,2-trichloroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-689

2,2,2-tribromoethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-690

n-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-691

3-fluoro-n-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-692

3-chloro-n-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-693

3-bromo-n-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-694

i-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-695

1,2-difluoro-2-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-696

1,3-difluoro-2-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-697

12-dichloro-2-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-698

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-699

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-700

n-butyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-701

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-702

i-butyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-703

s-butyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-704

vinyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-705

benzyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OC2F5

11-706

phenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-707

2,2,2-trichloroethyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

CF3

11-708

2,2,2-trichloroethyl

H

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

11-709

methyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-710

ethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-711

2-fluoroethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-712

2-chloroethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-713

2-bromoethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-714

2-iodoethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-715

2-cyanoethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

11-716

2,2-difluoroethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-717

2,2-dichloroethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-718

2,2,2-trifluoroethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-719

2,2,2-trichloroethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-720

2,2,2-tribromoethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-721

n-propyl

H

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

11-722

3-fluoro-n-propyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-723

3-chloro-n-propyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-724

3-bromo-n-propyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-725

i-propyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

11-726

1,2-difluoro-2-propyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-727

1,3-difluoro-2-propyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-728

1,3-dichloro-2-propyl

H

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

11-729

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-730

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-731

n-butyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-732

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-733

i-butyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-734

s-butyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-735

vinyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-736

benzyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-737

phenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-738

methyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-739

ethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

11-740

2-fluoroethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-741

2-chloroethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-742

2-bromoethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-743

2-iodoethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-744

2-cyanoethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-745

2,2-difluoroethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-746

2,2-dichloroethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-747

2,2,2-trifluoroethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-748

2,2,2-trichloroethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-749

2,2,2-tribromoethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-750

n-propyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-751

3-fluoro-n-propyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-752

3-chloro-n-propyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-753

3-bromo-n-propyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-754

i-propyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-755

1,2-difluoro-2-propyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-756

1,3-difluoro-2-propyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-757

1,3-dichloro-2-propyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-758

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-759

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-760

n-butyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-761

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-762

i-butyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-763

s-butyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-764

vinyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-765

benzyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-766

phenyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-767

methyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-768

ethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-769

2-fluoroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-770

2-chloroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-771

2-bromoethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-772

2-iodoethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-773

2-cyanoethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

C2F5

11-774

2,2-difluoroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-775

2,2-dichloroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-776

2,2,2-trifluoroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-777

2,2,2-trichloroethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-778

2,2,2-tribromoethyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-779

n-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-780

3-fluoro-n-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-781

3-chloro-n-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-782

3-bromo-n-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-783

1-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-784

1,2-difluoro-2-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

n-C3F7

11-785

1,3-difluoro-2-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-786

1,3-dichloro-2-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-787

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-788

3,3,3-fluoro-n-propyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-789

n-butyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-790

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-791

i-butyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-792

s-butyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-793

vinyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-794

benzyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-795

phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-796

methyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-797

ethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-798

2-fluoroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-799

2-chloroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-800

2-bromoethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-801

2-iodoethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-802

2-cyanoethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-803

2,2-difluoroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-804

2,2-dichloroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-805

2,2,2-trifluoroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-806

2,2,2-trichloroethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-807

2,2,2-tribromoethyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-808

n-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-809

3-fluoro-n-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-810

3-chloro-n-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-811

3-bromo-n-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-812

i-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-813

1,2-difluoro-2-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-814

1,3-difluoro-2-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-815

1,3-dichloro-2-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-816

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-817

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-818

n-butyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-819

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-820

i-butyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-821

s-butyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-822

vinyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-823

benzyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-824

phenyl

H

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

i-C3F7

11-825

methyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-826

ethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-827

2-fluoroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-828

2-chloroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-829

2-bromoethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-830

2-iodoethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-831

2-cyanoethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-832

2,2-difluoroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-833

2,2-dichloroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-834

2,2,2-trifluoroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-835

2,2,2-trichloroethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-836

2,2,2-tribromoethyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-837

n-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-838

3-fluoro-n-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-839

3-chloro-n-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-840

3-bromo-n-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

C2F5

11-841

i-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-842

1,2-difluoro-2-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-843

1,3-difluoro-2-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-844

1,3-dichloro-2-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-845

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-846

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-847

n-butyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-848

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-849

i-butyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-850

s-butyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-851

vinyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-852

benzyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-853

phenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

11-854

methyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-855

ethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-856

2-fluoroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-857

2-chloroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-858

2-bromoethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-859

2-iodoethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-860

2-cyanoethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-861

2,2-difluoroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-862

2,2-dichloroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-863

2,2,2-trifluoroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-864

2,2,2-trichloroethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-865

2,2,2-tribromoethyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-866

n-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-867

3-fluoro-n-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-868

3-chloro-n-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-869

3-bromo-n-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-870

i-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-871

1,2-difluoro-2-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-872

1,3-difluoro-2-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-873

1,3-dichloro-2-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-874

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-875

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-876

n-butyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-877

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-878

i-butyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-879

s-butyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-880

vinyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

i-C3F7

11-881

benzyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-882

phenyl

H

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-893

2,2,2-trichloroethyl

H

H

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

11-922

2,2,2-trichloroethyl

H

H

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

11-951

2,2,2-trichloroethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

11-980

2,2,2-trichloroethyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

11-999

methyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1000

ethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1001

2-fluoroethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1002

2-chloroethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1003

2-bromoethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1004

2-iodoethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1005

2-cyanoethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1006

2,2-difluoroethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1007

2,2-dichloroethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1008

2,2,2-trifluoroethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1009

2,2,2-trichloroethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1010

2,2,2-tribromoethyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1011

n-propyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1012

3-fluoro-n-propyl

H

H

F

H

H

H

C2F5

H

heptafluoroisopropyl

H

CF3

11-1013

3-chloro-n-propyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1014

3-bromo-n-propyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1015

i-propyl

H

H

F

H

H

H

i-C3F7

H

heptafluoroisopropyl

H

CF3

11-1016

1,2-difluoro-2-propyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1017

1,3-di6uoro-2-propyl

H

H

F

H

H

H

CF3

H

pentafluoroethyl

H

CF3

11-1018

1,3-dichloro-2-propyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1019

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1020

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1021

n-butyl

H

H

F

H

H

H

C2F5

H

heptafluoroisopropyl

H

C2F5

11-1022

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1023

i-butyl

H

H

F

H

H

H

C2F5

H

heptafluoroisopropyl

H

n-C3F7

11-1024

s-butyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1025

vinyl

H

H

F

H

H

H

n-C3F7

H

heptafluoroisopropyl

H

CF3

11-1026

benzyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1027

phenyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1030

2-fluoroethyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1031

2-chloroethyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1032

2-bromoethyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1033

2-iodoethyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1035

2,2-difluoroethyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1036

2,2-dichloroethyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1037

2,2,2-trifluoroethyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1038

2,2,2-trichloroethyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1039

2,2,2-tribromoethyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1041

3-fluoro-n-propyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1042

3-chloro-n-propyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1043

3-bromo-n-propyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1045

1,2-difluoro-2-propyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1046

1,3-difluoro-2-propyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1047

1,3-dichloro-2-propyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1048

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1049

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

n-C3F7

H

nonafluoro-2-butyl

H

i-C3F7

11-1051

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1057

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

heptafluoroisopropyl

H

F

11-1058

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

11-1069

2,2,2-trichloroethyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

11-1098

2,2,2-trichloroethyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

11-1127

2,2,2-trichloroethyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

11-1156

2,2,2-trichloroethyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

11-1185

2,2,2-trichloroethyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

I

11-1214

2,2,2-trichloroethyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

11-1233

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

heptafluoroisopropyl

H

Cl

11-1234

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

heptafluoroisopropyl

H

Br

11-1235

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

heptafluoroisopropyl

H

I

11-1236

2,2,2-trichloroethyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Br

11-1237

2,2,2-trichloroethyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

I

11-1238

2,2,2-trichloroethyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

I

11-1239

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

Cl

11-1240

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

Br

11-1241

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

I

11-1242

2,2,2-trichloroethyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Br

11-1243

2,2,2-trichloroethyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

I

11-1244

2,2,2-trichloroethyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

I

11-1245

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

heptafluoroisopropyl

H

OCF3

11-1246

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

OCF3

11-1257

2,2,2-trichloroethyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

11-1286

2,2,2-trichloroethyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

11-1315

2,2,2-trichloroethyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-1344

2,2,2-trichloroethyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-1373

2,2,2-trichloroethyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-1402

2,2,2-trichloroethyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-1421

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

heptafluoroisopropyl

H

CF3

11-1422

2,2,2-trichloroethyl

H

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

11-1433

2,2,2-trichloroethyl

H

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-1461

2,2,2-trifluoroethyl

H

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-1491

2,2,2-trichloroethyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-1504

4,4,4-trifluoro-n-butyl

H

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-1520

2,2,2-trichloroethyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-1533

4,4,4-trifluoro-n-butyl

H

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-1548

2,2,2-trifluoroethyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

11-1562

4,4,4-trifluoro-n-butyl

H

H

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

11-1578

2,2,2-trichloroethyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-1591

4,4,4-trifluoro-n-butyl

H

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-1607

2,2,2-trichloroethyl

H

H

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

11-1636

2,2,2-trichloroethyl

H

H

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

11-1665

2,2,2-trichloroethyl

H

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

11-1694

2,2,2-trichloroethyl

H

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

11-1723

2,2,2-trichloroethyl

H

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-1752

2,2,2-trichloroethyl

H

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-1771

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

heptafluoroisopropyl

H

F

11-1772

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

11-1783

2,2,2-trichloroethyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

11-1812

2,2,2-trichloroethyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

11-1841

2,2,2-trichloroethyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

11-1870

2,2,2-trichloroethyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

11-1899

2,2,2-trichloroethyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

I

11-1928

2,2,2-trichloroethyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

11-1947

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

heptafluoroisopropyl

H

Cl

11-1948

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

heptafluoroisopropyl

H

Br

11-1949

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

heptafluoroisopropyl

H

I

11-1950

2,2,2-trichloroethyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Br

11-1951

2,2,2-trichloroethyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

I

11-1952

2,2,2-trichloroethyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

I

11-1953

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

Cl

11-1954

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

Br

11-1955

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

I

11-1956

2,2,2-trichloroethyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Br

11-1957

2,2,2-trichloroethyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

I

11-1958

2,2,2-trichloroethyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

I

11-1959

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

heptafluoroisopropyl

H

OCF3

11-1960

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

OCF3

11-1971

2,2,2-trichloroethyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

11-2000

2,2,2-trichloroethyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2029

2,2,2-trichloroethyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-2058

2,2,2-trichloroethyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-2087

2,2,2-trichloroethyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-2116

2,2,2-trichloroethyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-2135

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

heptafluoroisopropyl

H

CF3

11-2136

2,2,2-trichloroethyl

H

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

11-2147

2,2,2-trichloroethyl

H

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-2176

2,2,2-trichloroethyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-2205

2,2,2-trichloroethyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-2218

4,4,4-trifluoro-n-butyl

H

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-2234

2,2,2-trichloroethyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-2247

4,4,4-trifluoro-n-butyl

H

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-2263

2,2,2-trichloroethyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

11-2276

4,4,4-trifluoro-n-butyl

H

H

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

11-2292

2,2,2-trichloroethyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-2305

4,4,4-trifluoro-n-butyl

H

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-2321

2,2,2-trichloroethyl

H

H

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

11-2350

2,2,2-trichloroethyl

H

H

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

11-2379

2,2,2-trichloroethyl

H

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

11-2408

2,2,2-trichloroethyl

H

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

11-2437

2,2,2-trichloroethyl

H

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-2466

2,2,2-trichloroethyl

H

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-2485

2,2,2-trichloroethyl

H

H

F

F

F

H

Cl

H

pentafluoroethyl

H

Cl

11-2486

2,2,2-trichloroethyl

H

H

F

F

F

H

Br

H

heptafluoroisopropyl

H

Br

11-2487

2,2,2-trichloroethyl

H

H

F

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

11-2488

2,2,2-trichloroethyl

H

H

F

F

F

H

I

H

heptafluoroisopropyl

H

CF3

11-2489

2,2,2-trichloroethyl

H

H

F

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

11-2490

2,2,2-trichloroethyl

H

H

F

F

F

H

I

H

nonafluoro-2-butyl

H

I

11-2491

2,2,2-trichloroethyl

H

H

F

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2492

2,2,2-trichloroethyl

H

H

F

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

11-2493

2,2,2-trichloroethyl

H

H

F

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-2494

2,2,2-trichloroethyl

H

H

H

H

F

H

Cl

H

pentafluoroethyl

H

Cl

11-2495

2,2,2-trichloroethyl

H

H

H

H

F

H

Br

H

heptafluoroisopropyl

H

Br

11-2496

2,2,2-trichloroethyl

H

H

H

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

11-2497

2,2,2-trichloroethyl

H

H

H

H

F

H

I

H

heptafluoroisopropyl

H

CF3

11-2498

2,2,2-trichloroethyl

H

H

H

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

11-2499

2,2,2-trichloroethyl

H

H

H

H

F

H

I

H

nonafluoro-2-butyl

H

I

11-2500

2,2,2-trichloroethyl

H

H

H

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2501

2,2,2-trichloroethyl

H

H

H

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

11-2502

2,2,2-trichloroethyl

H

H

H

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-2503

2,2,2-trichloroethyl

H

H

H

H

H

F

Cl

H

pentafluoroethyl

H

Cl

11-2504

2,2,2-trichloroethyl

H

H

H

H

H

F

Br

H

heptafluoroisopropyl

H

Br

11-2505

2,2,2-trichloroethyl

H

H

H

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

11-2506

2,2,2-trichloroethyl

H

H

H

H

H

F

I

H

heptafluoroisopropyl

H

CF3

11-2507

2,2,2-trichloroethyl

H

H

H

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

11-2508

2,2,2-trichloroethyl

H

H

H

H

H

F

I

H

nonafluoro-2-butyl

H

I

11-2509

2,2,2-trichloroethyl

H

H

H

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2510

2,2,2-trichloroethyl

H

H

H

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

11-2511

2,2,2-trichloroethyl

H

H

H

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

11-2512

2,2,2-trichloroethyl

H

H

F

H

F

H

Cl

H

pentafluoroethyl

H

Cl

11-2513

2,2,2-trichloroethyl

H

H

F

H

F

H

Br

H

heptafluoroisopropyl

H

Br

11-3514

2,2,2-trichloroethyl

H

H

F

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

11-2515

2,2,2-trichloroethyl

H

H

F

H

F

H

I

H

heptafluoroisopropyl

H

CF3

11-2516

2,2,2-trichloroethyl

H

H

F

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

11-2517

2,2,2-trichloroethyl

H

H

F

H

F

H

I

H

nonafluoro-2-butyl

H

I

11-2518

2,2,2-trichloroethyl

H

H

F

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2519

2,2,2-trichloroethyl

H

H

F

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

11-2520

2,2,2-trichloroethyl

H

H

F

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-2521

2,2,2-trichloroethyl

H

H

F

H

H

F

Cl

H

pentafluoroethyl

H

Cl

11-2522

2,2,2-trichloroethyl

H

H

F

H

H

F

Br

H

heptafluoroisopropyl

H

Br

11-2523

2,2,2-trichloroethyl

H

H

F

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

11-2524

2,2,2-trichloroethyl

H

H

F

H

H

F

I

H

heptafluoroisopropyl

H

CF3

11-2525

2,2,2-trichloroethyl

H

H

F

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

11-2526

2,2,2-trichloroethyl

H

H

F

H

H

F

I

H

nonafluoro-2-butyl

H

I

11-2527

2,2,2-trichloroethyl

H

H

F

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2528

2,2,2-trichloroethyl

H

H

F

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

11-2529

2,2,2-trichloroethyl

H

H

F

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

11-2530

2,2,2-trichloroethyl

H

H

H

F

F

H

Cl

H

pentafluoroethyl

H

Cl

11-2531

2,2,2-trichloroethyl

H

H

H

F

F

H

Br

H

heptafluoroisopropyl

H

Br

11-2532

2,2,2-trichloroethyl

H

H

H

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

11-2533

2,2,2-trichloroethyl

H

H

H

F

F

H

I

H

heptafluoroisopropyl

H

CF3

11-2534

2,2,2-trichloroethyl

H

H

H

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

11-2535

2,2,2-trichloroethyl

H

H

H

F

F

H

I

H

nonafluoro-2-butyl

H

I

11-2536

2,2,2-trichloroethyl

H

H

H

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2537

2,2,2-trichloroethyl

H

H

H

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

11-2538

2,2,2-trichloroethyl

H

H

H

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-2539

2,2,2-trichloroethyl

H

H

H

F

H

F

Cl

H

pentafluoroethyl

H

Cl

11-2540

2,2,2-trichloroethyl

H

H

H

F

H

F

Br

H

heptafluoroisopropyl

H

Br

11-2541

2,2,2-trichloroethyl

H

H

H

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

11-2542

2,2,2-trichloroethyl

H

H

H

F

H

F

I

H

heptafluoroisopropyl

H

CF3

11-2543

2,2,2-trichloroethyl

H

H

H

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

11-2544

2,2,2-trichloroethyl

H

H

H

F

H

F

I

H

nonafluoro-2-butyl

H

I

11-2545

2,2,2-trichloroethyl

H

H

H

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2546

2,2,2-trichloroethyl

H

H

H

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

11-2547

2,2,2-trichloroethyl

H

H

H

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

11-2548

2,2,2-trichloroethyl

H

H

H

H

F

F

Cl

H

pentafluoroethyl

H

Cl

11-2549

2,2,2-trichloroethyl

H

H

H

H

F

F

Br

H

heptafluoroisopropyl

H

Br

11-2550

2,2,2-trichloroethyl

H

H

H

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

11-2551

2,2,2-trichloroethyl

H

H

H

H

F

F

I

H

heptafluoroisopropyl

H

CF3

11-2552

2,2,2-trichloroethyl

H

H

H

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

11-2553

2,2,2-trichloroethyl

H

H

H

H

F

F

I

H

nonafluoro-2-butyl

H

I

11-2554

2,2,2-trichloroethyl

H

H

H

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2555

2,2,2-trichloroethyl

H

H

H

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

11-2556

2,2,2-trichloroethyl

H

H

H

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

11-2557

2,2,2-trichloroethyl

H

H

F

F

H

F

Cl

H

pentafluoroethyl

H

Cl

11-2558

2,2,2-trichloroethyl

H

H

F

F

H

F

Br

H

heptafluoroisopropyl

H

Br

11-2559

2,2,2-trichloroethyl

H

H

F

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

11-2560

2,2,2-trichloroethyl

H

H

F

F

H

F

I

H

heptafluoroisopropyl

H

CF3

11-2561

2,2,2-trichloroethyl

H

H

F

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

11-2562

2,2,2-trichloroethyl

H

H

F

F

H

F

I

H

nonafluoro-2-butyl

H

I

11-2563

2,2,2-trichloroethyl

H

H

F

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2564

2,2,2-trichloroethyl

H

H

F

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

11-2565

2,2,2-trichloroethyl

H

H

F

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

11-2566

2,2,2-trichloroethyl

H

H

F

H

F

F

Cl

H

pentafluoroethyl

H

Cl

11-2567

2,2,2-trichloroethyl

H

H

F

H

F

F

Br

H

heptafluoroisopropyl

H

Br

11-2568

2,2,2-trichloroethyl

H

H

F

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

11-2569

2,2,2-trichloroethyl

H

H

F

H

F

F

I

H

heptafluoroisopropyl

H

CF3

11-2570

2,2,2-trichloroethyl

H

H

F

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

11-2571

2,2,2-trichloroethyl

H

H

F

H

F

F

I

H

nonafluoro-2-butyl

H

I

11-2572

2,2,2-trichloroethyl

H

H

F

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2573

2,2,2-trichloroethyl

H

H

F

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

11-2574

2,2,2-trichloroethyl

H

H

F

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

11-2575

2,2,2-trichloroethyl

H

H

H

F

F

F

Cl

H

pentafluoroethyl

H

Cl

11-2576

2,2,2-trichloroethyl

H

H

H

F

F

F

Br

H

heptafluoroisopropyl

H

Br

11-2577

2,2,2-trichloroethyl

H

H

H

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

11-2578

2,2,2-trichloroethyl

H

H

H

F

F

F

I

H

heptafluoroisopropyl

H

CF3

11-2579

2,2,2-trichloroethyl

H

H

H

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

11-2580

2,2,2-trichloroethyl

H

H

H

F

F

F

i

H

nonafluoro-2-butyl

H

I

11-2581

2,2,2-trichloroethyl

H

H

H

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2582

2,2,2-trichloroethyl

H

H

H

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

11-2583

2,2,2-trichloroethyl

H

H

H

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

11-2584

2,2,2-trichloroethyl

H

H

F

F

F

F

Cl

H

pentafluoroethyl

H

Cl

11-2585

2,2,2-trichloroethyl

H

H

F

F

F

F

Br

H

heptafluoroisopropyl

H

Br

11-2586

2,2,2-trichloroethyl

H

H

F

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

11-2587

2,2,2-trichloroethyl

H

H

F

F

F

F

I

H

heptafluoroisopropyl

H

CF3

11-2588

2,2,2-trichloroethyl

H

H

F

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

11-2589

2,2,2-trichloroethyl

H

H

F

F

F

F

I

H

nonafluoro-2-butyl

H

I

11-2590

2,2,2-trichloroethyl

H

H

F

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2591

2,2,2-trichloroethyl

H

H

F

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

11-2592

2,2,2-trichloroethyl

H

H

F

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

11-2593

2,2,2-trichloroethyl

H

H

H

CN

H

H

F

H

heptafluoroisopropyl

H

OCF3

11-2594

2,2,2-trichloroethyl

H

H

H

CN

H

H

F

H

nonafluoro-2-butyl

H

OCF3

11-2605

2,2,2-trichloroethyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

11-2634

2,2,2-trichloroethyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

11-2663

2,2,2-trichloroethyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-2692

2,2,2-trichloroethyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-2721

2,2,2-trichloroethyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-2750

2,2,2-trichloroethyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-2769

2,2,2-trichloroethyl

H

H

H

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

11-2770

2,2,2-trichloroethyl

H

H

H

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

11-2781

2,2,2-trichloroethyl

H

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-2810

2,2,2-trichloroethyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-2839

2,2,2-trichloroethyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-2852

4,4,4-trifluoro-n-butyl

H

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-2868

2,2,2-trichloroethyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-2881

4,4,4-trifluoro-n-butyl

H

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-2897

2,2,2-trichloroethyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

11-2910

4,4,4-trifluoro-n-butyl

H

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

11-2926

2,2,2-trichloroethyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-2939

4,4,4-trifluoro-n-butyl

H

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-2955

2,2,2-trichloroethyl

H

H

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

11-2984

2,2,2-trichloroethyl

H

H

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

11-3013

2,2,2-trichloroethyl

H

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

11-3042

2,2,2-trichloroethyl

H

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

11-3071

2,2,2-trichloroethyl

H

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-3100

2,2,2-trichloroethyl

H

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-3119

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

heptafluoroisopropyl

H

F

11-3120

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

nonafluoro-2-butyl

H

F

11-3131

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

Cl

11-3160

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

11-3189

2,2,2-trichloroethyl

H

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

Br

11-3218

2,2,2-trichloroethyl

H

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

Br

11-3247

2,2,2-trichloroethyl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

I

11-3276

2,2,2-trichloroethyl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

I

11-3295

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

heptafluoroisopropyl

H

Cl

11-3296

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

heptafluoroisopropyl

H

Br

11-3297

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

heptafluoroisopropyl

H

I

11-3298

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

Br

11-3299

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

I

11-3300

2,2,2-trichloroethyl

H

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

I

11-3301

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

nonafluoro-2-butyl

H

Cl

11-3302

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

nonafluoro-2-butyl

H

Br

11-3303

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

nonafluoro-2-butyl

H

I

11-3304

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

Br

11-3305

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

I

11-3306

2,2,2-trichloroethyl

H

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

I

11-3307

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

heptafluoroisopropyl

H

OCF3

11-3308

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

nonafluoro-2-butyl

H

OCF3

11-3319

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

11-3348

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

11-3377

2,2,2-trichloroethyl

H

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

11-3406

2,2,2-trichloroethyl

H

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-3435

2,2,2-trichloroethyl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

11-3464

2,2,2-trichloroethyl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

11-3483

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

11-3484

2,2,2-trichloroethyl

H

H

F

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

11-3495

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

11-3524

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-3553

2,2,2-trichloroethyl

H

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-3566

4,4,4-trifluoro-n-butyl

H

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

11-3582

2,2,2-trichloroethyl

H

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-3595

4,4,4-trifluoro-n-butyl

H

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

11-3611

2,2,2-trichloroethyl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

11-3624

4,4,4-trifluoro-n-butyl

H

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

11-3640

2,2,2-trichloroethyl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-3653

4,4,4-trifluoro-n-butyl

H

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

11-3669

2,2,2-trichloroethyl

H

H

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

11-3698

2,2,2-tnchloroethyl

H

H

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

11-3727

2,2,2-trichloroethyl

H

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

11-3756

2,2,2-trichloroethyl

H

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

11-3785

2,2,2-trichloroethyl

H

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

11-3814

2,2,2-trichloroethyl

H

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

11-3833

2,2,2-trichloroethyl

H

H

F

CN

F

H

F

H

heptafluoroisopropyl

H

F

11-3834

2,2,2-trichloroethyl

H

H

F

CN

F

H

F

H

nonafluoro-2-butyl

H

F

11-3845

2,2,2-trichloroethyl

H

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

Cl

11-3874

2,2,2-trichloroethyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

Cl

11-3903

2,2,2-trichloroethyl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

Br

11-3932

2,2,2-trichloroethyl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

Br

11-3961

2,2,2-trichloroethyl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

I

11-3990

2,2,2-trichloroethyl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

I

11-4009

2,2,2-trichloroethyl

H

H

F

CN

F

H

F

H

heptafluoroisopropyl

H

Cl

11-4010

2,2,2-trichloroethyl

H

H

F

CN

F

H

F

H

heptafluoroisopropyl

H

Br

11-4011

2,2,2-trichloroethyl

H

H

F

CN

F

H

F

H

heptafluoroisopropyl

H

I

11-4012

2,2,2-trichloroethyl

H

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

Br

11-4013

2,2,2-trichloroethyl

H

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

I

11-4014

2,2,2-trichloroethyl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

I

11-4015

2,2,2-trichloroethyl

H

H

F

CN

F

H

F

H

nonafluoro-2-butyl

H

Cl

11-4016

2,2,2-trichloroethyl

H

H

F

CN

F

H

F

H

nonafluoro-2-butyl

H

Br

11-4017

2,2,2-trichloroethyl

H

H

F

CN

F

H

F

H

nonafluoro-2-butyl

H

I

11-4018

2,2,2-trichloroethyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

Br

11-4019

2,2,2-trichloroethyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

I

11-4020

2,2,2-trichloroethyl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

I

11-4021

2,2,2-trichloroethyl

H

H

F

CN

F

H

F

H

heptafluoroisopropyl

H

OCF3

11-4022

2,2,2-trichloroethyl

H

H

F

CN

F

H

F

H

nonafluoro-2-butyl

H

OCF3

11-4033

2,2,2-trichloroethyl

H

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

11-4062

2,2,2-trichloroethyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

11-4091

2,2,2-trichloroethyl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

11-4120

2,2,2-trichloroethyl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

11-4149

2,2,2-trichloroethyl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

11-4178

2,2,2-trichloroethyl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

11-4209

2,2,2-trichloroethyl

H

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

11-4238

2,2,2-trichloroethyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

11-4267

2,2,2-trichloroethyl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

11-4280

4,4,4-trifluoro-n-butyl

H

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

11-4296

2,2,2-trichloroethyl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

11-4309

4,4,4-trifluoro-n-butyl

H

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

11-4325

2,2,2-trichloroethyl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

11-4338

4,4,4-trifluoro-n-butyl

H

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

11-4354

2,2,2-trichloroethyl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

11-4367

4,4,4-trifluoro-n-butyl

H

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

11-4383

2,2,2-trichloroethyl

H

H

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

11-4412

2,2,2-trichloroethyl

H

H

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

11-4441

2,2,2-trichloroethyl

H

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

11-4470

2,2,2-trichloroethyl

H

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

11-4499

2,2,2-trichloroethyl

H

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

11-4528

2,2,2-trichloroethyl

H

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 12

compound

number

Q2

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

12-1

2,2,2-trichloroethyl

Me

H

H

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

12-2

2,2,2-trichloroethyl

Me

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

12-13

2,2,2-trichloroethyl

Me

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

12-42

2,2,2-trichloroethyl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

12-71

2,2,2-trichloroethyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

12-100

2,2,2-trichloroethyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

12-129

2,2,2-trichloroethyl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

12-158

2,2,2-trichloroethyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

12-177

2,2,2-trichloroethyl

Me

H

H

H

H

H

F

H

heptafluoroisopropyl

H

CF3

12-178

2,2,2-trichloroethyl

Me

H

H

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

12-189

2,2,2-trichloroethyl

Me

H

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

12-218

2,2,2-trichloroethyl

Me

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

12-247

2,2,2-trichloroethyl

Me

H

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-276

2,2,2-trichloroethyl

Me

H

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-305

2,2,2-trichloroethyl

Me

H

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-334

2,2,2-trichloroethyl

Me

H

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-363

2,2,2-trichloroethyl

Me

H

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

12-392

2,2,2-trichloroethyl

Me

H

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

12-421

2,2,2-trichloroethyl

Me

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

12-450

2,2,2-trichloroethyl

Me

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

12-479

2,2,2-trichloroethyl

Me

H

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

12-508

2,2,2-trichloroethyl

Me

H

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

12-527

2,2,2-trichloroethyl

Me

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

12-528

2,2,2-trichloroethyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

12-529

2,2,2-trichloroethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

12-530

2,2,2-trichloroethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

12-531

2,2,2-trichloroethyl

Me

H

F

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

12-532

2,2,2-trichloroethyl

Me

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

12-543

2,2,2-trichloroethyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

12-572

2,2,2-trichloroethyl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

12-601

2,2,2-trichloroethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

12-630

2,2,2-trichloroethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

12-659

2,2,2-trichloroethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

12-688

2,2,2-trichloroethyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

12-707

2,2,2-trichloroethyl

Me

H

F

H

H

H

F

H

heptafluoroisopropyl

H

CF3

12-708

2,2,2-trichloroethyl

Me

H

F

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

12-715

2-cyanoethyl

Et

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

12-719

2,2,2-trichloroethyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

12-721

n-propyl

Me

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

12-725

i-propyl

n-Pr

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

12-728

1,3-dichloro-2-propyl

Me

H

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

12-729

1-chloro-3-fluoro-2-propyl

i-Pr

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

12-733

i-butyl

CH2CH═CH2

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

12-739

ethyl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

12-744

2-cyanoethyl

CN

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

12-748

2,2,2-trichloroethyl

Me

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

12-750

n-propyl

CH2C≡CH

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

12-762

i-butyl

NH2

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

12-767

methyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-768

ethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-769

2-fluoroethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-770

2-chloroethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-771

2-bromoethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-772

2-iodoethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-773

2-cyanoethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

C2F5

12-774

2,2-difluoroethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-775

2,2-dichloroethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-776

2,2,2-trifluoroethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-777

2,2,2-trichloroethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-778

2,2,2-tribromoethyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-779

n-propyl

C(O)OMe

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-780

3-fluoro-n-propyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-781

3-chloro-n-propyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-782

3-bromo-n-propyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-783

i-propyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-784

1,2-difluoro-2-propyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

n-C3F7

12-785

1,3-difluoro-2-propyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-786

1,3-dichloro-2-propyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-787

1-chloro-3-fluoro-2-propyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-788

3,3,3-trifluoro-n-propyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-789

n-butyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-790

4,4,4-trifluoro-n-butyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-791

i-butyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-792

s-butyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-793

vinyl

C(O)C(O)OMe

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-794

benzyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-795

phenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-796

methyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-797

ethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-798

2-fluoroethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-799

2-chloroethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-800

2-bromoethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-801

2-iodoethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

GF3

12-802

2-cyanoethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-803

2,2-difluoroethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-804

2,2-dichloroethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-805

2,2,2-trifluoroethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-806

2,2,2-trichloroethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-807

2,2,2-tribromoethyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-808

n-propyl

C(O)OEt

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-809

3-fluoro-n-propyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-810

3-chloro-n-propyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-811

3-bromo-n-propyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-812

i-propyl

C(O)Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-813

1,2-difluoro-2-propyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-814

1,3-difluoro-2-propyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-815

1,3-dichloro-2-propyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-816

1-chloro-3-fluoro-2-propyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-817

3,3,3-trifluoro-n-propyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-818

n-butyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-819

4,4,4-trifluoro-n-butyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-820

i-butyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-821

s-butyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-822

vinyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-823

benzyl

Me

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-824

phenyl

C(O)C(O)OEt

H

F

H

H

H

Br

H

nonafluoro-2-butyl

H

i-C3F7

12-825

methyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-826

ethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-827

2-fluoroethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-828

2-chloroethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-829

2-bromoethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-830

2-iodoethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-831

2-cyanoethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-832

2,2-difluoroethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-833

2,2-dichloroethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-834

2,2,2-trifluoroethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-835

2,2,2-trichloroethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-836

2,2,2-tribromoethyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-837

n-propyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-838

3-fluoro-n-propyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-839

3-chloro-n-propyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-840

3-bromo-n-propyl

C(O)Et

H

F

H

H

H

I

H

heptafluoroisopropyl

H

C2F5

12-841

i-propyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-842

1,2-difluoro-2-propyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-843

1,3-difluoro-2-propyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-844

1,3-dichloro-2-propyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-845

1-chloro-3-fluoro-2-propyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-846

3,3,3-trifluoro-n-propyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-847

n-butyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-848

4,4,4-trifluoro-n-butyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-849

i-butyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-850

s-butyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-851

vinyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-852

benzyl

S(O)2Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-853

phenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

12-854

methyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-855

ethyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-856

2-fluoroethyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-857

2-chloroethyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-858

2-bromoethyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-859

2-iodoethyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-860

2-cyanoethyl

S(O)2Et

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-861

2,2-difluoroethyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-862

2,2-dichloroethyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-863

2,2,2-trifluoroethyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-864

2,2,2-trichloroethyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-865

2,2,2-tribromoethyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-866

n-propyl

CH2Ph

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

n-C3F7

12-867

3-fluoro-n-propyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-868

3-chloro-n-propyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-869

3-bromo-n-propyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-870

i-propyl

CH2(3-Py)

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-871

1,2-difluoro-2-propyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-872

1,3-difluoro-2-propyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-873

1,3-dichloro-2-propyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-874

1-chloro-3-fluoro-2-propyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-875

3,3,3-trifluoro-n-propyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-876

n-butyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-877

4,4,4-trifluoro-n-butyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-878

i-butyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-879

s-butyl

CH2(3-Py—N-

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

12-880

vinyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

i-C3F7

12-881

benzyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-882

phenyl

Me

H

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-893

2,2,2-trichloroethyl

Me

H

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

12-922

2,2,2-trichloroethyl

Me

H

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

12-951

2,2,2-trichloroethyl

Me

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

12-980

2,2,2-trichloroethyl

Me

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

12-1009

2,2,2-trichloroethyl

Me

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

12-1038

2,2,2-trichloroethyl

Me

H

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

12-1057

2,2,2-trichloroethyl

Me

H

H

F

H

H

F

H

heptafluoroisopropyl

H

F

12-1058

2,2,2-trichloroethyl

Me

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

12-1069

2,2,2-trichloroethyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

12-1098

2,2,2-trichloroethyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

12-1127

2,2,2-trichloroethyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

12-1156

2,2,2-trichloroethyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

12-1185

2,2,2-trichloroethyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

I

12-1214

2,2,2-trichloroethyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

12-1236

2,2,2-trichloroethyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Br

12-1245

2,2,2-trichloroethyl

Me

H

H

F

H

H

F

H

heptafluoroisopropyl

H

OCF3

12-1246

2,2,2-trichloroethyl

Me

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

OCF3

12-1257

2,2,2-trichloroethyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

12-1286

2,2,2-trichloroethyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

12-1315

2,2,2-trichloroethyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

12-1344

2,2,2-trichloroethyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

12-1373

2,2,2-trichloroethyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

12-1402

2,2,2-trichloroethyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

12-1421

2,2,2-trichloroethyl

Me

H

H

F

H

H

F

H

heptafluoroisopropyl

H

CF3

12-1422

2,2,2-trichloroethyl

Me

H

H

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

12-1433

2,2,2-trichloroethyl

Me

H

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

12-1462

2,2,2-trichloroethyl

Me

H

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

12-1491

2,2,2-trichloroethyl

Me

H

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-1520

2,2,2-trichloroethyl

Me

H

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-1549

2,2,2-trichloroethyl

Me

H

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

12-1578

2,2,2-trichloroethyl

Me

H

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-1607

2,2,2-trichloroethyl

Me

H

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

12-1636

2,2,2-trichloroethyl

Me

H

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

12-1665

2,2,2-trichloroethyl

Me

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

12-1694

2,2,2-trichloroethyl

Me

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

12-1723

2,2,2-trichloroethyl

Me

H

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

12-1752

2,2,2-trichloroethyl

Me

H

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

12-1771

2,2,2-trichloroethyl

Me

H

F

F

H

H

F

H

heptafluoroisopropyl

H

F

12-1772

2,2,2-trichloroethyl

Me

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

12-1783

2,2,2-trichloroethyl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

12-1812

2,2,2-trichloroethyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

12-1841

2,2,2-trichloroethyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

12-1870

2,2,2-trichloroethyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

12-1899

2,2,2-trichloroethyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

I

12-1928

2,2,2-trichloroethyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

12-1956

2,2,2-trichloroethyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Br

12-1959

2,2,2-trichloroethyl

Me

H

F

F

H

H

F

H

heptafluoroisopropyl

H

OCF3

12-1960

2,2,2-trichloroethyl

Me

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

OCF3

12-1971

2,2,2-trichloroethyl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

12-2000

2,2,2-trichloroethyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2029

2,2,2-trichloroethyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

12-2058

2,2,2-trichloroethyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

12-2087

2,2,2-trichloroethyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

12-2116

2,2,2-trichloroethyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

12-2135

2,2,2-trichloroethyl

Me

H

F

F

H

H

F

H

heptafluoroisopropyl

H

CF3

12-2136

2,2,2-trichloroethyl

Me

H

F

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

12-2147

2,2,2-trichloroethyl

Me

H

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

12-2176

2,2,2-trichloroethyl

Me

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

12-2205

2,2,2-trichloroethyl

Me

H

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-2234

2,2,2-trichloroethyl

Me

H

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-2263

2,2,2-trichloroethyl

Me

H

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

12-2292

2,2,2-trichloroethyl

Me

H

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-2321

2,2,2-trichloroethyl

Me

H

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

12-2350

2,2,2-trichloroethyl

Me

H

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

12-2379

2,2,2-trichloroethyl

Me

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

12-2408

2,2,2-trichloroethyl

Me

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

12-2437

2,2,2-trichloroethyl

Me

H

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

12-2466

2,2,2-trichloroethyl

Me

H

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

12-2485

2,2,2-trichloroethyl

Me

H

F

F

F

H

Cl

H

pentafluoroethyl

H

Cl

12-2486

2,2,2-trichloroethyl

Me

H

F

F

F

H

Br

H

heptafluoroisopropyl

H

Br

12-2487

2,2,2-trichloroethyl

Me

H

F

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

12-2488

2,2,2-trichloroethyl

Me

H

F

F

F

H

I

H

heptafluoroisopropyl

H

CF3

12-2489

2,2,2-trichloroethyl

Me

H

F

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

12-2490

2,2,2-trichloroethyl

Me

H

F

F

F

H

I

H

nonafluoro-2-butyl

H

I

12-2491

2,2,2-trichloroethyl

Me

H

F

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2492

2,2,2-trichloroethyl

Me

H

F

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

12-2493

2,2,2-trichloroethyl

Me

H

F

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

12-2494

2,2,2-trichloroethyl

Me

H

H

H

F

H

Cl

H

pentafluoroethyl

H

Cl

12-2495

2,2,2-trichloroethyl

Me

H

H

H

F

H

Br

H

heptafluoroisopropyl

H

Br

12-2496

2,2,2-trichloroethyl

Me

H

H

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

12-2497

2,2,2-trichloroethyl

Me

H

H

H

F

H

I

H

heptafluoroisopropyl

H

CF3

12-2498

2,2,2-trichloroethyl

Me

H

H

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

12-2499

2,2,2-trichloroethyl

Me

H

H

H

F

H

I

H

nonafluoro-2-butyl

H

I

12-2500

2,2,2-trichloroethyl

Me

H

H

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2501

2,2,2-trichloroethyl

Me

H

H

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

12-2502

2,2,2-trichloroethyl

Me

H

H

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

12-2503

2,2,2-trichloroethyl

Me

H

H

H

H

F

Cl

H

pentafluoroethyl

H

Cl

12-2504

2,2,2-trichloroethyl

Me

H

H

H

H

F

Br

H

heptafluoroisopropyl

H

Br

12-2505

2,2,2-trichloroethyl

Me

H

H

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

12-2506

2,2,2-trichloroethyl

Me

H

H

H

H

F

I

H

heptafluoroisopropyl

H

CF3

12-2507

2,2,2-trichloroethyl

Me

H

H

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

12-2508

2,2,2-trichloroethyl

Me

H

H

H

H

F

I

H

nonafluoro-2-butyl

H

I

12-2509

2,2,2-trichloroethyl

Me

H

H

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2510

2,2,2-trichloroethyl

Me

H

H

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

12-2511

2,2,2-trichloroethyl

Me

H

H

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

12-2512

2,2,2-trichloroethyl

Me

H

F

H

F

H

Cl

H

pentafluoroethyl

H

Cl

12-2513

2,2,2-trichloroethyl

Me

H

F

H

F

H

Br

H

heptafluoroisopropyl

H

Br

12-2514

2,2,2-trichloroethyl

Me

H

F

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

12-2515

2,2,2-trichloroethyl

Me

H

F

H

F

H

I

H

heptafluoroisopropyl

H

CF3

12-2516

2,2,2-trichloroethyl

Me

H

F

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

12-2517

2,2,2-trichloroethyl

Me

H

F

H

F

H

I

H

nonafluoro-2-butyl

H

I

12-2518

2,2,2-trichloroethyl

Me

H

F

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2519

2,2,2-trichloroethyl

Me

H

F

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

12-2520

2,2,2-trichloroethyl

Me

H

F

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

12-2521

2,2,2-trichloroethyl

Me

H

F

H

H

F

Cl

H

pentafluoroethyl

H

Cl

12-2522

2,2,2-trichloroethyl

Me

H

F

H

H

F

Br

H

heptafluoroisopropyl

H

Br

12-2523

2,2,2-trichloroethyl

Me

H

F

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

12-2524

2,2,2-trichloroethyl

Me

H

F

H

H

F

I

H

heptafluoroisopropyl

H

CF3

12-2525

2,2,2-trichloroethyl

Me

H

F

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

12-2526

2,2,2-trichloroethyl

Me

H

F

H

H

F

I

H

nonafluoro-2-butyl

H

I

12-2527

2,2,2-trichloroethyl

Me

H

F

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2528

2,2,2-trichloroethyl

Me

H

F

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

12-2529

2,2,2-trichloroethyl

Me

H

F

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

12-2530

2,2,2-trichloroethyl

Me

H

H

F

F

H

Cl

H

pentafluoroethyl

H

Cl

12-2531

2,2,2-trichloroethyl

Me

H

H

F

F

H

Br

H

heptafluoroisopropyl

H

Br

12-2532

2,2,2-trichloroethyl

Me

H

H

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

12-2533

2,2,2-trichloroethyl

Me

H

H

F

F

H

I

H

heptafluoroisopropyl

H

CF3

12-2534

2,2,2-trichloroethyl

Me

H

H

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

12-2535

2,2,2-trichloroethyl

Me

H

H

F

F

H

I

H

nonafluoro-2-butyl

H

I

12-2536

2,2,2-trichloroethyl

Me

H

H

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2537

2,2,2-trichloroethyl

Me

H

H

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

12-2538

2,2,2-trichloroethyl

Me

H

H

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

12-2539

2,2,2-trichloroethyl

Me

H

H

F

H

F

Cl

H

pentafluoroethyl

H

Cl

12-2540

2,2,2-trichloroethyl

Me

H

H

F

H

F

Br

H

heptafluoroisopropyl

H

Br

12-2541

2,2,2-trichloroethyl

Me

H

H

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

12-2542

2,2,2-trichloroethyl

Me

H

H

F

H

F

I

H

heptafluoroisopropyl

H

CF3

12-2543

2,2,2-trichloroethyl

Me

H

H

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

12-2544

2,2,2-trichloroethyl

Me

H

H

F

H

F

I

H

nonafluoro-2-butyl

H

I

12-2545

2,2,2-trichloroethyl

Me

H

H

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2546

2,2,2-trichloroethyl

Me

H

H

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

12-2547

2,2,2-trichloroethyl

Me

H

H

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

12-2548

2,2,2-trichloroethyl

Me

H

H

H

F

F

Cl

H

pentafluoroethyl

H

Cl

12-2549

2,2,2-trichloroethyl

Me

H

H

H

F

F

Br

H

heptafluoroisopropyl

H

Br

12-2550

2,2,2-trichloroethyl

Me

H

H

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

12-2551

2,2,2-trichloroethyl

Me

H

H

H

F

F

I

H

heptafluoroisopropyl

H

CF3

12-2552

2,2,2-trichloroethyl

Me

H

H

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

12-2553

2,2,2-trichloroethyl

Me

H

H

H

F

F

I

H

nonafluoro-2-butyl

H

I

12-2554

2,2,2-trichloroethyl

Me

H

H

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2555

2,2,2-trichloroethyl

Me

H

H

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

12-2556

2,2,2-trichloroethyl

Me

H

H

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

12-2557

2,2,2-trichloroethyl

Me

H

F

F

H

F

Cl

H

pentafluoroethyl

H

Cl

12-2558

2,2,2-trichloroethyl

Me

H

F

F

H

F

Br

H

heptafluoroisopropyl

H

Br

12-2559

2,2,2-trichloroethyl

Me

H

F

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

12-2560

2,2,2-trichloroethyl

Me

H

F

F

H

F

I

H

heptafluoroisopropyl

H

CF3

12-2561

2,2,2-trichloroethyl

Me

H

F

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

12-2562

2,2,2-trichloroethyl

Me

H

F

F

H

F

I

H

nonafluoro-2-butyl

H

I

12-2563

2,2,2-trichloroethyl

Me

H

F

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2564

2,2,2-trichloroethyl

Me

H

F

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

12-2565

2,2,2-trichloroethyl

Me

H

F

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

12-2566

2,2,2-trichloroethyl

Me

H

F

H

F

F

Cl

H

pentafluoroethyl

H

Cl

12-2567

2,2,2-trichloroethyl

Me

H

F

H

F

F

Br

H

heptafluoroisopropyl

H

Br

12-2568

2,2,2-trichloroethyl

Me

H

F

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

12-2569

2,2,2-trichloroethyl

Me

H

F

H

F

F

I

H

heptafluoroisopropyl

H

CF3

12-2570

2,2,2-trichloroethyl

Me

H

F

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

12-2571

2,2,2-trichloroethyl

Me

H

F

H

F

F

I

H

nonafluoro-2-butyl

H

I

12-2572

2,2,2-trichloroethyl

Me

H

F

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2573

2,2,2-trichloroethyl

Me

H

F

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

12-2574

2,2,2-trichloroethyl

Me

H

F

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

12-2575

2,2,2-trichloroethyl

Me

H

H

F

F

F

Cl

H

pentafluoroethyl

H

Cl

12-2576

2,2,2-trichloroethyl

Me

H

H

F

F

F

Br

H

heptafluoroisopropyl

H

Br

12-2577

2,2,2-trichloroethyl

Me

H

H

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

12-2578

2,2,2-trichloroethyl

Me

H

H

F

F

F

I

H

heptafluoroisopropyl

H

CF3

12-2579

2,2,2-trichloroethyl

Me

H

H

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

12-2580

2,2,2-trichloroethyl

Me

H

H

F

F

F

I

H

nonafluoro-2-butyl

H

I

12-2581

2,2,2-trichloroethyl

Me

H

H

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2582

2,2,2-trichloroethyl

Me

H

H

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

12-2583

2,2,2-trichloroethyl

Me

H

H

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

12-2584

2,2,2-trichloroethYl

Me

H

F

F

F

F

Cl

H

pentafluoroethyl

H

Cl

12-2585

2,2,2-trichloroethyl

Me

H

F

F

F

F

Br

H

heptafluoroisopropyl

H

Br

12-2586

2,2,2-trichloroethyl

Me

H

F

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

12-2587

2,2,2-trichloroethyl

Me

H

F

F

F

F

I

H

heptafluoroisopropyl

H

CF3

12-2588

2,2,2-trichloroethyl

Me

H

F

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

12-2589

2,2,2-trichloroethyl

Me

H

F

F

F

F

I

H

nonafluoro-2-butyl

H

I

12-2590

2,2,2-trichloroethyl

Me

H

F

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2591

2,2,2-trichloroethyl

Me

H

F

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

12-2592

2,2,2-trichloroethyl

Me

H

F

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

12-2593

2,2,2-trichloroethyl

Me

H

H

CN

H

H

F

H

heptafluoroisopropyl

H

OCF3

12-2594

2,2,2-trichloroethyl

Me

H

H

CN

H

H

F

H

nonafluoro-2-butyl

H

OCF3

12-2605

2,2,2-trichloroethyl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

12-2634

2,2,2-trichloroethyl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

12-2663

2,2,2-trichloroethyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

12-2692

2,2,2-trichloroethyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

12-2721

2,2,2-trichloroethyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

12-2750

2,2,2-trichloroethyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

12-2769

2,2,2-trichloroethyl

Me

H

H

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

12-2770

2,2,2-trichloroethyl

Me

H

H

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

12-2781

2,2,2-trichloroethyl

Me

H

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

12-2810

2,2,2-trichloroethyl

Me

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

12-2839

2,2,2-trichloroethyl

Me

H

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-2868

2,2,2-trichloroethyl

Me

H

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-2897

2,2,2-trichloroethyl

Me

H

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

12-2926

2,2,2-trichloroethyl

Me

H

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-2955

2,2,2-trichloroethyl

Me

H

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

12-2984

2,2,2-trichloroethyl

Me

H

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

12-3013

2,2,2-trichloroethyl

Me

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

12-3042

2,2,2-trichloroethyl

Me

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

12-3071

2,2,2-trichloroethyl

Me

H

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

12-3100

2,2,2-trichloroethyl

Me

H

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

12-3119

2,2,2-trichloroethyl

Me

H

F

CN

H

H

F

H

heptafluoroisopropyl

H

F

12-3120

2,2,2-trichloroethyl

Me

H

F

CN

H

H

F

H

nonafluoro-2-butyl

H

F

12-3131

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

Cl

12-3160

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

12-3189

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

Br

12-3218

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

Br

12-3247

2,2,2-trichloroethyl

Me

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

I

12-3276

2,2,2-trichloroethyl

Me

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

I

12-3298

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

Br

12-3307

2,2,2-trichloroethyl

Me

H

F

CN

H

H

F

H

heptafluoroisopropyl

H

OCF3

12-3308

2,2,2-trichloroethyl

Me

H

F

CN

H

H

F

H

nonafluoro-2-butyl

H

OCF3

12-3319

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

12-3348

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

12-3377

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

12-3406

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

12-3435

2,2,2-trichloroethyl

Me

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

12-3464

2,2,2-trichloroethyl

Me

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

12-3483

2,2,2-trichloroethyl

Me

H

F

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

12-3484

2,2,2-trichloroethyl

Me

H

F

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

12-3495

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

12-3524

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

12-3553

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

12-3582

2,2,2-trichloroethyl

Me

H

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

12-3611

2,2,2-trichloroethyl

Me

H

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

12-3640

2,2,2-trichloroethyl

Me

H

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

12-3669

2,2,2-trichloroethyl

Me

H

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

12-3698

2,2,2-trichloroethyl

Me

H

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

12-3727

2,2,2-trichloroethyl

Me

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

12-3756

2,2,2-trichloroethyl

Me

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

12-3785

2,2,2-trichloroethyl

Me

H

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

12-3814

2,2,2-trichloroethyl

Me

H

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

12-3833

2,2,2-trichloroethyl

Me

H

F

CN

F

H

F

H

heptafluoroisopropyl

H

F

12-3834

2,2,2-trichloroethyl

Me

H

F

CN

F

H

F

H

nonafluoro-2-butyl

H

F

12-3845

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

Cl

12-3874

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

Cl

12-3903

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

Br

12-3932

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

Br

12-3961

2,2,2-trichloroethyl

Me

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

I

12-3990

2,2,2-trichloroethyl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

I

12-4018

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

Br

12-4021

2,2,2-trichloroethyl

Me

H

F

CN

F

H

F

H

heptafluoroisopropyl

H

OCF3

12-4022

2,2,2-trichloroethyl

Me

H

F

CN

F

H

F

H

nonafluoro-2-butyl

H

OCF3

12-4033

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

12-4062

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

12-4091

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

12-4120

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

12-4149

2,2,2-trichloroethyl

Me

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

12-4178

2,2,2-trichloroethyl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

12-4197

2,2,2-trichloroethyl

Me

H

F

CN

F

H

F

H

heptafluoroisopropyl

H

CF3

12-4198

2,2,2-trichloroethyl

Me

H

F

CN

F

H

F

H

nonafluoro-2-butyl

H

CF3

12-4209

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

12-4238

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

12-4267

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

12-4296

2,2,2-trichloroethyl

Me

H

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

12-4325

2,2,2-trichloroethyl

Me

H

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

12-4354

2,2,2-trichloroethyl

Me

H

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

12-4383

2,2,2-trichloroethyl

Me

H

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

12-4412

2,2,2-trichloroethyl

Me

H

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

12-4441

2,2,2-trichloroethyl

Me

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

12-4470

2,2,2-trichloroethyl

Me

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

12-4499

2,2,2-trichloroethyl

Me

H

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

12-4528

2,2,2-trichloroethyl

Me

H

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 13

compound

number

Q2

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

13-1

2,2,2-trichloroethyl

H

Me

H

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

13-2

2,2,2-trichloroethyl

H

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

13-13

2,2,2-trichloroethyl

H

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

13-42

2,2,2-trichloroethyl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

13-71

2,2,2-trichloroethyl

H

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

13-100

2,2,2-trichloroethyl

H

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

13-129

2,2,2-trichloroethyl

H

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

13-158

2,2,2-trichloroethyl

H

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

13-177

2,2,2-trichloroethyl

H

Me

H

H

H

H

F

H

heptafluoroisopropyl

H

CF3

13-178

2,2,2-trichloroethyl

H

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

13-189

2,2,2-trichloroethyl

H

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

13-218

2,2,2-trichloroethyl

H

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

13-247

2,2,2-trichloroethyl

H

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

13-276

2,2,2-trichloroethyl

H

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

13-305

2,2,2-trichloroethyl

H

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

13-334

2,2,2-trichloroethyl

H

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

13-363

2,2,2-trichloroethyl

H

Me

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

13-392

2,2,2-trichloroethyl

H

Me

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

13-421

2,2,2-trichloroethyl

H

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

13-450

2,2,2-trichloroethyl

H

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

13-479

2,2,2-trichloroethyl

H

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

13-508

2,2,2-trichloroethyl

H

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

13-527

2,2,2-trichloroethyl

H

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

F

13-528

2,2,2-trichloroethyl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

13-529

2,2,2-trichloroethyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

13-530

2,2,2-trichloroethyl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

I

13-531

2,2,2-trichloroethyl

H

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

13-532

2,2,2-trichloroethyl

H

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

13-543

2,2,2-trichloroethyl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

13-572

2,2,2-trichloroethyl

H

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

13-601

2,2,2-trichloroethyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

13-630

2,2,2-trichloroethyl

H

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

13-659

2,2,2-trichloroethyl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

13-688

2,2,2-trichloroethyl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

13-707

2,2,2-trichloroethyl

H

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

CF3

13-708

2,2,2-trichloroethyl

H

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

13-715

2-cyanoethyl

H

Et

F

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

13-719

2,2,2-trichloroethyl

H

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

13-721

n-propyl

H

Me

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

13-725

i-propyl

H

n-Pr

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

13-728

1,3-dichloro-2-propyl

H

Me

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

13-729

1-chloro-3-fluoro-2-propyl

H

i-Pr

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

13-733

i-butyl

H

CH2CH═CH2

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

13-739

ethyl

H

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

13-744

2-cyanoethyl

H

CN

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

13-748

2,2,2-trichloroethyl

H

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

13-750

n-propyl

H

CH2C═CH

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

13-762

i-butyl

H

NH2

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

13-773

2-cyanoethyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

C2F5

13-777

2,2,2-trichloroethyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

13-779

n-propyl

H

C(O)OMe

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

13-784

1,2-difluoro-2-propyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

n-C3F7

13-790

4,4,4-trifluoro-n-butyl

H

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

13-793

vinyl

H

C(O)C(O)OMe

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

13-806

2,2,2-trichloroethyl

H

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

13-808

n-propyl

H

C(O)OEt

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

13-812

i-propyl

H

C(O)Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

13-819

4,4,4-trifluoro-n-butyl

H

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

13-824

phenyl

H

C(O)C(O)OEt

F

H

H

H

Br

H

nonafluoro-2-butyl

H

i-C3F7

13-835

2,2,2-trichloroethyl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

13-840

3-bromo-n-propyl

H

C(O)Et

F

H

H

H

I

H

heptafluoroisopropyl

H

C2F5

13-848

4,4,4-trifluoro-n-butyl

H

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

13-852

benzyl

H

S(O)2Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

13-860

2-cyanoethyl

H

S(O)2Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

13-864

2,2,2-trichloroethyl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

13-866

n-propyl

H

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

n-C3F7

13-870

i-propyl

H

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

13-877

4,4,4-trifluoro-n-butyl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

13-879

s-butyl

H

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

13-880

vinyl

H

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

i-C3F7

13-893

2,2,2-trichloroethyl

H

Me

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

13-922

2,2,2-trichloroethyl

H

Me

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

13-951

2,2,2-trichloroethyl

H

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

13-980

2,2,2-trichloroethyl

H

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

13-1009

2,2,2-trichloroethyl

H

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

13-1038

2,2,2-trichloroethyl

H

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

13-1057

2,2,2-trichloroethyl

H

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

F

13-1058

2,2,2-trichloroethYl

H

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

13-1069

2,2,2-trichloroethyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

13-1098

2,2,2-trichloroethyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

13-1127

2,2,2-trichloroethyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

13-1156

2,2,2-trichloroethyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

13-1185

2,2,2-trichloroethyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

I

13-1214

2,2,2-trichloroethyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

13-1236

2,2,2-trichloroethyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Br

13-1245

2,2,2-trichloroethyl

H

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

OCF3

13-1246

2,2,2-trichloroethyl

H

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

OCF3

13-1257

2,2,2-trichloroethyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

13-1286

2,2,2-trichloroethyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

13-1315

2,2,2-trichloroethyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

13-1344

2,2,2-trichloroethyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

13-1373

2,2,2-trichloroethyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

13-1402

2,2,2-trichloroethyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

13-1421

2,2,2-trichloroethyl

H

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

CF3

13-1422

2,2,2-trichloroethyl

H

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

13-1433

2,2,2-trichloroethyl

H

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

13-1462

2,2,2-trichloroethyl

H

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

13-1491

2,2,2-trichloroethyl

H

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

13-1520

2,2,2-trichloroethyl

H

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

13-1549

2,2,2-trichloroethyl

H

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

13-1578

2,2,2-trichloroethyl

H

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

13-1607

2,2,2-trichloroethyl

H

Me

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

13-1636

2,2,2-trichloroethyl

H

Me

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

13-1665

2,2,2-trichloroethyl

H

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

13-1694

2,2,2-trichloroethyl

H

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

13-1723

2,2,2-trichloroethyl

H

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

13-1752

2,2,2-trichloroethyl

H

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

13-1771

2,2,2-trichloroethyl

H

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

F

13-1772

2,2,2-trichloroethyl

H

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

13-1783

2,2,2-trichloroethyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

13-1812

2,2,2-trichloroethyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

13-1841

2,2,2-trichloroethyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

13-1870

2,2,2-trichloroethyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

13-1899

2,2,2-trichloroethyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

I

13-1928

2,2,2-trichloroethyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

13-1956

2,2,2-trichloroethyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Br

13-1959

2,2,2-trichloroethyl

H

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

OCF3

13-1960

2,2,2-trichloroethyl

H

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

OCF3

13-1971

2,2,2-trichloroethyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

13-2000

2,2,2-trichloroethyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2029

2,2,2-trichloroethyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

13-2058

2,2,2-trichloroethyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

13-2087

2,2,2-trichloroethyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

13-2116

2,2,2-trichloroethyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

13-2135

2,2,2-trichloroethyl

H

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

CF3

13-2136

2,2,2-trichloroethyl

H

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

13-2147

2,2,2-trichloroethyl

H

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

13-2176

2,2,2-trichloroethyl

H

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

13-2205

2,2,2-trichloroethyl

H

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

13-2234

2,2,2-trichloroethyl

H

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

13-2263

2,2,2-trichloroethyl

H

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

13-2292

2,2,2-trichloroethyl

H

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

13-2321

2,2,2-trichloroethyl

H

Me

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

13-2350

2,2,2-trichloroethyl

H

Me

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

13-2379

2,2,2-trichloroethyl

H

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

13-2408

2,2,2-trichloroethyl

H

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

13-2437

2,2,2-trichloroethyl

H

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

13-2439

n-propyl

H

S(O)2Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

13-2466

2,2,2-trichloroethyl

H

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

13-2485

2,2,2-trichloroethyl

H

Me

F

F

F

H

Cl

H

pentafluoroethyl

H

Cl

13-2486

2,2,2-trichloroethyl

H

Me

F

F

F

H

Br

H

heptafluoroisopropyl

H

Br

13-2487

2,2,2-trichloroethyl

H

Me

F

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

13-2488

2,2,2-trichloroethyl

H

Me

F

F

F

H

I

H

heptafluoroisopropyl

H

CF3

13-2489

2,2,2-trichloroethyl

H

Me

F

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

13-2490

2,2,2-trichloroethyl

H

Me

F

F

F

H

I

H

nonafluoro-2-butyl

H

I

13-2491

2,2,2-trichloroethyl

H

Me

F

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2492

2,2,2-trichloroethyl

H

Me

F

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

13-2493

2,2,2-trichloroethyl

H

Me

F

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

13-2494

2,2,2-trichloroethyl

H

Me

H

H

F

H

Cl

H

pentafluoroethyl

H

Cl

13-2495

2,2,2-trichloroethyl

H

Me

H

H

F

H

Br

H

heptafluoroisopropyl

H

Br

13-2496

2,2,2-trichloroethyl

H

Me

H

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

13-2497

2,2,2-trichloroethyl

H

Me

H

H

F

H

I

H

heptafluoroisopropyl

H

CF3

13-2498

2,2,2-trichloroethyl

H

Me

H

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

13-2499

2,2,2-trichloroethyl

H

Me

H

H

F

H

I

H

nonafluoro-2-butyl

H

I

13-2500

2,2,2-trichloroethyl

H

Me

H

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2501

2,2,2-trichloroethyl

H

Me

H

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

13-2502

2,2,2-trichloroethyl

H

Me

H

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

13-2503

2,2,2-trichloroethyl

H

Me

H

H

H

F

Cl

H

pentafluoroethyl

H

Cl

13-2504

2,2,2-trichloroethyl

H

Me

H

H

H

F

Br

H

heptafluoroisopropyl

H

Br

13-2505

2,2,2-trichloroethyl

H

Me

H

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

13-2506

2,2,2-trichloroethyl

H

Me

H

H

H

F

I

H

heptafluoroisopropyl

H

CF3

13-2507

2,2,2-trichloroethyl

H

Me

H

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

13-2508

2,2,2-trichloroethyl

H

Me

H

H

H

F

I

H

nonafluoro-2-butyl

H

I

13-2509

2,2,2-trichloroethyl

H

Me

H

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2510

2,2,2-trichloroethyl

H

Me

H

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

13-2511

2,2,2-trichloroethyl

H

Me

H

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

13-2512

2,2,2-trichloroethyl

H

Me

F

H

F

H

Cl

H

pentafluoroethyl

H

Cl

13-2513

2,2,2-trichloroethyl

H

Me

F

H

F

H

Br

H

heptafluoroisopropyl

H

Br

13-2514

2,2,2-trichloroethyl

H

Me

F

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

13-2515

2,2,2-trichloroethyl

H

Me

F

H

F

H

I

H

heptafluoroisopropyl

H

CF3

13-2516

2,2,2-trichloroethyl

H

Me

F

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

13-2517

2,2,2-trichloroethyl

H

Me

F

H

F

H

I

H

nonafluoro-2-butyl

H

I

13-2518

2,2,2-trichloroethyl

H

Me

F

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2519

2,2,2-trichloroethyl

H

Me

F

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

13-2520

2,2,2-trichloroethyl

H

Me

F

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

13-2521

2,2,2-trichloroethyl

H

Me

F

H

H

F

Cl

H

pentafluoroethyl

H

Cl

13-2522

2,2,2-trichloroethyl

H

Me

F

H

H

F

Br

H

heptafluoroisopropyl

H

Br

13-2523

2,2,2-trichloroethyl

H

Me

F

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

13-2524

2,2,2-trichloroethyl

H

Me

F

H

H

F

I

H

heptafluoroisopropyl

H

CF3

13-2525

2,2,2-trichloroethyl

H

Me

F

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

13-2526

2,2,2-trichloroethyl

H

Me

F

H

H

F

I

H

nonafluoro-2-butyl

H

I

13-2527

2,2,2-trichloroethyl

H

Me

F

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2528

2,2,2-trichloroethyl

H

Me

F

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

13-2529

2,2,2-trichloroethyl

H

Me

F

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

13-2530

2,2,2-trichloroethyl

H

Me

H

F

F

H

Cl

H

pentafluoroethyl

H

Cl

13-2531

2,2,2-trichloroethyl

H

Me

H

F

F

H

Br

H

heptafluoroisopropyl

H

Br

13-2532

2,2,2-trichloroethyl

H

Me

H

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

13-2533

2,2,2-trichloroethyl

H

Me

H

F

F

H

I

H

heptafluoroisopropyl

H

CF3

13-2534

2,2,2-trichloroethyl

H

Me

H

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

13-2535

2,2,2-trichloroethyl

H

Me

H

F

F

H

I

H

nonafluoro-2-butyl

H

I

13-2536

2,2,2-trichloroethyl

H

Me

H

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2537

2,2,2-trichloroethyl

H

Me

H

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

13-2538

2,2,2-trichloroethyl

H

Me

H

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

13-2539

2,2,2-trichloroethyl

H

Me

H

F

H

F

Cl

H

pentafluoroethyl

H

Cl

13-2540

2,2,2-trichloroethyl

H

Me

H

F

H

F

Br

H

heptafluoroisopropyl

H

Br

13-2541

2,2,2-trichloroethyl

H

Me

H

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

13-2542

2,2,2-trichloroethyl

H

Me

H

F

H

F

I

H

heptafluoroisopropyl

H

CF3

13-2543

2,2,2-trichloroethyl

H

Me

H

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

13-2544

2,2,2-trichloroethyl

H

Me

H

F

H

F

I

H

nonafluoro-2-butyl

H

I

13-2545

2,2,2-trichloroethyl

H

Me

H

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2546

2,2,2-trichloroethyl

H

Me

H

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

13-2547

2,2,2-trichloroethyl

H

Me

H

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

13-2548

2,2,2-trichloroethyl

H

Me

H

H

F

F

Cl

H

pentafluoroethyl

H

Cl

13-2549

2,2,2-trichloroethyl

H

Me

H

H

F

F

Br

H

heptafluoroisopropyl

H

Br

13-2550

2,2,2-trichloroethyl

H

Me

H

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

13-2551

2,2,2-trichloroethyl

H

Me

H

H

F

F

I

H

heptafluoroisopropyl

H

CF3

13-2552

2,2,2-trichloroethyl

H

Me

H

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

13-2553

2,2,2-trichloroethyl

H

Me

H

H

F

F

I

H

nonafluoro-2-butyl

H

I

13-2554

2,2,2-trichloroethyl

H

Me

H

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2555

2,2,2-trichloroethyl

H

Me

H

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

13-2556

2,2,2-trichloroethyl

H

Me

H

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

13-2557

2,2,2-trichloroethyl

H

Me

F

F

H

F

Cl

H

pentafluoroethyl

H

Cl

13-2558

2,2,2-trichloroethyl

H

Me

F

F

H

F

Br

H

heptafluoroisopropyl

H

Br

13-2559

2,2,2-trichloroethyl

H

Me

F

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

13-2560

2,2,2-trichloroethyl

H

Me

F

F

H

F

I

H

heptafluoroisopropyl

H

CF3

13-2561

2,2,2-trichloroethyl

H

Me

F

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

13-2562

2,2,2-trichloroethyl

H

Me

F

F

H

F

I

H

nonafluoro-2-butyl

H

I

13-2563

2,2,2-trichloroethyl

H

Me

F

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2564

2,2,2-trichloroethyl

H

Me

F

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

13-2565

2,2,2-trichloroethyl

H

Me

F

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

13-2566

2,2,2-trichloroethyl

H

Me

F

H

F

F

Cl

H

pentafluoroethyl

H

Cl

13-2567

2,2,2-trichloroethyl

H

Me

F

H

F

F

Br

H

heptafluoroisopropyl

H

Br

13-2568

2,2,2-trichloroethyl

H

Me

F

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

13-2569

2,2,2-trichloroethyl

H

Me

F

H

F

F

I

H

heptafluoroisopropyl

H

CF3

13-2570

2,2,2-trichloroethyl

H

Me

F

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

13-2571

2,2,2-trichloroethyl

H

Me

F

H

F

F

I

H

nonafluoro-2-butyl

H

I

13-2572

2,2,2-trichloroethyl

H

Me

F

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2573

2,2,2-trichloroethyl

H

Me

F

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

13-2574

2,2,2-trichloroethyl

H

Me

F

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

13-2575

2,2,2-trichloroethyl

H

Me

H

F

F

F

Cl

H

pentafluoroethyl

H

Cl

13-2576

2,2,2-trichloroethyl

H

Me

H

F

F

F

Br

H

heptafluoroisopropyl

H

Br

13-2577

2,2,2-trichloroethyl

H

Me

H

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

13-2578

2,2,2-trichloroethyl

H

Me

H

F

F

F

I

H

heptafluoroisopropyl

H

CF3

13-2579

2,2,2-trichloroethyl

H

Me

H

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

13-2580

2,2,2-trichloroethyl

H

Me

H

F

F

F

I

H

nonafluoro-2-butyl

H

I

13-2581

2,2,2-trichloroethyl

H

Me

H

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2582

2,2,2-trichloroethyl

H

Me

H

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

13-2583

2,2,2-trichloroethyl

H

Me

H

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

13-2584

2,2,2-trichloroethyl

H

Me

F

F

F

F

Cl

H

pentafluoroethyl

H

Cl

13-2585

2,2,2-trichloroethyl

H

Me

F

F

F

F

Br

H

heptafluoroisopropyl

H

Br

13-2586

2,2,2-trichloroethyl

H

Me

F

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

13-2587

2,2,2-trichloroethyl

H

Me

F

F

F

F

I

H

heptafluoroisopropyl

H

CF3

13-2588

2,2,2-trichloroethyl

H

Me

F

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

13-2589

2,2,2-trichloroethyl

H

Me

F

F

F

F

I

H

nonafluoro-2-butyl

H

I

13-2590

2,2,2-trichloroethyl

H

Me

F

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2591

2,2,2-trichloroethyl

H

Me

F

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

13-2592

2,2,2-trichloroethyl

H

Me

F

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

13-2593

2,2,2-trichloroethyl

H

Me

H

CN

H

H

F

H

heptafluoroisopropyl

H

OCF3

13-2594

2,2,2-trichloroethyl

H

Me

H

CN

H

H

F

H

nonafluoro-2-butyl

H

OCF3

13-2605

2,2,2-trichloroethyl

H

Me

H

ON

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

13-2634

2,2,2-trichloroethyl

H

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

13-2663

2,2,2-trichloroethyl

H

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

13-2692

2,2,2-trichloroethyl

H

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

13-2721

2,2,2-trichloroethyl

H

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

13-2750

2,2,2-trichloroethyl

H

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

13-2769

2,2,2-trichloroethyl

H

Me

H

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

13-2770

2,2,2-trichloroethyl

H

Me

H

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

13-2781

2,2,2-trichloroethyl

H

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

13-2810

2,2,2-trichloroethyl

H

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

13-2839

2,2,2-trichloroethyl

H

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

13-2868

2,2,2-trichloroethyl

H

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

13-2897

2,2,2-trichloroethyl

H

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

13-2926

2,2,2-trichloroethyl

H

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

13-2955

2,2,2-trichloroethyl

H

Me

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

13-2984

2,2,2-trichloroethyl

H

Me

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

13-3013

2,2,2-trichloroethyl

H

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

13-3042

2,2,2-trichloroethyl

H

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

13-3071

2,2,2-trichloroethyl

H

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

13-3100

2,2,2-trichloroethyl

H

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

13-3119

2,2,2-trichloroethyl

H

Me

F

CN

H

H

F

H

heptafluoroisopropyl

H

F

13-3120

2,2,2-trichloroethyl

H

Me

F

CN

H

H

F

H

nonafluoro-2-butyl

H

F

13-3131

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

Cl

13-3160

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

13-3189

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

Br

13-3218

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

Br

13-3247

2,2,2-trichloroethyl

H

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

I

13-3276

2,2,2-trichloroethyl

H

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

I

13-3298

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

Br

13-3307

2,2,2-trichloroethyl

H

Me

F

CN

H

H

F

H

heptafluoroisopropyl

H

OCF3

13-3308

2,2,2-trichloroethyl

H

Me

F

CN

H

H

F

H

nonafluoro-2-butyl

H

OCF3

13-3319

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

13-3348

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

13-3377

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

13-3406

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

13-3435

2,2,2-trichloroethyl

H

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

13-3464

2,2,2-trichloroethyl

H

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

13-3483

2,2,2-trichloroethyl

H

Me

F

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

13-3484

2,2,2-trichloroethyl

H

Me

F

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

13-3495

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

13-3524

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

13-3553

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

13-3582

2,2,2-trichloroethyl

H

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

13-3611

2,2,2-trichloroethyl

H

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

13-3640

2,2,2-trichloroethyl

H

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

13-3669

2,2,2-trichloroethyl

H

Me

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

13-3698

2,2,2-trichloroethyl

H

Me

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

13-3727

2,2,2-trichloroethyl

H

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

13-3756

2,2,2-trichloroethyl

H

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

13-3785

2,2,2-trichloroethyl

H

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

13-3814

2,2,2-trichloroethyl

H

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

13-3833

2,2,2-trichloroethyl

H

Me

F

CN

F

H

F

H

heptafluoroisopropyl

H

F

13-3834

2,2,2-trichloroethyl

H

Me

F

CN

F

H

F

H

nonafluoro-2-butyl

H

F

13-3845

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

Cl

13-3874

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

Cl

13-3903

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

Br

13-3932

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

Br

13-3961

2,2,2-trichloroethyl

H

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

I

13-3990

2,2,2-trichloroethyl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

I

13-4012

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

Br

13-4021

2,2,2-trichloroethyl

H

Me

F

CN

F

H

F

H

heptafluoroisopropyl

H

OCF3

13-4022

2,2,2-trichloroethyl

H

Me

F

CN

F

H

F

H

nonafluoro-2-butyl

H

OCF3

13-4033

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

13-4062

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

13-4091

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

13-4120

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

13-4149

2,2,2-trichloroethyl

H

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

OOF3

13-4178

2,2,2-trichloroethyl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

13-4197

2,2,2-trichloroethyl

H

Me

F

CN

F

H

F

H

heptafluoroisopropyl

H

CF3

13-4198

2,2,2-trichloroethyl

H

Me

F

CN

F

H

F

H

nonafluoro-2-butyl

H

CF3

13-4209

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

13-4238

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

13-4267

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

13-4296

2,2,2-trichloroethyl

H

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

13-4325

2,2,2-trichloroethyl

H

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

13-4354

2,2,2-trichloroethyl

H

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

13-4383

2,2,2-trichloroethyl

H

Me

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

13-4412

2,2,2-trichloroethyl

H

Me

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

13-4441

2,2,2-trichloroethyl

H

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

13-4470

2,2,2-trichloroethyl

H

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

13-4499

2,2,2-trichloroethyl

H

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

13-4528

2,2,2-trichloroethyl

H

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 14

compound

number

Q2

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

14-1

2,2,2-trichloroethyl

Me

Me

H

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

14-2

2,2,2-trichloroethyl

Me

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

14-13

2,2,2-trichloroethyl

Me

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

14-42

2,2,2-trichloroethyl

Me

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

14-71

2,2,2-trichloroethyl

Me

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

14-100

2,2,2-trichloroethyl

Me

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

14-129

2,2,2-trichloroethyl

Me

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

14-158

2,2,2-trichloroethyl

Me

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

14-373

2,2,2-trichloroethyl

Me

Me

H

H

H

H

F

H

heptafluoroisopropyl

H

CF3

14-374

2,2,2-trichloroethyl

Me

Me

H

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

14-385

2,2,2-trichloroethyl

Me

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-414

2,2,2-trichloroethyl

Me

Me

H

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-443

2,2,2-trichloroethyl

Me

Me

H

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

14-472

2,2,2-trichloroethyl

Me

Me

H

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-501

2,2,2-trichloroethyl

Me

Me

H

H

H

H

I

H

heptafluoroisopropyl

H

CF3

14-530

2,2,2-trichloroethyl

Me

Me

H

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-755

2,2,2-trichloroethyl

Me

Me

H

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

14-784

2,2,2-trichloroethyl

Me

Me

H

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

14-813

2,2,2-trichloroethyl

Me

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

14-842

2,2,2-trichloroethyl

Me

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

14-871

2,2,2-trichloroethyl

Me

Me

H

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

14-900

2,2,2-trichloroethyl

Me

Me

H

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

14-1115

2,2,2-trichloroethyl

Me

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

F

14-1116

2,2,2-trichloroethyl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

14-1117

2,2,2-trichloroethyl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

14-1118

2,2,2-trichloroethyl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

I

14-1119

2,2,2-trichloroethyl

Me

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

14-1120

2,2,2-trichloroethyl

Me

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

14-1131

2,2,2-trichloroethyl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

14-1160

2,2,2-trichloroethyl

Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

14-1189

2,2,2-trichloroethyl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

14-1218

2,2,2-trichloroethyl

Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

14-1247

2,2,2-trichloroethyl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

14-1276

2,2,2-trichloroethyl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

14-1491

2,2,2-trichloroethyl

Me

Me

F

H

H

H

F

H

heptafluoroisopropyl

H

CF3

14-1492

2,2,2-trichloroethyl

Me

Me

F

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

14-1498

2-iodoethyl

Me

Et

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-1499

2-cyanoethyl

Et

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

14-1503

2,2,2-trichloroethyl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-1505

n-propyl

Me

n-Pr

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

14-1509

i-propyl

n-Pr

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

14-1512

1,3-dichloro-2-propyl

Me

Me

F

H

H

H

Cl

H

pentafluoroethyl

H

CF3

14-1513

1-chloro-3-fluoro-2-propyl

i-Pr

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-1515

n-butyl

Me

i-Pr

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-1517

i-butyl

CH2CH═CH2

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-1518

s-butyl

Me

CH2CH═CH2

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-1519

vinyl

Me

CN

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-1523

ethyl

Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

14-1528

2-cyanoethyl

CN

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-1532

2,2,2-trichloroethyl

Me

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-1533

2,2,2-tribromoethyl

Me

CH2C≡CH

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-1534

n-propyl

CH2C≡CH

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-1544

n-butyl

Me

NH2

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-1546

i-butyl

NH2

Me

F

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-1557

2-cyanoethyl

Me

C(O)OMe

F

H

H

H

Br

H

heptafluoroisopropyl

H

C2F5

14-1561

2,2,2-trichloroethyl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

14-1563

n-propyl

C(O)OMe

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

14-1568

1,2-difluoro-2-propyl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

n-C3F7

14-1574

4,4,4-trifluoro-n-butyl

Me

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

14-1575

i-butyl

Me

C(O)C(O)OMe

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

14-1577

vinyl

C(O)C(O)OMe

Me

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

14-1586

2-cyanoethyl

Me

C(O)OEt

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-1590

2,2,2-trichloroethyl

Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-1592

n-propyl

C(O)OEt

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-1595

3-bromo-n-propyl

Me

C(O)Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-1596

i-propyl

C(O)Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-1603

4,4,4-trifluoro-n-butyl

Me

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-1604

i-butyl

Me

C(O)C(O)OEt

F

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-1608

phenyl

C(O)C(O)OEt

Me

F

H

H

H

Br

H

nonafluoro-2-butyl

H

i-C3F7

14-1619

2,2,2-trichloroethyl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

14-1621

n-propyl

Me

C(O)Et

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

14-1624

3-bromo-n-propyl

C(O)Et

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

C2F5

14-1632

4,4,4-trifluoro-n-butyl

Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

14-1633

i-butyl

Me

S(O)2Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

14-1636

benzyl

S(O)2Me

Me

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

14-1643

2-iodoethyl

Me

S(O)2Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1644

2-cyanoethyl

S(O)2Et

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1648

2,2,2-trichloroethyl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1649

2,2,2-tribromoethyl

Me

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1650

n-propyl

CH2Ph

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

n-C3F7

14-1654

i-propyl

CH2(3-Py)

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1660

n-butyl

Me

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1661

4,4,4-trifluoro-n-butyl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1663

s-butyl

CH2(3-Py—N-

Me

F

H

H

H

H

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1664

vinyl

Me

Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

i-C3F7

14-1666

phenyl

Me

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1667

2,2,2-trichloroethyl

Et

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1668

2,2,2-trichloroethyl

Et

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1669

2,2,2-trichloroethyl

Et

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1670

2,2,2-trichloroethyl

Et

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1671

2,2,2-trichloroethyl

Et

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1672

2,2,2-trichloroethyl

Et

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1673

2,2,2-trichloroethyl

Et

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1674

2,2,2-trichloroethyl

Et

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1675

2,2,2-trichloroethyl

Et

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1676

2,2,2-trichloroethyl

Et

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1677

2,2,2-trichloroethyl

Et

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1678

2,2,2-trichloroethyl

Et

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1679

2,2,2-trichloroethyl

Et

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1680

2,2,2-trichloroethyl

Et

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1681

2,2,2-trichloroethyl

n-Pr

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1682

2,2,2-trichloroethyl

n-Pr

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1683

2,2,2-trichloroethyl

n-Pr

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1684

2,2,2-trichloroethyl

n-Pr

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1685

2,2,2-trichloroethyl

n-Pr

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1686

2,2,2-trichloroethyl

n-Pr

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1687

2,2,2-trichloroethyl

n-Pr

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1688

2,2,2-trichloroethyl

n-Pr

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1689

2,2,2-trichloroethyl

n-Pr

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1690

2,2,2-trichloroethyl

n-Pr

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1691

2,2,2-trichloroethyl

n-Pr

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1692

2,2,2-trichloroethyl

n-Pr

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1693

2,2,2-trichloroethyl

n-Pr

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1694

2,2,2-trichloroethyl

n-Pr

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1695

2,2,2-trichloroethyl

i-Pr

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1696

2,2,2-trichloroethyl

i-Pr

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1697

2,2,2-trichloroethyl

i-Pr

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1698

2,2,2-trichloroethyl

i-Pr

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1699

2,2,2-trichloroethyl

i-Pr

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1700

2,2,2-trichloroethyl

i-Pr

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1701

2,2,2-trichloroethyl

i-Pr

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1702

2,2,2-trichloroethyl

i-Pr

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1703

2,2,2-trichloroethyl

i-Pr

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1704

2,2,2-trichloroethyl

i-Pr

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1705

2,2,2-trichloroethyl

i-Pr

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1706

2,2,2-trichloroethyl

i-Pr

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1707

2,2,2-trichloroethyl

i-Pr

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1708

2,2,2-trichloroethyl

i-Pr

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1709

2,2,2-trichloroethyl

CH2CH═CH2

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1710

2,2,2-trichloroethyl

CH2CH═CH2

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1711

2,2,2-trichloroethyl

CH2CH═CH2

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1712

2,2,2-trichloroethyl

CH2CH═CH2

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1713

2,2,2-trichloroethyl

CH2CH═CH2

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1714

2,2,2-trichloroethyl

CH2CH═CH2

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1715

2,2,2-trichloroethyl

CH2CH═CH2

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1716

2,2,2-trichloroethyl

CH2CH═CH2

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1717

2,2,2-trichloroethyl

CH2CH═CH2

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1718

2,2,2-trichloroethyl

CH2CH═CH2

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1719

2,2,2-trichloroethyl

CH2CH═CH2

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1720

2,2,2-trichloroethyl

CH2CH═CH2

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1721

2,2,2-trichloroethyl

CH2CH═CH2

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1722

2,2,2-trichloroethyl

CH2CH═CH2

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1723

2,2,2-trichloroethyl

CN

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1724

2,2,2-trichloroethyl

CN

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1725

2,2,2-trichloroethyl

CN

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1726

2,2,2-trichloroethyl

CN

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1727

2,2,2-trichloroethyl

CN

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1728

2,2,2-trichloroethyl

CN

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1729

2,2,2-trichloroethyl

CN

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1730

2,2,2-trichloroethyl

CN

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1731

2,2,2-trichloroethyl

CN

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1732

2,2,2-trichloroethyl

CN

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1733

2,2,2-trichloroethyl

CN

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1734

2,2,2-trichloroethyl

CN

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1735

2,2,2-trichloroethyl

CN

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1736

2,2,2-trichloroethyl

CN

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1737

2,2,2-trichloroethyl

CH2C≡CH

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1738

2,2,2-trichloroethyl

CH2C≡CH

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1739

2,2,2-trichloroethyl

CH2C≡CH

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1740

2,2,2-trichloroethyl

CH2C≡CH

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1741

2,2,2-trichloroethyl

CH2C≡CH

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1742

2,2,2-trichloroethyl

CH2C≡CH

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1743

2,2,2-trichloroethyl

CH2C≡CH

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1744

2,2,2-trichloroethyl

CH2C≡CH

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1745

2,2,2-trichloroethyl

CH2C≡CH

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1746

2,2,2-trichloroethyl

CH2C≡CH

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1747

2,2,2-trichloroethyl

CH2C≡CH

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1748

2,2,2-trichloroethyl

CH2C≡CH

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1749

2,2,2-trichloroethyl

CH2C≡CH

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1750

2,2,2-trichloroethyl

CH2C≡CH

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1751

2,2,2-trichloroethyl

NH2

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1752

2,2,2-trichloroethyl

NH2

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1753

2,2,2-trichloroethyl

NH2

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1754

2,2,2-trichloroethyl

NH2

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1755

2,2,2-trichloroethyl

NH2

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1756

2,2,2-trichloroethyl

NH2

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1757

2,2,2-trichloroethyl

NH2

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1758

2,2,2-trichloroethyl

NH2

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1759

2,2,2-trichloroethyl

NH2

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1760

2,2,2-trichloroethyl

NH2

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1761

2,2,2-trichloroethyl

NH2

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1762

2,2,2-trichloroethyl

NH2

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1763

2,2,2-trichloroethyl

NH2

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1764

2,2,2-trichloroethyl

NH2

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1765

2,2,2-trichloroethyl

C(O)OMe

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1766

2,2,2-trichloroethyl

C(O)OMe

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1767

2,2,2-trichloroethyl

C(O)OMe

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1768

2,2,2-trichloroethyl

C(O)OMe

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1769

2,2,2-trichloroethyl

C(O)OMe

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1770

2,2,2-trichloroethyl

C(O)OMe

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1771

2,2,2-trichloroethyl

C(O)OMe

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1772

2,2,2-trichloroethyl

C(O)OMe

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1773

2,2,2-trichloroethyl

C(O)OMe

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1774

2,2,2-trichloroethyl

C(O)OMe

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1775

2,2,2-trichloroethyl

C(O)OMe

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1776

2,2,2-trichloroethyl

C(O)OMe

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1777

2,2,2-trichloroethyl

C(O)OMe

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1778

2,2,2-trichloroethyl

C(O)OMe

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1779

2,2,2-trichloroethyl

C(O)C(O)OMe

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1780

2,2,2-trichloroethyl

C(O)C(O)OMe

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1781

2,2,2-trichloroethyl

C(O)C(O)OMe

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1782

2,2,2-trichloroethyl

C(O)C(O)OMe

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1783

2,2,2-trichloroethyl

C(O)C(O)OMe

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1784

2,2,2-trichloroethyl

C(O)C(O)OMe

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1785

2,2,2-trichloroethyl

C(O)C(O)OMe

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1786

2,2,2-trichloroethyl

C(O)C(O)OMe

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1787

2,2,2-trichloroethyl

C(O)C(O)OMe

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1788

2,2,2-trichloroethyl

C(O)C(O)OMe

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1789

2,2,2-trichloroethyl

C(O)C(O)OMe

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1790

2,2,2-trichloroethyl

C(O)C(O)OMe

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1791

2,2,2-trichloroethyl

C(O)C(O)OMe

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1792

2,2,2-trichloroethyl

C(O)C(O)OMe

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1793

2,2,2-trichloroethyl

C(O)Me

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1794

2,2,2-trichloroethyl

C(O)Me

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1795

2,2,2-trichloroethyl

C(O)Me

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1796

2,2,2-trichloroethyl

C(O)Me

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1797

2,2,2-trichloroethyl

C(O)Me

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1798

2,2,2-trichloroethyl

C(O)Me

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1799

2,2,2-trichloroethyl

C(O)Me

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1800

2,2,2-trichloroethyl

C(O)Me

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1801

2,2,2-trichloroethyl

C(O)Me

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1802

2,2,2-trichloroethyl

C(O)Me

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1803

2,2,2-trichloroethyl

C(O)Me

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1804

2,2,2-trichloroethyl

C(O)Me

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1805

2,2,2-trichloroethyl

C(O)Me

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1806

2,2,2-trichloroethyl

C(O)Me

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1807

2,2,2-trichloroethyl

S(O)2Me

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1808

2,2,2-trichloroethyl

S(O)2Me

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1809

2,2,2-trichloroethyl

S(O)2Me

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1810

2,2,2-trichloroethyl

S(O)2Me

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1811

2,2,2-trichloroethyl

S(O)2Me

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1812

2,2,2-trichloroethyl

S(O)2Me

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1813

2,2,2-trichloroethyl

S(O)2Me

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1814

2,2,2-trichloroethyl

S(O)2Me

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1815

2,2,2-trichloroethyl

S(O)2Me

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1816

2,2,2-trichloroethyl

S(O)2Me

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1817

2,2,2-trichloroethyl

S(O)2Me

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1818

2,2,2-trichloroethyl

S(O)2Me

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1819

2,2,2-trichloroethyl

S(O)2Me

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1820

2,2,2-trichloroethyl

S(O)2Me

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1821

2,2,2-trichloroethyl

CH2Ph

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1822

2,2,2-trichloroethyl

CH2Ph

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1823

2,2,2-trichloroethyl

CH2Ph

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1824

2,2,2-trichloroethyl

CH2Ph

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1825

2,2,2-trichloroethyl

CH2Ph

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1826

2,2,2-trichloroethyl

CH2Ph

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1827

2,2,2-trichloroethyl

CH2Ph

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1828

2,2,2-trichloroethyl

CH2Ph

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1829

2,2,2-trichloroethyl

CH2Ph

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1830

2,2,2-trichloroethyl

CH2Ph

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1831

2,2,2-trichloroethyl

CH2Ph

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1832

2,2,2-trichloroethyl

CH2Ph

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1833

2,2,2-trichloroethyl

CH2Ph

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1834

2,2,2-trichloroethyl

CH2Ph

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1835

2,2,2-trichloroethyl

CH2(3-Py)

