Carbamates and crop protection agents containing them

Abstract

Carbamates of the formula I where the substituents have the following meanings:Z is methoxy, NH.sub.2, NHCH.sub.3, N(CH.sub.3).sub.2, CH.sub.3, C.sub.2 H.sub.5, CF.sub.3 or CCl.sub.3,X and Y are identical or different and each is hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may be condensed together to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,R.sup.1 may also be substituted or unsubstituted and is O-alkyl, O-alkenyl, O-alkynyl, O-cycloalkyl, O-cycloalkenyl or O--CO.sub.2 -alkyl,A is --O--, --S--, --CR.sup.2 .dbd.CR.sup.3 --, CHR.sup.2 --O--, --CHR.sup.2 --S--, --CHR.sup.2 --O--N.dbd.C(R.sup.4)--, --CR.sup.2 .dbd.N--O--, --O--N.dbd.C(R.sup.4)--, --C.tbd.C--, --CHR.sup.2 --CHR.sup.3 --, --CHR.sup.2 --O--CO--, --O--CHR.sup.2 -- or a single bond,B is substituted or unsubstituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl, hydrogen, substituted or unsubstituted alkylaryl, substituted or unsubstituted alkylhetaryl, substituted or unsubstituted alkylcycloalkyl, substituted or unsubstituted alkylcycloalkenyl,R.sup.2 and R.sup.3 are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl,R.sup.4 is hydrogen, CN, alkyl, alkenyl, alkynyl, alkoxy or cycloalkyl,R.sup.5 is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl and plant-tolerated acid and base adducts thereof, and fungicides containing them.

Description

The present invention relates to carbamates and crop protection agents, in particular for controlling fungi, insects, nematodes and spider mites.

It is known that aniline derivatives, for example isopropyl N-phenylcarbamate or the corresponding 3-chlorophenyl ester (GB 574 995) or methyl N-3,4-dichlorophenylcarbamate (BE 612 550) can be used as crop protection agents. However, their fungicidal action is unsatisfactory.

It has now been found, surprisingly, that carbamates of the formula I ##STR1## where the substituents have the following meanings: Z is methoxy, NH.sub.2, NHCH.sub.3, N(CH.sub.3).sub.2, CH.sub.3, C.sub.2 H.sub.5, CF.sub.3 or CCl.sub.3, X and Y independently of one another are each hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form an unsubstituted or substituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

R.sup.1 is unsubstituted or substituted alkyl, alkenyl, cyclopropyl, cyclopropylmethyl, cyclobutyl, --CH.sub.2 --CN, --CH.sub.2 OCH.sub.3, --CO.sub.2 CH.sub.3 or --S--R.sup.5, O-alkyl, O-alkenyl, O-alkynyl, O-cycloalkyl, O-cycloalkenyl or O--CO.sub.2 -alkyl, A is --O--, --S--, --CR.sup.2 .dbd.CR.sup.3 --, CHR.sup.2 --O--, --CHR.sup.2 --S--, --CHR.sup.2 --O--N.dbd.C(R.sup.4)--, --CR.sup.2 .dbd.N--O--, --O--N.dbd.C(R.sup.4)--, --C.tbd.C--, --CHR.sup.2 --CHR.sup.3 --, --CHR.sup.2 --O--CO--, --O--CHR.sup.2 -- or a single bond, B can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl, hydrogen, unsubstituted or substituted alkylaryl, unsubstituted or substituted alkylhetaryl, unsubstituted or substituted alkylcycloalkyl or unsubstituted or substituted alkylcycloalkenyl, R.sup.2 and R.sup.3 independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, R.sup.4 is hydrogen, CN, alkyl, alkenyl, alkynyl, alkoxy or cycloalkyl, R.sup.5 is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl, and their plant-tolerated acid addition products and base addition products have a good fungicidal, acaricidal, insecticidal and nematocidal action.

Acids for addition products are, for example, mineral acids, such as hydrochloric acid, hydrobromic acid, phosphoric acid, sulfuric acid or nitric acid, or carboxylic acids, such as formic acid, acetic acid, oxalic acid, malonic acid, lactic acid, malic acid, succinic acid, tartaric acid, citric acid, salicylic acid, p-toluenesulfonic acid or dodecylbenzenesulfonic acid, as well as proton-acidic compounds generally, for example saccharin.

