Claims
- 1. A sterol conjugate compound of the formula ##STR14## wherein each R.sub.1, R.sub.2, R.sub.3 and R.sub.4 is individually selected from the group consisting of H, OH and OSO.sub.3 H; and wherein Y is NH(CH.sub.2).sub.3 NH(CH.sub.2).sub.4 NH(CH.sub.2).sub.3 NH.sub.2, NHCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 NH.sub.2, or NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NH.sub.2.
- 2. A compound according to claim 1 which is ##STR15## wherein Y is selected from the group consisting of NH(CH.sub.2).sub.3 NH(CH.sub.2).sub.4 NH(CH.sub.2).sub.3 NH.sub.2, NHCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 NH.sub.2, and NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NH.sub.2, and wherein X is selected from the group consisting of H and SO.sub.3 H.
- 3. A compound according to claim 2 wherein Y is NH(CH.sub.2).sub.3 NH(CH.sub.2).sub.4 NH(CH.sub.2).sub.3 NH.sub.2.
- 4. The compound according to claim 3 wherein X is H.
- 5. The compound according to claim 3 wherein X is SO.sub.3 H.
- 6. A compound according to claim 2 wherein Y is NHCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 NH.sub.2.
- 7. The compound according to claim 6 wherein X is H.
- 8. The compound according to claim 6 wherein X is SO.sub.3 H.
- 9. A compound according to claim 2 wherein Y is NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NH.sub.2.
- 10. The compound according to claim 9 wherein X is H.
- 11. The compound according to claim 9 wherein X is SO.sub.3 H.
- 12. The compound according to claim 1 which is ##STR16## wherein Y is selected from the group consisting of NH(CH.sub.2).sub.3 NH(CH.sub.2).sub.4 NH(CH.sub.2).sub.3 NH.sub.2, NHCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 NH.sub.2, and NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NH.sub.2, and wherein X is selected from the group consisting of H and SO.sub.3 H.
- 13. The compound according to claim 1 which is ##STR17## wherein Y is selected from the group consisting of NH(CH.sub.2).sub.3 NH(CH.sub.2).sub.4 NH(CH.sub.2).sub.3 NH.sub.2, NHCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 NH.sub.2, and NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NH.sub.2, and wherein X is selected from the group consisting of H and SO.sub.3 H.
- 14. The compound according to claim 1 which is ##STR18## wherein X is selected from the group consisting of H, OSO.sub.3 H, and OH, and Y is selected from the group consisting of NH(CH.sub.2).sub.3 NH(CH.sub.2).sub.4 NH(CH.sub.2).sub.3 NH.sub.2, NHCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 NH.sub.2, or NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NH.sub.2.
- 15. A compound according to claim 1 which is ##STR19## wherein Y is selected from the group consisting of NH(CH.sub.2).sub.3 NH(CH.sub.2).sub.4 NH(CH.sub.2).sub.3 NH.sub.2, NHCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 NH.sub.2, and NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NH.sub.2, and wherein X is selected from the group consisting of H and SO.sub.3 H.
- 16. A compound according to claim 1 which is ##STR20## wherein Y is selected from the group consisting of NH(CH.sub.2).sub.3 NH(CH.sub.2).sub.4 NH(CH.sub.2).sub.3 NH.sub.2, NHCH.sub.2 CH.sub.2 CH.sub.2 CH.sub.2 NH.sub.2, and NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NHCH.sub.2 CH.sub.2 NH.sub.2, and wherein X is selected from the group consisting of H and SO.sub.3 H.
Government Interests
Partial financial support in the making of the invention described herein was provided by the National Institutes of Health. In view of providing financial support to the making of the invention described herein, the United States government has certain statutory interests in the invention under 35 USC 200 et seq.
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