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1836

2,2,2-trichloroethyl

CH2(3-Py)

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1837

2,2,2-trichloroethyl

CH2(3-Py)

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1838

2,2,2-trichloroethyl

CH2(3-Py)

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1839

2,2,2-trichloroethyl

CH2(3-Py)

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1840

2,2,2-trichloroethyl

CH2(3-Py)

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1841

2,2,2-trichloroethyl

CH2(3-Py)

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1842

2,2,2-trichloroethyl

CH2(3-Py)

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1843

2,2,2-trichloroethyl

CH2(3-Py)

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1844

2,2,2-trichloroethyl

CH2(3-Py)

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1845

2,2,2-trichloroethyl

CH2(3-Py)

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1846

2,2,2-trichloroethyl

CH2(3-Py)

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1847

2,2,2-trichloroethyl

CH2(3-Py)

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-1848

2,2,2-trichloroethyl

CH2(3-Py)

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1849

2,2,2-trichloroethyl

CH2(3-Py—N-

Et

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1850

2,2,2-trichloroethyl

CH2(3-Py—N-

n-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1851

2,2,2-trichloroethyl

CH2(3-Py—N-

i-Pr

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1852

2,2,2-trichloroethyl

CH2(3-Py—N-

CH2CH═CH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1853

2,2,2-trichloroethyl

CH2(3-Py—N-

CN

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1854

2,2,2-trichloroethyl

CH2(3-Py—N-

CH2C≡CH

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1855

2,2,2-trichloroethyl

CH2(3-Py—N-

NH2

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1856

2,2,2-trichloroethyl

CH2(3-Py—N-

C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1857

2,2,2-trichloroethyl

CH2(3-Py—N-

C(O)C(O)OMe

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1858

2,2,2-trichloroethyl

CH2(3-Py—N-

C(O)Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1859

2,2,2-trichloroethyl

CH2(3-Py—N-

S(O)2Me

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1860

2,2,2-trichloroethyl

CH2(3-Py—N-

CH2Ph

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1861

2,2,2-trichloroethyl

CH2(3-Py—N-

CH2(3-Py)

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

14-1862

2,2,2-trichloroethyl

CH2(3-Py—N-

CH2(3-Py—N-

F

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

oxide)

14-1873

2,2,2-trichloroethyl

Me

Me

F

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

14-1902

2,2,2-trichloroethyl

Me

Me

F

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

14-1931

2,2,2-trichloroethyl

Me

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

14-1960

2,2,2-trichloroethyl

Me

Me

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

14-1989

2,2,2-trichloroethyl

Me

Me

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

14-2019

2,2,2-trichloroethyl

Me

CH2C≡CH

F

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

14-2233

2,2,2-trichloroethyl

Me

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

F

14-2234

2,2,2-trichloroethyl

Me

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

F

14-2245

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

14-2274

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

14-2303

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

Br

14-2332

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

14-2361

2,2,2-trichloroethyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

I

14-2390

2,2,2-trichloroethyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

I

13-1236

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

Br

14-2605

2,2,2-trichloroethyl

Me

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

OCF3

14-2606

2,2,2-trichloroethyl

Me

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

OCF3

14-2617

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

14-2646

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

14-2675

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

14-2704

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

14-2733

2,2,2-trichloroethyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

14-2762

2,2,2-trichloroethyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

14-2977

2,2,2-trichloroethyl

Me

Me

H

F

H

H

F

H

heptafluoroisopropyl

H

CF3

14-2978

2,2,2-trichloroethyl

Me

Me

H

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

14-2989

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-3018

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-3047

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

14-3076

2,2,2-trichloroethyl

Me

Me

H

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-3105

2,2,2-trichloroethyl

Me

Me

H

F

H

H

I

H

heptafluoroisopropyl

H

CF3

14-3134

2,2,2-trichloroethyl

Me

Me

H

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-3359

2,2,2-trichloroethyl

Me

Me

H

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

14-3388

2,2,2-trichloroethyl

Me

Me

H

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

14-3417

2,2,2-trichloroethyl

Me

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

14-3446

2,2,2-trichloroethyl

Me

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

14-3475

2,2,2-trichloroethyl

Me

Me

H

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

14-3504

2,2,2-trichloroethyl

Me

Me

H

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

14-3719

2,2,2-trichloroethyl

Me

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

F

14-3720

2,2,2-trichloroethyl

Me

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

F

14-3731

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Cl

14-3760

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

14-3789

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

Br

14-3818

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

Br

14-3847

2,2,2-trichloroethyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

I

14-3876

2,2,2-trichloroethyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

I

13-1950

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

Br

14-4091

2,2,2-trichloroethyl

Me

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

OCF3

14-4092

2,2,2-trichloroethyl

Me

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

OCF3

14-4103

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

14-4132

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

14-4161

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

OCF3

14-4190

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

14-4219

2,2,2-trichloroethyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

OCF3

14-4248

2,2,2-trichloroethyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

OCF3

14-4463

2,2,2-trichloroethyl

Me

Me

F

F

H

H

F

H

heptafluoroisopropyl

H

CF3

14-4464

2,2,2-trichloroethyl

Me

Me

F

F

H

H

F

H

nonafluoro-2-butyl

H

CF3

14-4475

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-4504

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-4533

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Br

H

heptafluoroisopropyl

H

CF3

14-4562

2,2,2-trichloroethyl

Me

Me

F

F

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-4591

2,2,2-trichloroethyl

Me

Me

F

F

H

H

I

H

heptafluoroisopropyl

H

CF3

14-4620

2,2,2-trichloroethyl

Me

Me

F

F

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-4845

2,2,2-trichloroethyl

Me

Me

F

F

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

14-4874

2,2,2-trichloroethyl

Me

Me

F

F

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

14-4903

2,2,2-trichloroethyl

Me

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

14-4932

2,2,2-trichloroethyl

Me

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

14-4961

2,2,2-trichloroethyl

Me

Me

F

F

H

H

CF3

H

heptafluoroisopropyl

H

CF3

14-4990

2,2,2-trichloroethyl

Me

Me

F

F

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

14-5205

2,2,2-trichloroethyl

Me

Me

F

F

F

H

Cl

H

pentafluoroethyl

H

Cl

14-5206

2,2,2-trichloroethyl

Me

Me

F

F

F

H

Br

H

heptafluoroisopropyl

H

Br

14-5207

2,2,2-trichloroethyl

Me

Me

F

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

14-5208

2,2,2-trichloroethyl

Me

Me

F

F

F

H

I

H

heptafluoroisopropyl

H

CF3

14-5209

2,2,2-trichloroethyl

Me

Me

F

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

14-5210

2,2,2-trichloroethyl

Me

Me

F

F

F

H

I

H

nonafluoro-2-butyl

H

I

14-5211

2,2,2-trichloroethyl

Me

Me

F

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5212

2,2,2-trichloroethyl

Me

Me

F

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

14-5213

2,2,2-trichloroethyl

Me

Me

F

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

14-5214

2,2,2-trichloroethyl

Me

Me

H

H

F

H

Cl

H

pentafluoroethyl

H

Cl

14-5215

2,2,2-trichloroethyl

Me

Me

H

H

F

H

Br

H

heptafluoroisopropyl

H

Br

14-5216

2,2,2-trichloroethyl

Me

Me

H

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

14-5217

2,2,2-trichloroethyl

Me

Me

H

H

F

H

I

H

heptafluoroisopropyl

H

CF3

14-5218

2,2,2-trichloroethyl

Me

Me

H

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

14-5219

2,2,2-trichloroethyl

Me

Me

H

H

F

H

I

H

nonafluoro-2-butyl

H

I

14-5220

2,2,2-trichloroethyl

Me

Me

H

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5221

2,2,2-trichloroethyl

Me

Me

H

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

14-5222

2,2,2-trichloroethyl

Me

Me

H

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

14-5223

2,2,2-trichloroethyl

Me

Me

H

H

H

F

Cl

H

pentafluoroethyl

H

Cl

14-5224

2,2,2-trichloroethyl

Me

Me

H

H

H

F

Br

H

heptafluoroisopropyl

H

Br

14-5225

2,2,2-trichloroethyl

Me

Me

H

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

14-5226

2,2,2-trichloroethyl

Me

Me

H

H

H

F

I

H

heptafluoroisopropyl

H

CF3

14-5227

2,2,2-trichloroethyl

Me

Me

H

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

14-5228

2,2,2-trichloroethyl

Me

Me

H

H

H

F

I

H

nonafluoro-2-butyl

H

I

14-5229

2,2,2-trichloroethyl

Me

Me

H

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5230

2,2,2-trichloroethyl

Me

Me

H

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

14-5231

2,2,2-trichloroethyl

Me

Me

H

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

14-5232

2,2,2-trichloroethyl

Me

Me

F

H

F

H

Cl

H

pentafluoroethyl

H

Cl

14-5233

2,2,2-trichloroethyl

Me

Me

F

H

F

H

Br

H

heptafluoroisopropyl

H

Br

14-5234

2,2,2-trichloroethyl

Me

Me

F

H

F

H

Br

H

heptafluoroisopropyl

H

OCF3

14-5235

2,2,2-trichloroethyl

Me

Me

F

H

F

H

I

H

heptafluoroisopropyl

H

CF3

14-5236

2,2,2-trichloroethyl

Me

Me

F

H

F

H

CF3

H

heptafluoroisopropyl

H

CF3

14-5237

2,2,2-trichloroethyl

Me

Me

F

H

F

H

I

H

nonafluoro-2-butyl

H

I

14-5238

2,2,2-trichloroethyl

Me

Me

F

H

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5239

2,2,2-trichloroethyl

Me

Me

F

H

F

H

Br

H

nonafluoro-2-butyl

H

CF3

14-5240

2,2,2-trichloroethyl

Me

Me

F

H

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

14-5241

2,2,2-trichloroethyl

Me

Me

F

H

H

F

Cl

H

pentafluoroethyl

H

Cl

14-5242

2,2,2-trichloroethyl

Me

Me

F

H

H

F

Br

H

heptafluoroisopropyl

H

Br

14-5243

2,2,2-trichloroethyl

Me

Me

F

H

H

F

Br

H

heptafluoroisopropyl

H

OCF3

14-5244

2,2,2-trichloroethyl

Me

Me

F

H

H

F

I

H

heptafluoroisopropyl

H

CF3

14-5245

2,2,2-trichloroethyl

Me

Me

F

H

H

F

CF3

H

heptafluoroisopropyl

H

CF3

14-5246

2,2,2-trichloroethyl

Me

Me

F

H

H

F

I

H

nonafluoro-2-butyl

H

I

14-5247

2,2,2-trichloroethyl

Me

Me

F

H

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5248

2,2,2-trichloroethyl

Me

Me

F

H

H

F

Br

H

nonafluoro-2-butyl

H

CF3

14-5249

2,2,2-trichloroethyl

Me

Me

F

H

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

14-5250

2,2,2-trichloroethyl

Me

Me

H

F

F

H

Cl

H

pentafluoroethyl

H

Cl

14-5251

2,2,2-trichloroethyl

Me

Me

H

F

F

H

Br

H

heptafluoroisopropyl

H

Br

14-5252

2,2,2-trichloroethyl

Me

Me

H

F

F

H

Br

H

heptafluoroisopropyl

H

OCF3

14-5253

2,2,2-trichloroethyl

Me

Me

H

F

F

H

I

H

heptafluoroisopropyl

H

CF3

14-5254

2,2,2-trichloroethyl

Me

Me

H

F

F

H

CF3

H

heptafluoroisopropyl

H

CF3

14-5255

2,2,2-trichloroethyl

Me

Me

H

F

F

H

I

H

nonafluoro-2-butyl

H

I

14-5256

2,2,2-trichloroethyl

Me

Me

H

F

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5257

2,2,2-trichloroethyl

Me

Me

H

F

F

H

Br

H

nonafluoro-2-butyl

H

CF3

14-5258

2,2,2-trichloroethyl

Me

Me

H

F

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

14-5259

2,2,2-trichloroethyl

Me

Me

H

F

H

F

Cl

H

pentafluoroethyl

H

Cl

14-5260

2,2,2-trichloroethyl

Me

Me

H

F

H

F

Br

H

heptafluoroisopropyl

H

Br

14-5261

2,2,2-trichloroethyl

Me

Me

H

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

14-5262

2,2,2-trichloroethyl

Me

Me

H

F

H

F

I

H

heptafluoroisopropyl

H

CF3

14-5263

2,2,2-trichloroethyl

Me

Me

H

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

14-5264

2,2,2-trichloroethyl

Me

Me

H

F

H

F

I

H

nonafluoro-2-butyl

H

I

14-5265

2,2,2-trichloroethyl

Me

Me

H

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5266

2,2,2-trichloroethyl

Me

Me

H

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

14-5267

2,2,2-trichloroethyl

Me

Me

H

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

14-5268

2,2,2-trichloroethyl

Me

Me

H

H

F

F

Cl

H

pentafluoroethyl

H

Cl

14-5269

2,2,2-trichloroethyl

Me

Me

H

H

F

F

Br

H

heptafluoroisopropyl

H

Br

14-5270

2,2,2-trichloroethyl

Me

Me

H

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

14-5271

2,2,2-trichloroethyl

Me

Me

H

H

F

F

I

H

heptafluoroisopropyl

H

CF3

14-5272

2,2,2-trichloroethyl

Me

Me

H

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

14-5273

2,2,2-trichloroethyl

Me

Me

H

H

F

F

I

H

nonafluoro-2-butyl

H

I

14-5274

2,2,2-trichloroethyl

Me

Me

H

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5275

2,2,2-trichloroethyl

Me

Me

H

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

14-5276

2,2,2-trichloroethyl

Me

Me

H

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

14-5277

2,2,2-trichloroethyl

Me

Me

F

F

H

F

Cl

H

pentafluoroethyl

H

Cl

14-5278

2,2,2-trichloroethyl

Me

Me

F

F

H

F

Br

H

heptafluoroisopropyl

H

Br

14-5279

2,2,2-trichloroethyl

Me

Me

F

F

H

F

Br

H

heptafluoroisopropyl

H

OCF3

14-5280

2,2,2-trichloroethyl

Me

Me

F

F

H

F

I

H

heptafluoroisopropyl

H

CF3

14-5281

2,2,2-trichloroethyl

Me

Me

F

F

H

F

CF3

H

heptafluoroisopropyl

H

CF3

14-5282

2,2,2-trichloroethyl

Me

Me

F

F

H

F

I

H

nonafluoro-2-butyl

H

I

14-5283

2,2,2-trichloroethyl

Me

Me

F

F

H

F

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5284

2,2,2-trichloroethyl

Me

Me

F

F

H

F

Br

H

nonafluoro-2-butyl

H

CF3

14-5285

2,2,2-trichloroethyl

Me

Me

F

F

H

F

CF3

H

nonafluoro-2-butyl

H

CF3

14-5286

2,2,2-trichloroethyl

Me

Me

F

H

F

F

Cl

H

pentafluoroethyl

H

Cl

14-5287

2,2,2-trichloroethyl

Me

Me

F

H

F

F

Br

H

heptafluoroisopropyl

H

Br

14-5288

2,2,2-trichloroethyl

Me

Me

F

H

F

F

Br

H

heptafluoroisopropyl

H

OCF3

14-5289

2,2,2-trichloroethyl

Me

Me

F

H

F

F

I

H

heptafluoroisopropyl

H

CF3

14-5290

2,2,2-trichloroethyl

Me

Me

F

H

F

F

CF3

H

heptafluoroisopropyl

H

CF3

14-5291

2,2,2-trichloroethyl

Me

Me

F

H

F

F

I

H

nonafluoro-2-butyl

H

I

14-5292

2,2,2-trichloroethyl

Me

Me

F

H

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5293

2,2,2-trichloroethyl

Me

Me

F

H

F

F

Br

H

nonafluoro-2-butyl

H

CF3

14-5294

2,2,2-trichloroethyl

Me

Me

F

H

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

14-5295

2,2,2-trichloroethyl

Me

Me

H

F

F

F

Cl

H

pentafluoroethyl

H

Cl

14-5296

2,2,2-trichloroethyl

Me

Me

H

F

F

F

Br

H

heptafluoroisopropyl

H

Br

14-5297

2,2,2-trichloroethyl

Me

Me

H

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

14-5298

2,2,2-trichloroethyl

Me

Me

H

F

F

F

I

H

heptafluoroisopropyl

H

CF3

14-5299

2,2,2-trichloroethyl

Me

Me

H

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

14-5300

2,2,2-trichloroethyl

Me

Me

H

F

F

F

I

H

nonafluoro-2-butyl

H

I

14-5301

2,2,2-trichloroethyl

Me

Me

H

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5302

2,2,2-trichloroethyl

Me

Me

H

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

14-5303

2,2,2-trichloroethyl

Me

Me

H

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

14-5304

2,2,2-trichloroethyl

Me

Me

F

F

F

F

Cl

H

pentafluoroethyl

H

Cl

14-5305

2,2,2-trichloroethyl

Me

Me

F

F

F

F

Br

H

heptafluoroisopropyl

H

Br

14-5306

2,2,2-trichloroethyl

Me

Me

F

F

F

F

Br

H

heptafluoroisopropyl

H

OCF3

14-5307

2,2,2-trichloroethyl

Me

Me

F

F

F

F

I

H

heptafluoroisopropyl

H

CF3

14-5308

2,2,2-trichloroethyl

Me

Me

F

F

F

F

CF3

H

heptafluoroisopropyl

H

CF3

14-5309

2,2,2-trichloroethyl

Me

Me

F

F

F

F

I

H

nonafluoro-2-butyl

H

I

14-5310

2,2,2-trichloroethyl

Me

Me

F

F

F

F

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5311

2,2,2-trichloroethyl

Me

Me

F

F

F

F

Br

H

nonafluoro-2-butyl

H

CF3

14-5312

2,2,2-trichloroethyl

Me

Me

F

F

F

F

CF3

H

nonafluoro-2-butyl

H

CF3

14-5313

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

F

H

heptafluoroisopropyl

H

OCF3

14-5314

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

F

H

nonafluoro-2-butyl

H

OCF3

14-5325

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

14-5354

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

14-5383

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

14-5412

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

14-5441

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

14-5470

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

14-5685

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

14-5686

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

14-5697

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-5726

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-5755

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

14-5784

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-5813

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

14-5842

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-6067

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

14-6096

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

14-6125

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

14-6154

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

14-6183

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

14-6212

2,2,2-trichloroethyl

Me

Me

H

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

14-6427

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

F

H

heptafluoroisopropyl

H

F

14-6428

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

F

H

nonafluoro-2-butyl

H

F

14-6439

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

Cl

14-6468

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

14-6497

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

Br

14-6526

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

Br

14-6555

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

I

14-6584

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

I

13-3306

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

I

14-6799

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

F

H

heptafluoroisopropyl

H

OCF3

14-6800

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

F

H

nonafluoro-2-butyl

H

OCF3

14-6811

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

14-6840

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

14-6869

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

OCF3

14-6898

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

14-6927

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

OCF3

14-6956

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

OCF3

14-7171

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

F

H

heptafluoroisopropyl

H

CF3

14-7172

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

F

H

nonafluoro-2-butyl

H

CF3

14-7183

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

H

CF3

14-7212

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-7241

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Br

H

heptafluoroisopropyl

H

CF3

14-7270

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

Br

H

nonafluoro-2-butyl

H

CF3

14-7299

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

I

H

heptafluoroisopropyl

H

CF3

14-7328

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

I

H

nonafluoro-2-butyl

H

CF3

14-7553

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

14-7582

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

14-7611

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

14-7640

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

14-7669

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

CF3

H

heptafluoroisopropyl

H

CF3

14-7698

2,2,2-trichloroethyl

Me

Me

F

CN

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

14-7913

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

F

H

heptafluoroisopropyl

H

F

14-7914

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

F

H

nonafluoro-2-butyl

H

F

14-7925

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

Cl

14-7954

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

Cl

14-7983

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

Br

14-8012

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

Br

14-8041

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

I

14-8070

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

I

13-4012

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

Br

14-8285

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

F

H

heptafluoroisopropyl

H

OCF3

14-8286

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

F

H

nonafluoro-2-butyl

H

OCF3

14-8297

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

OCF3

14-8326

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

OCF3

14-8355

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

OCF3

14-8384

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

OCF3

14-8413

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

OCF3

14-8442

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

OCF3

14-8657

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

F

H

heptafluoroisopropyl

H

CF3

14-8658

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

F

H

nonafluoro-2-butyl

H

CF3

14-8669

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Cl

H

heptafluoroisopropyl

H

CF3

14-8698

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Cl

H

nonafluoro-2-butyl

H

CF3

14-8727

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Br

H

heptafluoroisopropyl

H

CF3

14-8756

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

Br

H

nonafluoro-2-butyl

H

CF3

14-8785

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

I

H

heptafluoroisopropyl

H

CF3

14-8814

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

I

H

nonafluoro-2-butyl

H

CF3

14-9039

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

OCF3

H

heptafluoroisopropyl

H

OCF3

14-9068

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

14-9097

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

OCF3

14-9126

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

OCF3

14-9155

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

CF3

H

heptafluoroisopropyl

H

CF3

14-9184

2,2,2-trichloroethyl

Me

Me

F

CN

F

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 15

compound

number

Q2

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

15-9

2,2-dichloroethyl

H

Et

H

H

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

15-39

2,2,2-trifluoroethyl

H

H

H

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

15-144

methyl

H

H

H

H

H

H

Cl

F

heptafluoroisopropyl

H

CF3

15-147

2-chloroethyl

Me

Me

H

H

H

H

Cl

H

heptafluoroisopropyl

Cl

CF3

15-148

2-bromoethyl

H

H

H

H

H

H

F

Br

heptafluoroisopropyl

H

CF3

15-153

2,2,2-trifluoroethyl

H

H

H

H

H

H

Cl

F

heptafluoroisopropyl

Cl

CF3

15-165

3,3,3-trifluoro-n-propyl

H

H

H

H

H

H

Cl

I

nonafluoro-2-butyl

Cl

CF3

15-168

i-butyl

H

H

H

H

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

15-169

s-butyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

15-170

vinyl

i-Pr

H

H

H

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

15-171

benzyl

H

H

H

H

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

15-182

2,2,2-trifluoroethyl

H

H

H

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

15-183

2,2,2-trichloroethyl

H

H

H

H

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

15-189

i-propyl

H

H

H

H

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

15-190

1,2-difluoro-2-propyl

H

H

H

H

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

15-196

2-chloroethyl

H

H

H

H

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

15-197

2-bromoethyl

H

H

H

H

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

15-203

2,2,2-trichloroethyl

H

H

H

H

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

15-204

2,2,2-tribromoethyl

H

H

H

H

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

15-210

1,2-difluoro-2-propyl

H

H

H

H

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

15-211

1,3-difluoro-2-propyl

H

H

H

H

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

15-217

i-butyl

H

H

H

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

15-218

s-butyl

H

H

H

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

15-224

2-fluoroethyl

H

H

H

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

15-225

2-chloroethyl

H

H

H

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

15-231

2,2,2-trifluoroethyl

H

H

H

H

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

15-232

2,2,2-trichloroethyl

H

H

H

H

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

15-238

i-propyl

Et

i-Pr

H

H

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

15-239

1,2-difluoro-2-propyl

H

H

H

H

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

15-245

2-iodoethyl

H

H

H

H

H

H

I

Br

heptafluoroisopropyl

Me

CF3

15-246

2-cyanoethyl

H

H

H

H

H

H

I

Br

heptafluoroisopropyl

Et

CF3

15-252

n-propyl

n-Pr

Me

H

H

H

H

I

I

heptafluoroisopropyl

Me

CF3

15-253

3-fluoro-n-propyl

H

H

H

H

H

H

I

I

heptafluoroisopropyl

Et

CF3

15-259

1,3-dichloro-2-propyl

H

H

H

H

H

H

I

Me

heptafluoroisopropyl

F

C2F5

15-260

1-chloro-3-fluoro-2-propyl

H

H

H

H

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

15-263

4,4,4-trifluoro-n-butyl

H

H

H

H

H

H

I

Et

nonafluoro-2-butyl

F

CF3

15-264

i-butyl

H

H

H

H

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

15-267

benzyl

H

H

H

H

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

15-268

phenyl

H

H

H

H

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

15-271

2-fluoroethyl

H

H

H

H

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

15-272

2-chloroethyl

H

H

H

H

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

15-275

2-cyanoethyl

H

H

H

H

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

15-276

2,2-difluoroethyl

H

H

H

H

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

15-279

2,2,2-trichloroethyl

H

H

H

H

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

15-280

2,2,2-tribromoethyl

H

H

H

H

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

15-283

3-chloro-n-propyl

i-Pr

n-Pr

H

H

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

15-284

3-bromo-n-propyl

H

H

H

H

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

15-295

2,2-dichloroethyl

H

Et

H

H

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

15-325

2,2,2-trifluoroethyl

H

H

H

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

15-438

2,2-dichloroethyl

H

Et

H

H

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

15-468

2,2,2-trifluoroethyl

H

H

H

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

15-581

2,2-dichloroethyl

H

Et

H

H

H

H

CF3

F

heptafluoroisopropyl

F

CF3

15-611

2,2,2-trifluoroethyl

H

H

H

H

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

15-734

2,2-dichloroethyl

H

Et

F

H

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

15-764

2,2,2-trifluoroethyl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

15-869

methyl

H

H

F

H

H

H

Cl

F

heptafluoroisopropyl

H

CF3

15-870

ethyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

F

CF3

15-871

2-fluoroethyl

H

Me

F

H

H

H

Cl

Cl

heptafluoroisopropyl

H

CF3

15-872

2-chloroethyl

Me

Me

F

H

H

H

Cl

H

heptafluoroisopropyl

Cl

CF3

15-873

2-bromoethyl

H

H

F

H

H

H

F

Br

heptafluoroisopropyl

H

CF3

15-874

2-iodoethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

Br

CF3

15-875

2-cyanoethyl

Et

H

F

H

H

H

Cl

I

heptafluoroisopropyl

H

C2F5

15-876

2,2-difluoroethyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

I

CF3

15-877

2,2-dichloroethyl

H

Et

F

H

H

H

Cl

F

heptafluoroisopropyl

F

CF3

15-878

2,2,2-trifluoroethyl

H

H

F

H

H

H

Cl

F

heptafluoroisopropyl

Cl

CF3

15-879

2,2,2-trichloroethyl

H

H

F

H

H

H

Cl

F

heptafluoroisopropyl

Br

CF3

15-880

2,2,2-tribromoethyl

Et

Et

F

H

H

H

Cl

F

pentafluoroethyl

I

C2F5

15-881

n-propyl

H

H

F

H

H

H

Cl

Cl

pentafluoroethyl

F

CF3

15-882

3-fluoro-n-propyl

H

H

F

H

H

H

Cl

Cl

heptafluoroisopropyl

Cl

CF3

15-883

3-chloro-n-propyl

n-Pr

H

F

H

H

H

Cl

Cl

heptafluoroisopropyl

Br

CF3

15-884

3-bromo-n-propyl

H

H

F

H

H

H

Cl

Cl

heptafluoroisopropyl

I

n-C3F7

15-885

i-propyl

H

n-Pr

F

H

H

H

Cl

Br

heptafluoroisopropyl

F

CF3

15-886

1,2-difluoro-2-propyl

H

H

F

H

H

H

Cl

Br

heptafluoroisopropyl

Cl

CF3

15-887

1,3-difluoro-2-propyl

H

H

F

H

H

H

Cl

Br

heptafluoroisopropyl

Br

CF3

15-888

1,3-dichloro-2-propyl

n-Pr

n-Pr

F

H

H

H

Cl

Br

pentafluoroethyl

I

CF3

15-889

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

F

I

nonafluoro-2-butyl

F

CF3

15-890

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

Cl

I

nonafluoro-2-butyl

Cl

CF3

15-891

n-butyl

H

H

F

H

H

H

Cl

I

nonafluoro-2-butyl

Br

CF3

15-892

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

Cl

I

nonafluoro-2-butyl

I

CF3

15-893

i-butyl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

15-894

s-butyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

15-895

vinyl

i-Pr

H

F

H

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

15-896

benzyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

15-897

phenyl

H

H

F

H

H

H

Cl

n-Pr

nonafluoro-2-butyl

H

CF3

15-898

methyl

H

i-Pr

F

H

H

H

Cl

H

nonafluoro-2-butyl

n-Pr

CF3

15-899

ethyl

i-Pr

i-Pr

F

H

H

H

Cl

i-Pr

nonafluoro-2-butyl

H

CF3

15-900

2-fluoroethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

i-Pr

CF3

15-901

2-chloroethyl

H

H

F

H

H

H

Cl

n-Bu

nonafluoro-2-butyl

H

CF3

15-902

2-bromoethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

n-Bu

CF3

15-903

2-iodoethyl

H

H

F

H

H

H

Cl

i-Bu

nonafluoro-2-butyl

H

CF3

15-904

2-cyanoethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

i-Bu

CF3

15-905

2,2-difluoroethyl

H

H

F

H

H

H

Cl

s-Bu

nonafluoro-2-butyl

H

C2F5

15-906

2,2-dichloroethyl

H

H

F

H

H

H

Cl

H

nonafluoro-2-butyl

s-Bu

CF3

15-907

2,2,2-trifluoroethyl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

15-908

2,2,2-trichloroethyl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

15-909

2,2,2-tribromoethyl

C(O)Me

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

n-Pr

CF3

15-910

n-propyl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

i-Pr

CF3

15-911

3-fluoro-n-propyl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

n-Bu

CF3

15-912

3-chloro-n-propyl

H

H

F

H

H

H

Cl

Me

nonafluoro-2-butyl

i-Bu

CF3

15-913

3-bromo-n-propyl

H

C(O)Me

F

H

H

H

Cl

Me

nonafluoro-2-butyl

s-Bu

CF3

15-914

i-propyl

H

H

F

H

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

15-915

1,2-difluoro-2-propyl

H

H

F

H

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

15-916

1,3-difluoro-2-propyl

C(O)Me

C(O)Me

F

H

H

H

Cl

Et

nonafluoro-2-butyl

n-Pr

CF3

15-917

1,3-dichloro-2-propyl

H

H

F

H

H

H

Cl

Et

nonafluoro-2-butyl

i-Pr

CF3

15-918

methyl

H

H

F

H

H

H

Br

Et

heptafluoroisopropyl

n-Bu

CF3

15-919

ethyl

H

H

F

H

H

H

Br

Et

heptafluoroisopropyl

i-Bu

CF3

15-920

2-fluoroethyl

H

H

F

H

H

H

Br

Et

heptafluoroisopropyl

s-Bu

CF3

15-921

2-chloroethyl

H

H

F

H

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

15-922

2-bromoethyl

H

H

F

H

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

15-923

2-iodoethyl

Me

Et

F

H

H

H

Br

n-Pr

pentafluoroethyl

n-Pr

CF3

15-924

2-cyanoethyl

H

H

F

H

H

H

Br

n-Pr

heptafluoroisopropyl

i-Pr

CF3

15-925

2,2-difluoroethyl

H

H

F

H

H

H

Br

n-Pr

pentafluoroethyl

n-Bu

CF3

15-926

2,2-dichloroethyl

H

H

F

H

H

H

Br

n-Pr

heptafluoroisopropyl

i-Bu

CF3

15-927

2,2,2-trifluoroethyl

H

H

F

H

H

H

Br

n-Pr

heptafluoroisopropyl

s-Bu

CF3

15-928

2,2,2-trichloroethyl

H

H

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

15-929

2,2,2-tribromoethyl

H

H

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

15-930

n-propyl

Me

n-Pr

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

n-Pr

CF3

15-931

3-fluoro-n-propyl

H

H

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

i-Pr

CF3

15-932

3-chloro-n-propyl

H

H

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

n-Bu

CF3

15-933

3-bromo-n-propyl

H

H

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

i-Bu

CF3

15-934

i-propyl

Me

i-Pr

F

H

H

H

Br

i-Pr

heptafluoroisopropyl

s-Bu

CF3

15-935

1,2-difluoro-2-propyl

H

H

F

H

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

15-936

1,3-difluoro-2-propyl

H

H

F

H

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

15-937

1,3-dichloro-2-propyl

H

H

F

H

H

H

Br

n-Bu

heptafluoroisopropyl

n-Pr

CF3

15-938

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

Br

n-Bu

nonafluoro-2-butyl

i-Pr

CF3

15-939

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

Br

n-Bu

nonafluoro-2-butyl

n-Bu

CF3

15-940

n-butyl

H

H

F

H

H

H

Br

n-Bu

nonafluoro-2-butyl

i-Bu

CF3

15-941

4,4,4-trifluoro-n-butyl

Me

C(O)Me

F

H

H

H

Br

n-Bu

nonafluoro-2-butyl

s-Bu

CF3

15-942

i-butyl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

15-943

s-butyl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

15-944

vinyl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

n-Pr

CF3

15-945

benzyl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

i-Pr

CF3

15-946

phenyl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

n-Bu

CF3

15-947

methyl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

i-Bu

CF3

15-948

ethyl

H

H

F

H

H

H

Br

i-Bu

nonafluoro-2-butyl

s-Bu

C2F5

15-949

2-fluoroethyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

15-950

2-chloroethyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

15-951

2-bromoethyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

n-Pr

CF3

15-952

2-iodoethyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

i-Pr

CF3

15-953

2-cyanoethyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

n-Bu

CF3

15-954

2,2-difluoroethyl

H

H

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

i-Bu

CF3

15-955

2,2-dichloroethyl

Et

Me

F

H

H

H

Br

s-Bu

nonafluoro-2-butyl

s-Bu

CF3

15-956

2,2,2-trifluoroethyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

15-957

2,2,2-trichloroethyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

15-958

2,2,2-tribromoethyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

n-Pr

CF3

15-959

n-propyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

i-Pr

CF3

15-960

3-fluoro-n-propyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

n-Bu

CF3

15-961

3-chloro-n-propyl

H

H

F

H

H

H

Br

F

nonafluoro-2-butyl

i-Bu

CF3

15-962

3-bromo-n-propyl

Et

n-Pr

F

H

H

H

Br

F

nonafluoro-2-butyl

s-Bu

CF3

15-963

i-propyl

Et

i-Pr

F

H

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

15-964

1,2-difluoro-2-propyl

H

H

F

H

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

15-965

methyl

H

H

F

H

H

H

I

Cl

pentafluoroethyl

n-Pr

i-C3F7

15-966

ethyl

H

H

F

H

H

H

I

Cl

heptafluoroisopropyl

i-Pr

CF3

15-967

2-fluoroethyl

H

H

F

H

H

H

I

Cl

heptafluoroisopropyl

n-Bu

CF3

15-968

2-chloroethyl

Et

C(O)Me

F

H

H

H

I

Cl

heptafluoroisopropyl

i-Bu

CF3

15-969

2-bromoethyl

H

H

F

H

H

H

I

Cl

heptafluoroisopropyl

s-Bu

CF3

15-970

2-iodoethyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

Me

CF3

15-971

2-cyanoethyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

Et

CF3

15-972

2,2-difluoroethyl

H

H

F

H

H

H

I

Br

pentafluoroethyl

n-Pr

CF3

15-973

2,2-dichloroethyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

i-Pr

CF3

15-974

2,2,2-trifluoroethyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

n-Bu

CF3

15-975

2,2,2-trichloroethyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

i-Bu

CF3

15-976

2,2,2-tribromoethyl

H

H

F

H

H

H

I

Br

heptafluoroisopropyl

s-Bu

CF3

15-977

n-propyl

n-Pr

Me

F

H

H

H

I

I

heptafluoroisopropyl

Me

CF3

15-978

3-fluoro-n-propyl

H

H

F

H

H

H

I

I

heptafluoroisopropyl

Et

CF3

15-979

3-chloro-n-propyl

n-Pr

Et

F

H

H

H

I

I

heptafluoroisopropyl

n-Pr

CF3

15-980

3-bromo-n-propyl

H

H

F

H

H

H

I

I

heptafluoroisopropyl

i-Pr

CF3

15-981

i-propyl

H

H

F

H

H

H

I

I

heptafluoroisopropyl

n-Bu

CF3

15-982

1,2-difluoro-2-propyl

H

H

F

H

H

H

I

I

heptafluoroisopropyl

i-Bu

CF3

15-983

1,3-difluoro-2-propyl

H

H

F

H

H

H

I

I

heptafluoroisopropyl

s-Bu

CF3

15-984

1,3-dichloro-2-propyl

H

H

F

H

H

H

I

Me

heptafluoroisopropyl

F

C2F5

15-985

1-chloro-3-fluoro-2-propyl

H

H

F

H

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

15-986

3,3,3-trifluoro-n-propyl

H

H

F

H

H

H

I

Me

nonafluoro-2-butyl

Br

n-C3F7

15-987

n-butyl

H

H

F

H

H

H

I

Me

nonafluoro-2-butyl

I

i-C3F7

15-988

4,4,4-trifluoro-n-butyl

H

H

F

H

H

H

I

Et

nonafluoro-2-butyl

F

CF3

15-989

i-butyl

H

H

F

H

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

15-990

s-butyl

H

H

F

H

H

H

I

Et

nonafluoro-2-butyl

Br

CF3

15-991

vinyl

n-Pr

i-Pr

F

H

H

H

I

Et

nonafluoro-2-butyl

I

C2F5

15-992

benzyl

H

H

F

H

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

15-993

phenyl

H

H

F

H

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

15-994

methyl

H

H

F

H

H

H

I

n-Pr

nonafluoro-2-butyl

Br

CF3

15-995

ethyl

H

H

F

H

H

H

I

n-Pr

nonafluoro-2-butyl

I

n-C3F7

15-996

2-fluoroethyl

H

H

F

H

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

15-997

2-chloroethyl

H

H

F

H

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

15-998

2-bromoethyl

n-Pr

C(O)Me

F

H

H

H

I

i-Pr

nonafluoro-2-butyl

Br

CF3

15-999

2-iodoethyl

H

H

F

H

H

H

I

i-Pr

nonafluoro-2-butyl

I

CF3

15-1000

2-cyanoethyl

H

H

F

H

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

15-1001

2,2-difluoroethyl

H

H

F

H

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

15-1002

2,2-dichloroethyl

H

H

F

H

H

H

I

n-Bu

nonafluoro-2-butyl

Br

CF3

15-1003

2,2,2-trifluoroethyl

i-Pr

Me

F

H

H

H

I

n-Bu

nonafluoro-2-butyl

I

CF3

15-1004

2,2,2-trichloroethyl

H

H

F

H

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

15-1005

2,2,2-tribromoethyl

H

H

F

H

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

15-1006

n-propyl

H

H

F

H

H

H

I

i-Bu

nonafluoro-2-butyl

Br

CF3

15-1007

3-fluoro-n-propyl

i-Pr

Et

F

H

H

H

I

i-Bu

nonafluoro-2-butyl

I

CF3

15-1008

3-chloro-n-propyl

i-Pr

n-Pr

F

H

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

15-1009

3-bromo-n-propyl

H

H

F

H

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

15-1010

i-propyl

i-Pr

C(O)Me

F

H

H

H

I

s-Bu

nonafluoro-2-butyl

Br

CF3

15-1011

1,2-difluoro-2-propyl

H

H

F

H

H

H

I

s-Bu

nonafluoro-2-butyl

I

CF3

15-1020

2,2-dichloroethyl

H

Et

F

H

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

15-1050

2,2,2-trifluoroethyl

H

H

F

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

15-1163

2,2-dichloroethyl

H

Et

F

H

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

15-1193

2,2,2-trifluoroethyl

H

H

F

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

15-1306

2,2-dichloroethyl

H

Et

F

H

H

H

CF3

F

heptafluoroisopropyl

F

CF3

15-1336

2,2,2-trifluoroethyl

H

H

F

H

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

15-1449

2,2-dichloroethyl

H

Et

H

F

H

H

Cl

F

heptafluoroisopropyl

F

Cl

15-1479

2,2,2-trifluoroethyl

H

H

H

F

H

H

Cl

Me

nonafluoro-2-butyl

Me

I

15-1592

2,2-dichloroethyl

H

Et

H

F

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

15-1622

2,2,2-trifluoroethyl

H

H

H

F

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

15-1737

2,2,2-trichloroethyl

H

H

H

F

H

H

Cl

F

heptafluoroisopropyl

Br

CF3

15-1749

n-butyl

H

H

H

F

H

H

Cl

I

nonafluoro-2-butyl

Br

CF3

15-1766

2,2,2-trichloroethyl

H

H

H

F

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

15-1772

i-propyl

H

H

H

F

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

15-1773

1,2-difluoro-2-propyl

H

H

H

F

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

15-1779

2-chloroethyl

H

H

H

F

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

15-1780

2-bromoethyl

H

H

H

F

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

15-1786

2,2,2-trichloroethyl

H

H

H

F

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

15-1787

2,2,2-tribromoethyl

H

H

H

F

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

15-1793

1,2-difluoro-2-propyl

H

H

H

F

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

15-1794

1,3-difluoro-2-propyl

H

H

H

F

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

15-1800

i-butyl

H

H

H

F

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

15-1801

s-butyl

H

H

H

F

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

15-1807

2-fluoroethyl

H

H

H

F

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

15-1808

2-chloroethyl

H

H

H

F

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

15-1814

2,2,2-trifluoroethyl

H

H

H

F

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

15-1815

2,2,2-trichloroethyl

H

H

H

F

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

15-1821

i-propyl

Et

i-Pr

H

F

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

15-1822

1,2-difluoro-2-propyl

H

H

H

F

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

15-1828

2-iodoethyl

H

H

H

F

H

H

I

Br

heptafluoroisopropyl

Me

CF3

15-1829

2-cyanoethyl

H

H

H

F

H

H

I

Br

heptafluoroisopropyl

Et

CF3

15-1835

n-propyl

n-Pr

Me

H

F

H

H

I

I

heptafluoroisopropyl

Me

CF3

15-1836

3-fluoro-n-propyl

H

H

H

F

H

H

I

I

heptafluoroisopropyl

Et

CF3

15-1842

1,3-dichloro-2-propyl

H

H

H

F

H

H

I

Me

heptafluoroisopropyl

F

C2F5

15-1843

1-chloro-3-fluoro-2-propyl

H

H

H

F

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

15-1846

4,4,4-trifluoro-n-butyl

H

H

H

F

H

H

I

Et

nonafluoro-2-butyl

F

CF3

15-1847

i-butyl

H

H

H

F

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

15-1850

benzyl

H

H

H

F

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

15-1851

phenyl

H

H

H

F

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

15-1854

2-fluoroethyl

H

H

H

F

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

15-1855

2-chloroethyl

H

H

H

F

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

15-1858

2-cyanoethyl

H

H

H

F

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

15-1859

2,2-difluoroethyl

H

H

H

F

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

15-1862

2,2,2-trichloroethyl

H

H

H

F

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

15-1863

2,2,2-tribromoethyl

H

H

H

F

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

15-1866

3-chloro-n-propyl

i-Pr

n-Pr

H

F

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

15-1867

3-bromo-n-propyl

H

H

H

F

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

15-1878

2,2-dichloroethyl

H

Et

H

F

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

15-1908

2,2,2-trifluoroethyl

H

H

H

F

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

15-2021

2,2-dichloroethyl

H

Et

H

F

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

15-2051

2,2,2-trifluoroethyl

H

H

H

F

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

15-2164

2,2-dichloroethyl

H

Et

H

F

H

H

CF3

F

heptafluoroisopropyl

F

CF3

15-2194

2,2,2-trifluoroethyl

H

H

H

F

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

15-2307

2,2-dichloroethyl

H

Et

F

F

H

H

Cl

F

heptafluoroisopropyl

F

Cl

15-2337

2,2,2-trifluoroethyl

H

H

F

F

H

H

Cl

Me

nonafluoro-2-butyl

Me

I

15-2450

2,2-dichloroethyl

H

Et

F

F

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

15-2480

2,2,2-trifluoroethyl

H

H

F

F

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

15-2585

methyl

H

H

F

F

H

H

Cl

F

heptafluoroisopropyl

H

CF3

15-2591

2-cyanoethyl

Et

H

F

F

H

H

Cl

I

heptafluoroisopropyl

H

C2F5

15-2594

2,2,2-trifluoroethyl

H

H

F

F

H

H

Cl

F

heptafluoroisopropyl

Cl

CF3

15-2602

1,2-difluoro-2-propyl

H

H

F

F

H

H

Cl

Br

heptafluoroisopropyl

Cl

CF3

15-2609

i-butyl

H

H

F

F

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

15-2610

s-butyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

15-2611

vinyl

i-Pr

H

F

F

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

15-2612

benzyl

H

H

F

F

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

15-2623

2,2,2-trifluoroethyl

H

H

F

F

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

15-2624

2,2,2-trichloroethyl

H

H

F

F

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

15-2630

i-propyl

H

H

F

F

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

15-2631

1,2-difluoro-2-propyl

H

H

F

F

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

15-2637

2-chloroethyl

H

H

F

F

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

15-2638

2-bromoethyl

H

H

F

F

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

15-2644

2,2,2-trichloroethyl

H

H

F

F

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

15-2645

2,2,2-tribromoethyl

H

H

F

F

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

15-2651

1,2-difluoro-2-propyl

H

H

F

F

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

15-2652

1,3-difluoro-2-propyl

H

H

F

F

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

15-2658

i-butyl

H

H

F

F

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

15-2659

s-butyl

H

H

F

F

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

15-2665

2-fluoroethyl

H

H

F

F

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

15-2666

2-chloroethyl

H

H

F

F

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

15-2672

2,2,2-trifluoroethyl

H

H

F

F

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

15-2673

2,2,2-trichloroethyl

H

H

F

F

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

15-2679

i-propyl

Et

i-Pr

F

F

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

15-2680

1,2-difluoro-2-propyl

H

H

F

F

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

15-2686

2-iodoethyl

H

H

F

F

H

H

I

Br

heptafluoroisopropyl

Me

CF3

15-2687

2-cyanoethyl

H

H

F

F

H

H

I

Br

heptafluoroisopropyl

Et

CF3

15-2693

n-propyl

n-Pr

Me

F

F

H

H

I

I

heptafluoroisopropyl

Me

CF3

15-2694

3-fluoro-n-propyl

H

H

F

F

H

H

I

I

heptafluoroisopropyl

Et

CF3

15-2700

1,3-dichloro-2-propyl

H

H

F

F

H

H

I

Me

heptafluoroisopropyl

F

C2F5

15-2701

1-chloro-3-fluoro-2-propyl

H

H

F

F

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

15-2704

4,4,4-trifluoro-n-butyl

H

H

F

F

H

H

I

Et

nonafluoro-2-butyl

F

CF3

15-2705

i-butyl

H

H

F

F

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

15-2708

benzyl

H

H

F

F

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

15-2709

phenyl

H

H

F

F

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

15-2712

2-fluoroethyl

H

H

F

F

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

15-2713

2-chloroethyl

H

H

F

F

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

15-2716

2-cyanoethyl

H

H

F

F

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

15-2717

2,2-difluoroethyl

H

H

F

F

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

15-2720

2,2,2-trichloroethyl

H

H

F

F

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

15-2721

2,2,2-tribromoethyl

H

H

F

F

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

15-2724

3-chloro-n-propyl

i-Pr

n-Pr

F

F

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

15-2725

3-bromo-n-propyl

H

H

F

F

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

15-2736

2,2-dichloroethyl

H

Et

F

F

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

15-2766

2,2,2-trifluoroethyl

H

H

F

F

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

15-2879

2,2-dichloroethyl

H

Et

F

F

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

15-2909

2,2,2-trifluoroethyl

H

H

F

F

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

15-3022

2,2-dichloroethyl

H

Et

F

F

H

H

CF3

F

heptafluoroisopropyl

F

CF3

15-3052

2,2,2-trifluoroethyl

H

H

F

F

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

15-3157

2,2,2-trichloroethyl

H

H

F

F

F

H

Cl

F

pentafluoroethyl

H

Cl

15-3158

2,2,2-trichloroethyl

Me

H

F

F

F

H

Cl

H

heptafluoroisopropyl

F

Cl

15-3159

2,2,2-trichloroethyl

H

Me

F

F

F

H

Br

Cl

heptafluoroisopropyl

H

Br

15-3160

2,2,2-trichloroethyl

Me

Me

F

F

F

H

I

H

heptafluoroisopropyl

Cl

I

15-3161

2,2,2-trichloroethyl

H

H

F

F

F

H

Cl

Br

heptafluoroisopropyl

H

OCF3

15-3162

2,2,2-trichloroethyl

H

H

F

F

F

H

Br

H

heptafluoroisopropyl

Br

OCF3

15-3163

2,2,2-trichloroethyl

Et

H

F

F

F

H

I

I

heptafluoroisopropyl

H

OCF3

15-3164

2,2,2-trichloroethyl

H

H

F

F

F

H

Cl

H

heptafluoroisopropyl

I

CF3

15-3165

2,2,2-trichloroethyl

H

Et

F

F

F

H

Br

F

heptafluoroisopropyl

F

CF3

15-3166

2,2,2-trichloroethyl

H

H

F

F

F

H

I

F

heptafluoroisopropyl

Cl

CF3

15-3167

2,2,2-trichloroethyl

H

H

F

F

F

H

CF3

F

heptafluoroisopropyl

Br

CF3

15-3168

2,2,2-trichloroethyl

Et

Et

F

F

F

H

Cl

F

nonafluoro-2-butyl

I

Cl

15-3169

2,2,2-trichloroethyl

H

H

F

F

F

H

Br

Cl

nonafluoro-2-butyl

F

Br

15-3170

2,2,2-trichloroethyl

H

H

F

F

F

H

I

Cl

nonafluoro-2-butyl

Cl

I

15-3171

2,2,2-trichloroethyl

n-Pr

H

F

F

F

H

Cl

Cl

nonafluoro-2-butyl

Br

OCF3

15-3172

2,2,2-trichloroethyl

H

H

F

F

F

H

Br

Cl

nonafluoro-2-butyl

I

OCF3

15-3173

2,2,2-trichloroethyl

H

n-Pr

F

F

F

H

I

Br

nonafluoro-2-butyl

F

OCF3

15-3174

2,2,2-trichloroethyl

H

H

F

F

F

H

Cl

Br

nonafluoro-2-butyl

Cl

CF3

15-3175

2,2,2-trichloroethyl

H

H

F

F

F

H

Br

Br

nonafluoro-2-butyl

Br

CF3

15-3176

2,2,2-trichloroethyl

n-Pr

n-Pr

F

F

F

H

I

Br

nonafluoro-2-butyl

I

CF3

15-3177

2,2,2-trichloroethyl

H

H

F

F

F

H

CF3

I

nonafluoro-2-butyl

F

CF3

15-3178

2,2,2-trichloroethyl

H

H

H

H

F

H

Cl

I

pentafluoroethyl

Cl

Cl

15-3179

2,2,2-trichloroethyl

H

H

H

H

F

H

Cl

I

heptafluoroisopropyl

Br

Cl

15-3180

2,2,2-trichloroethyl

H

H

H

H

F

H

Br

I

heptafluoroisopropyl

I

Br

15-3181

2,2,2-trichloroethyl

H

H

H

H

F

H

I

Me

heptafluoroisopropyl

H

I

15-3182

2,2,2-trichloroethyl

H

H

H

H

F

H

Cl

H

heptafluoroisopropyl

Me

OCF3

15-3183

2,2,2-trichloroethyl

i-Pr

H

H

H

F

H

Br

Et

heptafluoroisopropyl

H

OCF3

15-3184

2,2,2-trichloroethyl

H

H

H

H

F

H

I

H

heptafluoroisopropyl

Et

OCF3

15-3185

2,2,2-trichloroethyl

H

H

H

H

F

H

Cl

n-Pr

heptafluoroisopropyl

H

CF3

15-3186

2,2,2-trichloroethyl

H

i-Pr

H

H

F

H

Br

H

heptafluoroisopropyl

n-Pr

CF3

15-3187

2,2,2-trichloroethyl

i-Pr

i-Pr

H

H

F

H

I

i-Pr

heptafluoroisopropyl

H

CF3

15-3188

2,2,2-trichloroethyl

H

H

H

H

F

H

CF3

H

heptafluoroisopropyl

i-Pr

CF3

15-3189

2,2,2-trichloroethyl

H

H

H

H

F

H

Cl

n-Bu

nonafluoro-2-butyl

H

Cl

15-3190

2,2,2-trichloroethyl

H

H

H

H

F

H

Br

H

nonafluoro-2-butyl

n-Bu

Br

15-3191

2,2,2-trichloroethyl

H

H

H

H

F

H

I

i-Bu

nonafluoro-2-butyl

H

I

15-3192

2,2,2-trichloroethyl

H

H

H

H

F

H

Cl

H

nonafluoro-2-butyl

i-Bu

OCF3

15-3193

2,2,2-trichloroethyl

H

H

H

H

F

H

Br

s-Bu

nonafluoro-2-butyl

H

OCF3

15-3194

2,2,2-trichloroethyl

H

H

H

H

F

H

I

H

nonafluoro-2-butyl

s-Bu

OCF3

15-3195

2,2,2-trichloroethyl

H

H

H

H

F

H

Cl

Me

nonafluoro-2-butyl

Me

CF3

15-3196

2,2,2-trichloroethyl

H

H

H

H

F

H

Br

Me

nonafluoro-2-butyl

Et

CF3

15-3197

2,2,2-trichloroethyl

C(O)Me

H

H

H

F

H

I

Me

nonafluoro-2-butyl

n-Pr

CF3

15-3198

2,2,2-trichloroethyl

H

H

H

H

F

H

CF3

Me

nonafluoro-2-butyl

i-Pr

CF3

15-3199

2,2,2-trichloroethyl

H

H

H

H

H

F

Cl

Me

pentafluoroethyl

n-Bu

Cl

15-3200

2,2,2-trichloroethyl

H

H

H

H

H

F

Br

Me

heptafluoroisopropyl

i-Bu

Br

15-3201

2,2,2-trichloroethyl

H

C(O)Me

H

H

H

F

Br

Me

heptafluoroisopropyl

s-Bu

OCF3

15-3202

2,2,2-trichloroethyl

H

H

H

H

H

F

I

Et

heptafluoroisopropyl

Me

CF3

15-3203

2,2,2-trichloroethyl

H

H

H

H

H

F

CF3

Et

heptafluoroisopropyl

Et

CF3

15-3204

2,2,2-trichloroethyl

C(O)Me

C(O)Me

H

H

H

F

I

Et

nonafluoro-2-butyl

n-Pr

I

15-3205

2,2,2-trichloroethyl

H

H

H

H

H

F

Cl

Et

nonafluoro-2-butyl

i-Pr

OCF3

15-3206

2,2,2-trichloroethyl

H

H

H

H

H

F

Br

Et

nonafluoro-2-butyl

n-Bu

CF3

15-3207

2,2,2-trichloroethyl

H

H

H

H

H

F

CF3

Et

nonafluoro-2-butyl

i-Bu

CF3

15-3208

2,2,2-trichloroethyl

H

H

F

H

F

H

Cl

Et

pentafluoroethyl

s-Bu

Cl

15-3209

2,2,2-trichloroethyl

H

H

F

H

F

H

Cl

n-Pr

heptafluoroisopropyl

Me

Cl

15-3210

2,2,2-trichloroethyl

H

H

F

H

F

H

Br

n-Pr

heptafluoroisopropyl

Et

Br

15-3211

2,2,2-trichloroethyl

Me

Et

F

H

F

H

I

n-Pr

heptafluoroisopropyl

n-Pr

I

15-3212

2,2,2-trichloroethyl

H

H

F

H

F

H

Cl

n-Pr

heptafluoroisopropyl

i-Pr

OCF3

15-3213

2,2,2-trichloroethyl

H

H

F

H

F

H

Br

n-Pr

heptafluoroisopropyl

n-Bu

OCF3

15-3214

2,2,2-trichloroethyl

H

H

F

H

F

H

I

n-Pr

heptafluoroisopropyl

i-Bu

OCF3

15-3215

2,2,2-trichloroethyl

H

H

F

H

F

H

Cl

n-Pr

heptafluoroisopropyl

s-Bu

CF3

15-3216

2,2,2-trichloroethyl

Me

n-Pr

F

H

F

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

15-3217

2,2,2-trichloroethyl

H

H

F

H

F

H

I

i-Pr

heptafluoroisopropyl

Et

CF3

15-3218

2,2,2-trichloroethyl

H

H

F

H

F

H

CF3

i-Pr

heptafluoroisopropyl

n-Pr

CF3

15-3219

2,2,2-trichloroethyl

H

H

F

H

F

H

Cl

i-Pr

nonafluoro-2-butyl

i-Pr

Cl

15-3220

2,2,2-trichloroethyl

H

H

F

H

F

H

Br

i-Pr

nonafluoro-2-butyl

n-Bu

Br

15-3221

2,2,2-trichloroethyl

H

H

F

H

F

H

I

i-Pr

nonafluoro-2-butyl

i-Bu

I

15-3222

2,2,2-trichloroethyl

Me

i-Pr

F

H

F

H

Cl

i-Pr

nonafluoro-2-butyl

s-Bu

OCF3

15-3223

2,2,2-trichloroethyl

H

H

F

H

F

H

Br

n-Bu

nonafluoro-2-butyl

Me

OCF3

15-3224

2,2,2-trichloroethyl

H

H

F

H

F

H

I

n-Bu

nonafluoro-2-butyl

Et

OCF3

15-3225

2,2,2-trichloroethyl

H

H

F

H

F

H

Br

n-Bu

nonafluoro-2-butyl

n-Pr

CF3

15-3226

2,2,2-trichloroethyl

H

H

F

H

F

H

I

n-Bu

nonafluoro-2-butyl

i-Pr

CF3

15-3227

2,2,2-trichloroethyl

H

H

F

H

F

H

CF3

n-Bu

nonafluoro-2-butyl

n-Bu

CF3

15-3228

2,2,2-trichloroethyl

H

H

F

H

H

F

Cl

n-Bu

pentafluoroethyl

i-Bu

Cl

15-3229

2,2,2-trichloroethyl

Me

C(O)Me

F

H

H

F

Br

n-Bu

heptafluoroisopropyl

s-Bu

Br

15-3230

2,2,2-trichloroethyl

H

H

F

H

H

F

Br

i-Bu

heptafluoroisopropyl

Me

OCF3

15-3231

2,2,2-trichloroethyl

H

H

F

H

H

F

I

i-Bu

heptafluoroisopropyl

Et

CF3

15-3232

2,2,2-trichloroethyl

H

H

F

H

H

F

CF3

i-Bu

heptafluoroisopropyl

n-Pr

CF3

15-3233

2,2,2-trichloroethyl

H

H

F

H

H

F

I

i-Bu

nonafluoro-2-butyl

i-Pr

I

15-3234

2,2,2-trichloroethyl

H

H

F

H

H

F

Cl

i-Bu

nonafluoro-2-butyl

n-Bu

OCF3

15-3235

2,2,2-trichloroethyl

H

H

F

H

H

F

Br

i-Bu

nonafluoro-2-butyl

i-Bu

CF3

15-3236

2,2,2-trichloroethyl

H

H

F

H

H

F

CF3

i-Bu

nonafluoro-2-butyl

s-Bu

CF3

15-3237

2,2,2-trichloroethyl

H

H

H

F

F

H

Cl

s-Bu

pentafluoroethyl

Me

Cl

15-3238

2,2,2-trichloroethyl

H

H

H

F

F

H

Br

s-Bu

heptafluoroisopropyl

Et

Br

15-3239

2,2,2-trichloroethyl

H

H

H

F

F

H

Br

s-Bu

heptafluoroisopropyl

n-Pr

OCF3

15-3240

2,2,2-trichloroethyl

H

H

H

F

F

H

I

s-Bu

heptafluoroisopropyl

i-Pr

CF3

15-3241

2,2,2-trichloroethyl

H

H

H

F

F

H

CF3

s-Bu

heptafluoroisopropyl

n-Bu

CF3

15-3242

2,2,2-trichloroethyl

H

H

H

F

F

H

I

s-Bu

nonafluoro-2-butyl

i-Bu

I

15-3243

2,2,2-trichloroethyl

Et

Me

H

F

F

H

Cl

s-Bu

nonafluoro-2-butyl

s-Bu

OCF3

15-3244

2,2,2-trichloroethyl

H

H

H

F

F

H

Br

F

nonafluoro-2-butyl

Me

CF3

15-3245

2,2,2-trichloroethyl

H

H

H

F

F

H

CF3

F

nonafluoro-2-butyl

Et

CF3

15-3246

2,2,2-trichloroethyl

H

H

H

F

H

F

Cl

F

pentafluoroethyl

n-Pr

Cl

15-3247

2,2,2-trichloroethyl

H

H

H

F

H

F

Br

F

heptafluoroisopropyl

i-Pr

Br

15-3248

2,2,2-trichloroethyl

H

H

H

F

H

F

Br

F

heptafluoroisopropyl

n-Bu

OCF3

15-3249

2,2,2-trichloroethyl

H

H

H

F

H

F

I

F

heptafluoroisopropyl

i-Bu

CF3

15-3250

2,2,2-trichloroethyl

Et

n-Pr

H

F

H

F

CF3

F

heptafluoroisopropyl

s-Bu

CF3

15-3251

2,2,2-trichloroethyl

Et

i-Pr

H

F

H

F

I

Cl

nonafluoro-2-butyl

Me

I

15-3252

2,2,2-trichloroethyl

H

H

H

F

H

F

Cl

Cl

nonafluoro-2-butyl

Et

OCF3

15-3253

2,2,2-trichloroethyl

H

H

H

F

H

F

Br

Cl

nonafluoro-2-butyl

n-Pr

CF3

15-3254

2,2,2-trichloroethyl

H

H

H

F

H

F

CF3

Cl

nonafluoro-2-butyl

i-Pr

CF3

15-3255

2,2,2-trichloroethyl

H

H

H

H

F

F

Cl

Cl

pentafluoroethyl

n-Bu

Cl

15-3256

2,2,2-trichloroethyl

Et

C(O)Me

H

H

F

F

Br

Cl

heptafluoroisopropyl

i-Bu

Br

15-3257

2,2,2-trichloroethyl

H

H

H

H

F

F

Br

Cl

heptafluoroisopropyl

s-Bu

OCF3

15-3258

2,2,2-trichloroethyl

H

H

H

H

F

F

I

Br

heptafluoroisopropyl

Me

CF3

15-3259

2,2,2-trichloroethyl

H

H

H

H

F

F

CF3

Br

heptafluoroisopropyl

Et

CF3

15-3260

2,2,2-trichloroethyl

H

H

H

H

F

F

I

Br

nonafluoro-2-butyl

n-Pr

I

15-3261

2,2,2-trichloroethyl

H

H

H

H

F

F

Cl

Br

nonafluoro-2-butyl

i-Pr

OCF3

15-3262

2,2,2-trichloroethyl

H

H

H

H

F

F

Br

Br

nonafluoro-2-butyl

n-Bu

CF3

15-3263

2,2,2-trichloroethyl

H

H

H

H

F

F

CF3

Br

nonafluoro-2-butyl

i-Bu

CF3

15-3264

2,2,2-trichloroethyl

H

H

F

F

H

F

Cl

Br

pentafluoroethyl

s-Bu

Cl

15-3265

2,2,2-trichloroethyl

n-Pr

Me

F

F

H

F

Br

I

heptafluoroisopropyl

Me

Br

15-3266

2,2,2-trichloroethyl

H

H

F

F

H

F

Br

I

heptafluoroisopropyl

Et

OCF3

15-3267

2,2,2-trichloroethyl

n-Pr

Et

F

F

H

F

I

I

heptafluoroisopropyl

n-Pr

CF3

15-3268

2,2,2-trichloroethyl

H

H

F

F

H

F

CF3

I

heptafluoroisopropyl

i-Pr

CF3

15-3269

2,2,2-trichloroethyl

H

H

F

F

H

F

I

I

nonafluoro-2-butyl

n-Bu

I

15-3270

2,2,2-trichloroethyl

H

H

F

F

H

F

Cl

I

nonafluoro-2-butyl

i-Bu

OCF3

15-3271

2,2,2-trichloroethyl

H

H

F

F

H

F

Br

I

nonafluoro-2-butyl

s-Bu

CF3

15-3272

2,2,2-trichloroethyl

H

H

F

F

H

F

CF3

Me

nonafluoro-2-butyl

F

CF3

15-3273

2,2,2-trichloroethyl

H

H

F

H

F

F

Cl

Me

pentafluoroethyl

Cl

Cl

15-3274

2,2,2-trichloroethyl

H

H

F

H

F

F

Br

Me

heptafluoroisopropyl

Br

Br

15-3275

2,2,2-trichloroethyl

H

H

F

H

F

F

Br

Me

heptafluoroisopropyl

I

OCF3

15-3276

2,2,2-trichloroethyl

H

H

F

H

F

F

I

Et

heptafluoroisopropyl

F

CF3

15-3277

2,2,2-trichloroethyl

H

H

F

H

F

F

CF3

Et

heptafluoroisopropyl

Cl

CF3

15-3278

2,2,2-trichloroethyl

H

H

F

H

F

F

I

Et

nonafluoro-2-butyl

Br

I

15-3279

2,2,2-trichloroethyl

n-Pr

i-Pr

F

H

F

F

Cl

Et

nonafluoro-2-butyl

I

OCF3

15-3280

2,2,2-trichloroethyl

H

H

F

H

F

F

Br

n-Pr

nonafluoro-2-butyl

F

CF3

15-3281

2,2,2-trichloroethyl

H

H

F

H

F

F

CF3

n-Pr

nonafluoro-2-butyl

Cl

CF3

15-3282

2,2,2-trichloroethyl

H

H

H

F

F

F

Cl

n-Pr

pentafluoroethyl

Br

Cl

15-3283

2,2,2-trichloroethyl

H

H

H

F

F

F

Br

n-Pr

heptafluoroisopropyl

I

Br

15-3284

2,2,2-trichloroethyl

H

H

H

F

F

F

Br

i-Pr

heptafluoroisopropyl

F

OCF3

15-3285

2,2,2-trichloroethyl

H

H

H

F

F

F

I

i-Pr

heptafluoroisopropyl

Cl

CF3

15-3286

2,2,2-trichloroethyl

n-Pr

C(O)Me

H

F

F

F

CF3

i-Pr

heptafluoroisopropyl

Br

CF3

15-3287

2,2,2-trichloroethyl

H

H

H

F

F

F

I

i-Pr

nonafluoro-2-butyl

I

I

15-3288

2,2,2-trichloroethyl

H

H

H

F

F

F

Cl

n-Bu

nonafluoro-2-butyl

F

OCF3

15-3289

2,2,2-trichloroethyl

H

H

H

F

F

F

Br

n-Bu

nonafluoro-2-butyl

Cl

CF3

15-3290

2,2,2-trichloroethyl

H

H

H

F

F

F

CF3

n-Bu

nonafluoro-2-butyl

Br

CF3

15-3291

2,2,2-trichloroethyl

i-Pr

Me

F

F

F

F

Cl

n-Bu

pentafluoroethyl

I

Cl

15-3292

2,2,2-trichloroethyl

H

H

F

F

F

F

Br

i-Bu

heptafluoroisopropyl

F

Br

15-3293

2,2,2-trichloroethyl

H

H

F

F

F

F

Br

i-Bu

heptafluoroisopropyl

Cl

OCF3

15-3294

2,2,2-trichloroethyl

H

H

F

F

F

F

I

i-Bu

heptafluoroisopropyl

Br

CF3

15-3295

2,2,2-trichloroethyl

i-Pr

Et

F

F

F

F

CF3

i-Bu

heptafluoroisopropyl

I

CF3

15-3296

2,2,2-trichloroethyl

i-Pr

n-Pr

F

F

F

F

I

s-Bu

nonafluoro-2-butyl

F

I

15-3297

2,2,2-trichloroethyl

H

H

F

F

F

F

Cl

s-Bu

nonafluoro-2-butyl

Cl

OCF3

15-3298

2,2,2-trichloroethyl

i-Pr

C(O)Me

F

F

F

F

Br

s-Bu

nonafluoro-2-butyl

Br

CF3

15-3299

2,2,2-trichloroethyl

H

H

F

F

F

F

CF3

s-Bu

nonafluoro-2-butyl

I

CF3

15-3308

2,2-dichloroethyl

H

Et

H

CN

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

15-3338

2,2,2-trifluoroethyl

H

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

15-3447

2-bromoethyl

H

H

H

CN

H

H

F

Br

heptafluoroisopropyl

H

CF3

15-3457

3-chloro-n-propyl

n-Pr

H

H

CN

H

H

Cl

Cl

heptafluoroisopropyl

Br

CF3

15-3464

3,3,3-trifluoro-n-propyl

H

H

H

CN

H

H

Cl

I

nonafluoro-2-butyl

Cl

CF3

15-3467

i-butyl

H

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

15-3468

s-butyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

15-3469

vinyl

i-Pr

H

H

CN

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

15-3470

benzyl

H

H

H

CN

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

15-3481

2,2,2-trifluoroethyl

H

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

15-3482

2,2,2-trichloroethyl

H

H

H

CN

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

15-3488

i-propyl

H

H

H

CN

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

15-3489

1,2-difluoro-2-propyl

H

H

H

CN

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

15-3495

2-chloroethyl

H

H

H

CN

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

15-3496

2-bromoethyl

H

H

H

CN

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

15-3502

2,2,2-trichloroethyl

H

H

H

CN

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

15-3503

2,2,2-tribromoethyl

H

H

H

CN

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

15-3509

1,2-difluoro-2-propyl

H

H

H

CN

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

15-3510

1,3-difluoro-2-propyl

H

H

H

CN

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

15-3516

i-butyl

H

H

H

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

15-3517

s-butyl

H

H

H

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

15-3523

2-fluoroethyl

H

H

H

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

15-3524

2-chloroethyl

H

H

H

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

15-3530

2,2,2-trifluoroethyl

H

H

H

CN

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

15-3531

2,2,2-trichloroethyl

H

H

H

CN

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

15-3537

i-propyl

Et

i-Pr

H

CN

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

15-3538

1,2-difluoro-2-propyl

H

H

H

CN

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

15-3544

2-iodoethyl

H

H

H

CN

H

H

I

Br

heptafluoroisopropyl

Me

CF3

15-3545

2-cyanoethyl

H

H

H

CN

H

H

I

Br

heptafluoroisopropyl

Et

CF3

15-3551

n-propyl

n-Pr

Me

H

CN

H

H

I

I

heptafluoroisopropyl

Me

CF3

15-3552

3-fluoro-n-propyl

H

H

H

CN

H

H

I

I

heptafluoroisopropyl

Et

CF3

15-3558

1,3-dichloro-2-propyl

H

H

H

CN

H

H

I

Me

heptafluoroisopropyl

F

C2F5

15-3559

1-chloro-3-fluoro-2-propyl

H

H

H

CN

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

15-3562

4,4,4-trifluoro-n-butyl

H

H

H

CN

H

H

I

Et

nonafluoro-2-butyl

F

CF3

15-3563

i-butyl

H

H

H

CN

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

15-3566

benzyl

H

H

H

CN

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

15-3567

phenyl

H

H

H

CN

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

15-3570

2-fluoroethyl

H

H

H

CN

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

15-3571

2-chloroethyl

H

H

H

CN

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

15-3574

2-cyanoethyl

H

H

H

CN

H

H

I

n-Bu

nonafluorc-2-butyl

F

CF3

15-3575

2,2-difluoroethyl

H

H

H

CN

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

15-3578

2,2,2-trichloroethyl

H

H

H

CN

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

15-3579

2,2,2-tribromoethyl

H

H

H

CN

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

15-3582

3-chloro-n-propyl

i-Pr

n-Pr

H

CN

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

15-3583

3-bromo-n-propyl

H

H

H

CN

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

15-3594

2,2-dichloroethyl

H

Et

H

CN

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

15-3624

2,2,2-trifluoroethyl

H

H

H

CN

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

15-3737

2,2-dichloroethyl

H

Et

H

CN

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

15-3767

2,2,2-trifluoroethyl

H

H

H

CN

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

15-3880

2,2-dichloroethyl

H

Et

H

CN

H

H

CF3

F

heptafluoroisopropyl

F

CF3

15-3910

2,2,2-trifluoroethyl

H

H

H

CN

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

15-4023

2,2-dichloroethyl

H

Et

F

CN

H

H

Cl

F

heptafluoroisopropyl

F

Cl

15-4053

2,2,2-trifluoroethyl

H

H

F

CN

H

H

Cl

Me

nonafluoro-2-butyl

Me

I

15-4166

2,2-dichloroethyl

H

Et

F

CN

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

15-4196

2,2,2-trifluoroethyl

H

H

F

CN

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

15-4304

2-chloroethyl

Me

Me

F

CN

H

H

Cl

H

heptafluoroisopropyl

Cl

CF3

15-4311

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

F

heptafluoroisopropyl

Br

CF3

15-4318

1,2-difluoro-2-propyl

H

H

F

CN

H

H

Cl

Br

heptafluoroisopropyl

Cl

CF3

15-4325

i-butyl

H

H

F

CN

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

15-4326

s-butyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

15-4327

vinyl

i-Pr

H

F

CN

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

15-4328

benzyl

H

H

F

CN

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

15-4339

2,2,2-trifluoroethyl

H

H

F

CN

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

15-4340

2,2,2-trichloroethyl

H

H

F

CN

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

15-4346

i-propyl

H

H

F

CN

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

15-4347

1,2-difluoro-2-propyl

H

H

F

CN

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

15-4353

2-chloroethyl

H

H

F

CN

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

15-4354

2-bromoethyl

H

H

F

CN

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

15-4360

2,2,2-trichloroethyl

H

H

F

CN

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

15-4361

2,2,2-tribromoethyl

H

H

F

CN

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

15-4367

1,2-difluoro-2-prooyl

H

H

F

CN

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

15-4368

1,3-difluoro-2-propyl

H

H

F

CN

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

15-4374

i-butyl

H

H

F

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

15-4375

s-butyl

H

H

F

CN

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

15-4381

2-fluoroethyl

H

H

F

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

15-4382

2-chloroethyl

H

H

F

CN

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

15-4388

2,2,2-trifluoroethyl

H

H

F

CN

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

15-4389

2,2,2-trichloroethyl

H

H

F

CN

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

15-4395

i-propyl

Et

i-Pr

F

CN

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

15-4396

1,2-difluoro-2-propyl

H

H

F

CN

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

15-4402

2-iodoethyl

H

H

F

CN

H

H

I

Br

heptafluoroisopropyl

Me

CF3

15-4403

2-cyanoethyl

H

H

F

CN

H

H

I

Br

heptafluoroisopropyl

Et

CF3

15-4409

n-propyl

n-Pr

Me

F

CN

H

H

I

I

heptafluoroisopropyl

Me

CF3

15-4410

3-fluoro-n-propyl

H

H

F

CN

H

H

I

I

heptafluoroisopropyl

Et

CF3

15-4416

1,3-dichloro-2-propyl

H

H

F

CN

H

H

I

Me

heptafluoroisopropyl

F

C2F5

15-4417

1-chloro-3-fluoro-2-propyl

H

H

F

CN

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

15-4420

4,4,4-trifluoro-n-butyl

H

H

F

CN

H

H

I

Et

nonafluoro-2-butyl

F

CF3

15-4421

i-butyl

H

H

F

CN

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

15-4424

benzyl

H

H

F

CN

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

15-4425

phenyl

H

H

F

CN

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

15-4428

2-fluoroethyl

H

H

F

CN

H

H

I

i-Pr

nonafluoro-2-butyl

F

I-C3F7

15-4429

2-chloroethyl

H

H

F

CN

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

15-4432

2-cyanoethyl

H

H

F

CN

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

15-4433

2,2-difluoroethyl

H

H

F

CN

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

15-4436

2,2,2-trichloroethyl

H

H

F

CN

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

15-4437

2,2,2-trichloroethyl

H

H

F

CN

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

15-4440

3-chloro-n-propyl

i-Pr

n-Pr

F

CN

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

15-4441

3-bromo-n-propyl

H

H

F

CN

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

15-4452

2,2-dichloroethyl

H

Et

F

CN

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

15-4482

2,2,2-trifluoroethyl

H

H

F

CN

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

15-4595

2,2-dichloroethyl

H

Et

F

CN

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

15-4625

2,2,2-trifluoroethyl

H

H

F

CN

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

15-4738

2,2-dichloroethyl

H

Et

F

CN

H

H

CF3

F

heptafluoroisopropyl

F

CF3

15-4768

2,2,2-trifluoroethyl

H

H

F

CN

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

15-4881

2,2-dichloroethyl

H

Et

F

CN

F

H

Cl

F

heptafluoroisopropyl

F

Cl

15-4911

2,2,2-trifluoroethyl

H

H

F

CN

F

H

Cl

Me

nonafluoro-2-butyl

Me

I

15-5024

2,2-dichloroethyl

H

Et

F

CN

F

H

Cl

F

heptafluoroisopropyl

F

OCF3

15-5054

2,2,2-trifluoroethyl

H

H

F

CN

F

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

15-5163

2-bromoethyl

H

H

F

CN

F

H

F

Br

heptafluoroisopropyl

H

CF3

15-5168

2,2,2-trifluoroethyl

H

H

F

CN

F

H

Cl

F

heptafluoroisopropyl

Cl

CF3

15-5180

3,3.3-trifluoro-n-propyl

H

H

F

CN

F

H

Cl

I

nonafluoro-2-butyl

Cl

CF3

15-5183

i-butyl

H

H

F

CN

F

H

Cl

Me

nonafluoro-2-butyl

H

CF3

15-5184

s-butyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

Me

CF3

15-5185

vinyl

i-Pr

H

F

CN

F

H

Cl

Et

nonafluoro-2-butyl

H

CF3

15-5186

benzyl

H

H

F

CN

F

H

Cl

H

nonafluoro-2-butyl

Et

CF3

15-5197

2,2,2-trifluoroethyl

H

H

F

CN

F

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

15-5198

2,2,2-trichloroethyl

H

H

F

CN

F

H

Cl

Me

nonafluoro-2-butyl

Et

I-C3F7

15-5204

i-propyl

H

H

F

CN

F

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

15-5205

1,2-difluoro-2-propyl

H

H

F

CN

F

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

15-5211

2-chloroethyl

H

H

F

CN

F

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

15-5212

2-bromoethyl

H

H

F

CN

F

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

15-5218

2,2,2-trichloroethyl

H

H

F

CN

F

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

15-5219

2,2,2-tribromoethyl

H

H

F

CN

F

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

15-5225

1,2-difluoro-2-propyl

H

H

F

CN

F

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

15-5226

1,3-difluoro-2-propyl

H

H

F

CN

F

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

15-5232

i-butyl

H

H

F

CN

F

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

15-5233

s-butyl

H

H

F

CN

F

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

15-5239

2-fluomethyl

H

H

F

CN

F

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

15-5240

2-chloroethyl

H

H

F

CN

F

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

15-5246

2,2,2-trifluoroethyl

H

H

F

CN

F

H

Br

F

nonafluoro-2-butyl

Me

CF3

15-5247

2,2,2-trichloroethyl

H

H

F

CN

F

H

Br

F

nonafluoro-2-butyl

Et

CF3

15-5253

i-propyl

Et

i-Pr

F

CN

F

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

15-5254

1,2-difluoro-2-propyl

H

H

F

CN

F

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

15-5260

2-iodoethyl

H

H

F

CN

F

H

I

Br

heptafluoroisopropyl

Me

CF3

15-5261

2-cyanoethyl

H

H

F

CN

F

H

I

Br

heptafluoroisopropyl

Et

CF3

15-5267

n-propyl

n-Pr

Me

F

CN

F

H

I

I

heptafluoroisopropyl

Me

CF3

15-5268

3-fluoro-n-propyl

H

H

F

CN

F

H

I

I

heptafluoroisopropyl

Et

CF3

15-5274

1,3-dichloro-2-propyl

H

H

F

CN

F

H

I

Me

heptafluoroisopropyl

F

C2F5

15-5275

1-chloro-3-fluoro-2-propyl

H

H

F

CN

F

H

I

Me

nonafluoro-2-butyl

Cl

CF3

15-5278

4,4,4-trifluoro-n-butyl

H

H

F

CN

F

H

I

Et

nonafluoro-2-butyl

F

CF3

15-5279

i-butyl

H

H

F

CN

F

H

I

Et

nonafluoro-2-butyl

Cl

CF3

15-5282

benzyl

H

H

F

CN

F

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

15-5283

phenyl

H

H

F

CN

F

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

15-5286

2-fluoroethyl

H

H

F

CN

F

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

15-5287

2-chloroethyl

H

H

F

CN

F

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

15-5290

2-cyanoethyl

H

H

F

CN

F

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

15-5291

2,2-difluoroethyl

H

H

F

CN

F

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

15-5294

2,2,2-trichloroethyl

H

H

F

CN

F

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

15-5295

2,2,2-tribromoethyl

H

H

F

CN

F

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

15-5298

3-chloro-n-propyl

i-Pr

n-Pr

F

CN

F

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

15-5299

3-bromo-n-propyl

H

H

F

CN

F

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

15-5310

2,2-dichloroethyl

H

Et

F

CN

F

H

OCF3

F

heptafluoroisopropyl

F

OCF3

15-5340

2,2,2-trifluoroethyl

H

H

F

CN

F

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

15-5453

2,2-dichloroethyl

H

Et

F

CN

F

H

OCF3

F

heptafluoroisopropyl

F

CF3

15-5483

2,2,2-trifluoroethyl

H

H

F

CN

F

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

15-5596

2,2-dichloroethyl

H

Et

F

CN

F

H

CF3

F

heptafluoroisopropyl

F

CF3

15-5626

2,2,2-trifluoroethyl

H

H

F

CN

F

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

TABLE 16

compound

number

Q1

R1

R2

A

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

16-1

phenyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

F

16-2

3-cyanophenyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

F

16-3

4-cyanophenyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

F

16-4

2-chloropyridin-3-yl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

F

16-5

phenyl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

16-6

3-cyanophenyl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

16-7

4-cyanophenyl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

16-8

2-chloropyridin-3-yl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

16-9

phenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

16-13

2-chlorophenyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

Cl

16-17

3-bromophenyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

Br

16-20

3-iodophenyl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

Cl

16-22

(2-trifluoromethyl)phenyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

I

16-25

2-nitrophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Br

16-28

2-cyanophenyl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

Cl

16-29

3-cyanophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

16-30

4-cyanophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

16-31

2,6-difluorophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

I

16-43

pyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

I

16-44

2-fluoropyridin-3-yl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

Cl

16-45

2-chloropyridin-3-yl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

16-63

5-nitropyridin-3-yl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

Cl

16-64

5-cyanopyridin-3-yl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

16-66

4-chloropyridin-3-yl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

16-86

4-cyanopyridin-2-yl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

Cl

16-87

phenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

16-107

3-cyanophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

16-108

4-cyanophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

16-123

2-chloropyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

16-165

phenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-166

2-fluorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-177

4-iodophenyl

H

H

N

H

H

H

Br

H

pentafluoroethyl

H

Br

16-185

3-cyanophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-186

4-cyanophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-200

2-fluoropyridin-3-yl

H

H

N

H

H

H

Br

H

pentafluoroethyl

H

Br

16-201

2-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-219

5-nitropyridin-3-yl

H

H

N

H

H

H

Br

H

pentafluoroethyl

H

Br

16-220

5-cyanopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-221

4-fluoropyridin-3-yl

H

H

N

H

H

H

Br

H

pentafluoroethyl

H

Br

16-242

4-cyanopyridin-2-yl

H

H

N

H

H

H

Br

H

pentafluoroethyl

H

Br

16-243

phenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

16-244

2-fluorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

16-263

3-cyanophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

16-264

4-cyanophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

16-279

2-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

16-321

phenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

I

16-328

2-bromophenyl

H

H

N

H

H

H

I

H

pentafluoroethyl

H

I

16-341

3-cyanophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

I

16-342

4-cyanophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

I

16-356

2-fluoropyridin-3-yl

H

H

N

H

H

H

I

H

pentafluoroethyl

H

I

16-357

2-chloropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

I

16-375

5-nitropyridin-3-yl

H

H

N

H

H

H

I

H

pentafluoroethyl

H

I

16-399

phenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

16-400

2-fluorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

16-419

3-cyanophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

16-420

4-cyanophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

16-435

2-chloropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

16-477

phenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

16-478

2-fluorophenyl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

OCF3

16-492

(4-trifluoromethyl)phenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OC2F5

16-493

2-nitrophenyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

16-496

2-cyanophenyl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

OC2F5

16-497

3-cyanophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

16-498

4-cyanophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

16-504

4-bromo-2-chlorophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OC2F5

16-512

2-fluoropyridin-3-yl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

OCF3

16-513

2-chloropyridin-3-yl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

16-555

phenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

16-565

2-iodophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

16-571

2-nitrophenyl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

16-572

3-nitrophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

16-573

4-nitrophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

16-581

2-chloro-4,5-difluorophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OC2F5

16-591

2-chloropyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

16-597

6-fluoropyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OC2F5

16-633

phenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

16-646

(2-trifluoromethyl)phenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

16-653

3-cyanophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

16-654

4-cyanophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

16-669

2-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

16-676

6-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

16-711

phenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

16-731

3-cyanophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

16-732

4-cyanophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

16-745

pyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

16-747

2-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

16-789

phenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

16-794

3-chlorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

16-809

3-cyanophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

16-810

4-cyanophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

16-825

2-chloropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

16-867

phenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

16-887

3-cyanophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

16-888

4-cyanophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

16-903

2-chloropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

16-945

phenyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

CF3

16-946

phenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

16-947

2-fluorophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

16-958

4-iodophenyl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

16-965

2-cyanophenyl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

C2F5

16-966

3-cyanophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

16-967

4-cyanophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

16-970

2,4-dichlorophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

16-974

2-bromo-4-chlorophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

16-981

2-fluoropyridin-3-yl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

16-982

2-chloropyridin-3-yl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

16-995

5-fluoropyridin-3-yl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

16-997

5-bromopyridin-3-yl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

16-998

5-iodopyridin-3-yl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

16-1000

5-nitropyridin-3-yl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

16-1002

4-fluoropyridin-3-yl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

16-1004

4-bromopyridin-3-yl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

16-1023

4-cyanopyridin-2-yl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

16-1024

phenyl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

16-1025

phenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

16-1038

(2-trifluoromethyl)phenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

16-1045

3-cyanophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

16-1046

4-cyanophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

16-1055

2-chloro-4-nitrophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

16-1061

2-chloropyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

16-1074

5-fluoropyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

16-1076

5-bromopyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

16-1077

5-iodopyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

16-1081

4-fluoropyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

16-1085

4-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

16-1086

4-nitropyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

16-1102

4-cyanopyridin-2-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

16-1103

phenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1104

2-fluorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1105

3-fluorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1106

4-fluorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1107

2-chlorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1108

3-chlorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1109

4-chlorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1110

2-bromophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1111

3-bromophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1112

4-bromophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1113

2-iodophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1114

3-iodophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1115

4-iodophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1116

(2-trifluoromethyl)phenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1117

(3-trifluoromethyl)phenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1118

(4-trifluoromethyl)phenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1119

2-nitrophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1120

3-nitrophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1121

4-nitrophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1122

2-cyanophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1123

3-cyanophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1124

4-cyanophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1125

2,6-difluorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1126

3,4-dichlorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1127

2,4-dichlorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1128

2-chloro-4-fluorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1129

2-chloro-4,5-difluorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1130

4-bromo-2-chlorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1131

2-bromo-4-chlorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1132

2-bromo-4-fluorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1133

2-chloro-4-nitrophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1134

3,5-dicyanophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1135

4-cyano-2-fluorophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1136

2-chloro-4-cyanophenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1137

pyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1138

2-fluoropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1139

2-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1140

2-bromopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1141

2-iodopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1142

2-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1143

2-nitropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1144

2-cyanopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1145

6-fluoropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1146

6-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1147

6-bromopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1148

6-iodopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1149

6-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1150

6-nitropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1151

6-cyanopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1152

5-fluoropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1153

5-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1154

5-bromopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1155

5-iodopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1156

5-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1157

5-nitropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1158

5-cyanopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1159

4-fluoropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1160

4-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1161

4-bromopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1162

4-iodopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1163

4-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1164

4-nitropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1165

4-cyanopyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1166

2,6-dichloropyridin-3-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1167

pyridin-3-yl N-oxide

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1168

pyridin-4-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1169

2-chloropyridin-4-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1170

3-bromopyridin-4-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1171

3,5-dichloropyridin-4-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1172

3-(trifluoromethyl)pyridin-4-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1173