Bases for base addition products are, for example, potassium hydroxide, sodium hydroxide, potassium carbonate, sodium carbonate and ammonium hydroxide.

The novel compounds of the formula I may be obtained in the preparation as mixtures of stereoisomers (E/Z isomers, diastereomers, enantiomers), which can be separated into the individual components in a conventional manner, for example by crystallization or chromatography. Both the individual isomers and mixtures thereof may be used as fungicides, acaricides, nematocides or insecticides, and form the subject of the present invention.

The abovementioned alkyl radicals may be substituted and are of 1 to 6 carbon atoms.

The abovementioned alkenyl and alkynyl radicals may be substituted and are of 2 to 6 carbon atoms.

The abovementioned cycloalkyl radicals are of 3 to 10 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R.sup.6.

The abovementioned aryl radicals are of 6, 10 or 14 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R.sup.6.

The abovementioned hetaryl radicals have 5 to 14 ring atoms, including from 1 to 4 hetero atoms selected from the group consisting of N, O and S, are unsaturated and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R.sup.6.

The abovementioned heterocyclyl radicals have 5 to 14 carbon atoms, including 1 to 4 hetero atoms selected from the group consisting of N, O and S, are saturated or partially unsaturated and are unsubstituted or substituted, for example by 1 to 4 identical or different substitutents R.sup.6.

The abovementioned cycloalkenyl radicals are of 5 to 14 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R.sup.6.

Two adjacent substituents R.sup.6, together with the carbon atoms of which they are substituents, may form a carbocyclic hydrogenated, partially unsaturated or aromatic ring having 3 to 14 carbon atoms or a heterocyclic hydrogenated, partially unsaturated or heteroaromatic ring having 3 to 14 carbon atoms, including 1 to 4 hetero atoms selected from the group consisting of N, O and S.

R.sup.6 may be unsubstituted or substituted, for example by 1 to 4 identical or different substituents R.sup.7, and R.sup.6 is, for example, hydrogen, halogen, cyano, nitro, haloalkyl, alkyl, haloalkoxy, alkenyl, alkynyl, cycloalkyl, aryl, hetaryl, heterocyclyl, cycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, aryloxy, hetaryloxy, heterocyclyloxy, cycloalkenyloxy, alkoximino, alkenyloximino, alkynyloximino, cycloalkoxyimino, cycloalkenyloximino, aryloximino, hetaryloximino, heterocyclyloximino, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkyloxycarbonyl, aryloxycarbonyl, hetaryloxycarbonyl, heterocyclyloxycarbonyl, cycloalkenyloxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkenylaminocarbonyl, dialkenylaminocarbonyl, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, arylthio, hetarylthio, heterocyclylthio, cycloalkenylthio, alkylamino, alkenylamino, alkynylamino, cycloalkylamino, arylamino, hetarylamino, heterocyclylamino, cycloalkenylamino, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, arylcarbonyl, hetarylcarbonyl, heterocyclylcarbonyl, cycloalkenylcarbonyl, alkylsulfoxyl, alkenylsulfoxyl, alkynylsulfoxyl, cycloalkylsulfoxyl, arylsulfoxyl, hetarylsulfoxyl, heterocyclylsulfoxyl, cycloalkenylsulfoxyl, alkylsulfonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, hetarylsulfonyl, heterocyclylsulfonyl, cycloalkenylsulfonyl, alkylsulfinyl, alkenylsulfinyl, alkynylsulfinyl, cycloalkylsulfinyl, arylsulfinyl, hetarylsulfinyl, heterocyclylsulfinyl or cycloalkenylsulfinyl.

