Claims
- 1. A 2-oxa-7,9-diazabicyclo[4,2,2]-decane derivative, which is selected from the group consisting of the following compounds: 5-benzyloxyimino-5-nor-bicyclomycin; 5-carboxymethoxyimino-5-nor-bicyclomycin; 5-methoxyimino-5-nor-bicyclomycin-6,1',3'-tri-tetrahydropyranyl ether; 5-nor-bicyclomycin-5-one phenylhydrazone, 5-nor-bicyclomycin-5-one semicarbazone, and 5-nor-bicyclomycin-5-one pyridinioacetylhydrazone chloride.
- 2. 5-Hydroxyimino-5-nor-bicyclomycin.
- 3. 5-Methoxyimino-5-nor-bicyclomycin.
- 4. 5-Methylcarbonylmethoxyimino-5-nor-bicyclomycin.
- 5. 5-Methoxyimino-5-nor-bicyclomycin-3'-benzoate.
- 6. Pharmaceutically tolerable non-toxic salts of compound of claims 1 to 5, provided they contain salt-forming groups.
- 7. A pharmaceutical preparation useful against bacteria, which contains an effective amount of one of the compound of any one of claims 1 to 6, together with pharmacologically useful carriers.
- 8. A method of treating anti-bacterial diseases which comprises enteral or parenteral administration of a therapeutically effective dose of a compound according to any one of claims 1 to 6.
- 9. A method of treating anti-bacterial diseases which comprises enteral or parenteral administration of a therapeautically effective dose of a pharmaceutical preparation according to claim 7.
Priority Claims (1)
Number |
Date |
Country |
Kind |
6445/76 |
May 1976 |
CHX |
|
Parent Case Info
This is a Continuation of application Ser. No. 796,286 filed on May 12, 1977, now abandoned.
US Referenced Citations (4)
Number |
Name |
Date |
Kind |
3873526 |
Kamiya et al. |
Mar 1975 |
|
3923790 |
Imanaka et al. |
Dec 1975 |
|
4145344 |
Muller et al. |
Mar 1979 |
|
4215043 |
Kamiya et al. |
Jul 1980 |
|
Foreign Referenced Citations (1)
Number |
Date |
Country |
1464962 |
Feb 1977 |
GBX |
Continuations (1)
|
Number |
Date |
Country |
Parent |
796286 |
May 1977 |
|