2,6-dicyanopyridin-4-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1174

pyridin-4-yl N-oxide

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1175

pyridin-2-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1176

3-chloropyridin-2-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1177

4-bromopyridin-2-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1178

5-iodopyridin-2-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1179

6-chloropyridin-2-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1180

4-cyanopyridin-2-yl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-1181

phenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1182

2-fluorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1183

3-fluorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1184

4-fluorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1185

2-chlorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1186

3-chlorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1187

4-chlorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1188

2-bromophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1189

3-bromophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1190

4-bromophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1191

2-iodophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1192

3-iodophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1193

4-iodophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1194

(2-trifluoromethyl)phenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1195

(3-trifluoromethyl)phenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1196

(4-trifluoromethyl)phenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1197

2-nitrophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1198

3-nitrophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1199

4-nitrophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1200

2-cyanophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1201

3-cyanophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1202

4-cyanophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1203

2,6-difluorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1204

3,4-dichlorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1205

2,4-dichlorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1206

2-chloro-4-fluorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1207

2-chloro-4,5-difluorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1208

4-bromo-2-chlorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1209

2-bromo-4-chlorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1210

2-bromo-4-fluorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1211

2-chloro-4-nitrophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1212

3,5-dicyanophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1213

4-cyano-2-fluorophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1214

2-chloro-4-cyanophenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1215

pyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1216

2-fluoropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1217

2-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1218

2-bromopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1219

2-iodopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1220

2-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1221

2-nitropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1222

2-cyanopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1223

6-fluoropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1224

6-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1225

6-bromopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1226

6-iodopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1227

6-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1228

6-nitropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1229

6-cyanopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1230

5-fluoropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1231

5-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1232

5-bromopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1233

5-iodopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1234

5-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1235

5-nitropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1236

5-cyanopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1237

4-fluoropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1238

4-chloropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1239

4-bromopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1240

4-iodopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1241

4-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1242

4-nitropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1243

4-cyanopyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1244

2,6-dichloropyridin-3-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1245

pyridin-3-yl N-oxide

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1246

pyridin-4-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1247

2-chloropyridin-4-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1248

3-bromopyridin-4-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1249

3,5-dichloropyridin-4-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1250

3-(trifluoromethyl)pyridin-4-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1251

2,6-dicyanopyridin-4-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1252

pyridin-4-yl N-oxide

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1253

pyridin-2-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1254

3-chloropyridin-2-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1255

4-bromopyridin-2-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1256

5-iodopyridin-2-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1257

6-chloropyridin-2-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1258

4-cyanopyridin-2-yl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-1259

phenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1260

2-fluorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1261

3-fluorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1262

4-fluorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1263

2-chlorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1264

3-chlorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1265

4-chlorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1266

2-bromophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1267

3-bromophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1268

4-bromophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1269

2-iodophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1270

3-iodophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1271

4-iodophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1272

(2-trifluoromethyl)phenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1273

(3-trifluoromethyl)phenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1274

(4-trifluoromethyl)phenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1275

2-nitrophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1276

3-nitrophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1277

4-nitrophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1278

2-cyanophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1279

3-cyanophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1280

4-cyanophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1281

2,6-difluorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1282

3,4-dichlorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1283

2,4-dichlorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1284

2-chloro-4-fluorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1285

2-chloro-4,5-difluorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1286

4-bromo-2-chlorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1287

2-bromo-4-chlorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1288

2-bromo-4-fluorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1289

2-chloro-4-nitrophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1290

3,5-dicyanophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1291

4-cyano-2-fluorophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1292

2-chloro-4-cyanophenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1293

pyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1294

2-fluoropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1295

2-chloropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1296

2-bromopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1297

2-iodopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1298

2-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1299

2-nitropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1300

2-cyanopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1301

6-fluoropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1302

6-chloropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1303

6-bromopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1304

6-iodopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1305

6-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1306

6-nitropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1307

6-cyanopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1308

5-fluoropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1309

5-chloropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1310

5-bromopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1311

5-iodopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1312

5-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1313

5-nitropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1314

5-cyanopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1315

4-fluoropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1316

4-chloropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1317

4-bromopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1318

4-iodopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1319

4-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1320

4-nitropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1321

4-cyanopyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1322

2,6-dichloropyridin-3-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1323

pyridin-3-yl N-oxide

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1324

pyridin-4-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1325

2-chloropyridin-4-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1326

3-bromopyridin-4-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1327

3,5-dichloropyridin-4-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1328

3-(trifluoromethyl)pyridin-4-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1329

2,6-dicyanopyridin-4-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1330

pyridin-4-yl N-oxide

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1331

pyridin-2-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1332

3-chloropyridin-2-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1333

4-bromopyridin-2-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1334

5-iodopyridin-2-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1335

6-chloropyridin-2-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1336

4-cyanopyridin-2-yl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-1337

phenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1338

2-fluorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1339

3-fluorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1340

4-fluorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1341

2-chlorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1342

3-chlorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1343

4-chlorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1344

2-bromophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1345

3-bromophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1346

4-bromophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1347

2-iodophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1348

3-iodophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1349

4-iodophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1350

(2-trifluoromethyl)phenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1351

(3-trifluoromethyl)phenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1352

(4-trifluoromethyl)phenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1353

2-nitrophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1354

3-nitrophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1355

4-nitrophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1356

2-cyanophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1357

3-cyanophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1358

4-cyanophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1359

2,6-difluorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1360

3,4-dichlorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1361

2,4-dichlorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1362

2-chloro-4-fluorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1363

2-chloro-4,5-difluorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1364

4-bromo-2-chlorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1365

2-bromo-4-chlorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1366

2-bromo-4-fluorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1367

2-chloro-4-nitrophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1368

3,5-dicyanophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1369

4-cyano-2-fluorophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1370

2-chloro-4-cyanophenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1371

pyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1372

2-fluoropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1373

2-chloropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1374

2-bromopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1375

2-iodopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1376

2-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1377

2-nitropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1378

2-cyanopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1379

6-fluoropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1380

6-chloropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1381

6-bromopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1382

6-iodopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1383

6-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1384

6-nitropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1385

6-cyanopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1386

5-fluoropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1387

5-chloropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1388

5-bromopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1389

5-iodopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1390

5-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1391

5-nitropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1392

5-cyanopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1393

4-fluoropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1394

4-chloropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1395

4-bromopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1396

4-iodopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1397

4-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1398

4-nitropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1399

4-cyanopyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1400

2,6-dichloropyridin-3-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1401

pyridin-3-yl N-oxide

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1402

pyridin-4-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1403

2-chloropyridin-4-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1404

3-bromopyridin-4-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1405

3,5-dichloropyridin-4-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1406

3-(trifluoromethyl)pyridin-4-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1407

2,6-dichloropyridin-4-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1408

pyridin-4-yl N-oxide

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1409

pyridin-2-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1410

3-chloropyridin-2-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1411

4-bromopyridin-2-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1412

5-iodopyridin-2-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1413

6-chloropyridin-2-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1414

4-cyanopyridin-2-yl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-1415

phenyl

H

H

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

16-1422

2-bromophenyl

H

H

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OC2F5

16-1427

4-iodophenyl

H

H

N

H

H

H

OCF3

H

pentafluoroethyl

H

OCF3

16-1430

3-cyanophenyl

H

H

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

16-1431

4-cyanophenyl

H

H

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

16-1436

2-chloro-4,5-difluorophenyl

H

H

N

H

H

H

OC2F5

H

heptafluoroisopropyl

H

OC2F5

16-1439

2-bromo-4-fluorophenyl

H

H

N

H

H

H

OC2F5

H

heptafluoroisopropyl

H

OCF3

16-1445

2-fluoropyridin-3-yl

H

H

N

H

H

H

OCF3

H

pentafluoroethyl

H

OCF3

16-1446

2-chloropyridin-3-yl

H

H

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

16-1471

phenyl

H

H

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

16-1478

2-bromophenyl

H

H

N

H

H

H

OC2F5

H

nonafluoro-2-butyl

H

OCF3

16-1484

(2-trifluoromethyl)phenyl

H

H

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OC2F5

16-1486

3-cyanophenyl

H

H

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

16-1487

4-cyanophenyl

H

H

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

16-1493

4-bromo-2-chlorophenyl

H

H

N

H

H

H

OC2F5

H

nonafluoro-2-butyl

H

OC2F5

16-1502

2-chloropyridin-3-yl

H

H

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

16-1527

phenyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

16-1534

2-bromophenyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OC2F5

16-1539

4-iodophenyl

H

H

N

H

H

H

CF3

H

pentafluoroethyl

H

OCF3

16-1540

(2-trifluoromethyl)phenyl

H

H

N

H

H

H

C2F5

H

heptafluoroisopropyl

H

OC2F5

16-1542

3-cyanophenyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

16-1543

4-cyanophenyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

16-1550

2-bromo-4-chlorophenyl

H

H

N

H

H

H

n-C3F7

H

heptafluoroisopropyl

H

OCF3

16-1554

4-cyano-2-fluorophenyl

H

H

N

H

H

H

i-C3F7

H

heptafluoroisopropyl

H

OCF3

16-1558

2-chloropyridin-3-yl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

16-1564

6-chloropyridin-3-yl

H

H

N

H

H

H

n-C3F7

H

heptafluoroisopropyl

H

OC2F5

16-1567

5-cyanopyridin-3-yl

H

H

N

H

H

H

i-C3F7

H

heptafluoroisopropyl

H

OC2F5

16-1568

4-chloropyridin-3-yl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

16-1583

phenyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-1594

3-iodophenyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OC2F5

16-1597

3-nitrophenyl

H

H

N

H

H

H

C2F5

H

nonafluoro-2-butyl

H

OCF3

16-1598

3-cyanophenyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-1599

4-cyanophenyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-1605

4-bromo-2-chlorophenyl

H

H

N

H

H

H

i-C3F7

H

nonafluoro-2-butyl

H

OCF3

16-1608

2-chloro-4-nitrophenyl

H

H

N

H

H

H

n-C3F7

H

nonafluoro-2-butyl

H

OCF3

16-1614

2-chloropyridin-3-yl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-1615

2-bromopyridin-3-yl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-1616

2-iodopyridin-3-yl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-1617

2-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-1618

2-nitropyridin-3-yl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-1619

2-cyanopyridin-3-yl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-1620

6-chloropyridin-3-yl

H

H

N

H

H

H

C2F5

H

nonafluoro-2-butyl

H

OC2F5

16-1625

4-cyanopyridin-3-yl

H

H

N

H

H

H

n-C3F7

H

nonafluoro-2-butyl

H

OC2F5

16-1636

5-iodopyridin-2-yl

H

H

N

H

H

H

i-C3F7

H

nonafluoro-2-butyl

H

OC2F5

16-1639

phenyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-1640

2-fluorophenyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-1651

4-iodophenyl

H

H

N

H

H

H

CF3

H

pentafluoroethyl

H

CF3

16-1653

(3-trifluoromethyl)phenyl

H

H

N

H

H

H

C2F5

H

heptafluoroisopropyl

H

CF3

16-1658

2-cyanophenyl

H

H

N

H

H

H

CF3

H

pentafluoroethyl

H

CF3

16-1659

3-cyanophenyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-1660

4-cyanophenyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-1666

4-bromo-2-chlorophenyl

H

H

N

H

H

H

n-C3F7

H

heptafluoroisopropyl

H

CF3

16-1671

4-cyano-2-fluorophenyl

H

H

N

H

H

H

i-C3F7

H

heptafluoroisopropyl

H

CF3

16-1675

2-chloropyridin-3-yl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-1676

2-bromopyridin-3-yl

H

H

N

H

H

H

C2F5

H

heptafluoroisopropyl

H

C2F5

16-1677

2-iodopyridin-3-yl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-1678

2-(trifluoromethyl)pyridin-3-yl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-1679

2-nitropyridin-3-yl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-1680

2-cyanopyridin-3-yl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-1681

6-fluoropyridin-3-yl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-1682

6-chloropyridin-3-yl

H

H

N

H

H

H

C2F5

H

heptafluoroisopropyl

H

n-C3F7

16-1691

4-cyanopyridin-3-yl

H

H

N

H

H

H

C2F5

H

heptafluoroisopropyl

H

i-C3F7

16-1707

phenyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

16-1708

2-fluorophenyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

16-1719

4-iodophenyl

H

H

N

H

H

H

C2F5

H

nonafluoro-2-butyl

H

CF3

16-1727

3-cyanophenyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

16-1728

4-cyanophenyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

16-1734

4-bromo-2-chlorophenyl

H

H

N

H

H

H

n-C3F7

H

nonafluoro-2-butyl

H

CF3

16-1739

4-cyano-2-fluorophenyl

H

H

N

H

H

H

i-C3F7

H

nonafluoro-2-butyl

H

CF3

16-1743

2-chloropyridin-3-yl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

16-1744

2-bromopyridin-3-yl

H

H

N

H

H

H

C2F5

H

nonafluoro-2-butyl

H

C2F5

16-1755

6-cyanopyridin-3-yl

H

H

N

H

H

H

C2F5

H

nonafluoro-2-butyl

H

n-C3F7

16-1759

4-cyanopyridin-3-yl

H

H

N

H

H

H

C2F5

H

nonafluoro-2-butyl

H

i-C3F7

16-1775

phenyl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

16-1776

3-cyanophenyl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

16-1777

4-cyanophenyl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

16-1778

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

16-1779

phenyl

H

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

16-1780

3-cyanophenyl

H

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

16-1781

4-cyanophenyl

H

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

16-1782

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

16-1783

phenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

16-1787

2-chlorophenyl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

Cl

16-1791

3-bromophenyl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

Br

16-1795

4-iodophenyl

H

H

N-oxide

H

H

H

Cl

H

pentafluoroethyl

H

Cl

16-1796

(2-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

I

16-1799

2-nitrophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Br

16-1803

3-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

16-1804

4-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

16-1805

2,6-difluorophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

I

16-1817

pyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

I

16-1818

2-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

pentafluoroethyl

H

Cl

16-1819

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

16-1861

phenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

16-1881

3-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

16-1882

4-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

16-1897

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

16-1939

phenyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-1951

4-iodophenyl

H

H

N-oxide

H

H

H

Br

H

pentafluoroethyl

H

Br

16-1959

3-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-1960

4-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-1973

pyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-1975

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-1982

6-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

16-2017

phenyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

16-2037

3-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

16-2038

4-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

16-2053

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

16-2095

phenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

16-2107

4-iodophenyl

H

H

N-oxide

H

H

H

I

H

pentafluoroethyl

H

I

16-2115

3-cyanophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

16-2116

4-cyanophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

16-2131

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

16-2160

pyridin-4-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

16-2173

phenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

16-2193

3-cyanophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

16-2194

4-cyanophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

16-2209

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

16-2251

phenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

16-2263

4-iodophenyl

H

H

N-oxide

H

H

H

Cl

H

pentafluoroethyl

H

OCF3

16-2266

(4-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OC2F5

16-2267

2-nitrophenyl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

16-2270

2-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

pentafluoroethyl

H

OC2F5

16-2271

3-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

16-2272

4-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

16-2287

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

16-2329

phenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

16-2345

2-nitrophenyl

H

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

16-2349

3-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

16-2350

4-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

16-2365

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

16-2407

phenyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

16-2427

3-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

16-2428

4-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

16-2444

2-bromopyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

16-2485

phenyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

16-2505

3-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

16-2506

4-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

16-2521

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

16-2563

phenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

16-2583

3-cyanophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

16-2584

4-cyanophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

16-2599

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

16-2641

phenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

16-2661

3-cyanophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

16-2662

4-cyanophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

16-2677

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

16-2719

phenyl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

CF3

16-2720

phenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

16-2721

2-fluorophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

16-2732

4-iodophenyl

H

H

N-oxide

H

H

H

Cl

H

pentafluoroethyl

H

CF3

16-2739

2-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

pentafluoroethyl

H

C2F5

16-2740

3-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

16-2741

4-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

16-2744

2,4-dichlorophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

16-2745

2-chloro-4-fluorophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

16-2748

2-bromo-4-chlorophenyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

16-2756

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

16-2769

5-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

16-2771

5-bromopyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

16-2772

5-iodopyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

16-2774

5-nitropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

pentafluoroethyl

H

CF3

16-2776

4-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

pentafluoroethyl

H

CF3

16-2778

4-bromopyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

16-2779

4-iodopyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

16-2796

6-chloropyridin-2-yl

H

H

N-oxide

H

H

H

Cl

H

pentafluoroethyl

H

CF3

16-2798

phenyl

H

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

16-2799

phenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

16-2811

4-iodophenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

16-2812

(2-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

16-2819

3-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

16-2820

4-cyanophenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

16-2829

2-chloro-4-nitrophenyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

16-2835

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

16-2848

5-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

16-2850

5-bromopyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

16-2851

5-iodopyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

16-2855

4-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

16-2859

4-(trifluoromethyl)pyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

16-2860

4-nitropyridin-3-yl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

16-2877

phenyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-2878

2-fluorophenyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-2897

3-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-2898

4-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-2913

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-2920

6-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-2942

pyridin-4-yl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

16-2955

phenyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-2963

3-bromophenyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-2969

(3-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-2975

3-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-2976

4-cyanophenyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-2991

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-2998

6-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-3005

5-chloropyridin-3-yl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-3020

pyridin-4-yl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

16-3033

phenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3034

2-fluorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3035

3-fluorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3036

4-fluorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3037

2-chlorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3038

3-chlorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3039

4-chlorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3040

2-bromophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3041

3-bromophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3042

4-bromophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3043

2-iodophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3044

3-iodophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3045

4-iodophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3046

(2-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3047

(3-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3048

(4-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3049

2-nitrophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3050

3-nitrophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3051

4-nitrophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3052

2-cyanophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3053

3-cyanophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3054

4-cyanophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3055

2,6-difluorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3056

3,4-dichlorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3057

2,4-dichlorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3058

2-chloro-4-fluorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3059

2-chloro-4,5-difluorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3060

4-bromo-2-chlorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3061

2-bromo-4-chlorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3062

2-bromo-4-fluorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3063

2-chloro-4-nitrophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3064

3,5-dicyanophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3065

4-cyano-2-fluorophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3066

2-chloro-4-cyanophenyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3067

pyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3068

2-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3069

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3070

2-bromopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3071

2-iodopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3072

2-(trifluoromethyl)pyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3073

2-nitropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3074

2-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3075

6-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3076

6-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3077

6-bromopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3078

6-iodopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3079

6-(trifluoromethyl)pyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3080

6-nitropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3081

6-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3082

5-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3083

5-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3084

5-bromopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3085

5-iodopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3086

5-(trifluoromethyl)pyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3087

5-nitropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3088

5-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3089

4-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3090

4-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3091

4-bromopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3092

4-iodopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3093

4-(trifluoromethyl)pyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3094

4-nitropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3095

4-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3096

2,6-dichloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3097

pyridin-3-yl N-oxide

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3098

pyridin-4-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3099

2-chloropyridin-4-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3100

3-bromopyridin-4-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3101

3,5-dichloropyridin-4-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3102

3-(trifluoromethyl)pyridin-4-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3103

2,6-dicyanopyridin-4-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3104

pyridin-4-yl N-oxide

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3105

pyridin-2-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3106

3-chloropyridin-2-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3107

4-bromopyridin-2-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3108

5-iodopyridin-2-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3109

6-chloropyridin-2-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3110

4-cyanopyridin-2-yl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

16-3111

phenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3112

2-fluorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3113

3-fluorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3114

4-fluorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3115

2-chlorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3116

3-chlorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3117

4-chlorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3118

2-bromophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3119

3-bromophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3120

4-bromophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3121

2-iodophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3122

3-iodophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3123

4-iodophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3124

(2-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3125

(3-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3126

(4-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3127

2-nitrophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3128

3-nitrophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3129

4-nitrophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3130

2-cyanophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3131

3-cyanophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3132

4-cyanophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3133

2,6-difluorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3134

3,4-dichlorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3135

2,4-dichlorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3136

2-chloro-4-fluorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3137

2-chloro-4,5-difluorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3138

4-bromo-2-chlorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3139

2-bromo-4-chlorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3140

2-bromo-4-fluorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3141

2-chloro-4-nitrophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3142

3,5-dicyanophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3143

4-cyano-2-fluorophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3144

2-chloro-4-cyanophenyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3145

pyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3146

2-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3147

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3148

2-bromopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3149

2-iodopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3150

2-(trifluoromethyl)pyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3151

2-nitropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3152

2-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3153

6-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3154

6-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3155

6-bromopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3156

6-iodopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3157

6-(trifluoromethyl)pyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3158

6-nitropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3159

6-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3160

5-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3161

5-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3162

5-bromopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3163

5-iodopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3164

5-(trifluoromethyl)pyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3165

5-nitropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3166

5-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3167

4-fluoropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3168

4-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3169

4-bromopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3170

4-iodopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3171

4-(trifluoromethyl)pyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3172

4-nitropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3173

4-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3174

2,6-dichloropyridin-3-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3175

pyridin-3-yl N-oxide

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3176

pyridin-4-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3177

2-chloropyridin-4-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3178

3-bromopyridin-4-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3179

3,5-dichloropyridin-4-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3180

3-(trifluoromethyl)pyridin-4-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3181

2,6-dicyanopyridin-4-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3182

pyridin-4-yl N-oxide

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3183

pyridin-2-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3184

3-chloropyridin-2-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3185

4-bromopyridin-2-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3186

5-iodopyridin-2-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3187

6-chloropyridin-2-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3188

4-cyanopyridin-2-yl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

16-3189

phenyl

H

H

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

16-3196

2-bromophenyl

H

H

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OC2F5

16-3201

4-iodophenyl

H

H

N-oxide

H

H

H

OCF3

H

pentafluoroethyl

H

OCF3

16-3204

3-cyanophenyl

H

H

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

16-3205

4-cyanophenyl

H

H

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

16-3213

2-bromo-4-fluorophenyl

H

H

N-oxide

H

H

H

OC2F5

H

heptafluoroisopropyl

H

OCF3

16-3220

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

16-3229

5-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

OC2F5

H

heptafluoroisopropyl

H

OC2F5

16-3231

4-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OC2F5

16-3245

phenyl

H

H

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

16-3252

2-bromophenyl

H

H

N-oxide

H

H

H

OC2F5

H

nonafluoro-2-butyl

H

OCF3

16-3258

(2-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OC2F5

16-3260

3-cyanophenyl

H

H

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

16-3261

4-cyanophenyl

H

H

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

16-3276

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

16-3283

6-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

OC2F5

H

nonafluoro-2-butyl

H

OCF3

16-3284

5-chloropyridin-3-yl

H

H

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OC2F5

16-3301

phenyl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

16-3308

2-bromophenyl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OC2F5

16-3313

4-iodophenyl

H

H

N-oxide

H

H

H

CF3

H

pentafluoroethyl

H

OCF3

16-3314

(2-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

C2F5

H

heptafluoroisopropyl

H

OC2F5

16-3315

3-nitrophenyl

H

H

N-oxide

H

H

H

C2F5

H

heptafluoroisopropyl

H

OCF3

16-3316

3-cyanophenyl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

16-3317

4-cyanophenyl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

16-3324

2-bromo-4-chlorophenyl

H

H

N-oxide

H

H

H

n-C3F7

H

heptafluoroisopropyl

H

OCF3

16-3328

4-cyano-2-fluorophenyl

H

H

N-oxide

H

H

H

i-C3F7

H

heptafluoroisopropyl

H

OCF3

16-3332

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

16-3338

6-chloropyridin-3-yl

H

H

N-oxide

H

H

H

n-C3F7

H

heptafluoroisopropyl

H

OC2F5

16-3341

5-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

i-C3F7

H

heptafluoroisopropyl

H

OC2F5

16-3357

phenyl

H

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-3368

3-iodophenyl

H

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OC2F5

16-3371

3-nitrophenyl

H

H

N-oxide

H

H

H

C2F5

H

nonafluoro-2-butyl

H

OCF3

16-3372

3-cyanophenyl

H

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-3373

4-cyanophenyl

H

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-3379

4-bromo-2-chlorophenyl

H

H

N-oxide

H

H

H

i-C3F7

H

nonafluoro-2-butyl

H

OCF3

16-3382

2-chloro-4-nitrophenyl

H

H

N-oxide

H

H

H

n-C3F7

H

nonafluoro-2-butyl

H

OCF3

16-3388

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

16-3397

5-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

C2F5

H

nonafluoro-2-butyl

H

OC2F5

16-3399

4-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

n-C3F7

H

nonafluoro-2-butyl

H

OC2F5

16-3410

5-iodopyridin-2-yl

H

H

N-oxide

H

H

H

i-C3F7

H

nonafluoro-2-butyl

H

OC2F5

16-3413

phenyl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-3425

4-iodophenyl

H

H

N-oxide

H

H

H

CF3

H

pentafluoroethyl

H

CF3

16-3427

(3-trifluoromethyl)phenyl

H

H

N-oxide

H

H

H

C2F5

H

heptafluoroisopropyl

H

CF3

16-3433

3-cyanophenyl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-3434

4-cyanophenyl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-3440

4-bromo-2-chlorophenyl

H

H

N-oxide

H

H

H

n-C3F7

H

heptafluoroisopropyl

H

CF3

16-3445

4-cyano-2-fluorophenyl

H

H

N-oxide

H

H

H

i-C3F7

H

heptafluoroisopropyl

H

CF3

16-3447

pyridin-3-yl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-3449

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

16-3450

2-bromopyridin-3-yl

H

H

N-oxide

H

H

H

C2F5

H

heptafluoroisopropyl

H

C2F5

16-3461

6-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

C2F5

H

heptafluoroisopropyl

H

n-C3F7

16-3465

4-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

C2F5

H

heptafluoroisopropyl

H

i-C3F7

16-3481

phenyl

H

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

16-3493

4-iodophenyl

H

H

N-oxide

H

H

H

C2F5

H

nonafluoro-2-butyl

H

CF3

16-3501

3-cyanophenyl

H

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

16-3502

4-cyanophenyl

H

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

16-3508

4-bromo-2-chlorophenyl

H

H

N-oxide

H

H

H

n-C3F7

H

nonafluoro-2-butyl

H

CF3

16-3513

4-cyano-2-fluorophenyl

H

H

N-oxide

H

H

H

i-C3F7

H

nonafluoro-2-butyl

H

CF3

16-3517

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

16-3518

2-bromopyridin-3-yl

H

H

N-oxide

H

H

H

C2F5

H

nonafluoro-2-butyl

H

C2F5

16-3529

6-cyanopyridin-3-yl

H

H

N-oxide

H

H

H

C2F5

H

nonafluoro-2-butyl

H

n-C3F7

16-3536

pyridin-4-yl

H

H

N-oxide

H

H

H

C2F5

H

nonafluoro-2-butyl

H

i-C3F7

TABLE 17

com-

pound

number

Q1

R1

R2

A

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

17-1

phenyl

Me

H

N

H

H

H

F

H

heptafluoroisopropyl

H

F

17-2

3-cyanophenyl

Me

H

N

H

H

H

F

H

heptafluoroisopropyl

H

F

17-3

4-cyanophenyl

Me

H

N

H

H

H

F

H

heptafluoroisopropyl

H

F

17-4

2-chloropyridin-3-yl

Me

H

N

H

H

H

F

H

heptafluoroisopropyl

H

F

17-5

phenyl

Me

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

17-6

3-cyanophenyl

Me

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

17-7

4-cyanophenyl

Me

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

17-8

2-chloropyridin-3-yl

Me

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

17-9

phenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

17-29

3-cyanophenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

17-30

4-cyanophenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

17-45

2-chloropyridin-3-yl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

17-87

phenyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

17-107

3-cyanophenyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

17-108

4-cyanophenyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

17-123

2-chloropyridin-3-yl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

17-165

phenyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

17-185

3-cyanophenyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

17-186

4-cyanophenyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

17-201

2-chloropyridin-3-yl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

17-243

phenyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

17-263

3-cyanophenyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

17-264

4-cyanophenyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

17-279

2-chloropyridin-3-yl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

17-321

phenyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

I

17-341

3-cyanophenyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

I

17-342

4-cyanophenyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

I

17-357

2-chloropyridin-3-yl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

I

17-399

phenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

17-400

2-fluorophenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

17-419

3-cyanophenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

17-420

4-cyanophenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

17-435

2-chloropyridin-3-yl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

17-477

phenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

17-497

3-cyanophenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

17-498

4-cyanophenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

17-513

2-chloropyridin-3-yl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

17-555

phenyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

17-575

3-cyanophenyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

17-576

4-cyanophenyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

17-591

2-chloropyridin-3-yl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

17-633

phenyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

17-653

3-cyanophenyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

17-654

4-cyanophenyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

17-669

2-chloropyridin-3-yl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

17-711

phenyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

17-731

3-cyanophenyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

17-732

4-cyanophenyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

17-747

2-chloropyridin-3-yl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

17-789

phenyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

17-809

3-cyanophenyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

17-810

4-cyanophenyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

17-825

2-chloropyridin-3-yl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

17-867

phenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

17-887

3-cyanophenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

17-888

4-cyanophenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

17-903

2-chloropyridin-3-yl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

17-945

phenyl

Me

H

N

H

H

H

F

H

heptafluoroisopropyl

H

CF3

17-946

phenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

17-957

3-iodophenyl

Me

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

17-958

4-iodophenyl

Me

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

17-965

2-cyanophenyl

Me

H

N

H

H

H

Cl

H

pentafluoroethyl

H

C2F5

17-966

3-cyanophenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

17-967

4-cyanophenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

17-970

2,4-dichlorophenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

17-971

2-chloro-4-fluorophenyl

n-Pr

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

17-974

2-bromo-4-chlorophenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

17-981

2-fluoropyridin-3-yl

Me

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

17-982

2-chloropyridin-3-yl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

17-988

6-fluoropyridin-3-yl

i-Pr

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

17-995

5-fluoropyridin-3-yl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

17-997

5-bromopyridin-3-yl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

17-998

5-iodopyridin-3-yl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

17-1000

5-nitropyridin-3-yl

Me

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

17-1002

4-fluoropyridin-3-yl

Me

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

17-1004

4-bromopyridin-3-yl

CH2CH═CH2

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

17-1005

4-iodopyridin-3-yl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

17-1011

pyridin-4-yl

CN

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

17-1023

4-cyanopyridin-2-yl

Me

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

17-1024

phenyl

Me

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

17-1025

phenyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-1033

3-bromophenyl

CH2C≡CH

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-1038

(2-trifluoromethyl)phenyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

17-1040

(4-trifluoromethyl)phenyl

NH2

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-1045

3-cyanophenyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-1046

4-cyanophenyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-1053

2-bromo-4-chlorophenyl

C(O)OMe

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-1055

2-chloro-4-nitrophenyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

17-1061

2-chloropyridin-3-yl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-1074

5-fluoropyridin-3-yl

C(O)OEt

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

17-1076

5-bromopyridin-3-yl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

17-1077

5-iodopyridin-3-yl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

17-1081

4-fluoropyridin-3-yl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

17-1083

4-bromopyridin-3-yl

C(O)C(O)Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-1085

4-(trifluoromethyl )pyridin-3-yl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

17-1086

4-nitropyridin-3-yl

C(O)C(O)Et

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

17-1100

5-iodopyridin-2-yl

C(O)Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-1102

4-cyanopyridin-2-yl

C(O)Et

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

17-1103

phenyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-1104

2-fluorophenyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-1117

(3-trifluoromethyl)phenyl

S(O)2Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-1135

4-cyano-2-fluorophenyl

S(O)2Et

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-1139

2-chloropyridin-3-yl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-1150

6-nitropyridin-3-yl

CH2Ph

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-1159

4-fluoropyridin-3-yl

CH2(3-Py)

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-1180

4-cyanopyridin-2-yl

CH2(3-Py—N-

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

17-1181

phenyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

17-1182

2-fluorophenyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

17-1201

3-cyanophenyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

17-1202

4-cyanophenyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

17-1208

4-bromo-2-chlorophenyl

Et

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

17-1217

2-chloropyridin-3-yl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

17-1234

5-(trifluoromethyl)pyridin-3-yl

CN

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

17-1259

phenyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

17-1260

2-fluorophenyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

17-1279

3-cyanophenyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

17-1280

4-cyanophenyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

17-1295

2-chloropyridin-3-yl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

17-1308

5-fluoropyridin-3-yl

C(O)Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

17-1337

phenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

17-1338

2-fluorophenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

17-1357

3-cyanophenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

17-1358

4-cyanophenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

17-1373

2-chloropyridin-3-yl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

17-1415

phenyl

Me

H

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

17-1446

2-chloropyridin-3-yl

Me

H

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

17-1471

phenyl

Me

H

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

17-1502

2-chloropyridin-3-yl

Me

H

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

17-1527

phenyl

Me

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

17-1558

2-chloropyridin-3-yl

Me

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

17-1583

phenyl

Me

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

17-1614

2-chloropyridin-3-yl

Me

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

17-1639

phenyl

Me

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

17-1659

3-cyanophenyl

Me

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

17-1660

4-cyanophenyl

Me

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

17-1675

2-chloropyridin-3-yl

Me

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

17-1707

phenyl

Me

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

17-1727

3-cyanophenyl

Me

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

17-1728

4-cyanophenyl

Me

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

17-1743

2-chloropyridin-3-yl

Me

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

17-1775

phenyl

Me

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

17-1776

3-cyanophenyl

Me

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

17-1777

4-cyanophenyl

Me

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

17-1778

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

17-1779

phenyl

Me

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

17-1780

3-cyanophenyl

Me

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

17-1781

4-cyanophenyl

Me

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

17-1782

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

17-1783

phenyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

17-1803

3-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

17-1804

4-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

17-1819

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

17-1861

phenyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

17-1881

3-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

17-1882

4-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

17-1897

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

17-1939

phenyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

17-1959

3-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

17-1960

4-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

17-1975

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

17-2017

phenyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

17-2037

3-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

17-2038

4-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

17-2053

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

17-2095

phenyl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

17-2114

2-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

pentafluoroethyl

H

I

17-2115

3-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

17-2131

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

17-2173

phenyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

17-2193

3-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

17-2194

4-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

17-2209

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

17-2251

phenyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

17-2271

3-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

17-2272

4-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

17-2287

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

17-2329

phenyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

17-2349

3-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

17-2350

4-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

17-2365

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

17-2407

phenyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

17-2427

3-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

17-2428

4-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

17-2443

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

17-2485

phenyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

17-2505

3-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

17-2506

4-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

17-2563

phenyl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

17-2583

3-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

17-2584

4-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

17-2599

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

17-2641

phenyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

17-2661

3-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

17-2662

4-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

17-2677

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

17-2719

phenyl

Me

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

CF3

17-2720

phenyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

17-2740

3-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

17-2741

4-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

17-2756

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

17-2798

phenyl

Me

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

17-2799

phenyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-2819

3-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-2820

4-cyanophenyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-2835

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

17-2877

phenyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-2897

3-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-2898

4-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-2913

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-2914

2-bromopyridin-3-yl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

17-2955

phenyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

17-2975

3-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

17-2976

4-cyanophenyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

17-2991

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

17-3033

phenyl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

17-3053

3-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

17-3054

4-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

17-3069

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

17-3111

phenyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

17-3131

3-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

17-3132

4-cyanophenyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

17-3147

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

17-3189

phenyl

Me

H

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

17-3220

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

17-3245

phenyl

Me

H

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

17-3276

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

17-3301

phenyl

Me

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

17-3332

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

17-3357

phenyl

Me

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

17-3388

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

17-3413

phenyl

Me

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

17-3433

3-cyanophenyl

Me

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

17-3434

4-cyanophenyl

Me

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

17-3449

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

17-3481

phenyl

Me

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

17-3501

3-cyanophenyl

Me

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

17-3502

4-cyanophenyl

Me

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

17-3517

2-chloropyridin-3-yl

Me

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 18

compound

number

Q1

R1

R2

A

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

18-1

phenyl

H

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

F

18-2

3-cyanophenyl

H

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

F

18-3

4-cyanophenyl

H

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

F

18-4

2-chloropyridin-3-yl

H

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

F

18-5

phenyl

H

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

18-6

3-cyanophenyl

H

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

18-7

4-cyanophenyl

H

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

18-8

2-chloropyridin-3-yl

H

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

18-9

phenyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

18-29

3-cyanophenyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

18-30

4-cyanophenyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

18-45

2-chloropyridin-3-yl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

18-87

phenyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

18-107

3-cyanophenyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

18-108

4-cyanophenyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

18-123

2-chloropyridin-3-yl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

18-165

phenyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

18-176

3-iodophenyl

H

Me

N

H

H

H

Br

H

pentafluoroethyl

H

Br

18-177

4-iodophenyl

H

Me

N

H

H

H

Br

H

pentafluoroethyl

H

Br

18-185

3-cyanophenyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

18-186

4-cyanophenyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

18-201

2-chloropyridin-3-yl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

18-243

phenyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

18-263

3-cyanophenyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

18-264

4-cyanophenyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

18-279

2-chloropyridin-3-yl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

18-321

phenyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

I

18-341

3-cyanophenyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

I

18-342

4-cyanophenyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

I

18-357

2-chloropyridin-3-yl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

I

18-399

phenyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

18-419

3-cyanophenyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

18-420

4-cyanophenyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

18-435

2-chloropyridin-3-yl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

18-477

phenyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

18-497

3-cyanophenyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

18-498

4-cyanophenyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

18-513

2-chloropyridin-3-yl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

18-555

phenyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

18-575

3-cyanophenyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

18-576

4-cyanophenyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

18-591

2-chloropyridin-3-yl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

18-633

phenyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

18-653

3-cyanophenyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

18-654

4-cyanophenyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

18-669

2-chloropyridin-3-yl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

18-711

phenyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

18-731

3-cyanophenyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

18-732

4-cyanophenyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

18-747

2-chloropyridin-3-yl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

18-789

phenyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

18-809

3-cyanophenyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

18-810

4-cyanophenyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

18-825

2-chloropyridin-3-yl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

18-867

phenyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

18-887

3-cyanophenyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

18-888

4-cyanophenyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

18-903

2-chloropyridin-3-yl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

18-945

phenyl

H

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

CF3

18-946

phenyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-957

3-iodophenyl

H

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

18-958

4-iodophenyl

H

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

18-960

(3-trifluoromethyl)phenyl

H

Et

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-965

2-cyanophenyl

H

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

C2F5

18-966

3-cyanophenyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-967

4-cyanophenyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-970

2,4-dichlorophenyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

18-971

2-chloro-4-fluorophenyl

H

n-Pr

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-974

2-bromo-4-chlorophenyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

18-981

2-fluoropyridin-3-yl

H

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

18-982

2-chloropyridin-3-yl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-988

6-fluoropyridin-3-yl

H

i-Pr

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-995

5-fluoropyridin-3-yl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

18-997

5-bromopyridin-3-yl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

18-998

5-iodopyridin-3-yl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

18-1000

5-nitropyridin-3-yl

H

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

18-1002

4-fluoropyridin-3-yl

H

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

18-1004

4-bromopyridin-3-yl

H

CH2CH═CH2

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

18-1005

4-iodopyridin-3-yl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

18-1011

pyridin-4-yl

H

CN

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-1023

4-cyanopyridin-2-yl

H

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

18-1024

phenyl

H

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

18-1025

phenyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-1033

3-bromophenyl

H

CH2C≡CH

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-1038

(2-trifluoromethyl)phenyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

18-1040

(4-trifluoromethyl)phenyl

H

NH2

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-1045

3-cyanophenyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-1046

4-cyanophenyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-1053

2-bromo-4-chlorophenyl

H

C(O)OMe

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-1055

2-chloro-4-nitrophenyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

18-1061

2-chloropyridin-3-yl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-1074

5-fluoropyndin-3-yl

H

C(O)OEt

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

18-1076

5-bromopyridin-3-yl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

18-1077

5-iodopyridin-3-yl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

18-1081

4-fluoropyridin-3-yl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

18-1083

4-bromopyridin-3-yl

H

C(O)C(O)Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-1085

4-(trifluoromethyl)pyridin-

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

3-yl

18-1086

4-nitropyridin-3-yl

H

C(O)C(O)Et

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

18-1100

5-iodopyridin-2-yl

H

C(O)Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-1102

4-cyanopyridin-2-yl

H

C(O)Et

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

18-1103

phenyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-1104

2-fluorophenyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-1117

(3-trifluoromethyl)phenyl

H

S(O)2Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-1123

3-cyanophenyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-1124

4-cyanophenyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-1135

4-cyano-2-fluorophenyl

H

S(O)2Et

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-1139

2-chloropyridin-3-yl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-1150

6-nitropyridin-3-yl

H

CH2Ph

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-1159

4-fluoropyridin-3-yl

H

CH2(3-Py)

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-1180

4-cyanopyridin-2-yl

H

CH2(3-Py—N-

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

18-1181

phenyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

18-1182

2-fluorophenyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

18-1201

3-cyanophenyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

18-1202

4-cyanophenyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

18-1208

4-bromo-2-chlorophenyl

H

Et

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

18-1217

2-chloropyridin-3-yl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

18-1234

5-(trifluoromethyl)pyridin-

H

CN

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

3-yl

18-1259

phenyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

18-1260

2-fluorophenyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

18-1279

3-cyanophenyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

18-1280

4-cyanophenyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

18-1295

2-chloropyridin-3-yl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

18-1308

5-fluoropyridin-3-yl

H

C(O)Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

18-1337

phenyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

18-1338

2-fluorophenyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

18-1357

3-cyanophenyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

18-1358

4-cyanophenyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

18-1373

2-chloropyridin-3-yl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

18-1415

phenyl

H

Me

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

18-1446

2-chloropyridin-3-yl

H

Me

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

18-1471

phenyl

H

Me

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

18-1502

2-chloropyridin-3-yl

H

Me

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

18-1527

phenyl

H

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

18-1558

2-chloropyridin-3-yl

H

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

18-1583

phenyl

H

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

18-1614

2-chloropyridin-3-yl

H

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

18-1639

phenyl

H

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

18-1659

3-cyanophenyl

H

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

18-1660

4-cyanophenyl

H

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

18-1675

2-chloropyridin-3-yl

H

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

18-1707

phenyl

H

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

18-1727

3-cyanophenyl

H

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

18-1728

4-cyanophenyl

H

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

18-1743

2-chloropyridin-3-yl

H

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

18-1775

phenyl

H

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

18-1776

3-cyanophenyl

H

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

18-1777

4-cyanophenyl

H

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

18-1778

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

18-1779

phenyl

H

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

18-1780

3-cyanophenyl

H

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

18-1781

4-cyanophenyl

H

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

18-1782

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

18-1783

phenyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

18-1803

3-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

18-1804

4-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

18-1819

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

18-1861

phenyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

18-1881

3-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

18-1882

4-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

18-1897

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

18-1939

phenyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

18-1959

3-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

18-1960

4-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

18-1975

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

18-2017

phenyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

18-2037

3-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

18-2038

4-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

18-2053

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

18-2095

phenyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

18-2115

3-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

18-2116

4-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

18-2131

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

18-2173

phenyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

18-2193

3-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

18-2194

4-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

18-2209

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

18-2251

phenyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

18-2271

3-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

18-2272

4-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

18-2287

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

18-2291

2-nitropyridin-3-yl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OC2F5

18-2329

phenyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

18-2349

3-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

18-2350

4-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

18-2365

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

18-2407

phenyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

18-2427

3-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

18-2428

4-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

18-2443

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

18-2485

phenyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

18-2505

3-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

18-2506

4-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

18-2521

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

18-2563

phenyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

18-2583

3-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

18-2584

4-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

18-2599

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

18-2641

phenyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

18-2661

3-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

18-2662

4-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

18-2677

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

18-2719

phenyl

H

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

CF3

18-2720

phenyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-2740

3-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-2741

4-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-2756

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

18-2798

phenyl

H

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

18-2799

phenyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-2819

3-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-2820

4-cyanophenyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-2835

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

18-2877

phenyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-2897

3-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-2898

4-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-2913

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

18-2955

phenyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

18-2975

3-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

18-2976

4-cyanophenyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

18-2991

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

18-3033

phenyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

18-3053

3-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

18-3054

4-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

18-3069

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

18-3111

phenyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

18-3131

3-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

18-3132

4-cyanophenyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

18-3147

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

18-3189

phenyl

H

Me

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

18-3220

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

18-3245

phenyl

H

Me

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

18-3276

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

18-3301

phenyl

H

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

18-3332

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

18-3357

phenyl

H

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

18-3388

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

18-3413

phenyl

H

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

18-3433

3-cyanophenyl

H

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

18-3434

4-cyanophenyl

H

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

18-3449

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

18-3481

phenyl

H

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

18-3501

3-cyanophenyl

H

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

18-3502

4-cyanophenyl

H

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

18-3517

2-chloropyridin-3-yl

H

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 19

com-

pound

number

Q1

R1

R2

A

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

19-1

phenyl

Me

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

F

19-2

3-cyanophenyl

Me

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

F

19-3

4-cyanophenyl

Me

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

F

19-4

2-chloropyridin-3-yl

Me

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

F

19-5

phenyl

Me

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

19-6

3-cyanophenyl

Me

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

19-7

4-cyanophenyl

Me

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

19-8

2-chloropyridin-3-yl

Me

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

Cl

19-9

phenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

19-11

3-fluorophenyl

Et

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

19-12

4-fluorophenyl

Me

Et

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

19-29

3-cyanophenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

19-30

4-cyanophenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

19-45

2-chloropyridin-3-yl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

19-87

phenyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

19-107

3-cyanophenyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

19-108

4-cyanophenyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

19-123

2-chloropyridin-3-yl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

19-165

phenyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

19-185

3-cyanophenyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

19-186

4-cyanophenyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

19-201

2-chloropyridin-3-yl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

19-243

phenyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

19-263

3-cyanophenyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

19-264

4-cyanophenyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

19-279

2-chloropyridin-3-yl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

19-321

phenyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

I

19-341

3-cyanophenyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

I

19-342

4-cyanophenyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

I

19-357

2-chloropyridin-3-yl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

I

19-399

phenyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

19-419

3-cyanophenyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

19-420

4-cyanophenyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

19-435

2-chloropyridin-3-yl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

19-673

phenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

19-693

3-cyanophenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

19-694

4-cyanophenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

19-709

2-chloropyridin-3-yl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

19-751

phenyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

19-771

3-cyanophenyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

19-772

4-cyanophenyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

19-787

2-chloropyndin-3-yl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

19-829

phenyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

19-849

3-cyanophenyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

19-850

4-cyanophenyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

19-865

2-chloropyridin-3-yl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

19-907

phenyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

19-927

3-cyanophenyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

19-928

4-cyanophenyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

19-943

2-chloropyridin-3-yl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

19-985

phenyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

19-1005

3-cyanophenyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

19-1006

4-cyanophenyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

19-1021

2-chloropyridin-3-yl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

19-1063

phenyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

19-1083

3-cyanophenyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

19-1084

4-cyanophenyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

19-1099

2-chloropyridin-3-yl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

19-1337

phenyl

Me

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

CF3

19-1338

phenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1349

3-iodophenyl

Me

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

19-1350

4-iodophenyl

Me

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

19-1352

(3-trifluoromethyl)phenyl

Et

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1353

(4-trifluoromethyl)phenyl

Me

Et

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1357

2-cyanophenyl

Me

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

C2F5

19-1358

3-cyanophenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1359

4-cyanophenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1362

2,4-dichlorophenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

19-1363

2-chloro-4-fluorophenyl

n-Pr

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1365

4-bromo-2-chlorophenyl

Me

n-Pr

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1366

2-bromo-4-chlorophenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

19-1373

2-fluoropyridin-3-yl

Me

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

19-1374

2-chloropyridin-3-yl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1378

2-nitropyridin-3-yl

Me

i-Pr

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1380

6-fluoropyridin-3-yl

i-Pr

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1387

5-fluoropyridin-3-yl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

19-1389

5-bromopyridin-3-yl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

19-1390

5-iodopyridin-3-yl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

19-1392

5-nitropyridin-3-yl

Me

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

19-1393

5-cyanopyridin-3-yl

Me

CH2CH═CH2

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1394

4-fluoropyridin-3-yl

Me

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

19-1396

4-bromopyridin-3-yl

CH2CH═CH2

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

19-1397

4-iodopyridin-3-yl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

i-C3F7

19-1400

4-cyanopyridin-3-yl

Me

CN

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1403

pyridin-4-yl

CN

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-1415

4-cyanopyridin-2-yl

Me

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

19-1416

phenyl

Me

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

19-1417

phenYI

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1425

3-bromophenyl

CH2C≡CH

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1429

4-iodophenyl

Me

CH2C≡CH

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1430

(2-trifluoromethyl)phenyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

19-1432

(4-trifluoromethyl)phenyl

NH2

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1436

2-cyanophenyl

Me

NH2

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1437

3-cyanophenyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1438

4-cyanophenyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1442

2-chloro-4-fluorophenyl

Me

C(O)OMe

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1445

2-bromo-4-chlorophenyl

C(O)OMe

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1447

2-chloro-4-nitrophenyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

19-1453

2-chloropyridin-3-yl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1464

6-nitropyridin-3-yl

Me

C(O)OEt

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1466

5-fluoropyridin-3-yl

C(O)OEt

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

19-1468

5-bromopyridin-3-yl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

19-1469

5-iodopyridin-3-yl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

19-1472

5-cyanopyridin-3-yl

Me

C(O)C(O)Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1473

4-fluoropyridin-3-yl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

19-1475

4-bromopyridin-3-yl

C(O)C(O)Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1477

4-(trifluoromethyl)pyridin-3-yl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

n-C3F7

19-1478

4-nitropyridin-3-yl

C(O)C(O)Et

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

19-1479

4-cyanopyridin-3-yl

Me

C(O)C(O)Et

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1484

3-bromopyridin-4-yl

Me

C(O)Et

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1491

4-bromopyridin-2-yl

Me

C(O)Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1492

5-iodopyridin-2-yl

C(O)Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-1494

4-cyanopyridin-2-yl

C(O)Et

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

C2F5

19-1495

phenyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1496

2-fluorophenyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1509

(3-trifluoromethyl)phenyl

S(O)2Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1514

2-cyanophenyl

Me

S(O)2Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1515

3-cyanophenyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1516

4-cyanophenyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1523

2-bromo-4-chlorophenyl

Me

S(O)2Et

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1527

4-cyano-2-fluorophenyl

S(O)2Et

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1531

2-chloropyridin-3-yl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1542

6-nitropyridin-3-yl

CH2Ph

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1546

5-bromopyridin-3-yl

Me

CH2Ph

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1551

4-fluoropyridin-3-yl

CH2(3-Py)

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1556

4-nitropyridin-3-yl

Me

CH2(3-Py)

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-1570

5-iodopyridin-2-yl

Me

CH2(3-Py—N-

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

19-1572

4-cyanopyridin-2-yl

CH2(3-Py—N-

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

oxide)

19-1573

phenyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-1574

2-fluorophenyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-1593

3-cyanophenyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-1594

4-cyanophenyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-1600

4-bromo-2-chlorophenyl

Et

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-1603

2-chloro-4-nitrophenyl

Me

Et

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-1609

2-chloropyridin-3-yl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-1626

5-(trifluoromethyl)pyridin-3-yl

CN

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-1627

5-nitropyridin-3-yl

Me

CN

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-1651

phenyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

19-1652

2-fluorophenyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

19-1671

3-cyanophenyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

19-1672

4-cyanophenyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

19-1687

2-chloropyridin-3-yl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

19-1700

5-fluoropyridin-3-yl

C(O)Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

19-1705

5-nitropyridin-3-yl

Me

C(O)Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

19-1729

phenyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

19-1730

2-fluorophenyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

19-1749

3-cyanophenyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

19-1750

4-cyanophenyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

19-1765

2-chloropyridin-3-yl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

19-2003

phenyl

Me

Me

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

19-2034

2-chloropyridin-3-yl

Me

Me

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

19-2059

phenyl

Me

Me

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

19-2090

2-chloropyridin-3-yl

Me

Me

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

19-2115

phenyl

Me

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

19-2146

2-chloropyridin-3-yl

Me

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

19-2171

phenol

Me

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

19-2202

2-chloropyridin-3-yl

Me

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

19-2227

phenyl

Me

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

19-2247

3-cyanophenyl

Me

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

19-2248

4-cyanophenyl

Me

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

19-2263

2-chloropyridin-3-yl

Me

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

19-2295

phenyl

Me

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

19-2315

3-cyanophenyl

Me

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

19-2316

4-cyanophenyl

Me

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

19-2331

2-chloropyridin-3-yl

Me

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

19-2559

phenyl

Me

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

19-2560

3-cyanophenyl

Me

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

19-2561

4-cyanophenyl

Me

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

19-2562

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

19-2563

phenyl

Me

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

19-2564

3-cyanophenyl

Me

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

19-2565

4-cyanophenyl

Me

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

19-2566

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

19-2567

phenyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

19-2587

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

19-2588

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

19-2603

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

19-2645

phenyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

19-2665

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

19-2666

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

19-2681

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

19-2723

phenyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

19-2743

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

19-2744

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

19-2759

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

19-2801

phenyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

19-2821

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

19-2822

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

19-2837

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

19-2879

phenyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

19-2899

3-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

19-2900

4-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

19-2915

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

19-2957

phenyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

19-2977

3-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

19-2978

4-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

19-2993

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

19-3231

phenyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

19-3251

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

19-3252

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

19-3267

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

19-3309

phenyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

19-3329

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

19-3330

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

19-3345

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

19-3387

phenyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

19-3407

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

19-3408

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

19-3423

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

19-3465

phenyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

19-3485

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

19-3486

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

19-3501

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

19-3543

phenyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

19-3563

3-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

19-3564

4-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

19-3579

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

19-3621

phenyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

19-3641

3-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

19-3642

4-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

19-3657

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

19-3895

phenyl

Me

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

CF3

19-3896

phenyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-3916

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-3917

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-3932

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

19-3974

phenyl

Me

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

19-3975

phenyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-3995

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-3996

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-4011

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

19-4053

phenyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-4073

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-4074

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-4089

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

19-4131

phenyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-4151

3-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-4152

4-cyanophenyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-4167

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

19-4209

phenyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

19-4229

3-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

19-4230

4-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

19-4245

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

19-4287

phenyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

19-4307

3-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

19-4308

4-cyanophenyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

19-4323

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

19-4561

phenyl

Me

Me

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

19-4592

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

19-4617

phenyl

Me

Me

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

19-4648

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

19-4673

phenyl

Me

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

19-4704

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

19-4729

phenyl

Me

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

19-4760

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

19-4785

phenyl

Me

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

19-4805

3-cyanophenyl

Me

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

19-4806

4-cyanophenyl

Me

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

19-4821

2-chloropyridin-3-yl

Me

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

19-4853

phenyl

Me

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

19-4873

3-cyanophenyl

Me

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

19-4874

4-cyanophenyl

Me

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

19-4889

2-chloropyridrn-3-yl

Me

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 20

compound

number

Q1

R1

R2

A

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

20-9

3-bromophenyl

H

Et

N

H

H

H

Cl

F

heptafluoroisopropyl

F

Cl

20-39

2-iodopyridin-3-yl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

I

20-152

3-bromophenyl

H

Et

N

H

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

20-182

2-iodopyridin-3-yl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

20-287

phenyl

H

H

N

H

H

H

Cl

F

heptafluoroisopropyl

H

CF3

20-288

2-fluorophenyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

F

CF3

20-289

3-fluorophenyl

H

Me

N

H

H

H

Cl

Cl

heptafluoroisopropyl

H

CF3

20-290

4-fluorophenyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

Cl

CF3

20-291

2-chlorophenyl

H

H

N

H

H

H

F

Br

heptafluoroisopropyl

H

CF3

20-292

3-chlorophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

Br

CF3

20-293

4-chlorophenyl

Et

H

N

H

H

H

Cl

I

heptafluoroisopropyl

H

C2F5

20-294

2-bromophenyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

I

CF3

20-295

3-bromophenyl

H

Et

N

H

H

H

Cl

F

heptafluoroisopropyl

F

CF3

20-296

4-bromophenyl

H

H

N

H

H

H

Cl

F

heptafluoroisopropyl

Cl

CF3

20-297

2-iodophenyl

H

H

N

H

H

H

Cl

F

heptafluoroisopropyl

Br

CF3

20-298

3-iodophenyl

Et

Et

N

H

H

H

Cl

F

pentafluoroethyl

I

C2F5

20-299

4-iodophenyl

H

H

N

H

H

H

Cl

Cl

pentafluoroethyl

F

CF3

20-300

(2-trifluoromethyl)phenyl

H

H

N

H

H

H

Cl

Cl

heptafluoroisopropyl

Cl

CF3

20-301

(3-trifluoromethyl)phenyl

n-Pr

H

N

H

H

H

Cl

Cl

heptafluoroisopropyl

Br

CF3

20-302

(4-trifluoromethyl)phenyl

H

H

N

H

H

H

Cl

Cl

heptafluoroisopropyl

I

n-C3F7

20-303

2-nitrophenyl

H

n-Pr

N

H

H

H

Cl

Br

heptafluoroisopropyl

F

CF3

20-304

3-nitrophenyl

H

H

N

H

H

H

Cl

Br

heptafluoroisopropyl

Cl

CF3

20-305

4-nitrophenyl

H

H

N

H

H

H

Cl

Br

heptafluoroisopropyl

Br

CF3

20-306

2-cyanophenyl

n-Pr

n-Pr

N

H

H

H

Cl

Br

pentafluoroethyl

I

CF3

20-307

3-cyanophenyl

H

H

N

H

H

H

F

I

nonafluoro-2-butyl

F

CF3

20-308

4-cyanophenyl

H

H

N

H

H

H

Cl

I

nonafluoro-2-butyl

Cl

CF3

20-309

2,6-difluorophenyl

H

H

N

H

H

H

Cl

I

nonafluoro-2-butyl

Br

CF3

20-310

3,4-dichlorophenyl

H

H

N

H

H

H

Cl

I

nonafluoro-2-butyl

I

CF3

20-311

2,4-dichlorophenyl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

20-312

2-chloro-4-fluorophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

20-313

2-chloro-4,5-difluorophenyl

i-Pr

H

N

H

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

20-314

4-bromo-2-chlorophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

20-315

2-bromo-4-chlorophenyl

H

H

N

H

H

H

Cl

n-Pr

nonafluoro-2-butyl

H

CF3

20-316

2-bromo-4-fluorophenyl

H

i-Pr

N

H

H

H

Cl

H

nonafluoro-2-butyl

n-Pr

CF3

20-317

2-chloro-4-nitrophenyl

i-Pr

i-Pr

N

H

H

H

Cl

i-Pr

nonafluoro-2-butyl

H

CF3

20-318

3,5-dicyanophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

i-Pr

CF3

20-319

4-cyano-2-fluorophenyl

H

H

N

H

H

H

Cl

n-Bu

nonafluoro-2-butyl

H

CF3

20-320

2-chloro-4-cyanophenyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

n-Bu

CF3

20-321

pyridin-3-yl

H

H

N

H

H

H

Cl

i-Bu

nonafluoro-2-butyl

H

CF3

20-322

2-fluoropyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

i-Bu

CF3

20-323

2-chloropyridin-3-yl

H

H

N

H

H

H

Cl

s-Bu

nonafluoro-2-butyl

H

C2F5

20-324

2-bromopyridin-3-yl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

s-Bu

CF3

20-325

2-iodopyridin-3-yl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

20-326

2-(trifluoromethyl)pyridin-

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

3-yl

20-327

2-nitropyridin-3-yl

C(O)Me

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

n-Pr

CF3

20-328

2-cyanopyridin-3-yl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

i-Pr

CF3

20-329

6-fluoropyridin-3-yl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

n-Bu

CF3

20-330

6-chloropyridin-3-yl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

i-Bu

CF3

20-331

6-bromopyridin-3-yl

H

C(O)Me

N

H

H

H

Cl

Me

nonafluoro-2-butyl

s-Bu

CF3

20-332

6-iodopyridin-3-yl

H

H

N

H

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

20-333

6-(trifluoromethyl)pyridin-

H

H

N

H

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

3-yl

20-334

6-nitropyridin-3-yl

C(O)Me

C(O)Me

N

H

H

H

Cl

Et

nonafluoro-2-butyl

n-Pr

CF3

20-335

6-cyanopyridir-3-yl

H

H

N

H

H

H

Cl

Et

nonafluoro-2-butyl

i-Pr

CF3

20-336

phenyl

H

H

N

H

H

H

Br

Et

heptafluoroisopropyl

n-Bu

CF3

20-337

5-fluoropyridin-3-yl

H

H

N

H

H

H

Br

Et

heptafluoroisopropyl

i-Bu

CF3

20-338

5-chloropyridin-3-yl

H

H

N

H

H

H

Br

Et

heptafluoroisopropyl

s-Bu

CF3

20-339

5-bromopyridin-3-yl

H

H

N

H

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

20-340

5-iodopyridin-3-yl

H

H

N

H

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

20-341

5-(trifluoromethyl)pyridin-

Me

Et

N

H

H

H

Br

n-Pr

pentafluoroethyl

n-Pr

CF3

3-yl

20-342

5-nitropyridin-3-yl

H

H

N

H

H

H

Br

n-Pr

heptafluoroisopropyl

i-Pr

CF3

20-343

5-cyanopyridin-3-yl

H

H

N

H

H

H

Br

n-Pr

pentafluoroethyl

n-Bu

CF3

20-344

4-fluoropyridin-3-yl

H

H

N

H

H

H

Br

n-Pr

heptafluoroisopropyl

i-Bu

CF3

20-345

4-chloropyridin-3-yl

H

H

N

H

H

H

Br

n-Pr

heptafluoroisopropyl

s-Bu

CF3

20-346

4-bromopyridin-3-yl

Me

n-Pr

N

H

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

20-347

4-iodopyridin-3-yl

H

H

N

H

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

20-348

4-(trifluoromethyl)pyridin-

H

H

N

H

H

H

Br

i-Pr

heptafluoroisopropyl

n-Pr

CF3

3-yl

20-349

4-nitropyridin-3-yl

H

H

N

H

H

H

Br

i-Pr

heptafluoroisopropyl

i-Pr

CF3

20-350

4-cyanopyridin-3-yl

H

H

N

H

H

H

Br

i-Pr

heptafluoroisopropyl

n-Bu

CF3

20-351

2,6-dichloropyridin-3-yl

H

H

N

H

H

H

Br

i-Pr

heptafluoroisopropyl

i-Bu

CF3

20-352

pyridin-3-yl N-oxide

Me

i-Pr

N

H

H

H

Br

i-Pr

heptafluoroisopropyl

s-Bu

CF3

20-353

pyridin-4-yl

H

H

N

H

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

20-354

2-chloropyridin-4-yl

H

H

N

H

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

20-355

3-bromopyridin-4-yl

H

H

N

H

H

H

Br

n-Bu

heptafluoroisopropyl

n-Pr

CF3

20-356

3,5-dichloropyridin-4-yl

H

H

N

H

H

H

Br

n-Bu

nonafluoro-2-butyl

i-Pr

CF3

20-357

3-(trifluoromethyl)pyridin-

H

H

N

H

H

H

Br

n-Bu

nonafluoro-2-butyl

n-Bu

CF3

4-yl

20-358

2,6-dicyanopyridin-4-yl

H

H

N

H

H

H

Br

n-Bu

nonafluoro-2-butyl

i-Bu

CF3

20-359

pyridin-4-yl N-oxide

Me

C(O)Me

N

H

H

H

Br

n-Bu

nonafluoro-2-butyl

s-Bu

CF3

20-360

pyridin-2-yl

H

H

N

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

20-361

3-chloropyridin-2-yl

H

H

N

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

20-362

4-bromopyridin-2-yl

H

H

N

H

H

H

Br

i-Bu

nonafluoro-2-butyl

n-Pr

CF3

20-363

5-iodopyridin-2-yl

H

H

N

H

H

H

Br

i-Bu

nonafluoro-2-butyl

i-Pr

CF3

20-364

6-chloropyridin-2-yl

H

H

N

H

H

H

Br

i-Bu

nonafluoro-2-butyl

n-Bu

CF3

20-365

4-cyanopyridin-2-yl

H

H

N

H

H

H

Br

i-Bu

nonafluoro-2-butyl

n-Bu

CF3

20-366

phenyl

H

H

N

H

H

H

Br

i-Bu

nonafluoro-2-butyl

s-Bu

C2F5

20-367

2-fluorophenyl

H

H

N

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

20-368

3-fluorophenyl

H

H

N

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

20-369

4-fluorophenyl

H

H

N

H

H

H

Br

s-Bu

nonafluoro-2-butyl

n-Pr

CF3

20-370

2-chlorophenyl

H

H

N

H

H

H

Br

s-Bu

nonafluoro-2-butyl

i-Pr

CF3

20-371

3-chlorophenyl

H

H

N

H

H

H

Br

s-Bu

nonafluoro-2-butyl

n-Bu

CF3

20-372

4-chlorophenyl

H

H

N

H

H

H

Br

s-Bu

nonafluoro-2-butyl

i-Bu

CF3

20-373

2-bromophenyl

Et

Me

N

H

H

H

Br

s-Bu

nonafluoro-2-butyl

s-Bu

CF3

20-374

3-bromophenyl

H

H

N

H

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

20-375

4-bromophenyl

H

H

N

H

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

20-376

2-iodophenyl

H

H

N

H

H

H

Br

F

nonafluoro-2-butyl

n-Pr

CF3

20-377

3-iodophenyl

H

H

N

H

H

H

Br

F

nonafluoro-2-butyl

i-Pr

CF3

20-378

4-iodophenyl

H

H

N

H

H

H

Br

F

nonafluoro-2-butyl

n-Bu

CF3

20-379

(2-trifluoromethyl)phenyl

H

H

N

H

H

H

Br

F

nonafluoro-2-butyl

i-Bu

CF3

20-380

(3-trifluoromethyl)phenyl

Et

n-Pr

N

H

H

H

Br

F

nonafluoro-2-butyl

s-Bu

CF3

20-381

(4-trifluoromethyl)phenyl

Et

i-Pr

N

H

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

20-382

2-nitrophenyl

H

H

N

H

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

20-383

phenyl

H

H

N

H

H

H

I

Cl

pentafluoroethyl

n-Pr

CF3

20-384

3-nitrophenyl

H

H

N

H

H

H

I

Cl

heptafluoroisopropyl

i-Pr

CF3

20-385

4-nitrophenyl

H

H

N

H

H

H

I

Cl

heptafluoroisopropyl

n-Bu

CF3

20-386

2-cyanophenyl

Et

C(O)Me

N

H

H

H

I

Cl

heptafluoroisopropyl

i-Bu

CF3

20-387

3-cyanophenyl

H

H

N

H

H

H

I

Cl

heptafluoroisopropyl

s-Bu

CF3

20-388

3-cyanophenyl

H

H

N

H

H

H

I

Br

heptafluoroisopropyl

Me

CF3

20-389

2,6-difluorophenyl

H

H

N

H

H

H

I

Br

heptafluoroisopropyl

Et

CF3

20-390

3,4-dichlorophenyl

H

H

N

H

H

H

I

Br

pentafluoroethyl

n-Pr

CF3

20-391

2,4-dichlorophenyl

H

H

N

H

H

H

I

Br

heptafluoroisopropyl

i-Pr

CF3

20-392

2-chloro-fluorophenyl

H

H

N

H

H

H

I

Br

heptafluoroisopropyl

n-Bu

CF3

20-393

2-chloro-4,5-difluorophenyl

H

H

N

H

H

H

I

Br

heptafluoroisopropyl

i-Bu

CF3

20-394

4-bromo-2-chlorophenyl

H

H

N

H

H

H

I

Br

heptafluoroisopropyl

s-Bu

CF3

20-395

2-bromo-4-chlorophenyl

n-Pr

Me

N

H

H

H

I

I

heptafluoroisopropyl

Me

CF3

20-396

2-bromo-4-flulorophenyl

H

H

N

H

H

H

I

I

heptafluoroisopropyl

Et

CF3

20-397

2-chloro-4-nitrophenyl

n-Pr

Et

N

H

H

H

I

I

heptafluoroisopropyl

n-Pr

CF3

20-398

3,5-dicyanophenyl

H

H

N

H

H

H

I

I

heptafluoroisopropyl

i-Pr

CF3

20-399

4-cyano-2-flulorophenyl

H

H

N

H

H

H

I

I

heptafluoroisopropyl

n-Bu

CF3

20-400

4-cyano-2-cyanophenyl

H

H

N

H

H

H

I

I

heptafluoroisopropyl

i-Bu

CF3

20-401

pyridin-3-yl

H

H

N

H

H

H

I

I

heptafluoroisopropyl

s-Bu

CF3

20-402

2-fluoropyridin-3-yl

H

H

N

H

H

H

I

Me

heptafluoroisopropyl

F

C2F5

20-403

2-chloropyridin-3-yl

H

H

N

H

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

20-404

2-bromopyridin-3-yl

H

H

N

H

H

H

I

Me

nonafluoro-2-butyl

Br

n-C3F7

20-405

2-iodopyridin-3-yl

H

H

N

H

H

H

I

Me

nonafluoro-2-butyl

I

i-C3F7

20-406

2-(trifluoromethyl)pyridin-

H

H

N

H

H

H

I

Et

nonafluoro-2-butyl

F

CF3

3-yl

20-407

2-nitropyridin-3-yl

H

H

N

H

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

20-408

2-cyanopyridin-3-yl

H

H

N

H

H

H

I

Et

nonafluoro-2-butyl

Br

CF3

20-409

6-fluoropyridin-3-yl

n-Pr

i-Pr

N

H

H

H

I

Et

nonafluoro-2-butyl

I

C2F5

20-410

6-chloropyridin-3-yl

H

H

N

H

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

20-411

6-bromopyridin-3-yl

H

H

N

H

H

H

I

n-Pr

nonafluoro-2-butyl

Cl

CF3

20-412

6-iodopyridin-3-yl

H

H

N

H

H

H

I

n-Pr

nonafluoro-2-butyl

Br

CF3

20-413

6-(trifluoromethyl)pyridin-

H

H

N

H

H

H

I

n-Pr

nonafluoro-2-butyl

I

n-C3F7

3-yl

20-414

6-nitropyridin-3-yl

H

H

N

H

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

20-415

5-cyanopyridin-3-yl

H

H

N

H

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

20-416

5-fluoropyridin-3-yl

n-Pr

C(O)Me

N

H

H

H

I

i-Pr

nonafluoro-2-butyl

Br

CF3

20-417

5-chloropyridin-3-yl

H

H

N

H

H

H

I

i-Pr

nonafluoro-2-butyl

I

CF3

20-418

5-bromopyridin-3-yl

H

H

N

H

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

20-419

5-iodopyridin-3-yl

H

H

N

H

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

20-420

5-(trifluoromethyl)pyridin-

H

H

N

H

H

H

I

n-Bu

nonafluoro-2-butyl

Br

CF3

3-yl

20-421

5-nitropyridin-3-yl

i-Pr

Me

N

H

H

H

I

n-Bu

nonafluoro-2-butyl

I

CF3

20-422

5-cyanopyridin-3-yl

H

H

N

H

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

20-423

4-fluoropyridin-3-yl

H

H

N

H

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

20-424

4-chloropyridin-3-yl

H

H

N

H

H

H

I

i-Bu

nonafluoro-2-butyl

Br

CF3

20-425

4-bromopyridin-3-yl

i-Pr

Et

N

H

H

H

I

i-Bu

nonafluoro-2-butyl

I

CF3

20-426

4-iodopyridin-3-yl

i-Pr

n-Pr

N

H

H

H

I

s-Bu

nonafluoro-2-butyl

F

CF3

20-427

4-(trifluoromethyl)pyridin-

H

H

N

H

H

H

I

s-Bu

nonafluoro-2-butyl

Cl

CF3

3-yl

20-428

4-nitropyridin-3-yl

i-Pr

C(O)Me

N

H

H

H

I

s-Bu

nonafluoro-2-butyl

Br

CF3

20-429

4-cyanopyridin-3-yl

H

H

N

H

H

H

I

s-Bu

nonafluoro-2-butyl

I

CF3

20-438

3-bromophenyl

H

Et

N

H

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

20-468

2-iodopyridin-3-yl

H

H

N

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

20-581

3-bromophenyl

H

Et

N

H

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

20-611

2-iodopyridin-3-yl

H

H

N

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

20-724

3-bromophenyl

H

Et

N

H

H

H

CF3

F

heptafluoroisopropyl

F

CF3

20-754

2-iodopyridin-3-yl

H

H

N

H

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

20-887

3-bromophenyl

H

Et

N-oxide

H

H

H

Cl

F

heptafluoroisopropyl

F

Cl

20-897

2-iodopyridin-3-yl

H

H

N-oxide

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

I

20-1010

3-bromophenyl

H

Et

N-oxide

H

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

20-1040

2-iodopyridin-3-yl

H

H

N-oxide

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

20-1154

4-bromophenyl

H

H

N-oxide

H

H

H

Cl

F

heptafluoroisopropyl

Cl

CF3

20-1169

2,4-dichlorophenyl

H

H

N-oxide

H

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

20-1233

4-bromophenyl

H

H

N-oxide

H

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

20-1261

2-chloropyridin-3-yl

H

H

N-oxide

H

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

20-1296

3-bromophenyl

H

Et

N-oxide

H

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

20-1326

2-iodopyridin-3-yl

H

H

N-oxide

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

20-1439

3-bromophenyl

H

Et

N-oxide

H

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

20-1469

2-iodopyridin-3-yl

H

H

N-oxide

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

20-1582

3-bromophenyl

H

Et

N-oxide

H

H

H

CF3

F

heptafluoroisopropyl

F

CF3

20-1612

2-iodopyridin-3-yl

H

H

N-oxide

H

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

TABLE 21

compound

number

Q2

R1

R2

A

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

21-1

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

F

21-2

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

21-13

2,2,2-trichloroethyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

21-14

2,2,2-tribromoethyl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

Cl

21-22

1,3-dichloro-2-propyl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

Cl

21-26

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

21-42

2,2,2-trichloroethyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

21-55

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

21-71

2,2,2-trichloroethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

21-74

3-fluoro-n-propyl

H

H

N

H

H

H

Br

H

pentafluoroethyl

H

Br

21-80

1,3-dichloro-2-propyl

H

H

N

H

H

H

Br

H

pentafluoroethyl

H

Br

21-84

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

21-100

2,2,2-trichloroethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

21-113

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

21-129

2,2,2-trichloroethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

I

21-131

n-propyl

H

H

N

H

H

H

I

H

pentafluoroethyl

H

I

21-138

1,3-dichloro-2-propyl

H

H

N

H

H

H

I

H

pentafluoroethyl

H

I

21-142

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

I

21-158

2,2,2-trichloroethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

21-171

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

21-177

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

Cl

21-178

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

Br

21-179

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

I

21-180

2,2,2-trichloroethyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Br

21-181

2,2,2-trichloroethyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

I

21-182

2,2,2-trichloroethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

I

21-183

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

Cl

21-184

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

Br

21-185

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

I

21-186

2,2,2-trichloroethyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Br

21-187

2,2,2-trichloroethyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

I

21-188

2,2,2-trichloroethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

I

21-189

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

21-190

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

21-201

2,2,2-trichloroethyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

21-202

2,2,2-tribromoethyl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

OCF3

21-206

3-bromo-n-propyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OC2F5

21-210

1,3-dichloro-2-propyl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

OC2F5

21-214

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

21-226

2-cyanoethyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OC2F5

21-230

2,2,2-trichloroethyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

21-243

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

21-245

s-butyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OC2F5

21-254

2-iodoethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OC2F5

21-259

2,2,2-trichloroethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

21-260

2,2,2-tribromoethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

21-272

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

21-288

2,2,2-trichloroethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

21-289

2,2,2-tribromoethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OC2F5

21-301

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

21-317

2,2,2-trichloroethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

21-321

3-chloro-n-propyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OC2F5

21-330

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

21-346

2,2,2-trichloroethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

21-359

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

21-363

benzyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OC2F5

21-365

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

heptafluoroisopropyl

H

CF3

21-366

2,2,2-trichloroethyl

H

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

21-373

2-cyanoethyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

21-377

2,2,2-trichloroethyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

21-378

2,2,2-tribromoethyl

H

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

21-383

i-propyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

21-390

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

21-397

ethyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

21-406

2,2,2-trichloroethyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

21-419

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

21-425

methyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-426

ethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-427

2-fluoroethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-428

2-chloroethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-429

2-bromoethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-430

2-iodoethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-431

2-cyanoethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

C2F5

21-432

2,2-difluoroethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-433

2,2-dichloroethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-434

2,2,2-trifluoroethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-435

2,2,2-trichloroethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-436

2,2,2-tribromoethyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-437

n-propyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-438

3-fluoro-n-propyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-439

3-chloro-n-propyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-440

3-bromo-n-propyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-441

i-propyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-442

1,2-difluoro-2-propyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

n-C3F7

21-443

1,3-difluoro-2-propyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-444

1,3-dichloro-2-propyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-445

1-chloro-3-fluoro-2-propyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-446

3,3,3-trifluoro-n-propyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-447

n-butyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-448

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-449

i-butyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-450

s-butyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-451

vinyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-452

benzyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-453

phenyl

H

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-454

methyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-455

ethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-456

2-fluoroethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-457

2-chloroethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-458

2-bromoethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-459

2-iodoethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-460

2-cyanoethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-461

2,2-difluoroethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-462

2,2-dichloroethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-463

2,2,2-trifluoroethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-464

2,2,2-trichloroethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-465

2,2,2-tribromoethyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-466

n-propyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-467

3-fluoro-n-propyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-468

3-chloro-n-propyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-469

3-bromo-n-propyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-470

i-propyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-471

1,2-difluoro-2-propyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-472

1,3-difluoro-2-propyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-473

1,3-dichloro-2-propyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-474

1-chloro-3-fluoro-2-propyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-475

3,3,3-trifluoro-n-propyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-476

n-butyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-477

4,4,4-trifluoro-n-propyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-478

i-butyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-479

s-butyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-480

vinyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-481

benzyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-482

phenyl

H

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

i-C3F7

21-483

methyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-484

ethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-485

2-fluoroethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-486

2-chloroethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-487

2-bromoethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-488

2-iodoethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-489

2-cyanoethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-490

2,2-difluoroethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-491

2,2-dichloroethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-492

2,2,2-trifluoroethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-493

2,2,2-trichloroethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-494

2,2,2-tribromoethyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-495

n-propyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-496

3-fluoro-n-propyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-497

3-chloro-n-propyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-498

3-bromo-n-propyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

C2F5

21-499

i-propyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-500

1,2-difluoro-2-propyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-501

1,3-difluoro-2-propyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-502

1,3-dichloro-2-propyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-503

1-chloro-3-fluoro-2-propyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-504

3,3,3-trifluoro-n-propyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-505

n-butyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-506

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-507

i-butyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-508

s-butyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-509

vinyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-510

benzyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-511

phenyl

H

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-512

methyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-513

ethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-514

2-fluoroethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-515

2-chloroethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-516

2-bromoethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-517

2-iodoethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-518

2-cyanoethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-519

2,2-difluoroethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-520

2,2-dichloroethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-521

2,2,2-trifluoroethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-522

2,2,2-trichloroethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-523

2,2,2-tribromoethyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-524

n-propyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

n-C3F7

21-525

3-fluoro-n-propyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-526

3-chloro-n-propyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-527

3-bromo-n-propyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-528

i-propyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-529

1,2-difluoro-2-propyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-530

1,3-difluoro-2-propyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-531

1,3-dichloro-2-propyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-532

1-chloro-3-fluoro-2-propyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-533

3,3,3-trifluoro-n-propyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-534

n-butyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-535

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-536

i-butyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-537

s-butyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-538

vinyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

i-C3F7

21-539

benzyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-540

phenyl

H

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-547

2-cyanoethyl

H

H

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OC2F5

21-551

2,2,2-trichloroethyl

H

H

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

21-552

2,2,2-tribromoethyl

H

H

N

H

H

H

OCF3

H

pentafluoroethyl

H

OCF3

21-561

1-chloro-3-fluoro-2-propyl

H

H

N

H

H

H

OC2F5

H

heptafluoroisopropyl

H

OC2F5

21-564

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

21-566

s-butyl

H

H

N

H

H

H

OC2F5

H

heptafluoroisopropyl

H

OCF3

21-576

2-cyanoethyl

H

H

N

H

H

H

OC2F5

H

nonafluoro-2-butyl

H

OCF3

21-580

2,2,2-trichloroethyl

H

H

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

21-581

2,2,2-tribromoethyl

H

H

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OC2F5

21-592

n-butyl

H

H

N

H

H

H

OC2F5

H

nonafluoro-2-butyl

H

OC2F5

21-593

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

21-605

2-cyanoethyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OC2F5

21-609

2,2,2-trichloroethyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

21-610

2,2,2-tribromoethyl

H

H

N

H

H

H

C2F5

H

heptafluoroisopropyl

H

OC2F5

21-621

n-butyl

H

H

N

H

H

H

n-C3F7

H

heptafluoroisopropyl

H

OCF3

21-622

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

21-625

vinyl

H

H

N

H

H

H

i-C3F7

H

heptafluoroisopropyl

H

OCF3

21-633

2-iodoethyl

H

H

N

H

H

H

C2F5

H

nonafluoro-2-butyl

H

OCF3

21-638

2,2,2-trichloroethyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

21-640

n-propyl

H

H

N

H

H

H

n-C3F7

H

nonafluoro-2-butyl

H

OCF3

21-644

i-propyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OC2F5

21-651

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

21-652

i-butyl

H

H

N

H

H

H

i-C3F7

H

nonafluoro-2-butyl

H

OCF3

21-655

benzyl

H

H

N

H

H

H

n-C3F7

H

nonafluoro-2-butyl

H

OC2F5

21-656

phenyl

H

H

N

H

H

H

i-C3F7

H

nonafluoro-2-butyl

H

OC2F5

21-667

2,2,2-trichloroethyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

21-670

3-fluoro-n-propyl

H

H

N

H

H

H

C2F5

H

heptafluoroisopropyl

H

CF3

21-673

i-propyl

H

H

N

H

H

H

i-C3F7

H

heptafluoroisopropyl

H

CF3

21-675

1,3-difluoro-2-propyl

H

H

N

H

H

H

CF3

H

pentafluoroethyl

H

CF3

21-679

n-butyl

H

H

N

H

H

H

C2F5

H

heptafluoroisopropyl

H

C2F5

21-680

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

21-681

i-butyl

H

H

N

H

H

H

C2F5

H

heptafluoroisopropyl

H

n-C3F7

21-683

vinyl

H

H

N

H

H

H

n-C3F7

H

heptafluoroisopropyl

H

CF3

21-696

2,2,2-trichloroethyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

21-708

n-butyl

H

H

N

H

H

H

C2F5

H

nonafluoro-2-butyl

H

i-C3F7

21-709

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

21-712

vinyl

H

H

N

H

H

H

n-C3F7

H

nonafluoro-2-butyl

H

i-C3F7

21-715

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

21-716

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

21-727

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

21-756

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

21-785

2,2,2-trichloroethyl

H

H

N-oxtde

H

H

H

Br

H

heptafluoroisopropyl

H

Br

21-814

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

21-843

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

21-872

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

21-894

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Br

21-903

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

21-904

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

21-915

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

21-944

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

21-973

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

21-1002

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

21-1031

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

21-1060

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

21-1079

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

CF3

21-1080

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

21-1091

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

21-1120

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

21-1149

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

21-1178

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

21-1207

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

21-1236

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

21-1265

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

21-1294

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

21-1323

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

21-1352

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

21-1381

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

21-1410

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 22

compound

number

Q2

R1

R2

A

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

22-1

2,2,2-trichloroethyl

Me

H

N

H

H

H

F

H

heptafluoroisopropyl

H

F

22-2

2,2,2-trichloroethyl

Me

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

22-13

2,2,2-trichloroethyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

22-42

2,2,2-trichloroethyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

22-71

2,2,2-trichloroethyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

22-100

2,2,2-trichloroethyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

22-129

2,2,2-trichloroethyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

I

22-158

2,2,2-trichloroethyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

22-186

2,2,2-trichloroethyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Br

22-189

2,2,2-trichloroethyl

Me

H

N

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

22-190

2,2,2-trichloroethyl

Me

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

22-201

2,2,2-trichloroethyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

22-230

2,2,2-trichloroethyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

22-259

2,2,2-trichloroethyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

22-288

2,2,2-trichloroethyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

22-317

22,2-trichloroethyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

22-346

22,2-trichloroethyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

22-365

2,2,2-trichloroethyl

Me

H

N

H

H

H

F

H

heptafluoroisopropyl

H

CF3

22-366

2,2,2-trichloroethyl

Me

H

N

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

22-373

2-cyanoethyl

Et

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

22-377

2,2,2-trichloroethyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

22-379

n-propyl

Me

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

22-383

i-propyl

n-Pr

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

22-386

1,3-dichloro-2-propyl

Me

H

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

22-387

1-chloro-3-fluoro-2-propyl

i-Pr

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

22-390

4,4.4-trifluoro-n-butyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

22-391

i-butyl

CH2CH═CH2

H

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

22-397

ethyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

22-402

2-cyanoethyl

CN

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

22-406

2,2,2-trichloroethyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

22-408

n-propyl

CH2C≡CH

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

22-419

4,4,4-trifluoro-n-butyl

Me

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

22-420

i-butyl

NH2

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

22-431

2-cyanoethyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

C2F5

22-435

2,2,2-trichloroethyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

22-438

3-fluoro-n-propyl

C(O)OMe

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

22-442

1,2-difluoro-2-propyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

n-C3F7

22-448

4,4,4-trifluoro-n-butyl

Me

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

22-451

vinyl

C(O)C(O)OMe

H

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

22-464

2,2,2-trichloroethyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

22-466

n-propyl

C(O)OEt

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

22-470

i-propyl

C(O)Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

22-477

4,4,4-trifluoro-n-butyl

Me

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

22-482

phenyl

C(O)C(O)OEt

H

N

H

H

H

Br

H

nonafluoro-2-butyl

H

i-C3F7

22-493

2,2,2-trichloroethyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

22-498

3-bromo-n-propyl

C(O)Et

H

N

H

H

H

I

H

heptafluoroisopropyl

H

C2F5

22-506

4,4,4-trifluoro-n-butyl

Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

22-510

benzyl

S(O)2Me

H

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

22-518

2-cyanoethyl

S(O)2Et

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

22-522

2,2,2-trichloroethyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

22-523

2,2,2-tribromoethyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

22-524

n-propyl

CH2Ph

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

n-C3F7

22-528

i-propyl

CH2(3-Py)

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

22-535

4,4,4-trifluoro-n-butyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

22-537

s-butyl

CH2(3-Py—N-

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

22-538

vinyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

i-C3F7

22-539

benzyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

22-540

phenyl

Me

H

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

22-551

2,2,2-trichloroethyl

Me

H

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

22-580

2,2,2-trichloroethyl

Me

H

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

22-609

2,2,2-trichloroethyl

Me

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

22-638

2,2,2-trichloroethyl

Me

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

22-667

2,2,2-trichloroethyl

Me

H

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

22-696

2,2,2-trichloroethyl

Me

H

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

22-715

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

22-716

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

22-727

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

22-756

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

22-785

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

22-814

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

22-843

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

22-872

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

22-894

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Br

22-903

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

22-904

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

22-915

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

22-944

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

22-973

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

22-1002

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

22-1031

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

22-1060

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

22-1079

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

CF3

22-1080

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

22-1091

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

22-1120

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

22-1149

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

22-1178

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

22-1207

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

22-1236

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

22-1265

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

22-1294

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

22-1323

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

22-1352

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

22-1381

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

22-1410

2,2,2-trichloroethyl

Me

H

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 23

compound

number

Q2

R1

R2

A

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

23-1

2,2,2-trichloroethyl

H

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

F

23-2

2,2,2-trichloroethyl

H

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

23-13

2,2,2-trichloroethyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

23-42

2,2,2-trichloroethyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

23-100

2,2,2-trichloroethyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

23-129

2,2,2-trichloroethyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

I

23-158

2,2,2-trichloroethyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

23-186

2,2,2-trichloroethyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Br

23-189

2,2,2-trichloroethyl

H

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

23-190

2,2,2-trichloroethyl

H

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

23-201

2,2,2-trichloroethyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

23-230

2,2,2-trichloroethyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

23-259

2,2,2-trichloroethyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

23-288

2,2,2-trichloroethyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

23-317

2,2,2-trichloroethyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

23-346

2,2,2-trichloroethyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

23-365

2,2,2-trichloroethyl

H

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

CF3

23-366

2,2,2-trichloroethyl

H

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

23-373

2-cyanoethyl

H

Et

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

23-377

2,2,2-trichloroethyl

H

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

23-379

n-propyl

H

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

23-383

i-propyl

H

n-Pr

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

23-386

1,3-dichloro-2-propyl

H

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

23-387

1-chloro-3-fluoro-2-propyl

H

i-Pr

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

23-391

i-butyl

H

CH2CH═CH2

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

23-397

ethyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

23-402

2-cyanoethyl

H

CN

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

23-406

2,2,2-trichloroethyl

H

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

23-408

n-propyl

H

CH2C≡CH

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

23-420

i-butyl

H

NH2

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

23-431

2-cyanoethyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

C2F5

23-435

2,2,2-trichloroethyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

23-437

n-propyl

H

C(O)OMe

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

23-442

1,2-difluoro-2-propyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

n-C3F7

23-448

4,4,4-trifluoro-n-butyl

H

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

23-451

vinyl

H

C(O)C(O)OMe

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

23-464

2,2,2-trichloroethyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

23-466

n-propyl

H

C(O)OEt

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

23-470

i-propyl

H

C(O)Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

23-477

4,4,4-trifluoro-n-butyl

H

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

23-482

phenyl

H

C(O)C(O)OEt

N

H

H

H

Br

H

nonafluoro-2-butyl

H

i-C3F7

23-493

2,2,2-trichloroethyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

23-498

3-bromo-n-propyl

H

C(O)Et

N

H

H

H

I

H

heptafluoroisopropyl

H

C2F5

23-506

4,4,4-trifluoro-n-butyl

H

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

23-510

benzyl

H

S(O)2Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

23-518

2-cyanoethyl

H

S(O)2Et

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

23-522

2,2,2-trichloroethyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

23-524

n-propyl

H

CH2Ph

N

H

H

H

I

H

nonafluoro-2-butyl

H

n-C3F7

23-528

i-propyl

H

CH2(3-Py)