R.sup.7 is any substituent and is, for example, hydrogen, halogen, cyano, nitro, haloalkyl, alkyl, haloalkoxy, alkenyl, alkynyl, cycloalkyl, aryl, hetaryl, heterocyclyl, cycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, aryloxy, hetaryloxy, heterocyclyloxy, cycloalkenyloxy, alkoximino, alkenyloximino, alkynyloximino, cycloalkoximino, cycloalkenyloximino, aryloximino, hetaryloximino, heterocyclyloximino, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkyloxycarbonyl, aryloxycarbonyl, hetaryloxycarbonyl, heterocyclyloxycarbonyl, cycloalkenyloxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkenylaminocarbonyl, dialkenylaminocarbonyl, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, arylthio, hetarylthio, heterocyclylthio, cycloalkenylthio, alkylamino, alkenylamino, alkynylamino, cycloalkylamino, arylamino, hetarylamino, heterocyclylamino, cycloalkenylamino, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, arylcarbonyl, hetarylcarbonyl, heterocyclylcarbonyl, cycloalkenylcarbonyl, alkylsulfoxyl; alkenylsulfoxyl, alkynylsulfoxyl, cycloalkylsulfoxyl, arylsulfoxyl, hetarylsulfoxyl, heterocyclylsulfoxyl, cycloalkenylsulfoxyl, alkylsulfonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, hetarylsulfonyl, heterocyclylsulfonyl, cycloalkenylsulfonyl, alkylsulfinyl, alkenylsulfinyl, alkynylsulfinyl, cycloalkylsulfinyl, arylsulfinyl, hetarylsulfinyl, heterocyclylsulfinyl or cycloalkenylsulfinyl.

The abovementioned alkyl radicals may be substituted, are preferably of 1 to 6 carbon atoms and are, in particular, methyl, ethyl, propyl, such as n-propyl or isopropyl, butyl, such as n-butyl, isobutyl, tert-butyl or sec-butyl, pentyl or hexyl.

The abovementioned alkenyl radicals may be substituted, are preferably of 2 to 6 carbon atoms and are, in particular, ethenyl, propenyl, such as prop-1-enyl, prop-2-enyl or prop-1-en-2-yl, butenyl, such as but-1-enyl, but-2-enyl, but-3-enyl, but-1-en-3-yl, but-2-en-2-yl, but-1-en-2-yl, 2-methyl-1-propenyl or 2-methyl-2-propenyl, pentenyl or hexenyl.

The abovementioned alkynyl radicals may be substituted, are preferably of 2 to 6 carbon atoms and are, in particular, ethynyl, propynyl, such as prop-1-ynyl or prop-3-ynyl, butynyl, such as but-1-ynyl, but-2-ynyl, but-3-ynyl or 1-methylprop-2-ynyl, pentynyl or hexynyl.

The abovementioned halogens are fluorine, chlorine, bromine or iodine.

The abovementioned cycloalkyl radicals are preferably cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, cycloheptyl, cyclooctyl, cyclononyl, cyclodecyl, bornanyl, norbornanyl, dicyclohexyl, bicyclo[3.3.0]octyl, bicyclo[3.2.1]octyl, bicyclo[2.2.2]octyl or bicyclo[3.3.1]nonyl.

The abovementioned cycloalkenyl radicals are preferably cyclopropenyl, cyclobutenyl, cyclopentenyl, cyclohexenyl, cycloheptenyl, cyclooctenyl, cyclononenyl, cyclodecenyl, bornenyl, norbornenyl, bicyclo[3.3.0]octenyl, bicyclo[3.2.1]octenyl, bicyclo[2.2.2]octenyl or bicyclo[3.3.1]nonenyl.

The abovementioned haloalkyl radicals are preferably C.sub.1 -C.sub.4 -haloalkyl, in particular C.sub.1 - or C.sub.2 -haloalkyl, such as chloromethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluoromethyl, dichlorofluoromethyl, chlorodifluoromethyl, 1-fluoroethyl, 2-fluoroethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2-difluoroethyl, 2,2-dichloro-2-fluoroethyl, 2,2,2-trichloroethyl or pentafluoroethyl.

The abovementioned haloalkoxy radicals are preferably C.sub.2 -C.sub.4 -haloalkoxy, in particular C.sub.1 - or C.sub.2 -haloalkoxy, such as chloromethoxy, dichloromethoxy, trichloromethoxy, fluoromethoxy, difluoromethoxy, trifluoromethoxy, chlorofluoromethoxy, dichlorofluoromethoxy, chlorodifluoromethoxy, 1-fluoroethoxy, 2-fluoroethoxy, 2,2-difluoroethoxy, 2,2,2-trifluoroethoxy, 2-chloro-2-fluoroethoxy, 2-chloro-2,2-difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy or pentafluoroethoxy.

The abovementioned aryl radicals are preferably phenyl, 1-naphthyl, 2-naphtyl, 1-anthracenyl, 2-anthracenyl or 9-anthracenyl.

The abovementioned hetaryl radicals are preferably furyl, such as 2-furyl or 3-furyl, thienyl, such as 2-thienyl or 3-thienyl, pyrrolyl, such as 1-pyrrolyl, 2-pyrrolyl or 3-pyrrolyl, isoxazolyl, such as 3-isoxazolyl, 4-isoxazolyl or 5-isoxazolyl, isothiazolyl, such as 3-isothiazolyl, 4-isothiazolyl or 5-isothiazolyl, pyrazolyl, such as 1-pyrazolyl, 3-pyrazolyl, 4-pyrazolyl or 5-pyrazolyl, oxazolyl, such as 2-oxazolyl, 4-oxazolyl or 5-oxazolyl, thiazolyl, such as 2-thiazolyl, 4-thiazolyl or 5-thiazolyl, imidazolyl, such as 1-imidazolyl, 2-imidazolyl, 4-imidazolyl or 5-imidazolyl, 1,2,3-thiadiazolyl, 1,2,4-thiadiazolyl, 1,2,5-thiadiazolyl, 1,3,4-thiadiazolyl, tetrazolyl, 1,2,3,4-thiatriazolyl, 1,2,3,4-oxatriazolyl, pyridyl, such as 2-pyridyl or 4-pyridyl, pyridazinyl, such as 3-pyridazinyl or 4-pyridazinyl, pyrimidinyl, such as 2-pyrimidinyl, 4-pyrimidinyl or 5-pyrimidinyl, pyrazinyl, such as 2-pyrazinyl or 3-pyrazinyl, 1,2,4-triazinyl, 1,3,5-triazinyl or 1,2,4,5-tetrazinyl.

Adjacent substituents of the hetero atoms may be condensed to form an aromatic or heteroaromatic ring, so that hetaryl also comprises fused ring systems, eg. benzofuranyl, isobenzofuranyl, 1-benzothienyl, 2-benzothienyl, indolyl, isoindolyl, benzisoxazolyl, benzoxazolyl, benzisothiazolyl, benzothiazolyl, such as 2-benzothiazolyl, 4-benzothiazolyl, 5-benzothiazolyl, 6-benzothiazolyl or 7-benzothiazolyl, indazolyl, benzimidazolyl, benzofurazanyl, dibenzofuranyl, dibenzothienyl, acridinyl, phenanthridinyl, carbazolyl, quinolyl, isoquinolyl, phthalazinyl, quinazolinyl, quinoxalinyl, cinnolinyl, 1,5-naphthyridinyl, 1,6-naphthyridinyl, 1,7-naphthyridinyl, 1,8-naphthyridinyl, pteridinyl, pyrrolopyridinyl, pyrrolopyridazinyl, pyrrolopyrimidinyl, pyrrolopyrazinyl, pyrrolotriazinyl, furopyridyl, furopyridazinyl, furopyrimidinyl, furopyrazinyl, furotriazinyl, thienopyridyl, thienopyridazinyl, thienopyrimidinyl, thienopyrazinyl, thienotriazinyl, imidazopyridazinyl, imidazopyrimidinyl, imidazopyrazinyl, pyrazolopyridyl, pyrazolopyridazinyl, pyrazolopyrimidinyl, pyrazopyrazinyl, isoxazolopyrazinyl, oxazolopyridyl, oxazolopyridazinyl, oxazolopyrimidinyl, oxazolopyrazinyl, thiazolopyridyl, thiazolopyridazinyl, isothiazolopyrazinyl, triazolopyridyl, triazolopyridazinyl, triazolopyrimidinyl or triazolopyrazinyl.