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

23-535

4,4,4-trifluoro-n-butyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

23-537

s-butyl

H

CH2(3-Py—N-

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

23-538

vinyl

H

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

i-C3F7

23-551

2,2,2-trichloroethyl

H

Me

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

23-580

2,2.2-trichloroethyl

H

Me

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

23-609

2,2,2-trichloroethyl

H

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

23-638

2,2,2-trichloroethyl

H

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

23-667

2,2,2-trichloroethyl

H

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

23-696

2,2,2-trichloroethyl

H

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

23-715

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

23-716

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

23-727

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

23-756

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

23-785

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

23-814

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

23-843

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

23-872

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

23-895

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

I

23-903

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

23-904

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

23-915

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

23-944

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

23-973

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

23-1002

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

23-1031

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

23-1060

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

23-1079

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

CF3

23-1080

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

23-1091

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

23-1120

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

23-1149

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

23-1178

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

23-1207

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

23-1236

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

23-1265

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

23-1294

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

23-1323

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

23-1352

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

23-1381

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

23-1410

2,2,2-trichloroethyl

H

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 24

compound

number

Q2

R1

R2

A

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

24-1

2,2,2-trichloroethyl

Me

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

F

24-2

2,2,2-trichloroethyl

Me

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

F

24-13

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

24-42

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

24-71

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

Br

24-100

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

24-129

2,2,2-trichloroethyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

I

24-158

2,2,2-trichloroethyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

I

24-376

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

Br

24-385

2,2,2-trichloroethyl

Me

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

24-386

2,2,2-trichloroethyl

Me

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

24-397

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

24-426

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

24-455

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

24-484

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

24-513

2,2,2-trichloroethyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

24-542

2,2,2-trichloroethyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

24-757

2,2,2-trichloroethyl

Me

Me

N

H

H

H

F

H

heptafluoroisopropyl

H

CF3

24-758

2,2,2-trichloroethyl

Me

Me

N

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

24-764

2-iodoethyl

Me

Et

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

24-765

2-cyanoethyl

Et

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

24-769

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

24-771

n-propyl

Me

n-Pr

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

24-775

i-propyl

n-Pr

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

24-778

1,3-dichloro-2-propyl

Me

Me

N

H

H

H

Cl

H

pentafluoroethyl

H

CF3

24-779

1-chloro-3-fluoro-2-propyl

i-Pr

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

24-781

n-butyl

Me

i-Pr

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

24-783

i-butyl

CH2CH═CH2

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

24-784

s-butyl

Me

CH2CH═CH2

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

24-785

vinyl

Me

CN

N

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

24-789

ethyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

i-C3F7

24-794

2-cyanoethyl

CN

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

24-798

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

24-799

2,2,2-tribromoethyl

Me

CH2C≡CH

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

24-800

n-propyl

CH2C≡CH

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

24-810

n-butyl

Me

NH2

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

24-812

i-butyl

NH2

Me

N

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

24-823

2-cyanoethyl

Me

C(O)OMe

N

H

H

H

Br

H

heptafluoroisopropyl

H

C2F5

24-827

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

24-829

n-propyl

C(O)OMe

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

24-834

1,2-difluoro-2-propyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

n-C3F7

24-840

4,4,4-trifluoro-n-butyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

24-841

i-butyl

Me

C(O)C(O)OMe

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

24-842

s-butyl

Me

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

24-843

vinyl

C(O)C(O)OMe

Me

N

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

24-852

2-cyanoethyl

Me

C(O)OEt

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

24-856

2,2,2-trichloroethyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

24-858

n-propyl

C(O)OEt

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

24-861

3-bromo-n-propyl

Me

C(O)Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

24-862

i-propyl

C(O)Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

24-869

4,4,4-trifluoro-n-butyl

Me

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

24-870

i-butyl

Me

C(O)C(O)OEt

N

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

24-874

phenyl

C(O)C(O)OEt

Me

N

H

H

H

Br

H

nonafluoro-2-butyl

H

i-C3F7

24-885

2,2,2-trichloroethyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

24-887

n-propyl

Me

C(O)Et

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

24-890

3-bromo-n-propyl

C(O)Et

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

C2F5

24-898

4,4,4-trifluoro-n-butyl

Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

24-899

i-butyl

Me

S(O)2Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

24-902

benzyl

S(O)2Me

Me

N

H

H

H

I

H

heptafluoroisopropyl

H

CF3

24-909

2-iodoethyl

Me

S(O)2Et

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

24-910

2-cyanoethyl

S(O)2Et

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

24-914

2,2,2-trichloroethyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

24-915

2,2,2-tribromoethyl

Me

CH2Ph

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

24-916

n-propyl

CH2Ph

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

n-C3F7

24-920

i-propyl

CH2(3-Py)

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

24-926

n-butyl

Me

CH2(3-Py)

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

24-927

4,4,4-trifluoro-n-butyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

24-929

s-butyl

CH2(3-Py—N-

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

24-930

vinyl

Me

Me

N

H

H

H

I

H

nonafluoro-2-butyl

H

i-C3F7

24-932

phenyl

Me

CH2(3-Py—N-

N

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

oxide)

24-1139

2,2,2-trichloroethyl

Me

Me

N

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

24-1168

2,2,2 trichloroethyl

Me

Me

N

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

24-1197

2,2,2-trichloroethyl

Me

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

24-1226

2,2,2-trichloroethyl

Me

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

24-1255

2,2,2-trichloroethyl

Me

Me

N

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

24-1284

2,2,2-trichloroethyl

Me

Me

N

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

24-1499

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

F

24-1500

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

F

24-1511

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

24-1540

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

Cl

24-1569

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

Br

24-1598

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

Br

24-1627

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

I

24-1656

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

I

24-1875

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

I

24-1883

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

OCF3

24-1884

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

OCF3

24-1895

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

OCF3

24-1924

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

OCF3

24-1953

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

OCF3

24-1982

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

OCF3

24-2011

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

OCF3

24-2040

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

OCF3

24-2255

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

F

H

heptafluoroisopropyl

H

CF3

24-2256

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

F

H

nonafluoro-2-butyl

H

CF3

24-2267

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

24-2296

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Cl

H

nonafluoro-2-butyl

H

CF3

24-2325

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

24-2354

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

Br

H

nonafluoro-2-butyl

H

CF3

24-2383

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

I

H

heptafluoroisopropyl

H

CF3

24-2412

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

I

H

nonafluoro-2-butyl

H

CF3

24-2637

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

OCF3

H

heptafluoroisopropyl

H

OCF3

24-2666

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

OCF3

H

nonafluoro-2-butyl

H

OCF3

24-2695

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

OCF3

24-2724

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

OCF3

24-2753

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

24-2782

2,2,2-trichloroethyl

Me

Me

N-oxide

H

H

H

CF3

H

nonafluoro-2-butyl

H

CF3

TABLE 25

compound

number

Q2

R1

R2

A

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

25-9

2,2-dichloroethyl

H

Et

N

H

H

H

Cl

F

heptafluoroisopropyl

F

Cl

25-39

2,2,2-trifluoroethyl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

I

25-152

2,2-dichloroethyl

H

Et

N

H

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

25-182

2,2,2-trifluoroethyl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

25-287

methyl

H

H

N

H

H

H

Cl

F

heptafluoroisopropyl

H

CF3

25-288

ethyl

Me

H

N

H

H

H

Cl

H

heptafluoroisopropyl

F

CF3

25-289

2-fluoroethyl

H

Me

N

H

H

H

Cl

Cl

heptafluoroisopropyl

H

CF3

25-290

2-chloroethyl

Me

Me

N

H

H

H

Cl

H

heptafluoroisopropyl

Cl

CF3

25-291

2-bromoethyl

H

H

N

H

H

H

F

Br

heptafluoroisopropyl

H

CF3

25-292

2-iodoethyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

Br

CF3

25-293

2-cyanoethyl

Et

H

N

H

H

H

Cl

Cl

heptafluoroisopropyl

H

C2F5

25-294

2,2-difluoroethyl

H

H

N

H

H

H

Cl

H

heptafluoroisopropyl

I

CF3

25-295

2,2-dichloroethyl

H

Et

N

H

H

H

Cl

F

heptafluoroisopropyl

F

CF3

25-296

22,2-trifluoroethyl

H

H

N

H

H

H

Cl

F

heptafluoroisopropyl

Cl

CF3

25-299

n-propyl

H

H

N

H

H

H

Cl

Cl

pentafluoroethyl

F

CF3

25-300

3-fluoro-n-propyl

H

H

N

H

H

H

Cl

Cl

heptafluoroisopropyl

Cl

CF3

25-303

i-propyl

H

n-Pr

N

H

H

H

Cl

Br

heptafluoroisopropyl

F

CF3

25-304

1,2-difluoro-2-propyl

H

H

N

H

H

H

Cl

Br

heptafluoroisopropyl

Cl

CF3

25-307

1-chloro-3-fluoro-2-propyl

H

H

N

H

H

H

F

I

nonafluoro-2-butyl

F

CF3

25-308

3,3,3-trifluoro-n-propyl

H

H

N

H

H

H

Cl

I

nonafluoro-2-butyl

Cl

CF3

25-311

i-butyl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

H

CF3

25-312

s-butyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

Me

CF3

25-313

vinyl

i-Pr

H

N

H

H

H

Cl

Et

nonafluoro-2-butyl

H

CF3

25-314

benzyl

H

H

N

H

H

H

Cl

H

nonafluoro-2-butyl

Et

CF3

25-325

2,2,2-trifluoroethyl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

n-C3F7

25-326

2,2,2-trichloroethyl

H

H

N

H

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

25-332

i-propyl

H

H

N

H

H

H

Cl

Et

nonafluoro-2-butyl

Me

n-C3F7

25-333

1,2-difluoro-2-propyl

H

H

N

H

H

H

Cl

Et

nonafluoro-2-butyl

Et

i-C3F7

25-339

2-chloroethyl

H

H

N

H

H

H

Br

n-Pr

heptafluoroisopropyl

Me

CF3

25-340

2-bromoethyl

H

H

N

H

H

H

Br

n-Pr

heptafluoroisopropyl

Et

CF3

25-346

2,2,2-trichloroethyl

H

H

N

H

H

H

Br

i-Pr

heptafluoroisopropyl

Me

CF3

25-347

2,2,2-tribromoethyl

H

H

N

H

H

H

Br

i-Pr

heptafluoroisopropyl

Et

CF3

25-353

1,2-difluoro-2-propyl

H

H

N

H

H

H

Br

n-Bu

heptafluoroisopropyl

Me

CF3

25-354

1,3-difluoro-2-propyl

H

H

N

H

H

H

Br

n-Bu

heptafluoroisopropyl

Et

CF3

25-360

i-butyl

H

H

N

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Me

CF3

25-361

s-butyl

H

H

N

H

H

H

Br

i-Bu

nonafluoro-2-butyl

Et

CF3

25-367

2-fluoroethyl

H

H

N

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Me

CF3

25-368

2-chloroethyl

H

H

N

H

H

H

Br

s-Bu

nonafluoro-2-butyl

Et

CF3

25-374

2,2,2-trifluoroethyl

H

H

N

H

H

H

Br

F

nonafluoro-2-butyl

Me

CF3

25-375

2,2,2-trifluoroethyl

H

H

N

H

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

25-381

i-propyl

Et

i-Pr

N

H

H

H

Br

Cl

nonafluoro-2-butyl

Me

CF3

25-382

1,2-difluoro-2-propyl

H

H

N

H

H

H

Br

Cl

nonafluoro-2-butyl

Et

CF3

25-388

2-iodoethyl

H

H

N

H

H

H

I

Br

heptafluoroisopropyl

Me

CF3

25-389

2-cyanoethyl

H

H

N

H

H

H

I

Br

heptafluoroisopropyl

Et

CF3

25-395

n-propyl

n-Pr

Me

N

H

H

H

I

I

heptafluoroisopropyl

Me

CF3

25-396

3-fluoro-n-propyl

H

H

N

H

H

H

I

I

heptafluoroisopropyl

Et

CF3

25-402

1,3-difluoro-2-propyl

H

H

N

H

H

H

I

Me

heptafluoroisopropyl

F

C2F5

25-403

1-chloro-3-fluoro-2-propyl

H

H

N

H

H

H

I

Me

nonafluoro-2-butyl

Cl

CF3

25-406

4,4,4-trifluoro-n-butyl

H

H

N

H

H

H

I

Et

nonafluoro-2-butyl

F

CF3

25-407

i-butyl

H

H

N

H

H

H

I

Et

nonafluoro-2-butyl

Cl

CF3

25-410

benzyl

H

H

N

H

H

H

I

n-Pr

nonafluoro-2-butyl

F

CF3

25-413

ethyl

H

H

N

H

H

H

I

n-Pr

nonafluoro-2-butyl

I

N-C3F7

25-414

2-fluoroethyl

H

H

N

H

H

H

I

i-Pr

nonafluoro-2-butyl

F

i-C3F7

25-415

2-chloroethyl

H

H

N

H

H

H

I

i-Pr

nonafluoro-2-butyl

Cl

CF3

25-418

2-cyanoethyl

H

H

N

H

H

H

I

n-Bu

nonafluoro-2-butyl

F

CF3

25-419

2,2-diftuoroethyl

H

H

N

H

H

H

I

n-Bu

nonafluoro-2-butyl

Cl

CF3

25-422

2,2,2-trichloroethyl

H

H

N

H

H

H

I

i-Bu

nonafluoro-2-butyl

F

CF3

25-423

2,2,2-tribromoethyl

H

H

N

H

H

H

I

i-Bu

nonafluoro-2-butyl

Cl

CF3

25-426

3-chloro-n-propyl

i-Pr

n-Pr

N

H

H

H

1

s-Bu

nonafluoro-2-butyl

F

CF3

25-427

3-bromo-n-propyl

H

H

N

H

H

H

1

s-Bu

nonafluoro-2-butyl

Cl

CF3

25-438

2,2-dichloroethyl

H

Et

N

H

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

25-468

2,2,2-trifluoroethyl

H

H

N

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

25-581

2,2-dichloroethyl

H

Et

N

H

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

25-611

2,2,2-trifluoroethyl

H

H

N

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

25-724

2,2-dichloroethyl

H

Et

N

H

H

H

CF3

F

heptafluoroisopropyl

F

CF3

25-754

2,2,2-trifluoroethyl

H

H

N

H

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

25-867

2,2-dichloroethyl

H

Et

N-oxide

H

H

H

Cl

F

heptafluoroisopropyl

F

Cl

25-897

2,2,2-trifluoroethyl

H

H

N-oxide

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

I

25-1010

2,2-dichloroethyl

H

Et

N-oxide

H

H

H

Cl

F

heptafluoroisopropyl

F

OCF3

25-1040

2,2,2-trifluoroethyl

H

H

N-oxide

H

H

H

Cl

Me

nonafluoro-2-butyl

Me

OCF3

25-1155

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Cl

F

heptafluoroisopropyl

Br

CF3

25-1168

4,4,4-trifluoro-n-butyl

H

H

N-oxide

H

H

H

Cl

I

nonafluoro-2-butyl

I

CF3

25-1184

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Cl

Me

nonafluoro-2-butyl

Et

i-C3F7

25-1233

2,2,2-trichloroethyl

H

H

N-oxide

H

H

H

Br

F

nonafluoro-2-butyl

Et

CF3

25-1264

4,4,4-trrfluoro-n-butyl

H

H

N-oxide

H

H

H

I

Et

nonafluoro-2-butyl

F

CF3

25-1296

2,2-dichloroethyl

H

Et

N-oxide

H

H

H

OCF3

F

heptafluoroisopropyl

F

OCF3

25-1326

2,2,2-trifluoroethyl

H

H

N-oxide

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

OCF3

25-1439

2,2-dichloroethyl

H

Et

N-oxide

H

H

H

OCF3

F

heptafluoroisopropyl

F

CF3

25-1469

2,2,2-trifluoroethyl

H

H

N-oxide

H

H

H

OCF3

Me

nonafluoro-2-butyl

Me

CF3

25-1582

2,2-dichloroethyl

H

Et

N-oxide

H

H

H

CF3

F

heptafluoroisopropyl

F

CF3

25-1612

2,2,2-trifluoroethyl

H

H

N-oxide

H

H

H

CF3

Me

nonafluoro-2-butyl

Me

CF3

TABLE 26
compound
number	Q1	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
26-1	phenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
26-4	4-fluorophenyl	H	H	Cl	Cl	H	heptafluoroisopropyl	H	OCF3
26-12	3-iodophenyl	H	H	H	Cl	H	pentafluoroethyl	H	OCF3
26-13	4-iodophenyl	H	H	H	Cl	H	pentafluoroethyl	H	OCF3
26-16	(4-trifluoromethyl)phenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OC2F5
26-17	2-nitrophenyl	H	H	H	F	H	heptafluoroisopropyl	H	OCF3
26-20	2-cyanophenyl	H	H	H	Cl	H	pentafluoroethyl	H	OC2F5
26-21	3-cyanophenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
26-22	4-cyanophenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
26-28	4-bromo-2-chlorophenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OC2F5
26-36	2-fluoropyridin-3-yl	H	H	H	Cl	H	pentafluoroethyl	H	OCF3
26-37	2-chloropyridin-3-yl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
26-41	2-nitropyridin-3-yl	H	H	H	Cl	H	heptafluoroisopropyl	H	OC2F5
26-50	5-fluoropyridin-3-yl	H	H	H	Cl	H	heptafluoroisopropyl	H	OC2F5
26-55	5-nitropyridin-3-yl	H	H	H	Cl	H	pentafluoroethyl	H	OCF3
26-59	4-bromopyridin-3-yl	H	H	H	Cl	H	heptafluoroisopropyl	H	OC2F5
26-60	4-iodopyridin-3-yl	H	H	H	Cl	H	heptafluoroisopropyl	H	OC2F5
26-78	4-cyanopyridin-2-yl	H	H	H	Cl	H	pentafluoroethyl	H	OCF3
26-79	phenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
26-95	2-nitrophenyl	H	H	H	F	H	nonafluoro-2-butyl	H	OCF3
26-99	3-cyanophenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
26-100	4-cyanophenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
26-105	2-chloro-4,5-difluorophenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OC2F5
26-115	2-chloropyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
26-121	6-fluoropyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OC2F5
26-130	5-bromopyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OC2F5
26-131	5-iodopyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OC2F5
26-139	4-(trifluoromethyl)pyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OC2F5
26-140	4-nitropyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OC2F5
26-157	phenyl	H	H	H	Br	H	heptafluoroisopropyl	H	OCF3
26-158	2-fluorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	OCF3
26-177	3-cyanophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	OCF3
26-178	4-cyanophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	OCF3
26-193	2-chloropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	OCF3
26-235	phenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
26-236	2-fluorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
26-255	3-cyanophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
26-256	4-cyanophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
26-271	2-chloropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
26-313	phenyl	H	H	H	I	H	heptafluoroisopropyl	H	OCF3
26-314	2-fluorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	OCF3
26-333	3-cyanophenyl	H	H	H	I	H	heptafluoroisopropyl	H	OCF3
26-334	4-cyanophenyl	H	H	H	I	H	heptafluoroisopropyl	H	OCF3
26-349	2-chloropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	OCF3
26-391	phenyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
26-392	2-fluorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
26-411	3-cyanophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
26-412	4-cyanophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
26-427	2-chloropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
26-469	phenyl	H	H	H	F	H	heptafluoroisopropyl	H	CF3
26-470	phenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
26-471	2-fluorophenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
26-481	3-iodophenyl	H	H	H	Cl	H	pentafluoroethyl	H	CF3
26-482	4-iodophenyl	H	H	H	Cl	H	pentafluoroethyl	H	CF3
26-489	2-cyanophenyl	H	H	H	Cl	H	pentafluoroethyl	H	C2F5
26-490	3-cyanophenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
26-491	4-cyanophenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
26-494	2,4-dichlorophenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	C2F5
26-498	2-bromo-4-chlorophenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
26-505	2-fluoropyridin-3-yl	H	H	H	Cl	H	pentafluoroethyl	H	CF3
26-506	2-chloropyridin-3-yl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
26-510	2-nitropyridin-3-yl	H	H	Cl	Cl	H	heptafluoroisopropyl	H	CF3
26-519	5-fluoropyridin-3-yl	H	H	H	Cl	H	heptafluoroisopropyl	H	C2F5
26-521	5-bromopyridin-3-yl	H	H	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
26-522	5-iodopyridin-3-yl	H	H	H	Cl	H	heptafluoroisopropyl	H	i-C3F7
26-524	5-nitropyridin-3-yl	H	H	H	Cl	H	pentafluoroethyl	H	CF3
26-526	4-fluoropyridin-3-yl	H	H	H	Cl	H	pentafluoroethyl	H	CF3
26-528	4-bromopyridin-3-yl	H	H	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
26-529	4-iodopyridin-3-yl	H	H	H	Cl	H	heptafluoroisopropyl	H	i-C3F7
26-548	phenyl	H	H	H	F	H	nonafluoro-2-butyl	H	CF3
26-549	phenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
26-550	2-fluorophenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
26-562	(2-trifluoromethyl)phenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	C2F5
26-569	3-cyanophenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
26-570	4-cyanophenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
26-579	2-chloro-4-nitrophenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
26-585	2-chloropyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
26-598	5-fluoropyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	C2F5
26-600	5-bromopyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	n-C3F7
26-601	5-iodopyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
26-605	4-fluoropyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	C2F5
26-609	4-(trifluoromethyl)pyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	n-C3F7
26-610	4-nitropyridin-3-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
26-626	4-cyanopyridin-2-yl	H	H	H	Cl	H	nonafluoro-2-butyl	H	C2F5
26-627	phenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-628	2-fluorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-629	3-fluorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-630	4-fluorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-631	2-chlorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-632	3-chlorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-633	4-chlorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-634	2-bromophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-635	3-bromophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-636	4-bromophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-637	2-iodophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-638	3-iodophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-639	4-iodophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-640	(2-trifluoromethyl)phenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-641	(3-trifluoromethyl)phenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-642	(4-trifluoromethyl)phenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-643	2-nitrophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-644	3-nitrophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-645	4-nitrophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-646	2-cyanophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-647	3-cyanophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-648	4-cyanophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-649	2,6-difluorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-650	3,4-dichlorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-651	2,4-dichlorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-652	2-chloro-4-fluorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-653	2-chloro-4,5-difluorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-654	4-bromo-2-chlorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-655	2-bromo-4-chlorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-656	2-bromo-4-fluorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-657	2-chloro-4-nitrophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-658	3,5-dicyanophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-659	4-cyano-2-fluorophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-660	2-chloro-4-cyanophenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-661	pyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-662	2-fluoropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-663	2-chloropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-664	2-bromopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-665	2-iodopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-666	2-(trifluoromethyl)pyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-667	2-nitropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-668	2-cyanopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-669	6-fluoropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-670	6-chloropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-671	6-bromopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-672	6-iodopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-673	6-(trifluoromethyl)pyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-674	6-nitropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-675	6-cyanopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-676	5-fluoropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-677	5-chloropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-678	5-bromopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-679	5-iodopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-680	5-(trifluoromethyl)pyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-681	5-nitropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-682	5-cyanopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-683	4-fluoropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-684	4-chloropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-685	4-bromopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-686	4-iodopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-687	4-(trifluoromethyl)pyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-688	4-nitropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-689	4-cyanopyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-690	2,6-dichloropyridin-3-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-691	pyridin-3-yl N-oxide	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-692	pyridin-4-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-693	2-chloropyridin-4-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-694	3-bromopyridin-4-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-695	3,5-dichloropyridin-4-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-696	3-(trifluoromethyl)pyridin-4-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-697	2,6-dicyanopyridin-4-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-698	pyridin-4-yl N-oxide	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-699	pyridin-2-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-700	3-chloropyridin-2-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-701	4-bromopyridin-2-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-702	5-iodopyridin-2-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-703	6-chloropyridin-2-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-704	4-cyanopyridin-2-yl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
26-705	phenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-706	2-fluorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-707	3-fluorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-708	4-fluorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-709	2-chlorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-710	3-chlorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-711	4-chlorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-712	2-bromophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-713	3-bromophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-714	4-bromophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-715	2-iodophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-716	3-iodophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-717	4-iodophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-718	(2-trifluoromethyl)phenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-719	(3-trifluoromethyl)phenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-720	(4-trifluoromethyl)phenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-721	2-nitrophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-722	3-nitrophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-723	4-nitrophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-724	2-cyanophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-725	3-cyanophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-726	4-cyanophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-727	2,6-difluorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-728	3,4-dichlorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-729	2,4-dichlorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-730	2-chloro-4-fluorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-731	2-chloro-4,5-difluorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-732	4-bromo-2-chlorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-733	2-bromo-4-chlorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-734	2-bromo-4-fluorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-735	2-chloro-4-nitrophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-736	3,5-dicyanophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-737	4-cyano-2-fluorophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-738	2-chloro-4-cyanophenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-739	pyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-740	2-fluoropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-741	2-chloropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-742	2-bromopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-743	2-iodopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-744	2-(trifluoromethyl)pyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-745	2-nitropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-746	2-cyanopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-747	6-fluoropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-748	6-chloropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-749	6-bromopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-750	6-iodopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-751	6-(trifluoromethyl)pyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-752	6-nitropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-753	6-cyanopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-754	5-fluoropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-755	5-chloropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-756	5-bromopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-757	5-iodopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-758	5-(trifluoromethyl)pyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-759	5-nitropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-760	5-cyanopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-761	4-fluoropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-762	4-chloropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-763	4-bromopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-764	4-iodopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-765	4-(trifluoromethyl)pyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-766	4-nitropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-767	4-cyanopyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-768	2,6-dichloropyridin-3-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-769	pyridin-3-yl N-oxide	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-770	pyridin-4-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-771	2-chloropyridin-4-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-772	3-bromopyridin-4-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-773	3,5-dichloropyridin-4-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-774	3-(trifluoromethyl)pyridin-4-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-775	2,6-dicyanopyridin-4-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-776	pyridin-4-yl N-oxide	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-777	pyridin-2-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-778	3-chloropyridin-2-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-779	4-bromopyridin-2-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-780	5-iodopyridin-2-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-781	6-chloropyridin-2-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-782	4-cyanopyridin-2-yl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
26-783	phenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-784	2-fluorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-785	3-fluorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-786	4-fluorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-787	2-chlorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-788	3-chlorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-789	4-chlorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-790	2-bromophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-791	3-bromophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-792	4-bromophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-793	2-iodophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-794	3-iodophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-795	4-iodophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-796	(2-trifluoromethyl)phenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-797	(3-trifluoromethyl)phenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-798	(4-trifluoromethyl)phenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-799	2-nitrophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-800	3-nitrophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-801	4-nitrophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-802	2-cyanophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-803	3-cyanophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-804	4-cyanophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-805	2,6-difluorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-806	3,4-dichlorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-807	2,4-dichlorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-808	2-chloro-4-fluorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-809	2-chloro-4,5-difluorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-810	4-bromo-2-chlorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-811	2-bromo-4-chlorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-812	2-bromo-4-fluorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-813	2-chloro-4-nitrophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-814	3,5-dicyanophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-815	4-cyano-2-fluorophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-816	2-chloro-4-cyanophenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-817	pyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-818	2-fluoropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-819	2-chloropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-820	2-bromopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-821	2-iodopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-822	2-(trifluoromethyl)pyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-823	2-nitropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-824	2-cyanopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-825	6-fluoropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-826	6-chloropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-827	6-bromopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-828	6-iodopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-829	6-(trifluoromethyl)pyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-830	6-nitropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-831	6-cyanopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-832	5-fluoropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-833	5-chloropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-834	5-bromopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-835	5-iodopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-836	5-(trifluoromethyl)pyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-837	5-nitropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-838	5-cyanopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-839	4-fluoropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-840	4-chloropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-841	4-bromopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-842	4-iodopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-843	4-(trifluoromethyl)pyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-844	4-nitropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-845	4-cyanopyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-846	2,6-dichloropyridin-3-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-847	pyridin-3-yl N-oxide	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-848	pyridin-4-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-849	2-chloropyridin-4-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-850	3-bromopyridin-4-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-851	3,5-dichloropyridin-4-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-852	3-(trifluoromethyl)pyridin-4-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-853	2,6-dicyanopyridin-4-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-854	pyridin-4-yl N-oxide	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-855	pyridin-2-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-856	3-chloropyridin-2-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-857	4-bromopyridin-2-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-858	5-iodopyridin-2-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-859	6-chloropyridin-2-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-860	4-cyanopyridin-2-yl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
26-861	phenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-862	2-fluorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-863	3-fluorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-864	4-fluorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-865	2-chlorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-866	3-chlorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-867	4-chlorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-868	2-bromophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-869	3-bromophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-870	4-bromophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-871	2-iodophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-872	3-iodophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-873	4-iodophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-874	(2-trifluoromethyl)phenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-875	(3-trifluoromethyl)phenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-876	(4-trifluoromethyl)phenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-877	2-nitrophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-878	3-nitrophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-879	4-nitrophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-880	2-cyanophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-881	3-cyanophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-882	4-cyanophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-883	2,6-difluorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-884	3,4-dichlorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-885	2,4-dichlorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-886	2-chloro-4-fluorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-887	2-chloro-4,5-difluorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-888	4-bromo-2-chlorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-889	2-bromo-4-chlorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-890	2-bromo-4-fluorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-891	2-chloro-4-nitrophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-892	3,5-dicyanophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-893	4-cyano-2-fluorophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-894	2-chloro-4-cyanophenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-895	pyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-896	2-fluoropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-897	2-chloropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-898	2-bromopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-899	2-iodopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-900	2-(trifluoromethyl)pyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-901	2-nitropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-902	2-cyanopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-903	6-fluoropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-904	6-chloropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-905	6-bromopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-906	6-iodopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-907	6-(trifluoromethyl)pyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-908	6-nitropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-909	6-cyanopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-910	5-fluoropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-911	5-chloropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-912	5-bromopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-913	5-iodopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-914	5-(trifluoromethyl)pyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-915	5-nitropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-916	5-cyanopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-917	4-fluoropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-918	4-chloropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-919	4-bromopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-920	4-iodopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-921	4-(trifluoromethyl)pyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-922	4-nitropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-923	4-cyanopyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-924	2,6-dichloropyridin-3-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-925	pyridin-3-yl N-oxide	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-926	pyridin-4-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-927	2-chloropyridin-4-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-928	3-bromopyridin-4-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-929	3,5-dichloropyridin-4-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-930	3-(trifluoromethyl)pyridin-4-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-931	2,6-dichloropyridin-4-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-932	pyridin-4-yl N-oxide	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-933	pyridin-2-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-934	3-chloropyridin-2-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-935	4-bromopyridin-2-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-936	5-iodopyridin-2-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-937	6-chloropyridin-2-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-938	4-cyanopyridin-2-yl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
26-939	phenyl	H	H	H	OCF3	H	heptafluoroisopropyl	H	OCF3
26-946	2-bromophenyl	H	H	H	OCF3	H	heptafluoroisopropyl	H	OC2F5
26-950	3-iodophenyl	H	H	H	OCF3	H	pentafluoroethyl	H	OCF3
26-951	4-iodophenyl	H	H	H	OCF3	H	pentafluoroethyl	H	OCF3
26-954	3-cyanophenyl	H	H	H	OCF3	H	heptafluoroisopropyl	H	OCF3
26-955	4-cyanophenyl	H	H	H	OCF3	H	heptafluoroisopropyl	H	OCF3
26-960	2-chloro-4,5-difluorophenyl	H	H	H	OC2F5	H	heptafluoroisopropyl	H	OC2F5
26-963	2-bromo-4-fluorophenyl	H	H	H	OC2F5	H	heptafluoroisopropyl	H	OCF3
26-964	2-chloro-4-nitrophenyl	H	H	Cl	OCF3	H	heptafluoroisopropyl	H	OCF3
26-969	2-fluoropyridin-3-yl	H	H	H	OCF3	H	pentafluoroethyl	H	OCF3
26-970	2-chloropyridin-3-yl	H	H	H	OCF3	H	heptafluoroisopropyl	H	OCF3
26-979	5-cyanopyridin-3-yl	H	H	H	OC2F5	H	heptafluoroisopropyl	H	OC2F5
26-981	4-cyanopyridin-3-yl	H	H	H	OCF3	H	heptafluoroisopropyl	H	OC2F5
26-994	4-cyanopyridin-2-yl	H	H	H	OCF3	H	pentafluoroethyl	H	OCF3
26-995	phenyl	H	H	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
26-1002	2-bromophenyl	H	H	H	OC2F5	H	nonafluoro-2-butyl	H	OCF3
26-1008	(2-trifluoromethyl)phenyl	H	H	H	OCF3	H	nonafluoro-2-butyl	H	OC2F5
26-1010	3-cyanophenyl	H	H	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
26-1011	4-cyanophenyl	H	H	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
26-1017	4-bromo-2-chlorophenyl	H	H	H	OC2F5	H	nonafluoro-2-butyl	H	OC2F5
26-1026	2-chloropyridin-3-yl	H	H	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
26-1033	6-cyanopyridin-3-yl	H	H	H	OC2F5	H	nonafluoro-2-butyl	H	OCF3
26-1035	5-cyanopyridin-3-yl	H	H	H	OCF3	H	nonafluoro-2-butyl	H	OC2F5
26-1037	4-cyanopyridin-3-yl	H	H	H	OC2F5	H	nonafluoro-2-butyl	H	OC2F5
26-1051	phenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	OCF3
26-1058	2-bromophenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	OC2F5
26-1062	3-iodophenyl	H	H	H	CF3	H	pentafluoroethyl	H	OCF3
26-1063	4-iodophenyl	H	H	H	CF3	H	pentafluoroethyl	H	OCF3
26-1064	(2-trifluoromethyl)phenyl	H	H	H	C2F5	H	heptafluoroisopropyl	H	OC2F5
26-1065	3-nitrophenyl	H	H	H	C2F5	H	heptafluoroisopropyl	H	OCF3
26-1066	3-cyanophenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	OCF3
26-1067	4-cyanophenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	OCF3
26-1074	2-bromo-4-chlorophenyl	H	H	H	n-C3F7	H	heptafluoroisopropyl	H	OCF3
26-1078	4-cyano-2-fluorophenyl	H	H	H	i-C3F7	H	heptafluoroisopropyl	H	OCF3
26-1081	2-fluoropyridin-3-yl	H	H	H	CF3	H	pentafluoroethyl	H	OCF3
26-1082	2-chloropyridin-3-yl	H	H	H	CF3	H	heptafluoroisopropyl	H	OCF3
26-1089	6-cyanopyridin-3-yl	H	H	H	n-C3F7	H	heptafluoroisopropyl	H	OC2F5
26-1091	5-cyanopyridin-3-yl	H	H	H	i-C3F7	H	heptafluoroisopropyl	H	OC2F5
26-1106	4-cyanopyridin-2-yl	H	H	H	CF3	H	pentafluoroethyl	H	OCF3
26-1107	phenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	OCF3
26-1118	3-iodophenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	OC2F5
26-1121	3-nitrophenyl	H	H	H	C2F5	H	nonafluoro-2-butyl	H	OCF3
26-1122	3-cyanophenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	OCF3
26-1123	4-cyanophenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	OCF3
26-1129	4-bromo-2-chlorophenyl	H	H	H	i-C3F7	H	nonafluoro-2-butyl	H	OCF3
26-1132	2-chloro-4-nitrophenyl	H	H	H	n-C3F7	H	nonafluoro-2-butyl	H	OCF3
26-1138	2-chloropyridin-3-yl	H	H	H	CF3	H	nonafluoro-2-butyl	H	OCF3
26-1147	5-cyanopyridin-3-yl	H	H	H	C2F5	H	nonafluoro-2-butyl	H	OC2F5
26-1149	4-cyanopyridin-3-yl	H	H	H	n-C3F7	H	nonafluoro-2-butyl	H	OC2F5
26-1160	5-iodopyridin-2-yl	H	H	H	i-C3F7	H	nonafluoro-2-butyl	H	OC2F5
26-1163	phenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
26-1174	3-iodophenyl	H	H	H	CF3	H	pentafluoroethyl	H	CF3
26-1175	4-iodophenyl	H	H	H	CF3	H	pentafluoroethyl	H	CF3
26-1177	(3-trifluoromethyl)phenyl	H	H	H	C2F5	H	heptafluoroisopropyl	H	CF3
26-1183	3-cyanophenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
26-1184	4-cyanophenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
26-1190	4-bromo-2-chlorophenyl	H	H	H	n-C3F7	H	heptafluoroisopropyl	H	CF3
26-1195	4-cyano-2-fluorophenyl	H	H	H	i-C3F7	H	heptafluoroisopropyl	H	CF3
26-1198	2-fluoropyridin-3-yl	H	H	H	CF3	H	pentafluoroethyl	H	CF3
26-1199	2-chloropyridin-3-yl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
26-1200	2-bromopyridin-3-yl	H	H	H	C2F5	H	heptafluoroisopropyl	H	C2F5
26-1203	2-nitropyridin-3-yl	H	H	Cl	CF3	H	heptafluoroisopropyl	H	CF3
26-1211	6-cyanopyridin-3-yl	H	H	H	C2F5	H	heptafluoroisopropyl	H	n-C3F7
26-1215	4-cyanopyridin-3-yl	H	H	H	C2F5	H	heptafluoroisopropyl	H	i-C3F7
26-1230	4-cyanopyridin-2-yl	H	H	H	CF3	H	pentafluoroethyl	H	CF3
26-1231	phenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
26-1243	4-iodophenyl	H	H	H	C2F5	H	nonafluoro-2-butyl	H	CF3
26-1251	3-cyanophenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
26-1252	4-cyanophenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
26-1258	4-bromo-2-chlorophenyl	H	H	H	n-C3F7	H	nonafluoro-2-butyl	H	CF3
26-1263	4-cyano-2-fluorophenyl	H	H	H	i-C3F7	H	nonafluoro-2-butyl	H	CF3
26-1267	2-chloropyridin-3-yl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
26-1268	2-bromopyridin-3-yl	H	H	H	C2F5	H	nonafluoro-2-butyl	H	C2F5
26-1279	6-cyanopyridin-3-yl	H	H	H	C2F5	H	nonafluoro-2-butyl	H	n-C3F7
26-1283	4-cyanopyridin-3-yl	H	H	H	C2F5	H	nonafluoro-2-butyl	H	i-C3F7

TABLE 27
compound
number	Q1	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
27-1	phenyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
27-21	3-cyanophenyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
27-22	4-cyanophenyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
27-37	2-chloropyridin-3-yl	Me	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
27-79	phenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
27-99	3-cyanophenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
27-100	4-cyanophenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
27-115	2-chloropyridin-3-yl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
27-157	phenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
27-177	3-cyanophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
27-178	4-cyanophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
27-193	2-chloropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
27-235	phenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
27-255	3-cyanophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
27-256	4-cyanophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
27-271	2-chloropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
27-313	phenyl	Me	H	H	I	H	heptafluoroisopropyl	H	OCF3
27-333	3-cyanophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	OCF3
27-334	4-cyanophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	OCF3
27-349	2-chloropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	OCF3
27-391	phenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	OCF3
27-411	3-cyanophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	OCF3
27-412	4-cyanophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	OCF3
27-427	2-chloropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	OCF3
27-469	phenyl	Me	H	H	F	H	heptafluoroisopropyl	H	CF3
27-470	phenyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	CF3
27-484	(3-trifluoromethyl)phenyl	Et	H	H	Cl	H	heptafluoroisopropyl	H	CF3
27-489	2-cyanophenyl	Me	H	H	Cl	H	pentafluoroethyl	H	C2F5
27-490	3-cyanophenyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	CF3
27-491	4-cyanophenyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	CF3
27-494	2,4-dichlorophenyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	C2F5
27-495	2-chloro-4-fluorophenyl	n-Pr	H	H	Cl	H	heptafluoroisopropyl	H	CF3
27-498	2-bromo-4-chlorophenyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
27-506	2-chloropyridin-3-yl	Me	H	H	Cl	H	heptafluoroisopropyl	H	CF3
27-510	2-nitropyridin-3-yl	Me	H	Cl	Cl	H	heptafluoroisopropyl	H	CF3
27-512	6-fluoropyridin-3-yl	i-Pr	H	H	Cl	H	heptafluoroisopropyl	H	CF3
27-519	5-fluoropyridin-3-yl	Me	H	H	Cl	H	heptafluoroisopropyl	H	C2F5
27-521	5-bromopyridin-3-yl	Me	H	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
27-522	5-iodopyridin-3-yl	Me	H	H	Cl	H	heptafluoroisopropyl	H	i-C3F7
27-528	4-bromopyridin-3-yl	CH2CH═CH2	H	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
27-529	4-iodopyridin-3-yl	Me	H	H	Cl	H	heptafluoroisopropyl	H	i-C3F7
27-535	pyridin-4-yl	CN	H	H	Cl	H	heptafluoroisopropyl	H	CF3
27-548	phenyl	Me	H	H	F	H	nonafluoro-2-butyl	H	CF3
27-549	phenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
27-557	3-bromophenyl	CH2C≡CH	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
27-562	(2-trifluoromethyl)phenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	C2F5
27-564	(4-trifluoromethyl)phenyl	NH2	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
27-569	3-cyanophenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
27-570	4-cyanophenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
27-577	2-bromo-4-chlorophenyl	C(O)OMe	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
27-579	2-chloro-4-nitrophenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
27-585	2-chloropyridin-3-yl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
27-598	5-fluoropyridin-3-yl	C(O)OEt	H	H	Cl	H	nonafluoro-2-butyl	H	C2F5
27-600	5-bromopyridin-3-yl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	n-C3F7
27-601	5-iodopyridin-3-yl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
27-605	4-fluoropyridin-3-yl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	C2F5
27-607	4-bromopyridin-3-yl	C(O)C(O)Me	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
27-609	4-(trifluoromethyl)pyridin-3-yl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	n-C3F7
27-610	4-nitropyridin-3-yl	C(O)C(O)Et	H	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
27-624	5-iodopyridin-2-yl	C(O)Me	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
27-626	4-cyanopyridin-2-yl	C(O)Et	H	H	Cl	H	nonafluoro-2-butyl	H	C2F5
27-627	phenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-628	2-fluorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-629	3-fluorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-630	4-fluorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-631	2-chlorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-632	3-chlorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-633	4-chlorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-634	2-bromophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-635	3-bromophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-636	4-bromophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-637	2-iodophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-638	3-iodophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-639	4-iodophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-640	(2-trifluoromethyl)phenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-641	(3-trifluoromethyl)phenyl	S(O)2Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-642	(4-trifluoromethyl)phenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-643	2-nitrophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-644	3-nitrophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-645	4-nitrophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-646	2-cyanophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-647	3-cyanophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-648	4-cyanophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-649	2,6-difluorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-650	3,4-dichlorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-651	2,4-dichlorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-652	2-chloro-4-fluorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-653	2-chloro-4,5-difluorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-654	4-bromo-2-chlorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-655	2-bromo-4-chlorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-656	2-bromo-4-fluorophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-657	2-chloro-4-nitrophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-658	3,5-dicyanophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-659	4-cyano-2-fluorophenyl	S(O)2Et	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-660	2-chloro-4-cyanophenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-661	pyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-662	2-fluoropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-663	2-chloropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-664	2-bromopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-665	2-iodopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-666	2-(trifluoromethyl)pyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-667	2-nitropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-668	2-cyanopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-669	6-fluoropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-670	6-chloropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-671	6-bromopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-672	6-iodopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-673	6-(trifluoromethyl)pyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-674	6-nitropyridin-3-yl	CH2Ph	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-675	6-cyanopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-676	5-fluoropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-677	5-chloropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-678	5-bromopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-679	5-iodopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-680	5-(trifluoromethyl)pyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-681	5-nitropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-682	5-cyanopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-683	4-fluoropyridin-3-yl	CH2(3-Py)	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-684	4-chloropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-685	4-bromopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-686	4-iodopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-687	4-(trifluoromethyl)pyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-688	4-nitropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-689	4-cyanopyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-690	2,6-dichloropyridin-3-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-691	pyridin-3-yl N-oxide	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-692	pyridin-4-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-693	2-chloropyridin-4-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-694	3-bromopyridin-4-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-695	3,5-dichloropyridin-4-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-696	3-(trifluoromethyl)pyridin-4-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-697	2,6-dicyanopyridin-4-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-698	pyridin-4-yl N-oxide	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-699	pyridin-2-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-700	3-chloropyridin-2-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-701	4-bromopyridin-2-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-702	5-iodopyridin-2-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-703	6-chloropyridin-2-yl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
27-704	4-cyanopyridin-2-yl	CH2(3-Py—N-	H	H	Br	H	heptafluoroisopropyl	H	CF3
		oxide)
27-705	phenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-706	2-fluorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-707	3-fluorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-708	4-fluorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-709	2-chlorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-710	3-chlorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-711	4-chlorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-712	2-bromophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-713	3-bromophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-714	4-bromophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-715	2-iodophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-716	3-iodophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-717	4-iodophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-718	(2-trifluoromethyl)phenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-719	(3-trifluoromethyl)phenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-720	(4-trifluoromethyl)phenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-721	2-nitrophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-722	3-nitrophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-723	4-nitrophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-724	2-cyanophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-725	3-cyanophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-726	4-cyanophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-727	2,6-difluorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-728	3,4-dichlorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-729	2,4-dichlorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-730	2-chloro-4-fluorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-731	2-chloro-4,5-difluorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-732	4-bromo-2-chlorophenyl	Et	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-733	2-bromo-4-chlorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-734	2-bromo-4-fluorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-735	2-chloro-4-nitrophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-736	3,5-dicyanophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-737	4-cyano-2-fluorophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-738	2-chloro-4-cyanophenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-739	pyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-740	2-fluoropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-741	2-chloropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-742	2-bromopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-743	2-iodopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-744	2-(trifluoromethyl)pyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-745	2-nitropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-746	2-cyanopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-747	6-fluoropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-748	6-chloropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-749	6-bromopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-750	6-iodopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-751	6-(trifluoromethyl)pyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-752	6-nitropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-753	6-cyanopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-754	5-fluoropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-755	5-chloropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-756	5-bromopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-757	5-iodopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-758	5-(trifluoromethyl)pyridin-3-yl	CN	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-759	5-nitropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-760	5-cyanopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-761	4-fluoropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-762	4-chloropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-763	4-bromopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-764	4-iodopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-765	4-(trifluoromethyl)pyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-766	4-nitropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-767	4-cyanopyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-768	2,6-dichloropyridin-3-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-769	pyridin-3-yl N-oxide	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-770	pyridin-4-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-771	2-chloropyridin-4-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-772	3-bromopyridin-4-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-773	3,5-dichloropyridin-4-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-774	3-(trifluoromethyl)pyridin-4-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-775	2,6-dicyanopyridin-4-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-776	pyridin-4-yl N-oxide	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-777	pyridin-2-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-778	3-chloropyridin-2-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-779	4-bromopyridin-2-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-780	5-iodopyridin-2-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-781	6-chloropyridin-2-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-782	4-cyanopyridin-2-yl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
27-783	phenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-784	2-fluorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-785	3-fluorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-786	4-fluorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-787	2-chlorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-788	3-chlorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-789	4-chlorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-790	2-bromophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-791	3-bromophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-792	4-bromophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-793	2-iodophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-794	3-iodophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-795	4-iodophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-796	(2-trifluoromethyl)phenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-797	(3-trifluoromethyl)phenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-798	(4-trifluoromethyl)phenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-799	2-nitrophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-800	3-nitrophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-801	4-nitrophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-802	2-cyanophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-803	3-cyanophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-804	4-cyanophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-805	2,6-difluorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-806	3,4-dichlorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-807	2,4-dichlorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-808	2-chloro-4-fluorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-809	2-chloro-4,5-difluorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-810	4-bromo-2-chlorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-811	2-bromo-4-chlorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-812	2-bromo-4-fluorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-813	2-chloro-4-nitrophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-814	3,5-dicyanophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-815	4-cyano-2-fluorophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-816	2-chloro-4-cyanophenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-817	pyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-818	2-fluoropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-819	2-chloropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-820	2-bromopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-821	2-iodopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-822	2-(trifluoromethyl)pyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-823	2-nitropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-824	2-cyanopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-825	6-fluoropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-826	6-chloropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-827	6-bromopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-828	6-iodopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-829	6-(trifluoromethyl)pyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-830	6-nitropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-831	6-cyanopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-832	5-fluoropyridin-3-yl	C(O)Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-833	5-chloropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-834	5-bromopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-835	5-iodopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-836	5-(trifluoromethyl)pyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-837	5-nitropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-838	5-cyanopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-839	4-fluoropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-840	4-chloropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-841	4-bromopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-842	4-iodopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-843	4-(trifluoromethyl)pyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-844	4-nitropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-845	4-cyanopyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-846	2,6-dichloropyridin-3-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-847	pyridin-3-yl N-oxide	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-848	pyridin-4-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-849	2-chloropyridin-4-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-850	3-bromopyridin-4-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-851	3,5-dichloropyridin-4-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-852	3-(trifluoromethyl)pyridin-4-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-853	2,6-dicyanopyridin-4-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-854	pyridin-4-yl N-oxide	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-855	pyridin-2-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-856	3-chloropyridin-2-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-857	4-bromopyridin-2-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-858	5-iodopyridin-2-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-859	6-chloropyridin-2-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-860	4-cyanopyridin-2-yl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
27-861	phenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-862	2-fluorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-863	3-fluorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-864	4-fluorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-865	2-chlorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-866	3-chlorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-867	4-chlorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-868	2-bromophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-869	3-bromophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-870	4-bromophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-871	2-iodophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-872	3-iodophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-873	4-iodophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-874	(2-trifluoromethyl)phenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-875	(3-trifluoromethyl)phenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-876	(4-trifluoromethyl)phenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-877	2-nitrophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-878	3-nitrophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-879	4-nitrophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-880	2-cyanophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-881	3-cyanophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-882	4-cyanophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-883	2,6-difluorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-884	3,4-dichlorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-885	2,4-dichlorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-886	2-chloro-4-fluorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-887	2-chloro-4,5-difluorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-888	4-bromo-2-chlorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-889	2-bromo-4-chlorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-890	2-bromo-4-fluorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-891	2-chloro-4-nitrophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-892	3,5-dicyanophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-893	4-cyano-2-fluorophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-894	2-chloro-4-cyanophenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-895	pyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-896	2-fluoropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-897	2-chloropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-898	2-bromopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-899	2-iodopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-900	2-(trifluoromethyl)pyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-901	2-nitropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-902	2-cyanopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-903	6-fluoropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-904	6-chloropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-905	6-bromopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-906	6-iodopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-907	6-(trifluoromethyl)pyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-908	6-nitropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-909	6-cyanopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-910	5-fluoropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-911	5-chloropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-912	5-bromopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-913	5-iodopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-914	5-(trifluoromethyl)pyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-915	5-nitropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-916	5-cyanopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-917	4-fluoropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-918	4-chloropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-919	4-bromopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-920	4-iodopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-921	4-(trifluoromethyl)pyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-922	4-nitropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-923	4-cyanopyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-924	2,6-dichloropyridin-3-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-925	pyridin-3-yl N-oxide	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-926	pyridin-4-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-927	2-chloropyridin-4-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-928	3-bromopyridin-4-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-929	3,5-dichloropyridin-4-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-930	3-(trifluoromethyl)pyridin-4-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-931	2,6-dicyanopyridin-4-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-932	pyridin-4-yl N-oxide	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-933	pyridin-2-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-934	3-chloropyridin-2-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-935	4-bromopyridin-2-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-936	5-iodopyridin-2-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-937	6-chloropyridin-2-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-938	4-cyanopyridin-2-yl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
27-939	phenyl	Me	H	H	OCF3	H	heptafluoroisopropyl	H	OCF3
27-970	2-chloropyridin-3-yl	Me	H	H	OCF3	H	heptafluoroisopropyl	H	OCF3
27-995	phenyl	Me	H	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
27-1026	2-chloropyridin-3-yl	Me	H	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
27-1051	phenyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	OCF3
27-1082	2-chloropyridin-3-yl	Me	H	H	CF3	H	heptafluoroisopropyl	H	OCF3
27-1107	phenyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	OCF3
27-1138	2-chloropyridin-3-yl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	OCF3
27-1163	phenyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
27-1183	3-cyanophenyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
27-1184	4-cyanophenyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
27-1199	2-chloropyridin-3-yl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
27-1231	phenyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
27-1251	3-cyanophenyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
27-1252	4-cyanophenyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
27-1267	2-chloropyridin-3-yl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3

TABLE 28
compound
number	Q1	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
28-1	phenyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
28-21	3-cyanophenyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
28-22	4-cyanophenyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
28-37	2-chloropyridin-3-yl	H	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
28-79	phenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
28-99	3-cyanophenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
28-100	4-cyanophenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
28-115	2-chloropyridin-3-yl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
28-157	phenyl	H	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
28-177	3-cyanophenyl	H	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
28-178	4-cyanophenyl	H	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
28-193	2-chloropyridin-3-yl	H	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
28-235	phenyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
28-255	3-cyanophenyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
28-256	4-cyanophenyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
28-271	2-chloropyridin-3-yl	H	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
28-313	phenyl	H	Me	H	I	H	heptafluoroisopropyl	H	OCF3
28-333	3-cyanophenyl	H	Me	H	I	H	heptafluoroisopropyl	H	OCF3
28-334	4-cyanophenyl	H	Me	H	I	H	heptafluoroisopropyl	H	OCF3
28-349	2-chloropyridin-3-yl	H	Me	H	I	H	heptafluoroisopropyl	H	OCF3
28-391	phenyl	H	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
28-411	3-cyanophenyl	H	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
28-412	4-cyanophenyl	H	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
28-427	2-chloropyridin-3-yl	H	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
28-469	phenyl	H	Me	H	F	H	heptafluoroisopropyl	H	CF3
28-470	phenyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
28-481	3-iodophenyl	H	Me	H	Cl	H	pentafluoroethyl	H	CF3
28-482	4-iodophenyl	H	Me	H	Cl	H	pentafluoroethyl	H	CF3
28-484	(3-trifluoromethyl)phenyl	H	Et	H	Cl	H	heptafluoroisopropyl	H	CF3
28-489	2-cyanophenyl	H	Me	H	Cl	H	pentafluoroethyl	H	C2F5
28-490	3-cyanophenyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
28-491	4-cyanophenyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
28-494	2,4-dichlorophenyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	C2F5
28-495	2-chloro-4-fluorophenyl	H	n-Pr	H	Cl	H	heptafluoroisopropyl	H	CF3
28-498	2-bromo-4-chlorophenyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
28-505	2-fluoropyridin-3-yl	H	Me	H	Cl	H	pentafluoroethyl	H	CF3
28-506	2-chloropyridin-3-yl	H	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
28-512	6-fluoropyridin-3-yl	H	i-Pr	H	Cl	H	heptafluoroisopropyl	H	CF3
28-519	5-fluoropyridin-3-yl	H	Me	H	Cl	H	heptafluoroisopropyl	H	C2F5
28-521	5-bromopyridin-3-yl	H	Me	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
28-522	5-iodopyridin-3-yl	H	Me	H	Cl	H	heptafluoroisopropyl	H	i-C3F7
28-524	5-nitropyridin-3-yl	H	Me	H	Cl	H	pentafluoroethyl	H	CF3
28-526	4-fluoropyridin-3-yl	H	Me	H	Cl	H	pentafluoroethyl	H	CF3
28-528	4-bromopyridin-3-yl	H	CH2CH═CH2	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
28-529	4-iodopyridin-3-yl	H	Me	H	Cl	H	heptafluoroisopropyl	H	i-C3F7
28-531	4-nitropyridin-3-yl	H	Me	Cl	Cl	H	heptafluoroisopropyl	H	CF3
28-535	pyridin-4-yl	H	CN	H	Cl	H	heptafluoroisopropyl	H	CF3
28-547	4-cyanopyridin-2-yl	H	Me	H	Cl	H	pentafluoroethyl	H	CF3
28-548	phenyl	H	Me	H	F	H	nonafluoro-2-butyl	H	CF3
28-549	phenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
28-557	3-bromophenyl	H	CH2C≡CH	H	Cl	H	nonafluoro-2-butyl	H	CF3
28-562	(2-trifluoromethyl)phenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	C2F5
28-564	(4-trifluoromethyl)phenyl	H	NH2	H	Cl	H	nonafluoro-2-butyl	H	CF3
28-569	3-cyanophenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
28-570	4-cyanophenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
28-577	2-bromo-4-chlorophenyl	H	C(O)OMe	H	Cl	H	nonafluoro-2-butyl	H	CF3
28-579	2-chloro-4-nitrophenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
28-585	2-chloropyridin-3-yl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
28-598	5-fluoropyridin-3-yl	H	C(O)OEt	H	Cl	H	nonafluoro-2-butyl	H	C2F5
28-600	5-bromopyridin-3-yl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	n-C3F7
28-601	5-iodopyridin-3-yl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
28-605	4-fluoropyridin-3-yl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	C2F5
28-607	4-bromopyridin-3-yl	H	C(O)C(O)Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
28-609	4-(trifluoromethyl)pyridin-3-yl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	n-C3F7
28-610	4-nitropyridin-3-yl	H	C(O)C(O)Et	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
28-624	5-iodopyridin-2-yl	H	C(O)Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
28-626	4-cyanopyridin-2-yl	H	C(O)Et	H	Cl	H	nonafluoro-2-butyl	H	C2F5
28-627	phenyl	H	Me	H	Br	H	heptafluoroisopropyl	H	CF3
28-628	2-fluorophenyl	H	Me	H	Br	H	heptafluoroisopropyl	H	CF3
28-641	(3-trifluoromethyl)phenyl	H	S(O)2Me	H	Br	H	heptafluoroisopropyl	H	CF3
28-647	3-cyanophenyl	H	Me	H	Br	H	heptafluoroisopropyl	H	CF3
28-648	4-cyanophenyl	H	Me	H	Br	H	heptafluoroisopropyl	H	CF3
28-659	4-cyano-2-fluorophenyl	H	S(O)2Et	H	Br	H	heptafluoroisopropyl	H	CF3
28-663	2-chloropyridin-3-yl	H	Me	H	Br	H	heptafluoroisopropyl	H	CF3
28-674	6-nitropyridin-3-yl	H	CH2Ph	H	Br	H	heptafluoroisopropyl	H	CF3
28-683	4-fluoropyridin-3-yl	H	CH2(3-Py)	H	Br	H	heptafluoroisopropyl	H	CF3
28-704	4-cyanopyridin-2-yl	H	CH2(3-Py—N-	H	Br	H	heptafluoroisopropyl	H	CF3
			oxide)
28-705	phenyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
28-706	2-fluorophenyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
28-725	3-cyanophenyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
28-726	4-cyanophenyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
28-732	4-bromo-2-chlorophenyl	H	Et	H	Br	H	nonafluoro-2-butyl	H	CF3
28-741	2-chloropyridin-3-yl	H	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
28-758	5-(trifluoromethyl)pyridin-3-yl	H	CN	H	Br	H	nonafluoro-2-butyl	H	CF3
28-783	phenyl	H	Me	H	I	H	heptafluoroisopropyl	H	CF3
28-784	2-fluorophenyl	H	Me	H	I	H	heptafluoroisopropyl	H	CF3
28-803	3-cyanophenyl	H	Me	H	I	H	heptafluoroisopropyl	H	CF3
28-804	4-cyanophenyl	H	Me	H	I	H	heptafluoroisopropyl	H	CF3
28-819	2-chloropyridin-3-yl	H	Me	H	I	H	heptafluoroisopropyl	H	CF3
28-832	5-fluoropyridin-3-yl	H	C(O)Me	H	I	H	heptafluoroisopropyl	H	CF3
28-861	phenyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
28-862	2-fluorophenyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
28-881	3-cyanophenyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
28-882	4-cyanophenyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
28-897	2-chloropyridin-3-yl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
28-939	phenyl	H	Me	H	OCF3	H	heptafluoroisopropyl	H	OCF3
28-970	2-chloropyridin-3-yl	H	Me	H	OCF3	H	heptafluoroisopropyl	H	OCF3
28-995	phenyl	H	Me	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
28-1026	2-chloropyridin-3-yl	H	Me	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
28-1051	phenyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	OCF3
28-1082	2-chloropyridin-3-yl	H	Me	H	CF3	H	heptafluoroisopropyl	H	OCF3
28-1107	phenyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	OCF3
28-1138	2-chloropyridin-3-yl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	OCF3
28-1163	phenyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
28-1183	3-cyanophenyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
28-1184	4-cyanophenyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
28-1199	2-chloropyridin-3-yl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
28-1231	phenyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
28-1251	3-cyanophenyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
28-1252	4-cyanophenyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
28-1267	2-chloropyridin-3-yl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3

TABLE 29
compound
number	Q1	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
29-1	phenyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
29-21	3-cyanophenyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
29-22	4-cyanophenyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
29-37	2-chloropyridin-3-yl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
29-79	phenyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
29-99	3-cyanophenyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
29-100	4-cyanophenyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
29-115	2-chloropyridin-3-yl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
29-157	phenyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
29-177	3-cyanophenyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
29-178	4-cyanophenyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
29-193	2-chloropyridin-3-yl	Me	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
29-235	phenyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
29-255	3-cyanophenyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
29-256	4-cyanophenyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
29-271	2-chloropyridin-3-yl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
29-313	phenyl	Me	Me	H	I	H	heptafluoroisopropyl	H	OCF3
29-333	3-cyanophenyl	Me	Me	H	I	H	heptafluoroisopropyl	H	OCF3
29-334	4-cyanophenyl	Me	Me	H	I	H	heptafluoroisopropyl	H	OCF3
29-349	2-chloropyridin-3-yl	Me	Me	H	I	H	heptafluoroisopropyl	H	OCF3
29-391	phenyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
29-411	3-cyanophenyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
29-412	4-cyanophenyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
29-427	2-chloropyridin-3-yl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
29-665	phenyl	Me	Me	H	F	H	heptafluoroisopropyl	H	CF3
29-666	phenyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
29-677	3-iodophenyl	Me	Me	H	Cl	H	pentafluoroethyl	H	CF3
29-678	4-iodophenyl	Me	Et	H	Cl	H	pentafluoroethyl	H	CF3
29-680	(3-trifluoromethyl)phenyl	Et	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
29-682	2-nitrophenyl	Me	Me	Cl	Cl	H	heptafluoroisopropyl	H	CF3
29-685	2-cyanophenyl	Me	Me	H	Cl	H	pentafluoroethyl	H	C2F5
29-686	3-cyanophenyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
29-687	4-cyanophenyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
29-689	3,4-dichlorophenyl	Me	n-Pr	H	Cl	H	heptafluoroisopropyl	H	CF3
29-690	2,4-dichlorophenyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	C2F5
29-691	2-chloro-4-fluorophenyl	n-Pr	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
29-694	2-bromo-4-chlorophenyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
29-701	2-fluoropyridin-3-yl	Me	Me	H	Cl	H	pentafluoroethyl	H	CF3
29-702	2-chloropyridin-3-yl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
29-706	2-nitropyridin-3-yl	Me	i-Pr	H	Cl	H	heptafluoroisopropyl	H	CF3
29-708	6-fluoropyridin-3-yl	i-Pr	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
29-715	5-fluoropyridin-3-yl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	C2F5
29-717	5-bromopyridin-3-yl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
29-718	5-iodopyridin-3-yl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	i-C3F7
29-720	5-nitropyridin-3-yl	Me	Me	H	Cl	H	pentafluoroethyl	H	CF3
29-722	4-fluoropyridin-3-yl	Me	CH2CH═CH2	H	Cl	H	pentafluoroethyl	H	CF3
29-724	4-bromopyridin-3-yl	CH2CH═CH2	Me	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
29-725	4-iodopyridin-3-yl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	i-C3F7
29-729	2,6-dichloropyridin-3-yl	Me	CN	H	Cl	H	heptafluoroisopropyl	H	CF3
29-731	pyridin-4-yl	CN	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
29-743	4-cyanopyridin-2-yl	Me	Me	H	Cl	H	pentafluoroethyl	H	CF3
29-744	phenyl	Me	Me	H	F	H	nonafluoro-2-butyl	H	CF3
29-745	phenyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-751	4-chlorophenyl	Me	CH2C≡CH	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-753	3-bromophenyl	CH2C≡CH	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-758	(2-trifluoromethyl)phenyl	Me	NH2	H	Cl	H	nonafluoro-2-butyl	H	C2F5
29-760	(4-trifluoromethyl)phenyl	NH2	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-765	3-cyanophenyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-766	4-cyanophenyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-771	2-chloro-4,5-difluorophenyl	Me	C(O)OMe	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-773	2-bromo-4-chlorophenyl	C(O)OMe	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-775	2-chloro-4-nitrophenyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
29-781	2-chloropyridin-3-yl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-792	6-nitropyridin-3-yl	Me	C(O)OEt	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-794	5-fluoropyridin-3-yl	C(O)OEt	Me	H	Cl	H	nonafluoro-2-butyl	H	C2F5
29-796	5-bromopyridin-3-yl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	n-C3F7
29-797	5-iodopyridin-3-yl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
29-801	4-fluoropyridin-3-yl	Me	C(O)C(O)Me	H	Cl	H	nonafluoro-2-butyl	H	C2F5
29-803	4-bromopyridin-3-yl	C(O)C(O)Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-804	4-iodopyridin-3-yl	Me	C(O)C(O)Et	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-805	4-(trifluoromethyl)pyridin-3-yl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	n-C3F7
29-806	4-nitropyridin-3-yl	C(O)C(O)Et	Me	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
29-818	3-chloropyridin-2-yl	Me	C(O)Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-820	5-iodopyridin-2-yl	C(O)Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-821	6-chloropyridin-2-yl	Me	C(O)Et	H	Cl	H	nonafluoro-2-butyl	H	CF3
29-822	4-cyanopyridin-2-yl	C(O)Et	Me	H	Cl	H	nonafluoro-2-butyl	H	C2F5
29-823	phenyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
29-824	2-fluorophenyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
29-835	4-iodophenyl	Me	S(O)2Me	H	Br	H	heptafluoroisopropyl	H	CF3
29-837	(3-trifluoromethyl)phenyl	S(O)2Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
29-843	3-cyanophenyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
29-844	4-cyanophenyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
29-853	2-chloro-4-nitrophenyl	Me	S(O)2Et	H	Br	H	heptafluoroisopropyl	H	CF3
29-855	4-cyano-2-fluorophenyl	S(O)2Et	Me	H	Br	H	heptafluoroisopropyl	H	CF3
29-859	2-chloropyridin-3-yl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
29-868	6-iodopyridin-3-yl	Me	CH2Ph	H	Br	H	heptafluoroisopropyl	H	CF3
29-870	6-nitropyridin-3-yl	CH2Ph	Me	H	Br	H	heptafluoroisopropyl	H	CF3
29-877	5-nitropyridin-3-yl	Me	CH2(3-Py)	H	Br	H	heptafluoroisopropyl	H	CF3
29-879	4-fluoropyridin-3-yl	CH2(3-Py)	Me	H	Br	H	heptafluoroisopropyl	H	CF3
29-898	5-iodopyridin-2-yl	Me	CH2(3-Py—N-	H	Br	H	heptafluoroisopropyl	H	CF3
			oxide)
29-900	4-cyanopyridin-2-yl	CH2(3-Py—N-	Me	H	Br	H	heptafluoroisopropyl	H	CF3
		oxide)
29-901	phenyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
29-902	2-fluorophenyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
29-921	3-cyanophenyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
29-922	4-cyanophenyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
29-926	2-chloro-4-fluorophenyl	Me	Et	H	Br	H	nonafluoro-2-butyl	H	CF3
29-928	4-bromo-2-chlorophenyl	Et	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
29-937	2-chloropyridin-3-yl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
29-952	5-bromopyridin-3-yl	Me	CN	H	Br	H	nonafluoro-2-butyl	H	CF3
29-954	5-(trifluoromethyl)pyridin-3-yl	CN	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
29-979	phenyl	Me	Me	H	I	H	heptafluoroisopropyl	H	CF3
29-980	2-fluorophenyl	Me	Me	H	I	H	heptafluoroisopropyl	H	CF3
29-999	3-cyanophenyl	Me	Me	H	I	H	heptafluoroisopropyl	H	CF3
29-1000	4-cyanophenyl	Me	Me	H	I	H	heptafluoroisopropyl	H	CF3
29-1015	2-chloropyridin-3-yl	Me	Me	H	I	H	heptafluoroisopropyl	H	CF3
29-1026	6-nitropyridin-3-yl	Me	C(O)Me	H	I	H	heptafluoroisopropyl	H	CF3
29-1028	5-fluoropyridin-3-yl	C(O)Me	Me	H	I	H	heptafluoroisopropyl	H	CF3
29-1057	phenyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	CF3
29-1058	2-fluorophenyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	CF3
29-1077	3-cyanophenyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	CF3
29-1078	4-cyanophenyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	CF3
29-1093	2-chloropyridin-3-yl	Me	Me	H	I	H	nonafluoro-2-butyl	H	CF3
29-1331	phenyl	Me	Me	H	OCF3	H	heptafluoroisopropyl	H	OCF3
29-1362	2-chloropyridin-3-yl	Me	Me	H	OCF3	H	heptafluoroisopropyl	H	OCF3
29-1387	phenyl	Me	Me	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
29-1418	2-chloropyridin-3-yl	Me	Me	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
29-1443	phenyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	OCF3
29-1474	2-chloropyridin-3-yl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	OCF3
29-1499	phenyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	OCF3
29-1530	2-chloropyridin-3-yl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	OCF3
29-1555	phenyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
29-1575	3-cyanophenyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
29-1576	4-cyanophenyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
29-1591	2-chloropyridin-3-yl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
29-1623	phenyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
29-1643	3-cyanophenyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
29-1644	4-cyanophenyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
29-1659	2-chloropyridin-3-yl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3

TABLE 30
compound
number	Q1	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
30-9	3-bromophenyl	H	Et	H	Cl	F	heptafluoroisopropyl	F	OCF3
30-39	2-iodopyridin-3-yl	H	H	H	Cl	Me	nonafluoro-2-butyl	Me	OCF3
30-144	phenyl	H	H	H	Cl	F	heptafluoroisopropyl	H	CF3
30-154	2-iodophenyl	H	H	H	Cl	F	heptafluoroisopropyl	Br	CF3
30-161	3-nitrophenyl	H	H	H	Cl	Br	heptafluoroisopropyl	Cl	CF3
30-168	2,4-dichlorophenyl	H	H	H	Cl	Me	nonafluoro-2-butyl	H	CF3
30-182	2-iodopyridin-3-yl	H	H	H	Cl	Me	nonafluoro-2-butyl	Me	n-C3F7
30-183	2-(trifluoromethyl)pyridin-3-yl	H	H	H	Cl	Me	nonafluoro-2-butyl	Et	i-C3F7
30-189	6-iodopyridin-3-yl	H	H	H	Cl	Et	nonafluoro-2-butyl	Me	n-C3F7
30-190	6-(trifluoromethyl)pyridin-3-yl	H	H	H	Cl	Et	nonafluoro-2-butyl	Et	i-C3F7
30-196	5-bromopyridin-3-yl	H	H	H	Br	n-Pr	heptafluoroisopropyl	Me	CF3
30-197	5-iodopyridin-3-yl	H	H	H	Br	n-Pr	heptafluoroisopropyl	Et	CF3
30-203	4-bromopyridin-3-yl	Me	n-Pr	H	Br	i-Pr	heptafluoroisopropyl	Me	CF3
30-204	4-iodopyridin-3-yl	H	H	H	Br	i-Pr	heptafluoroisopropyl	Et	CF3
30-210	pyridin-4-yl	H	H	H	Br	n-Bu	heptafluoroisopropyl	Me	CF3
30-211	2-chloropyridin-4-yl	H	H	H	Br	n-Bu	heptafluoroisopropyl	Et	CF3
30-217	pyridin-2-yl	H	H	H	Br	i-Bu	nonafluoro-2-butyl	Me	CF3
30-218	3-chloropyridin-2-yl	H	H	H	Br	i-Bu	nonafluoro-2-butyl	Et	CF3
30-224	2-fluorophenyl	H	H	H	Br	s-Bu	nonafluoro-2-butyl	Me	CF3
30-225	3-fluorophenyl	H	H	H	Br	s-Bu	nonafluoro-2-butyl	Et	CF3
30-231	3-bromophenyl	H	H	H	Br	F	nonafluoro-2-butyl	Me	CF3
30-232	4-bromophenyl	H	H	H	Br	F	nonafluoro-2-butyl	Et	CF3
30-238	(4-trifluoromethyl)phenyl	Et	i-Pr	H	Br	Cl	nonafluoro-2-butyl	Me	CF3
30-239	2-nitrophenyl	H	H	H	Br	Cl	nonafluoro-2-butyl	Et	CF3
30-245	4-cyanophenyl	H	H	H	I	Br	heptafluoroisopropyl	Me	CF3
30-246	2,6-difluorophenyl	H	H	H	I	Br	heptafluoroisopropyl	Et	CF3
30-252	2-bromo-4-chlorophenyl	n-Pr	Me	H	I	I	heptafluoroisopropyl	Me	CF3
30-253	2-bromo-4-fluorophenyl	H	H	H	I	I	heptafluoroisopropyl	Et	CF3
30-259	2-fluoropyridin-3-yl	H	H	H	I	Me	heptafluoroisopropyl	F	C2F5
30-260	2-chloropyridin-3-yl	H	H	H	I	Me	nonafluoro-2-butyl	Cl	CF3
30-263	2-(trifluoromethyl)pyridin-3-yl	H	H	H	I	Et	nonafluoro-2-butyl	F	CF3
30-264	2-nitropyridin-3-yl	H	H	H	I	Et	nonafluoro-2-butyl	Cl	CF3
30-267	6-chloropyridin-3-yl	H	H	H	I	n-Pr	nonafluoro-2-butyl	F	CF3
30-268	6-bromopyridin-3-yl	H	H	H	I	n-Pr	nonafluoro-2-butyl	Cl	CF3
30-271	6-nitropyridin-3-yl	H	H	H	I	i-Pr	nonafluoro-2-butyl	F	i-C3F7
30-272	6-cyanopyridin-3-yl	H	H	H	I	i-Pr	nonafluoro-2-butyl	Cl	CF3
30-275	5-bromopyridin-3-yl	H	H	H	I	n-Bu	nonafluoro-2-butyl	F	CF3
30-276	5-iodopyridin-3-yl	H	H	H	I	n-Bu	nonafluoro-2-butyl	Cl	CF3
30-279	5-cyanopyridin-3-yl	H	H	H	I	i-Bu	nonafluoro-2-butyl	F	CF3
30-280	4-fluoropyridin-3-yl	H	H	H	I	i-Bu	nonafluoro-2-butyl	Cl	CF3
30-283	4-iodopyridin-3-yl	i-Pr	n-Pr	H	I	s-Bu	nonafluoro-2-butyl	F	CF3
30-284	4-(trifluoromethyl)pyridin-3-yl	H	H	H	I	s-Bu	nonafluoro-2-butyl	Cl	CF3
30-295	3-bromophenyl	H	Et	H	OCF3	F	heptafluoroisopropyl	F	OCF3
30-325	2-iodopyridin-3-yl	H	H	H	OCF3	Me	nonafluoro-2-butyl	Me	OCF3
30-438	3-bromophenyl	H	Et	H	OCF3	F	heptafluoroisopropyl	F	CF3
30-468	2-iodopyridin-3-yl	H	H	H	OCF3	Me	nonafluoro-2-butyl	Me	CF3
30-581	3-bromophenyl	H	Et	H	CF3	F	heptafluoroisopropyl	F	CF3
30-611	2-iodopyridin-3-yl	H	H	H	CF3	Me	nonafluoro-2-butyl	Me	CF3

TABLE 31
compound
number	Q2	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
31-1	2,2,2-trichloroethyl	H	H	H	F	H	heptafluoroisopropyl	H	OCF3
31-2	2,2,2-trichloroethyl	H	H	H	F	H	nonafluoro-2-butyl	H	OCF3
31-9	2-chloroethyl	H	H	Cl	Cl	H	heptafluoroisopropyl	H	OCF3
31-13	2,2,2-trichloroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
31-16	3-fluoro-n-propyl	H	H	H	Cl	H	pentafluoroethyl	H	OCF3
31-18	3-bromo-n-propyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OC2F5
31-22	1,3-dichloro-2-propyl	H	H	H	Cl	H	pentafluoroethyl	H	OC2F5
31-26	4,4,4-trifluoro-n-butyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
31-36	2-bromoethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OC2F5
31-42	2,2,2-trichloroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
31-55	4,4,4-trifluoro-n-butyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
31-57	s-butyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OC2F5
31-66	2-iodoethyl	H	H	H	Br	H	heptafluoroisopropyl	H	OC2F5
31-71	2,2,2-trichloroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	OCF3
31-84	4,4,4-trifluoro-n-butyl	H	H	H	Br	H	heptafluoroisopropyl	H	OCF3
31-100	2,2,2-trichloroethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
31-102	n-propyl	H	H	H	Br	H	nonafluoro-2-butyl	H	OC2F5
31-113	4,4,4-trifluoro-n-butyl	H	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
31-129	2,2,2-trichloroethyl	H	H	H	I	H	heptafluoroisopropyl	H	OCF3
31-133	3-chloro-n-propyl	H	H	H	I	H	heptafluoroisopropyl	H	OC2F5
31-142	4,4,4-trifluoro-n-butyl	H	H	H	I	H	heptafluoroisopropyl	H	OCF3
31-158	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
31-171	4,4,4-trifluoro-n-butyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
31-175	benzyl	H	H	H	I	H	nonafluoro-2-butyl	H	OC2F5
31-177	2,2,2-trichloroethyl	H	H	H	F	H	heptafluoroisopropyl	H	CF3
31-178	2,2,2-trichloroethyl	H	H	H	F	H	nonafluoro-2-butyl	H	CF3
31-179	methyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-180	ethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-181	2-fluoroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-182	2-chloroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-183	2-bromoethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-184	2-iodoethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-185	2-cyanoethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	C2F5
31-186	2,2-difluoroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-187	2,2-dichloroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-188	2,2,2-trifluoroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-189	2,2,2-trichloroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-190	2,2,2-tribromoethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-191	n-propyl	H	H	H	Cl	H	pentafluoroethyl	H	CF3
31-192	3-fluoro-n-propyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-193	3-chloro-n-propyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-194	3-bromo-n-propyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-195	i-propyl	H	H	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
31-196	1,2-difluoro-2-propyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-197	1,3-difluoro-2-propyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-198	1,3-dichloro-2-propyl	H	H	H	Cl	H	pentafluoroethyl	H	CF3
31-199	1-chloro-3-fluoro-2-propyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-200	3,3,3-trifluoro-n-propyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-201	n-butyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-202	4,4,4-trifluoro-n-butyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-203	i-butyl	H	H	Cl	Cl	H	heptafluoroisopropyl	H	CF3
31-204	s-butyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-205	vinyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-206	benzyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-207	phenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
31-208	methyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-209	ethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
31-210	2-fluoroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-211	2-chloroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-212	2-bromoethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-213	2-iodoethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-214	2-cyanoethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-215	2,2-difluoroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-216	2,2-dichloroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-217	2,2,2-trifluoroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-218	2,2,2-trichloroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-219	2,2,2-tribromoethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-220	n-propyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-221	3-fluoro-n-propyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-222	3-chloro-n-propyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-223	3-bromo-n-propyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-224	i-propyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-225	1,2-difluoro-2-propyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-226	1,3-difluoro-2-propyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-227	1,3-dichloro-2-propyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-228	1-chloro-3-fluoro-2-propyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-229	3,3,3-trifluoro-n-propyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-230	n-butyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-231	4,4,4-trifluoro-n-butyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-232	i-butyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-233	s-butyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-234	vinyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-235	benzyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-236	phenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
31-237	methyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-238	ethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-239	2-fluoroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-240	2-chloroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-241	2-bromoethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-242	2-iodoethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-243	2-cyanoethyl	H	H	H	Br	H	heptafluoroisopropyl	H	C2F5
31-244	2,2-difluoroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-245	2,2-dichloroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-246	2,2,2-trifluoroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-247	2,2,2-trichloroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-248	2,2,2-tribromoethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-249	n-propyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-250	3-fluoro-n-propyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-251	3-chloro-n-propyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-252	3-bromo-n-propyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-253	i-propyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-254	1,2-difluoro-2-propyl	H	H	H	Br	H	heptafluoroisopropyl	H	n-C3F7
31-255	1,3-difluoro-2-propyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-256	1,3-dichloro-2-propyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-257	1-chloro-3-fluoro-2-propyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-258	3,3,3-trifluoro-n-propyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-259	n-butyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-260	4,4,4-trifluoro-n-butyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-261	i-butyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-262	s-butyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-263	vinyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-264	benzyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-265	phenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
31-266	methyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-267	ethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-268	2-fluoroethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-269	2-chloroethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-270	2-bromoethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-271	2-iodoethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-272	2-cyanoethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-273	2,2-difluoroethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-274	2,2-dichloroethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-275	2,2,2-trifluoroethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-276	2,2,2-trichloroethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-277	2,2,2-tribromoethyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-278	n-propyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-279	3-fluoro-n-propyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-280	3-chloro-n-propyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-281	3-bromo-n-propyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-282	i-propyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-283	1,2-difluoro-2-propyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-284	1,3-difluoro-2-propyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-285	1,3-dichloro-2-propyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-286	1-chloro-3-fluoro-2-propyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-287	3,3,3-trifluoro-n-propyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-288	n-butyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-289	4,4,4-trifluoro-n-butyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-290	i-butyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-291	s-butyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-292	vinyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-293	benzyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
31-294	phenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	i-C3F7
31-295	methyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-296	ethyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-297	2-fluoroethyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-298	2-chloroethyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-299	2-bromoethyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-300	2-iodoethyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-301	2-cyanoethyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-302	2,2-difluoroethyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-303	2,2-dichloroethyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-304	2,2,2-trifluoroethyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-305	2,2,2-trichloroethyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-306	2,2,2-tribromoethyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-307	n-propyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-308	3-fluoro-n-propyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-309	3-chloro-n-propyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-310	3-bromo-n-propyl	H	H	H	I	H	heptafluoroisopropyl	H	C2F5
31-311	i-propyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-312	1,2-difluoro-2-propyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-313	1,3-difluoro-2-propyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-314	1,3-dichloro-2-propyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-315	1-chloro-3-fluoro-2-propyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-316	3,3,3-trifluoro-n-propyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-317	n-butyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-318	4,4,4-trifluoro-n-butyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-319	i-butyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-320	s-butyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-321	vinyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-322	benzyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-323	phenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
31-324	methyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-325	ethyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-326	2-fluoroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-327	2-chloroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-328	2-bromoethyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-329	2-iodoethyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-330	2-cyanoethyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-331	2,2-difluoroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-332	2,2-dichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-333	2,2,2-trifluoroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-334	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-335	2,2,2-tribromoethyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-336	n-propyl	H	H	H	I	H	nonafluoro-2-butyl	H	n-C3F7
31-337	3-fluoro-n-propyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-338	3-chloro-n-propyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-339	3-bromo-n-propyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-340	i-propyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-341	1,2-difluoro-2-propyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-342	1,3-difluoro-2-propyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-343	1,3-dichloro-2-propyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-344	1-chloro-3-fluoro-2-propyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-345	3,3,3-trifluoro-n-propyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-346	n-butyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-347	4,4,4-trifluoro-n-butyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-348	i-butyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-349	s-butyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-350	vinyl	H	H	H	I	H	nonafluoro-2-butyl	H	i-C3F7
31-351	benzyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-352	phenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
31-359	2-cyanoethyl	H	H	H	OCF3	H	heptafluoroisopropyl	H	OC2F5
31-363	2,2,2-trichloroethyl	H	H	H	OCF3	H	heptafluoroisopropyl	H	OCF3
31-364	2,2,2-tribromoethyl	H	H	H	OCF3	H	pentafluoroethyl	H	OCF3
31-373	1-chloro-3-fluoro-2-propyl	H	H	H	OC2F5	H	heptafluoroisopropyl	H	OC2F5
31-376	4,4,4-trifluoro-n-butyl	H	H	H	OCF3	H	heptafluoroisopropyl	H	OCF3
31-378	s-butyl	H	H	H	OC2F5	H	heptafluoroisopropyl	H	OCF3
31-391	2,2,2-trifluoroethyl	H	H	H	OC2F5	H	nonafluoro-2-butyl	H	OCF3
31-392	2,2,2-trichloroethyl	H	H	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
31-394	n-propyl	H	H	Cl	OCF3	H	nonafluoro-2-butyl	H	OC2F5
31-403	3,3,3-trifluoro-n-propyl	H	H	H	OC2F5	H	nonafluoro-2-butyl	H	OC2F5
31-405	4,4,4-trifluoro-n-butyl	H	H	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
31-417	2-cyanoethyl	H	H	H	CF3	H	heptafluoroisopropyl	H	OC2F5
31-421	2,2,2-trichloroethyl	H	H	H	CF3	H	heptafluoroisopropyl	H	OCF3
31-423	n-propyl	H	H	H	C2F5	H	heptafluoroisopropyl	H	OC2F5
31-427	i-propyl	H	H	H	CF3	H	pentafluoroethyl	H	OCF3
31-432	3,3,3-trifluoro-n-propyl	H	H	Cl	n-C3F7	H	heptafluoroisopropyl	H	OCF3
31-434	4,4,4-trifluoro-n-butyl	H	H	H	CF3	H	heptafluoroisopropyl	H	OCF3
31-437	vinyl	H	H	H	i-C3F7	H	heptafluoroisopropyl	H	OCF3
31-445	2-iodoethyl	H	H	H	C2F5	H	nonafluoro-2-butyl	H	OCF3
31-450	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	OCF3
31-452	n-propyl	H	H	H	n-C3F7	H	nonafluoro-2-butyl	H	OCF3
31-456	i-propyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	OC2F5
31-463	4,4,4-trifluoro-n-butyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	OCF3
31-464	i-butyl	H	H	H	i-C3F7	H	nonafluoro-2-butyl	H	OCF3
31-467	benzyl	H	H	H	n-C3F7	H	nonafluoro-2-butyl	H	OC2F5
31-468	phenyl	H	H	H	i-C3F7	H	nonafluoro-2-butyl	H	OC2F5
31-479	2,2,2-trichloroethyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
31-482	3-fluoro-n-propyl	H	H	H	C2F5	H	heptafluoroisopropyl	H	CF3
31-485	i-propyl	H	H	H	i-C3F7	H	heptafluoroisopropyl	H	CF3
31-487	1,3-difluoro-2-propyl	H	H	H	CF3	H	pentafluoroethyl	H	CF3
31-490	3,3,3-trifluoro-n-propyl	H	H	H	C2F5	H	heptafluoroisopropyl	H	C2F5
31-492	4,4,4-trifluoro-n-butyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
31-493	i-butyl	H	H	H	C2F5	H	heptafluoroisopropyl	H	n-C3F7
31-495	vinyl	H	H	H	n-C3F7	H	heptafluoroisopropyl	H	CF3
31-508	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
31-520	n-butyl	H	H	H	C2F5	H	nonafluoro-2-butyl	H	i-C3F7
31-521	4,4,4-trifluoro-n-butyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
31-522	i-butyl	H	H	Cl	CF3	H	nonafluoro-2-butyl	H	CF3
31-524	vinyl	H	H	H	n-C3F7	H	nonafluoro-2-butyl	H	i-C3F7

TABLE 32
compound
number	Q2	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
32-1	2,2,2-trichloroethyl	Me	H	H	F	H	heptafluoroisopropyl	H	OCF3
32-2	2,2,2-trichloroethyl	Me	H	H	F	H	nonafluoro-2-butyl	H	OCF3
32-13	2,2,2-trichloroethyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
32-42	2,2,2-trichloroethyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
32-71	2,2,2-trichloroethyl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
32-100	2,2,2-trichloroethyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
32-129	2,2,2-trichloroethyl	Me	H	H	I	H	heptafluoroisopropyl	H	OCF3
32-158	2,2,2-trichloroethyl	Me	H	H	I	H	nonafluoro-2-butyl	H	OCF3
32-177	2,2,2-trichloroethyl	Me	H	H	F	H	heptafluoroisopropyl	H	CF3
32-178	2,2,2-trichloroethyl	Me	H	H	F	H	nonafluoro-2-butyl	H	CF3
32-185	2-cyanoethyl	Et	H	H	Cl	H	heptafluoroisopropyl	H	C2F5
32-189	2,2,2-trichloroethyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	CF3
32-191	n-propyl	Me	H	H	Cl	H	pentafluoroethyl	H	CF3
32-195	i-propyl	n-Pr	H	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
32-198	1,3-dichloro-2-propyl	Me	H	H	Cl	H	pentafluoroethyl	H	CF3
32-199	1-chloro-3-fluoro-2-propyl	i-Pr	H	H	Cl	H	heptafluoroisopropyl	H	CF3
32-202	4,4,4-trifluoro-n-butyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	CF3
32-203	i-butyl	CH2CH═CH2	H	H	Cl	H	heptafluoroisopropyl	H	CF3
32-207	phenyl	Me	H	Cl	Cl	H	heptafluoroisopropyl	H	CF3
32-209	ethyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
32-214	2-cyanoethyl	CN	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
32-218	2,2,2-trichloroethyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
32-220	n-propyl	CH2C≡CH	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
32-231	4,4,4-trifluoro-n-butyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
32-232	i-butyl	NH2	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
32-243	2-cyanoethyl	Me	H	H	Br	H	heptafluoroisopropyl	H	C2F5
32-247	2,2,2-trichloroethyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
32-249	n-propyl	C(O)OMe	H	H	Br	H	heptafluoroisopropyl	H	CF3
32-254	1,2-difluoro-2-propyl	Me	H	H	Br	H	heptafluoroisopropyl	H	n-C3F7
32-260	4,4,4-trifluoro-n-butyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
32-263	vinyl	C(O)C(O)OMe	H	H	Br	H	heptafluoroisopropyl	H	CF3
32-276	2,2,2-trichloroethyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
32-278	n-propyl	C(O)OEt	H	H	Br	H	nonafluoro-2-butyl	H	CF3
32-282	i-propyl	C(O)Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
32-289	4,4,4-trifluoro-n-butyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
32-294	phenyl	C(O)C(O)OEt	H	H	Br	H	nonafluoro-2-butyl	H	i-C3F7
32-305	2,2,2-trichloroethyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
32-310	3-bromo-n-propyl	C(O)Et	H	H	I	H	heptafluoroisopropyl	H	C2F5
32-318	4,4,4-trifluoro-n-butyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
32-322	benzyl	S(O)2Me	H	H	I	H	heptafluoroisopropyl	H	CF3
32-330	2-cyanoethyl	S(O)2Et	H	H	I	H	nonafluoro-2-butyl	H	CF3
32-334	2,2,2-trichloroethyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
32-336	n-propyl	CH2Ph	H	H	I	H	nonafluoro-2-butyl	H	n-C3F7
32-340	i-propyl	CH2(3-Py)	H	H	I	H	nonafluoro-2-butyl	H	CF3
32-347	4,4,4-trifluoro-n-butyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
32-349	s-butyl	CH2(3-Py—N-	H	H	I	H	nonafluoro-2-butyl	H	CF3
		oxide)
32-350	vinyl	Me	H	H	I	H	nonafluoro-2-butyl	H	i-C3F7
32-363	2,2,2-trichloroethyl	Me	H	H	OCF3	H	heptafluoroisopropyl	H	OCF3
32-392	2,2,2-trichloroethyl	Me	H	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
32-421	2,2,2-trichloroethyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	OCF3
32-450	2,2,2-trichloroethyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	OCF3
32-479	2,2,2-trichloroethyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
32-508	2,2,2-trichloroethyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3