The abovementioned heterocycyl radicals are preferably 2-tetrahydrofuranyl, oxiranyl, 3-tetrahydrofuranyl, 2-tetrahydrothienyl, 3-tetrahydrothienyl, 2-pyrrolidinyl, 3-pyrrolidinyl, 3-isoxazolidinyl, 4-isoxazolidinyl, 5-isoxazolidinyl, 3-isothiazolidinyl, 4-isothiazolidinyl, 5-isothiazolidinyl, 3-pyrazolidinyl, 4-pyrazolidinyl, 5-pyrazolidinyl, 2-oxazolidinyl, 4-oxazolidinyl, 5-oxazolidinyl, 2-thiazolidinyl, 4-thiazolidinyl, 5-thiazolidinyl, 2-imidazolidinyl, 4-imidazolidinyl, 1,2,4-oxadiazolidin-3-yl, 1,2,4-oxadiazolidin-5-yl, 1,2,4-thiadiazolidin-3-yl, 1,2,4-thiadiazolidin-5-yl, 1,2,5-triazolidin-3-yl, 1,3,4-oxadiazolidin-2-yl, 1,3,4-thiadiazolidin-2-yl, 1,3,4-triazolidin-2-yl, 2,3-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,5-dihydrofur-2-yl, 2,5-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,3-dihydrothieno-2-yl, 2,3-dihydrothien-3-yl, 2,5-dihydrothien-2-yl, 2,4-pyrrolin-2-yl, 2,3-pyrrolin-3-yl, 2,5-pyrrolin-2-yl, 2,5-pyrrolin-3-yl, 2,3-isoxazolidin-3-yl, 3,4-isoxazolin-3-yl, 4,5-isoxazolin-2-yl, 2,3-isoxazolin-4-yl, 3,4-isoxazolin-3-yl, 4,5-isoxazolin-4-yl, 2,3-isoxazolin-5-yl, 3,4-isoxazolin-5-yl, 4,5-isoxazolin-5-yl, 2,3-isothiazolin-3-yl, 3,4-isothiazolin-3-yl, 4,5-isothiazolin-3-yl, 2,3-isothiazolin-4-yl, 3,4-isothiazolin-4-yl, 4,5-isothiazolin-4-yl, 2,3-isothiazolin-5-yl, 3,4-isothiazolin-5-yl, 4,5-isothiazolin-5-yl, 2,3-dihydropyrazol-1-yl, 2,3-dihydropyrazol-2-yl, 2,3-dihydropyrazol-3-yl, 2,3-dihydropyrazol-4-yl, 2,3-dihydropyrazol-5-yl, 3,4-dihydropyrazol-1-yl, 3,4-dihydropyrazol-2-yl, 3,4-dihydropyrazol-4-yl, 3,4-dihydropyrazol-5-yl, 4,5-dihydropyrazol-1-yl, 4,5-dihydropyrazol-3-yl, 4,5-dihydropyrazol-4-yl, 4,5-dihydropyrazol-5-yl, 3,4-dihydrooxazol-2-yl, 2,3-dihydrooxazol-3-yl, 2,3-dihydrooxazol-4-yl, 2,3-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 3,4-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 2-piperidinyl, 3-piperidinyl, 4-piperidinyl, 3-tetrahydropyridazinyl, 4-tetrahydropyridazinyl, 2-tetrahydropyrimidinyl, 4-tetrahydropyrimidinyl, 5-tetrahydropyrimidinyl, 2-tetrahydropyrazinyl, 1,3,5-tetrahydrotriazin-2-yl, 1,2,4-tetrahydrotriazin-3-yl, 1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, oxazol-2-in-2-yl, 2-tetrahydropyranyl, 1,3-dioxolan-2-yl, thiazol-2-in-2-yl, 3,4,5,6-tetrahydropyridin-2-yl, 4H-1,3-thiazin-2-yl, 4H-3,1-benzothiazin-2-yl, 1,1-dioxo-2,3,4,5-tetrahydrothien-2-yl, 2H-1,4-benzothiazin-3-yl, 2H-1,4-benzoxazin-3-yl, 1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, N-morpholinyl or dihydroquinazolinyl.

The invention furthermore relates to carbamates of the formula I ##STR2## where the substituents have the following meanings: Z is methoxy, NH.sub.2, NHCH.sub.3 or CH.sub.3,

X and Y independently of one another are each hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form a phenyl ring, R.sup.1 is hydrogen, alkyl, alkenyl alkynyl cyclopropyl, cyclopropylmethyl, cyclobutyl, --CH.sub.2 --CN, --CH.sub.2 --O--CH.sub.3, --CO.sub.2 CH.sub.3 or --S--R.sup.5, A is --O--, --CR.sup.2 .dbd.CR.sup.3 --, --C.tbd.C--, --CHR.sup.2 --O--, --CHR.sup.2 --S--, --CHR.sup.2 --O--N.dbd.C(R.sup.4)--, --CR.sup.2 .dbd.N--O-- or --O--N.dbd.C(R.sup.4)--, a) B is substituted phenyl when A is --CR.sup.2 .tbd.CR.sup.3 --, --C.dbd.C--, --CHR.sup.2 --O--, --CHR.sup.2 --S--, --CR.sup.2 --O--N.dbd.C(R.sup.4)--, --CR.sup.2 .dbd.N--O-- or --O--N.dbd.C(R.sup.4), b) or B is unsubstituted or substituted cyclolalkyl, unsubstituted or substituted cycloalkenyl, unsubstituted or substituted heterocyclyl, unsubstituted or substituted hetaryl, unsubstituted or substituted naphthyl, unsubstituted or substituted arylalkyl, unsubstituted or substituted hetarylalkyl, unsubstituted or substituted cycloalkylalkyl, unsubstituted or substituted cycloalkenylalkyl or unsubstituted or substituted anthracenyl, R.sup.2 and R.sup.3 independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, R.sup.4 is CN, alkyl, alkenyl, alkynyl or cycloalkyl and R.sup.5 is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl, and their plant-tolerated acid addition products and base addition products.