TABLE 33
compound
number	Q2	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
33-1	2,2,2-trichloroethyl	H	Me	H	F	H	heptafluoroisopropyl	H	OCF3
33-2	2,2,2-trichloroethyl	H	Me	H	F	H	nonafluoro-2-butyl	H	OCF3
33-13	2,2,2-trichloroethyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
33-42	2,2,2-trichloroethyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
33-71	2,2,2-trichloroethyl	H	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
33-100	2,2,2-trichloroethyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
33-129	2,2,2-trichloroethyl	H	Me	H	I	H	heptafluoroisopropyl	H	OCF3
33-158	2,2,2-trichloroethyl	H	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
33-177	2,2,2-trichloroethyl	H	Me	H	F	H	heptafluoroisopropyl	H	CF3
33-178	2,2,2-trichloroethyl	H	Me	H	F	H	nonafluoro-2-butyl	H	CF3
33-185	2-cyanoethyl	H	Et	H	Cl	H	heptafluoroisopropyl	H	C2F5
33-189	2,2,2-trichloroethyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
33-191	n-propyl	H	Me	H	Cl	H	pentafluoroethyl	H	CF3
33-195	i-propyl	H	n-Pr	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
33-198	1,3-dichloro-2-propyl	H	Me	H	Cl	H	pentafluoroethyl	H	CF3
33-199	1-chloro-3-fluoro-2-propyl	H	i-Pr	H	Cl	H	heptafluoroisopropyl	H	CF3
33-203	i-butyl	H	CH2CH═CH2	H	Cl	H	heptafluoroisopropyl	H	CF3
33-207	phenyl	H	Me	Cl	Cl	H	heptafluoroisopropyl	H	CF3
33-209	ethyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
33-214	2-cyanoethyl	H	CN	H	Cl	H	nonafluoro-2-butyl	H	CF3
33-218	2,2,2-trichloroethyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
33-220	n-propyl	H	CH2C≡CH	H	Cl	H	nonafluoro-2-butyl	H	CF3
33-232	i-butyl	H	NH2	H	Cl	H	nonafluoro-2-butyl	H	CF3
33-243	2-cyanoethyl	H	Me	H	Br	H	heptafluoroisopropyl	H	C2F5
33-247	2,2,2-trichloroethyl	H	Me	H	Br	H	heptafluoroisopropyl	H	CF3
33-249	n-propyl	H	C(O)OMe	H	Br	H	heptafluoroisopropyl	H	CF3
33-254	1,2-difluoro-2-propyl	H	Me	H	Br	H	heptafluoroisopropyl	H	n-C3F7
33-260	4,4,4-trifluoro-n-butyl	H	Me	H	Br	H	heptafluoroisopropyl	H	CF3
33-263	vinyl	H	C(O)C(O)OMe	H	Br	H	heptafluoroisopropyl	H	CF3
33-276	2,2,2-trichloroethyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
33-278	n-propyl	H	C(O)OEt	H	Br	H	nonafluoro-2-butyl	H	CF3
33-282	i-propyl	H	C(O)Me	H	Br	H	nonafluoro-2-butyl	H	CF3
33-289	4,4,4-trifluoro-n-butyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
33-294	phenyl	H	C(O)C(O)OEt	H	Br	H	nonafluoro-2-butyl	H	i-C3F7
33-305	2,2,2-trichloroethyl	H	Me	H	I	H	heptafluoroisopropyl	H	CF3
33-310	3-bromo-n-propyl	H	C(O)Et	H	I	H	heptafluoroisopropyl	H	C2F5
33-318	4,4,4-trifluoro-n-butyl	H	Me	H	I	H	heptafluoroisopropyl	H	CF3
33-322	benzyl	H	S(O)2Me	H	I	H	heptafluoroisopropyl	H	CF3
33-330	2-cyanoethyl	H	S(O)2Et	H	I	H	nonafluoro-2-butyl	H	CF3
33-334	2,2,2-trichloroethyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
33-336	n-propyl	H	CH2Ph	H	I	H	nonafluoro-2-butyl	H	n-C3F7
33-340	i-propyl	H	CH2(3-Py)	H	I	H	nonafluoro-2-butyl	H	CF3
33-347	4,4,4-trifluoro-n-butyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
33-349	s-butyl	H	CH2(3-Py—N-	H	I	H	nonafluoro-2-butyl	H	CF3
			oxide)
33-350	vinyl	H	Me	H	I	H	nonafluoro-2-butyl	H	i-C3F7
33-363	2,2,2-trichloroethyl	H	Me	H	OCF3	H	heptafluoroisopropyl	H	OCF3
33-392	2,2,2-trichloroethyl	H	Me	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
33-421	2,2,2-trichloroethyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	OCF3
33-450	2,2,2-trichloroethyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	OCF3
33-479	2,2,2-trichloroethyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
33-508	2,2,2-trichloroethyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3

TABLE 34
compound
number	Q2	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
34-1	2,2,2-trichloroethyl	Me	Me	H	F	H	heptafluoroisopropyl	H	OCF3
34-2	2,2,2-trichloroethyl	Me	Me	H	F	H	nonafluoro-2-butyl	H	OCF3
34-13	2,2,2-trichloroethyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
34-42	2,2,2-trichloroethyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
34-71	2,2,2-trichloroethyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
34-100	2,2,2-trichloroethyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
34-129	2,2,2-trichloroethyl	Me	Me	H	I	H	heptafluoroisopropyl	H	OCF3
34-158	2,2,2-trichloroethyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
34-373	2,2,2-trichloroethyl	Me	Me	H	F	H	heptafluoroisopropyl	H	CF3
34-374	2,2,2-trichloroethyl	Me	Me	H	F	H	nonafluoro-2-butyl	H	CF3
34-380	2-iodoethyl	Me	Et	H	Cl	H	heptafluoroisopropyl	H	CF3
34-381	2-cyanoethyl	Et	Me	H	Cl	H	heptafluoroisopropyl	H	C2F5
34-385	2,2,2-trichloroethyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
34-387	n-propyl	Me	n-Pr	H	Cl	H	pentafluoroethyl	H	CF3
34-391	i-propyl	n-Pr	Me	H	Cl	H	heptafluoroisopropyl	H	n-C3F7
34-394	1,3-dichloro-2-propyl	Me	Me	H	Cl	H	pentafluoroethyl	H	CF3
34-395	1-chloro-3-fluoro-2-propyl	i-Pr	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
34-397	n-butyl	Me	i-Pr	H	Cl	H	heptafluoroisopropyl	H	CF3
34-399	i-butyl	CH2CH═CH2	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
34-400	s-butyl	Me	CH2CH═CH2	H	Cl	H	heptafluoroisopropyl	H	CF3
34-401	vinyl	Me	CN	H	Cl	H	heptafluoroisopropyl	H	CF3
34-405	ethyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	i-C3F7
34-410	2-cyanoethyl	CN	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
34-414	2,2,2-trichloroethyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
34-415	2,2,2-tribromoethyl	Me	CH2C≡CH	H	Cl	H	nonafluoro-2-butyl	H	CF3
34-416	n-propyl	CH2C≡CH	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
34-420	i-propyl	Me	Me	Cl	Cl	H	nonafluoro-2-butyl	H	CF3
34-426	n-butyl	Me	NH2	H	Cl	H	nonafluoro-2-butyl	H	CF3
34-428	i-butyl	NH2	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
34-439	2-cyanoethyl	Me	C(O)OMe	H	Br	H	heptafluoroisopropyl	H	C2F5
34-443	2,2,2-trichloroethyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
34-445	n-propyl	C(O)OMe	Me	H	Br	H	heptafluoroisopropyl	H	CF3
34-450	1,2-difluoro-2-propyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	n-C3F7
34-456	4,4,4-trifluoro-n-butyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
34-457	i-butyl	Me	C(O)C(O)OMe	H	Br	H	heptafluoroisopropyl	H	CF3
34-459	vinyl	C(O)C(O)OMe	Me	H	Br	H	heptafluoroisopropyl	H	CF3
34-468	2-cyanoethyl	Me	C(O)OEt	H	Br	H	nonafluoro-2-butyl	H	CF3
34-472	2,2,2-trichloroethyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
34-474	n-propyl	C(O)OEt	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
34-477	3-bromo-n-propyl	Me	C(O)Me	H	Br	H	nonafluoro-2-butyl	H	CF3
34-478	i-propyl	C(O)Me	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
34-485	4,4,4-trifluoro-n-butyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
34-486	i-butyl	Me	C(O)C(O)OEt	H	Br	H	nonafluoro-2-butyl	H	CF3
34-490	phenyl	C(O)C(O)OEt	Me	H	Br	H	nonafluoro-2-butyl	H	i-C3F7
34-501	2,2,2-trichloroethyl	Me	Me	H	I	H	heptafluoroisopropyl	H	CF3
34-503	n-propyl	Me	C(O)Et	H	I	H	heptafluoroisopropyl	H	CF3
34-506	3-bromo-n-propyl	C(O)Et	Me	H	I	H	heptafluoroisopropyl	H	C2F5
34-514	4,4,4-trifluoro-n-butyl	Me	Me	H	I	H	heptafluoroisopropyl	H	CF3
34-515	i-butyl	Me	S(O)2Me	H	I	H	heptafluoroisopropyl	H	CF3
34-518	benzyl	S(O)2Me	Me	H	I	H	heptafluoroisopropyl	H	CF3
34-525	2-iodoethyl	Me	S(O)2Et	H	I	H	nonafluoro-2-butyl	H	CF3
34-526	2-cyanoethyl	S(O)2Et	Me	H	I	H	nonafluoro-2-butyl	H	CF3
34-530	2,2,2-trichloroethyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	CF3
34-531	2,2,2-tribromoethyl	Me	CH2Ph	H	I	H	nonafluoro-2-butyl	H	CF3
34-532	n-propyl	CH2Ph	Me	H	I	H	nonafluoro-2-butyl	H	n-C3F7
34-536	i-propyl	CH2(3-Py)	Me	H	I	H	nonafluoro-2-butyl	H	CF3
34-542	n-butyl	Me	CH2(3-Py)	H	I	H	nonafluoro-2-butyl	H	CF3
34-543	4,4,4-trifluoro-n-butyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	CF3
34-545	s-butyl	CH2(3-Py—N-	Me	H	I	H	nonafluoro-2-butyl	H	CF3
		oxide)
34-546	vinyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	i-C3F7
34-548	phenyl	Me	CH2(3-Py—N-	H	I	H	nonafluoro-2-butyl	H	CF3
			oxide)
34-755	2,2,2-trichloroethyl	Me	Me	H	OCF3	H	heptafluoroisopropyl	H	OCF3
34-784	2,2,2-trichloroethyl	Me	Me	H	OCF3	H	nonafluoro-2-butyl	H	OCF3
34-813	2,2,2-trichloroethyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	OCF3
34-842	2,2,2-trichloroethyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	OCF3
34-871	2,2,2-trichloroethyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
34-900	2,2,2-trichloroethyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3

TABLE 35
compound
number	Q2	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
35-9	2,2-dichloroethyl	H	Et	H	Cl	F	heptafluoroisopropyl	F	OCF3
35-39	2,2,2-trifluoroethyl	H	H	H	Cl	Me	nonafluoro-2-butyl	Me	OCF3
35-154	2,2,2-trichloroethyl	H	H	H	Cl	F	heptafluoroisopropyl	Br	CF3
35-183	2,2,2-trichloroethyl	H	H	H	Cl	Me	nonafluoro-2-butyl	Et	i-C3F7
35-189	i-propyl	H	H	Cl	Cl	Et	nonafluoro-2-butyl	Me	n-C3F7
35-190	1,2-difluoro-2-propyl	H	H	H	Cl	Et	nonafluoro-2-butyl	Et	i-C3F7
35-196	2-chloroethyl	H	H	H	Br	n-Pr	heptafluoroisopropyl	Me	CF3
35-197	2-bromoethyl	H	H	H	Br	n-Pr	heptafluoroisopropyl	Et	CF3
35-203	2,2,2-trichloroethyl	H	H	H	Br	i-Pr	heptafluoroisopropyl	Me	CF3
35-204	2,2,2-tribromoethyl	H	H	H	Br	i-Pr	heptafluoroisopropyl	Et	CF3
35-210	1,2-difluoro-2-propyl	H	H	H	Br	n-Bu	heptafluoroisopropyl	Me	CF3
35-211	1,3-difluoro-2-propyl	H	H	H	Br	n-Bu	heptafluoroisopropyl	Et	CF3
35-217	i-butyl	H	H	H	Br	i-Bu	nonafluoro-2-butyl	Me	CF3
35-218	s-butyl	H	H	H	Br	i-Bu	nonafluoro-2-butyl	Et	CF3
35-224	2-fluoroethyl	H	H	H	Br	s-Bu	nonafluoro-2-butyl	Me	CF3
35-225	2-chloroethyl	H	H	H	Br	s-Bu	nonafluoro-2-butyl	Et	CF3
35-231	2,2,2-trifluoroethyl	H	H	H	Br	F	nonafluoro-2-butyl	Me	CF3
35-232	2,2,2-trichloroethyl	H	H	H	Br	F	nonafluoro-2-butyl	Et	CF3
35-238	i-propyl	Et	i-Pr	H	Br	Cl	nonafluoro-2-butyl	Me	CF3
35-239	1,2-difluoro-2-propyl	H	H	H	Br	Cl	nonafluoro-2-butyl	Et	CF3
35-245	2-iodoethyl	H	H	H	I	Br	heptafluoroisopropyl	Me	CF3
35-246	2-cyanoethyl	H	H	H	I	Br	heptafluoroisopropyl	Et	CF3
35-252	n-propyl	n-Pr	Me	H	I	I	heptafluoroisopropyl	Me	CF3
35-253	3-fluoro-n-propyl	H	H	H	I	I	heptafluoroisopropyl	Et	CF3
35-259	1,3-dichloro-2-propyl	H	H	H	I	Me	heptafluoroisopropyl	F	C2F5
35-260	1-chloro-3-fluoro-2-propyl	H	H	H	I	Me	nonafluoro-2-butyl	Cl	CF3
35-261	3,3,3-trifluoro-n-propyl	H	H	H	I	Me	nonafluoro-2-butyl	Br	n-C3F7
35-262	n-butyl	H	H	H	I	Me	nonafluoro-2-butyl	I	i-C3F7
35-263	4,4,4-trifluoro-n-butyl	H	H	H	I	Et	nonafluoro-2-butyl	F	CF3
35-264	i-butyl	H	H	H	I	Et	nonafluoro-2-butyl	Cl	CF3
35-265	s-butyl	H	H	H	I	Et	nonafluoro-2-butyl	Br	CF3
35-266	vinyl	n-Pr	i-Pr	H	I	Et	nonafluoro-2-butyl	I	C2F5
35-267	benzyl	H	H	H	I	n-Pr	nonafluoro-2-butyl	F	CF3
35-268	phenyl	H	H	H	I	n-Pr	nonafluoro-2-butyl	Cl	CF3
35-271	2-fluoroethyl	H	H	H	I	i-Pr	nonafluoro-2-butyl	F	i-C3F7
35-272	2-chloroethyl	H	H	H	I	i-Pr	nonafluoro-2-butyl	Cl	CF3
35-273	2-bromoethyl	n-Pr	C(O)Me	H	I	i-Pr	nonafluoro-2-butyl	Br	CF3
35-274	2-iodoethyl	H	H	H	I	i-Pr	nonafluoro-2-butyl	I	CF3
35-275	2-cyanoethyl	H	H	H	I	n-Bu	nonafluoro-2-butyl	F	CF3
35-276	2,2-difluoroethyl	H	H	H	I	n-Bu	nonafluoro-2-butyl	Cl	CF3
35-279	2,2,2-trichloroethyl	H	H	H	I	i-Bu	nonafluoro-2-butyl	F	CF3
35-280	2,2,2-tribromoethyl	H	H	H	I	i-Bu	nonafluoro-2-butyl	Cl	CF3
35-283	3-chloro-n-propyl	i-Pr	n-Pr	H	I	s-Bu	nonafluoro-2-butyl	F	CF3
35-284	3-bromo-n-propyl	H	H	H	I	s-Bu	nonafluoro-2-butyl	Cl	CF3
35-301	3-chloro-n-propyl	n-Pr	H	H	OCF3	Cl	heptafluoroisopropyl	Br	OCF3
35-454	i-butyl	H	H	H	OCF3	Me	nonafluoro-2-butyl	H	CF3
35-582	2,2,2-trifluoroethyl	H	H	H	CF3	F	heptafluoroisopropyl	Cl	CF3

TABLE 36
compound
number	Q1	R1	R2	X2	Y1	Y2	Y3	Y4	Y5
36-1	phenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
36-2	phenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
36-3	phenyl	H	H	Cl	Br	H	heptafluoroisopropyl	H	CF3
36-4	phenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
36-5	phenyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
36-6	phenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
36-7	phenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
36-8	phenyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
36-9	phenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
36-10	phenyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
36-11	phenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	OCF3
36-12	phenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
36-13	phenyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
36-14	phenyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
36-15	phenyl	H	Me	H	Br	H	heptafluoroisopropyl	H	CF3
36-16	phenyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
36-17	phenyl	H	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
36-18	phenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
36-19	phenyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
36-20	phenyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
36-21	phenyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
36-22	phenyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
36-23	phenyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
36-24	phenyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
36-25	phenyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
36-26	phenyl	H	H	H	Cl	F	heptafluoroisopropyl	H	OCF3
36-27	phenyl	Me	H	H	Br	H	heptafluoroisopropyl	F	CF3
36-28	phenyl	H	Me	H	CF3	Cl	heptafluoroisopropyl	H	CF3
36-29	phenyl	H	H	H	I	H	nonafluoro-2-butyl	Cl	OCF3
36-30	phenyl	H	H	H	Cl	Br	nonafluoro-2-butyl	H	CF3
36-31	phenyl	H	H	H	Br	H	nonafluoro-2-butyl	I	CF3
36-32	phenyl	H	H	H	I	Me	nonafluoro-2-butyl	H	CF3
36-33	phenyl	H	H	H	CF3	H	nonafluoro-2-butyl	Et	CF3

TABLE 37
compound
number	Q1	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
37-1	phenyl	H	H	H	Br	H	heptafluoroisopropyl	H	OCF3
37-2	phenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
37-3	phenyl	H	H	Cl	I	H	heptafluoroisopropyl	H	CF3
37-4	phenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
37-5	phenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
37-6	phenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
37-7	phenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
37-8	phenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
37-9	phenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
37-10	phenyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
37-11	phenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
37-12	phenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
37-13	phenyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
37-14	phenyl	H	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
37-15	phenyl	H	Me	H	I	H	heptafluoroisopropyl	H	CF3
37-16	phenyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
37-17	phenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
37-18	phenyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
37-19	phenyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
37-20	phenyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
37-21	phenyl	Me	Me	H	I	H	heptafluoroisopropyl	H	CF3
37-22	phenyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
37-23	phenyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
37-24	phenyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
37-25	phenyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
37-26	phenyl	Me	H	H	Br	F	heptafluoroisopropyl	H	OCF3
37-27	phenyl	H	H	H	I	H	heptafluoroisopropyl	F	CF3
37-28	phenyl	H	Me	H	CF3	Cl	heptafluoroisopropyl	H	CF3
37-29	phenyl	H	H	H	Cl	H	nonafluoro-2-butyl	Cl	OCF3
37-30	phenyl	H	H	H	Br	Br	nonafluoro-2-butyl	H	CF3
37-31	phenyl	H	H	H	I	H	nonafluoro-2-butyl	I	CF3
37-32	phenyl	H	H	H	Cl	Me	nonafluoro-2-butyl	H	CF3
37-33	phenyl	H	H	H	CF3	H	nonafluoro-2-butyl	Et	CF3

TABLE 38
compound
number	Q1	R1	R2	X2	Y1	Y2	Y3	Y4	Y5
38-1	phenyl	H	H	H	I	H	heptafluoroisopropyl	H	OCF3
38-2	phenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	CF3
38-3	phenyl	H	H	Cl	Cl	H	heptafluoroisopropyl	H	CF3
38-4	phenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
38-5	phenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
38-6	phenyl	H	H	H	I	H	nonafluoro-2-butyl	H	CF3
38-7	phenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
38-8	phenyl	Me	H	H	I	H	heptafluoroisopropyl	H	OCF3
38-9	phenyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	CF3
38-10	phenyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
38-11	phenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
38-12	phenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	CF3
38-13	phenyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
38-14	phenyl	H	Me	H	I	H	heptafluoroisopropyl	H	OCF3
38-15	phenyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
38-16	phenyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
38-17	phenyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
38-18	phenyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
38-19	phenyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
38-20	phenyl	Me	Me	H	I	H	heptafluoroisopropyl	H	OCF3
38-21	phenyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
38-22	phenyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
38-23	phenyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
38-24	phenyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	CF3
38-25	phenyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
38-26	phenyl	H	H	H	I	F	heptafluoroisopropyl	H	OCF3
38-27	phenyl	H	H	H	Cl	H	heptafluoroisopropyl	F	CF3
38-28	phenyl	Me	H	H	CF3	Cl	heptafluoroisopropyl	H	CF3
38-29	phenyl	H	H	H	Br	H	nonafluoro-2-butyl	Cl	OCF3
38-30	phenyl	H	Me	H	I	Br	nonafluoro-2-butyl	H	CF3
38-31	phenyl	H	H	H	Cl	H	nonafluoro-2-butyl	I	CF3
38-32	phenyl	H	H	H	Br	Me	nonafluoro-2-butyl	H	CF3
38-33	phenyl	H	H	H	CF3	H	nonafluoro-2-butyl	Et	CF3

TABLE 39
compound
number	Q1	R1	R2	X1	Y1	Y2	Y3	Y4	Y5
39-1	phenyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
39-2	phenyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
39-3	phenyl	H	H	Cl	Br	H	heptafluoroisopropyl	H	CF3
39-4	phenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
39-5	phenyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
39-6	phenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
39-7	phenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
39-8	phenyl	Me	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
39-9	phenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	CF3
39-10	phenyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
39-11	phenyl	Me	H	H	I	H	nonafluoro-2-butyl	H	OCF3
39-12	phenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
39-13	phenyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
39-14	phenyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
39-15	phenyl	H	Me	H	Br	H	heptafluoroisopropyl	H	CF3
39-16	phenyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
39-17	phenyl	H	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
39-18	phenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
39-19	phenyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
39-20	phenyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
39-21	phenyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
39-22	phenyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
39-23	phenyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
39-24	phenyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
39-25	phenyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
39-26	phenyl	H	H	H	Cl	F	heptafluoroisopropyl	H	OCF3
39-27	phenyl	Me	H	H	Br	H	heptafluoroisopropyl	F	CF3
39-28	phenyl	H	Me	H	CF3	Cl	heptafluoroisopropyl	H	CF3
39-29	phenyl	H	H	H	I	H	nonafluoro-2-butyl	Cl	OCF3
39-30	phenyl	H	H	H	Cl	Br	nonafluoro-2-butyl	H	CF3
39-31	phenyl	H	H	H	Br	H	nonafluoro-2-butyl	I	CF3
39-32	phenyl	H	H	H	I	Me	nonafluoro-2-butyl	H	CF3
39-33	phenyl	H	H	H	CF3	H	nonafluoro-2-butyl	Et	CF3

TABLE 40
compound
number	Q1	R1	R2	X1	Y1	Y2	Y3	Y4	Y5
40-1	phenyl	H	H	H	Br	H	heptafluoroisopropyl	H	OCF3
40-2	phenyl	H	H	H	I	H	heptafluoroisopropyl	H	CF3
40-3	phenyl	H	H	Cl	I	H	heptafluoroisopropyl	H	CF3
40-4	phenyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
40-5	phenyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
40-6	phenyl	H	H	H	Br	H	nonafluoro-2-butyl	H	CF3
40-7	phenyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
40-8	phenyl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
40-9	phenyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
40-10	phenyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
40-11	phenyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
40-12	phenyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
40-13	phenyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
40-14	phenyl	H	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
40-15	phenyl	H	Me	H	I	H	heptafluoroisopropyl	H	CF3
40-16	phenyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
40-17	phenyl	H	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
40-18	phenyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
40-19	phenyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
40-20	phenyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	OCF3
40-21	phenyl	Me	Me	H	I	H	heptafluoroisopropyl	H	CF3
40-22	phenyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
40-23	phenyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	OCF3
40-24	phenyl	Me	Me	H	Br	H	nonafluoro-2-butyl	H	CF3
40-25	phenyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
40-26	phenyl	H	H	H	Br	F	heptafluoroisopropyl	H	OCF3
40-27	phenyl	H	H	H	I	H	heptafluoroisopropyl	F	CF3
40-28	phenyl	Me	H	H	CF3	Cl	heptafluoroisopropyl	H	CF3
40-29	phenyl	H	H	H	Cl	H	nonafluoro-2-butyl	Cl	OCF3
40-30	phenyl	H	H	H	Br	Br	nonafluoro-2-butyl	H	CF3
40-31	phenyl	H	H	H	I	H	nonafluoro-2-butyl	I	CF3
40-32	phenyl	H	H	H	Cl	Me	nonafluoro-2-butyl	H	CF3
40-33	phenyl	H	Me	H	CF3	H	nonafluoro-2-butyl	Et	CF3

TABLE 41
compound
number	Q2	R1	R2	X2	Y1	Y2	Y3	Y4	Y5
41-1	2,2,2-trichloroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
41-2	2,2,2-trichloroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
41-3	2,2,2-trichloroethyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
41-4	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
41-5	2,2,2-trichloroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
41-6	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
41-7	2,2,2-trichloroethyl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
41-8	2,2,2-trichloroethyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
41-9	2,2,2-trichloroethyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
41-10	2,2,2-trichloroethyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
41-11	2,2,2-trichloroethyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
41-12	2,2,2-trichloroethyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
41-13	2,2,2-trichloroethyl	H	Me	H	I	H	heptafluoroisopropyl	H	OCF3
41-14	2,2,2-trichloroethyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
41-15	2,2,2-trichloroethyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
41-16	2,2,2-trichloroethyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
41-17	2,2,2-trichloroethyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
41-18	2,2,2-trichloroethyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
41-19	2,2,2-trichloroethyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
41-20	2,2,2-trichloroethyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
41-21	2,2,2-trichloroethyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
41-22	2,2,2-trichloroethyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
41-23	2,2,2-trichloroethyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
41-24	2,2,2-trichloroethyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
41-25	2,2,2-trichloroethyl	H	H	H	Br	F	heptafluoroisopropyl	H	OCF3
41-26	2,2,2-trichloroethyl	H	H	H	I	H	heptafluoroisopropyl	Cl	CF3
41-27	2,2,2-trichloroethyl	H	H	H	CF3	Br	heptafluoroisopropyl	H	CF3
41-28	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	I	OCF3
41-29	2,2,2-trichloroethyl	H	H	H	Br	Me	nonafluoro-2-butyl	H	CF3
41-30	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	Et	CF3
41-31	2,2,2-trichloroethyl	H	H	Cl	Br	H	heptafluoroisopropyl	H	CF3

TABLE 42
compound
number	Q2	R1	R2	X3	Y1	Y2	Y3	Y4	Y5
42-1	2,2,2-trichloroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
42-2	2,2,2-trichloroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
42-3	2,2,2-trichloroethyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
42-4	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
42-5	2,2,2-trichloroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
42-6	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
42-7	2,2,2-trichloroethyl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
42-8	2,2,2-trichloroethyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
42-9	2,2,2-trichloroethyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
42-10	2,2,2-trichloroethyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
42-11	2,2,2-trichloroethyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
42-12	2,2,2-trichloroethyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
42-13	2,2,2-trichloroethyl	H	Me	H	I	H	heptafluoroisopropyl	H	OCF3
42-14	2,2,2-trichloroethyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
42-15	2,2,2-trichloroethyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
42-16	2,2,2-trichloroethyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
42-17	2,2,2-trichloroethyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
42-18	2,2,2-trichloroethyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
42-19	2,2,2-trichloroethyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
42-20	2,2,2-trichloroethyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
42-21	2,2,2-trichloroethyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
42-22	2,2,2-trichloroethyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
42-23	2,2,2-trichloroethyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
42-24	2,2,2-trichloroethyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
42-25	2,2,2-trichloroethyl	H	H	H	Br	F	heptafluoroisopropyl	H	OCF3
42-26	2,2,2-trichloroethyl	H	H	H	I	H	heptafluoroisopropyl	Cl	CF3
42-27	2,2,2-trichloroethyl	H	H	H	CF3	Br	heptafluoroisopropyl	H	CF3
42-28	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	I	OCF3
42-29	2,2,2-trichloroethyl	H	H	H	Br	Me	nonafluoro-2-butyl	H	CF3
42-30	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	Et	CF3
42-31	2,2,2-trichloroethyl	H	H	Cl	Br	H	heptafluoroisopropyl	H	CF3

TABLE 43
compound
number	Q2	R1	R2	X2	Y1	Y2	Y3	Y4	Y5
43-1	2,2,2-trichloroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
43-2	2,2,2-trichloroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
43-3	2,2,2-trichloroethyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
43-4	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
43-5	2,2,2-trichloroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
43-6	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
43-7	2,2,2-trichloroethyl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
43-8	2,2,2-trichloroethyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
43-9	2,2,2-trichloroethyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
43-10	2,2,2-trichloroethyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
43-11	2,2,2-trichloroethyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
43-12	2,2,2-trichloroethyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
43-13	2,2,2-trichloroethyl	H	Me	H	I	H	heptafluoroisopropyl	H	OCF3
43-14	2,2,2-trichloroethyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
43-15	2,2,2-trichloroethyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
43-16	2,2,2-trichloroethyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
43-17	2,2,2-trichloroethyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
43-18	2,2,2-trichloroethyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
43-19	2,2,2-trichloroethyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
43-20	2,2,2-trichloroethyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
43-21	2,2,2-trichloroethyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
43-22	2,2,2-trichloroethyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
43-23	2,2,2-trichloroethyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
43-24	2,2,2-trichloroethyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
43-25	2,2,2-trichloroethyl	H	H	H	Br	F	heptafluoroisopropyl	H	OCF3
43-26	2,2,2-trichloroethyl	H	H	H	I	H	heptafluoroisopropyl	Cl	CF3
43-27	2,2,2-trichloroethyl	H	H	H	CF3	Br	heptafluoroisopropyl	H	CF3
43-28	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	I	OCF3
43-29	2,2,2-trichloroethyl	H	H	H	Br	Me	nonafluoro-2-butyl	H	CF3
43-30	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	Et	CF3
43-31	2,2,2-trichloroethyl	H	H	Cl	Br	H	heptafluoroisopropyl	H	CF3

TABLE 44
compound
number	Q2	R1	R2	X1	Y1	Y2	Y3	Y4	Y5
44-1	2,2,2-trichloroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
44-2	2,2,2-trichloroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
44-3	2,2,2-trichloroethyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
44-4	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
44-5	2,2,2-trichloroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
44-6	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
44-7	2,2,2-trichloroethyl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
44-8	2,2,2-trichloroethyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
44-9	2,2,2-trichloroethyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
44-10	2,2,2-trichloroethyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
44-11	2,2,2-trichloroethyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
44-12	2,2,2-trichloroethyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
44-13	2,2,2-trichloroethyl	H	Me	H	I	H	heptafluoroisopropyl	H	OCF3
44-14	2,2,2-trichloroethyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
44-15	2,2,2-trichloroethyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
44-16	2,2,2-trichloroethyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
44-17	2,2,2-trichloroethyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
44-18	2,2,2-trichloroethyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
44-19	2,2,2-trichloroethyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
44-20	2,2,2-trichloroethyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
44-21	2,2,2-trichloroethyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
44-22	2,2,2-trichloroethyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
44-23	2,2,2-trichloroethyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
44-24	2,2,2-trichloroethyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
44-25	2,2,2-trichloroethyl	H	H	H	Br	F	heptafluoroisopropyl	H	OCF3
44-26	2,2,2-trichloroethyl	H	H	H	I	H	heptafluoroisopropyl	Cl	CF3
44-27	2,2,2-trichloroethyl	H	H	H	CF3	Br	heptafluoroisopropyl	H	CF3
44-28	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	I	OCF3
44-29	2,2,2-trichloroethyl	H	H	H	Br	Me	nonafluoro-2-butyl	H	CF3
44-30	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	Et	CF3
44-31	2,2,2-trichloroethyl	H	H	Cl	Br	H	heptafluoroisopropyl	H	CF3

TABLE 45
compound
number	Q2	R1	R2	X1	Y1	Y2	Y3	Y4	Y5
45-1	2,2,2-trichloroethyl	H	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
45-2	2,2,2-trichloroethyl	H	H	H	Br	H	heptafluoroisopropyl	H	CF3
45-3	2,2,2-trichloroethyl	H	H	H	CF3	H	heptafluoroisopropyl	H	CF3
45-4	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	H	OCF3
45-5	2,2,2-trichloroethyl	H	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
45-6	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
45-7	2,2,2-trichloroethyl	Me	H	H	Br	H	heptafluoroisopropyl	H	OCF3
45-8	2,2,2-trichloroethyl	Me	H	H	I	H	heptafluoroisopropyl	H	CF3
45-9	2,2,2-trichloroethyl	Me	H	H	CF3	H	heptafluoroisopropyl	H	CF3
45-10	2,2,2-trichloroethyl	Me	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
45-11	2,2,2-trichloroethyl	Me	H	H	Br	H	nonafluoro-2-butyl	H	CF3
45-12	2,2,2-trichloroethyl	Me	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
45-13	2,2,2-trichloroethyl	H	Me	H	I	H	heptafluoroisopropyl	H	OCF3
45-14	2,2,2-trichloroethyl	H	Me	H	Cl	H	heptafluoroisopropyl	H	CF3
45-15	2,2,2-trichloroethyl	H	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
45-16	2,2,2-trichloroethyl	H	Me	H	Br	H	nonafluoro-2-butyl	H	OCF3
45-17	2,2,2-trichloroethyl	H	Me	H	I	H	nonafluoro-2-butyl	H	CF3
45-18	2,2,2-trichloroethyl	H	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
45-19	2,2,2-trichloroethyl	Me	Me	H	Cl	H	heptafluoroisopropyl	H	OCF3
45-20	2,2,2-trichloroethyl	Me	Me	H	Br	H	heptafluoroisopropyl	H	CF3
45-21	2,2,2-trichloroethyl	Me	Me	H	CF3	H	heptafluoroisopropyl	H	CF3
45-22	2,2,2-trichloroethyl	Me	Me	H	I	H	nonafluoro-2-butyl	H	OCF3
45-23	2,2,2-trichloroethyl	Me	Me	H	Cl	H	nonafluoro-2-butyl	H	CF3
45-24	2,2,2-trichloroethyl	Me	Me	H	CF3	H	nonafluoro-2-butyl	H	CF3
45-25	2,2,2-trichloroethyl	H	H	H	Br	F	heptafluoroisopropyl	H	OCF3
45-26	2,2,2-trichloroethyl	H	H	H	I	H	heptafluoroisopropyl	Cl	CF3
45-27	2,2,2-trichloroethyl	H	H	H	CF3	Br	heptafluoroisopropyl	H	CF3
45-28	2,2,2-trichloroethyl	H	H	H	I	H	nonafluoro-2-butyl	I	OCF3
45-29	2,2,2-trichloroethyl	H	H	H	Br	Me	nonafluoro-2-butyl	H	CF3
45-30	2,2,2-trichloroethyl	H	H	H	CF3	H	nonafluoro-2-butyl	Et	CF3
45-31	2,2,2-trichloroethyl	H	H	Cl	Br	H	heptafluoroisopropyl	H	CF3

TABLE 46
compound
number	Q1	R1	R2	A	X2	X3	Y1	Y2	Y3	Y4	Y5
46-1	phenyl	H	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
46-2	phenyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
46-3	phenyl	H	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-4	phenyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
46-5	phenyl	H	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
46-6	phenyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-7	phenyl	H	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
46-8	phenyl	H	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
46-9	phenyl	H	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-10	phenyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
46-11	phenyl	H	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
46-12	phenyl	H	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-13	phenyl	H	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
46-14	phenyl	H	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
46-15	phenyl	H	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-16	phenyl	H	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
46-17	phenyl	H	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
46-18	phenyl	H	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-19	phenyl	Me	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
46-20	phenyl	Me	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
46-21	phenyl	Me	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-22	phenyl	Me	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
46-23	phenyl	Me	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
46-24	phenyl	Me	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-25	phenyl	Me	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
46-26	phenyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
46-27	phenyl	Me	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-28	phenyl	Me	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
46-29	phenyl	Me	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
46-30	phenyl	Me	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-31	phenyl	Me	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
46-32	phenyl	Me	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
46-33	phenyl	Me	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-34	phenyl	Me	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
46-35	phenyl	Me	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
46-36	phenyl	Me	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-37	phenyl	H	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
46-38	phenyl	H	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
46-39	phenyl	H	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-40	phenyl	H	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
46-41	phenyl	H	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
46-42	phenyl	H	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-43	phenyl	H	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
46-44	phenyl	H	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
46-45	phenyl	H	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-46	phenyl	H	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
46-47	phenyl	H	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
46-48	phenyl	H	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-49	phenyl	H	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
46-50	phenyl	H	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
46-51	phenyl	H	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-52	phenyl	H	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
46-53	phenyl	H	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
46-54	phenyl	H	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-55	phenyl	Me	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
46-56	phenyl	Me	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
46-57	phenyl	Me	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-58	phenyl	Me	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
46-59	phenyl	Me	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
46-60	phenyl	Me	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-61	phenyl	Me	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
46-62	phenyl	Me	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
46-63	phenyl	Me	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-64	phenyl	Me	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
46-65	phenyl	Me	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
46-66	phenyl	Me	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-67	phenyl	Me	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
46-68	phenyl	Me	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
46-69	phenyl	Me	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
46-70	phenyl	Me	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
46-71	phenyl	Me	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
46-72	phenyl	Me	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
46-73	phenyl	Me	H	S	H	H	Cl	F	heptafluoroisopropyl	H	OCF3
46-74	phenyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	F	CF3
46-75	phenyl	H	H	S	H	H	CF3	Cl	heptafluoroisopropyl	H	CF3
46-76	phenyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	Cl	OCF3
46-77	phenyl	H	H	S	H	H	Cl	Br	nonafluoro-2-butyl	H	CF3
46-78	phenyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	Br	CF3
46-79	phenyl	H	H	O	H	H	Br	I	heptafluoroisopropyl	H	OCF3
46-80	phenyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	I	CF3
46-81	phenyl	H	H	O	H	H	CF3	Me	heptafluoroisopropyl	H	CF3
46-82	phenyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	Me	OCF3
46-83	phenyl	H	H	O	H	H	Br	F	nonafluoro-2-butyl	F	CF3
46-84	phenyl	H	H	O	H	H	CF3	Cl	nonafluoro-2-butyl	Cl	CF3
46-85	phenyl	H	H	NH	H	H	I	Br	heptafluoroisopropyl	Br	OCF3
46-86	phenyl	H	H	NH	H	H	Cl	I	heptafluoroisopropyl	I	CF3
46-87	phenyl	Me	H	NH	H	H	CF3	F	heptafluoroisopropyl	Me	CF3
46-88	phenyl	H	H	NH	H	H	Br	Cl	nonafluoro-2-butyl	Me	OCF3
46-89	phenyl	H	H	NH	H	H	I	Br	nonafluoro-2-butyl	Me	CF3
46-90	phenyl	H	H	NH	H	H	CF3	I	nonafluoro-2-butyl	Me	CF3

TABLE 47
compound
number	Q1	R1	R2	A	X1	X3	Y1	Y2	Y3	Y4	Y5
47-1	phenyl	H	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
47-2	phenyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
47-3	phenyl	H	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-4	phenyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
47-5	phenyl	H	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
47-6	phenyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-7	phenyl	H	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
47-8	phenyl	H	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
47-9	phenyl	H	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-10	phenyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
47-11	phenyl	H	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
47-12	phenyl	H	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-13	phenyl	H	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
47-14	phenyl	H	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
47-15	phenyl	H	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-16	phenyl	H	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
47-17	phenyl	H	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
47-18	phenyl	H	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-19	phenyl	Me	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
47-20	phenyl	Me	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
47-21	phenyl	Me	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-22	phenyl	Me	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
47-23	phenyl	Me	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
47-24	phenyl	Me	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-25	phenyl	Me	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
47-26	phenyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
47-27	phenyl	Me	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-28	phenyl	Me	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
47-29	phenyl	Me	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
47-30	phenyl	Me	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-31	phenyl	Me	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
47-32	phenyl	Me	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
47-33	phenyl	Me	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-34	phenyl	Me	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
47-35	phenyl	Me	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
47-36	phenyl	Me	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-37	phenyl	H	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
47-38	phenyl	H	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
47-39	phenyl	H	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-40	phenyl	H	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
47-41	phenyl	H	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
47-42	phenyl	H	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-43	phenyl	H	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
47-44	phenyl	H	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
47-45	phenyl	H	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-46	phenyl	H	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
47-47	phenyl	H	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
47-48	phenyl	H	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-49	phenyl	H	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
47-50	phenyl	H	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
47-51	phenyl	H	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-52	phenyl	H	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
47-53	phenyl	H	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
47-54	phenyl	H	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-55	phenyl	Me	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
47-56	phenyl	Me	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
47-57	phenyl	Me	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-58	phenyl	Me	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
47-59	phenyl	Me	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
47-60	phenyl	Me	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-61	phenyl	Me	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
47-62	phenyl	Me	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
47-63	phenyl	Me	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-64	phenyl	Me	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
47-65	phenyl	Me	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
47-66	phenyl	Me	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-67	phenyl	Me	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
47-68	phenyl	Me	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
47-69	phenyl	Me	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
47-70	phenyl	Me	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
47-71	phenyl	Me	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
47-72	phenyl	Me	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
47-73	phenyl	Me	H	S	H	H	Cl	F	heptafluoroisopropyl	H	OCF3
47-74	phenyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	F	CF3
47-75	phenyl	H	H	S	H	H	CF3	Cl	heptafluoroisopropyl	H	CF3
47-76	phenyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	Cl	OCF3
47-77	phenyl	H	H	S	H	H	Cl	Br	nonafluoro-2-butyl	H	CF3
47-78	phenyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	Br	CF3
47-79	phenyl	H	H	O	H	H	Br	I	heptafluoroisopropyl	H	OCF3
47-80	phenyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	I	CF3
47-81	phenyl	H	H	O	H	H	CF3	Me	heptafluoroisopropyl	H	CF3
47-82	phenyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	Me	OCF3
47-83	phenyl	H	H	O	H	H	Br	F	nonafluoro-2-butyl	F	CF3
47-84	phenyl	H	H	O	H	H	CF3	Cl	nonafluoro-2-butyl	Cl	CF3
47-85	phenyl	H	H	NH	H	H	I	Br	heptafluoroisopropyl	Br	OCF3
47-86	phenyl	H	H	NH	H	H	Cl	I	heptafluoroisopropyl	I	CF3
47-87	phenyl	Me	H	NH	H	H	CF3	F	heptafluoroisopropyl	Me	CF3
47-88	phenyl	H	H	NH	H	H	Br	Cl	nonafluoro-2-butyl	Me	OCF3
47-89	phenyl	H	H	NH	H	H	I	Br	nonafluoro-2-butyl	Me	CF3
47-90	phenyl	H	H	NH	H	H	CF3	I	nonafluoro-2-butyl	Me	CF3

TABLE 48
compound
number	Q1	R1	R2	A	X1	X2	Y1	Y2	Y3	Y4	Y5
48-1	phenyl	H	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
48-2	phenyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
48-3	phenyl	H	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-4	phenyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
48-5	phenyl	H	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
48-6	phenyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-7	phenyl	H	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
48-8	phenyl	H	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
48-9	phenyl	H	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-10	phenyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
48-11	phenyl	H	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
48-12	phenyl	H	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-13	phenyl	H	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
48-14	phenyl	H	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
48-15	phenyl	H	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-16	phenyl	H	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
48-17	phenyl	H	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
48-18	phenyl	H	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-19	phenyl	Me	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
48-20	phenyl	Me	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
48-21	phenyl	Me	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-22	phenyl	Me	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
48-23	phenyl	Me	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
48-24	phenyl	Me	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-25	phenyl	Me	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
48-26	phenyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
48-27	phenyl	Me	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-28	phenyl	Me	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
48-29	phenyl	Me	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
48-30	phenyl	Me	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-31	phenyl	Me	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
48-32	phenyl	Me	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
48-33	phenyl	Me	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-34	phenyl	Me	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
48-35	phenyl	Me	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
48-36	phenyl	Me	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-37	phenyl	H	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
48-38	phenyl	H	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
48-39	phenyl	H	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-40	phenyl	H	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
48-41	phenyl	H	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
48-42	phenyl	H	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-43	phenyl	H	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
48-44	phenyl	H	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
48-45	phenyl	H	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-46	phenyl	H	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
48-47	phenyl	H	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
48-48	phenyl	H	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-49	phenyl	H	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
48-50	phenyl	H	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
48-51	phenyl	H	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-52	phenyl	H	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
48-53	phenyl	H	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
48-54	phenyl	H	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-55	phenyl	Me	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
48-56	phenyl	Me	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
48-57	phenyl	Me	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-58	phenyl	Me	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
48-59	phenyl	Me	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
48-60	phenyl	Me	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-61	phenyl	Me	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
48-62	phenyl	Me	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
48-63	phenyl	Me	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-64	phenyl	Me	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
48-65	phenyl	Me	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
48-66	phenyl	Me	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-67	phenyl	Me	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
48-68	phenyl	Me	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
48-69	phenyl	Me	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
48-70	phenyl	Me	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
48-71	phenyl	Me	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
48-72	phenyl	Me	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
48-73	phenyl	Me	H	S	H	H	Cl	F	heptafluoroisopropyl	H	OCF3
48-74	phenyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	F	CF3
48-75	phenyl	H	H	S	H	H	CF3	Cl	heptafluoroisopropyl	H	CF3
48-76	phenyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	Cl	OCF3
48-77	phenyl	H	H	S	H	H	Cl	Br	nonafluoro-2-butyl	H	CF3
48-78	phenyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	Br	CF3
48-79	phenyl	H	H	O	H	H	Br	I	heptafluoroisopropyl	H	OCF3
48-80	phenyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	I	CF3
48-81	phenyl	H	H	O	H	H	CF3	Me	heptafluoroisopropyl	H	CF3
48-82	phenyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	Me	OCF3
48-83	phenyl	H	H	O	H	H	Br	F	nonafluoro-2-butyl	F	CF3
48-84	phenyl	H	H	O	H	H	CF3	Cl	nonafluoro-2-butyl	Cl	CF3
48-85	phenyl	H	H	NH	H	H	I	Br	heptafluoroisopropyl	Br	OCF3
48-86	phenyl	H	H	NH	H	H	Cl	I	heptafluoroisopropyl	I	CF3
48-87	phenyl	Me	H	NH	H	H	CF3	F	heptafluoroisopropyl	Me	CF3
48-88	phenyl	H	H	NH	H	H	Br	Cl	nonafluoro-2-butyl	Me	OCF3
48-89	phenyl	H	H	NH	H	H	I	Br	nonafluoro-2-butyl	Me	CF3
48-90	phenyl	H	H	NH	H	H	CF3	I	nonafluoro-2-butyl	Me	CF3

TABLE 49
compound
number	Q2	R1	R2	A	X2	X3	Y1	Y2	Y3	Y4	Y5
49-1	2,2,2-trichloroethyl	H	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
49-2	2,2,2-trichloroethyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
49-3	2,2,2-trichloroethyl	H	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-4	2,2,2-trichloroethyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
49-5	2,2,2-trichloroethyl	H	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
49-6	2,2,2-trichloroethyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-7	2,2,2-trichloroethyl	H	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
49-8	2,2,2-trichloroethyl	H	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
49-9	2,2,2-trichloroethyl	H	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-10	2,2,2-trichloroethyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
49-11	2,2,2-trichloroethyl	H	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
49-12	2,2,2-trichloroethyl	H	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-13	2,2,2-trichloroethyl	H	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
49-14	2,2,2-trichloroethyl	H	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
49-15	2,2,2-trichloroethyl	H	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-16	2,2,2-trichloroethyl	H	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
49-17	2,2,2-trichloroethyl	H	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
49-18	2,2,2-trichloroethyl	H	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-19	2,2,2-trichloroethyl	Me	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
49-20	2,2,2-trichloroethyl	Me	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
49-21	2,2,2-trichloroethyl	Me	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-22	2,2,2-trichloroethyl	Me	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
49-23	2,2,2-trichloroethyl	Me	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
49-24	2,2,2-trichloroethyl	Me	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-25	2,2,2-trichloroethyl	Me	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
49-26	2,2,2-trichloroethyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
49-27	2,2,2-trichloroethyl	Me	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-28	2,2,2-trichloroethyl	Me	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
49-29	2,2,2-trichloroethyl	Me	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
49-30	2,2,2-trichloroethyl	Me	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-31	2,2,2-trichloroethyl	Me	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
49-32	2,2,2-trichloroethyl	Me	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
49-33	2,2,2-trichloroethyl	Me	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-34	2,2,2-trichloroethyl	Me	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
49-35	2,2,2-trichloroethyl	Me	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
49-36	2,2,2-trichloroethyl	Me	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-37	2,2,2-trichloroethyl	H	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
49-38	2,2,2-trichloroethyl	H	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
49-39	2,2,2-trichloroethyl	H	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-40	2,2,2-trichloroethyl	H	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
49-41	2,2,2-trichloroethyl	H	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
49-42	2,2,2-trichloroethyl	H	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-43	2,2,2-trichloroethyl	H	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
49-44	2,2,2-trichloroethyl	H	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
49-45	2,2,2-trichloroethyl	H	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-46	2,2,2-trichloroethyl	H	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
49-47	2,2,2-trichloroethyl	H	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
49-48	2,2,2-trichloroethyl	H	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-49	2,2,2-trichloroethyl	H	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
49-50	2,2,2-trichloroethyl	H	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
49-51	2,2,2-trichloroethyl	H	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-52	2,2,2-trichloroethyl	H	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
49-53	2,2,2-trichloroethyl	H	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
49-54	2,2,2-trichloroethyl	H	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-55	2,2,2-trichloroethyl	Me	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
49-56	2,2,2-trichloroethyl	Me	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
49-57	2,2,2-trichloroethyl	Me	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-58	2,2,2-trichloroethyl	Me	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
49-59	2,2,2-trichloroethyl	Me	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
49-60	2,2,2-trichloroethyl	Me	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-61	2,2,2-trichloroethyl	Me	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
49-62	2,2,2-trichloroethyl	Me	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
49-63	2,2,2-trichloroethyl	Me	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-64	2,2,2-trichloroethyl	Me	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
49-65	2,2,2-trichloroethyl	Me	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
49-66	2,2,2-trichloroethyl	Me	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-67	2,2,2-trichloroethyl	Me	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
49-68	2,2,2-trichloroethyl	Me	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
49-69	2,2,2-trichloroethyl	Me	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
49-70	2,2,2-trichloroethyl	Me	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
49-71	2,2,2-trichloroethyl	Me	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
49-72	2,2,2-trichloroethyl	Me	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
49-73	2,2,2-trichloroethyl	Me	H	S	H	H	Cl	F	heptafluoroisopropyl	H	OCF3
49-74	2,2,2-trichloroethyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	F	CF3
49-75	2,2,2-trichloroethyl	H	H	S	H	H	CF3	Cl	heptafluoroisopropyl	H	CF3
49-76	2,2,2-trichloroethyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	Cl	OCF3
49-77	2,2,2-trichloroethyl	H	H	S	H	H	Cl	Br	nonafluoro-2-butyl	H	CF3
49-78	2,2,2-trichloroethyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	Br	CF3
49-79	2,2,2-trichloroethyl	H	H	O	H	H	Br	I	heptafluoroisopropyl	H	OCF3
49-80	2,2,2-trichloroethyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	I	CF3
49-81	2,2,2-trichloroethyl	H	H	O	H	H	CF3	Me	heptafluoroisopropyl	H	CF3
49-82	2,2,2-trichloroethyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	Me	OCF3
49-83	2,2,2-trichloroethyl	H	H	O	H	H	Br	F	nonafluoro-2-butyl	F	CF3
49-84	2,2,2-trichloroethyl	H	H	O	H	H	CF3	Cl	nonafluoro-2-butyl	Cl	CF3
49-85	2,2,2-trichloroethyl	H	H	NH	H	H	I	Br	heptafluoroisopropyl	Br	OCF3
49-86	2,2,2-trichloroethyl	H	H	NH	H	H	Cl	I	heptafluoroisopropyl	I	CF3
49-87	2,2,2-trichloroethyl	Me	H	NH	H	H	CF3	F	heptafluoroisopropyl	Me	CF3
49-88	2,2,2-trichloroethyl	H	H	NH	H	H	Br	Cl	nonafluoro-2-butyl	Me	OCF3
49-89	2,2,2-trichloroethyl	H	H	NH	H	H	I	Br	nonafluoro-2-butyl	Me	CF3
49-90	2,2,2-trichloroethyl	H	H	NH	H	H	CF3	I	nonafluoro-2-butyl	Me	CF3

TABLE 50
compound
number	Q2	R1	R2	A	X1	X3	Y1	Y2	Y3	Y4	Y5
50-1	2,2,2-trichloroethyl	H	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
50-2	2,2,2-trichloroethyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
50-3	2,2,2-trichloroethyl	H	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-4	2,2,2-trichloroethyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
50-5	2,2,2-trichloroethyl	H	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
50-6	2,2,2-trichloroethyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-7	2,2,2-trichloroethyl	H	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
50-8	2,2,2-trichloroethyl	H	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
50-9	2,2,2-trichloroethyl	H	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-10	2,2,2-trichloroethyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
50-11	2,2,2-trichloroethyl	H	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
50-12	2,2,2-trichloroethyl	H	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-13	2,2,2-trichloroethyl	H	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
50-14	2,2,2-trichloroethyl	H	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
50-15	2,2,2-trichloroethyl	H	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-16	2,2,2-trichloroethyl	H	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
50-17	2,2,2-trichloroethyl	H	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
50-18	2,2,2-trichloroethyl	H	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-19	2,2,2-trichloroethyl	Me	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
50-20	2,2,2-trichloroethyl	Me	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
50-21	2,2,2-trichloroethyl	Me	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-22	2,2,2-trichloroethyl	Me	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
50-23	2,2,2-trichloroethyl	Me	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
50-24	2,2,2-trichloroethyl	Me	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-25	2,2,2-trichloroethyl	Me	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
50-26	2,2,2-trichloroethyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
50-27	2,2,2-trichloroethyl	Me	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-28	2,2,2-trichloroethyl	Me	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
50-29	2,2,2-trichloroethyl	Me	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
50-30	2,2,2-trichloroethyl	Me	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-31	2,2,2-trichloroethyl	Me	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
50-32	2,2,2-trichloroethyl	Me	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
50-33	2,2,2-trichloroethyl	Me	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-34	2,2,2-trichloroethyl	Me	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
50-35	2,2,2-trichloroethyl	Me	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
50-36	2,2,2-trichloroethyl	Me	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-37	2,2,2-trichloroethyl	H	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
50-38	2,2,2-trichloroethyl	H	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
50-39	2,2,2-trichloroethyl	H	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-40	2,2,2-trichloroethyl	H	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
50-41	2,2,2-trichloroethyl	H	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
50-42	2,2,2-trichloroethyl	H	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-43	2,2,2-trichloroethyl	H	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
50-44	2,2,2-trichloroethyl	H	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
50-45	2,2,2-trichloroethyl	H	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-46	2,2,2-trichloroethyl	H	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
50-47	2,2,2-trichloroethyl	H	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
50-48	2,2,2-trichloroethyl	H	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-49	2,2,2-trichloroethyl	H	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
50-50	2,2,2-trichloroethyl	H	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
50-51	2,2,2-trichloroethyl	H	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-52	2,2,2-trichloroethyl	H	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
50-53	2,2,2-trichloroethyl	H	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
50-54	2,2,2-trichloroethyl	H	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-55	2,2,2-trichloroethyl	Me	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
50-56	2,2,2-trichloroethyl	Me	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
50-57	2,2,2-trichloroethyl	Me	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-58	2,2,2-trichloroethyl	Me	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
50-59	2,2,2-trichloroethyl	Me	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
50-60	2,2,2-trichloroethyl	Me	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-61	2,2,2-trichloroethyl	Me	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
50-62	2,2,2-trichloroethyl	Me	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
50-63	2,2,2-trichloroethyl	Me	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-64	2,2,2-trichloroethyl	Me	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
50-65	2,2,2-trichloroethyl	Me	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
50-66	2,2,2-trichloroethyl	Me	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-67	2,2,2-trichloroethyl	Me	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
50-68	2,2,2-trichloroethyl	Me	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
50-69	2,2,2-trichloroethyl	Me	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
50-70	2,2,2-trichloroethyl	Me	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
50-71	2,2,2-trichloroethyl	Me	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
50-72	2,2,2-trichloroethyl	Me	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
50-73	2,2,2-trichloroethyl	Me	H	S	H	H	Cl	F	heptafluoroisopropyl	H	OCF3
50-74	2,2,2-trichloroethyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	F	CF3
50-75	2,2,2-trichloroethyl	H	H	S	H	H	CF3	Cl	heptafluoroisopropyl	H	CF3
50-76	2,2,2-trichloroethyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	Cl	OCF3
50-77	2,2,2-trichloroethyl	H	H	S	H	H	Cl	Br	nonafluoro-2-butyl	H	CF3
50-78	2,2,2-trichloroethyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	Br	CF3
50-79	2,2,2-trichloroethyl	H	H	O	H	H	Br	I	heptafluoroisopropyl	H	OCF3
50-80	2,2,2-trichloroethyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	I	CF3
50-81	2,2,2-trichloroethyl	H	H	O	H	H	CF3	Me	heptafluoroisopropyl	H	CF3
50-82	2,2,2-trichloroethyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	Me	OCF3
50-83	2,2,2-trichloroethyl	H	H	O	H	H	Br	F	nonafluoro-2-butyl	F	CF3
50-84	2,2,2-trichloroethyl	H	H	O	H	H	CF3	Cl	nonafluoro-2-butyl	Cl	CF3
50-85	2,2,2-trichloroethyl	H	H	NH	H	H	I	Br	heptafluoroisopropyl	Br	OCF3
50-86	2,2,2-trichloroethyl	H	H	NH	H	H	Cl	I	heptafluoroisopropyl	I	CF3
50-87	2,2,2-trichloroethyl	Me	H	NH	H	H	CF3	F	heptafluoroisopropyl	Me	CF3
50-88	2,2,2-trichloroethyl	H	H	NH	H	H	Br	Cl	nonafluoro-2-butyl	Me	OCF3
50-89	2,2,2-trichloroethyl	H	H	NH	H	H	I	Br	nonafluoro-2-butyl	Me	CF3
50-90	2,2,2-trichloroethyl	H	H	NH	H	H	CF3	I	nonafluoro-2-butyl	Me	CF3

TABLE 51
compound
number	Q2	R1	R2	A	X1	X2	Y1	Y2	Y3	Y4	Y5
51-1	2,2,2-trichloroethyl	H	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
51-2	2,2,2-trichloroethyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
51-3	2,2,2-trichloroethyl	H	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-4	2,2,2-trichloroethyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
51-5	2,2,2-trichloroethyl	H	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
51-6	2,2,2-trichloroethyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-7	2,2,2-trichloroethyl	H	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
51-8	2,2,2-trichloroethyl	H	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
51-9	2,2,2-trichloroethyl	H	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-10	2,2,2-trichloroethyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
51-11	2,2,2-trichloroethyl	H	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
51-12	2,2,2-trichloroethyl	H	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-13	2,2,2-trichloroethyl	H	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
51-14	2,2,2-trichloroethyl	H	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
51-15	2,2,2-trichloroethyl	H	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-16	2,2,2-trichloroethyl	H	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
51-17	2,2,2-trichloroethyl	H	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
51-18	2,2,2-trichloroethyl	H	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-19	2,2,2-trichloroethyl	Me	H	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
51-20	2,2,2-trichloroethyl	Me	H	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
51-21	2,2,2-trichloroethyl	Me	H	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-22	2,2,2-trichloroethyl	Me	H	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
51-23	2,2,2-trichloroethyl	Me	H	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
51-24	2,2,2-trichloroethyl	Me	H	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-25	2,2,2-trichloroethyl	Me	H	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
51-26	2,2,2-trichloroethyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	H	CF3
51-27	2,2,2-trichloroethyl	Me	H	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-28	2,2,2-trichloroethyl	Me	H	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
51-29	2,2,2-trichloroethyl	Me	H	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
51-30	2,2,2-trichloroethyl	Me	H	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-31	2,2,2-trichloroethyl	Me	H	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
51-32	2,2,2-trichloroethyl	Me	H	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
51-33	2,2,2-trichloroethyl	Me	H	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-34	2,2,2-trichloroethyl	Me	H	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
51-35	2,2,2-trichloroethyl	Me	H	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
51-36	2,2,2-trichloroethyl	Me	H	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-37	2,2,2-trichloroethyl	H	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
51-38	2,2,2-trichloroethyl	H	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
51-39	2,2,2-trichloroethyl	H	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-40	2,2,2-trichloroethyl	H	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
51-41	2,2,2-trichloroethyl	H	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
51-42	2,2,2-trichloroethyl	H	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-43	2,2,2-trichloroethyl	H	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
51-44	2,2,2-trichloroethyl	H	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
51-45	2,2,2-trichloroethyl	H	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-46	2,2,2-trichloroethyl	H	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
51-47	2,2,2-trichloroethyl	H	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
51-48	2,2,2-trichloroethyl	H	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-49	2,2,2-trichloroethyl	H	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
51-50	2,2,2-trichloroethyl	H	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
51-51	2,2,2-trichloroethyl	H	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-52	2,2,2-trichloroethyl	H	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
51-53	2,2,2-trichloroethyl	H	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
51-54	2,2,2-trichloroethyl	H	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-55	2,2,2-trichloroethyl	Me	Me	S	H	H	Cl	H	heptafluoroisopropyl	H	OCF3
51-56	2,2,2-trichloroethyl	Me	Me	S	H	H	Br	H	heptafluoroisopropyl	H	CF3
51-57	2,2,2-trichloroethyl	Me	Me	S	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-58	2,2,2-trichloroethyl	Me	Me	S	H	H	I	H	nonafluoro-2-butyl	H	OCF3
51-59	2,2,2-trichloroethyl	Me	Me	S	H	H	Cl	H	nonafluoro-2-butyl	H	CF3
51-60	2,2,2-trichloroethyl	Me	Me	S	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-61	2,2,2-trichloroethyl	Me	Me	O	H	H	Br	H	heptafluoroisopropyl	H	OCF3
51-62	2,2,2-trichloroethyl	Me	Me	O	H	H	I	H	heptafluoroisopropyl	H	CF3
51-63	2,2,2-trichloroethyl	Me	Me	O	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-64	2,2,2-trichloroethyl	Me	Me	O	H	H	Cl	H	nonafluoro-2-butyl	H	OCF3
51-65	2,2,2-trichloroethyl	Me	Me	O	H	H	Br	H	nonafluoro-2-butyl	H	CF3
51-66	2,2,2-trichloroethyl	Me	Me	O	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-67	2,2,2-trichloroethyl	Me	Me	NH	H	H	I	H	heptafluoroisopropyl	H	OCF3
51-68	2,2,2-trichloroethyl	Me	Me	NH	H	H	Cl	H	heptafluoroisopropyl	H	CF3
51-69	2,2,2-trichloroethyl	Me	Me	NH	H	H	CF3	H	heptafluoroisopropyl	H	CF3
51-70	2,2,2-trichloroethyl	Me	Me	NH	H	H	Br	H	nonafluoro-2-butyl	H	OCF3
51-71	2,2,2-trichloroethyl	Me	Me	NH	H	H	I	H	nonafluoro-2-butyl	H	CF3
51-72	2,2,2-trichloroethyl	Me	Me	NH	H	H	CF3	H	nonafluoro-2-butyl	H	CF3
51-73	2,2,2-trichloroethyl	Me	H	S	H	H	Cl	F	heptafluoroisopropyl	H	OCF3
51-74	2,2,2-trichloroethyl	H	H	S	H	H	Br	H	heptafluoroisopropyl	F	CF3
51-75	2,2,2-trichloroethyl	H	H	S	H	H	CF3	Cl	heptafluoroisopropyl	H	CF3
51-76	2,2,2-trichloroethyl	H	H	S	H	H	I	H	nonafluoro-2-butyl	Cl	OCF3
51-77	2,2,2-trichloroethyl	H	H	S	H	H	Cl	Br	nonafluoro-2-butyl	H	CF3
51-78	2,2,2-trichloroethyl	H	H	S	H	H	CF3	H	nonafluoro-2-butyl	Br	CF3
51-79	2,2,2-trichloroethyl	H	H	O	H	H	Br	I	heptafluoroisopropyl	H	OCF3
51-80	2,2,2-trichloroethyl	Me	H	O	H	H	I	H	heptafluoroisopropyl	I	CF3
51-81	2,2,2-trichloroethyl	H	H	O	H	H	CF3	Me	heptafluoroisopropyl	H	CF3
51-82	2,2,2-trichloroethyl	H	H	O	H	H	Cl	H	nonafluoro-2-butyl	Me	OCF3
51-83	2,2,2-trichloroethyl	H	H	O	H	H	Br	F	nonafluoro-2-butyl	F	CF3
51-84	2,2,2-trichloroethyl	H	H	O	H	H	CF3	Cl	nonafluoro-2-butyl	Cl	CF3
51-85	2,2,2-trichloroethyl	H	H	NH	H	H	I	Br	heptafluoroisopropyl	Br	OCF3
51-86	2,2,2-trichloroethyl	H	H	NH	H	H	Cl	I	heptafluoroisopropyl	I	CF3
51-87	2,2,2-trichloroethyl	Me	H	NH	H	H	CF3	F	heptafluoroisopropyl	Me	CF3
51-88	2,2,2-trichloroethyl	H	H	NH	H	H	Br	Cl	nonafluoro-2-butyl	Me	OCF3
51-89	2,2,2-trichloroethyl	H	H	NH	H	H	I	Br	nonafluoro-2-butyl	Me	CF3
51-90	2,2,2-trichloroethyl	H	H	NH	H	H	CF3	I	nonafluoro-2-butyl	Me	CF3

Hereinbelow, Table 52 shows the physical properties of the representative compounds of the amide derivative of the present invention. The ¹H-NMR chemical shill values shown therein are based on tetramethylsilane as an internal standard substance unless specified otherwise.