The invention furthermore relates to carbamates of the formula II ##STR3## where X, Y, R.sup.1 and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula III ##STR4## where X, Y, R.sup.1 and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula I as claimed in claim 2, where A is --CH.dbd.CH-- and X, Y, R.sup.1 and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula VII ##STR5## where the substituents have the following meanings: X and Y independently of one another are each hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form an unsubstituted or substituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

R.sup.1 can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO.sub.2 -alkyl, A is --O--, --S--, --CR.sup.2 .dbd.CR.sup.3 --, CHR.sup.2 --O--, --CHR.sup.2 --S--, --CHR.sup.2 --O.dbd.N--C(R.sup.4)--, --CR.sup.2 .dbd.N--O--, --O--N.dbd.C(R.sup.4)--, --C.tbd.C--, --CHR.sup.2 --CHR.sup.3 --, --CHR.sup.2 --O--CO--, --O--CHR.sup.2 -- or a single bond, B can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl or hydrogen, R.sup.2 and R.sup.3 independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl and R.sup.4 is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy, and their plant-tolerated acid addition products and base addition products.

The invention furthermore relates to carbamates of the formula VIII ##STR6## where A, B and R.sup.1 have the meanings stated in claim 9.

The invention furthermore relates to carbamates of the formula IX ##STR7## where R.sup.1 and B have the meanings stated in claim 1.

The invention furthermore relates to carbamates of the formula X ##STR8## where R.sup.1 and B have the meanings stated in claim 1.

The novel compounds can be prepared, for example, by the following processes:

The nitrobenzenes 1 obtainable by standard processes are reduced to the anilines 2, for example with hydrogen or hydrogen transfer agents, such as ammonium formate, in the presence of suitable catalysts, such as Pd, Pt or Ni, with complex reducing agents, eg. Collman's reagent (Na.sub.2 Fe(CO).sub.4) or by other methods known from the literature (J. March, Advanced Organic Chemistry, 3rd Edition,. 1985, page 1103 et seq.). The anilines 2 are reacted under alkaline conditions with methyl chloroformate to give the carbamates 3. The reaction of the carbamates 3 under alkaline conditions with the corresponding alkylating agents, acylating agents or R.sup.5 --S--S(.dbd.O).sub.2 --R.sup.5 gives the derivatives 4 (Scheme 1). ##STR9##

The nitrobenzenes 5 can be converted into the carbamates 6 similarly to Scheme 1. The halogen derivatives 7 (Z=Cl or Br) are obtainable by acidic cleavage of the methyl ether of 6 (Scheme 2). ##STR10##

Alternatively, the halogen derivatives 7 (Z=Cl or Br) are obtainable from the derivatives 9 by free radical halogenation. The carbamates 9 are in turn prepared from the corresponding starting materials 8, similarly to Scheme 1 (Scheme 3). ##STR11##

The halogen derivatives 7 (Z=Cl or Br) can be converted into the active ingredients 10 under alkaline conditions. Alternatively, the compounds 7 are converted into the phosphorus compounds 11a and 11b by reaction with P(C.sub.6 H.sub.5).sub.3 or P(O-Alkyl).sub.3, or into the carbonyl compounds 12 by oxidation (for example with N-methylmorpholine N-oxide) (Scheme 4). ##STR12## A=--CHR.sup.2 --O-- --CHR.sup.2 --S-- --CHR.sup.2 --O--N.dbd.C(R.sup.4)--

The corresponding stilbenes 13 are obtainable from the phosphonium salts 11a or phosphonates 11b or carbonyl compounds 12 by a Wittig reaction (Scheme 5). ##STR13##

Partial reduction of the nitroaromatics 21 (for example with zinc (similarly to Bamberger et al., Ann. Chem. 316 (1901), 278) or with hydrogen in the presence of suitable catalysts such as platinum (similarly to European Patent 85,890)) gives the hydroxylamines 22, which can be reacted under alkaline conditions with an acylating agent (eg. propionyl chloride) or a carbamoylating agent (eg. methyl isocyanate) to give the compound 23 and then with an electrophile, for example with an alkylating agent, to give the active ingredients 24 (scheme 11). ##STR14##

In addition, the hydroxylamine 25 can be acylated or aminoacylated (for example with methyl isocyanate) (similarly to Bamberger et al., Ann. Chem. 316 (1901), 278; European Patent 85,890) to give the compound 26, which can then be alkylated or alkoxyacylated (for example with chloroformates) to give the hydroxylamine derivative 27. The free radical halogenation of 27, for example with N-bromosuccinamide, bromine, chlorine or SO.sub.2 Cl.sub.2 in the presence of free radical initiator, eg. azobisisobutyronitrile, or with exposure to UV light, then gives the halide 28 (Hal=Cl or Br; Scheme 12). ##STR15##

The halides 28 can then be converted into the compounds 29 with the corresponding nucelphiles (Scheme 13). ##STR16##

In addition, the halides 28 can be converted by free radical reaction to the dihalide 30 and then converted with H.sub.2 O/MeOH in the presence of AgNO.sub.3 into the carbonyl compound 31 or reacted directly with N-methylmorpholine N-oxide to give the carbonyl compound 11. Furthermore, the phosphonates, phosphonium salts or phosphine oxides 32 (P is the particular organophosphorus radical) are obtainable from the halides 8 (Scheme 14). ##STR17##

The carbonyl compounds 31 can then be reacted with the corresponding hydroxylamines to give the oximes 33 or can be subjected to a Wittig reaction to give the olefins 34, The olefins 34 are also obtainable by a Wittig reaction starting from the phosphonates, phosphonium salts or phosphine oxides 32 (Scheme 15). ##STR18##

The saturated compounds 35 can be prepared from the olefins 34 by reduction or, where R.sup.2 and R.sup.3 are each H, the acetylenes 36 can be prepared from said olefins by halogen addition (Hal=Cl, Br or I) and subsequent two-fold elimination of hydrogen halide (Scheme 16). ##STR19##

Alternatively, the ureas 39 can be synthesized by acylation of the hydroxylamines 22 to the compounds 37, subsequent alkylation or acylation to the compounds 38 and substitution of the nucleofugic leaving group V (V is, for example, OCH.sub.3, OCCl.sub.3, CCl.sub.3, O-phenyl or O-p-nitrophenyl) by NH.sub.3, H.sub.2 N--CH.sub.3 or HN(CH.sub.3).sub.2 (Scheme 17). ##STR20##

Alternatively, ureas of the formula 39 can also be obtained by alkylating ureas of the formula 41, which in turn are obtainable from 17 by reacting 17 with the corresponding amines, or directly from 22 by aminocarbonylation (for example with dimethylcarbamoyl chloride or methyl isocyanate) (cf. for example Houben-Weyl, volume E16a, page 208).

Furthermore, ureas of the formula 39 can also be obtained from the N-aryl-O-alkylhydroxylamines of the formula 42 in a similar manner by aminocarbonylation.

The compounds of the formula 42 are in turn obtainable by methods known from the literature, from hydroxylamines of the formula 2 (cf. for example Houben-Weyl, volume E16a, pages 271 and 282-289).

In addition, the hydroxylamines 22 are obtainable from the anilines 43 by formation of the imines 44, oxidation of the compounds 44 with the m-chloroperbenzoic acid and reaction of the oxaziridines 45 with hydroxylamine (Scheme 18; similarly to G. Grundke et al., Synthesis 1987, 1115). ##STR21##

The Examples which follow illustrate the preparation of the novel compounds.

EXAMPLES

Example 1

Methyl N-ethyl-N-(2-(2'-methylphenoxymethyl)-phenyl)-carbamate (Table 7, No. 2)

a) Methyl N-(o-methylphenyl)-carbamate

50 g (0.53 mol) of methyl chloroformate are added dropwise to 53 g (0.5 mol) of o-toluidene in 500 ml of methylene chloride. During this procedure, the reaction solution heats up to the boiling point and a colorless solid is precipitated.