TABLE 52
com-
pound
number  1H-NMR (CDCl3, ppm)
1-470   δ 7.55-7.68 (3H, m), 7.80-7.99 (6H, m), 8.58 (1H, s), 8.61 (1H, s), 9.12 (1H, d, J = 1.5 Hz).
1-491   δ 7.34-7.91 (4H, m), 8.00 (1H, s), 8.08 (2H, dd, J = 1.9, 6.8 Hz), 8.00 (1H, s), 8.49 (1H, s), 8.59 (1H, s),
        9.04 (1H, s).
1-506   δ 7.48 (1H, dd, J = 4.9, 7.81 Hz), 7.83-7.90 (3H, m), 8.00 (1H, s), 8.31 (1H, dd, J = 1.9, 7.8 Hz), 8.34 (1H, s),
        8.61 (1H, dd, J = 1.9, 4.9 Hz), 9.09 (1H, s), 9.10 (1H, s).
1-513   δ 7.54 (1H, d, J = 7.8 Hz), 7.83-7.90 (3H, m), 8.00 (1H, s), 8.21 (1H, dd, J = 2.4, 8.3 Hz), 8.31 (1H, s),
        8.51 (1H, s), 9.00 (1H, s), 9.01 (1H, d, J = 7.8 Hz).
1-627   δ 7.56-7.59 (3H, m), 7.64-7.66 (1H, m), 7.80-7.87 (2H, m), 7.94-7.97 (2H, m), 8.16 (1H, s), 8.46 (1H, s),
        8.57 (1H, s), 9.16 (1H, s).
1-1925  δ 7.52-7.59 (2H, m), 7.65-7.71 (2H, m), 7.93-7.95 (2H, m), 8.00-8.02 (2H, m), 8.12-8.16 (2H, m), 8.52 (1H, d, J = 11.2 Hz).
1-1968  δ 7.54 (1H, d J = 8.8 Hz), 7.72 (1H, d J = 8.8 Hz), 7.93 (1H, s), 8.09 (1H, s), 8.17-8.18 (2H, m), 8.27 (1H, dd, J = 2.4,
        8.8 Hz), 8.38 (1H, d J = 10.8 Hz), 8.98 (1H, d, J = 2.4 Hz).
2-491   δ 3.81 (3H, broad-s), 7.52-7.84 (8H, m), 7.89 (1H, s), 8.00 (1H, s).
2-513   δ 3.58 (3H, s), 7.34-7.36 (1H, m), 7.81-8.00 (8H, m).
2-518   δ 3.59 (3H, s), 7.69 (1H, broad-s), 7.81-8.01 (7H, m), 8.50 (1H, broad-s).
6-38    δ 7.51-7.62 (4H, m), 7.75-8.00 (8H, m), 8.32 (1H, s).
6-39    δ 7.22 (1H, dd, J = 8.0, 12.4 Hz), 7.32-7.36 (1H, m), 7.51-7.55 (2H, m), 7.78 (1H, d, J = 7.6 Hz),
        7.86-7.90 (3H, m), 8.11 (1H, s), 8.17-8.18 (1H, m), 8.35 (1H, s), 8.62-8.67 (1H, m).
6-45    δ 7.57-7.59 (1H, m), 7.65-7.69 (1H, m), 7.77-7.79 (1H, m), 7.89-7.9 (5H, m), 8.14-8.29 (4H, m).
6-46    δ 7.55-7.59 (1H, m), 7.77-8.07 (10H, m), 8.27 (1H, s).
6-47    δ 7.01-7.05 (2H, m), 7.44-7.56 (2H, m), 7.78-7.86 (4H, m), 8.03 (1H, s), 8.11 (1H, s), 8.33 (1H, s).
6-57    δ 7.28-7.32 (1H, m), 7.45-7.67 (4H, m), 7.76-8.02 (5H, m), 8.30 (1H, s).
6-60    δ 7.50-7.60 (2H, m), 7.78-8.02 (6H, m), 8.19-8.27 (2H, m), 8.91 (1H, s).
6-71    δ 7.51-7.62 (4H, m), 7.78-7.80 (1H, d, J = 8.0 Hz), 7.90-7.92 (3H, m), 8.06-8.09 (4H, m), 8.34 (1H, s).
6-72    δ 7.22-7.25 (1H, m), 7.35 (1H, t, J = 8.0 Hz), 7.55-7.60 (2H, m), 7.80 (1H, d, J = 8.0 Hz), 7.92 (1H, d, J = 8.0 Hz),
        8.01 (1H, s), 8.10 (2H, s), 8.20 (1H, t, J = 8.0 Hz), 8.37 (1H, s), 8.65 (1H, d, J = 16.8 Hz).
6-78    δ 7.58 (1H, t, J = 7.8 Hz), 7.68 (1H, t, J = 7.8), 7.80 (1H, d, J = 8.0 Hz), 7.87 (1H, d, 8.0 Hz), 7.95 (1H, d, J = 8.0 Hz),
        8.00 (1H, s), 8.09 (2H, s), 8.15 (1H, d, J = 8.0 Hz), 8.23 (1H, s), 8.26 (1H, s), 8.30 (1H, s).
6-79    δ 7.58 (1H, t, J = 8.2 Hz), 7.79-7.83 (3H, m), 7.97 (2H, s), 8.01 (2H, d, J = 8.0 Hz), 8.09 (2H, s), 8.18 (1H, s),
        8.29 (1H, s).
6-80    δ 7.05 (2H, t, J = 8.2 Hz), 7.48 (1H, t, J = 6.6 Hz), 7.56 (1H, t, J = 7.8 Hz), 7.81 (1H, d, J = 8.0 Hz), 7.89-7.91 (2H,
        m), 7.98 (1H, s), 8.10 (2H, s), 8.33 (1H, s).
6-90    δ 7.43-7.46 (1H, m), 7.59 (1H, t, J = 7.2 Hz), 7.82 (1H, d, J = 7.2 Hz), 7.93 (2H, d, J = 9.6 Hz), 8.10 (2H, s),
        8.24 (1H, d, J = 6.4 Hz), 8.33 (1H, s), 8.44 (1H, s), 8.56 (1H, s).
6-93    δ 7.51 (1H, d, J = 8.4 Hz), 7.59 (1H, t, J = 7.6 Hz), 7.81 (1H, d, J = 7.6 Hz), 7.94 (2H, s), 8.10-8.11 (3H, m),
        8.20 (1H, d, J = 8.0 Hz), 8.28 (1H, s), 8.91 (1H, s).
6-111   (DMSO-d6) δ 7.50-7.60 (4H, m), 7.70-7.73 (1H, m), 7.93-8.00 (3H, m), 8.04-8.08 (1H, m), 8.34-8.36 (2H, m),
        10.48 (1H, s), 10.60 (1H, s).
6-147   (DMSO-d6) δ 7.55-7.61 (2H, m), 7.74 (1H, d, J = 7.9 Hz), 7.94-7.97 (2H, m), 8.10 (1H, dd, J = 2.0, 7.6 Hz),
        8.27 (1H, s), 8.34 (1H, s), 8.54 (1H, dd, J = 2.0, 4.9 Hz), 10.65 (1H, s), 10.89 (1H, s).
6-268   δ 7.50-7.61 (4H, m), 7.70 (1H, d, J = 7.8 Hz), 7.85-7.92 (4H, m), 7.96-8.01 (2H, m), 8.14 (1H, s), 8.24 (1H, t,
        J = 2.0 Hz).
6-269   δ 7.22-7.25 (1H, m), 7.36 (1H, t, J = 8.0 Hz), 7.56-7.57 (2H, m), 7.75 (1H, d, J = 8.0 Hz), 7.90-8.00 (2H, m),
        8.07 (1H, s), 8.17-8.20 (2H, m), 8.33 (1H, s), 8.65 (1H, d, J = 16.4 Hz).
6-270   δ 7.25 (1H, t, J = 8.0 Hz), 7.43-7.53 (2H, m), 7.77-7.81 (4H, m), 7.85 (1H, d, J = 8.0 Hz), 7.91 (1H, s), 8.13 (1H,
        s), 8.19 (1H, d, J = 8.0 Hz), 8.24 (1H, s).
6-271   δ 7.09-7.22 (2H, m), 7.55 (1H, t, J = 7.8 Hz), 7.71 (1H, d, J = 8.0 Hz), 7.89-7.93 (4H, m), 8.03 (2H, d, J = 8.0 Hz),
        8.14 (1H, s), 8.23 (1H, s).
6-272   δ 7.40-7.50 (4H, m), 7.56 (1H, t, J = 8.0 Hz), 7.80 (2H, t, J = 8.4 Hz), 7.87 (2H, s), 7.91 (1H, d, J = 7.9 Hz),
        8.09 (1H, s), 8.32 (1H, s).
6-288   δ 7.54-7.55 (1H, m), 7.65-7.66 (1H, m), 7.72 (1H, d, J = 7.8 Hz), 7.85 (1H, d, J = 7.8 Hz), 7.91 (1H, s),
        7.95-7.98 (2H, m), 8.13-8.23 (4H, m), 8.36 (1H, s).
6-289   δ 7.55-7.56 (1H, m), 7.71 (1H, d, J = 7.8 Hz), 7.80 (2H, d, J = 8.3 Hz), 7.91-7.96 (3H, m), 7.99 (2H, d, J = 8.3 Hz),
        8.20 (1H, s), 8.21-8.22 (2H, m).
6-290   δ 7.01-7.05 (2H, m), 7.42-7.44 (1H, m), 7.55 (1H, t, J = 8.0 Hz), 7.75 (1H, d, J = 8.0 Hz), 7.90-7.95 (3H, m),
        8.01 (1H, s), 8.14 (1H, s), 8.26 (1H, s).
6-293   δ 7.14 (1H, t, J = 8.0 Hz), 7.22-7.29 (2H, m), 7.54 (1H, t, J = 7.8 Hz), 7.74 (1H, d, J = 7.8 Hz), 7.84-7.88 (3H, m),
        8.11 (1H, s), 8.15 (1H, s), 8.25 (1H, s).
6-300   δ 7.06-7.59 (2H, m), 7.62 (1H, dd, J = 1.5, 7.8 Hz), 7.81 (1H, d, J = 7.8 Hz), 7.92 (1H, s), 8.08-8.16 (4H, m),
        9.35-9.40 (1H, m), 9.51 (1H, broad-s).
6-304   δ 7.44 (1H, dd, J = 4.9, 7.8 Hz), 7.58 (1H, t, J = 7.8 Hz), 7.75 (1H, d, J = 7.8 Hz), 7.81 (1H, s), 7.92-7.96 (2H,
        m), 8.15 (1H, s), 8.22-8.26 (2H, m), 8.38 (1H, s), 8.55 (1H, dd, J = 2.0, 4.9 Hz).
6-306   δ 7.42-7.45 (1H, m), 7.58 (1H, t, J = 7.8 Hz), 7.75 (1H, d, J = 7.8 Hz), 7.88 (1H, broad-s), 7.93-7.95 (2H, m),
        8.15 (1H, broad-s), 8.23 (1H, dd, J = 2.0, 7.8 Hz), 8.24 (1H, s), 8.39 (1H, broad-s), 8.55 (1H, dd, J = 2.0, 4.8 Hz).
6-311   δ 7.45-7.52 (1H, m), 7.74 (1H, d, J = 8.0 Hz), 7.92-7.96 (1H, m), 8.00 (1H, s), 8.14 (1H, s), 8.22-8.23 (3H, m),
        8.29 (1H, d, J = 8.0 Hz), 8.91 (1H, s), 9.07 (1H, s).
6-346   δ 7.50-7.62 (4H, m), 7.71-7.73 (1H, m), 7.89-7.93 (4H, m), 8.02-8.04 (2H, m), 8.13 (1H, s), 8.27 (1H, s).
6-347   δ 7.19-7.25 (1H, m), 7.33-7.37 (1H, m), 7.52-7.59 (2H, m), 7.73-7.75 (1H, m), 7.89-7.91 (2H, m),
        8.09-8.21 (3H, m), 8.31 (1H, s), 8.65 (1H, s).
6-348   δ 7.30-7.31 (1H, m), 7.48-7.74 (5H, m), 7.91-7.92 (2H, m), 8.02 (1H, s), 8.07 (1H, s), 8.13 (1H, s),
        8.25 (1H, s).
6-349   δ 7.17-7.21 (2H, m), 7.51-7.55 (1H, m), 7.70-7.72 (1H, m), 7.88-7.93 (4H, m), 8.04 (1H, s), 8.11-8.23 (2H,
        m), 8.23 (1H, s).
6-366   δ 7.53-7.55 (1H, m), 7.62-7.72 (2H, m), 7.84-7.94 (3H, m), 8.09-8.16 (3H, m), 8.22-8.24 (2H, m), 8.40 (1H,
        s).
6-367   δ 7.54-7.58 (1H, m), 7.72-7.74 (1H, m), 7.80-7.83 (2H, m), 7.91-7.94 (2H, m), 8.00-8.07 (2H, m), 8.13 (1H,
        s), 8.18 (1H, s), 8.23 (1H, s), 8.24 (1H, s).
6-368   δ 7.01-7.06 (2H, m), 7.44-7.57 (3H, m), 7.74-7.76 (1H, m), 7.86-7.91 (2H, m), 8.07 (1H, s), 8.13-8.14 (1H,
        m), 8.28 (1H, s).
6-382   δ 7.43-7.46 (1H, m), 7.56-7.60 (1H, m), 7.76-7.78 (1H, m), 7.90-7.91 (2H, m), 8.02 (1H, s), 8.14 (1H, s),
        8.25 (2H, s), 8.43 (1H, s), 8.54-8.56 (1H, m).
6-389   δ 7.30-7.60 (2H, m), 7.74-7.76 (1H, m), 7.91-7.98 (3H, m), 8.07 (1H, s), 8.14 (1H, s), 8.19-8.23 (2H, m),
        8.90 (1H, s).
6-424   δ 7.51-7.62 (4H, m), 7.73 (1H, d, J = 8.3 Hz), 7.89-7.94 (4H, m), 8.01 (1H, s), 8.10 (1H, s), 8.27 (1H, t, J = 1.5 Hz),
        8.35 (1H, s).
6-425   δ 7.20-7.25 (1H, m), 7.34-7.37 (1H, m), 7.54-7.58 (2H, m), 7.75 (1H, d, J = 7.6 Hz), 7.88-7.95 (2H, m),
        8.18-8.22 (2H, m), 8.33-8.34 (2H, m), 8.66 (1H, d, J = 16.4 Hz).
6-426   δ 7.28-7.30 (1H, m), 7.46-7.66 (5H, m), 7.71-7.94 (2H, m), 8.11-8.24 (3H, m), 8.34 (1H, s).
6-427   δ 7.18-7.22 (2H, m), 7.52-7.57 (1H, m), 7.73 (1H, d, J = 7.6 Hz), 7.89-8.03 (5H, m), 8.22-8.25 (2H, m),
        8.35 (1H, s).
6-428   δ 7.42-7.50 (4H, m), 7.56 (1H, t, J = 8.0 Hz), 7.75 (1H, d, J = 8.0 Hz), 7.81 (1H, d, J = 7.8 Hz), 7.95-7.96 (2H, m),
        8.09 (1H, s), 8.28 (1H, s), 8.36 (1H, s).
6-444   δ 7.56 (1H, t, J = 7.8 Hz), 7.66 (1H, t, J = 7.8 Hz), 7.73 (1H, t, J = 7.8 Hz), 7.86 (1H, dd, J = 1.5, 7.8 Hz),
        7.93-7.96 (2H, m), 8.07 (1H, s), 8.14-8.16 (1H, m), 8.22-8.26 (3H, m), 8.34 (1H, s).
6-445   δ 7.57 (1H, t, J = 7.8 Hz), 7.74 (1H, d, J = 7.8 Hz), 7.81-7.83 (2H, m), 7.95 (1H, s), 7.97-8.04 (4H, m),
        8.12 (1H, broad-s), 8.23 (1H, t, J = 2.0 Hz), 8.35 (1H, broad-s).
6-446   δ 7.01-7.05 (2H, m), 7.43-7.57 (2H, m), 7.75-7.77 (1H, m), 7.88-7.94 (3H, m), 8.13 (1H, s), 8.27 (1H, s),
        8.35 (1H, s).
6-448   δ 7.39-7.41 (1H, m), 7.51-7.58 (2H, m), 7.74-7.78 (2H, m), 7.90-7.95 (2H, m), 8.04 (1H, s), 8.15 (1H, s),
        8.26 (1H, s), 8.35 (1H, s).
6-449   δ 7.12-7.36 (3H, m), 7.52-7.58 (1H, m), 7.75-7.95 (4H, m), 8.21-8.35 (3H, m).
6-450   6.82-6.86 (1H, m), 7.00-7.01 (1H, m), 7.15 (1H, t, J = 7.8 Hz), 7.56 (1H, t, J = 8.2 Hz), 7.74 (1H, d, J = 8.1 Hz),
        7.84 (1H, t, J = 8.8 Hz), 7.90-7.91 (1H, m), 7.95 (1H, s), 8.04 (1H, s), 8.42 (1H, s).
6-451   δ 7.23-7.69 (8H, m), 7.85 (1H, s), 8.04 (1H, s), 8.42 (1H, s).
6-452   δ 7.44 (1H, dd, J = 2.0, 8.3 Hz), 7.59 (1H, t, J = 8.3 Hz), 7.66 (1H, d, J = 8.3 Hz), 7.70 (1H, d, J = 2.0 Hz),
        7.75 (1H, d, J = 8.3 Hz), 7.86 (2H, broad-s), 7.95 (2H, broad-s), 8.24 (1H, broad-s), 8.37 (1H, broad-s).
6-453   δ 7.15 (1H, dt, J = 2.4, 8.3 Hz), 7.40 (1H, dd, J = 2.4, 8.3 Hz), 7.60 (1H, t, J = 8.3 Hz), 7.68-7.74 (2H, m),
        7.95-8.02 (4H, m), 8.24 (1H, s), 8.35 (1H, s).
6-454   δ 7.59 (1H, t, J = 7.8 Hz), 7.75 (1H, d, J = 7.8 Hz), 7.93 (1H, s), 7.95-7.99 (3H, m), 8.10 (1H, broad-s),
        8.23-8.26 (2H, m), 8.36 (2H, d, J = 1.9 Hz).
6-460   δ 7.43-7.46 (1H, m), 7.58 (1H, t, J = 7.8 Hz), 7.77 (1H, d, J = 7.8 Hz), 7.91-7.95 (2H, m), 8.01 (1H, s),
        8.24 (1H, dd, J = 2.0, 7.8 Hz), 8.28 (1H, s), 8.36 (1H, s), 8.41 (1H, s), 8.54-8.56 (1H, m).
6-461   δ 7.45 (1H, dd, J = 4.9, 7.3 Hz), 7.59 (1H, t, J = 7.8 Hz), 7.77 (1H, d, J = 7.8 Hz), 7.92-7.99 (3H, m),
        8.24-8.29 (2H, m), 8.36-8.39 (2H, m), 8.55 (1H, dd, J = 2.0, 4.9 Hz).
6-467   δ 7.45-7.60 (2H, m), 7.74 (1H, d, J = 8.0 Hz), 7.95-7.97 (2H, m), 8.03 (1H, s), 8.12 (1H, s), 8.19-8.35 (2H,
        m), 8.35 (1H, s), 8.90 (1H, s).
6-502   δ 7.51-7.62 (4H, m), 7.73 (1H, d, J = 7.6 Hz), 7.89-7.95 (4H, m), 8.01 (2H, d, J = 14.4 Hz), 8.27 (1H, s), 8.34 (1H,
        s).
6-503   δ 7.20-7.23 (1H, m), 7.34 (1H, t, J = 7.8 Hz), 7.54-7.60 (2H, m), 7.74 (1H, d, J = 7.8 Hz), 7.94 (2H, s), 8.05 (1H,
        s), 8.19 (1H, t, J = 7.8 Hz), 8.33 (2H, d, J = 12.0 Hz), 8.65 (1H, d, J = 16.0 Hz).
6-504   δ 7.47-7.69 (5H, m), 7.73 (1H, d, J = 7.8 Hz), 7.93 (2H, s), 8.05 (2H, d, J = 11.0 Hz), 8.25 (1H, s), 8.34 (1H, s).
6-505   δ 7.20 (2H, t, J = 7.8 Hz), 7.56 (1H, t, J = 8.0 Hz), 7.73 (1H, d, J = 8.2 Hz), 7.91-7.94 (5H, m), 8.02 (1H, s),
        8.24 (1H, s), 8.35 (1H, s).
6-522   δ 7.68-7.75 (2H, m), 7.86 (1H, d, J = 8.2 Hz), 7.93-7.96 (2H, m), 8.08 (1H, s), 8.14 (1H, d, J = 8.0 Hz), 8.24 (2H,
        d, J = 8.2 Hz), 8.28 (1H, s), 8.33 (1H, s), 8.62 (1H, s).
6-523   δ 7.57 (1H, t, J = 7.8 Hz), 7.82 (2H, d, J = 8.0 Hz), 7.93-8.02 (6H, m), 8.14 (1H, s), 8.23 (1H, s), 8.34 (1H, s).
6-524   δ 7.05 (2H, t, J = 8.0 Hz), 7.43-7.50 (1H, m), 7.56 (1H, t, J = 8.0 Hz), 7.75 (1H, d, J = 7.8 Hz), 7.86 (1H, s),
        7.92 (2H, d, J = 8.2 Hz), 8.00 (1H, s), 8.27 (1H, s), 8.34 (1H, s).
6-538   δ 7.45 (1H, t, J = 7.6 Hz), 7.59 (2H, s), 7.70 (1H, d, J = 4.0 Hz), 7.93 (2H, d, J = 7.6 Hz), 7.98 (1H, s), 8.28 (1H, s),
        8.34 (2H, d, J = 7.6 Hz), 8.41 (1H, s).
6-545   δ 7.56-7.60 (1H, m), 7.75 (1H, d, J = 8.0 Hz), 7.92-8.00 (4H, m), 8.09 (1H, s), 8.19-8.23 (2H, m), 8.35 (1H, s),
        8.90 (1H, s).
6-804   δ 7.50-7.62 (4H, m), 7.68-7.70 (1H, m), 7.85-7.91 (3H, m), 8.10 (1H, s), 8.16-8.22 (4H, m).
6-824   δ 7.55-7.59 (2H, m), 7.66-7.76 (2H, m), 7.86-7.92 (2H, m), 7.99-8.08 (2H, m), 8.13-8.22 (2H, m),
        8.39-8.43 (2H, m).
6-825   δ 7.55-7.59 (2H, m), 7.66-7.70 (2H, m), 7.72-7.73 (2H, m), 7.86-7.92 (2H, m), 7.99-8.22 (3H, m),
        8.40-8.42 (1H, m).
6-840   δ 7.42-7.45 (1H, m), 7.55-7.59 (1H, t, J = 7.8 Hz), 7.71-7.30 (1H, d, J = 7.8 Hz), 7.88-7.91 (1H, m), 8.00 (1H,
        s), 8.20-8.24 (4H, m), 8.41 (1H, s), 8.54-8.55 (1H, m).
6-1104  δ 7.40 (1H, t, J = 7.8 Hz), 7.53-7.64 (3H, m), 7.89 (2H, s), 7.90-7.95 (3H, m), 8.11-8.14 (2H, m),
        8.69-8.70 (1H, m).
6-1105  δ 7.22-7.26 (1H, m), 7.35-7.41 (2H, m), 7.58 (1H, d, J = 8.0 Hz), 7.88-7.92 (3H, m), 8.15-8.25 (2H, m),
        8.74-8.75 (2H, m).
6-1106  δ 7.35-7.34 (1H, m), 7.417.42 (1H, m), 7.53-7.54 (1H, m), 7.67-7.68 (2H, m), 7.89-7.90 (3H, m),
        8.09-8.10 (2H, m), 8.66-8.68 (1H, m).
6-1107  δ 7.21-7.26 (2H, m), 7.39-7.41 (1H, m), 7.89-7.96 (4H, m), 8.05-8.13 (3H, m), 8.70-8.72 (1H, m).
6-1124  δ 7.42-7.43 (1H, m), 7.70-7.72 (1H, m), 7.89-7.92 (4H, m), 8.09-8.17 (3H, m), 8.22 (1H, s), 8.62-8.63 (1H,
        m).
6-1125  δ 7.42-7.44 (1H, m), 7.84-7.94 (5H, m), 8.02-8.11 (4H, m), 8.63-8.64 (1H, m).
6-1126  δ 7.05-7.09 (2H, m), 7.38-7.42 (1H, m), 7.49-7.50 (1H, m), 7.88-7.99 (4H, m), 8.09-8.12 (1H, m),
        8.71-8.72 (1H, m).
6-1140  δ 7.40-7.49 (2H, m), 7.89 (2H, s), 7.94-7.96 (1H, m), 8.13 (1H, d, J = 12.7 Hz), 8.32-8.34 (1H, m),
        8.57-8.59 (1H, m), 8.67-8.71 (1H, m), 8.75 (1H, broad-s).
6-1147  δ 7.39-7.44 (1H, m), 7.52-7.55 (1H, m), 7.89 (1H, s), 7.96-7.98 (1H, m), 8.05-8.11 (3H, m), 8.21-8.23 (1H,
        m), 8.61-8.62 (1H, m), 8.93 (1H, s).
6-1182  δ 7.37-7.41 (1H, m), 7.53-7.64 (3H, m), 7.87-7.94 (5H, m), 8.11-8.14 (2H, m), 8.67-8.71 (1H, m).
6-1183  δ 7.35-7.41 (2H, m), 7.58-7.61 (1H, m), 7.86-7.92 (3H, m), 8.17-8.25 (2H, m), 8.61 (1H, s), 8.74 (1H, t, J = 7.8 Hz),
        8.90-8.93 (1H, m).
6-1184  δ 7.33 (1H, t, J = 8.0 Hz), 7.40 (1H, t, J = 7.8 Hz), 7.50-7.56 (1H, m), 7.64-7.69 (2H, m), 7.88 (2H, s), 7.92 (1H, t,
        J = 7.8 Hz), 8.09-8.12 (2H, m), 8.63 (1H, t, J = 8.2 Hz).
6-1185  δ 7.22 (2H, t, J = 7.8 Hz), 7.29-7.30 (1H, m), 7.40 (1H, t, J = 8.0 Hz), 7.88 (2H, s), 7.90-7.97 (2H, m), 8.05 (1H, s),
        8.10-8.13 (1H, m), 8.64 (1H, t, J = 7.8 Hz).
6-1202  δ 7.42-7.44 (1H, m), 7.68-7.72 (1H, m), 7.88-7.94 (4H, m), 8.10-8.23 (4H, m), 8.60-8.65 (1H, m).
6-1203  δ 7.39-7.44 (1H, m), 7.84-7.88 (4H, m), 7.92-7.95 (1H, m), 8.02-8.13 (4H, m), 8.61-8.65 (1H, m).
6-1204  δ 7.05 (2H, t, J = 8.0 Hz), 7.40 (1H, t, J = 8.0 Hz), 7.48-7.52 (1H, m), 7.87 (2H, s), 7.92 (1H, t, J = 8.0 Hz),
        8.01 (1H, s), 8.11-8.14 (1H, m), 8.68 (1H, t, J = 7.4 Hz).
6-1218  δ 7.40-7.49 (2H, m), 7.95 (2H, s), 7.94 (1H, t, J = 7.8 Hz), 8.12-8.16 (1H, m), 8.34 (1H, d, J = 8.0 Hz), 8.58 (1H,
        s), 8.70 (1H, t, J = 7.8 Hz), 8.77 (1H, s).
6-1225  δ 7.42 (1H, t, J = 8.2 Hz), 7.53 (1H, d, J = 8.0 Hz), 7.88 (2H, s), 7.94 (1H, t, J = 7.0 Hz), 8.06 (1H, s),
        8.09-8.12 (1H, m), 8.20-8.23 (1H, m), 8.60 (1H, t, J = 8.0 Hz), 8.93 (1H, s).
6-1260  δ 7.39 (1H, t, J = 7.8 Hz), 7.52-7.57 (4H, m), 7.60-7.63 (2H, m), 7.93-7.94 (4H, m), 8.70 (1H, t, J = 6.3 Hz).
6-1261  δ 7.22-7.28 (1H, m), 7.35-7.42 (2H, m), 7.59-7.61 (1H, m), 7.94-7.95 (1H, m), 8.12 (2H, s), 8.15-8.25 (2H,
        m), 8.78 (1H, t, J = 1.5 Hz), 9.00 (1H, d, J = 7.8 Hz).
6-1262  δ 7.30-7.33 (1H, m), 7.40-7.44 (1H, m), 7.52-7.55 (2H, m), 7.64-7.70 (3H, m), 7.95-7.96 (1H, m),
        8.09-8.13 (2H, m), 8.67-8.68 (1H, m).
6-1263  δ 7.20-7.26 (3H, m), 7.38-7.42 (1H, m), 7.91-7.98 (3H, m), 8.07-8.12 (3H, m), 8.63-8.67 (1H, m).
6-1280  δ 7.41-7.45 (1H, m), 7.68-7.72 (1H, m), 7.90-7.99 (2H, m), 8.08-8.25 (5H, m), 8.22-8.24 (1H, m),
        8.56-8.65 (1H, m).
6-1281  δ 7.41-7.50 (1H, m), 7.86-7.87 (2H, m), 7.95-7.98 (1H, m), 8.03-8.13 (6H, m), 8.65-8.67 (1H, m).
6-1282  δ 7.06 (2H, t, J = 8.3 Hz), 7.38-7.42 (1H, m), 7.47-7.52 (1H, m), 7.93-7.97 (1H, m), 8.01 (1H, s),
        8.11-8.13 (3H, m), 8.68-8.72 (1H, m).
6-1296  δ 7.41-7.52 (2H, m), 7.96-8.00 (1H, m), 8.12-8.14 (3H, m), 8.33-8.35 (1H, m), 8.57-8.59 (1H, m),
        8.68-8.76 (2H, m).
6-1303  δ 7.41-7.45 (1H, m), 7.51-7.54 (1H, m), 7.96-7.99 (1H, m), 8.06-8.24 (5H, m), 8.61 (1H, m), 8.94 (1H, m).
6-1338  δ 7.38-7.42 (1H, m), 7.52-7.64 (3H, m), 7.90-7.94 (3H, m), 8.11-8.15 (4H, m), 8.67-8.71 (1H, m).
6-1339  δ 7.35-7.42 (2H, m), 7.60 (1H, d, J = 8.0 Hz), 7.94 (1H, t, J = 8.0 Hz), 8.11 (2H, s), 8.17-8.25 (2H, m), 8.62 (1H,
        s), 8.74 (1H, t, J = 7.4 Hz), 8.92 (1H, d, J = 16.4 Hz).
6-1340  δ 7.28-7.35 (2H, m), 7.40 (1H, t, J = 8.0 Hz), 7.51-7.56 (1H, m), 7.64-7.70 (2H, m), 7.94 (1H, t, J = 8.0 Hz),
        8.10 (2H, s), 8.14 (1H, s), 8.65 (1H, t, J = 8.0 Hz).
6-1341  δ 7.20-7.25 (2H, m), 7.40 (1H, t, J = 8.0 Hz), 7.92-7.97 (3H, m), 8.09 (1H, d, J = 8.0 Hz), 8.11 (2H, s), 8.14 (1H,
        s), 8.64 (1H, t, J = 8.0 Hz).
6-1358  δ 7.41-7.45 (1H, m), 7.68-7.72 (1H, m), 7.89-7.98 (2H, m), 8.10-8.23 (6H, m), 8.60-8.64 (1H, m).
6-1359  δ 7.41-7.45 (1H, m), 7.83-7.89 (2H, m), 7.94-7.99 (1H, m), 8.03-8.14 (6H, m), 8.62-8.66 (1H, m).
6-1360  δ 7.05 (1H, t, J = 8.8 Hz), 7.41-7.46 (1H, m), 7.52 (1H, t, J = 7.8 Hz), 7.95 (1H, t, J = 7.8 Hz), 8.03 (1H, s),
        8.10 (2H, s), 8.15 (1H, s), 8.61 (1H, s), 8.70 (1H, t, J = 8.0 Hz).
6-1374  δ 7.41-7.49 (2H, m), 8.00 (1H, t, J = 8.0 Hz), 8.11 (2H, s), 8.16 (1H, s), 8.34 (1H, d, J = 7.2 Hz), 8.58 (1H, d, J = 2.0 Hz),
        8.70 (1H, t, J = 7.8 Hz), 8.78 (1H, s).
6-1381  δ 7.43 (1H, t, J = 8.0 Hz), 7.53 (1H, d, J = 8.0 Hz), 7.97 (1H, t, J = 7.8 Hz), 8.11-8.12 (3H, m), 8.14 (1H, s),
        8.22 (1H, d, J = 8.0 Hz), 8.57 (1H, t, J = 8.0 Hz), 8.94 (1H, s).
6-1574  δ 7.37-7.41 (1H, m), 7.53-7.64 (3H, m), 7.86-7.94 (4H, m), 8.13-8.22 (3H, m), 8.67-8.72 (1H, m).
6-1575  δ 7.22-7.27 (1H, m), 7.35-7.41 (2H, m), 7.57-7.60 (1H, m), 7.88-7.93 (2H, m), 8.16 (1H, s), 8.20-8.25 (2H,
        m), 8.74-8.75 (1H, m), 8.77-9.00 (1H, m).
6-1576  δ 7.27-7.37 (2H, m), 7.48-7.53 (1H, m), 7.72-7.80 (3H, m), 7.92 (1H, s), 8.15 (1H, s), 8.27-8.31 (1H, m),
        9.16 (1H, s), 9.35 (1H, d, J = 7.3 Hz).
6-1577  δ 7.20-7.23 (3H, m), 7.24-7.26 (1H, m), 7.39-7.40 (3H, m), 7.86-7.97 (1H, m), 8.06 (1H, d, J = 2.4 Hz),
        8.16-8.20 (1H, m), 8.62-8.67 (1H, m).
6-1594  δ 7.41-7.42 (1H, m), 7.70-7.71 (1H, m), 7.93-8.89 (3H, m), 8.12-8.24 (5H, m), 8.60-8.61 (1H, m).
6-1595  δ 7.41 (1H, t, J = 7.8 Hz), 7.84-7.87 (2H, m), 7.90-7.94 (2H, m), 8.03-8.05 (2H, m), 8.12-8.18 (3H, m),
        8.62-8.66 (1H, m).
6-1596  δ 7.00-7.09 (2H, m), 7.40-7.41 (1H, m), 7.46-7.53 (1H, m), 7.89-7.92 (2H, m), 8.00 (1H, s),
        8.16-8.19 (2H, m), 8.71-8.72 (1H, m).
6-1610  δ 7.42-7.49 (2H, m), 7.93-7.94 (2H, m), 8.15-8.21 (2H, m), 8.31-8.34 (1H, m), 8.57-8.59 (1H, m),
        8.63-8.69 (2H, m).
6-1617  δ 7.31-7.38 (1H, m), 7.49 (1H, d, J = 8.3 Hz), 7.82-7.86 (1H, m), 7.92 (1H, s), 8.15 (1H, s), 8.19-8.23 (1H,
        m), 8.30 (1H, dd, J = 2.4, 8.3 Hz), 9.04-9.09 (2H, m), 9.53 (1H, s).
6-1652  δ 7.40 (1H, t, J = 7.8 Hz), 7.53-7.64 (3H, m), 7.86-7.94 (4H, m), 8.13-8.20 (3H, m), 8.71-8.72 (1H, m).
6-1653  δ 7.22-7.25 (1H, m), 7.35-7.41 (2H, m), 7.57-7.60 (1H, m), 7.88-7.92 (2H, m), 8.15 (1H, s), 8.20-8.29 (2H,
        m), 8.71-8.75 (1H, m), 8.89-8.93 (1H, m).
6-1654  δ 7.32-7.34 (1H, m), 7.38-7.42 (1H, m), 7.50-7.56 (1H, m), 7.63-7.70 (2H, m), 7.88-7.91 (2H, m),
        8.09-8.20 (3H, m), 8.63-8.68 (1H, m).
6-1655  δ 7.21-7.30 (2H, m), 7.37-7.41 (1H, m), 7.86-7.97 (4H, m), 8.06-8.21 (3H, m), 8.63-8.67 (1H, m).
6-1672  δ 7.37-7.41 (1H, m), 7.67-7.71 (1H, m), 7.88-7.91 (3H, m), 8.15-8.18 (2H, m), 8.24-8.28 (3H, m),
        8.52-8.56 (1H, m).
6-1673  δ 7.39-7.44 (1H, m), 7.85-7.93 (4H, m), 8.03-8.05 (2H, m), 8.13-8.18 (3H, m), 8.61-8.65 (1H, m).
6-1674  δ 7.04-7.09 (2H, m), 7.38-7.42 (1H, m), 7.47-7.52 (1H, m), 7.89-7.93 (2H, m), 8.00 (1H, s), 8.14-8.20 (2H,
        m), 8.69-8.73 (1H, m).
6-1688  δ 7.42 (1H, t, J = 7.8 Hz), 7.47 (1H, dd, J = 4.9, 7.8 Hz), 7.92-7.96 (2H, m), 8.14 (1H, s), 8.19 (1H, d, J = 12.7 Hz),
        8.33 (1H, dd, J = 2.0, 7.8 Hz), 8.58 (1H, dd, J = 2.0, 4.9 Hz), 8.70-8.71 (1H, m), 8.74 (1H, s).
6-1695  δ 7.39-7.43 (1H, m), 7.52-7.54 (1H, m), 7.92-7.95 (2H, m), 8.08-8.09 (1H, m), 8.15 (1H, s), 8.17-8.23 (2H,
        m), 8.57-8.93 (1H, m), 8.94 (1H, s).
6-1730  δ 7.40 (1H, t, J = 7.8 Hz), 7.53-7.64 (3H, m), 7.87-7.95 (4H, m), 8.14 (1H, s), 8.22 (1H, d, J = 12.7 Hz),
        8.37 (1H, s), 8.71-8.72 (1H, m).
6-1731  δ 7.22-7.25 (1H, m), 7.35-7.37 (2H, m), 7.58-7.60 (1H, m), 7.90 (1H, t, J = 8.6 Hz), 7.96 (1H, s), 8.22 (1H, t, J = 8.8 Hz),
        8.29-8.32 (1H, d, J = 12.4 Hz), 8.37 (1H, s), 8.73 (1H, m), 8.94 (1H, s).
6-1732  δ 7.32-7.33 (1H, m), 7.37 (1H, t, J = 8.0 Hz), 7.52-7.54 (1H, m), 7.64-7.70 (2H, m), 7.90 (1H, t, J = 6.4 Hz),
        7.96 (1H, s), 8.10 (1H, s), 8.23 (1H, d, J = 12.0 Hz), 8.37 (1H, s), 8.65 (1H, t, J = 8.0 Hz).
6-1733  δ 7.19-7.25 (2H, m), 7.35 (1H, t, J = 7.8 Hz), 7.87-7.97 (4H, m), 8.08 (1H, s), 8.25 (1H, d, J = 12.0 Hz), 8.37 (1H,
        s), 8.65 (1H, t, J = 8.0 Hz).
6-1734  δ 7.43-7.52 (5H, m), 7.87-7.95 (3H, m), 8.22 (1H, d, J = 10.0 Hz), 8.35 (1H, d, J = 8.2 Hz), 8.74 (1H, t, J = 8.4 Hz).
6-1750  δ 7.40 (1H, t, J = 8.2 Hz), 7.68 (1H, t, J = 8.0 Hz), 7.88-7.95 (2H, m), 8.12 (1H, s), 8.16 (1H, d, J = 8.0 Hz),
        8.23-8.25 (2H, m), 8.30-8.33 (1H, m), 8.36 (1H, s), 8.53 (1H, t, J = 7.4 Hz).
6-1751  δ 7.44 (1H, t, J = 8.0 Hz), 7.86 (2H, d, J = 8.0 Hz), 7.91-7.96 (2H, m), 8.03 (2H, d, J = 7.6 Hz), 8.13-8.22 (2H, m),
        8.37 (1H, s), 8.64 (1H, t, J = 8.6 Hz).
6-1752  δ 7.04-7.11 (2H, m), 7.38-7.53 (2H, m), 7.90-7.95 (2H, m), 8.01 (1H, s), 8.22 (1H, d, J = 12.8 Hz), 8.37 (1H, s),
        8.69-8.73 (1H, m).
6-1754  δ 7.39-7.44 (2H, m), 7.54 (1H, s), 7.85 (1H, d, J = 8.0 Hz), 7.90-7.95 (2H, m), 8.22 (1H, d, J = 12.0 Hz), 8.68 (1H,
        s), 8.70 (1H, s), 8.69 (1H, t, J = 7.8 Hz).
6-1755  δ 7.16-7.19 (1H, m), 7.40 (1H, t, J = 8.0 Hz), 7.92-7.95 (2H, m), 8.07 (2H, t, J = 4.8 Hz), 8.24 (1H, d, J = 12.8 Hz),
        8.37 (1H, s), 8.42 (1H, s), 8.70 (1H, t, J = 8.0 Hz).
6-1766  δ 7.41-7.49 (2H, m), 7.93-7.97 (2H, m), 8.22 (1H, d, J = 13.2 Hz), 8.33 (1H, dd, J = 2.0, 7.3 Hz), 8.37 (1H, s),
        8.58 (1H, dd, J = 2.0, 4.9 Hz), 8.70-8.73 (2H, m).
6-1773  δ 7.40 (1H, t, J = 8.2 Hz), 7.52 (1H, d, J = 8.0 Hz), 7.91-7.96 (2H, m), 8.12-8.28 (3H, m), 8.37 (1H, s), 8.57 (1H,
        s), 8.94 (1H, s).
6-1808  δ 7.38-7.42 (1H, m), 7.53-7.64 (3H, m), 7.87-7.94 (4H, m), 8.14 (1H, s), 8.23-8.26 (1H, m), 8.36 (1H, s),
        8.68-8.71 (1H, m).
6-1809  δ 7.22-7.25 (2H, m), 7.38 (1H, t, J = 8.0 Hz), 7.58-7.61 (1H, m), 7.89-7.94 (2H, m), 8.23 (1H, t, J = 6.3 Hz),
        8.29 (1H, d, J = 13.2 Hz), 8.36 (1H, s), 8.74 (1H, t, J = 6.3 Hz), 8.93-8.94 (1H, m).
6-1810  δ 7.30-7.33 (2H, m), 7.40 (1H, t, J = 7.8 Hz), 7.51-7.56 (1H, m), 7.64-7.70 (2H, m), 7.88-7.94 (1H, m), 8.10 (1H,
        s), 8.23 (1H, d, J = 12.2 Hz), 8.36 (1H, s), 8.67 (1H, t, J = 7.8 Hz).
6-1811  δ 7.39 (1H, t, J = 8.3 Hz), 7.86-7.97 (3H, m), 8.08 (2H, s), 8.25 (1H, d, J = 12.2 Hz), 8.36 (2H, s), 8.65 (2H, t, J = 6.3 Hz).
6-1828  δ 7.30-7.33 (2H, m), 7.41 (1H, t, J = 7.6 Hz), 7.68-7.73 (1H, m), 7.89-7.94 (2H, m), 8.16 (1H, d, J = 7.6 Hz),
        8.23-8.27 (1H, m), 8.41 (1H, s), 8.63-8.64 (2H, m).
6-1829  δ 7.29-7.31 (1H, m), 7.42 (1H, t, J = 8.0 Hz), 7.90-7.94 (2H, m), 8.04 (2H, d, J = 4.4 Hz), 8.15 (1H, s), 8.23 (1H, d,
        J = 12.0 Hz), 8.36 (1H, s), 8.60-8.66 (2H, m).
6-1830  δ 7.06 (1H, t, J = 8.3 Hz), 7.41 (1H, t, J = 7.8 Hz), 7.67-7.69 (1H, m), 7.90-7.93 (2H, m), 8.03 (1H, s), 8.25 (1H, d,
        J = 12.7 Hz), 8.35 (1H, s), 8.61 (1H, s), 8.70 (1H, t, J = 7.8 Hz).
6-1851  δ 7.42 (1H, t, J = 8.0 Hz), 7.53 (1H, d, J = 7.9 Hz), 7.92-7.94 (2H, m), 8.09 (1H, s), 8.21-8.24 (2H, m), 8.36 (1H,
        s), 8.59 (1H, t, J = 8.0 Hz), 8.94 (1H, s).
6-2110  δ 7.36-7.40 (1H, m), 7.53-7.64 (3H, m), 7.84-7.97 (1H, m), 7.92-7.94 (2H, m), 8.04-8.07 (1H, m),
        8.08-8.13 (1H, m), 8.20 (2H, s), 8.68-8.72 (1H, m).
6-3348  δ 7.29-7.34 (1H, m), 7.53-7.65 (3H, m), 7.80-7.84 (1H, m), 7.90-7.92 (3H, m), 8.14 (1H, broad-s), 8.20 (1H, d,
        J = 2.9 Hz), 8.25 (1H, broad-s), 9.10 (1H, dd, J = 1.9, 7.3 Hz).
6-3384  δ 7.32-7.36 (1H, m), 7.45-7.48 (1H, m), 7.83-7.87 (1H, m), 7.93 (1H, broad-s), 8.10 (1H, broad-s), 8.15 (1H,
        broad-s), 8.30 (1H, dd, J = 1.5, 7.3 Hz), 8.57-8.79 (1H, m), 8.78 (1H, broad-s), 9.09 (1H, dd, J = 2.4, 7.3 Hz).
6-5902  (DMSO-d6) δ 7.39 (1H, t, J = 7.8 Hz), 7.52-7.64 (4H, m), 7.81 (1H, t, J = 6.8 Hz), 7.95 (1H, s), 7.98-8.01 (3H,
        m), 10.29 (1H, s), 10.68 (1H, s).
6-5903  δ 7.50-7.67 (5H, m), 7.79 (1H, d, J = 8.0 Hz), 7.92 (1H, d, J = 8.0 Hz), 8.01 (2H, d, J = 8.0 Hz), 8.10 (2H, s),
        8.31 (1H, s).
6-5904  δ 7.19-7.23 (1H, m), 7.28-7.31 (1H, m), 7.58 (1H, t, J = 8.2 Hz), 7.78 (1H, d, J = 8.0 Hz), 7.91-7.94 (3H, m),
        8.01 (2H, d, J = 8.0 Hz), 8.30 (2H, s), 8.61 (1H, s).
6-5905  δ 7.26 (1H, s), 7.43-7.46 (1H, m), 7.56-7.60 (1H, m), 7.80-7.94 (5H, m), 8.22-8.56 (4H, m).
6-5906  δ 7.18-7.12 (2H, m), 7.53-7.57 (1H, m), 7.76 (1H, d, J = 7.6 Hz), 7.86-8.28 (7H, m), 8.28 (1H, s).
6-5907  δ 7.39 (1H, t, J = 7.8 Hz), 7.52-7.64 (4H, m), 7.85-7.94 (4H, m), 8.06 (1H, d, J = 12.2 Hz), 8.14 (1H, broad-s),
        8.67-8.71 (1H, m).
6-5908  δ 7.39-7.49 (2H, m), 7.59 (1H, s), 7.88-7.94 (2H, m), 8.07 (1H, d, J = 12.2 Hz), 8.31-8.33 (1H, m),
        8.57-8.58 (1H, m), 8.60-8.70 (1H, m), 8.74 (1H, broad-s).
6-5909  δ 7.42 (1H, t, J = 7.8 Hz), 7.59 (1H, s), 7.85-7.92 (4H, m), 7.99 (1H, broad-s), 8.02-8.05 (2H, m), 8.10 (1H,
        broad-s), 8.61-8.67 (1H, m).
6-5910  δ 7.39 (1H, t, J = 8.3 Hz), 7.53-7.64 (3H, m), 7.88-7.94 (4H, m), 8.13 (1H, broad-s), 8.19 (1H, broad-s),
        8.24 (1H, d, J = 13.2 Hz), 8.70-8.72 (1H, m).
6-5911  δ 7.41 (1H, t, J = 8.3 Hz), 7.84-7.87 (3H, m), 7.91-7.95 (1H, m), 8.03-8.05 (2H, m), 8.10 (1H, broad-s),
        8.17-8.20 (2H, m), 8.63-8.67 (1H, m).
6-5912  δ 3.10 (3H, s), 7.59 (1H, t, J = 7.8 Hz), 7.76 (1H, d, J = 7.8 hz), 7.77-8.00 (5H, m), 8.03 (1H, s), 8.19 (1H, s),
        8.24 (1H, s), 8.36 (1H, s).
6-5913  δ 7.51-7.62 (4H, m), 7.72 (1H, dd, J = 1.5, 7.8 Hz), 7.89-8.00 (6H, m), 8.14 (1H, s), 8.27 (1H, t, J = 2.0 Hz).
6-5914  δ 7.44 (1H, dd, J = 4.9, 7.8 Hz), 7.56-7.60 (1H, m), 7.76 (1H, d, J = 7.8 Hz), 7.92 (3H, broad-s), 8.14 (1H, s),
        8.22-8.27 (1H, m), 8.27 (1H, s), 8.41 (1H, s), 8.55 (1H, dd, J = 2.0, 4.4 Hz).
7-38    δ 3.57 (3H, s), 7.21-7.24 (1H, m), 7.32-7.34 (4H, m), 7.40-7.44 (2H, m), 7.59 (1H, s), 7.71 (1H, d, J = 8.0 Hz),
        7.84 (3H, s).
7-39    δ 3.54 (3H, s), 7.06-7.19 (1H, m), 7.28-7.34 (2H, m), 7.43-7.48 (2H, m), 7.57 (1H, s), 7.69 (1H, s), 7.75 (1H, d, J = 8.0 Hz),
        7.90 (1H, d, J = 8.0 Hz), 8.06 (2H, s).
7-45    δ 3.57 (3H, s), 7.29-7.30 (2H, m), 7.48 (1H, t, J = 8.0 Hz), 7.59 (1H, s), 7.68-7.71 (3H, m), 7.77 (1H, d, J = 7.8 Hz),
        7.85 (2H, s), 8.24 (1H, s).
7-46    δ 3.57 (3H, s), 7.41-7.45 (3H, m), 7.52 (2H, s), 7.55 (1H, d, J = 8.0 Hz), 7.69 (1H, s), 7.74 (1H, d, J = 7.8 Hz),
        7.86 (2H, s), 8.62 (1H, s).
7-47    δ 3.56 (3H, s), 6.97-7.05 (3H, m), 7.17-7.19 (1H, m), 7.43-7.50 (3H, m), 7.73 (1H, s), 7.85 (2H, s).
7-57    δ 3.57 (3H, s), 7.15 (1H, t, J = 6.0 Hz), 7.41 (2H, s), 7.50 (1H, s), 7.52 (1H, s), 7.60 (1H, d, J = 6.4 Hz), 7.73 (1H,
        s), 7.85 (2H, s), 8.27 (1H, s).
7-60    3.57 (3H, s), 7.30 (1H, d, J = 8.0 Hz), 7.47 (1H, t, J = 8.0 Hz), 7.61 (1H, s), 7.76 (2H, s), 7.78-7.81 (1H, m),
        7.85 (2H, s), 8.11 (1H, s), 8.24 (1H, s).
7-71    δ 3.56 (3H, s), 7.20-7.25 (1H, m), 7.33-7.38 (3H, m), 7.43-7.47 (3H, m), 7.56 (1H, s), 7.74 (1H, d, J = 6.8 Hz),
        8.06-8.10 (3H, m).
7-72    δ 3.55 (3H, s), 7.06-7.10 (1H, m), 7.30-7.36 (2H, m), 7.43-7.48 (2H, m), 7.57 (1H, s), 7.68 (1H, s), 7.78 (1H, d, J = 8.0 Hz),
        7.90 (1H, d, J = 8.0 Hz), 8.07 (2H, s).
7-78    δ 3.57 (3H, s), 7.29-7.64 (2H, m), 7.70 (1H, s), 7.79 (1H, d, J = 8.0 Hz), 7.86 (1H, d, J = 8.0 Hz), 7.95 (1H, t, J = 8.0 Hz),
        8.08 (2H, s), 8.33 (1H, d, J = 8.0 Hz), 8.40 (1H, s), 8.71 (1H, s).
7-79    δ 3.58 (3H, s), 7.42-7.53 (3H, m), 7.60-7.66 (1H, m), 7.77 (1H, d, J = 8.0 Hz), 7.89 (1H, t, J = 8.0 Hz), 8.08 (2H,
        s), 8.21 (1H, d, J = 8.0 Hz), 8.70 (2H, s).
7-80    δ 3.56 (3H, s), 7.02 (1H, t, J = 8.0 Hz), 7.42-7.44 (1H, m), 7.55 (1H, t, J = 8.0 Hz), 7.75 (1H, d, J = 8.0 Hz),
        7.90-7.95 (3H, m), 8.01 (1H, s), 8.14 (1H, s), 8.26 (1H, s).
7-90    δ 3.59 (3H, s), 7.59 (1H, s), 7.60 (1H, d, J = 6.0 Hz), 7.80-7.83 (1H, m), 8.08 (2H, s), 8.26-8.30 (2H, m), 8.53 (1H,
        d, J = 4.0 Hz), 8.69 (2H, s).
7-93    δ 3.58 (3H, s), 7.34-7.52 (3H, m), 7.63 (1H, d, J = 16.0 Hz), 7.69 (1H, d, J = 8.0 Hz), 7.80 (1H, d, J = 8.0 Hz),
        7.85 (1H, t, J = 8.0 Hz), 8.25 (1H, s), 8.29 (1H, d, J = 8.0 Hz), 8.69 (1H, s).
7-132   δ 3.57 (3H, s), 7.26-7.28 (1H, m), 7.41-7.46 (3H, m), 7.52-7.54 (3H, m), 7.63 (1H, s), 7.68 (1H, d, J = 7.8 Hz),
        7.87 (1H, s), 7.98 (1H, s).
7-147   δ 3.58 (3H, s), 7.14 (1H, dd, J = 4.9, 7.8 Hz), 7.41-7.42 (2H, m), 7.52 (1H, s), 7.59 (1H, dd, J = 1.5, 7.8 Hz),
        7.67 (2H, broad-s), 7.87 (1H, s), 7.97 (1H, s), 8.26 (1H, dd, J = 1.5, 4.9 Hz).
7-268   δ 3.49 (3H, s), 7.12-7.16 (2H, m), 7.21-7.28 (4H, m), 7.35 (1H, t, J = 7.8 Hz), 7.64 (1H, s), 7.70 (1H, dd, J = 1.5,
        8.8 Hz), 7.86 (1H, s), 8.07 (1H, d, J = 1.5 Hz), 8.29 (1H, s).
7-269   δ 3.54 (3H, s), 6.80-6.81 (1H, m), 7.70-7.08 (1H, m), 7.25-7.26 (1H, m), 7.39-7.41 (4H, m), 7.52-7.53 (1H,
        m), 7.70-7.71 (1H, m), 7.90 (1H, s), 8.12 (1H, s).
7-270   δ 3.55 (3H, s), 6.97-6.99 (1H, m), 7.04-7.06 (2H, m), 7.15-7.21 (1H, m), 7.32-7.34 (1H, m), 7.44 (1H, t, J = 7.8 Hz),
        7.58-7.59 (2H, m), 7.70 (1H, d, J = 7.8 Hz), 7.90 (1H, s), 8.12 (1H, s).
7-271   δ 3.55 (3H, s), 6.88-6.92 (2H, m), 7.30-7.34 (3H, m), 7.43 (1H, t, J = 7.8 Hz), 7.57-7.58 (2H, m),
        7.67-7.69 (1H, m), 7.90-7.91 (1H, m), 8.13-8.14 (1H, m).
7-285   δ 3.59 (3H, s), 7.34-7.52 (3H, m), 7.65-7.73 (4H, m), 7.90 (1H, s), 8.13-8.16 (3H, m).
7-286   δ 3.59 (3H, s), 7.29-7.30 (1H, m), 7.42-7.52 (4H, m), 7.63 (1H, s), 7.69 (1H, d, J = 7.8 Hz), 7.91 (1H, s),
        8.08-8.13 (3H, m).
7-288   δ 3.57 (3H, s), 7.15-7.37 (2H, m), 7.47-7.48 (1H, m), 7.52-7.62 (5H, m), 7.72 (1H, d, J = 7.8 Hz), 7.91 (1H,
        s), 8.14 (1H, s).
7-289   δ 3.57 (3H, s), 7.26-7.29 (1H, m), 7.40-7.46 (3H, m), 7.52 (2H, d, J = 8.3 Hz), 7.58-7.61 (2H, m), 7.70 (1H,
        d, J = 7.8 Hz), 7.92 (1H, s), 8.14 (1H, s).
7-290   δ 3.55 (3H, s), 6.70-6.74 (2H, m), 7.14-7.19 (1H, m), 7.43-7.44 (2H, m), 7.52 (1H, s), 7.67 (1H, s),
        7.74-7.77 (1H, m), 7.91 (1H, s), 8.13 (1H, s).
7-299   δ 3.58 (3H, s), 7.33 (1H, d, J = 6.8 Hz), 7.52 (1H, t, J = 7.8 Hz), 7.64-7.65 (2H, m), 7.75-7.79 (3H, m),
        7.83 (1H, s), 7.92 (1H, s), 8.14 (1H, s).
7-300   δ 3.56 (3H, broad-s), 7.14 (1H, broad-d, J = 8.3 Hz), 7.33-7.53 (4H, m), 7.59-7.60 (2H, m), 7.71-7.72 (1H,
        m), 7.92 (1H, s), 8.14 (1H, s).
7-301   δ 3.57 (3H, s), 7.33-7.59 (4H, m), 7.60 (1H, s), 7.64 (1H, s), 7.68-7.70 (2H, m), 7.92 (1H, s), 8.15 (1H, s).
7-303   δ 3.56 (3H, s), 7.17-7.12 (1H, m), 7.39-7.45 (2H, m), 7.55 (2H, s), 7.69 (1H, d, J = 7.8 Hz), 7.90 (2H, s),
        8.13-8.14 (2H, m).
7-304   δ 3.54 (3H, s), 7.10 (1H, dd, J = 4.9, 7.8 Hz), 7.35-7.40 (2H, m), 7.56 (1H, dd, J = 1.5, 7.8 Hz), 7.70 (2H, s),
        7.88-7.90 (2H, m), 8.12 (1H, s), 8.22 (1H, dd, J = 1.5, 4.9 Hz).
7-305   δ 3.57 (3H, s), 7.13 (1H, dd, J = 4.9, 7.8 Hz), 7.41-7.42 (2H, m), 7.57-7.62 (2H, m), 7.67-7.69 (2H, m),
        7.91 (1H, s), 8.13 (1H, s), 8.24-8.26 (1H, m).
7-311   δ 3.57 (3H, s), 7.23-7.31 (2H, m), 7.47-7.48 (1H, m), 7.66-7.73 (4H, m), 7.92 (1H, s), 8.14 (1H, s),
        8.23 (1H, d, J = 1.9 Hz).
7-316   δ 3.59 (3H, s), 7.27-7.30 (1H, m), 7.48-7.49 (1H, m), 7.60-7.67 (3H, m), 7.73 (1H, d, J = 7.8 Hz), 7.85 (1H,
        dd, J = 1.9, 7.8 Hz), 7.92 (1H, s), 8.15 (1H, d, J = 1.5 Hz), 8.52 (1H, s).
7-346   δ 3.54 (3H, s), 7.18-7.34 (4H, m), 7.40 (1H, t, J = 7.8 Hz), 7.57 (1H, s), 7.67-7.69 (1H, m), 7.88 (1H, s), 8.10 (1H,
        s).
7-347   δ 3.53 (3H, s), 6.82 (1H, s), 7.07 (1H, s), 7.23-7.70 (7H, m), 7.89 (1H, s), 8.11 (1H, s).
7-348   δ 3.53 (3H, s), 6.96-6.99 (1H, m), 7.00-7.06 (2H, m), 7.15-7.19 (1H, m), 7.32-7.34 (1H, m), 7.42-7.46 (1H,
        m), 7.60 (1H, s), 7.68-7.71 (2H, m), 7.89 (1H, s), 8.11 (1H, s).
7-349   δ 3.54 (3H, s), 6.88-6.92 (2H, m), 7.29-7.34 (3H, m), 7.41-7.44 (2H, m), 7.59 (1H, s), 7.68-7.70 (1H, m),
        7.89 (1H, s), 8.11 (1H, s).
7-366   δ 3.64 (3H, s), 7.31-7.36 (2H, m), 7.44-7.48 (2H, m), 7.52-7.58 (1H, m), 7.61 (2H, s), 7.71-7.73 (2H, m),
        7.89 (1H, s), 8.12 (1H, s).
7-367   δ 3.56 (3H, s), 7.22-7.31 (3H, m), 7.44-7.48 (1H, m), 7.66-7.77 (4H, m), 7.90 (1H, s), 8.12 (1H, s),
        8.22 (1H, s).
7-368   δ 3.52 (3H, s), 6.67-6.72 (2H, m), 7.00 (1H, s), 7.13-7.17 (1H, m), 7.41-7.42 (2H, m), 7.72-7.89 (3H, m),
        8.11 (1H, s).
7-382   δ 3.58 (3H, s), 7.13-7.16 (1H, m), 7.43-7.61 (4H, m), 7.67 (2H, s), 7.90 (1H, s), 8.13 (1H, s), 8.26-8.27 (1H,
        m).
7-389   δ 3.57 (3H, s), 7.29 (1H, s), 7.40-7.46 (3H, m), 7.52-7.54 (2H, m), 7.59-7.62 (1H, m), 7.69-7.70 (1H, m),
        7.90 (1H, s), 8.13 (1H, s).
7-424   δ 3.56 (3H, s), 7.19-7.37 (6H, m), 7.44-7.45 (1H, m), 7.54 (1H, s), 7.60 (1H, broad-s), 7.68 (1H, d, J = 7.8 Hz),
        7.92 (1H, s), 8.31 (1H, s).
7-425   δ 3.54 (3H, broad-s), 6.82 (1H, broad-s), 7.07 (1H, broad-s), 7.23-7.30 (2H, m), 7.31-7.51 (3H, m),
        7.52-7.56 (1H, m), 7.71 (1H, broad-s), 7.92 (1H, s), 8.33 (1H, s).
7-426   δ 3.56 (3H, s), 6.96-7.00 (1H, m), 7.05-7.07 (2H, m), 7.15-7.21 (1H, m), 7.34-7.36 (1H, m), 7.46-7.47 (1H,
        m), 7.58-7.66 (2H, m), 7.71 (1H, d, J = 7.3 Hz), 7.93 (1H, s), 8.33 (1H, s).
7-427   δ 3.56 (3H, s), 6.88-6.92 (2H, m), 7.31-7.34 (2H, m), 7.45-7.46 (1H, m), 7.56 (1H, s), 7.62 (1H, s),
        7.65 (1H, s), 7.70 (1H, d, J = 7.3 Hz), 7.93 (1H, s), 8.33 (1H, s).
7-428   δ 3.58 (3H, s), 7.00-7.24 (4H, m), 7.42-7.43 (3H, m), 7.62 (1H, s), 7.66 (1H, s), 7.94 (1H, s), 8.34 (1H, s).
7-444   δ 3.57 (3H, s), 7.33-7.37 (2H, m), 7.48-7.49 (1H, m), 7.52-7.61 (4H, m), 7.69-7.74 (2H, m), 7.93 (1H, s),
        8.34 (1H, s).
7-445   δ 3.58 (3H, s), 7.30 (1H, d, J = 9.5 Hz), 7.41-7.48 (3H, m), 7.51-7.53 (3H, m), 7.59 (1H, s), 7.70 (1H, d, J = 7.9 Hz),
        7.94 (1H, s), 8.34 (1H, s).
7-446   δ 3.56 (3H, s), 6.69-6.73 (2H, m), 7.14-7.18 (1H, m), 7.44-7.45 (2H, m), 7.61 (1H, s), 7.69 (1H, s),
        7.75-7.77 (1H, m), 7.93 (1H, s), 8.34 (1H, s).
7-449   δ 3.51 (3H, s), 6.82-6.86 (1H, m), 6.94-6.98 (1H, m), 7.14-7.24 (1H, m), 7.28-7.29 (2H, m), 7.41 (1H, s),
        7.64 (1H, s), 7.69 (1H, d, J = 5.9 Hz), 7.94 (1H, s), 8.34 (1H, s).
7-460   δ 3.59 (3H, s), 7.13 (1H, dd, J = 4.8, 7.1 Hz), 7.43-7.44 (2H, m), 7.52 (1H, s), 7.58-7.60 (1H, m), 7.67 (2H,
        broad-s), 7.94 (1H, s), 8.26 (1H, dd, J = 1.6, 4.8 Hz), 8.34 (1H, s).
7-467   δ 3.58 (3H, s), 7.23 (1H, d, J = 8.3 Hz), 7.33 (1H, d, J = 7.8 Hz), 7.49-7.50 (1H, m), 7.62 (1H, s),
        7.67-7.68 (2H, m), 7.73 (1H, d, J = 7.8 Hz), 7.93 (1H, s), 8.23 (1H, d, J = 2.0 Hz), 8.34 (1H, s).
7-502   δ 3.57 (3H, s), 7.20-7.26 (3H, m), 7.27-7.37 (3H, m), 7.45 (1H, t, J = 7.6 Hz), 7.56 (1H, s), 7.68 (1H, s), 7.71 (1H,
        d, J = 8.0 Hz), 7.91 (1H, s), 8.31 (1H, s).
7-504   3.56 (3H, s), 6.96-7.01 (1H, m), 7.06 (2H, d, J = 7.2 Hz), 7.18 (1H, t, J = 6.8 Hz), 7.35 (1H, d, J = 8.0 Hz), 7.45 (1H,
        t, J = 8.0 Hz), 7.56 (2H, s), 7.71 (1H, d, J = 8.0 Hz), 7.91 (1H, s), 8.32 (1H, s).
7-505   δ 3.57 (3H, s), 6.90 (2H, t, J = 8.8 Hz), 7.31-7.35 (3H, m), 7.45 (1H, t, J = 8.0 Hz), 7.54 (2H, d, J = 13.6 Hz),
        7.69 (1H, d, J = 8.0 Hz), 7.91 (1H, s), 8.32 (1H, s).
7-522   δ 3.57 (3H, s), 7.32-7.37 (2H, m), 7.46 (1H, t, J = 8.0 Hz), 7.55 (1H, t, J = 7.6 Hz), 7.59 (2H, d, J = 8.0 Hz),
        7.75 (1H, d, J = 8.0 Hz), 7.88 (1H, s), 7.92 (2H, s), 8.33 (1H, s).
7-523   δ 3.56 (3H, s), 7.41-7.47 (4H, m), 7.53 (2H, d, J = 8.2 Hz), 7.61 (1H, s), 7.71-7.72 (2H, m), 7.92 (1H, s), 8.33 (1H,
        s).
7-538   δ 3.58 (3H, s), 7.14 (1H, t, J = 6.0 Hz), 7.40-7.43 (2H, m), 7.56-7.58 (2H, m), 7.68-7.69 (2H, m), 7.92 (1H, s),
        8.26 (1H, s), 8.33 (1H, s).
7-804   δ 3.55 (3H, s), 7.19-7.52 (9H, m), 7.62 (1H, d, J = 7.8 Hz), 8.16 (2H, s).
7-824   δ 3.57 (3H, s), 7.33-7.75 (7H, m), 7.98-7.99 (1H, m), 8.12 (2H, s), 8.18-8.43 (1H, m).
7-825   δ 3.57 (3H, s), 7.22-7.66 (7H, m), 7.85-7.88 (1H, m), 7.97-7.99 (2H, m), 8.17-8.27 (1H, m).
7-840   δ 3.57 (3H, s), 7.13-7.26 (1H, m), 7.40-7.44 (2H, m), 7.58-7.71 (3H, m), 8.18-8.23 (4H, m).
7-948   δ 3.49 (3H, s), 7.23-7.52 (8H, m), 7.66 (2H, s), 8.00 (1H, t, J = 6.8 Hz).
7-969   δ 3.51 (3H, s), 7.45-7.46 (3H, m), 7.53-7.55 (3H, m), 7.67 (2H, s), 7.92-7.93 (1H, m), 8.05-8.06 (1H, m).
7-984   δ 3.53 (3H, s), 7.13-7.16 (1H, m), 7.20-7.24 (1H, m), 7.52-7.53 (1H, m), 7.65-7.68 (3H, m), 7.99-8.03 (2H,
        m), 8.28-8.30 (1H, m).
7-1104  δ 3.51 (3H, s), 7.22-7.44 (7H, m), 7.86 (2H, s), 8.00-8.03 (2H, m).
7-1105  δ 3.52 (3H, s), 6.82 (1H, t, J = 8.8 Hz), 7.06-7.08 (1H, m), 7.18-7.24 (2H, m), 7.40-7.44 (2H, m), 7.87 (3H, s),
        8.01-8.05 (1H, m).
7-1106  δ 3.50 (3H, s), 7.00-7.23 (4H, m), 7.29-7.31 (1H, m), 7.45 (1H, s), 7.87 (3H, s), 8.03-8.07 (1H, m).
7-1107  δ 3.49 (3H, s), 6.91-6.93 (2H, m), 7.28-7.44 (4H, m), 7.86 (2H, s), 8.00-8.10 (2H, m).
7-1124  δ 3.52 (3H, s), 7.30-7.34 (2H, m), 7.46-7.59 (3H, m), 7.71 (1H, broad-s), 7.87 (2H, s), 7.97-8.09 (2H, m).
7-1125  δ 3.52 (3H, s), 7.29-7.32 (1H, m), 7.45-7.52 (5H, m), 7.84 (2H, s), 7.95-8.06 (2H, m).
7-1126  δ 3.49 (3H, s), 6.72-6.76 (2H, m), 7.16-7.23 (2H, m), 7.43-7.50 (1H, m), 7.88 (2H, s), 8.02-8.06 (1H, m),
        8.13-8.17 (1H, m).
7-1140  δ 3.54 (3H, s), 7.13-7.16 (1H, m), 7.21-7.26 (1H, m), 7.43-7.46 (1H, m), 7.52 (1H, broad-s), 7.65-7.69 (1H, m),
        7.88 (2H, s), 8.00-8.04 (1H, m), 8.28-8.30 (1H, m).
7-1147  δ 3.52 (3H, s), 7.22-7.26 (1H, m), 7.34 (1H, t, J = 7.8 Hz), 7.46-7.52 (1H, m), 7.62-7.68 (1H, m), 7.87 (2H,
        s), 7.91-7.95 (1H, m), 8.07-8.11 (1H, m), 8.34 (1H, broad-s).
7-1182  δ 3.51 (3H, s), 7.22-7.44 (7H, m), 7.85 (2H, s), 8.00-8.03 (2H, m).
7-1183  δ 3.51 (3H, s), 6.79-6.83 (1H, m), 7.05 (1H, t, J = 7.8 Hz), 7.17-7.23 (2H, m), 7.40-7.43 (2H, m), 7.85 (2H, s),
        7.98-8.00 (2H, m).
7-1184  δ 3.52 (3H, s), 6.99-7.22 (4H, m), 7.28-7.30 (1H, m), 7.44-7.45 (1H, m), 7.88 (2H, s), 8.02-8.06 (2H, m).
7-1185  δ 3.49 (3H, s), 6.91-7.00 (2H, m), 7.26-7.44 (4H, m), 7.85 (2H, s), 8.01-8.10 (2H, m).
7-1202  δ 3.52 (3H, s), 7.26-7.32 (1H, m), 7.45-7.52 (5H, m), 7.86 (2H, s), 7.84-7.95 (1H, m), 8.06-8.08 (1H, m).
7-1203  δ 3.52 (3H, s), 7.26-7.32 (1H, m), 7.45-7.52 (5H, m), 7.86 (2H, s), 7.84-7.95 (1H, m), 8.06-8.08 (1H, m).
7-1204  δ 3.51 (3H, s), 7.02 (1H, t, J = 8.8 Hz), 7.39-7.44 (1H, m), 7.50 (1H, t, J = 7.4 Hz), 7.93 (1H, t, J = 7.8 Hz),
        8.02 (1H, s), 8.10 (2H, s), 8.13 (1H, s), 8.68 (1H, t, J = 8.0 Hz).
7-1218  δ 3.52 (3H, s), 7.39-7.47 (1H, m), 7.96 (1H, t, J = 8.0 Hz), 8.11 (2H, s), 8.16 (1H, s), 8.33 (1H, d, J = 7.2 Hz),
        8.58-8.59 (1H, m), 8.68 (1H, t, J = 7.8 Hz), 8.78 (1H, s).
7-1225  δ 3.52 (3H, s), 7.22-7.24 (1H, m), 7.32-7.36 (1H, m), 7.46-7.50 (1H, m), 7.66-7.68 (1H, m), 7.85 (2H, s),
        7.93-7.96 (1H, m), 8.07-8.11 (1H, m), 8.34 (1H, broad-s).
7-1260  δ 4.09 (3H, s), 7.21-7.49 (7H, m), 7.99-8.08 (4H, m).
7-1261  δ 3.53 (3H, s), 6.79-6.83 (1H, m), 7.03-7.07 (1H, m), 7.19-7.23 (2H, m), 7.42-7.43 (2H, m), 8.01-8.10 (4H,
        m).
7-1262  δ 3.51 (3H, s), 6.99-7.00 (1H, m), 7.08-7.14 (2H, m), 7.29-7.33 (2H, m), 7.46-7.47 (1H, m), 8.05-8.12 (4H,
        m).
7-1263  δ 3.52 (3H, s), 6.88-6.93 (2H, m), 7.29-7.37 (3H, m), 7.46-7.48 (1H, m), 8.04-8.09 (4H, m).
7-1280  δ 3.52 (3H, s), 7.31-7.47 (2H, m), 7.49 (1H, s), 7.57 (2H, m), 7.69 (1H, s), 8.07-8.10 (4H, m).
7-1281  δ 3.53 (3H, s), 7.23-7.52 (6H, m), 7.90-8.09 (4H, m).
7-1282  δ 3.55 (3H, s), 6.72-6.76 (2H, m), 7.17-7.24 (2H, m), 7.48-7.49 (1H, m), 8.04-8.16 (4H, m).
7-1296  δ 3.55 (3H, s), 7.12-7.15 (1H, m), 7.46-7.51 (1H, broad-s), 7.67-7.69 (1H, m), 8.03-8.12 (5H, m),
        8.27-8.29 (1H, m).
7-1303  δ 3.54 (3H, s), 7.20-7.23 (1H, m), 7.35-7.39 (1H, m), 7.52-7.53 (1H, m), 7.65 (1H, s), 7.97 (1H, broad-s),
        8.09-8.14 (3H, m), 8.34-8.35 (1H, m).
7-1338  δ 3.52 (3H, s), 7.10-7.35 (6H, m), 7.45-7.52 (1H, m), 8.02-8.07 (4H, m).
7-1339  δ 3.53 (3H, s), 6.80 (1H, t, J = 8.0 Hz), 7.04 (1H, t, J = 8.0 Hz), 7.29-7.32 (1H, m), 7.43 (1H, t, J = 8.0 Hz),
        7.68-7.71 (1H, m), 8.01-8.04 (2H, m), 8.09 (2H, s), 8.63 (1H, s).
7-1340  δ 3.56 (3H, s), 7.04-7.08 (1H, m), 7.30-7.33 (1H, m), 7.43-7.48 (2H, m), 7.57 (1H, s), 7.64 (1H, s), 7.77 (1H, d, J = 8.0 Hz),
        7.90 (1H, d, J = 8.0 Hz), 8.07 (2H, s).
7-1341  δ 3.52 (3H, s), 6.91-6.92 (2H, m), 7.30 (1H, t, J = 8.0 Hz), 7.36 (2H, s), 7.47 (1H, t, J = 8.0 Hz), 8.00-8.06 (2H, m),
        8.08 (2H, s).
7-1358  δ 3.53 (3H, s), 7.31-7.40 (2H, m), 7.45-7.60 (3H, m), 7.69 (1H, s), 7.99-8.11 (4H, m).
7-1359  δ 3.53 (3H, s), 7.26-7.34 (1H, m), 7.40-7.60 (5H, m), 7.83-7.95 (1H, m), 8.01-8.06 (3H, m).
7-1360  δ 3.55 (3H, s), 6.72-6.76 (2H, m), 7.22-7.24 (1H, m), 7.42-7.44 (1H, m), 7.49 (1H, t, J = 8.0 Hz), 8.05 (1H, d, J = 8.0 Hz),
        8.10 (2H, s), 8.17 (1H, d, J = 8.0 Hz).
7-1374  δ 3.55 (3H, s), 7.12-7.15 (1H, m), 7.52-7.53 (2H, m), 7.68 (1H, d, J = 8.0 Hz), 8.02-8.06 (2H, m), 8.11 (2H, s),
        8.28 (1H, s).
7-1381  δ 3.54 (3H, s), 7.19-7.22 (1H, m), 7.37 (1H, t, J = 8.0 Hz), 7.54 (1H, t, J = 6.0 Hz), 7.66 (1H, d, J = 6.8 Hz),
        7.93-7.96 (1H, m), 8.09-8.13 (3H, m), 8.35 (1H, s).
7-1417  δ 3.49 (3H, s), 7.23-7.26 (3H, m), 7.27-7.33 (3H, m), 7.52-7.53 (1H, m), 7.85 (1H, s), 7.96-8.06 (3H, m).
7-1574  δ 3.50 (3H, s), 6.99-7.33 (6H, m), 7.43-7.45 (1H, m), 7.90 (1H, s), 7.97-8.06 (2H, m), 8.13 (1H, s).
7-1575  δ 3.52 (3H, s), 6.82-6.83 (1H, m), 7.06-7.07 (1H, m), 7.19-7.26 (2H, m), 7.39-7.46 (2H, m), 7.91 (1H, s),
        7.99-8.01 (1H, m), 8.07-8.14 (2H, m).
7-1576  δ 3.50 (3H, s), 7.01-7.17 (4H, m), 7.27-7.31 (1H, m), 7.46-7.52 (1H, m), 7.91 (1H, s), 8.01-8.05 (2H, m),
        8.13 (1H, s).
7-1577  δ 3.50 (3H, s), 6.90-6.94 (2H, m), 7.26-7.35 (3H, m), 7.45-7.46 (1H, m), 7.90 (1H, s), 8.00-8.07 (2H, m),
        8.13 (1H, s).
7-1594  δ 3.52 (3H, s), 7.29-7.36 (2H, m), 7.50 (2H, broad-s), 7.60 (1H, broad-d, J = 6.8 Hz), 7.70 (1H, broad-s),
        7.91 (1H, broad-s), 8.04-8.07 (2H, m), 8.14 (1H, s).
7-1595  δ 3.51 (3H, s), 7.29-7.31 (2H, m), 7.44-7.52 (4H, m), 7.92 (1H, s), 8.03-8.06 (2H, m), 8.14 (1H, broad-s).
7-1596  δ 3.54 (3H, s), 6.75 (2H, broad-s), 7.17-7.26 (2H, m), 7.50-7.51 (1H, m), 7.92 (1H, s), 8.01-8.05 (1H, m),
        8.14-8.20 (2H, m).
7-1605  δ 3.53 (3H, s), 7.41 (1H, t, J = 7.8 Hz), 7.53-7.55 (1H, m), 7.82-7.86 (3H, m), 7.91 (1H, s), 7.99-8.01 (1H,
        m), 8.10-8.14 (2H, m).
7-1606  δ 2.53 (3H, s), 7.15-7.17 (1H, m), 7.24-7.28 (1H, m), 7.39-7.41 (1H, m), 7.41-7.44 (1H, m), 7.53-7.56 (1H,
        m), 7.93 (1H, s), 8.04-8.08 (2H, m), 8.15 (1H, s).
7-1608  δ 3.52 (3H, s), 7.22-7.23 (1H, m), 7.29-7.33 (1H, m), 7.48-7.52 (1H, m), 7.71-7.72 (1H, m), 7.90 (1H, s),
        8.00-8.03 (2H, m), 8.13 (1H, s), 8.54-8.55 (2H, m).
7-1610  δ 3.54 (3H, s), 7.14-7.17 (2H, m), 7.45-7.70 (2H, m), 7.96 (1H, s), 8.00-8.07 (3H, m), 8.28-8.30 (1H, m).
7-1616  δ 3.52 (3H, s), 7.27-7.23 (1H, m), 7.35-7.36 (1H, m), 7.49-7.51 (1H, m), 7.68 (1H, d, J = 6.8 Hz), 7.91 (1H,
        s), 8.09-8.05 (2H, m), 8.13 (1H, s), 8.30 (1H, s).
7-1617  δ 3.52 (3H, s), 7.23-7.27 (1H, m), 7.33-7.37 (1H, m), 7.47-7.51 (1H, m), 7.67-7.68 (1H, m), 7.91 (1H, s),
        8.05-8.09 (1H, m), 8.13 (2H, s), 8.30 (1H, s).
7-1638  δ 3.50 (3H, s), 7.19-7.27 (2H, m), 7.32-7.33 (1H, m), 7.40-7.42 (1H, m), 7.91 (1H, s), 8.00-8.02 (1H, m),
        7.09-8.11 (1H, m), 8.14 (1H, s), 8.18 (1H, s), 8.56 (1H, d, J = 8.8 Hz).
7-1639  δ 3.52 (3H, broad-s), 7.00-7.29 (3H, m), 7.44 (1H, broad-s), 7.52 (1H, s), 7.91-8.14 (3H, m), 8.51 (2H,
        broad-s).
7-1645  δ 3.50 (3H, s), 7.22-7.27 (2H, m), 7.33-7.37 (1H, m), 7.43-7.47 (1H, m), 7.92 (1H, s), 8.02-8.10 (3H, m),
        8.15-8.19 (2H, m).
7-1652  δ 3.50 (3H, s), 7.23-7.26 (2H, m), 7.27-7.32 (4H, m), 7.44-7.45 (1H, m), 7.88 (1H, s), 7.98 (1H, t, J = 6.8 Hz),
        8.04-8.08 (1H, m), 8.11 (1H, s).
7-1672  δ 3.51 (3H, s), 7.29-7.35 (2H, m), 7.49-7.50 (2H, m), 7.60 (1H, d, J = 6.3 Hz), 7.69 (1H, s), 7.89 (1H, s),
        8.03-8.06 (2H, m), 8.12 (1H, s).
7-1673  δ 3.52 (3H, s), 7.29-7.32 (1H, m), 7.44-7.52 (5H, m), 7.89 (1H, s), 8.02-8.06 (2H, m), 8.12 (1H, s).
7-1730  δ 3.51 (3H, s), 7.21-7.23 (2H, m), 7.27-7.33 (4H, m), 7.44-7.46 (1H, m), 7.92 (1H, s), 8.00 (1H, t, J = 6.3 Hz),
        8.08-8.09 (1H, m), 8.33 (1H, s).
7-1731  δ 3.51 (3H, s), 6.79-6.83 (1H, m), 7.05 (1H, t, J = 7.6 Hz), 7.18-7.46 (4H, m), 7.94-8.00 (2H, m), 8.20 (1H, d, J = 12.4 Hz),
        8.34 (1H, s).
7-1732  δ 3.50 (3H, s), 7.00-7.18 (4H, m), 7.27-7.31 (1H, m), 7.45-7.48 (1H, m), 7.93 (1H, s), 8.01-8.03 (1H, m),
        8.12 (1H, broad-s), 8.34 (1H, s).
7-1733  δ 3.50 (3H, s), 6.91 (2H, s), 6.93-7.35 (3H, m), 7.47 (1H, t, J = 7.0 Hz), 7.93 (1H, s), 8.01-8.10 (1H, m), 8.13 (1H,
        broad-s), 8.34 (1H, s).
7-1750  δ 3.52 (3H, s), 7.28-7.71 (6H, m), 7.93 (1H, s), 8.06 (1H, t, J = 8.4 Hz), 8.34 (1H, s), 8.60 (1H, s).
7-1751  δ 3.52 (3H, s), 7.32 (1H, t, J = 8.3 Hz), 7.44-7.52 (5H, m), 7.93 (1H, s), 8.04-8.07 (2H, m), 8.34 (1H, s).
7-1752  δ 3.54 (3H, s), 6.74 (2H, s), 7.16-7.24 (2H, m), 7.50 (1H, t, J = 7.4 Hz), 7.94 (1H, s), 8.01-8.05 (1H, m), 8.25 (1H,
        broad-s), 8.35 (1H, s).
7-1764  δ 3.53 (3H, s), 7.20-7.21 (1H, m), 7.32 (1H, t, J = 7.8 Hz), 7.50 (1H, t, J = 7.8 Hz), 7.70-7.71 (1H, m),
        7.92 (1H, s), 8.01-8.04 (2H, m), 8.33 (1H, s), 8.53-8.54 (2H, m).
7-1766  δ 3.53 (3H, s), 7.14-7.17 (1H, m), 7.23-7.25 (1H, m), 7.54-7.55 (1H, m), 7.68 (1H, d, J = 8.0 Hz), 7.95 (1H, s),
        8.00 (1H, t, J = 7.0 Hz), 8.10-8.20 (1H, m), 8.28 (1H, d, J = 4.8 Hz), 8.36 (1H, s).
7-1773  δ 3.53 (3H, s), 7.19-7.40 (3H, m), 7.52-7.53 (1H, m), 7.67-7.68 (1H, m), 7.93 (2H, s), 8.07-8.09 (1H, m),
        8.32 (1H, d, J = 14.4 Hz), 8.35 (1H, s).
7-1794  δ 3.51 (3H, s), 7.18-7.23 (2H, m), 7.32 (1H, t, J = 7.8 Hz), 7.43-7.46 (1H, m), 7.92 (1H, s), 7.98-8.01 (1H,
        m), 8.08-8.09 (1H, m), 8.23-8.24 (1H, m), 8.32 (1H, s), 8.56-8.59 (1H, m).
7-1808  δ 3.51 (3H, s), 7.23-7.43 (6H, m), 7.44-7.60 (1H, m), 7.91 (1H, s), 7.98-8.01 (1H, m), 8.10 (1H, broad-s),
        8.32 (1H, s).
7-1809  δ 3.52 (3H, s), 6.80 (1H, t, J = 8.8 Hz), 7.06 (1H, t, J = 3.6 Hz), 7.17-7.23 (2H, m), 7.39-7.44 (1H, m),
        7.92-7.93 (2H, m), 7.99 (1H, t, J = 5.2 Hz), 8.16 (1H, d, J = 13.2 Hz), 8.33 (1H, s).
7-1810  δ 3.48 (3H, s), 6.99-7.16 (3H, m), 7.28-7.34 (2H, m), 7.43-7.45 (1H, m), 7.72 (1H, t, J = 8.0 Hz), 7.92 (1H, s),
        8.00 (1H, t, J = 8.0 Hz), 8.33 (1H, s).
7-1811  δ 3.53 (3H, s), 6.90 (2H, t, J = 8.0 Hz), 7.28-7.40 (3H, m), 7.46 (1H, t, J = 7.2 Hz), 7.92 (1H, s), 8.02 (1H, t, J = 8.0 Hz),
        8.13 (1H, d, J = 12.4 Hz), 8.33 (1H, s).
7-1828  δ 3.52 (3H, s), 7.32-7.35 (2H, m), 7.49-7.60 (3H, m), 7.69 (1H, s), 7.92 (1H, s), 8.05-8.08 (2H, m), 8.36 (1H, s).
7-1829  δ 3.53 (3H, s), 7.30-7.34 (1H, m), 7.45-7.52 (5H, m), 7.92 (1H, s), 8.04-8.07 (2H, m), 8.34 (1H, s).
7-1844  δ 3.54 (3H, s), 7.15 (1H, t, J = 5.2 Hz), 7.52-7.54 (1H, m), 7.68-7.71 (2H, m), 7.94 (1H, s), 8.00 (1H, t, J = 5.2 Hz),
        8.15-8.16 (1H, m), 8.28 (1H, d, J = 4.8 Hz), 8.34 (1H, s).
7-1851  δ 3.52 (3H, s), 7.65 (1H, d, J = 6.8 Hz), 7.92 (1H, s), 8.05-8.08 (2H, m), 8.11-8.18 (3H, m), 8.26-8.31 (1H, m),
        8.33 (1H, s).
7-3348  δ 3.48 (3H, s), 7.18-7.30 (6H, m), 7.45 (1H, broad-s), 7.52 (1H, broad-s), 7.74-7.76 (1H, m), 7.89 (1H, s),
        8.11 (1H, s).
7-3369  δ 3.49 (3H, s), 7.18-7.22 (1H, m), 7.45-7.53 (5H, m), 7.56 (2H, broad-s), 7.92 (1H, s), 8.14 (1H, s).
7-3384  δ 3.52 (3H, s), 7.15-7.20 (2H, m), 7.45-7.85 (4H, m), 7.92 (1H, s), 8.12-8.15 (1H, m), 8.27-8.29 (1H, m).
7-5902  δ 3.51 (3H, s), 7.00-7.52 (7H, m), 7.88 (1H, d, J = 1.5 Hz), 8.01-8.06 (3H, m).
7-5903  δ 3.55 (3H, s), 7.14 (1H, dd, J = 4.8, 7.8 Hz), 7.24-7.26 (1H, m), 7.40-7.60 (1H, m), 7.66-7.68 (1H, m),
        7.91 (1H, s), 8.01-8.05 (2H, m), 8.08 (1H, d, J = 1.5 Hz), 8.28 (1H, dd, J = 2.0, 4.8 Hz).
7-5904  δ 3.56 (3H, s), 7.05-7.09 (1H, m), 7.30-7.36 (2H, m), 7.43-7.48 (2H, m), 7.56 (1H, s), 7.65 (1H, s), 7.77 (1H, d, J = 8.0 Hz),
        7.90 (1H, d, J = 8.0 Hz), 8.07 (2H, s).
7-5905  δ 3.57 (3H, s), 6.89 (1H, t, J = 8.0 Hz), 7.15 (1H, t, J = 8.0 Hz), 7.32-7.36 (2H, m), 7.47 (1H, t, J = 8.0 Hz),
        7.53 (1H, s), 7.61 (1H, s), 7.77 (1H, d, J = 8.0 Hz), 8.09 (2H, s), 8.70 (1H, broad-s).
7-5906  δ 3.55 (3H, s), 7.00 (1H, t, J = 8.0 Hz), 7.07 (2H, d, J = 7.8 Hz), 7.16-7.22 (1H, m), 7.32 (1H, d, J = 6.8 Hz),
        7.44 (1H, t, J = 8.0 Hz), 7.57 (1H, s), 7.65-7.67 (1H, m), 7.74 (1H, d, J = 8.0 Hz), 7.85 (2H, s).
7-5907  δ 3.57 (3H, s), 6.90 (2H, t, J = 7.8 Hz), 7.29-7.34 (3H, m), 7.44 (1H, t, J = 7.8 Hz), 7.49 (1H, s), 7.62 (1H, s),
        7.73 (1H, d, J = 7.8 Hz), 7.85 (2H, s).
7-5908  δ 2.99 (3H, s), 3.58 (3H, s), 7.27-7.30 (1H, m), 7.43-7.44 (1H, m), 7.51 (2H, d, J = 8.3 Hz), 7.65-7.70 (3H,
        m), 7.81 (2H, d, J = 8.3 Hz), 7.91 (1H, s), 8.14 (1H, s).
7-5909  δ 3.60 (3H, s), 7.33 (1H, d, J = 7.9 Hz), 7.50 (1H, t, J = 7.9 Hz), 7.63 (1H, s), 7.70 (1H, s), 7.75 (1H, d, J = 7.9 Hz),
        7.94 (1H, s), 8.34 (1H, s), 8.65 (2H, s), 9.10 (1H, s).
7-5910  δ 3.53 (3H, s), 3.89 (3H, s), 7.32 (1H, t, J = 7.8 Hz), 7.48-7.49 (1H, m), 7.83-7.91 (2H, m), 8.01 (1H, t, J = 7.3 Hz),
        8.10-8.14 (3H, m), 8.22-8.23 (1H, m).
7-5911  δ 3.57 (3H, s), 7.20-7.35 (6H, m), 7.41-7.45 (2H, m), 7.53 (1H, s), 7.67 (1H, d, J = 7.8 Hz), 7.89 (1H, s),
        8.11 (1H, s).
7-5912  δ 3.58 (3H, s), 7.14 (1H, dd, J = 4.9, 7.8 Hz), 7.42-7.43 (2H, m), 7.55 (1H, s), 7.59 (1H, dd, J = 2.0, 7.8 Hz),
        7.67-7.68 (2H, m), 7.91 (1H, s), 8.13 (1H, s), 8.26 (1H, dd, J = 2.0, 4.9 Hz).
8-268   δ 3.28 (2/3*3H, s), 3.39 (1/3*3H, s), 7.13-7.14 (1/3*1H, m), 7.15-7.17 (1/3*1H, m), 7.34 (1/3*1H, s),
        7.36 (1/3*1H, s), 7.46-7.57 (12/3*1H, m), 7.74-7.90 (13/3*1H, m), 7.94 (2/3*1H, s), 8.05 (1/3*1H, s),
        8.15 (2/3*1H, s), 8.24 (2/3*1H, s).
8-288   (CDCl3 + DMSO-d6) δ 3.30 (3/4*3H, s), 3.40 (1/4*3H, s), 7.10-7.15 (1/4*1H, m), 7.20-7.25 (1/4*1H, m),
        7.35 (1/4*1H, s), 7.37 (1/4*1H, s), 7.50 (3/4*1H, t, J = 7.8 Hz), 7.62-7.66 (6/4*1H, m), 7.82-7.84 (5/4*1H,
        m), 7.94 (1/4*1H, s), 7.95 (3/4*1H, s), 8.00 (3/4*1H, t, J = 1.5 Hz), 8.08-8.10 (4/4*1H, m), 8.17 (3/4*1H,
        s), 8.18-8.19 (1/4*1H, m), 8.32-8.36 (4/4*1H, m), 8.48 (3/4*1H, t, J = 1.5 Hz), 10.00 (1/4*1H, s),
        10.29 (3/4*1H, s).
8-289   δ 3.26 (2/3*3H, s), 3.38 (1/3*3H, s), 7.08-7.09 (1/3*1H, m), 7.12-7.14 (1/3*1H, m), 7.32 (2/3*1H, d, J = 7.8 Hz),
        7.45-7.49 (3/3*1H, m), 7.72-7.76 (9/*13H, m), 7.83 (1/3*1H, s), 7.85-7.89 (4/3*1H, m),
        7.95 (2/3*1H, s), 7.98-8.00 (4/3*1H, m), 8.04 (2/3*1H, d, J = 6.3 Hz), 8.16 (2/3*1H, s), 8.57 (2/3*1H, s).
8-304   δ 3.29 (3/5*3H, s), 3.38 (2/5*3H, s), 7.14-7.18 (4/5*1H, m), 7.37-7.41 (8/5*1H, m), 7.50-7.52 (5/5*1H,
        m), 7.72 (2/5*1H, s), 7.83-7.86 (8/5*1H, m), 7.95 (3/5*1H, s), 8.05-8.07 (4/5*1H, m), 8.14-8.17 (6/5*1H,
        m), 8.30 (2/5*1H, s), 8.51-8.53 (5/5*1H, m), 8.57 (3/5*1H, s).
8-804   δ 3.31 (3H, s), 7.30-7.33 (1H, m), 7.48-7.52 (3H, m), 7.56-7.60 (1H, m), 7.72-7.74 (1H, m), 7.86-7.91 (3H,
        m), 8.06 (1H, s), 8.22 (2H, s).
8-824   (DMSO-d6) δ 3.32 (12/13*3H, s), 3.43 (1/13*3H, s), 7.01-7.02 (1/13*1H, m), 7.20-7.21 (1/13*1H, m),
        7.28 (12/13*1H, d, J = 7.8 Hz), 7.50 (12/13*1H, t, J = 7.8 Hz), 7.60-7.61 (1/13*1H, m), 7.65 (12/13*1H, t, J = 7.8 Hz),
        7.83-7.84 (13/13*1H, m), 7.85 (1/13*1H, d, J = 1.5 Hz), 7.94 (12/13*1H, d, J = 1.5 Hz),
        8.10-8.12 (12/13*1H, m), 8.14 (1/13*2H, s), 8.21-8.22 (1/13*1H, m), 8.23 (12/13*2H, s), 8.32-8.35 (13/13*1H, m),
        8.47-8.48 (13/13*1H, m), 10.05 (1/13*1H, s), 10.37 (12/13*1H, s).
8-840   δ 3.30 (10/11*3H, s), 3.43 (1/11*3H, s), 7.17-7.18 (1/11*1H, m), 7.19-7.20 (1/11*1H, m),
        7.33-7.42 (22/11*1H, m), 7.52 (10/11*1H, t, J = 7.8 Hz), 7.71 (1/11*1H, s), 7.75 (10/11*1H, s), 7.87 (10/11*1H, d, J = 8.3 Hz),
        8.12-8.13 (1/11*1H, m), 8.14 (1/11*2H, s), 8.17 (10/11*1H, dd, J = 2.0, 7.8 Hz), 8.23 (10/11*2H,
        s), 8.47-8.50 (11/11*1H, m), 8.52-8.53 (11/11*1H, m).
9-270   δ 2.64 (3/4*3H, s), 3.28 (1/4*3H, s), 3.37 (1/4*3H, s), 3.56 (3/4*3H, s), 6.70-6.71 (1/4*1H, m),
        6.80-6.81 (1/4*1H, m), 7.02-7.03 (4/4*1H, m), 7.16-7.26 (16/4*1H, m), 7.34-7.36 (10/4*1H, m),
        7.39-7.40 (1/4*1H, m), 7.46 (3/4*1H, t, J = 7.8 Hz), 7.80 (1/4*1H, s), 7.91 (3/4*1H, s), 8.01 (1/4*1H, s),
        8.11 (3/4*1H, s).
9-290   δ 2.88 (2/3*3H, s), 3.33 (1/3*3H, s), 3.37 (1/3*3H, s), 3.56 (2/3*3H, s), 6.70-6.71 (1/3*1H, m),
        6.95-6.98 (2/3*1H, m), 7.10 (2/3*1H, s), 7.28-7.42 (9/3*1H, m), 7.47-7.60 (6/3*1H, m), 7.62-7.63 (4/3*1H,
        m), 7.86 (1/3*1H, s), 7.93 (2/3*1H, s), 8.08 (1/3*1H, s), 8.14 (2/3*1H, s).
9-291   δ 2.82 (2/3*3H, s), 3.30 (1/3*3H, s), 3.37 (1/3*3H, s), 3.56 (2/3*3H, s), 6.75-6.76 (1/3*1H, m),
        6.95 (1/3*1H, t, J = 7.8 Hz), 7.00-7.01 (1/3*1H, m), 7.06 (2/3*1H, s), 7.28-7.32 (4/3*1H, m),
        7.39-7.54 (15/3*1H, m), 7.83 (1/3*1H, s), 7.93 (2/3*1H, s), 8.04 (1/3*1H, s), 8.14 (2/3*1H, s).
9-306   δ 2.89 (2/3*3H, s), 3.30 (1/3*3H, s), 3.36 (1/3*3H, s), 3.57 (2/3*3H, s), 6.96-6.97 (1/3*1H, m),
        7.04-7.05 (2/3*1H, m), 7.13-7.17 (2/3*1H, m), 7.27-7.41 (10/3*1H, m), 7.60-7.63 (3/3*1H, m), 7.81 (1/3*1H,
        s), 7.94 (2/3*1H, s), 8.02 (1/3*1H, s), 8.15 (2/3*1H, s), 8.24-8.25 (3/3*1H, m).
9-2164  δ 2.18-2.19 (3H, m), 3.48 (3H, s), 7.21-7.25 (4H, m), 7.32-7.40 (4H, m), 7.92 (1H, s), 8.13 (1H, s).
9-2322  δ 2.71-2.72 (3H, m), 3.47 (3H, s), 6.95-6.96 (1H, m), 7.11-7.16 (3H, m), 7.38-7.39 (2H, m), 7.95 (1H, s),
        8.02 (1H, s), 8.34 (1H, s).
11-777  δ 4.88 (2H, s), 7.20-7.21 (1H, m), 7.36 (1H, t, J = 7.8 Hz), 7.84-7.87 (1H, m), 7.92 (1H, s), 8.14-8.17 (2H,
        m), 8.36 (1H, broad-s).
11-835  δ 4.88 (2H, s), 7.22-7.23 (1H, m), 7.36 (1H, t, J = 7.8 Hz), 7.85-7.88 (1H, m), 7.95 (1H, s), 8.19 (1H, d, J = 13.1 Hz),
        8.36-8.37 (2H, m).
12-777  δ 3.39 (3H, s), 4.74 (2H, broad-s), 7.37 (1H, t, J = 7.8 Hz), 7.52-7.56 (1H, m), 7.92 (1H, s), 8.11-8.14 (2H,
        m), 8.25 (1H, d, J = 14.1 Hz).
12-835  δ 3.40 (3H, s), 4.74 (2H, broad-s), 7.37 (1H, t, J = 7.8 Hz), 7.55-7.58 (1H, m), 7.95 (1H, s), 8.12-8.13 (1H,
        m), 8.28-8.31 (1H, m), 8.36 (1H, s).
12-864  δ 3.40 (3H, s), 4.74 (2H, broad-s), 7.37 (1H, t, J = 7.8 Hz), 7.52-7.58 (1H, m), 7.93 (1H, s), 8.12-8.15 (1H,
        m), 8.28-8.34 (2H, m).
17-1103 δ 3.65 (3H, s), 7.28-7.41 (6H, m), 7.77 (1H, t, J = 7.8 Hz), 7.91 (1H, s), 8.00-8.02 (1H, m), 8.14 (1H, s),
        9.39 (1H, s).
22-435  δ 3.63 (3H, s), 4.90 (2H, s), 7.92-7.97 (2H, m), 8.08-8.15 (3H, m), 9.72 (1H, s).
27-627  δ 3.72 (3H, s), 7.51-7.60 (5H, m), 7.90 (1H, s), 8.05 (1H, s), 8.14 (1H, s), 9.11 (1H, s).
27-628  δ 3.67 (3H, s), 6.99-7.24 (1H, m), 7.29-7.35 (1H, m), 7.52-7.59 (2H, m), 7.90 (1H, s), 8.06 (1H, s),
        8.14 (1H, s), 9.08 (1H, s).
27-663  δ 3.63 (3H, s), 7.44-7.47 (1H, m), 7.80 (1H, dd, J = 2.0, 7.8 Hz), 7.90 (1H, s), 8.10 (1H, s), 8.14 (1H, s),
        8.58-8.60 (1H, m), 9.04 (1H, s).
32-247  δ 3.77-3.78 (3H, m), 4.96 (2H, s), 7.90 (1H, s), 8.00 (1H, s), 8.14 (1H, s), 9.02 (1H, s).

The pest control agent including the compound of the present invention as an active ingredient can effectively control, at a low concentration thereof, any pests such as insects including various agricultural pests damaging agricultural/horticultural crops, trees, and the like, insanitary pests adversely affecting the living environment of humans such as houses and the like in various manners, stored grain pests damaging grain and the like stored in a warehouse, wood-eating pests damaging wood such as buildings and the like, and mites, crustaceans, molluscs, and nematodes which propagate and cause damage in a manner similar to that in the case of the insects.

Specific examples of the insects, the mites, the crustaceans, molluscs and nematodes which can be controlled using the compound of the present invention include lepidopteran insects such as Adoxophyes honmai, Adoxophyes orana faciata, Archips breviplicanus, Grapholita inopinata, Archips fuscocupreanus, Grapholita molesta, Choristoneura magnanima, Leguminivora glycinivorella, Olethreutes mori, Caloptilia zachrysa, Argyresthia conjugella, Spulerrina astaurota, Matsumuraeses phaseoli, Pandemis heparana, Bucculatrix pyrivorella, Lyonetia clerkella, Carposina niponensis, Lyonetia prunifoliella malinella, Caloptilia theivora, Phyllonorycter ringoniella, Phyllocnistis citrella, Acrolepiopsis sapporensis, Acrolepiopsis suzukiella, Plutella xylostella, Stathmopoda masinissa, Helcystogramma triannulella, Pectinophora gossypiella, Carposina sasakii, Chilo suppressalis, Cnaphalocrocis medinalis, Ephestia elutella, Conogethes punctiferalis, Diaphania indica, Etiella zinckenella, Glyphodes pyloalis, Scirpophaga incertulas, Hellula undalis, Ostrinia furnacalis, Ostrinia scapulalis, Parapediasia teterrella, Parnara guttata, Pieris brassicae, Pieris rapae crucivora, Papilio xuthus, Ascotis selenaria, Pseudoplusia includens, Euproctis pseudoconspersa, Lymantria dispar, Orgyia thyellina, Hyphantria cunea, Lemyra imparilis, Adris tyrannus, Aedia leucomelas, Agrotis ipsilon, Agrotis segetum, Autographa nigrisigna, Ctenoplusia agnata, Cydla pomonella, Helicoverpa armigera, Helicoverpa assulta, Helicoverpa zea, Heliothis virescens, Ostrinia nubilalis, Mamestra brassicae, Mythimna separata, Sesamia inferens, Naranga aenescens, Spodoptera eridania, Spodoptera exigua, Spodoptera frugiperda, Spodoptera littoralis, Spodoptera litura, Spodoptera depravata, Trichoplusia ni, Endopiza viteana, Manduca quinquemaculata, Manduca sexta, and the like;

Hemipteran insects such as Arboridia apicalis, Balclutha saltuella, Epiacanthus stramineus, Empoascafabae, Empoasca nipponica, Empoasca onukii, Empoasca sakaii, Macrosteles striifrons, Nephotettix cinctinceps, Psuedatomoscelis seriatus, Laodelphax striatella, Nilaparvata lugens, Sogatellafurcfera, Diaphorina citri, Psylla pyrisuga, Aleurocanthus spiniferus, Bemisia argentifolii, Bemisia tabaci, Dialeurodes citri, Trialeurodes vaporariorum, Aleurolobus taonabae, Viteus vitifolii, Lipaphis erysimi, Aphis gossypii, Aphis spiraecola, Myzus persicae, Toxoptera aurantii, Drosicha corpulenta, Icerya purchasi, Phenacoccus solani, Pulvinaria aurantii, Planococcus citri, Pseudaonidia duplex, Planococcus kuraunhiae, Pseudococcus comstocki, Comstockaspis perniciosa, Ceroplastes ceriferus, Ceroplastes rubens, Aonidiella aurantii, Fiorinia theae, Pseudaonidia paeoniae, Pseudaulacaspis pentagona, Pseudaulacaspis prunicola, Unaspis euonymi, Unaspis yanonensis, Cimex lectularius, Dolycoris baccarum, Eurydema rugosum, Eysarcoris aeneus, Eysarcoris lewisi, Eysarcoris ventralis, Glaucias subpunctatus, Halyomorpha halys, Nezara antennata, Nezara viridula, Piezodorus hybneri, Plautia crossota, Scotinophora lurida, Cletus punctiger, Leptocorisa chinensis, Riptortus clavatus, Rhopalus msculatus, Cavelerius saccharivorus, Togo hemipterus, Dysdercus cingulatus, Stephanitis pyrioides, Halticus insularis, Lygus lineolaris, Stenodema sibiricum, Stenotus rubrovittatus, Trigonotylus caelestialium, and the like;

Coleopteran insects such as Anomala cuprea, Anomala rufocuprea, Gametis jucunda, Heptophylla picea, Popillia japonica, Lepinotarsa decemlineata, Epilachna varivestis, Melanotus fortnumi, Melanotus tamsuyensis, Lasioderma serricorne, Lyctusbrunneus, Tomicus piniperda, Rhizopertha dominica, Epuraea domina, Epilachna varivestis, Epilachna vigintioctopunctata, Tenebrio molitor, Tribolium castaneum, Anoplophora malasiaca, Monochamus alternatus, Psacothea hilaris, Xylotrechus pyrrhoderus, Callosobruchus chinensis, Aulacophora femoralis, Oulema oryzae, Chaetocnema concinna, Diabrotica undecimpunctata, Diabrotica virgifera, Diabrotica barberi, Phyllotreta striolata, Psylliodes angusticollis, Rhynchites heros, Cylas formicarius, Anthonomus grandis, Echinocnemus squameus, Euscepes postfasciatus, Hypera postica, Lissohoptrus oryzophilus, Otiorhynchus sulcatus, Sitophilus granarius, Sitophilus zeamais, Sphenophorus venatus vestitus, Paederus fuscipes, and the like;

Thysanopteran insects such as Frankliniella intonsa, Thrips flavus, Frankliniella occidentalis, Heliothrips haemorrhoidalis, Scirtothrips dorsalis, Thrips palmi, Thrips tabaci, Ponticulothrips diospyrosi, and the like;

Dipterous insects such as Asphondylia yushimai, Sitodiplosis mosellana, Bactrocera cucurbitae, Bactrocera dorsalis, Ceratitis capitata, Hydrellia griseola, Drosophila suzukii, Agromyza oryzae, Chromatomyia horticola, Liriomyza bryoniae, Liriomyza chinensis, Liriomyza sativae, Liriomyza trifolii, Delia platura, Delia antique, Pegomya cunicularia, Rhagoletis pomonella, Mayetiola destructo, Musca domestica, Stomoxys calcitrans, Melophagus ovinus, Hypoderma bovis, Hypoderma lineatum, Oestrus ovis, Glossina palpalis, Glossina morsitans, Pmsimulium yezoensis, Tabanus trigonus, Telmatoscopus albipunctatus, Leptoconops nipponensis, Culex pipiens pallens, Aedes aegypti, Aedes albopicutus, Anopheles hyracanus sinesis, and the like;

Hymenopteran insects such as Apethymus kuri, Athalia rosae, Arge pagana, Neodiprion sertifer, Dryocosmus kuriphilus, Eciton burchelli, Eciton schmitti, Camponotus japonicus, Vespa mandarina, Myrmecia spp., Solenopsis spp., Monomorium pharaonis, and the like;

Orthopteran insects such as Teleogryllus emma, Gryllotalpa orientalis, Locusta migratoria, Oxya yezoensis, Schistocerca gregaria, and the like;

Collembolan insects such as Onychiurus folsomi, Onychiurus sibiricus, Bourletiella hortensis, and the like;

Dictyopteran insects such as Periplaneta fuliginosa, Periplaneta japonica, Blattella germanica, Periplaneta Americana, and the like;

Isopterous insects such as Coptotermes formosanus, Reticulitermes speratus, Odontotermes formosanus, and the like;

Isopterous insects such as Ctenocephalidae felis, Ctenocephalides canis, Echidnophaga gallinacea, Pulex irritans, Xenopsylla cheopis, and the like;

Mallophaga insects such as Menacanthus stramineus, Bovicola bovis, and the like;

Anoplura insects such as Haematopinus eurysternus, Haematopinus suis, Linognathus vituli, Solenopotes capillatus, and the like;

Tarsonemidae such as Phytonemus pallidus, Polyphagotarsonemus latus, Tarsonemus bilobatus, and the like;

Eupodidae such as Penthaleus erythrocephalus, Penthaleus major, and the like;

Tetranychidae such as Oligonychus shinkajii, Panonychus citri, Panonychus mori, Panonychus ulmi, Tetranychus kanzawai, Tetranychus urticae, and the like;

Eriophydae such as Acaphylla theavagrans, Aceria tulipae, Aculops lycopersici, Aculops pelekassi, Aculus schlechtendali, Eriophyes chibaensis, Phyllocoptruta oleivora, and the like;

Acaridae such as Rhizoglyphus robini, Tyrophagus putrescentiae, Tyrophagus similis, and the like;

Varroidae such as Varroa jacobsoni, and the like;

Ixodidae such as Boophilus microplus, Rhipicephalus sanguineus, Haemaphysalis longicornis, Haemophysalis flava, Haemophysalis campanulata, Ixodes ovatus, Ixodes persulcatus, Amblyomma spp., Dermacentor spp., and the like;

Cheyletidae such as Cheyletiella yasguri, Cheyletiella blakei, and the like;

Demodicidae such as Demodex canis, Demodex cati, and the like;

Psoroptidae such as Psoroptes ovis, and the like;

Sarcoptidae such as Sarcoptes scabiei, Notoedres cati, Knemidocoptes spp., and the like;

Crustacea such as Armadillidium vulgare, and the like;

Gastropoda such as Pomacea canaliculata, Achatina fulica, Meghimatium bilineatum, Limax Valentiana, Acusta despecta sieboldiana, Euhadra peliomphala, and the like; and

Nematoda such as Prathylenchus coffeae, Prathylenchus penetrans, Prathylenchus vulnus, Globodera rostochiensis, Heterodera glycines, Meloidogyne hapla, Meloidogyne incognita, Aphelenchoides besseyi, Bursaphelenchus xylophilus, and the like, but the present invention is not limited thereto.

The pest control agent including the compound according to the present invention as an active ingredient has a significant control effect against the above-described harmful crops which damage lowland crops, upland crops, fruit trees, vegetables, and other crops and ornamental flowers, and therefore, the effect as a pest control agent of the present invention can be obtained by treating the paddy field water, plant stems and leaves, or soil of the crops of lowland, upland, fruit trees, vegetables, other crops, ornamental flowers, and the like during the seasons in which the appearance of such pests is expected, or before or at the point when the pest appearance is observed.

The pest control agent including the compound according to the present invention as an active ingredient has a significant control effect against stored grain pests and the like generated during storage of the harvest. That is, the the pest control agent having the compound of the present invention as an active ingredient may be subjected to a treatment after the harvest (post harvest) such as spray-spreading, coating, dipping, dressing, fumigation/smoking, pressurized injection, and the like with respect to the harvest or the place for storage of the harvest.

Further, the pest control agent including the compound according to the present invention as an active ingredient can be applied to plant seeds to prevent the damage caused by pests generated in the plants after seeding. That is, the pest control agent having the compound of the present invention as an active ingredient may be subjected to a treatment such as spray-spreading, dipping, dressing, and the like on the plant seeds in an effective amount for controlling the pests as it is, as an adequate dilution with water or the like, or as a suspension to bring the compound of the present invention into contact with the plant seeds.

The plant seeds refer to those used for breeding in agriculture by storing the nutrients for seedling germination, and examples thereof include seeds such as corn, soybeans, red beans, cotton, rice, sugar beet, wheat, barley, sunflower, tomato, cucumber, eggplant, spinach, sting beans, squash, sugarcane, tobacco, pimento, canola, and the like, seed tubers such as taro, potato, sweet potato, konjac, and the like, bulbs such as edible lily, tulips, and the like, and seed balls such as rakkyo and the like.

The pest control agent having the compound of the present invention as an active ingredient has a significant control effect against insanitary pests such as Diptera pests (Culex pipiens pallens, Culex pipiens, Chironomidae, houseflies, sandflies, horsefly, and the like) Dictyoptera pests (Blattella germanica, Periplaneta fuliginosa, Periplaneta americana, and the like), and other pests.

The pest control agent having the compound of the present invention as an active ingredient has a significant control effect against wood-feeding pests such as termites, Lyctusbrunneus, Rhizopertha dominica, Anobiidae, Cerambycidae, and the like, thus, the above-described wood-feeding pests can be controlled by treatment of wood, soil, buildings, and the like with the pest control agent.

Since the compound of the present invention exhibits a control effect against various pests and also exhibits an effect of protecting useful crops and an excellent control effect as a pesticide or a miticide at a low dose, it has an effect of contributing to reduction in an environmental impact. In addition, the compound of the present invention also exerts an excellent control effect when used in combination with other agricultural/horticultural pesticides, miticides, nematocides, fungicides, herbicides, plant growth regulators, biological agricultural chemicals, or the like.

For the use of the compound of the present invention, the compound can be put to practical use as a preparation in any form such as a soluble concentrate, an emulsifiable concentrate, a wettable powder, a water-soluble powder, a water dispersible granule, a water-soluble granule, a suspension concentrate, a concentrated emulsion, a suspoemulsion, a microemulsion, a dustable powder, a granule, a tablet, and an emulsifiable gel, typically by mixing the compound with a suitable solid carrier or liquid carrier, further if desired by adding to the resultant mixture, a surfactant, a penetrant, a spreader, a thickener, an antifreezing agent, a binder, an anticaking agent, a disintegrant, a defoaming agent, an antiseptic or a stabilizer. In addition, from the labor-saving and safety-enhancing viewpoints, the compound can be put to use by encapsulating the above preparation in any form in a water-soluble packaging material such as a water-soluble capsule and a bag of water-soluble film.

The inert carrier which can be used in the present invention may be solids or liquids, and examples thereof include soybean powders, grain powders, wood powders, bark powders, sawdust powders, tobacco stem powders, walnut shell powders, brans, cellulose powders, residues from plant extraction, synthetic polymers such as pulverized synthetic resins, clays (for example, kaolin, bentonite, acidic white clay), talcs (for examples, talc, pyrophyllite, etc.), silica (for examples, diatomaceous earth, sand, mica, white carbon [hydrous silica powders, synthetic high dispersity silicates called hydrous silicate, there are also products containing calcium silicate as a main component]), activated carbon, sulfur powder, pumice, calcined diatomaceous powders, pulverized bricks, fly ash, sand, inorganic mineral powders such as calcium carbonate, calcium phosphate, and the like, chemical fertilizers such as ammonium sulfate, ammonium phosphate, ammonium nitrate, urea, ammonium chloride, and the like, a compost, and others, which are used alone or as a mixture of two or more kinds thereof.

Materials which can be used as the liquid inert carrier are selected from those having the function as solvent, as well as those capable of dispersing the active ingredient compound with the aid of an adjuvant even if the inert carrier does not have a function as a solvent. Representative examples thereof include the carriers listed below: water, alcohols (for example, methanol, ethanol, isopropanol, butanol, ethylene glycol, and the like), ketones (for example, acetone, methyl ethyl ketone, methyl isobutyl ketone, diisobutylketone, cyclohexanone, and the like), ethers (for example, diethyl ether, dioxane, cellosolve, diisopropyl ether, tetrahydrofuran, and the like), aliphatic hydrocarbons (for example, kerosene, mineral oil, and the like), aromatic hydrocarbons (for example, benzene, toluene, xylene, solvent naphtha, alkyl naphthalene, and the like), halogenated hydrocarbons (for example, dichloromethane, chloroform, tetrachlorocarbon, chlorobenzene, and the like), esters (for example, ethyl acetate, butyl acetate, ethyl propionate, diisobutyl phthalate, dibutyl phthalate, dioctyl phthalate, and the like), amides (for example, dimethyl formamide, diethyl formamide, dimethyl acetamide, and the like), and nitriles (for example, acetonitrile, and the like), which are used alone or as mixtures of two or more kinds thereof.

These solid and liquid carriers may be used alone or in a combination of two or more kinds thereof.

Examples of the surfactant include nonionic surfactants such as polyoxyethylene alkyl ethers, polyoxyethylene alkyl (mono- or di-)phenyl ethers, polyoxyethylene (mono-, di-, or tri-)styryl phenyl ethers, polyoxyethylene-polyoxypropylene block copolymers, polyoxyethylene aliphatic acid (mono- or di-) esters, sorbitan aliphatic acid esters, polyoxyethylene sorbitan aliphatic acid esters, castor oil ethylene-oxide adducts, acetylene glycol, acetylene alcohols, acetylene glycol ethylene-oxide adducts, acetylene alcohol ethylene-oxide adducts, alkylglucosides, and the like; anionic surfactants such as alkyl sulfate ester salts, alkylbenzene sulfonates, lignin sulfonates, alkyl sulfosuccinates, naphthalene sulfonates, alkylnaphthalene sulfonates, salts of naphthalene sulfonate formalin condensate, salts of alkylnaphthalene sulfonate formalin condensate, polyoxyethylenealkylether sulfate or phosphate esters salts, polyoxyethylene (mono- or di-) alkylphenyl ether sulfate or phosphate esters, polyoxyethylene (mono-, di-, or tri-) styrylphenyl ether sulfate or phosphate esters, polycarboxylic acid salts (such as polyacrylic acid salts, polymaleic acid salts, maleic acid-olefin copolymers, and the like), polystyrene sulfonates, and the like; cationic surfactants such as alkylamine salts, alkyl quaternary ammonium salts, and the like; amphoteric surfactants such as amino acid-type surfactants, betaine-type surfactants, and the like; silicone-based surfactants; and fluorinated surfactants.

The content of these surfactants is not particularly limited, but it is preferably in the range of usually 0.05 part by weight to 20 parts by weight, with respect to 100 parts by weight of the preparation of the present invention. In addition, these surfactants may be used alone or in combination of two or more kinds thereof.

In order to control various pests, an amount effective for blight control can be applied as it is or as an adequate dilution with water or the like, or as a suspension, to the crops on which appearance of the corresponding pests is expected or to places where such occurrence is not preferable. The amount of use depends on various factors such as, for example, the purpose, the pest to be controlled, the state of plant growth, trends in pest appearance, climate, environmental conditions, Formulation, method of use, place of use, timing of use, and the like, but it is preferable to use the active ingredient in the concentration of 0.0001 ppm to 5000 ppm, and preferably 0.01 ppm to 1000 ppm. The dose that can be used per 10 a is generally in the range of 1 g to 300 g of the active ingredient.

The amount of the active ingredient of the compound of the present invention is usually 0.1% by weight to 20% by weight for powders, 5% by weight to 50% by weight for emulsifiable concentrates, 3% by weight to 90% by weight for wettable powders, 0.1% by weight to 20% by weight for granules, 5% by weight to 90% by weight for flowable Formulations, or 3% by weight to 90% by weight for water dispersible granules. The amount of the carrier in each form is usually 60% by weight to 99.9% by weight for powders, 40% by weight to 95% by weight for emulsifiable concentrates, 10% by weight to 90% by weight for wettable powders, 80% by weight to 99.9% by weight for granules, 10% by weight to 95% by weight for flowable Formulations, or 10% by weight to 90% by weight for water dispersible granules. Further, the amount of the adjuvant is usually 0.1% by weight to 20% by weight for powders, 1% by weight to 20% by weight for emulsifiable concentrates, 0.1% by weight to 20% by weight for wettable powders, 0.1% by weight to 20% by weight for granules, 0.1% by weight to 20% by weight for flowable Formulations, and 0.1% by weight to 20% by weight for water dispersible granules.

When the compound of the present invention is used as an agricultural chemical, it may be used, if required, as a mixture with other herbicides, various pesticides, miticides, nematocides, fungicides, plant growth regulators, synergists, fertilizers, soil conditioners, or the like to be applied during the preparation or the dusting.

All literature, patent applications, and technical specifications cited in the present specification are herein incorporated by reference as if each such individual piece of literature, patent application, and technical specification were specifically and individually indicated to be incorporated herein by reference.

EXAMPLES

Representative Examples of the present invention will be described with reference to the following Examples, but the present invention is not limited thereto. In the present Examples, DMF means N,N-dimethyl formamide, THF means tetrahydrofuran, IPE means isopropyl ether, DMI means 1,3-dimethyl-2-imidazolidinone, and DMSO means dimethylsulfoxide.

Furthermore, “%” is based on mass unless specified otherwise.

Example 1

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide (Compound No. 7-1574)

<1-1>

Preparation of 4-(perfluoropropan-2-yl)-2-(trifluoromethyl)aniline

100 g (0.608 mol) of 2-(trifluoromethyl)aniline, 131 g (0.639 mol) of 85% sodium hydrosulfite, and 20.9 g (0.0608 mol) of tetrabutylammonium hydrogen sulfate were charged to a mixed solution of 1500 ml of ethyl acetate and 1500 ml of water, and 53.9 g (0.639 mol) of sodium hydrogen carbonate was added thereto. 198 g (0.669 mol) of heptafluoroisopropyl iodide was added dropwise thereto at room temperature, followed by stirring at room temperature for 6 hours. After the liquid separation, the solvent of the organic layer was evaporated under reduced pressure, and 500 ml of ethyl acetate was charged thereto. 160 g (0.608 mol) of a 4 M hydrogen chloride/ethyl acetate solution was added dropwise thereto, followed by stirring at room temperature for 30 minutes, and then stirring at 5° C. for 1 hour. After the filtration, the filtrate was washed with water and a saturated aqueous sodium hydrogen carbonate in this order, and then dried over anhydrous magnesium sulfate, and the solvent was evaporated under reduced pressure. The obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=10:1) to prepare 60.0 g (yield 30%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 4.49 (2H, broad-s), 6.81 (1H, d, J=8.3 Hz), 7.48 (1H, d, J=8.3 Hz), 7.64 (1H, s).

<1-2>

Preparation of 2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline

100 g (0.273 mol) of 4-(perfluoropropan-2-yl)-2-(trifluoromethyl)aniline was charged to 500 ml of DMF, and 52.1 g (0.287 mol) of N-bromosuccinimide was charged in separate portions thereto over 30 minutes. After stirring at 60° C. for 2 hours, and then cooling to room temperature, the mixture was discharged to 2000 ml of water. The mixture was extracted with ethyl acetate, then washed with saturated brine, and dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=20:1) to prepare 89.0 g (yield 80%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 5.03 (2H, broad-s), 7.61 (1H, s), 7.79 (1H, s).

<1-3>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-chloro-3-nitrobenzamide

3.60 g (8.82 mmol) of 2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline was charged to 20 ml of anhydrous THF, and cooled to −70° C. under a nitrogen atmosphere. 4.85 ml (9.70 mmol) of a 2.0 M lithium diisopropyl amide hexane solution was added dropwise thereto, then 2.34 g (10.7 mmol) of acid chloride which was prepared from 2-chloro-3-nitrobenzoic acid and thionyl chloride was dissolved in 5 ml of anhydrous THF, and was added dropwise thereto, followed by stirring at −70° C. for 30 minutes and then stirring at room temperature for 30 minutes. The mixture was discharged to an aqueous ammonium chloride solution, then extracted with ethyl acetate, and dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=10:1→8:2→3:1) to prepare 1.76 g (yield: 34%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.61 (1H, t, J=7.8 Hz), 7.67 (1H, broad-s), 7.93-7.97 (3H, m), 8.18 (1H, broad-s).

<1-4>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-nitrobenzamide

To a solution of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-chloro-3-nitrobenzamide 4.89 g (8.27 mmol) in 50 ml of anhydrous DMF was added 2.40 g (41.3 mmol) of potassium fluoride (spray-dried product) under a flow of nitrogen, followed by stirring at 130° C. for 10 hours. Liquid separation was carried out by adding ethyl acetate, hexane, and water to the reaction mixture, and then the organic layer was washed with water and saturated brine, and dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=10:1) to prepare 0.940 g (yield 20%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.53 (1H, t, J=7.3 Hz), 7.93 (1H, broad-s), 8.17-8.18 (2H, m), 8.28-8.32 (1H, m), 8.44-8.48 (1H, m).

<1-5>

Preparation of 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluorobenzamide

0.940 g (1.63 mmol) of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-nitrobenzamide and 0.960 g (5.05 mmol) of stannous chloride (anhydrous) were added to 10 ml of ethanol, and 1.02 ml (9.78 mmol) of concentrated hydrochloric acid was added thereto, followed by stirring at 60° C. for 4 hours. The reaction mixture was adjusted to pH 10 by the addition of an aqueous sodium hydroxide solution, and the precipitated insolubles were removed by filtration using Celite. The filtrate on Celite was washed with ethyl acetate. The filtrate was extracted with ethyl acetate, and the organic layer was washed with a 20% aqueous sodium hydroxide solution and saturated brine, and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=4:1) to prepare 0.930 g (yield 99%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 3.93 (2H, broad-s), 6.99-7.04 (1H, m), 7.11 (1H, t, J=7.8 Hz), 7.47-7.49 (1H, m), 7.91 (1H, s), 8.14 (1H, s), 8.28 (1H, d, J=14.6 Hz).

<1-6>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(methylamino)benzamide

0.930 g (1.71 mmol) of 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluorobenzamide was added to 5 ml of concentrated sulfuric acid, and 10 ml of a 37% aqueous formaldehyde solution was charged dropwise thereto at 40° C. The reaction mixture was poured into ice-water, adjusted to pH 10 using an aqueous sodium hydroxide solution, and extracted with the addition of ethyl acetate. The organic layer was washed with a 20% aqueous sodium hydroxide solution and saturated brine, and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=8:1) to prepare 0.690 g (yield 72%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 2.94 (3H, s), 4.14 (1H, broad-s), 6.88-6.93 (1H, m), 7.18 (1H, t, J=7.8 Hz), 7.37-7.41 (1H, m), 7.90 (1H, s), 8.13 (1H, s), 8.27 (1H, d, J=14.6 Hz).

[1-7] Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide (Compound No. 7-1574)

To a solution of 1.54 g (2.75 mmol) of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(methylamino)benzamide and 0.330 g (4.13 mmol) of pyridine in 5 ml of THF was added 0.460 g (3.30 mmol) of benzoyl chloride, followed by stirring at 60° C. for 5 hours. To the reaction mixture were added water and ethyl acetate, and the organic layer was washed with 1 M hydrochloric acid, a saturated aqueous sodium hydrogen carbonate solution, and saturated brine, and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=8:1), and the obtained solid was washed with IPE to prepare 1.45 g (yield 80%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 3.50 (3H, s), 6.99-7.33 (6H, m), 7.43-7.45 (1H, m), 7.90 (1H, s), 7.97-8.06 (2H, m), 8.13 (1H, s).

Example 2

Preparation of 2-chloro-N-(3-(2,6-dibromo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)nicotinamide (Compound No. 6-1140)

<2-1>

Preparation of 4-(perfluoropropan-2-yl)aniline

100 g (1.02 mol) of aniline, 230 g (1.12 mol) of 85% sodium hydrosulfite, and 35.1 g (0.100 mol) of tetrabutylammonium hydrogen sulfate were charged to a mixed solution of 1500 ml of t-butyl methyl ether and 1500 ml of water, and 94.7 g (1.12 mol) of sodium hydrogen carbonate was added thereto. 350 g (1.12 mol) of heptafluoroisopropyl iodide was added dropwise thereto at room temperature, followed by stirring at room temperature for 6 hours. After the liquid separation, the organic layer was washed with 1 M hydrochloric acid, water, and a saturated aqueous sodium hydrogen carbonate solution, and then dried over anhydrous sodium sulfate. The solvent was evaporated under reduced pressure, and 500 ml of ethyl acetate was charged thereto. 255 g (1.02 mol) of a 4 M hydrogen chloride/ethyl acetate solution was added dropwise thereto, followed by stirring at room temperature for 30 minutes and at 5° C. for 1 hour. The precipitated solid was separated by filtration, and the solid was charged to 1000 ml of ethyl acetate, adjusted to pH 8 to 9 by the addition of 1000 ml of a saturated aqueous sodium hydrogen carbonate solution at 20° C. or lower, and subjected to liquid separation. The organic layer was dried over anhydrous sodium sulfate, and then the solvent was evaporated under reduced pressure to prepare 188 g (yield 71%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 3.92 (2H, broad-s), 6.69-6.74 (2H, m), 7.35 (2H, d, J=9.3 Hz).

<2-2>

Preparation of 2,6-dibromo-4-(perfluoropropan-2-yl)aniline

216 g (0.802 mol) of 4-(perfluoropropan-2-yl)aniline was charged to 863 ml of DMF, followed by cooling to 5° C. 285 g (1.60 mol) of N-bromosuccinimide was charged in separate portions thereto over 1 hour. The mixture was stirred at room temperature for 1 hour and then stirred at 37° C. for 2 hours. The mixture was discharged to 2000 ml of water, extracted with 2000 ml of ethyl acetate, and washed with 1000 ml of saturated brine. After dried over anhydrous magnesium sulfate, the solvent was evaporated under reduced pressure. The obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=20:1) to prepare 304 g (yield 90%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 4.88 (2H, broad-s), 7.59 (2H, s).

<2-3>

Preparation of 2-chloro-N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-3-nitrobenzamide

According to the method of 1-3 of Example 1, a target compound was prepared from 2,6-dibromo-4-(perfluoropropan-2-yl)aniline.

¹H-NMR (CDCl₃, ppm) δ 7.58 (1H, t, J=7.8 Hz), 7.66 (1H, broad-s), 7.90 (2H, s), 7.93 (1H, dd, J=1.5, 7.8 Hz), 7.98 (1H, d, J=7.8 Hz).

<2-4>

Preparation of N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide

According to the method of 1-4 of Example 1, a target compound was prepared from 2-chloro-N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 7.51-7.55 (1H, m), 7.90 (2H, s), 8.16 (1H, d, J=11.7 Hz), 8.27-8.31 (1H, m), 8.48 (1H, t, J=6.3 Hz).

<2-5>

Preparation of 3-amino-N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.93 (2H, broad-s), 6.99-7.04 (1H, m), 7.11 (1H, t, J=7.8 Hz), 7.47-7.49 (1H, m), 7.91 (1H, s), 8.14 (1H, s), 8.28 (1H, d, J=14.6 Hz).

<2-6>

Preparation of 2-chloro-N-(3-(2,6-dibromo-4-(perfluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)nicotinamide (Compound No. 6-1140)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-N-(2,6-dibromo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide and 2-chloronicotinic acid chloride.

¹H-NMR (CDCl₃, ppm) δ 7.40-7.49 (2H, m), 7.89 (2H, s), 7.94-7.96 (1H, m), 8.13 (1H, d, J=12.7 Hz), 8.32-8.34 (1H, m), 8.57-8.59 (1H, m), 8.67-8.71 (1H, m), 8.75 (1H, broad-s).

Example 3

Preparation of 3-benzamide-2-fluoro-N-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)benzamide (Compound No. 6-2110)

<3-1>

Preparation of 2,6-diiodo-4-(perfluoropropan-2-yl)aniline

To a solution of 5.74 g (22.0 mmol) of 4-(perfluoropropan-2-yl)aniline obtained in 2-1 of Example 2 in 50 ml of ethanol was added 2.16 g (22.0 mmol) of concentrated sulfuric acid at 5° C. The reaction mixture was warmed to room temperature, and 10.0 g (44.0 mmol) of N-iodosuccinimide was added thereto, followed by stirring for 3 hours. The reaction mixture was neutralized with a saturated aqueous sodium hydrogen carbonate solution. The precipitated crystals were filtered, washed with water, and then dried to prepare 9.00 g (yield 80%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 4.95 (2H, broad-s), 7.79 (2H, s).

<3-2>

Preparation of 2-chloro-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-3-nitrobenzamide

To a solution of 40.0 g (78.0 mmol) of 2,6-diiodo-4-(perfluoropropan-2-yl)aniline in 100 ml of DMI was added 20.6 g (94.0 mmol) of 2-chloro-3-nitrobenzoyl chloride, followed by stirring at 135° C. for 3 hours. After cooling to room temperature, the reaction mixture was poured into 1000 ml of water. After extraction with the addition of 1000 ml of ethyl acetate, the organic layer was washed with water and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was washed with hexane to prepare 56.2 g (yield 99%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.58 (1H, t, J=8.3 Hz), 7.70 (1H, d, J=3.4 Hz), 7.93 (1H, dd, J=1.5, 6.3 Hz), 8.08-8.10 (1H, m), 8.13 (2H, s).

<3-3>

Preparation of N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide

According to the method of 1-4 of Example 1, a target compound was prepared from 2-chloro-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-3-nitrobenzamide.

1H-NMR (CDCl3, ppm) δ 7.52-7.55 (1H, m), 8.12-8.18 (3H, m), 8.29-8.32 (1H, m), 8.48-8.51 (1H, m).

<3-4>

Preparation of 3-amino-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.93 (2H, broad-s), 6.99-7.04 (1H, m), 7.08 (1H, t, J=7.8 Hz), 7.39-7.43 (1H, m), 8.10 (2H, s), 8.72 (1H, d, J=11.2 Hz).

<3-5>

Preparation of 3-benzamide-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide (Compound No. 6-1260)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide.

¹H-NMR (CDCl₃, ppm) δ 7.39 (1H, t, J=7.8 Hz), 7.52-7.57 (4H, m), 7.60-7.63 (2H, m), 7.93-7.94 (4H, m), 8.70 (1H, t, J=6.3 Hz).

<3-6>

Preparation of 3-benzamide-2-fluoro-N-(4-(perfluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)benzamide (Compound No. 6-2110)

A solution of 1.95 g (2.59 mmol) of 3-benzamide-N-(2,6-diiodo-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide, 0.10 g (0.520 mmol) of copper iodide, and 1.24 g (6.48 mmol) of methyl fluorosulfonyl difluoroacetate in 50 ml of DMF was stirred at 100° C. for 6 hours. The reaction mixture was cooled to room temperature, and then 10 ml of water and 100 ml of ethyl acetate were added thereto, followed by filtration through Celite. The organic layer of the liquid was washed with water and a saturated aqueous sodium hydrogen carbonate solution, and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=1:1). The obtained solid was washed with hexane to prepare 0.840 g (yield 51%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.36-7.40 (1H, m), 7.53-7.64 (3H, m), 7.84-7.97 (1H, m), 7.92-7.94 (2H, m), 8.04-8.07 (1H, m), 8.08-8.13 (1H, m), 8.20 (2H, s), 8.68-8.72 (1H, m).

Example 4

Preparation of N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide (Compound No. 7-1182)

<4-1>

Preparation of 4-(perfluorobutan-2-yl)aniline

4.90 g (52.6 mmol) of aniline, 10.1 g (58.0 mmol) of 85% sodium hydrosulfite, and 1.90 g (5.77 mmol) of tetrabutylammonium hydrogen sulfate were charged to a mixed solution of 150 ml of t-butyl methyl ether and 150 ml of water using a light-shielded reaction vessel, and 4.84 g (57.6 mmol) of sodium hydrogen carbonate was added thereto. 20.0 g (57.8 mmol) of nonafluoro-s-butyliodide was added dropwise thereto at room temperature, followed by stirring at room temperature for 5 hours. The organic phase was collected by separation, washed with 2 mol/L of an aqueous hydrochloric acid solution twice, and then washed with saturated brine, an aqueous sodium hydrogen carbonate solution, and saturated brine. The organic layer was dried over anhydrous magnesium sulfate, and then the solvent was evaporated under reduced pressure to prepare 8.32 g (yield 51%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 3.92 (2H, broad-s), 6.72 (2H, d, J=8.8 Hz), 7.34 (2H, d, J=8.8 Hz).

<4-2>

Preparation of 2,6-dibromo-4-(perfluorobutan-2-yl)aniline

According to the method of 2-2 of Example 2, a target compound was prepared from 4-(perfluorobutan-2-yl)aniline.

¹H-NMR (CDCl₃, ppm) δ 4.89 (2H, broad-s), 7.57 (2H, s).

<4-3>

Preparation of 2-chloro-N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-3-nitrobenzamide

To 27 ml of DMI were added 9.90 g (21.1 mmol) of 2,6-dibromo-4-(perfluorobutan-2-yl)aniline and 4.60 g (20.9 mmol) of 2-chloro-3-nitrobenzoyl chloride, followed by stirring at 140° C. for 4 hours. To the reaction solution were added water and ethyl acetate, and the organic phase was extracted, and washed with 1 mol/L of an aqueous sodium hydroxide solution, saturated brine, and dried over anhydrous magnesium sulfate. Then, the solvent was evaporated under reduced pressure. The obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=20:1→10:1→5:1→3:1) to prepare 5.44 g (yield 40%) of a target compound.

¹H-NMR (CDCl3, ppm) δ 7.52-7.61 (2H, m), 7.89 (2H, s), 7.94 (1H, dd, J=1.5, 8.3 Hz), 7.99 (1H, d, J=7.8 Hz).

<4-4>

Preparation of N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide

To 108 ml of DMSO were added 5.44 g (8.34 mmol) of 2-chloro-N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-3-nitrobenzamide and 4.90 g (84.3 mmol) of potassium fluoride (spray-dried product), followed by stirring at 145° C. for 2 hours. The reaction solution was poured into ice-water to precipitate the crystal, and the obtained crystals were filtered and washed with hexane. The obtained crystals were purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=5:1) to prepare 2.42 g (yield 46%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.53-7.54 (1H, m), 7.89 (2H, s), 8.17 (1H, d, J=12.2 Hz), 8.29-8.30 (1H, m), 8.48-8.49 (1H, m).

<4-5>

Preparation of 3-amino-N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.92 (2H, broad-s), 6.99-7.04 (1H, m), 7.11-7.12 (1H, m), 7.48-7.52 (1H, m), 7.86 (2H, s), 8.22 (1H, d, J=14.1 Hz).

<4-6>

Preparation of N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(methylamino)benzamide

According to the method of 1-6 of Example 1, a target compound was prepared from 3-amino-N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluorobenzamide.

¹H-NMR (CDCl₃, ppm) δ 2.95 (3H, s), 4.14 (1H, broad-s), 6.91-6.92 (1H, m), 7.17-7.21 (1H, m), 7.39-7.43 (1H, m), 7.85 (2H, s), 8.21 (1H, d, J=14.1 Hz).

<4-7>

Preparation of N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide (Compound No. 7-1182)

According to the method of 1-7 of Example 1, a target compound was prepared from N-(2,6-dibromo-4-(perfluorobutan-2-yl)phenyl)-2-fluoro-3-(methylamino)benzamide.

¹H-NMR (CDCl₃, ppm) δ 3.51 (3H, s), 7.22-7.44 (7H, m), 7.85 (2H, s), 8.00-8.03 (2H, m).

Example 5

Preparation of N-(2-bromo-6-(perfluoroethyl)-4-(perfluoropropan-2-yl)phenyl)-3-(4-cyanobenzamide)-2-fluorobenzamide (Compound No. 6-5911)

5-1>

Preparation of 2-(perfluoroethyl)-4-(perfluoropropan-2-yl)aniline

According to the method of 1-1 of Example 1, a target compound was prepared from 4-(perfluoropropan-2-yl)aniline obtained in Example 2-1 and 1,1,2,2,2-pentafluoroethyliodide.

¹H-NMR (CDCl₃, ppm) δ 4.56 (2H, broad-s), 6.79 (1H, d, J=8.8 Hz), 7.47 (1H, d, J=8.8 Hz), 7.53 (1H, s).

<5-2>

Preparation of 2-bromo-6-(perfluoroethyl)-4-(perfluoropropan-2-yl)aniline

According to the method of 1-2 of Example 1, a target compound was prepared from 2-(perfluoroethyl)-4-(perfluoropropan-2-yl)aniline.

¹H-NMR (CDCl₃, ppm) δ 5.14 (2H, broad-s), 7.58 (1H, s), 7.81 (1H, s).

<5-3>

Preparation of N-(2-bromo-6-(perfluoroethyl)-4-(perfluoropropan-2-yl)phenyl)-2-chloro-3-nitrobenzamide

According to the method of 4-3 of Example 4, a target compound was prepared from 2-bromo-6-(perfluoroethyl)-4-(perfluoropropan-2-yl)aniline.

¹H-NMR (CDCl₃, ppm) δ 7.56-7.61 (1H, m), 7.73 (1H, s), 7.88 (1H, d, J=1.5 Hz), 7.92-7.98 (2H, m), 8.21 (1H, s).

<5-4>

Preparation of N-(2-bromo-6-(perfluoroethyl)-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide

According to the method of 1-4 of Example 1, a target compound was prepared from N-(2-bromo-6-(perfluoroethyl)-4-(perfluoropropan-2-yl)phenyl)-2-chloro-3-nitrobenzamide.

APCI-MS m/z (M+1):626

<5-5>

Preparation of 3-amino-N-(2-bromo-6-(perfluoroethyl)-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2-bromo-6-(perfluoroethyl)-4-(perfluoropropan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.92 (2H, broad-s), 6.99-7.04 (1H, m), 7.05-7.18 (1H, m), 7.46-7.51 (1H, m), 7.85 (1H, broad-s), 8.17 (1H, broad-s), 8.34 (1H, d, J=15.1 Hz).

<5-6>

Preparation of N-(2-bromo-6-(perfluoroethyl)-4-(perfluoropropan-2-yl)phenyl)-3-(4-cyanobenzamide)-2-fluorobenzamide (Compound No. 6-5911)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-N-(2-bromo-6-(perfluoroethyl)-4-(perfluoropropan-2-yl)phenyl)-2-fluorobenzamide and 4-cyanobenzoylchloride.

¹H-NMR (CDCl₃, ppm) δ 7.41 (1H, t, J=8.3 Hz), 7.84-7.87 (3H, m), 7.91-7.95 (1H, m), 8.03-8.05 (2H, m), 8.10 (1H, broad-s), 8.17-8.20 (2H, m), 8.63-8.67 (1H, m).

Example 6

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-6-(N-methylbenzamide)picolinamide (Compound No. 17-1103)

<6-1>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-6-chloropicoline amide

According to the method of 1-3 of Example 1, a target compound was prepared from 2-chloropyridine-6-carboxylic acid chloride prepared from 2-chloropyridine-6-carboxylic acid and thionyl chloride, and 2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline obtained in 1-2 of Example 1.

¹H-NMR (CDCl₃, ppm) δ 7.59 (1H, d, J=7.3 Hz), 7.90-7.93 (2H, m), 8.14 (1H, s), 8.20-8.24 (1H, m), 9.60 (1H, s).

<6-2>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-6-(methylamino)picolinamide

To a solution of 0.100 g (0.180 mmol) of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-6-chloropicoline amide in 5 ml of 1,4-dioxane were added 0.00600 g (0.0360 mmol) of copper sulfate and 0.140 g (1.80 mmol) of a 40% aqueous methylamine solution, followed by stirring at an oil bath temperature 80° C. for 3 hours under an enclosed condition. The reaction liquid was returned to room temperature and opened, and water and ethyl acetate were added thereto. The organic layer was washed with water and saturated brine, and dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=2:1) to prepare 0.0700 g (yield 69%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 2.64 (3H, s), 3.79 (1H, broad-s), 7.56-7.60 (1H, m), 7.87-7.93 (2H, m), 8.14-8.15 (1H, m), 8.20-8.23 (1H, m), 9.60 (1H, s).

<6-3>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-6-(N-methylbenzamide)picolinamide (Compound No. 17-1103)

According to the method of 1-7 of Example 1, a target compound was prepared from N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-6-(methylamino)picolinamide.

¹H-NMR (CDCl₃, ppm) δ 3.65 (3H, s), 7.28-7.41 (6H, m), 7.77 (1H, t, J=7.8 Hz), 7.91 (1H, s), 8.00-8.02 (1H, m), 8.14 (1H, s), 9.39 (1H, s).

Example 7

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-(2-fluoro-N-methylbenzamide)thiazole-4-carboxamide (Compound No. 27-628)

<7-1>

Preparation of 2-aminothiazole-4-carboxylic acid

To 40 ml of an aqueous solution of 4.00 g (23.2 mmol) of ethyl 2-aminothiazole-4-carboxylate was added 1.86 g (46.5 mmol) of sodium hydroxide, followed by stirring at room temperature for 5 hours. The reaction liquid was adjusted to pH 1 by the addition of concentrated hydrochloric acid, and the precipitated crystals were collected by filtration to prepare 2.84 g (yield 85%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.18 (2H, broad-s), 7.38 (1H, s).

The proton of the carboxylic acid was not detected.

<7-2>

Preparation of 2-chlorothiazole-4-carboxylic acid

To a solution of 2.84 g (19.7 mmol) of 2-aminothiazole-4-carboxylic acid in 30 ml of 1,4-dioxane was added 50 ml of concentrated hydrochloric acid, followed by cooling to 0° C., and 10 ml of an aqueous solution of 2.04 g (29.6 mmol) of sodium nitrite was added charged dropwise thereto at 0° C. to 5° C. The reaction liquid was stirred at 0° C. for 2 hours, and then 2.93 g (29.6 mmol) of copper chloride was charged in separate portions thereto. The reaction liquid was returned to room temperature, followed by stirring for 8 hours. To the reaction liquid were added water and ethyl acetate, followed by extraction with ethyl acetate four times. The organic layer was washed with saturated brine, and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure to prepare 1.77 g (yield 55%) of a target compound.

¹H-NMR (DMSO-d₆, ppm) δ 8.41 (1H, s).

The proton of the carboxylic acid was not detected.

<7-3>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-chlorothiazole-4-carboxamide

According to the method of 4-3 of Example 4, a target compound was prepared from 2-chlorothiazole-4-carbonylchloride prepared from 2-chlorothiazole-4-carboxylic acid and thionyl chloride, and 2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline obtained in 1-2 of Example 1.

¹H-NMR (CDCl₃, ppm) δ 7.91 (1H, s), 8.13 (1H, s), 8.19 (1H, s), 8.82 (1H, s).

<7-4>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-(methylamino)thiazole-4-carboxamide

According to the method of 6-2 of Example 6, a target compound was prepared from N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-chlorothiazole-4-carboxamide.

¹H-NMR (CDCl₃, ppm) δ 3.03 (3H, s), 5.11-5.12 (1H, m), 7.50 (1H, s), 7.88 (1H, s), 8.11 (1H, s), 8.99 (1H, s).

<7-5>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-(2-fluoro-N-methylbenzamide)thiazole-4-carboxamide (Compound No. 27-628)

According to the method of 1-7 of Example 1, a target compound was prepared from N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-(methylamino)thiazole-4-carboxamide and 2-fluorobenzoyl chloride.

¹H-NMR (CDCl₃, ppm) δ 3.67 (3H, s), 6.99-7.24 (1H, m), 7.29-7.35 (1H, m), 7.52-7.59 (2H, m), 7.90 (1H, s), 8.06 (1H, s), 8.14 (1H, s), 9.08 (1H, s).

Example 8

Preparation of 2,2,2-trichloroethyl 2-fluoro-3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl(methyl)carbamate (Compound No. 12-864)

<8-1>

Preparation of 4-(perfluorobutan-2-yl)-2-(trifluoromethyl)aniline

According to the method of 1-1 of Example 1, a target compound was prepared from 2-(trifluoromethyl)aniline and nonafluoro-s-butyliodide under the light-shielding reaction condition.

¹H-NMR (CDCl₃, ppm) δ 4.49 (2H, broad-s), 6.81 (1H, d, J=8.8 Hz), 7.47 (1H, d, J=8.8 Hz), 7.61 (1H, s).

<8-2>

Preparation of 2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)aniline

To 100 mL of ethanol was added 17.0 g (44.8 mmol) of 4-(perfluorobutan-2-yl)-2-(trifluoromethyl)aniline, and 5.28 g (53.8 mmol) of concentrated sulfuric acid and 12.6 g (55.8 mmol) of N-iodosuccinimide were added thereto under ice-cooling, followed by stirring at room temperature for 1 hour and 30 minutes and at 40° C. for 4 hours. To the reaction solution was added a 4 M aqueous sodium hydroxide solution to neutralize the reaction solution, and then ethyl acetate was added thereto to extract the organic phase. The organic phase was washed with saturated brine, and dried over anhydrous magnesium sulfate, and then the solvent was evaporated under reduced pressure. The obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=10:1) to prepare 14.6 g (yield 65%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 5.04 (2H, broad-s), 7.62 (1H, s), 7.97 (1H, s).

<8-3>

Preparation of 2-chloro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide

According to the method of 4-3 of Example 4, a target compound was prepared from 2-iodo-4-(perfluorobutan-2-yl)-6-(trifluormethyl)aniline.

¹H-NMR (CDCl₃, ppm) δ 7.60-7.61 (1H, m), 7.77 (1H, s), 7.89-7.96 (2H, m), 8.03-8.04 (1H, m), 8.38 (1H, s).

<8-4>

Preparation of 2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide

According to the method of 1-4 of Example 1, a target compound was prepared from 2-chloro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 7.53-7.54 (1H, m), 7.95 (1H, s), 8.24-8.32 (2H, m), 8.36 (1H, s), 8.44-8.48 (1H, m).

<8-5>

Preparation of 3-amino-2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide

According to the method of 1-5 of Example 1, a target compound was prepared from 2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.93 (2H, broad-s), 7.02-7.03 (1H, m), 7.11-7.13 (1H, m), 7.47-7.51 (1H, m), 7.92 (1H, s), 8.31-8.34 (2H, m).

<8-6>

Preparation of 2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(methylamino)benzamide

According to the method of 1-6 of Example 1, a target compound was prepared from 3-amino-2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)benzamide.

¹H-NMR (CDCl₃, ppm) δ 2.95-2.96 (3H, m), 4.15 (1H, broad-s), 6.91-6.93 (1H, m), 7.19-7.20 (1H, m), 7.38-7.42 (1H, m), 7.92 (1H, s), 8.32 (1H, d, J=14.1 Hz), 8.34 (1H, s).

<8-7>

Preparation of 2,2,2-trichloroethyl 2-fluoro-3-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl(methyl)carbamate (Compound No. 12-864)

According to the method of 1-7 of Example 1, a target compound was prepared from 2-fluoro-N-(2-iodo-4-(perfluorobutan-2-yl)-6-(trifluoromethyl)phenyl)-3-(methylamino)benzamide and 2,2,2-trichloroethoxycarbonylchloride.

¹H-NMR (CDCl₃, ppm) δ 3.40 (3H, s), 4.74 (2H, broad-s), 7.37 (1H, t, J=7.8 Hz), 7.52-7.58 (1H, m), 7.93 (1H, s), 8.12-8.15 (1H, m), 8.28-8.34 (2H, m).

Example 9

Preparation of N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyano-3-(4-cyano-N-methylbenzamide)benzamide (Compound No. 2-491)

<9-1>

Preparation of 2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline

According to the method of 1-2 of Example 1, a target compound was prepared from 4-(perfluoropropan-2-yl)-2-(trifluoromethyl)aniline obtained in 1-1 of Example 1 and N-chlorosuccinimide.

¹H-NMR (CDCl₃, ppm) δ 4.97 (2H, broad-s), 7.57 (1H, s), 7.64 (1H, s).

<9-2>

Preparation of N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-iodo-3-nitrobenzamide

According to the method of 1-3 of Example 1, a target compound was prepared from 4-iodo-3-nitrobenzoyl chloride prepared from 4-iodo-3-nitrobenzoic acid and thionyl chloride, and 2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline.

¹H-NMR (CDCl₃, ppm) δ 7.52-7.81 (2H, m), 7.89 (1H, s), 8.00 (1H, s), 8.25 (1H, d, J=8.3 Hz), 8.38 (1H, d, J=1.9 Hz).

<9-3>

Preparation of 3-amino-N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-iodobenzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-iodo-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 4.35 (2H, s), 6.92 (1H, dd, J=1.9, 8.3 Hz), 7.29 (1H, d, J=1.9 Hz), 7.60 (1H, s), 7.79 (1H, d, J=8.3 Hz), 7.86 (1H, s), 7.97 (1H, s).

<9-4>

Preparation of N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-iodo-3-(methylamino)benzamide

According to the method of 1-6 of Example 1, a target compound was prepared from 3-amino-N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-iodobenzamide.

¹H-NMR (CDCl₃, ppm) δ 2.97 (3H, s), 4.46 (1H, broad-s), 6.89 (1H, dd, J=1.9, 8.3 Hz), 7.07 (1H, d, J=1.9 Hz), 7.65 (1H, s), 7.80 (1H, d, J=8.3 Hz), 7.86 (1H, s), 7.97 (1H, s).

<9-5>

Preparation of N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyano-3-(methylamino)benzamide

To 10 mL of DMF were added 0.350 g (0.560 mmol) of N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-iodo-3-(methylamino)benzamide and 0.200 g (2.25 mmol) of copper (I) cyanide, followed by stirring at 140° C. for 1 hour and 30 minutes. A saturated aqueous sodium thiosulfate solution was poured into the reaction solution to quench the reaction, and the organic layer was collected with ethyl acetate and washed with saturated brine. The organic layer was dried over anhydrous magnesium sulfate, and then the solvent was evaporated under reduced pressure. The obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=5:1→3:1) to prepare 0.250 g (yield 86%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 3.01 (1/2*3H, s), 3.03 (1/2*3H, s), 4.89 (1/2*1H, s), 4.90 (1/2*1H, s), 7.80 (1H, dd, J=1.5, 8.3 Hz), 7.21-7.22 (1H, m), 7.54 (1H, d, J=8.3 Hz), 7.67 (1H, s), 7.88 (1H, s), 7.99 (1H, s).

<9-6>

Preparation of N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyano-3-(4-cyano-N-methylbenzamide)benzamide (Compound No. 2-491)

According to the method of 1-7 of Example 1, a target compound was prepared from N-(2-chloro-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyano-3-(methylamino)benzamide and 4-cyanobenzoylchloride.

¹H-NMR (CDCl3, ppm) δ 3.81 (3H, broad-s), 7.52-7.84 (8H, m), 7.89 (1H, s), 8.00 (1H, s).

Example 10

Preparation of N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-6-cyano-2-fluorophenyl)-6-chloronicotinamide (Compound No. 1-1968)

<10-1>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyano-2,3-difluorobenzamide

To a solution of 0.840 g (4.59 mmol) of 4-cyano-2,3-difluorobenzoic acid in 10 ml of dichloromethane were added one drop of DMF and 0.470 ml (5.51 mmol) of oxalyl chloride, followed by stirring at room temperature for 1 hour. The solvent was evaporated under reduced pressure and the obtained 4-cyano-2,3-difluorobenzoyl chloride was added to a solution of 1.56 g (3.83 mmol) of 2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline obtained in 1-2 of Example 1 in 5 ml of DMI, followed by stirring at 130° C. for 5 hours. To the reaction liquid were added water and ethyl acetate, and the organic layer was washed with a saturated aqueous sodium hydrogen carbonate solution and saturated brine, and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=1:0-+10:1) to prepare 0.58 g (yield 27%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.52-7.62 (1H, m), 7.92-7.94 (1H, m), 8.02-8.06 (1H, m), 8.13-8.16 (2H, m).

<10-2>

Preparation of 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyano-2-fluorobenzamide

To a solution of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyano-2,3-difluorobenzamide in 5 ml of DMSO was added 49.0 mg of ammonium carbonate, followed by stirring 100° C. for 5 hours. To the reaction liquid were added water and ethyl acetate, and the organic layer was washed with water, and then and dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=8:1→4:1) to prepare 0.30 g (yield 51%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 4.71 (2H, broad-s), 7.35-7.39 (1H, m), 7.40-7.44 (1H, m), 7.92 (1H, s), 8.12-8.15 (2H, m).

<10-3>

Preparation of N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-6-cyano-2-fluorophenyl)-6-chloronicotinamide (Compound No. 1-1968)

To a solution of 0.0500 g (0.0877 mol) of 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyano-2-fluorobenzamide in 0.200 ml of DMI was added 0.0308 g (0.175 mmol) of 6-chloronicotinoylchloride, followed by stirring at 130° C. for 6 hours. To the reaction liquid were added water and ethyl acetate, and the organic layer was washed with 1 M hydrochloric acid, a saturated aqueous sodium hydrogen carbonate solution, and saturated brine, and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=2:1) to prepare 0.0100 g (yield 16%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.54 (1H, d, J=8.8 Hz), 7.72 (1H, d, J=8.8 Hz), 7.93 (1H, s), 8.09 (1H, s), 8.17-8.18 (2H, m), 8.27 (1H, dd, J=2.4 Hz 8.8 Hz), 8.38 (1H, d, J=10.8 Hz), 8.98 (1H, d, J=2.4 Hz).

Example 11

Preparation of 3-(4-cyanobenzamide)-N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)benzamide (Compound No. 6-79)

<11-1>

Preparation of 2,6-diiodo-4-(perfluorobutan-2-yl)aniline

According to the method of 3-1 of Example 3, a target compound was prepared from 4-(perfluorobutan-2-yl)aniline obtained in 4-1 of Example 4.

¹H-NMR (CDCl₃, ppm) δ 4.95 (2H, broad-s), 7.78 (2H, s).

<11-2>

Preparation of N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-3-nitrobenzamide

According to the method of 4-3 of Example 4, a target compound was prepared from 2,6-diiodo-4-(perfluorobutan-2-yl)aniline and 3-nitrobenzoyl chloride.

¹H-NMR (CDCl₃, ppm) δ 7.74 (1H, t, J=8.0 Hz), 8.11 (2H, s), 8.42 (1H, d, J=7.6 Hz), 8.46 (1H, d, J=8.4 Hz), 8.90 (1H, d, J=12.4 Hz), 8.92 (1H, s).

<11-3>

Preparation of 3-amino-N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)benzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 5.39 (2H, broad-s), 6.89-6.93 (1H, m), 7.29-7.31 (3H, m), 7.68 (1H, s), 8.08 (2H, s).

<11-4>

Preparation of 3-(4-cyanobenzamide)-N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)benzamide (Compound No. 6-79)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-N-(2,6-diiodo-4-(perfluorobutan-2-yl)phenyl)benzamide and 4-cyanobenzoylchloride.

¹H-NMR (CDCl₃, ppm) δ 7.58 (1H, t, J=8.2 Hz), 7.79-7.83 (3H, m), 7.97 (2H, s), 8.01 (2H, d, J=8.0 Hz), 8.09 (2H, s), 8.18 (1H, s), 8.29 (1H, s).

Example 12

Preparation of N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)phenylcarbamoyl)-2-fluorophenyl)-2-chloronicotinamide (Compound No. 6-5908)

<12-1>

Preparation of 4-(perfluoropropan-2-yl)-2-(trifluoromethoxy)aniline

According to the method of 1-1 of Example 1, a target compound was prepared from 2-trifluoromethoxy aniline.

¹H-NMR (CDCl₃, ppm) δ 4.19 (2H, broad-s), 6.86 (1H, d, J=8.8 Hz), 7.30 (1H, d, J=8.8 Hz), 7.36 (1H, s).

<12-2>

Preparation of 2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)aniline

According to the method of 1-2 of Example 1, a target compound was prepared from 4-(perfluoropropan-2-yl)-2-(trifluoromethoxy)aniline.

¹H-NMR (CDCl₃, ppm) δ 4.65 (2H, broad-s), 7.33 (1H, s), 7.71 (1H, s).

<12-3>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)phenyl)-2-chloro-3-nitrobenzamide

According to the method of 1-3 of Example 1, a target compound was prepared from 2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)aniline.

¹H-NMR (CDCl₃, ppm) δ 7.49-7.61 (3H, m), 7.80-7.96 (3H, m).

<12-4>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)phenyl)-2-fluoro-3-nitrobenzamide

According to the method of 1-4 of Example 1, a target compound was prepared from N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)phenyl)-2-chloro-3-nitrobenzamide.

¹H-NMR (CDCl3, ppm) δ 7.53 (1H, t, J=7.8 Hz), 7.60 (1H, broad-s), 7.89 (1H, d, J=1.5 Hz), 8.07 (1H, broad-d, J=12.7 Hz), 8.29-8.30 (1H, m), 8.43-8.47 (1H, m).

<12-5>

Preparation of 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)phenyl)-2-fluorobenzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.92 (2H, broad-s), 6.99-7.04 (1H, m), 7.11 (1H, t, J=7.8 Hz), 7.45-7.49 (1H, m), 7.57 (1H, broad-s), 7.87 (1H, d, J=2.0 Hz), 8.14 (1H, d, J=14.2 Hz).

<12-6>

Preparation of N-(3-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)phenylcarbamoyl)-2-fluorophenyl)-2-chloronicotinamide (Compound No. 6-5908)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethoxy)phenyl)-2-fluorobenzamide and 2-chloronicotinoylchloride.

¹H-NMR (CDCl₃, ppm) δ 7.39-7.49 (2H, m), 7.59 (1H, s), 7.88-7.94 (2H, m), 8.07 (1H, d, J=12.2 Hz), 8.31-8.33 (1H, m), 8.57-8.58 (1H, m), 8.60-8.70 (1H, m), 8.74 (1H, broad-s).

Example 13

Preparation of 3-benzamide-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-fluorobenzamide (Compound No. 6-3348)

<13-1>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-fluoro-3-nitrobenzamide

According to the method of 1-3 of Example 1, a target compound was prepared from 4-fluoro-3-nitrobenzoyl chloride prepared from 4-fluoro-3-nitrobenzoic acid and thionyl chloride, and 2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline obtained in 1-2 of Example 1.

¹H-NMR (CDCl₃, ppm) δ 7.47-7.50 (1H, m), 7.92 (2H, d, J=5.9 Hz), 8.16 (1H, s), 8.23-8.28 (1H, m), 8.65-8.67 (1H, m).

<13-2>

Preparation of 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-fluorobenzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-fluoro-3-nitrobenzamide.

APCI-MS m/z (M+1): 546

<13-3>

Preparation of 3-benzamide-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-fluorobenzamide (Compound No. 6-3348)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-fluorobenzamide.

¹H-NMR (CDCl₃, ppm) δ 7.29-7.34 (1H, m), 7.53-7.65 (3H, m), 7.80-7.84 (1H, m), 7.90-7.92 (3H, m), 8.14 (1H, broad-s), 8.20 (1H, d, J=2.9 Hz), 8.25 (1H, broad-s), 9.10 (1H, dd, J=1.9, 7.3 Hz).

Example 14

Preparation of 2-chloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide (Compound No. 6-460)

<14-1>

Preparation of 2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline

According to the method of 8-2 of Example 8, a target compound was prepared from 4-(perfluoropropan-2-yl)-2-(trifluoromethyl)aniline obtained in 1-1 of Example 1 and N-iodosuccinimide.

¹H-NMR (CDCl₃, ppm) δ 5.04 (2H, broad-s), 7.64 (1H, s), 7.99 (1H, s).

<14-2>

Preparation of N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide

According to the method of 4-3 of Example 4, a target compound was prepared from 2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline and 3-nitrobenzoyl chloride.

¹H-NMR (CDCl₃, ppm) δ 7.76-7.80 (2H, m), 7.97 (1H, s), 8.28, 8.30 (1H, m), 8.37 (1H, s), 8.49-8.52 (1H, m), 8.78 (1H, s).

<14-3>

Preparation of 3-amino-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl3, ppm) δ 3.89 (2H, broad-s), 6.89-6.92 (1H, m), 7.23-7.32 (3H, m), 7.68 (1H, s), 7.93 (1H, s), 8.34-8.36 (1H, m).

<14-4>

Preparation of 2-chloro-N-(3-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)nicotinamide (Compound No. 6-460)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide and 2-chloronicotinoylchloride.

¹H-NMR (CDCl₃, ppm) δ 7.43-7.46 (1H, m), 7.58 (1H, t, J=7.8 Hz), 7.77 (1H, d, J=7.8 Hz), 7.91-7.95 (2H, m), 8.01 (1H, s), 8.24 (1H, dd, J=2.0, 7.8 Hz), 8.28 (1H, s), 8.36 (1H, s), 8.41 (1H, s), 8.54-8.56 (1H, m).

Example 15

Preparation of 2-fluoro-3-(4-fluoro-N-methylbenzamide)-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide (Compound No. 7-1733)

<15-1>

Preparation of 2-chloro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide

According to the method of 4-3 of Example 4, a target compound was prepared from 2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline obtained in 14-1 of Example 14 and 2-chloro-3-nitrobenzoyl chloride.

¹H-NMR (CDCl₃, ppm) δ 7.60 (1H, t, J=7.8 Hz), 7.76 (1H, s), 7.94 (1H, dd, J=1.5, 7.8 Hz), 7.97 (1H, s), 8.03 (1H, dd, J=1.5, 7.8 Hz), 8.39 (11, s).

<15-2>

Preparation of 2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide

According to the method of 1-4 of Example 1, a target compound was prepared from 2-chloro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 7.51-7.55 (1H, m), 7.97 (1H, s), 8.23 (1H, d, J=12.2 Hz), 8.28-8.32 (1H, m), 8.37 (1H, s), 8.44-8.48 (1H, m).

<15-3>

Preparation of 3-amino-2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide

According to the method of 1-5 of Example 1, a target compound was prepared from 2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.92 (2H, broad-s), 7.02-7.04 (1H, m), 7.11 (1H, t, J=7.8 Hz), 7.47-7.52 (1H, m), 7.94 (1H, s), 8.30-8.35 (2H, m).

<15-4>

Preparation of 2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(methylamino)benzamide

According to the method of 1-6 of Example 1, a target compound was prepared from 3-amino-2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide.

¹H-NMR (CDCl₃, ppm) δ 2.95 (3H, s), 4.15 (1H, broad-s), 6.90 (1H, t, J=8.2 Hz), 7.19 (1H, t, J=7.8 Hz), 7.40 (1H, t, J=7.8 Hz), 7.92 (1H, s), 8.30 (1H, s), 8.34 (1H, s).

<15-5>

Preparation of 2-fluoro-3-(4-fluoro-N-methylbenzamide)-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide (Compound No. 7-1733)

According to the method of 1-7 of Example 1, a target compound was prepared from 2-fluoro-N-(2-iodo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(methylamino)benzamide and 4-fluorobenzoyl chloride.

¹H-NMR (CDCl₃, ppm) δ 3.50 (3H, s), 6.91 (2H, s), 6.93-7.35 (3H, m), 7.46 (1H, t, J=7.0 Hz), 7.93 (1H, s), 8.01-8.10 (1H, m), 8.13 (1H, broad-s), 8.34 (1H, s).

Example 16

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-N-methyl-3-(N-methylbenzamide)benzamide (Compound No. 9-2164)

To a solution of 0.100 g (0.150 mmol) of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide obtained in 1-7 of Example 1 in 5 ml of DMF was added 0.00900 g (0.230 mmol) of sodium hydride (60% in oil), followed by stirring at room temperature for 40 minutes. To the reaction liquid was added 0.0300 g (0.180 mmol) of methyl iodide, followed by stirring at the same temperature for 6 hours. To the reaction liquid were added water and ethyl acetate, and the organic layer was washed with water and saturated brine, and dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=4:1) to prepare 0.106 g of a target compound quantitatively.

¹H-NMR (CDCl₃, ppm) δ 2.18-2.19 (3H, m), 3.48 (3H, s), 7.21-7.25 (4H, m), 7.32-7.40 (4H, m), 7.92 (1H, s), 8.13 (1H, s).

Example 17

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-cyanobenzamide)-N-methylbenzamide (Compound No. 8-289)

<17-1>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide

According to the method of 4-3 of Example 4, a target compound was prepared from 2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline obtained in 1-2 of Example 1 and 3-nitrobenzoyl chloride.

¹H-NMR (CDCl₃, ppm) δ 7.75-7.79 (2H, m), 7.94 (1H, s), 8.17 (1H, d, J=1.0 Hz), 8.28 (1H, dd, J=1.5, 7.8 Hz), 8.48-8.51 (1H, m), 8.76-8.77 (1H, m).

<17-2>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-N-methyl-3-nitrobenzamide

According to the method of Example 16, a target compound was prepared from N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.28 (1/2*3H, s), 3.44 (1/2*3H, s), 7.41 (1/2*1H, t, J=7.8 Hz), 7.71-7.76 (2/2*1H, m), 7.84 (1/2*1H, s), 7.93-7.95 (1/2*1H, m), 7.98 (1/2*1H, s), 8.07-8.09 (2/2*1H, m), 8.14-8.16 (1/2*1H, m), 8.19 (1/2*1H, s), 8.39-8.41 (1/2*1H, m), 8.45-8.46 (1/2*1H, m).

<17-3>

Preparation of 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-N-methylbenzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-N-methyl-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.24 (3/4*3H, s), 3.37 (1/4*3H, s), 3.80 (2H, broad-s), 6.47 (1/4*1H, d, J=7.8 Hz), 6.54-6.57 (1/4*1H, m), 6.78-6.84 (5/4*1H, m), 6.86 (3/4*11H, t, J=2.0 Hz), 6.96 (3/4*1H, d, J=7.8 Hz), 7.23-7.27 (3/4*1H, m), 7.79 (1/4*1H, s), 7.94 (3/4*1H, s), 8.00 (1/4*1H, s), 8.15 (3/4*1H, s).

<17-4>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(4-cyanobenzamide)-N-methylbenzamide (Compound No. 8-289)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-N-methylbenzamide and 4-cyanobenzoylchloride.

¹H-NMR (CDCl₃, ppm) δ 3.26 (2/3*3H, s), 3.38 (1/3*3H, s), 7.08-7.09 (1/3*1H, m), 7.12-7.14 (1/3*1H, m), 7.32 (2/3*1H, d, J=7.8 Hz), 7.45-7.49 (3/3*1H, m), 7.72-7.76 (9/3*1H, m), 7.83 (1/3*1H, s), 7.85-7.89 (4/3*1H, m), 7.95 (2/3*1H, s), 7.98-8.00 (4/3*1H, m), 8.04 (2/3*1H, d, J=6.3 Hz), 8.16 (2/3*1H, s), 8.57 (2/3*1H, s).

Example 18

Preparation of 3-benzamide-N-(2-bromo-4-(perfluoroethyl)-6-(trifluoromethyl)phenyl)benzamide (Compound No. 6-5913)

<18-1>

Preparation of 4-(perfluoroethyl)-2-(trifluoromethyl)aniline

To 40 ml of an aqueous solution of 7.04 g (40.4 mmol) of 85% sodium hydrosulfite and 3.40 g (40.4 mmol) of sodium hydrogen carbonate were added 13.6 g (33.7 mmol) of 2-(trifluoromethyl)aniline and 40 ml of DMF. To this reaction liquid was added 50 ml of a solution of 11.2 g (45.5 mmol) of 1,1,2,2,2-pentafluoroethyliodide in DMF (DMF was cooled to −30° C., and 1,1,2,2,2-pentafluoroethyl iodide was dissolved therein), and placed in an autoclave, followed by stirring at 110° C. for 9 hours. After being left to stand at room temperature overnight, water and ethyl acetate were added to the reaction liquid, followed by extraction with ethyl acetate. The organic layer was washed with water, a saturated aqueous sodium hydrogen carbonate solution, and saturated brine. The organic layer was dried over anhydrous sodium sulfate, then the solvent was evaporated under reduced pressure, and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=10:1→5:1) to prepare 1.95 g (yield 21%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 4.53 (2H, broad-s), 6.81 (1H, d, J=8.3 Hz), 7.48 (1H, d, J=8.3 Hz), 7.63 (1H, broad-s).

<18-2>

Preparation of 2-bromo-4-(perfluoroethyl)-6-(trifluoromethyl)aniline

According to the method of 1-2 of Example 1, a target compound was prepared from 4-(perfluoroethyl)-2-(trifluoromethyl)aniline.

¹H-NMR (CDCl₃, ppm) δ 5.08 (2H, broad-s), 7.62 (1H, s), 7.80 (1H, s).

<18-3>

Preparation of N-(2-bromo-4-(perfluoroethyl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide

To a solution of 2.50 g (6.99 mmol) of 2-bromo-4-(perfluoroethyl)-6-(trifluoromethyl)aniline in 20 ml of pyridine was added 2.72 g (14.7 mmol) of 3-nitrobenzoyl chloride, followed by stirring at 100° C. for 12 hours. To the reaction liquid were added water and ethyl acetate, followed by extraction with ethyl acetate. The organic layer was washed with 1 M hydrochloric acid, a saturated aqueous sodium hydrogen carbonate solution, and saturated brine. The organic layer was dried over anhydrous sodium sulfate, and then the solvent was evaporated under reduced pressure. To the obtained residue were added THF and an aqueous sodium hydroxide solution, followed by stirring at room temperature for 8 hours. The reaction liquid was extracted/dried in the same manner as described above, and the solvent was evaporated under reduced pressure. The obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=7:1-5:1) to prepare 0.202 g (yield 6%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.75 (1H, s), 7.78 (1H, t, J=7.8 Hz), 7.94 (1H, s), 8.17 (1H, s), 8.29-8.30 (1H, m), 8.50-8.52 (1H, m), 8.78 (1H, t, J=2.0 Hz).

<18-4>

Preparation of 3-amino-N-(2-bromo-4-(perfluoroethyl)-6-(trifluoromethyl)phenyl)benzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2-bromo-4-(perfluoroethyl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.89 (2H, broad-s), 6.90-6.92 (1H, m), 7.23-7.32 (3H, m), 7.64 (1H, s), 7.90 (1H, s), 8.13 (1H, s).

<18-5>

Preparation of 3-benzamide-N-(2-bromo-4-(perfluoroethyl)-6-(trifluoromethyl)phenyl)benzamide (Compound No. 6-5913)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-N-(2-bromo-4-(perfluoroethyl)-6-(trifluoromethyl)phenyl)benzamide.

¹H-NMR (CDCl₃, ppm) δ 7.51-7.62 (4H, m), 7.72 (1H, dd, J=1.5, 7.8 Hz), 7.89-8.00 (6H, m), 8.14 (1H, s), 8.27 (1H, t, J=2.0 Hz).

Example 19

Preparation of 3-benzamide-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyanobenzamide (Compound No. 1-627)

<19-1>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-fluoro-3-nitrobenzamide

According to the method of 4-3 of Example 4, a target compound was prepared from 4-fluoro-3-nitrobenzoyl chloride prepared from 4-fluoro-3-nitrobenzoic acid and thionyl chloride, and 2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)aniline obtained in 1-2 of Example 1.

¹H-NMR (CDCl₃, ppm) δ 7.47-7.50 (1H, m), 7.92 (2H, d, J=5.9 Hz), 8.16 (1H, s), 8.23-8.28 (1H, m), 8.65-8.67 (1H, m).

<19-2>

Preparation of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyano-3-nitrobenzamide

To a solution of 0.500 g (0.870 mmol) of N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-fluoro-3-nitrobenzamide in 5 ml of DMF was added 0.0639 g (1.31 mmol) of sodium cyanide, followed by stirring at room temperature for 10 hours. To the reaction liquid were added water and ethyl acetate, followed by extraction with ethyl acetate. The organic layer was washed with a 10% aqueous sodium hydroxide solution and saturated brine. The organic layer was dried over anhydrous sodium sulfate, and then the solvent was evaporated under reduced pressure. The obtained residue was purified by silica gel column chromatography to prepare 0.0500 g (yield 10%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.80 (1H, s), 7.96 (1H, s), 8.12-8.14 (1H, m), 8.18 (1H, s), 8.36 (1H, dd, J=2.0, 8.3 Hz), 8.84 (1H, d, J=1.5 Hz).

<19-3>

Preparation of 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyanobenzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyano-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 4.68 (2H, broad-s), 7.18 (1H, dd, J=1.9, 8.3 Hz), 7.29 (1H, s), 7.52-7.55 (1H, m), 7.68 (1H, s), 7.92 (1H, s), 8.14 (1H, d, J=1.5 Hz).

<19-4>

Preparation of 3-benzamide-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyanobenzamide (Compound No. 1-627)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-N-(2-bromo-4-(perfluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-4-cyanobenzamide.

¹H-NMR (CDCl₃, ppm) δ 7.56-7.59 (3H, m), 7.64-7.66 (1H, m), 7.80-7.87 (2H, m), 7.94-7.97 (2H, m), 8.16 (1H, s), 8.46 (1H, s), 8.57 (1H, s), 9.16 (1H, s).

Next, Preparation Examples in which the compound of the present invention is contained as an active ingredient will be shown, but the present invention is not limited thereto. Further, in Preparation Examples, parts represent parts by weight.

Preparation Example 1

20 parts of the compound represented by Formula (1) of the present invention, 10 parts of polyoxyethylene styrylphenyl ether, and 70 parts of xylene were mixed uniformly to obtain an emulsion.

Preparation Example 2

10 parts of the compound represented by Formula (1) of the present invention, 2 parts of sodium lauryl sulfate, 2 parts of dialkyl sulfosuccinate, 1 part of a 0-naphthalene sulfonic acid formalin condensate sodium salt, and 85 parts of diatomaceous earth were stirred and mixed uniformly to obtain a wettable powder.

Preparation Example 3

0.3 parts of the compound represented by Formula (1) of the present invention and 0.3 parts of white carbon were mixed uniformly, and 99.2 parts of clay and 0.2 parts of DRILESS A (manufactured by Sankyo Agro Co., Ltd.) were added thereto, followed by pulverizing and mixing uniformly, thereby obtaining powders.

Preparation Example 4

3 parts of the compound represented by Formula (1) of the present invention, 1.5 parts of a polyoxyethylene/polyoxypropylene condensate, 3 parts of carboxymethyl cellulose, 64.8 parts of clay, and 27.7 parts of talc were pulverized and mixed uniformly, and water was added thereto, followed by kneading, granulating, and drying, thereby obtaining powders.

Preparation Example 5

10 parts of the compound represented by Formula (1) of the present invention, 3 parts of a β-naphthalene sulfonic acid formalin condensate sodium salt, 1 part of tristyrylphenol, 5 parts of propylene glycol, 0.5 parts of a silicon-based defoaming agent, and 33.5 parts of water were sufficiently stirred and mixed, and then 0.3 parts of xanthan gum and 46.7 parts of water were mixed therewith, followed by stirring and mixing again, thereby obtaining a flowable Formulation.

Preparation Example 6

20 parts of the compound represented by Formula (1) of the present invention, 6 parts of a naphthalene sulfonic acid formaldehyde condensate metal salt, 1 part of dialkylsulfosuccinate metal salt, and 73 parts of calcium carbonate were pulverized and mixed uniformly, and water was added thereto, followed by kneading, granulating, and drying, thereby obtaining a granule wettable powder.

For the use of Formulations obtained above, Formulation was diluted to 1-fold to 10000-fold with water or was not diluted, and then directly sprayed.

Next, the usefulness of the compound of the present invention as a pest control agent will be described specifically with reference to the following Test Examples, but the present invention is not limited thereto.

Test Example 1

Pesticidal Test Against Spodoptera litura

A piece of a cabbage leaf was immersed for 30 seconds in a chemical solution in which a test compound had been prepared at a predetermined concentration, and air-dried, and then put into a 7 cm polyethylene cup having a filter paper laid on the bottom thereof, and 2-stage larvae of Spodoptera litura were released. They were left to stand in a thermostatic chamber at 25° C., and the numbers of the living pests and the dead pests were examined after 6 days. The test was carried out with five larvae per group in two replicates.

Further, the following compound (A) disclosed in the pamphlet of International Publication WO 2005/073165 was used as a comparative compound.

As the results of the above tests, the compounds of Compound Nos. 1-470, 1-491, 1-513, 1-627, 1-1925, 2-491, 6-38, 6-39, 6-45, 6-46, 6-47, 6-57, 6-60, 6-71, 6-72, 6-78, 6-79, 6-80, 6-90, 6-93, 6-111, 6-147, 6-268, 6-269, 6-270, 6-271, 6-272, 6-288, 6-289, 6-290, 6-293, 6-300, 6-304, 6-306, 6-311, 6-346, 6-347, 6-348, 6-349, 6-366, 6-367, 6-368, 6-382, 6-389, 6-424, 6-425, 6-426, 6-427, 6-428, 6-444, 6-445, 6-446, 6-448, 6-449, 6-450, 6-452, 6-453, 6-460, 6-461, 6-467, 6-502, 6-503, 6-504, 6-505, 6-522, 6-523, 6-524, 6-538, 6-545, 6-804, 6-824, 6-825, 6-840, 6-1104, 6-1105, 6-1106, 6-1107, 6-1124, 6-1125, 6-1126, 6-1140, 6-1147, 6-1182, 6-1183, 6-1184, 6-1185, 6-1202, 6-1203, 6-1204, 6-1218, 6-1225, 6-1260, 6-1261, 6-1262, 6-1263, 6-1280, 6-1281, 6-1282, 6-1296, 6-1303, 6-1338, 6-1339, 6-1340, 6-1341, 6-1358, 6-1359, 6-1360, 6-1374, 6-1381, 6-1574, 6-1575, 6-1576, 6-1577, 6-1594, 6-1595, 6-1596, 6-1610, 6-1617, 6-1652, 6-1653, 6-1654, 6-1655, 6-1672, 6-1673, 6-1674, 6-1688, 6-1695, 6-1730, 6-1731, 6-1732, 6-1733, 6-1734, 6-1750, 6-1751, 6-1752, 6-1754, 6-1755, 6-1766, 6-1773, 6-1808, 6-1809, 6-1810, 6-1811, 6-1828, 6-1829, 6-1830, 6-1851, 6-2110, 6-3348, 6-3384, 6-5902, 6-5903, 6-5904, 6-5905, 6-5906, 6-5907, 6-5908, 6-5909, 6-5910, 6-5911, 6-5912, 7-38, 7-39, 7-45, 7-46, 7-47, 7-57, 7-60, 7-71, 7-72, 7-78, 7-79, 7-80, 7-90, 7-93, 7-132, 7-147, 7-268, 7-269, 7-270, 7-271, 7-285, 7-286, 7-288, 7-289, 7-290, 7-299, 7-300, 7-301, 7-303, 7-304, 7-305, 7-311, 7-346, 7-347, 7-348, 7-349, 7-366, 7-367, 7-368, 7-382, 7-389, 7-424, 7-425, 7-426, 7-427, 7-428, 7-444, 7-445, 7-446, 7-449, 7-460, 7-467, 7-502, 7-504, 7-505, 7-522, 7-523, 7-538, 7-804, 7-824, 7-825, 7-840, 7-948, 7-969, 7-984, 7-1104, 7-1105, 7-1106, 7-1107, 7-1124, 7-1125, 7-1126, 7-1140, 7-1147, 7-1182, 7-1183, 7-1184, 7-1185, 7-1202, 7-1203, 7-1204, 7-1218, 7-1225, 7-1260, 7-1261, 7-1262, 7-1263, 7-1280, 7-1281, 7-1282, 7-1296, 7-1303, 7-1338, 7-1339, 7-1340, 7-1341, 7-1358, 7-1359, 7-1360, 7-1374, 7-1381, 7-1417, 7-1574, 7-1575, 7-1576, 7-1577, 7-1594, 7-1595, 7-1596, 7-1605, 7-1606, 7-1608, 7-1610, 7-1616, 7-1617, 7-1638, 7-1639, 7-1645, 7-1652, 7-1672, 7-1673, 7-1730, 7-1731, 7-1732, 7-1733, 7-1750, 7-1751, 7-1752, 7-1764, 7-1766, 7-1773, 7-1794, 7-1808, 7-1809, 7-1810, 7-1811, 7-1828, 7-1829, 7-1844, 7-1851, 7-3348, 7-3369, 7-3384, 7-5902, 7-5903, 7-5904, 7-5905, 7-5906, 7-5907, 7-5910, 8-268, 8-288, 8-289, 8-304, 8-804, 8-824, 8-840, 9-270, 9-290, 9-291, 9-306, 9-2164, 9-2322, 11-777, 11-835, 12-777, 12-835, 12-864, 27-627, and 27-663 each showed a pesticidal rate of 70% or more at a concentration of 1 ppm.

Furthermore, the compounds of Compound Nos. 1-506, 1-1968, 2-513, 2-518, 6-454, 6-5913, 6-5914, 7-316, 7-5911, 7-5912, 7-5908, 7-5909, 17-1103, and 27-628 each showed a pesticidal rate of 70% or more at a concentration of 10 ppm.

Meanwhile, the compound (A) had a pesticidal rate of 50% or less at a concentration of 10 ppm.

Test Example 2

Pesticidal Test Against Plutella xylostella

A piece of a cabbage leaf was immersed for 30 seconds in a chemical solution in which a test compound had been prepared at a predetermined concentration, and air-dried, and then put into a 7 cm polyethylene cup having a filter paper laid on the bottom thereof, and 2-stage larvae of Plutella xylostella were released. They were left to stand in a thermostatic chamber at 25° C., and the numbers of the living pests and the dead pests were examined after 6 days. The test was carried out with five larvae per group in two replicates.

Further, the above compound (A) was used as a comparative compound.

As the results of the above tests, the compounds of Compound Nos. 1-491, 1-513, 1-627, 1-1925, 1-1968, 2-491, 2-513, 6-38, 6-39, 6-45, 6-46, 6-47, 6-57, 6-71, 6-72, 6-78, 6-79, 6-80, 6-90, 6-111, 6-147, 6-268, 6-270, 6-271, 6-272, 6-288, 6-289, 6-290, 6-293, 6-300, 6-304, 6-306, 6-346, 6-347, 6-348, 6-349, 6-366, 6-367, 6-368, 6-382, 6-389, 6-424, 6-425, 6-426, 6-427, 6-428, 6-444, 6-445, 6-446, 6-449, 6-450, 6-453, 6-460, 6-461, 6-467, 6-502, 6-503, 6-504, 6-505, 6-522, 6-523, 6-524, 6-538, 6-545, 6-804, 6-824, 6-825, 6-840, 6-1104, 6-1105, 6-1106, 6-1107, 6-1124, 6-1125, 6-1126, 6-1140, 6-1147, 6-1182, 6-1183, 6-1184, 6-1185, 6-1202, 6-1203, 6-1204, 6-1218, 6-1225, 6-1260, 6-1261, 6-1262, 6-1263, 6-1280, 6-1281, 6-1282, 6-1296, 6-1303, 6-1338, 6-1339, 6-1340, 6-1341, 6-1358, 6-1359, 6-1360, 6-1374, 6-1381, 6-1574, 6-1575, 6-1576, 6-1577, 6-1594, 6-1595, 6-1596, 6-1610, 6-1617, 6-1652, 6-1653, 6-1654, 6-1655, 6-1672, 6-1673, 6-1674, 6-1688, 6-1695, 6-1730, 6-1731, 6-1732, 6-1733, 6-1734, 6-1750, 6-1751, 6-1752, 6-1754, 6-1755, 6-1766, 6-1773, 6-1808, 6-1809, 6-1810, 6-1811, 6-1828, 6-1829, 6-1830, 6-1851, 6-2110, 6-3348, 6-3384, 6-5903, 6-5904, 6-5905, 6-5906, 6-5907, 6-5908, 6-5909, 6-5910, 6-5911, 6-5912, 7-38, 7-39, 7-45, 7-46, 7-47, 7-57, 7-60, 7-71, 7-72, 7-78, 7-79, 7-80, 7-90, 7-93, 7-132, 7-147, 7-268, 7-271, 7-286, 7-288, 7-289, 7-290, 7-299, 7-300, 7-301, 7-303, 7-304, 7-305, 7-311, 7-346, 7-347, 7-348, 7-349, 7-366, 7-367, 7-368, 7-382, 7-389, 7-424, 7-425, 7-426, 7-427, 7-428, 7-444, 7-445, 7-446, 7-449, 7-460, 7-467, 7-502, 7-504, 7-505, 7-522, 7-523, 7-538, 7-824, 7-840, 7-948, 7-969, 7-984, 7-1104, 7-1105, 7-1106, 7-1107, 7-1124, 7-1125, 7-1126, 7-1140, 7-1147, 7-1182, 7-1183, 7-1184, 7-1185, 7-1202, 7-1203, 7-1204, 7-1218, 7-1225, 7-1260, 7-1261, 7-1262, 7-1263, 7-1280, 7-1281, 7-1282, 7-1296, 7-1303, 7-1338, 7-1339, 7-1340, 7-1341, 7-1358, 7-1359, 7-1360, 7-1374, 7-1381, 7-1417, 7-1574, 7-1575, 7-1576, 7-1577, 7-1594, 7-1595, 7-1596, 7-1605, 7-1606, 7-1608, 7-1610, 7-1616, 7-1617, 7-1638, 7-1639, 7-1645, 7-1652, 7-1672, 7-1673, 7-1730, 7-1731, 7-1732, 7-1733, 7-1750, 7-1751, 7-1752, 7-1764, 7-1766, 7-1773, 7-1794, 7-1808, 7-1809, 7-1810, 7-1811, 7-1828, 7-1829, 7-1844, 7-1851, 7-3348, 7-3369, 7-3384, 7-5902, 7-5903, 7-5904, 7-5905, 7-5906, 7-5907, 7-5909, 7-5910, 8-268, 8-288, 8-289, 8-304, 8-824, 9-270, 9-290, 9-291, 9-306, 9-2164, 9-2322, 11-777, 11-835, 12-777, 12-835, and 12-864 each showed a pesticidal rate of 70% or more at a concentration of 1 ppm.

Furthermore, the compounds of Compound Nos. 1-470, 1-506, 2-518, 6-60, 6-93, 6-269, 6-311, 6-448, 6-452, 6-454, 6-5913, 6-5914, 7-269, 7-270, 7-285, 7-316, 7-804, 7-825, 7-5908, 7-5911, 7-5912, 8-804, 8-840, 17-1103, 27-627, 27-628, and 27-663 each showed a pesticidal rate of 70% or more at a concentration of 10 ppm.

Meanwhile, the compound (A) had a pesticidal rate of 50% or less at a concentration of 10 ppm.

Test Example 3

Pesticidal Test Against Adoxophyes honmai

A thinly sliced artificial feed was immersed for 30 seconds in a chemical solution in which a test compound had been prepared at a predetermined concentration, and air-dried, and then put into a 7 cm polyethylene cup having a filter paper laid on the bottom thereof, and 2-stage larvae of Adoxophyes honmai were released. They were left to stand in a thermostatic chamber at 25° C., and the numbers of the living pests and the dead pests were examined after 6 days. The test was carried out with five larvae per group in two replicates.

Further, the above compound (A) was used as a comparative compound.

As the results of the above tests, the compounds of Compound Nos. 6-72, 6-80, 6-90, 6-347, 6-348, 6-349, 6-366, 6-382, 6-427, 6-446, 6-449, 6-460, 6-503, 6-504, 6-505, 6-522, 6-524, 6-538, 6-1106, 6-1182, 6-1202, 6-1260, 6-1262, 6-1263, 6-1341, 6-1358, 6-1574, 6-1576, 6-1594, 6-1596, 6-1652, 6-1654, 6-1655, 6-1672, 6-1674, 6-1688, 6-1730, 6-1732, 6-1733, 6-1750, 6-1809, 6-1811, 6-1828, 6-1830, 7-348, 7-366, 7-382, 7-502, 7-505, 7-522, 7-538, 7-1106, 7-1202, 7-1262, 7-1280, 7-1303, 7-1338, 7-1358, 7-1574, 7-1576, 7-1594, 7-1605, 7-1652, 7-1730, 7-1732, 7-1733, 7-1750, 7-1764, 7-1808, 7-1809, 7-1810, and 7-1811 each showed a pesticidal rate of 70% or more at a concentration of 1 ppm.

Furthermore, the compounds of Compound Nos. 6-271, 6-367, 6-389, 6-426, 6-523, 6-1104, 6-1577, 6-1695, 6-1851, 6-2110, 7-424, 7-444, 7-523, 7-1104, 7-1124, 7-1260, 7-1263, 7-1577, 7-1616, 7-1731, 7-1773, and 7-1851 each showed a pesticidal rate of 70% or more at a concentration of 10 ppm.

Meanwhile, the compound (A) had a pesticidal rate of 50% or less at a concentration of 10 ppm.

Test Example 4

Pesticidal Test Against Choristoneura magnanima

A thinly sliced artificial feed was immersed for 30 seconds in a chemical solution in which a test compound had been prepared at a predetermined concentration, and air-dried, and then put into a 7 cm polyethylene cup having a filter paper laid on the bottom thereof; and 2-stage larvae of Choristoneura magnanima were released. They were left to stand in a thermostatic chamber at 25° C., and the numbers of the living pests and the dead pests were examined after 6 days. The test was carried out with five larvae per group in two replicates.

Further, the above compound (A) was used as a comparative compound.

As the results of the above tests, the compounds of Compound Nos. 6-72, 6-80, 6-90, 6-271, 6-349, 6-366, 6-367, 6-426, 6-427, 6-1104, 6-1106, 6-1182, 6-1260, 6-1263, 6-1358, 6-1574, 6-1577, 6-1595, 6-1596, 6-1652, 6-1654, 6-1655, 6-1672, 6-1673, 6-1674, 6-1695, 6-1730, 6-1732, 6-1733, 6-1750, 6-1751, 6-1809, 6-1811, 6-1828, 6-1829, 6-1830, 6-1851, 7-90, 7-348, 7-366, 7-382, 7-389, 7-444, 7-502, 7-504, 7-505, 7-523, 7-1104, 7-1106, 7-1107, 7-1124, 7-1125, 7-1260, 7-1262, 7-1263, 7-1280, 7-1281, 7-1303, 7-1358, 7-1359, 7-1574, 7-1576, 7-1577, 7-1594, 7-1595, 7-1605, 7-1616, 7-1617, 7-1652, 7-1730, 7-1732, 7-1733, 7-1750, 7-1764, 7-1773, 7-1808, 7-1809, 7-1810, 7-1811, 7-1829, and 7-1851 each showed a pesticidal rate of 70% or more at a concentration of 1 ppm.

Furthermore, the compounds of Compound Nos. 6-382, 6-446, 6-460, 6-2110, 7-424, 7-538, and 7-1606 each showed a pesticidal rate of 70% or more at a concentration of 10 ppm.

Meanwhile, the compound (A) had a pesticidal rate of 50% or less at a concentration of 10 ppm.

Test Example 5

Pesticidal Test Against Helicoverpa armigera

A cabbage leaf disk was immersed for 30 seconds in a chemical solution in which a test compound had been prepared at a predetermined concentration, and air-dried. The leaf disk was put into a 6-hole plastic cup having a filter paper laid on the bottom thereof, and 2-stage larvae of Helicoverpa armigera were released with one insect being released per hole. They were left to stand in a thermostatic chamber at 25° C., and the numbers of the living pests and the dead pests were examined after 3 days. The test was carried out with five larvae per group in two replicates.

Further, the above compound (A) was used as a comparative compound.

As the results of the above tests, the compounds of Compound Nos. 6-72, 6-80, 6-90, 6-271, 6-347, 6-348, 6-349, 6-366, 6-367, 6-382, 6-389, 6-426, 6-427, 6-446, 6-449, 6-460, 6-503, 6-504, 6-505, 6-522, 6-523, 6-524, 6-538, 6-1104, 6-1106, 6-1260, 6-1262, 6-1263, 6-1281, 6-1341, 6-1358, 6-1359, 6-1574, 6-1576, 6-1577, 6-1594, 6-1595, 6-1596, 6-1652, 6-1654, 6-1655, 6-1672, 6-1673, 6-1674, 6-1695, 6-1730, 6-1732, 6-1733, 6-1750, 6-1751, 6-1808, 6-1809, 6-1811, 6-1828, 6-1829, 6-1830, 6-1851, 6-2110, 7-90, 7-348, 7-366, 7-382, 7-389, 7-424, 7-444, 7-502, 7-505, 7-522, 7-523, 7-538, 7-1106, 7-1107, 7-1125, 7-1262, 7-1263, 7-1280, 7-1303, 7-1338, 7-1358, 7-1359, 7-1574, 7-1576, 7-1577, 7-1594, 7-1595, 7-1605, 7-1606, 7-1616, 7-1617, 7-1652, 7-1730, 7-1731, 7-1732, 7-1733, 7-1750, 7-1751, 7-1764, 7-1773, 7-1808, 7-1809, 7-1810, 7-1811, 7-1829, and 7-1851 each showed a pesticidal rate of 70% or more at a concentration of 1 ppm.

Furthermore, the compound of Compound No. 7-1104 showed a pesticidal rate of 70% or more at a concentration of 10 ppm.

Meanwhile, the compound (A) had a pesticidal rate of 50% or less at a concentration of 10 ppm.

Test Example 6

Pesticidal Test Against Laodelphax striatellus

2.5 ml of an acetone solution in which a test compound had been prepared at a predetermined concentration was sprayed on rice seedlings, air-dried, and then put into a glass tube having a diameter of 3 cm and a height of 13 cm, having water therein, and 3-stage larvae of Laodelphax striatellus were released and the tube was capped. They were left to stand in a thermostatic chamber at 25° C., and the numbers of the living pests and the dead pests were examined after 6 days. The test was carried out with ten larvae per group in two replicates.

As the results of the above tests, the compounds of Compound Nos. 1-491, 1-627, 2-491, 6-39, 6-45, 6-47, 6-57, 6-71, 6-72, 6-79, 6-80, 6-90, 6-147, 6-268, 6-269, 6-270, 6-271, 6-290, 6-304, 6-306, 6-311, 6-346, 6-347, 6-368, 6-382, 6-425, 6-427, 6-444, 6-445, 6-446, 6-460, 6-461, 6-503, 6-1104, 6-1106, 6-1107, 6-1124, 6-1126, 6-1140, 6-1147, 6-1182, 6-1183, 6-1184, 6-1185, 6-1202, 6-1203, 6-1204, 6-1218, 6-1225, 6-1260, 6-1261, 6-1262, 6-1263, 6-1280, 6-1281, 6-1282, 6-1296, 6-1303, 6-1338, 6-1339, 6-1340, 6-1341, 6-1358, 6-1359, 6-1360, 6-1374, 6-1381, 6-1574, 6-1575, 6-1576, 6-1577, 6-1594, 6-1595, 6-1596, 6-1610, 6-1617, 6-1652, 6-1653, 6-1654, 6-1655, 6-1672, 6-1673, 6-1674, 6-1688, 6-1695, 6-1730, 6-1731, 6-1732, 6-1733, 6-1734, 6-1750, 6-1751, 6-1752, 6-1754, 6-1766, 6-1773, 6-1808, 6-1809, 6-1810, 6-1811, 6-1828, 6-1829, 6-1830, 6-1851, 6-2110, 6-3348, 6-3384, 6-5903, 6-5904, 6-5905, 6-5906, 6-5907, 6-5908, 6-5909, 6-5910, 6-5911, 6-5914, 7-47, 7-57, 7-90, 7-268, 7-285, 7-286, 7-288, 7-289, 7-301, 7-303, 7-304, 7-305, 7-311, 7-316, 7-346, 7-348, 7-368, 7-382, 7-389, 7-424, 7-426, 7-427, 7-444, 7-445, 7-446, 7-460, 7-467, 7-538, 7-825, 7-840, 7-948, 7-984, 7-1104, 7-1105, 7-1106, 7-1107, 7-1124, 7-1125, 7-1126, 7-1140, 7-1147, 7-1182, 7-1183, 7-1184, 7-1185, 7-1202, 7-1203, 7-1204, 7-1218, 7-1225, 7-1260, 7-1261, 7-1262, 7-1263, 7-1280, 7-1281, 7-1282, 7-1296, 7-1303, 7-1338, 7-1339, 7-1340, 7-1341, 7-1358, 7-1359, 7-1360, 7-1374, 7-1381, 7-1417, 7-1574, 7-1575, 7-1576, 7-1577, 7-1594, 7-1595, 7-1596, 7-1605, 7-1606, 7-1608, 7-1610, 7-1616, 7-1617, 7-1638, 7-1639, 7-1645, 7-1652, 7-1672, 7-1673, 7-1730, 7-1731, 7-1732, 7-1733, 7-1750, 7-1751, 7-1752, 7-1764, 7-1766, 7-1773, 7-1794, 7-1808, 7-1809, 7-1810, 7-1811, 7-1828, 7-1829, 7-1844, 7-1851, 7-3348, 7-3369, 7-5902, 7-5903, 7-5904, 7-5906, 7-5907, 7-5909, 7-5912, 8-289, 8-304, 8-840, 9-270, 9-290, 9-291, 9-306, 9-2164, 9-2322, 12-835, and 12-864 each showed a pesticidal rate of 70% or more at a concentration of 100 ppm.

Test Example 7

Pesticidal Test Against Musca domestica

1 ml of an acetone solution in which a test compound had been prepared at a predetermined concentration was added dropwise to a petri dish having a diameter of 9 cm, and air-dried, and then the female adults of Musca domestica were released and the petri dish was capped. They were left to stand in a thermostatic chamber at 25° C., and the numbers of the living pests and the dead pests were examined after 1 day. The test was carried out with five larvae per group in two replicates.

As the results of the above tests, the compounds of Compound Nos. 1-1925, 1-1968, 6-39, 6-47, 6-72, 6-272, 6-293, 6-346, 6-347, 6-348, 6-366, 6-368, 6-382, 6-389, 6-426, 6-427, 6-428, 6-450, 6-452, 6-453, 6-460, 6-503, 6-504, 6-505, 6-522, 6-523, 6-524, 6-538, 6-1105, 6-1107, 6-1124, 6-1125, 6-1126, 6-1147, 6-1184, 6-1204, 6-1218, 6-1260, 6-1281, 6-1338, 6-1341, 6-1358, 6-1359, 6-1360, 6-1374, 6-1575, 6-1576, 6-1577, 6-1594, 6-1596, 6-1617, 6-1652, 6-1672, 6-1673, 6-1695, 6-1730, 6-1731, 6-1732, 6-1733, 6-1734, 6-1750, 6-1751, 6-1752, 6-1773, 6-1808, 6-1809, 6-1810, 6-1811, 6-1828, 6-1829, 6-1830, 6-1851, 6-2110, 6-5905, 7-39, 7-57, 7-90, 7-268, 7-346, 7-348, 7-349, 7-366, 7-367, 7-368, 7-382, 7-389, 7-424, 7-428, 7-444, 7-446, 7-449, 7-504, 7-522, 7-538, 7-1104, 7-1105, 7-1106, 7-1107, 7-1126, 7-1262, 7-1280, 7-1282, 7-1296, 7-1303, 7-1338, 7-1340, 7-1358, 7-1359, 7-1360, 7-1381, 7-1417, 7-1574, 7-1575, 7-1576, 7-1577, 7-1596, 7-1652, 7-1731, 7-1732, 7-1733, 7-1750, 7-1752, 7-1764, 7-1766, 7-1730, 7-1773, 7-1794, 7-1808, 7-1809, 7-1810, 7-1811, 7-1828, 7-1829, 7-1851, 9-2164, 9-2322, 11-777, 11-835, 12-777, 12-835, 12-864, 17-1103, and 27-627 each showed a pesticidal rate of 70% or more at a concentration of 100 ppm.

Test Example 8

Pesticidal Test Against Blattella germanica

1 ml of an acetone solution in which a test compound had been prepared at a predetermined concentration was added dropwise to a petri dish having a diameter of 9 cm, and air-dried, and then the female adults of Blattella germanica were released and the petri dish was capped. They were left to stand in a thermostatic chamber at 25° C., and the numbers of the living pests and the dead pests were examined after 1 day. The test was carried out with five larvae per group in two replicates.

As the results of the above tests, the compounds of Compound Nos. 1-1925, 6-39, 6-47, 6-346, 6-347, 6-367, 6-368, 6-382, 6-389, 6-426, 6-427, 6-503, 6-538, 6-1105, 6-1106, 6-1107, 6-1124, 6-1125, 6-1126, 6-1147, 6-1184, 6-1204, 6-1218, 6-1280, 6-1296, 6-1338, 6-1358, 6-1359, 6-1575, 6-1576, 6-1577, 6-1594, 6-1595, 6-1596, 6-1610, 6-1617, 6-1730, 6-1731, 6-1732, 6-1733, 6-1750, 6-1751, 6-1752, 6-1773, 6-1811, 6-5905, 7-57, 7-268, 7-305, 7-347, 7-349, 7-367, 7-382, 7-389, 7-424, 7-444, 7-446, 7-502, 7-505, 7-538, 7-1104, 7-1105, 7-1106, 7-1107, 7-1125, 7-1126, 7-1261, 7-1262, 7-1280, 7-1282, 7-1296, 7-1303, 7-1381, 7-1574, 7-1575, 7-1576, 7-1577, 7-1594, 7-1595, 7-1596, 7-1617, 7-1731, 7-1732, 7-1733, 7-1750, 7-1752, 7-1766, 7-1773, and 7-1851 each showed a pesticidal rate of 70% or more at a concentration of 100 ppm.

Test Example 9

Pesticidal Test Against Culex pipiens Molestus

1 ml of an acetone solution in which a test compound had been prepared at a predetermined concentration was added dropwise to a petri dish having a diameter of 9 cm, and air-dried, and then the female adults of Culex pipiens molestus were released and the petri dish was capped. They were left to stand in a thermostatic chamber at 25° C., and the numbers of the living pests and the dead pests were examined after 1 day of treatment. The test was carried out with five larvae per group in two replicates.

As the results of the above tests, the compounds of Compound Nos. Compound No. 7-424, 7-1574, 7-1577, 7-1730, 7-1732, and 7-1733 each showed a pesticidal rate of 70% or more at a concentration of 1000 ppm.

Test Example 10

Pesticidal Test Against Coptotermes formosanus

20 μl of an acetone solution in which a test compound had been prepared at a predetermined concentration was added dropwise to the filter paper having a diameter of 2.6 mm included in a polypropylene cup, and air-dried, and then 20 dl of water was added thereto. Coptotermes formosanus was released and the cup was capped. They were left to stand in a thermostatic chamber at 28° C., and the numbers of the living pests and the dead pests were examined after 5 days of treatment. The test was carried out with ten larvae per group in two replicates.

As the results of the above tests, the compounds of Compound Nos. Compound No. 6-460, 6-1260, 6-1652, 7-268, 7-424, 7-1104, 7-1574, 7-1577, 7-1730, 7-1732, and 7-1733 each showed a pesticidal rate of 70% or more at a concentration of 30 ppm.

According to the present invention, it becomes possible to provide a novel amide derivative. The amide derivative shows a significant effect for a pest control activity, and has a high industrial availability.

The present invention also provides a composition and method for exterminating animal parasites.

WO2005/21488, WO2005/73165, WO2006/137376, and WO2006/137395 disclose various compounds which are amide derivatives having the ability to control pests, and methods for using them. Further WO2009/080203 discloses amide derivatives which are animal parasiticides, and methods for using them.

In addition, conventional parasiticides for administration to an animal to exterminate animal parasites include formulations of imidacloprid, fipronil, etc.

However, some parasites are impossible or difficult to exterminate with said animal parasiticides.

Thus, an objective of the invention is to provide a composition that has excellent activity for exterminating animal parasites, and a method for exterminating animal parasites.

As the result of earnest research for solving the above problem, the present inventors found that an aromatic carboxamide derivative represented by Formula (A1) of the present invention is a novel compound that is not disclosed in the literature, and a composition containing the present aromatic carboxamide derivative as an active ingredient has excellent activity for exterminating animal parasites, thereby completing the present invention.

A first aspect of the present invention provides a composition for exterminating animal parasites which comprises as an active ingredient at least one amide derivative represented by the following Formula (A1).

In Formula (A1), Q₁ represents a phenyl group or a phenyl group substituted with a halogen atom; X₁ represents a fluorine atom, and X₂, X₃, and X₄ are each a hydrogen atom; R₁ represents a hydrogen atom or a C₁-C₃ alkyl group; R₂ is a hydrogen atom; Y₁ and Y₅ each independently represent a halogen atom or a C₁-C₃ haloalkyl group; Y₂ and Y₄ each represent a hydrogen atom; and Y₃ represents a heptafluoroisopropyl group.

In Formula (A1), Q₁ represents a phenyl group or a phenyl group substituted with a single fluorine atom; R₁ represents a hydrogen atom or a methyl group; and Y₁ and Y₅ each independently represent a bromine or iodine atom or a trifluoromethyl group preferably.

The amide derivative represented by Formula (A1) is preferably 2-fluoro-3-(N-methylbenzamide)-N-(2-bromo-6-trifluoromethyl-4-(heptafluoropropan-2-yl)phenyl)benzamide, 2-fluoro-3-(4-fluoro-N-methylbenzamide)-N-(2-iodo-6-trifluoromethyl-4-(heptafluoropropan-2-yl)phenyl)benzamide, 2-fluoro-3-(3-fluoro-N-methylbenzamide)-N-(2-iodo-6-trifluoromethyl-4-(heptafluoropropan-2-yl)phenyl)benzamide, 2-fluoro-3-(4-fluorobenzamide)-N-(2-iodo-6-trifluoromethyl-4-(heptafluoropropan-2-yl)phenyl)benzamide, or 2-fluoro-3-(N-methylbenzamide)-N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)benzamide.

In Formula (A1), Q₁ represents preferably a phenyl group, a 2-fluorophenyl group, a 3-fluorophenyl group, a 4-fluorophenyl group, a 2-chlorophenyl group, a 3-chlorophenyl group, a 4-chlorophenyl group, a 2-bromophenyl group, a 3-bromophenyl group, a 4-bromophenyl group, a 2-iodophenyl group, a 3-iodophenyl group, or a 4-iodophenyl group.

The amide derivative represented by Formula (A1) is preferably 3-benzamide-N-(2-bromo-chloro-4-(heptafluoropropan-2-yl)phenyl)-2-fluorobenzamide, 3-benzamide-N-(2,6-d iodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluorobenzamide, 3-benzamide-N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluorobenzamide, N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide, N-(2,6-dichloro-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide, N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide, N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(2-fluorobenzamide)benzamide, N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(4-fluorobenzamide)benzamide, 3-(2,6-difluorobenzamide)-N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluorobenzamide, N-(2-bromo-6-iodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide,

N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(3-fluorobenzamide)benzamide, N-(3-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2-fluoro-N-methylbenzamide, N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(3-fluoro-N-methylbenzamide)benzamide, N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(4-fluoro-N-methylbenzamide)benzamide, N-(3-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2,6-difluoro-N-methylbenzamide, N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(2-fluorobenzamide)benzamide, N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(3-fluorobenzamide)benzamide, N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(4-fluorobenzamide)benzamide, N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-3-(2,6-difluorobenzamide)-2-fluorobenzamide, N-(3-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2-fluoro-N-methylbenzamide, N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(3-fluoro-N-methylbenzamide)benzamide, N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(4-fluoro-N-methylbenzamide)benzamide, N-(3-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenylcarbamoyl)-2-fluorophenyl)-2,6-difluoro-N-methylbenzamide,

3-benzamide-N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluorobenzamide, N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide, 3-benzamide-2-fluoro-N-(4-(heptafluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)benzamide, 3-benzamide-2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 3-benzamide-N-(2-bromo-6-(pentafluoroethyl)-4-(heptafluoropropan-2-yl)phenyl)-2-fluorobenzamide, 2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(N-methylbenzamide)benzamide, 2-fluoro-N-(2-fluoro-3-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 2-fluoro-3-(3-fluoro-N-methylbenzamide)-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-3-(4-fluoro-N-methylbenzamide)-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2,6-difluoro-N-(2-fluoro-3-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)phenyl)-N-methylbenzamide, 2-fluoro-3-(2-fluorobenzamide)-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 2-fluoro-3-(3-fluorobenzamide)-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, N-(3-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-2-fluoro-N-methylbenzamide, N-(3-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenylcarbamoyl)-2-fluorophenyl)-2,6-difluoro-N-methylbenzamide, N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(3-fluoro-N-methylbenzamide)benzamide, N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(4-fluoro-N-methylbenzamide)benzamide, N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethy)phenyl)-2-fluoro-3-(2-fluowobenzamide)benzamide, N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(3-fluorobenzamide)benzamide, N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(4-fluorobenzamide)benzamide,

2-fluoro-3-(4-fluorobenzamide)-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 3-(2,6-difluorobenzamide)-2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethy)phenyl)benzamide, N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(2,6-difluorobenzamide)-2-fluorobenzamide, 3-(2,4-dichlorobenzamide)-2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 3-(2-chloro-4-fluorobenzamide)-2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, 3-(2-chlorobenzamide)-2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide, or N-(2-chloro-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide.

A second aspect of the present invention provides a method for exterminating animal parasites comprising administering to the animal the composition for exterminating animal parasites

Wherein, the animal parasite is preferably an ectoparasite and the ectoparasite is more preferably Siphonaptera pests or the ectoparasite is Acarina pests.

According to the present invention, a composition which has excellent activity for exterminating animal parasites and a method for exterminating animal parasites are provided.

A composition for exterminating animal parasites according to the present invention includes at least one amide derivative represented by the following Formula (A1).

By adopting such a constitution, it becomes possible to show excellent activity for exterminating animal parasites in the case of giving the composition to an animal.

In Formula (A1), Q₁ represents a phenyl group or a phenyl group substituted with a halogen atom. X, represents a fluorine atom, and X₂, X₃, and X₄ are each a hydrogen atom. R₁ represents a hydrogen atom or a C1-C3 alkyl group, and R₂ is a hydrogen atom. Y₁ and Y₅ each independently represent a halogen atom or a C1-C3 haloalkyl group, Y₂ and Y₄ each represent a hydrogen atom, and Y₃ represents a heptafluoroisopropyl group.

The terms used in the formulae including the Formula (A1) and the like according to the present invention, have the same meanings as described below in the definitions.

The “halogen atom” represents a fluorine atom, a chlorine atom, a bromine atom, or an iodine atom.

The expression “Ca-Cb (wherein a and b represent an integer of 1 or more)”, for example, “C1-C3” means the number of carbon atoms of from 1 to 3, the “C2-C6” means the number of carbon atoms of from 2 to 6.

The “C1-C3 alkyl group” in the present invention represents, for example, a linear or branched alkyl group having from 1 to 3 carbon atoms such as methyl, ethyl, n-propyl, i-propyl, and the like.

The “C1-C3 haloalkyl group” represents, for example, a linear or branched alkyl group having from 1 to 3 carbon atoms, that is substituted with one or more halogen atoms which may be the same as or different from each other, such as trifluoromethyl, pentafluoroethyl, heptafluoro-n-propyl, heptafluoro-i-propyl, 2,2-difluoroethyl, 2,2-dichloroethyl, 2,2,2-trifluoroethyl, 2-fluoroethyl, 2-chloroethyl, 2-bromoethyl, 2-iodoethyl, 2,2,2-trichloroethyl, 2,2,2-tribromoethyl, 1,3-difluoro-2-propyl, 1,3-dichloro-2-propyl, 1-chloro-3-fluoro-2-propyl, 1,1,1-trifluoro-2-propyl, 2,3,3,3-trifluoro-n-propyl, 1,1,1,3,3,3-hexafluoro-2-propyl, 1,1,1,3,3,3-hexafluoro-2-chloro-2-propyl, 1,1,1,3,3,3-hexafluoro-2-bromo-2-propyl, 1,1,2,3,3,3-hexafluoro-2-chloro-n-propyl, 1,1,2,3,3,3-hexafluoro-2-bromo-n-propyl, 1,1,2,3,3,3-hexafluoro-1-bromo-2-propyl, 2,2,3,3,3-pentafluoro-n-propyl, 3-fluoro-n-propyl, 3-chloro-n-propyl, 3-bromo-n-propyl, and the like.

The “C1-C6 alkyl group” in the present invention represents, for example, a linear or branched alkyl group having from 1 to 6 carbon atoms such as methyl, ethyl, n-propyl, i-propyl, n-butyl, s-butyl, t-butyl, n-pentyl, 2-pentyl, neopentyl, 4-methyl-2-pentyl, n-hexyl, 3-methyl-n-pentyl, and the like.

The “C3-C9 cycloalkyl group” represents, for example, a cycloalkyl group having from 3 to 9 carbon atoms, that has a cyclic structure, such as cyclopropyl, cyclobutyl, cyclopentyl, 2-methylcyclopentyl, 3-methylcyclopentyl, cyclohexyl, 2-methylcyclohexyl, 3-methylcyclohexyl, 4-methylcyclohexyl, and the like.

The “C2-C6 alkenyl group” represents, for example, an alkenyl group having from 2 to 6 carbon atoms, that has a double bond in the carbon chain, such as vinyl, allyl, 2-butenyl, 3-butenyl, and the like.

The “C2-C6 alkynyl group” represents, for example, an alkynyl group having from 2 to 6 carbon atoms, that has a triple bond in the carbon chain, such as propargyl, 1-butyn-3-yl, l-butyn-3-methyl-3-yl, and the like.

The compounds represented by Formula (A1) according to the present invention may include one or plural chiral carbon atoms or chiral centers in their structural Formulae, and thus two or more optical isomers may exist. However, the present invention includes each of the optical isomers and a mixture thereof at any proportions. Further, the compounds represented by Formula (A1) according to the present invention may include two or more kinds of geometrical isomers derived from carbon-carbon double bonds in the structural Formulae. The present invention includes each of the geometrical isomers and a mixture thereof at any proportions.

The representative methods for producing the compound according to the present invention are shown below, and the method for producing the amide derivative according to the present invention is not limited to the preparation methods below.

In Formula shown in the following preparation method, X₁, X₂, X₃, X₄, R₁, R₂, Q₁, Y₁, Y₂, Y₃, Y₄, and Y₅ represent the same definitions as X₁, X₂, X₃, X₄, R₁, R₂, Q₁, Y₁, Y₂, Y₃, Y₄, and Y₅, respectively, in Formula (A1). LG represents a functional group having a leaving ability, such as a halogen atom, a hydroxy group, or the like, Hal represents a chlorine atom or a bromine atom, and Xa and Xb represent chlorine atoms, bromine atoms, or iodine atoms. R3 represents a C1-C6 alkyl group, a C3-C9 cycloalkyl group, a C2-C6 alkenyl group, a C2-C6 alkynyl group.

Preparation Method 1

1-(i): Formula (A11)+Formula (A12)→Formula (A13))

A nitro aromatic carboxamide derivative represented by Formula (A13) can be prepared by reacting a nitro aromatic carboxylic acid derivative having a leaving group represented by Formula (A11) with an aromatic amine derivative represented by Formula (A 12) in a suitable solvent or without a solvent. In the present step, a suitable base can be used.

The solvent may be any of those which do not inhibit the present reaction significantly. Examples thereof may include water and aromatic hydrocarbons such as benzene, toluene, xylene, and the like, halogenated hydrocarbons such as dichloromethane, chloroform, carbon tetrachloride, and the like, chained or cyclic ethers such as diethyl ether, dioxane, tetrahydrofuran, 1,2-dimethoxy ethane, and the like, esters such as ethyl acetate, butyl acetate, and the like, alcohols such as methanol, ethanol, and the like, ketones such as acetone, methyl isobutyl ketone, cyclohexanone, and the like, amides such as dimethyl formamide, dimethylacetamide, and the like, nitriles such as acetonitrile and the like, and inert solvents such as 1,3-dimethyl-2-imidazolidinone and the like. These solvents may be used alone or as a mixture of two or more kinds thereof.

Furthermore, examples of the base may include organic bases such as triethylamine, tri-n-butyl amine, pyridine, 4-dimethylamino pyridine, and the like, alkali metal hydroxides such as sodium hydroxide, potassium hydroxide, and the like, carbonates such as sodium hydrogen carbonate, potassium carbonate, and the like, phosphates such as dipotassium monohydrogen phosphate, trisodium phosphate, and the like, alkali metal hydride salts such as sodium hydride and the like, alkali metal alkoxides such as sodium methoxide, sodium ethoxide, and the like, and lithium amides such as lithium diisopropyl amide, and the like.

These bases may be appropriately used in an amount in the range from 0.01-fold molar equivalent to 5-fold molar equivalents with respect to the compound represented by Formula (A11).

The reaction temperature may be appropriately selected from −20° C. to the reflux temperature of the solvent used. Further, the reaction time may be appropriately selected within the range from several minutes to 96 hours.

Among the compounds represented by Formula (A11), the aromatic carbonyl halide derivative can be prepared easily by a general method using a halogenating agent from an aromatic carboxylic acid. Examples of the halogenating agent include thionyl chloride, thionyl bromide, phosphorus oxychloride, oxalyl chloride, phosphorus trichloride, and the like.

Meanwhile, it is possible to prepare the compound represented by Formula (A13) from the nitro aromatic carboxylic acid derivative and the compound represented by Formula (A12) without using a halogenating agent. Examples of the method may include a method described in, for example, Chem. Ber. p. 788 (1970), in which a condensing agent such as N,N′-dicyclohexylcarbodiimide and the like is appropriately used, suitably with the use of an additive such as 1-hydroxybenzotriazole and the like. Other condensing agents that can be used in this case may include 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide, 1,1′-carbonylbis-1H-imidazole, and the like.

Furthermore, examples of other methods for producing the compound represented by Formula (A13) may include a mixed acid anhydride method using chloroformic acid esters, and examples thereof include a method described in J. Am. Chem. Soc., p. 5012 (1967), whereby the compound represented by Formula (A13) can be prepared. Examples of the chloroformic acid esters used in this case may include isobutyl chloroformate, isopropyl chloroformate and the like. In addition to chloroformic acid esters, diethylacetyl chloride, trimethylacetyl chloride and the like may also be included.

Both the method using a condensing agent and the mixed acid anhydride method are not limited by the solvent, the reaction temperature, and the reaction time according to the literature above. An inert solvent may be used which does not inhibit the progress of the appropriate reaction significantly, and the reaction temperature and the reaction time may also be selected appropriately according to the progress of the reaction.

1-(ii): Formula (A13)→Formula (A14)

An aromatic carboxamide derivative having an amino group represented by Formula (A14) can be derived from the aromatic carboxamide derivative having a nitro group represented by Formula (A13) by means of a reduction reaction. Examples of such reduction include a method using a hydrogenation reaction and a method using a metal compound (for example, stannous chloride (anhydride), iron powder, zinc powder, and the like).

The reaction of the former method can be carried out in a suitable solvent in the presence of a catalyst at normal pressure or a higher pressure under a hydrogen atmosphere. Examples of the catalyst may include palladium catalysts such as palladium-carbon and the like, nickel catalysts such as Raney-nickel and the like, cobalt catalysts, ruthenium catalysts, rhodium catalysts, platinum catalysts, and the like, and examples of the solvent may include water; alcohols such as methanol, ethanol, and the like; aromatic hydrocarbons such as benzene, toluene, and the like; chained or cyclic ethers such as ether, dioxane, tetrahydrofuran, and the like; and esters such as ethyl acetate and the like. The pressure may be appropriately selected within a range of 0.1 MPa to 10 MPa, the reaction temperature may be appropriately selected within a range of −20° C. to the reflux temperature of the solvent used, and the reaction time may be appropriately selected within a range of several minutes to 96 hours, whereby the compound of Formula (14) can be efficiently prepared.

Examples of the latter method include a method using stannous chloride (anhydride) as a metal compound under the conditions described in “Organic Syntheses” Coll. Vol. III, P. 453.

1-(iii): Formula (A14)→Formula (A15)

(Method A)

A compound represented by Formula (A15) can be prepared by reacting the compound represented by Formula (A14) with an aldehyde or a ketone in a solvent, and reacting them under a hydrogen atmosphere with the addition of a catalyst.

The solvent may be any of those which do not inhibit the progress of the reaction significantly, and examples thereof may include aliphatic hydrocarbons such as hexane, cyclohexane, methylcyclohexane, and the like, aromatic hydrocarbons such as benzene, xylene, toluene, and the like, halogenated hydrocarbons such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, and the like, ethers such as diethyl ether, dioxane, tetrahydrofuran, 1,2-dimethoxy ethane, and the like, amides such as dimethyl formamide, dimethylacetamide, and the like, nitriles such as acetonitrile, propionitrile, and the like, ketones such as acetone, methyl isobutyl ketone, cyclohexanone, methyl ethyl ketone, and the like, esters such as ethyl acetate, butyl acetate, and the like, alcohols such as methanol, ethanol, and the like, inert solvents such as 1,3-dimethyl-2-imidazolidinone, sulfolane, dimethylsulfoxide, and the like, water, and the like. These solvents may be used alone or as a mixture of two or more kinds thereof.

Examples of the catalyst may include palladium catalysts such as palladium-carbon, palladium hydroxide-carbon, and the like, nickel catalysts such as Raney-nickel and the like, cobalt catalysts, platinum catalysts, ruthenium catalysts, rhodium catalysts, and the like.

Examples of the aldehydes may include formaldehyde, acetaldehyde, propionaldehyde, trifluoroacetaldehyde, difluoroacetaldehyde, fluoroacetaldehyde, chloroacetaldehyde, dichloroacetaldehyde, trichloroacetaldehyde, bromoacetaldehyde, and the like.

Examples of the ketones may include acetone, perfluoroacetone, methyl ethyl ketone, and the like.

The reaction pressure may be appropriately selected within the range of 1 atm to 100 atm. The reaction temperature may be appropriately selected within the range from −20° C. to the reflux temperature of the solvent used. Further, the reaction time may be appropriately selected within the range from several minutes to 96 hours.

(Method B)

A compound represented by Formula (A 15) can be prepared by reacting the compound represented by Formula (A14) with an aldehyde or a ketone in a solvent, and treating the product with a reducing agent.

The solvent may be any of those which do not inhibit the progress of the reaction significantly, and examples thereof may include aliphatic hydrocarbons such as hexane, cyclohexane, methylcyclohexane, and the like, aromatic hydrocarbons such as benzene, xylene, toluene, and the like, halogenated hydrocarbons such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, and the like, ethers such as diethyl ether, dioxane, tetrahydrofuran, 1,2-dimethoxy ethane, and the like, amides such as dimethyl formamide, dimethylacetamide, and the like, nitriles such as acetonitrile, propionitrile, and the like, ketones such as acetone, methyl isobutyl ketone, cyclohexanone, methyl ethyl ketone, and the like, esters such as ethyl acetate, butyl acetate, and the like, alcohols such as methanol, ethanol, and the like, inert solvents such as 1,3-dimethyl-2-imidazolidinone, sulfolane, dimethylsulfoxide, and the like, water, and the like. These solvents may be used alone or as a mixture of two or more kinds thereof.

Examples of the reducing agent may include, for example, borohydrides such as sodium borohydride, sodium cyanoborohydride, sodium triacetate borohydride, and the like.

Examples of the aldehydes may include formaldehyde, acetaldehyde, propionaldehyde, trifluoroacetaldehyde, difluoroacetaldehyde, fluoroacetaldehyde, chloroacetaldehyde, dichloroacetaldehyde, trichloroacetaldehyde, bromoacetaldehyde, and the like.

Examples of the ketones may include acetone, perfluoroacetone, methyl ethyl ketone, and the like.

The reaction temperature may be appropriately selected within the range from −20° C. to the reflux temperature of the solvent used. Further, the reaction time may be appropriately selected within the range from several minutes to 96 hours.

(Method C)

A compound of Formula (A15) can be prepared by reacting the compound represented by Formula (A14) with an aldehyde in a solvent or without a solvent.

The solvent may be any of those which do not inhibit the progress of the reaction significantly, and examples thereof may include aliphatic hydrocarbons such as hexane, cyclohexane, methylcyclohexane, and the like, aromatic hydrocarbons such as benzene, xylene, toluene, and the like, halogenated hydrocarbons such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, and the like, ethers such as diethyl ether, dioxane, tetrahydrofuran, 1,2-dimethoxy ethane, and the like, amides such as dimethyl formamide, dimethylacetamide, and the like, nitriles such as acetonitrile, propionitrile, and the like, ketones such as acetone, methyl isobutyl ketone, cyclohexanone, methyl ethyl ketone, and the like, esters such as ethyl acetate, butyl acetate, and the like, alcohols such as methanol, ethanol, and the like, inert solvents such as 1,3-dimethyl-2-imidazolidinone, sulfolane, dimethylsulfoxide, and the like, inorganic acids such as sulfuric acid, hydrochloric acid, and the like, organic acids such as formic acid, acetic acid, and the like, water, and the like. These solvents may be used alone or as a mixture of two or more kinds thereof.

Examples of the aldehydes may include formaldehyde, acetaldehyde, propionaldehyde, and the like.

The reaction temperature may be appropriately selected within the range from −20° C. to the reflux temperature of the solvent used, and the reaction time may be appropriately selected within the range from several minutes to 96 hours.

1-(iv): Formula (A15)+Formula (A16)→Formula (A1)

An aromatic carboxamide derivative represented by Formula (A1) can be prepared by reacting the aromatic amine derivative represented by Formula (A 15) with the carboxylic acid derivative or the carbonate ester derivative having a leaving group represented by Formula (A16) in a suitable solvent. In the present step, a suitable base or solvent can be used, and as the base or solvent, those exemplified in 1-(i) can be used. Examples of the reaction temperature, the reaction time, and the like may include those exemplified in 1-(i).

In Formula (A16), the carbonyl chloride derivative can be prepared easily from a carboxylic acid derivative by a general method using a halogenating agent. The halogenating agent may include those exemplified in 1-(i).

There may be exemplified a method for producing a compound represented by Formula (A1) from the carboxylic acid derivative (A16) and the compound represented by Formula (A15) without the use of a halogenating agent, and the preparation can be conducted according to the method exemplified in 1-(i).

Preparation Method 2

2-(i): Formula (A17)+Formula (A12)→Formula (A18)

A compound represented by Formula (A18) can be prepared by reacting the compound represented by Formula (A17) with a compound represented by Formula (A12) under the condition described in 1-(i).

2-(ii): Formula (A18)→Formula (A15)

A compound represented by Formula (A15) can be prepared by carrying out an amination reaction using an amination agent such as ammonia and the like according to the conditions described, for example, in J. Org. Chem. p. 280 (1958). However, the conditions such as a reaction solvent and the like are not restricted to those described in the literature, and an inert solvent which does not inhibit the proper progress of the reaction significantly may be used. The reaction temperature and reaction time may be suitably selected as the reaction proceeds. Further, examples of the amination agent include methylamine, ethylamine or the like, in addition to ammonia.

2-(iii): Formula (A15)+Formula (A16)→Formula (A1)

The compound represented by Formula (A1) can be prepared by reacting the compound represented by Formula (A15) with a compound represented by Formula (A16) according to the conditions described in l-(i).

Preparation Method 3

3-(i): Formula (A19)+Formula (A12)→Formula (A20)

A compound represented by Formula (A20) can be prepared by reacting the compound represented by Formula (A19) and the compound represented by Formula (A12) according to the conditions described in 1-(i).

3-(ii): Formula (A20)→Formula (A21)

A compound represented by Formula (A21) can be prepared by reacting the nitro aromatic carboxamide derivative represented by Formula (A20) with a suitable fluorinating agent in a suitable solvent or without a solvent.

The solvent may be any of those which do not inhibit the progress of the reaction significantly, and examples thereof may include aliphatic hydrocarbons such as hexane, cyclohexane, methylcyclohexane, and the like, aromatic hydrocarbons such as benzene, toluene, xylene, and the like, halogenated hydrocarbons such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, and the like, chained or cyclic ethers such as diethyl ether, dioxane, tetrahydrofuran, 1,2-dimethoxy ethane, and the like, esters such as ethyl acetate, butyl acetate, and the like, ketones such as acetone, methyl isobutyl ketone, cyclohexanone, methyl ethyl ketone, and the like, nitriles such as acetonitrile, propionitrile, and the like, and aprotic polar solvents such as 1,3-dimethyl-2-imidazolidinone, sulfolane, dimethylsulfoxide, N,N-dimethyl formamide, N-methyl pyrrolidone, N,N-dimethylacetamide, and the like. These solvents may be used alone or as a mixture of two or more kinds thereof.

Examples of the fluorinating agent may include 1,1,2,2-tetrafluoroethyl diethylamine, 2-chloro-1,1,2-trifluoroethyl diethylamine, trifluorodiphenylphospholane, difluorotriphenylphospholane, fluoroformic acid esters, sulfur tetrafluoride, potassium fluoride, potassium hydrogen fluoride, cesium fluoride, rubidium fluoride, sodium fluoride, lithium fluoride, antimony (III) fluoride, antimony (V) fluoride, zinc fluoride, cobalt fluoride, lead fluoride, copper fluoride, mercury (II) fluoride, silver fluoride, silver fluoroborate, thallium (I) fluoride, molybdenum (VI) fluoride, arsenic (III) fluoride, bromine fluoride, selenium tetrafluoride, tris(dimethylamino)sulfonium difluorotrimethylsilicate, sodium hexafluorosilicate, quaternary ammonium fluorides, (2-chloroethyl) diethylamine, diethylaminosulfur trifluoride, morpholinosulfur trifluoride, silicon tetrafluoride, hydrogen fluoride, hydrofluoric acid, hydrogen fluoride-pyridine complex, hydrogen fluoride-triethylamine complex, hydrogen fluoride salts, bis(2-methoxyethyl)amino sulfurtrifluoride, 2,2-difluoro-1,3-dimethyl-2-imidazolidinone, iodine pentafluoride, tris(diethylamino)phosphonium 2,2,3,3,4,4-hexafluorocyclobutanilide, triethylammonium hexafluorocylcobutanilide, hexafluoropropene, and the like. These fluorinating agents may be used alone or as a mixture of two or more kinds thereof.

The fluorinating agent may be appropriately selected and used as a solvent, in the range of 1-fold molar equivalent to 10-fold molar equivalents with respect to the nitro aromatic carboxamide derivative represented by Formula (A20).

Additives may be used, and examples thereof may include crown ethers such as 18-crown-6 and the like, phase transfer catalysts such as a tetraphenylphosphonium salt and the like, inorganic salts such as calcium fluoride, calcium chloride, and the like, metal oxides such as mercury oxide and the like, ion exchange resins, and the like. These additives may not only be added to the reaction system but also used as a pretreating agent for the fluorinating agent.

The reaction temperature may be appropriately selected within the range from −80° C. to the reflux temperature of the solvent used, and the reaction time may be appropriately selected within the range from several minutes to 96 hours.

Preparation Method 4

4-(i): Formula (A22)+Formula (A16)→Formula (A23)

A carboxylic acid having an acylamino group represented by Formula (A23) can be prepared by reacting a compound represented by Formula (A22) as a starting material with a compound represented by Formula (A16) according to the conditions described in 1-(i).

4-(ii): Formula (A23)+Formula (A24)→Formula (A25)

The compound represented by Formula (A25) can be prepared by reacting the amide compound represented by Formula (A23) with the compound having a leaving group such as a halogen and the like, represented by Formula (A24) in a solvent or without a solvent. In the present step, a suitable base or solvent can be used, and as the base or solvent, those exemplified in 1-(i) can be used. Examples of the reaction temperature, the reaction time, and the like may include those exemplified in l-(i).

4-(iii): Formula (A25)→Formula (A26)

The compound represented by Formula (A26) can be prepared from the compound represented by Formula (A25) through hydrolysis conducted by a general technique or a method using a Pd catalyst. In the hydrolysis, the compound can be obtained by base hydrolysis using one equivalent to 5-fold molar amount of aqueous or alcoholic lithium hydroxide, sodium hydroxide, or potassium hydroxide in a single solvent of methanol, ethanol, tetrahydrofuran, or dioxane, or a combination thereof. Also in a non-aqueous solvent such as toluene and xylene, hydrolysis can be conducted with the combination of a base such as aqueous sodium hydroxide, potassium hydroxide, or lithium hydroxide and a phase-transfer catalyst such as tetrabutylammonium bromide, benzyltriethylammonium chloride, or crown ether. Alternatively, acid hydrolysis can be conducted with inorganic acid such as hydrochloric acid and sulfuric acid, organic acid such as acetic acid and trifluoroacetic acid, or strongly acidic resin.

The reaction temperature may be appropriately selected in the range from −20° C. to the reflux temperature of the solvent to be used. And the reaction time may be appropriately selected in the range from a few minutes to 96 hours.

The method using Pd can include, for example, the method described in Tetrahedron Letters p. 4371 (1987). The conditions such as the solvent and the reaction temperature are not limited to those described in the reference.

4-(iv): Formula (A26)→Formula (A27)

The compound represented by Formula (A27) can be prepared according to the known routine procedure in which the compound represented by Formula (A26) is reacted with thionyl chloride, oxalyl chloride, phosgene, phosphorus oxychloride, phosphorus pentachloride, phosphorous trichloride, thionyl bromide, phosphorus tribromide, diethylaminosulfur trifluoride, or the like.

4-(v): Formula (A27)+Formula (A12)→Formula (A1)

The compound represented by Formula (A1) can be produced by reacting the compound represented by Formula (A27) with the compound represented by Formula (A12) according to the conditions described in 1-(i).

4-(vi): Formula (A26)+Formula (A12)→Formula (A1)

The amide derivative represented by Formula (A1) can be produced by reacting the compound represented by Formula (A26) with the compound represented by Formula (A 12) according to the conditions of the method in which a condensing agent is used or the mixed anhydride method both described in 1-(i).

Production Method 5

5-(i): Formula (A28)→Formula (A29)

The compound represented by Formula (A29) can be produced by fluorinating the compound represented by Formula (A28) according to the conditions described in 3-(ii).

5-(ii): Formula (A29)→Formula (A30)

The compound represented by Formula (A30) can be produced by reducing the compound represented by Formula (A29) according to the conditions described in 1-(ii).

In all of the preparation methods as described above, a desired product may be isolated from the reaction system after the reaction is completed according to a general method, but if required, purification can be carried out by operations such as recrystallization, column chromatography, distillation, and the like. In addition, the desired product can be also provided to the subsequent reaction process without being separated from the reaction system.

Hereinbelow, examples of the representative compounds of the amide derivative represented by Formula (A1) as an active ingredient for the composition for exterminating animal parasites according to the present invention will be given in Table A1 and Table A2 below, but the present invention is not limited thereto.

In addition, in the tables, “Me” represents a methyl group, “n-Pr” represents a normal propyl group, “CF3” represents a trifluoromethyl group, “C2F5” represents a pentafluoroethyl group, “n-C3F7” represents a heptafluoronormalpropyl group, “H” represents a hydrogen atom, “F” represents a fluorine atom, “Cl” represents a chlorine atom, “Br” represents a bromine atom, and “I” represents an iodine atom, respectively.

TABLE A1

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

6-940

phenyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

6-948

phenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

6-952

2-chlorophenyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

Cl

6-956

3-bromophenyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

Br

6-970

2,6-difluorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

I

6-1104

phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1105

2-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1106

3-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1107

4-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1126

2,6-difluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

6-1260

phenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1261

2-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1262

3-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1263

4-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1282

2,6-difluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

6-1416

phenyl

H

H

F

H

H

H

F

H

heptafluoroisopropyl

H

CF3

6-1417

phenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1418

2-fluorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1422

3-chlorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1426

4-bromophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1439

2,6-difluorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1440

3,4-dichlorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1441

2,4-dichlorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

6-1442

2-chloro-4-fluorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1445

2-bromo-4-chlorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

6-1446

2-bromo-4-fluorophenyl

H

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

6-1574

phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1575

2-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1576

3-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1577

4-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1578

2-chlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1579

3-chlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1580

4-chlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1581

2-bromophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1582

3-bromophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1583

4-bromophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1584

2-iodophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1585

3-iodophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1586

4-iodophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1596

2,6-difluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1597

3,4-dichlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1598

2,4-dichlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1599

2-chloro-4-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1600

2-chloro-4,5-difluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1601

4-bromo-2-chlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1602

2-bromo-4-chlorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1603

2-bromo-4-fluorophenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

6-1730

phenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1731

2-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1732

3-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1733

4-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1734

2-chlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1735

3-chlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1736

4-chlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1737

2-bromophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1738

3-bromophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1739

4-bromophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1740

2-iodophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1741

3-iodophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1742

4-iodophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1752

2,6-difluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1753

3,4-dichlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1754

2,4-dichlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1755

2-chloro-4-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1756

2-chloro-4,5-difluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1757

4-bromo-2-chlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1758

2-bromo-4-chlorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-1759

2-bromo-4-fluorophenyl

H

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

6-2110

phenyl

H

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

6-5902

phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Cl

6-5910

phenyl

H

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

C2F5

TABLE A2

compound

number

Q1

R1

R2

X1

X2

X3

X4

Y1

Y2

Y3

Y4

Y5

7-940

phenyl

Me

H

F

H

H

H

F

H

heptafluoroisopropyl

H

F

7-948

phenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

Cl

7-1104

phenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1105

2-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1106

3-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1107

4-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1126

2,6-difluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

Br

7-1260

phenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1261

2-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1262

3-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1263

4-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1282

2,6-difluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

I

7-1416

phenyl

Me

H

F

H

H

H

F

H

heptafluoroisopropyl

H

CF3

7-1417

phenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-1441

2,4-dichlorophenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

C2F5

7-1442

2-chloro-4-fluorophenyl

n-Pr

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

CF3

7-1445

2-bromo-4-chlorophenyl

Me

H

F

H

H

H

Cl

H

heptafluoroisopropyl

H

n-C3F7

7-1574

phenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1575

2-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1576

3-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1577

4-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1578

2-chlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1579

3-chlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1580

4-chlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1581

2-bromophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1582

3-bromophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1583

4-bromophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1584

2-iodophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1585

3-iodophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1586

4-iodophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1596

2,6-difluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1597

3,4-dichlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1598

2,4-dichlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1599

2-chloro-4-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1600

2-chloro-4,5-difluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1601

4-bromo-2-chlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1602

2-bromo-4-chlorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1603

2-bromo-4-fluorophenyl

Me

H

F

H

H

H

Br

H

heptafluoroisopropyl

H

CF3

7-1730

phenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1731

2-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1732

3-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1733

4-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1734

2-chlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1735

3-chlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1736

4-chlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1737

2-bromophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1738

3-bromophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1739

4-bromophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1740

2-iodophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1741

3-iodophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1742

4-iodophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1752

2,6-difluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1753

3,4-dichlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1754

2,4-dichlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1755

2-chloro-4-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1756

2-chloro-4,5-difluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1757

4-bromo-2-chlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1758

2-bromo-4-chlorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-1759

2-bromo-4-fluorophenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

CF3

7-2110

phenyl

Me

H

F

H

H

H

CF3

H

heptafluoroisopropyl

H

CF3

7-5902

phenyl

Me

H

F

H

H

H

I

H

heptafluoroisopropyl

H

Br

Hereinbelow, Table A3 shows the physical properties of the representative compounds of the amide derivative according to the present invention. The ¹H-NMR chemical shift values shown therein are based on tetramethylsilane as an internal standard substance unless specified otherwise.

TABLE A3
compound
number 1H-NMR (CDCl3, ppm)
6-1104 δ 7.40 (1H, t, J = 7.8 Hz), 7.53-7.64 (3H, m), 7.89 (2H, s), 7.90-7.95 (3H, m), 8.11-8.14 (2H, m),
       8.69-8.70 (1H, m).
6-1105 δ 7.22-7.26 (1H, m), 7.35-7.41 (2H, m), 7.58 (1H, d, J = 8.0 Hz), 7.88-7.92 (3H, m), 8.15-8.25 (2H, m),
       8.74-8.75 (2H, m).
6-1106 δ 7.35-7.34 (1H, m), 7.417.42 (1H, m), 7.53-7.54 (1H, m), 7.67-7.68 (2H, m), 7.89-7.90 (3H, m),
       8.09-8.10 (2H, m), 8.66-8.68 (1H, m).
6-1107 δ 7.21-7.26 (2H, m), 7.39-7.41 (1H, m), 7.89-7.96 (4H, m), 8.05-8.13 (3H, m), 8.70-8.72 (1H, m).
6-1126 δ 7.05-7.09 (2H, m), 7.38-7.42 (1H, m), 7.49-7.50 (1H, m), 7.88-7.99 (4H, m), 8.09-8.12 (1H, m),
       8.71-8.72 (1H, m).
6-1260 δ 7.39 (1H, t, J = 7.8 Hz), 7.52-7.57 (4H, m), 7.60-7.63 (2H, m), 7.93-7.94 (4H, m), 8.70 (1H, t, J = 6.3 Hz).
6-1261 δ 7.22-7.28 (1H, m), 7.35-7.42 (2H, m), 7.59-7.61 (1H, m), 7.94-7.95 (1H, m), 8.12 (2H, s), 8.15-8.25 (2H,
       m), 8.78 (1H, t, J = 1.5 Hz), 9.00 (1H, d, J = 7.8 Hz).
6-1262 δ 7.30-7.33 (1H, m), 7.40-7.44 (1H, m), 7.52-7.55 (2H, m), 7.64-7.70 (3H, m), 7.95-7.96 (1H, m),
       8.09-8.13 (2H, m), 8.67-8.68 (1H, m).
6-1263 δ 7.20-7.26 (3H, m), 7.38-7.42 (1H, m), 7.91-7.98 (3H, m), 8.07-8.12 (3H, m), 8.63-8.67 (1H, m).
6-1282 δ 7.06 (2H, t, J = 8.3 Hz), 7.38-7.42 (1H, m), 7.47-7.52 (1H, m), 7.93-7.97 (1H, m), 8.01 (1H, s),
       8.11-8.13 (3H, m), 8.68-8.72 (1H, m).
6-1574 δ 7.37-7.41 (1H, m), 7.53-7.64 (3H, m), 7.86-7.94 (4H, m), 8.13-8.22 (3H, m), 8.67-8.72 (1H, m).
6-1575 δ 7.22-7.27 (1H, m), 7.35-7.41 (2H, m), 7.57-7.60 (1H, m), 7.88-7.93 (2H, m), 8.16 (1H, s), 8.20-8.25 (2H,
       m), 8.74-8.75 (1H, m), 8.77-9.00 (1H, m).
6-1576 δ 7.27-7.37 (2H, m), 7.48-7.53 (1H, m), 7.72-7.80 (3H, m), 7.92 (1H, s), 8.15 (1H, s), 8.27-8.31 (1H, m),
       9.16 (1H, s), 9.35 (1H, d, J = 7.3 Hz).
6-1577 δ 7.20-7.23 (3H, m), 7.24-7.26 (1H, m), 7.39-7.40 (3H, m), 7.86-7.97 (1H, m), 8.06 (1H, d, J = 2.4 Hz),
       8.16-8.20 (1H, m), 8.62-8.67 (1H, m).
6-1596 δ 7.00-7.09 (2H, m), 7.40-7.41 (1H, m), 7.46-7.53 (1H, m), 7.89-7.92 (2H, m), 8.00 (1H, s),
       8.16-8.19 (2H, m), 8.71-8.72 (1H, m).
6-1730 δ 7.40 (1H, t, J = 7.8 Hz), 7.53-7.64 (3H, m), 7.87-7.95 (4H, m), 8.14 (1H, s), 8.22 (1H, d, J = 12.7 Hz),
       8.37 (1H, s), 8.71-8.72 (1H, m).
6-1731 δ 7.22-7.25 (1H, m), 7.35-7.37 (2H, m), 7.58-7.60 (1H, m), 7.90 (1H, t, J = 8.6 Hz), 7.96 (1H, s), 8.22 (1H, t, J = 8.8 Hz),
       8.29-8.32 (1H, d, J = 12.4 Hz), 8.37 (1H, s), 8.73 (1H, m), 8.94 (1H, s).
6-1732 δ 7.32-7.33 (1H, m), 7.37 (1H, t, J = 8.0 Hz), 7.52-7.54 (1H, m), 7.64-7.70 (2H, m), 7.90 (1H, t, J = 6.4 Hz),
       7.96 (1H, s), 8.10 (1H, s), 8.23 (1H, d, J = 12.0 Hz), 8.37 (1H, s), 8.65 (1H, t, J = 8.0 Hz).
6-1733 δ 7.19-7.25 (2H, m), 7.35 (1H, t, J = 7.8 Hz), 7.87-7.97 (4H, m), 8.08 (1H, s), 8.25 (1H, d, J = 12.0 Hz), 8.37 (1H,
       s), 8.65 (1H, t, J = 8.0 Hz).
6-1734 δ 7.43-7.52 (5H, m), 7.87-7.95 (3H, m), 8.22 (1H, d, J = 10.0 Hz), 8.35 (1H, d, J = 8.2 Hz), 8.74 (1H, t, J = 8.4 Hz).
6-2110 δ 7.36-7.40 (1H, m), 7.53-7.64 (3H, m), 7.84-7.97 (1H, m), 7.92-7.94 (2H, m), 8.04-8.07 (1H, m),
       8.08-8.13 (1H, m), 8.20 (2H, s), 8.68-8.72 (1H, m).
6-5902 (DMSO-d6) δ 7.39 (1H, t, J = 7.8 Hz), 7.52-7.64 (4H, m), 7.81 (1H, t, J = 6.8 Hz), 7.95 (1H, s), 7.98-8.01 (3H,
       m), 10.29 (1H, s), 10.68 (1H, s).
6-5910 δ 7.39 (1H, t, J = 8.3 Hz), 7.53-7.64 (3H, m), 7.88-7.94 (4H, m), 8.13 (1H, broad-s), 8.19 (1H, broad-s),
       8.24 (1H, d, J = 13.2 Hz), 8.70-8.72 (1H, m).
7-948  δ 3.49 (3H, s), 7.23-7.52 (8H, m), 7.66 (2H, s), 8.00 (1H, t, J = 6.8 Hz).
7-1104 δ 3.51 (3H, s), 7.22-7.44 (7H, m), 7.86 (2H, s), 8.00-8.03 (2H, m).
7-1105 δ 3.52 (3H, s), 6.82 (1H, t, J = 8.8 Hz), 7.06-7.08 (1H, m), 7.18-7.24 (2H, m), 7.40-7.44 (2H, m), 7.87 (3H, s),
       8.01-8.05 (1H, m).
7-1106 δ 3.50 (3H, s), 7.00-7.23 (4H, m), 7.29-7.31 (1H, m), 7.45 (1H, s), 7.87 (3H, s), 8.03-8.07 (1H, m).
7-1107 δ 3.49 (3H, s), 6.91-6.93 (2H, m), 7.28-7.44 (4H, m), 7.86 (2H, s), 8.00-8.10 (2H, m).
7-1126 δ 3.49 (3H, s), 6.72-6.76 (2H, m), 7.16-7.23 (2H, m), 7.43-7.50 (1H, m), 7.88 (2H, s), 8.02-8.06 (1H, m),
       8.13-8.17 (1H, m).
7-1260 δ 4.09 (3H, s), 7.21-7.49 (7H, m), 7.99-8.08 (4H, m).
7-1261 δ 3.53 (3H, s), 6.79-6.83 (1H, m), 7.03-7.07 (1H, m), 7.19-7.23 (2H, m), 7.42-7.43 (2H, m), 8.01-8.10 (4H,
       m).
7-1417 δ 3.49 (3H, s), 7.23-7.26 (3H, m), 7.27-7.33 (3H, m), 7.52-7.53 (1H, m), 7.85 (1H, s), 7.96-8.06 (3H, m).
7-1574 δ 3.50 (3H, s), 6.99-7.33 (6H, m), 7.43-7.45 (1H, m), 7.90 (1H, s), 7.97-8.06 (2H, m), 8.13 (1H, s).
7-1575 δ 3.52 (3H, s), 6.82-6.83 (1H, m), 7.06-7.07 (1H, m), 7.19-7.26 (2H, m), 7.39-7.46 (2H, m), 7.91 (1H, s),
       7.99-8.01 (1H, m), 8.07-8.14 (2H, m).
7-1576 δ 3.50 (3H, s), 7.01-7.17 (4H, m), 7.27-7.31 (1H, m), 7.46-7.52 (1H, m), 7.91 (1H, s), 8.01-8.05 (2H, m),
       8.13 (1H, s).
7-1577 δ 3.50 (3H, s), 6.90-6.94 (2H, m), 7.26-7.35 (3H, m), 7.45-7.46 (1H, m), 7.90 (1H, s), 8.00-8.07 (2H, m),
       8.13 (1H, s).
7-1596 δ 3.54 (3H, s), 6.75 (2H, broad-s), 7.17-7.26 (2H, m), 7.50-7.51 (1H, m), 7.92 (1H, s), 8.01-8.05 (1H, m),
       8.14-8.20 (2H, m).
7-1730 δ 3.51 (3H, s), 7.21-7.23 (2H, m), 7.27-7.33 (4H, m), 7.44-7.46 (1H, m), 7.92 (1H, s), 8.00 (1H, t, J = 6.3 Hz),
       8.08-8.09 (1H, m), 8.33 (1H, s).
7-1731 δ 3.51 (3H, s), 6.79-6.83 (1H, m), 7.05 (1H, t, J = 7.6 Hz), 7.18-7.46 (4H, m), 7.94-8.00 (2H, m), 8.20 (1H, d, J = 12.4 Hz),
       8.34 (1H, s).
7-1732 δ 3.50 (3H, s), 7.00-7.18 (4H, m), 7.27-7.31 (1H, m), 7.45-7.48 (1H, m), 7.93 (1H, s), 8.01-8.03 (1H, m),
       8.12 (1H, broad-s), 8.34 (1H, s).
7-1733 δ 3.50 (3H, s), 6.91 (2H, s), 6.93-7.35 (3H, m), 7.47 (1H, t, J = 7.0 Hz), 7.93 (1H, s), 8.01-8.10 (1H, m), 8.13 (1H,
       broad-s), 8.34 (1H, s).
7-1752 δ 3.54 (3H, s), 6.74 (2H, s), 7.16-7.24 (2H, m), 7.50 (1H, t, J = 7.4 Hz), 7.94 (1H, s), 8.01-8.05 (1H, m), 8.25 (1H,
       broad-s), 8.35 (1H, s).
7-5902 δ 3.51 (3H, s), 7.00-7.52 (7H, m), 7.88 (1H, d, J = 1.5 Hz), 8.01-8.06 (3H, m).

In particular, for example, animal parasites that can be exterminated by the composition for exterminating animal parasites according to the invention include the followings, although the invention is not limited thereto. The ectoparasites include Siphonaptera pests such as Ctenocephalides felis, Ctenocephalides canis, Xenopsylla cheopis, Echidnophaga gallinacea), and Pulex irritans;

acarine pests such as Haemaphyxalislongicornis, Haemaphysalis japonica, Rhipicephalus sanguineus, Boophilus microplus, Dermacentor recticulatus, Dermacentor taiwanensis, Haemaphysalis flava, Ixodes ovatus, Ixodes persulcatus, Amblyomma americanum, Amblyomma maculatum, Dermacentor andersoni, Dermacentor occidentalis, Dermacentor variabilis, Haemaphysalis campanulata, Haemaphysalis megaspinosa, Ixodes nipponensis, Ixodes pacifcus, Ixodes ricinus, and Ixodes scapularisand;

dipterous pests such as Musca hervei, Musca bezzii, Haematobia irritans, Simulium iwatens, Culicoides oxystoma, Tabanus chrysurus, Culex pipiens, and Aedes albopictus;

Phthiraptera pests such as Haematopinus eurysternus and Damalinia ovis; and the like.

The endoparasites include:

Protozoa such as Rhizopoda including Endamoeba histolytica, Mastigophora including Leishmania and Tichomonas, Sporozoea including Plasmodium and Toxoplasma, and Ciliophora including Balantidium coli;

helminths such as Nematoda including Ascaris lumbricoides and Ancylostoma, Acannthocephala including Macracanthorhynchus hirudinaceus, Nematomorpha including Paragordius tricuspidatus, Tematoda including Clonorchis sinensis, and Cestoda including Taenia saginata;

nematodes such as Ascaris, Toxocara, Toxascaris, Parascaris, Ascaridia, Heterakis, Oxyuris, Capillaria, Trichinella, Strongylus, Triodontophorus, Trichonema, Stephanurus, Desophagostomum, Chabertia, Syngamus, Ancylostoma, Uncinaria, Necator, Bunostomum, Trichostrongylus, Cooperia, Nematodirus, Haemonchus, Ostertagia, Dictyocaulus, Metastrongylus, Dirofilaria, Parafilaria, Setaria, Onchocerca, Habronema, Arduenna, and Acuaria;

cestodes such as Diphyllobothrium, Anoplocephara, Moniezia, Dipylidium, Taenia, Dithyridium, Raillietina, and Echinococcus;

flukes such as Schistosoma, Paramphistomum, and Fasciola; and the like.

In the invention, said animal parasites are preferably ectoparasites from the viewpoint of parasiticidal activity, and they are preferably at least one of Siphonaptera pests (especially preferably Ctenocephalides felis) and Acarina pests (especially preferably Haemaphyxalislongicornis, Rhipicephalus sanguineus, and Boophilus microplus).

The animals to which the composition for exterminating animal parasites according to the invention can be applied include domestic animals such as human, horses, cows, pigs, sheep, goats, rabbits, camels, buffalos, deer, minks, and chinchillas; fowls such as chickens, ducks, geese, and turkeys; pets such as dogs, cats, small birds, and monkeys; laboratory animals such as rats, mice, golden hamsters, and guinea pigs; and the like, although the invention is not limited thereto.

The composition for exterminating animal parasites according to the invention can be used as a parasiticide by any of the methods normally used, with no particular restriction.

In particular, for example, the composition may be dissolved, suspended, mixed, impregnated, adsorbed, or adhered on suitable solid and/or liquid carriers according to a formulation generally used, and, if required, together with adjuvant in a suitable proportion. And the composition may be prepared into an appropriate form in accordance with the intended use.

The solid or liquid carrier for use in the invention may be those normally used in agents for animals. From the viewpoint of easiness of treatment on the target animals, it is preferable to use a liquid carrier. The liquid carrier includes, for example, alcohol such as methyl alcohol, ethyl alcohol, isopropyl alcohol, tertiary butyl alcohol, and benzyl alcohol; propylene carbonate; N-methyl-2-pyrrolidone; water, and the like. As the adjuvant, surfactant, antioxidant, emulsifier, and the like can be used. The adjuvant can include, for example, surfactant such as polyoxyethylene alkylaryl ether, polyoxyethylene sorbitan monolaurate, alkyl allyl sorbitan monolaurate, alkylbenzenesulfonate, alkylnaphthalene sulfonic acid, ligninsulfonic acid salts, higher alcohol sulfate salts, glycol monoalkyl ethers, and glycols; emulsifier such as sorbitan monooleate, sorbitan monolaurate, caprylic acid monoglyceride, capric acid monoglyceride, isostearic acid monoglyceride, and propylene glycol monocaprylate; and antioxidant such as BHA and BHT.

The composition for exterminating animal parasites according to the invention may be administered orally or parenterally to an animal.

If the composition for exterminating animal parasites according to the invention is administered orally, the composition may be in the form of capsules, tablets, pills, powders, granules, fine granules, syrups, enteric agents, suspensions, paste, or beverage or feeds mixed with the drug.

If the composition for exterminating animal parasites according to the invention is administered parenterally, the composition may be in the form of injectables, drips, suppositories, emulsions, suspensions, drops, ointments, creams, solutions, lotions, sprays, aerosols, cataplasms, and tapes.

The method for administration includes the spot-on method in which drops are dropped on the skin of the back shoulder region and the like of the target animal to exterminate ectoparasites; local methods such as the pour-on method in which a liquid agent is applied along the back center line of the target animal to allow the applied agent to diffuse on the body surface, resulting in control of ectoparasites; the methods in which the agent is released from a collar containing the agent; the methods in which a liquid agent, ointment, or the like is directly applied to the body surface; the methods in which an aerosol or the like is applied with a spray or the like; the methods in which an injectable is injected intramuscularly, subcutaneously, or the like; and rectal administration with a suppository.

In addition to extermination of endoparasites and exoparasites, the composition for exterminating animal parasites according to the invention also can prophylactically prevent parasitic infections by applying it to the environments which are to be the infection routes. For example, the composition can prevent soil infections from soils of upland fields and parks; percutaneous infections from aqueous systems such as river, lake, wetland, and paddy field; oral infections from excrements of animals such as dogs and cats; and oral infections from raw meats of sea water fish, fresh water fish, Crustaceae, shellfish, domestic animals, and the like; and infections from mosquitoes, horseflies, flies, cockroaches, ticks, fleas, lice, assassin bugs, chiggers, etc.; and the like.

If the composition for exterminating animal parasites according to the invention is used to exterminate parasites in the animals that are mammals or birds, the optimal dosage varies depending on whether it is used for therapeutic purposes or for preventive purposes, and also varies with the type of infected parasites, the type and extent of infection, dosage form, etc. But generally, in case of oral administration, the dosage is in the range from about 0.0001 to 10,000 mg per kilogram of body weight per day. In case of parenteral administration, the dosage is in the range from about 0.0001 to 10,000 mg per kilogram of body weight per day, and the composition is administered in single or in divided doses.

The concentration of the active ingredient in the composition for exterminating animal parasites according to the invention is typically from 0.0001 to 100% by weight, preferably from 0.001 to 99% by weight, and more preferably from 0.005 to 80% by weight. In general, the parasiticides may be provided as a high-concentrated composition to be diluted to the appropriate concentration prior to use.

In addition to the amide derivatives represented by Formula (1) according to the invention, the composition for exterminating animal parasites according to the invention can further contain other insecticidal components that are generally known. The other insecticidal components can include, for example, pyrethroid compounds such as permethrin, d-phenothrin, allethrin, pyrethrum, prallethrin, cyphenothrin, cyfluthrin, fenvalerate, fenpropathrin, transfluthrin, metofluthrin, resmethrin, cypermethrin, alpha-cypermethrin, bifenthrin, deltamethrin, lambda-cyhalothrin, d,d-trans-cyphenothrin, tetramethrin, and ethofenprox; organic phosphorus compounds such as dichlorvos, tetrachlorvinphos, fenthion, chlorpyrifos, chlorpyrifos-methyl, malathion, pirimiphos-methyl, fenitrothion, and diazinon; N-phenylpyrazole compounds such as fipronil; carbamate compounds such as propoxur, carbaryl, metoxadiazone, and fenocarb; neonicotinoid compounds such as imidacloprid, clothianidin, thiamethoxam, acetamiprid, nitenpyram, and dinotefuran; growth inhibitors for insect such as methoprene, pyriproxyfen, lufenuron, fenoxycarb, triflumuron, and chromafenozide; milbemycin oxime; milbemectin; lepimectin; abamectin; ivermectin; selamectin; spinosad; rotenone; and the like.

The disclosure of Japanese Patent Application JP 2010-019747 is incorporated herein in its entirety.

All publications, patent applications, and technical specifications cited herein are incorporated herein by reference to the same extent as if each individual publication, patent application, and technical specification were specifically and individually indicated to be incorporated by reference.

EXAMPLES

Representative Examples of the present invention will be described with reference to the following Examples, but the present invention is not limited thereto. In the present Examples, DMF means N,N-dimethyl formamide, THF means tetrahydrofuran, IPE means isopropyl ether, and DMI means 1,3-dimethyl-2-imidazolidinone. Furthermore, “%” is based on mass unless specified otherwise.

Example 1

Preparation of N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide (Compound No. 7-1574)

1-1>

Preparation of 4-(heptafluoropropan-2-yl)-2-(trifluoromethyl)aniline

100 g (0.608 mol) of 2-(trifluoromethyl)aniline, 131 g (0.639 mol) of 85% sodium hydrosulfite, and 20.9 g (0.0608 mol) of tetrabutylammonium hydrogen sulfate were charged to a mixed solution of 1500 ml of ethyl acetate and 1500 ml of water, and 53.9 g (0.639 mol) of sodium hydrogen carbonate was added thereto. 198 g (0.669 mol) of heptafluoroisopropyl iodide was added dropwise thereto at room temperature, followed by stirring at room temperature for 6 hours. After the liquid separation, the solvent of the organic layer was evaporated under reduced pressure, and 500 ml of ethyl acetate was charged thereto. 160 g (0.608 mol) of a 4 M hydrogen chloride/ethyl acetate solution was added dropwise thereto, followed by stirring at room temperature for 30 minutes, and then stirring at 5° C. for 1 hour. After the filtration, the filtrate was washed with water and a saturated aqueous sodium hydrogen carbonate in this order, and then dried over anhydrous magnesium sulfate, and the solvent was evaporated under reduced pressure. The obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=10:1) to prepare 60.0 g (yield 30%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 4.49 (2H, broad-s), 6.81 (1H, d, J=8.3 Hz), 7.48 (1H, d, J=8.3 Hz), 7.64 (1H, s).

<1-2>

Preparation of 2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)aniline

100 g (0.273 mol) of 4-(heptafluoropropan-2-yl)-2-(trifluoromethyl)aniline was charged to 500 ml of DMF, and 52.1 g (0.287 mol) of N-bromosuccinimide was charged in separate portions thereto over 30 minutes. After stirring at 60° C. for 2 hours, and then cooling to room temperature, the mixture was discharged to 2000 ml of water. The mixture was extracted with ethyl acetate, then washed with saturated brine, and dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=20:1) to prepare 89.0 g (yield 80%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 5.03 (2H, broad-s), 7.61 (1H, s), 7.79 (1H, s).

<1-3>

Preparation of N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-chloro-3-nitrobenzamide

3.60 g (8.82 mmol) of 2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)aniline was charged to 20 ml of anhydrous THF, and cooled to −70° C. under a nitrogen atmosphere. 4.85 ml (9.70 mmol) of a 2.0 M lithium diisopropyl amide hexane solution was added dropwise thereto, then 2.34 g (10.7 mmol) of acid chloride which was prepared from 2-chloro-3-nitrobenzoic acid and thionyl chloride was dissolved in 5 ml of anhydrous TIF, and was added dropwise thereto, followed by stirring at −70° C. for 30 minutes and then stirring at room temperature for 30 minutes. The mixture was discharged to an aqueous ammonium chloride solution, then extracted with ethyl acetate, and dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=10:1→8:2→3:1) to prepare 1.76 g (yield: 34%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.61 (1H, t, J=7.8 Hz), 7.67 (1H, broad-s), 7.93-7.97 (3H, m), 8.18 (1H, broad-s).

<1-4>

Preparation of N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-nitrobenzamide

To a solution of N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-chloro-3-nitrobenzamide 4.89 g (8.27 mmol) in 50 ml of anhydrous DMF was added 2.40 g (41.3 mmol) of potassium fluoride (spray-dried product) under a flow of nitrogen, followed by stirring at 130° C. for 10 hours. Liquid separation was carried out by adding ethyl acetate, hexane, and water to the reaction mixture, and then the organic layer was washed with water and saturated brine, and dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=10:1) to prepare 0.940 g (yield 20%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.53 (1H, t, J=7.3 Hz), 7.93 (1H, broad-s), 8.17-8.18 (2H, m), 8.28-8.32 (1H, m), 8.44-8.48 (1H, m).

<1-5>

Preparation of 3-amino-N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluorobenzamide

0.940 g (1.63 mmol) of N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-nitrobenzamide and 0.960 g (5.05 mmol) of stannous chloride (anhydrous) were added to 10 ml of ethanol, and 1.02 ml (9.78 mmol) of concentrated hydrochloric acid was added thereto, followed by stirring at 60° C. for 4 hours. The reaction mixture was adjusted to pH 10 by the addition of an aqueous sodium hydroxide solution, and the precipitated insolubles were removed by filtration using Celite. The filtrate on Celite was washed with ethyl acetate. The filtrate was extracted with ethyl acetate, and the organic layer was washed with a 20% aqueous sodium hydroxide solution and saturated brine, and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=4:1) to prepare 0.930 g (yield 99%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 3.93 (2H, broad-s), 6.99-7.04 (1H, m), 7.11 (1H, t, J=7.8 Hz), 7.47-7.49 (1H, m), 7.91 (1H, s), 8.14 (1H, s), 8.28 (1H, d, J=14.6 Hz).

<1-6>

Preparation of N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(methylamino)benzamide

0.930 g (1.71 mmol) of 3-amino-N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluorobenzamide was added to 5 ml of concentrated sulfuric acid, and 10 ml of a 37% aqueous formaldehyde solution was charged dropwise thereto at 40° C. The reaction mixture was poured into ice-water, adjusted to pH 10 using an aqueous sodium hydroxide solution, and extracted with the addition of ethyl acetate. The organic layer was washed with a 20% aqueous sodium hydroxide solution and saturated brine, and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=8:1) to prepare 0.690 g (yield 72%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 2.94 (3H, s), 4.14 (1H, broad-s), 6.88-6.93 (1H, m), 7.18 (1H, t, J=7.8 Hz), 7.37-7.41 (1H, m), 7.90 (1H, s), 8.13 (1H, s), 8.27 (1H, d, J=14.6 Hz).

<1-7> Preparation of N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide (Compound No. 7-1574)

To a solution of 1.54 g (2.75 mmol) of N-(2-bromo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-2-fluoro-3-(methylamino)benzamide and 0.330 g (4.13 mmol) of pyridine in 5 ml of THF was added 0.460 g (3.30 mmol) of benzoyl chloride, followed by stirring at 60° C. for 5 hours. To the reaction mixture were added water and ethyl acetate, and the organic layer was washed with 1 M hydrochloric acid, a saturated aqueous sodium hydrogen carbonate solution, and saturated brine, and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=8:1), and the obtained solid was washed with IPE to prepare 1.45 g (yield 80%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 3.50 (3H, s), 6.99-7.33 (6H, m), 7.43-7.45 (1H, m), 7.90 (1H, s), 7.97-8.06 (2H, m), 8.13 (1H, s).

Example 2

Preparation of N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide (Compound No. 7-1104)

<2-1>

Preparation of 4-(heptafluoropropan-2-yl)aniline

100 g (1.02 mol) of aniline, 230 g (1.12 mol) of 85% sodium hydrosulfite, and 35.1 g (0.100 mol) of tetrabutylammonium hydrogen sulfate were charged to a mixed solution of 1500 ml of t-butyl methyl ether and 1500 ml of water, and 94.7 g (1.12 mol) of sodium hydrogen carbonate was added thereto. 350 g (1.12 mol) of heptafluoroisopropyl iodide was added dropwise thereto at room temperature, followed by stirring at room temperature for 6 hours. After the liquid separation, the organic layer was washed with 1 M hydrochloric acid, water, and a saturated aqueous sodium hydrogen carbonate solution, and then dried over anhydrous sodium sulfate. The solvent was evaporated under reduced pressure, and 500 ml of ethyl acetate was charged thereto. 255 g (1.02 mol) of a 4 M hydrogen chloride/ethyl acetate solution was added dropwise thereto, followed by stirring at room temperature for 30 minutes and at 5° C. for 1 hour. The precipitated solid was separated by filtration, and the solid was charged to 1000 ml of ethyl acetate, adjusted to pH 8 to 9 by the addition of 1000 ml of a saturated aqueous sodium hydrogen carbonate solution at 20° C. or lower, and subjected to liquid separation. The organic layer was dried over anhydrous sodium sulfate, and then the solvent was evaporated under reduced pressure to prepare 188 g (yield 71%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 3.92 (2H, broad-s), 6.69-6.74 (2H, m), 7.35 (2H, d, J-=9.3 Hz).

<2-2>

Preparation of 2,6-dibromo-4-(heptafluoropropan-2-yl)aniline

216 g (0.802 mol) of 4-(heptafluoropropan-2-yl)aniline was charged to 863 ml of DMF, followed by cooling to 5° C. 285 g (1.60 mol) of N-bromosuccinimide was charged in separate portions thereto over 1 hour. The mixture was stirred at room temperature for 1 hour and then stirred at 37° C. for 2 hours. The mixture was discharged to 2000 ml of water, extracted with 2000 ml of ethyl acetate, and washed with 1000 ml of saturated brine. After dried over anhydrous magnesium sulfate, the solvent was evaporated under reduced pressure. The obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=20:1) to prepare 304 g (yield 90%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 4.88 (2H, broad-s), 7.59 (2H, s).

<2-3>

Preparation of 2-chloro-N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-3-nitrobenzamide

According to the method of 1-3 of Example 1, a target compound was prepared from 2,6-dibromo-4-(heptafluoropropan-2-yl)aniline.

¹H-NMR (CDCl₃, ppm) δ 7.58 (1H, t, J=7.8 Hz), 7.66 (1H, broad-s), 7.90 (2H, s), 7.93 (1H, dd, J=1.5, 7.8 Hz), 7.98 (1H, d, J=7.8 Hz).

<2-4>

Preparation of N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide

According to the method of 1-4 of Example 1, a target compound was prepared from 2-chloro-N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 7.51-7.55 (1H, m), 7.90 (2H, s), 8.16 (1H, d, J=11.7 Hz), 8.27-8.31 (1H, m), 8.48 (1H, t, J=6.3 Hz).

<2-5>

Preparation of 3-amino-N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluorobenzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.93 (2H, broad-s), 6.99-7.04 (1H, m), 7.11 (1H, t, J=7.8 Hz), 7.47-7.49 (1H, m), 7.91 (1H, s), 8.14 (1H, s), 8.28 (1H, d, J=14.6 Hz).

<2-6>

Preparation of N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(methylamino)benzamide

According to the method of 1-6 of Example 1, a target compound was prepared from 3-amino-N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluorobenzamide.

¹H-NMR (CDCl₃, ppm) δ 2.94 (3H, d, J=5.6 HZ), 4.87-4.91 (1H, m), 6.91 (1H, t, J=7.9 Hz), 7.18 (1H, t, J=7.9 Hz), 7.41 (11H, t, J=7.1 Hz), 7.87 (2H, s), 8.20 (11H, d, J=13.5 Hz).

<2-7>

Preparation of N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(N-methylbenzamide)benzamide (Compound No. 7-1104)

According to the method of 1-7 of Example 1, a target compound was prepared from N-(2,6-dibromo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-(methylamino)benzamide and benzoyl chloride.

¹H-NMR (CDCl₃, ppm) δ 3.51 (3H, s), 7.22-7.44 (7H, m), 7.86 (2H, s), 8.00-8.03 (2H, m).

Example 3

Preparation of 3-benzamide-2-fluoro-N-(4-(heptafluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)benzamide (Compound No. 6-2110)

<3-1>

Preparation of 2,6-diiodo-4-(heptafluoropropan-2-yl)aniline

To a solution of 5.74 g (22.0 mmol) of 4-(heptafluoropropan-2-yl)aniline obtained in 2-1 of Example 2 in 50 ml of ethanol was added 2.16 g (22.0 mmol) of concentrated sulfuric acid at 5° C. The reaction mixture was warmed to room temperature, and 10.0 g (44.0 mmol) of N-iodosuccinimide was added thereto, followed by stirring for 3 hours. The reaction mixture was neutralized with a saturated aqueous sodium hydrogen carbonate solution. The precipitated crystals were filtered, washed with water, and then dried to prepare 9.00 g (yield 80%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 4.95 (2H, broad-s), 7.79 (2H, s).

<3-2>

Preparation of 2-chloro-N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-3-nitrobenzamide

To a solution of 40.0 g (78.0 mmol) of 2,6-diiodo-4-(heptafluoropropan-2-yl)aniline in 100 ml of DMI was added 20.6 g (94.0 mmol) of 2-chloro-3-nitrobenzoyl chloride, followed by stirring at 135° C. for 3 hours. After cooling to room temperature, the reaction mixture was poured into 1000 ml of water. After extraction with the addition of 1000 ml of ethyl acetate, the organic layer was washed with water and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was washed with hexane to prepare 56.2 g (yield 99%) of a target compound.

1H-NMR (CDCl₃, ppm) δ 7.58 (1H, t, J=8.3 Hz), 7.70 (1H, d, J=3.4 Hz), 7.93 (1H, dd, J=1.5, 6.3 Hz), 8.08-8.10 (1H, m), 8.13 (2H, s).

<3-3>

Preparation of N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide

According to the method of 1-4 of Example 1, a target compound was prepared from 2-chloro-N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 7.52-7.55 (1H, m), 8.12-8.18 (3H, m), 8.29-8.32 (1H, m), 8.48-8.51 (1H, m).

<3-4>

Preparation of 3-amino-N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluorobenzamide

According to the method of 1-5 of Example 1, a target compound was prepared from N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.93 (2H, broad-s), 6.99-7.04 (1H, m), 7.08 (1H, t, J=7.8 Hz), 7.39-7.43 (1H, m), 8.10 (2H, s), 8.72 (1H, d, J=11.2 Hz).

<3-5>

Preparation of 3-benzamide-N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluorobenzamide (Compound No. 6-1260)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluorobenzamide.

¹H-NMR (CDCl₃, ppm) δ 7.39 (1H, t, J=7.8 Hz), 7.52-7.57 (4H, m), 7.60-7.63 (2H, m), 7.93-7.94 (4H, m), 8.70 (1H, t, J=6.3 Hz).

<3-6>

Preparation of 3-benzamide-2-fluoro-N-(4-(heptafluoropropan-2-yl)-2,6-bis(trifluoromethyl)phenyl)benzamide (Compound No. 6-2110)

A solution of 1.95 g (2.59 mmol) of 3-benzamide-N-(2,6-diiodo-4-(heptafluoropropan-2-yl)phenyl)-2-fluorobenzamide, 0.10 g (0.520 mmol) of copper iodide, and 1.24 g (6.48 mmol) of methyl fluorosulfonyl difluoroacetate in 50 ml of DMF was stirred at 100° C. for 6 hours. The reaction mixture was cooled to room temperature, and then 10 ml of water and 100 ml of ethyl acetate were added thereto, followed by filtration through Celite. The organic layer of the liquid was washed with water and a saturated aqueous sodium hydrogen carbonate solution, and then dried over anhydrous magnesium sulfate. The solvent was evaporated under reduced pressure and the obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=1:1). The obtained solid was washed with hexane to prepare 0.840 g (yield 51%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 7.36-7.40 (1H, m), 7.53-7.64 (3H, m), 7.84-7.97 (1H, m), 7.92-7.94 (2H, m), 8.04-8.07 (1H, m), 8.08-8.13 (1H, m), 8.20 (2H, s), 8.68-8.72 (1H, m).

Example 4

Preparation of 2-fluoro-3-(4-fluoro-N-methylbenzamide)-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide (Compound No. 7-1733)

<4-1>

Preparation of 2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)aniline

To 1200 mL of ethanol was added 200 g (0.600 mol) of 4-(heptafluoropropan-2-yl)-2-(trifluoromethyl)aniline which was obtained in 1-1 of example 1, and 63.2 g (0.630 mol) of concentrated sulfuric acid and 155 g (0.660 mol) of N-iodosuccinimide were added thereto under ice-cooling, followed by stirring at room temperature for 1 hour and 30 minutes and at 40° C. for 4 hours. To the reaction solution was added a 4 M aqueous sodium hydroxide solution to neutralize the reaction solution, and then ethyl acetate was added thereto to extract the organic phase. The organic phase was washed with saturated brine, and dried over anhydrous magnesium sulfate, and then the solvent was evaporated under reduced pressure. The obtained residue was purified by silica gel column chromatography (eluent solvent; hexane:ethyl acetate=10:1) to prepare 216 g (yield 80%) of a target compound.

¹H-NMR (CDCl₃, ppm) δ 5.04 (2H, broad-s), 7.64 (1H, s), 7.99 (1H, s).

<4-2>

Preparation of 2-chloro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide

According to the method of 3-2 of Example 3, a target compound was prepared from 2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)aniline and 2-chloro-3-nitrobenzoyl chloride.

¹H-NMR (CDCl₃, ppm) δ 7.60 (1H, t, J=7.8 Hz), 7.76 (1H, s), 7.94 (1H, dd, J=1.5, 7.8 Hz), 7.97 (1H, s), 8.03 (1H, dd, J=1.5, 7.8 Hz), 8.39 (1H, s).

<4-3>

Preparation of 2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide

According to the method of 1-4 of Example 1, a target compound was prepared from 2-chloro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 7.51-7.55 (1H, m), 7.97 (1H, s), 8.23 (1H, d, J=12.2 Hz), 8.28-8.32 (1H, m), 8.37 (1H, s), 8.44-8.48 (1H, m).

<4-4>

Preparation of 3-amino-2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide

According to the method of 1-5 of Example 1, a target compound was prepared from 2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-nitrobenzamide.

¹H-NMR (CDCl₃, ppm) δ 3.92 (2H, broad-s), 7.02-7.04 (1H, m), 7.11 (1H, t, J=7.8 Hz), 7.47-7.52 (1H, m), 7.94 (1H, s), 8.30-8.35 (2H, m).

<4-5>

Preparation of 2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(methylamino)benzamide

According to the method of 1-6 of Example 1, a target compound was prepared from 3-amino-2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide.

¹H-NMR (CDCl₃, ppm) δ 2.95 (3H, s), 4.15 (1H, broad-s), 6.90 (1H, t, J=8.2 Hz), 7.19 (1H, t, J=7.8 Hz), 7.40 (1H, t, J=7.8 Hz), 7.92 (1H, s), 8.30 (1H, s), 8.34 (1H, s).

<4-6>

Preparation of 2-fluoro-3-(4-fluoro-N-methylbenzamide)-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide (Compound No. 7-1733)

According to the method of 1-7 of Example 1, a target compound was prepared from 2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(methylamino)benzamide and 4-fluorobenzoyl chloride.

¹H-NMR (CDCl₃, ppm) δ 3.50 (3H, s), 6.91 (2H, s), 6.93-7.35 (3H, m), 7.46 (1H, t, J=7.0 Hz), 7.93 (1H, s), 8.01-8.10 (1H, m), 8.13 (1H, broad-s), 8.34 (1H, s).

Example 5

Preparation of 2-fluoro-3-(3-fluoro-N-methylbenzamide)-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide (Compound No. 7-1732)

According to the method of 1-7 of Example 1, a target compound was prepared from 2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)-3-(methylamino)benzamide and 3-fluorobenzoyl chloride.

¹H-NMR (CDCl₃, ppm) δ 3.50 (3H, s), 6.91 (2H, s), 7.00-7.18 (4H, m), 7.27-7.31 (1H, m), 7.45-7.48 (1H, m), 7.93 (1H, s), 8.01-8.03 (1H, m), 8.12 (1H, broad-s), 8.34 (1H, s).

Example 6

Preparation of 2-fluoro-3-(4-fluorobenzamide)-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide (Compound No. 6-1733)

According to the method of 1-7 of Example 1, a target compound was prepared from 3-amino-2-fluoro-N-(2-iodo-4-(heptafluoropropan-2-yl)-6-(trifluoromethyl)phenyl)benzamide and 4-fluorobenzoyl chloride.

¹H-NMR (CDCl₃, ppm) δ 7.19-7.25 (2H, m), 7.35 (1H, t, J=7.8 Hz), 7.87-7.97 (4H, m), 8.08 (1H, s), 8.25 (1H, d, J=12.0 Hz), 8.37 (1H, s), 8.65 (1H, t, J=8.0 Hz).

Now, the representative examples of the formulations according to the invention will be shown, although the invention is not limited thereto. “Parts” in Formulation Examples indicates “parts by weight”.

Formulation Example 1 (Emulsion)

10 parts of Compound No. 7-1574 or 7-1733, 6 parts of Sol Pol 355S (surfactant available from Toho Chemical Industry Co.), and 84 parts of Solvesso 150 (available from ExxonMobil Chemical Co.) were homogeneously mixed with stirring to obtain as emulsion the composition for exterminating animal parasites.

Formulation Example 2 (Ointment)

1 part of Compound No. 7-1574 or 7-1733, 50 parts of white beeswax, and 49 parts of white petrolatum were thoroughly mixed to obtain as ointment the composition for exterminating animal parasites.

Formulation Example 3 (Tablets)

2 parts of Compound No. 7-1574 or 7-1733, 10 parts of vegetable oil (olive oil), 3 parts of crystalline cellulose, 20 parts of white carbon, and 65 parts of kaolin were thoroughly mixed and then compressed to obtain as tablets the composition for exterminating animal parasites.

Formulation Example 4 (Injectable)

10 parts of Compound No. 7-1574 or 7-1733, 10 parts of propylene glycol for food additives, 80 parts of vegetable oil (corn oil) were mixed to obtain as injectable the composition for exterminating animal parasites.

Formulation Example 5 (Solution)

5 parts of Compound No. 7-1574 or 7-1733, 20 parts of surfactant, and 75 parts of ion-exchanged water were thoroughly mixed to obtain as solution the composition for exterminating animal parasites.

Next, the utility of the composition of the invention as a parasiticide will be concretely explained in the following Test Examples, although the invention is not limited thereto.

Test Example 1

Insecticidal Test for Ctenocephalides Felis

0.5 ml of a solution of acetone, the active ingredient, prepared to the prescribed concentration was added dropwise to a glass tube with a flat bottom (internal diameter 2.6 cm, bottom area: 5.3 cm², height: 12 cm), and the solvent was evaporated at room temperature to form a dry film of the agent on the bottom surface. About 10 adults of Ctenocephalides Felis per glass tube were added, and the adults were contact-exposed to the test compound. After 24 hours of the exposure, the conditions of the adults were examined and classified into “alive” and “dead (including a moribund condition)” to determine the death rate (in triplicate). The results are shown in Table A4.

As the comparative compounds, the following Compounds (A), (B), and (C) disclosed in WO2009/080203, and fipronil were used.

	TABLE A4
	active ingredient	concentration	death rate
	(compound number)	(μg/ml)	(%)
	7-1574	0.1	100.0
	7-1733	0.1	100.0
	7-1732	0.1	76.7
	6-1733	0.1	70.0
	7-1104	0.1	73.3
	compound (A)	1.0	0.0
	compound (B)	1.0	3.2
	compound (C)	1.0	0.0
	fipronil	0.1	92.1
	only acetone	—	4.7

The amide derivatives of Compound No. 7-1574 and 7-1104 were found to be effective even in the examination after 12 hours of the exposure. In addition, they showed immediate effect as compared with the fipronil.

Test Example 2

Insecticidal Test for Haemaphyxalis longicornis

1 ml of a solution of acetone, the active ingredient, prepared to the prescribed concentration was added dropwise to filter paper inside a petri dish with a diameter of 9 cm, and the acetone was evaporated at room temperature. About 100 larvae of Haemaphyxalis longicornis per dish were added to the filter paper. The dish was covered by a polyethylene sheet, sealed with a rubber band, and placed in a dark place at a temperature of 25° C. and a relative humidity of 100% to expose the larvae to the test substance. After 24 hours of the exposure, the conditions of the larvae were examined and classified into “alive” and “dead (including a moribund condition)”. As a result, the amide derivatives according to the invention were found to be effective in killing Haemaphyxalis longicornis.

Test Example 3

Insecticidal Test for Ctenocephalides felis

0.96 ml of a solution of acetone, the active ingredient, prepared to the prescribed concentration was added dropwise to a glass tube with a flat bottom (internal diameter: 3.6 cm, height: 12 cm), and the solvent was evaporated at room temperature to form a dry film of the agent on the bottom surface. About 10 adults of Ctenocephalides felis per glass tube were added, and they were contact-exposed to the test compound. After 24 hours of the exposure, the conditions of the adults were examined and classified into “alive” and “dead (including a moribund condition)” to determine the death rate was determined (in triplicate). The results are shown in Table A5.

As the comparative compounds, the following Compounds (D) and (E) disclosed in WO2009/080203, and fipronil were used.

	TABLE A5
	active ingredient	concentration	death rate
	(compound number)	(μg/ml)	(%)
	7-1574	0.03	72.0
		0.1	98.9
	7-1733	0.03	21.1
		0.1	91.6
	componud (D)	0.3	22.0
		1	61.4
	compound (E)	1	0.0
	fipronil	0.03	70.0
		0.1	100.0
	only acetone	—	1.4

Test Example 4

Insecticidal Test for Rhipicephalus sanguineus

0.5 ml of a solution of acetone, the active ingredient, prepared to the prescribed dose was added dropwise into a glass petri dish with a diameter of 10 cm, and the acetone was evaporated at room temperature. About 10 adults of Rhipicephalus sanguineus per dish were added, and the dish was covered by another glass petri dish that was treated with the active ingredient in the same manner described above. After 18 hour exposure to the test substance, the adults were transferred into a glass petri dish that was not treated with the active ingredient. After 48 hours of the exposure, the conditions of the adults were examined and classified into “alive” and “dead (including a moribund condition)” to determine the death rate (in single). The results are shown in Table A6.

As the comparative compounds, said Compounds (B), (C), and (D), and the following Compound (F) disclosed in WO2009/080203, and fipronil were used.

	TABLE A6
	active ingredient	concentration	death rate
	(compound number)	(mg/m2)	(%)
	7-1574	0.0431	10.0
		0.0861	100.0
		0.172	100.0
	7-1733	0.0431	0.0
		0.0861	80.0
		0.172	100.0
	compound (B)	0.673	0.0
		2.69	20.0
		10.8	50.0
	compound (C)	0.673	0.0
		2.69	11.1
		10.8	10.0
	compound (D)	0.673	0.0
		2.69	10.0
		10.8	50.0
	compound (F)	0.673	0.0
		2.69	0.0
		10.8	0.0
	fipronil	0.0431	0.0
		0.172	45.5
		0.673	100.0

As the composition for exterminating animal parasites according to the invention has excellent activity for exterminating animal parasites, the composition has wide industrial applicability.

The foregoing description of the exemplary embodiments of the present invention has been provided for the purposes of illustration and description. It is not intended to be exhaustive or to limit the invention to the precise forms disclosed. Obviously, many modifications and variations will be apparent to practitioners skilled in the art. The exemplary embodiments were chosen and described in order to best explain the principles of the invention and its practical applications, thereby enabling others skilled in the art to understand the invention for various embodiments and with the various modifications as are suited to the particular use contemplated. It is intended that the scope of the invention be defined by the following claims and their equivalents.

All publications, patent applications, and technical standards mentioned in this specification are herein incorporated by reference to the same extent as if each individual publication, patent application, or technical standard was specifically and individually indicated to be incorporated by reference.

Claims

1. An amide derivative represented by the following Formula (1a):

2. The amide derivative according to claim 1, wherein in Formula (1a): Q1 represents a phenyl group which may have a halogen atom or a pyridyl group which may have a halogen atom;R1 represents and a C1-C6 alkyl group; andR2 represents a hydrogen atom or a C1-C6 alkyl group.

3. The amide derivative according to claim 2, wherein in Formula (1a): Q1 represents a phenyl group which may have a fluorine atom or a pyridyl group which may have a chlorine atom;Y1 represents a bromine atom, and Y5 represents a trifluoromethyl group;Y3 represents a heptafluoroisopropyl group;R1 represents a methyl group; andR2 represents a hydrogen atom or a methyl group.

4. The amide derivative according to claim 3, wherein in Formula (1 a): T represents —C(=G1)-Q1.

5. A pest control agent comprising at least one amide derivative according to claim 1 as an active ingredient.

6. The pest control agent according to claim 5, wherein the pest is an animal parasite.

7. The amide derivative according to claim 2, wherein in Formula (1a): Q2 represents a C1-C6 haloalkyl group.

8. The amide derivative according to claim 1, wherein in Formula (1a): Q2 represents a 2,2,2-trifluoroethyl group.