Stirring is carried out for one hour, after which 200 ml of 10% strength sodium hydroxide solution are added dropwise, the colorless solid going into solution. The organic phase is dried over MgSO.sub.4 and evaporated down under reduced pressure. The remaining solid is stirred with n-hexane and filtered off under suction. 84 g (0.5 mol, quantitative yield) of the title compound are obtained as a colorless solid.

mp.=61-62.degree. C.

.sup.1 H-NMR (DMSO-d.sub.6 ; .delta. (ppm)): 8.85 (s, 1H, NH); 7.35 (d, broad, 1H, aromatic); 7.1 (m, 3H, aromatic); 3.6 (s, 3H, OCH.sub.3); 2.2 (s, 3H, CH.sub.3).

b) Methyl N-ethyl-N-(o-methylphenyl)-carbamate

5.1 g (0.2 mol) of sodium hydride are added a little at a time to 30 g (0.18 mol) of methyl N-(o-methylphenyl)-carbamate (Example 1a) in 200 ml of dimethylformamide. After the evolution of gas has ceased, 30 g (0.2 mol) of ethyl iodide are added dropwise, the reaction mixture being lightly cooled in a water bath. A white solid is precipitated. After about 4 hours, the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The organic phase is dried over MgSO.sub.4 and evaporated down. The residue is distilled. 32.5 g (0.17 mol=93%) of the title compound are obtained as a colorless oil.

bp..sup.0.5 =74.degree. C.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm): 7.2 (m, 3H, aromatic); 7.1 (m, 1H, aromatic); 3.8 (m, 1H, N--CH.sub.A); 3.6 (s, 3H, OCH.sub.3); 3.5 (m, 1H, N--CH.sub.B); 2.2 (s, 3H, CH.sub.3); 1.1 (t, 3H, CH.sub.3).

c) Methyl N-ethyl-N-(o-bromomethylphenyl)-carbamate

A mixture of 30 g (0.155 mol) of methyl N-ethyl-N-(o-methylphenyl)-carbamate (Example 1b), 33 g (0.185 mol) of N-bromosuccinimide and 0.1 g of azoisobutyronitrile in 300 ml of carbon tetrachloride is exposed to a 300 W UV lamp for 6 hours. During this procedure, the contents of the flask heat up to about 70.degree. C. Thereafter, the reaction mixture is washed four times with water, dried and evaporated down. The residue obtained comprises 41 g of a brown oil which contains the title compound in about 50% purity and is used without further purification in the next reaction.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.2 (m, 4H, aromatic); 4.45 (s, 2H, CH.sub.2 --Br); 3.8 (m, 1H, N--CH.sub.A); 3.6 (s, 3H, OCH.sub.3); 3.5 (m, 1H, N--CH.sub.B); 1.15 (t, 3H, J=8 Hz, CH.sub.3).

d) Methyl N-ethyl-N-(2-(2'-methylphenoxymethyl)phenyl)-carbamate (Table 7, No. 2)

2.4 g (17 mmol) of sodium hydride are added a little at a time to 8.6 g (80 mmol) of o-cresol in 100 ml of dimethylformamide. Stirring is carried out for 30 minutes at room temperature (20.degree. C.), after which 20.5 g of methyl N-ethyl-N-(o-bromomethylphenyl)-carbamate (Example 1c, about 50% purity, about 37 mmol) are added. Stirring is carried out overnight at room temperature, after which the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The combined ether phases are dried over MgSO.sub.4 and evaporated down. The residue is distilled in a kugelrohr (bulb tube) apparatus. 10 g of a yellow oil are obtained at 220.degree. C. and 0.2 mbar, and the oil is then purified by chromatography with cyclohexane/ethyl acetate mixtures over silica gel and then over alumina. The product thus obtained is purified again by kugelrohr distillation. 3.6 g (12 mmol=32%) of the title compound are obtained as a colorless oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.6 (m, 1H, aromatic); 7.35 (m, 2H, aromatic); 7.15 (m, 3H, aromatic); 6.85 (m, 2H, aromatic); 5.0 (dd, broad, 2H, O--CH.sub.2); 3.8 (m, 1H, N--CH.sub.A); 3.6 (s, 3H, O--CH.sub.3); 3.5 (m, 1H, N--CH.sub.6); 2.3 (s, 3H, CH.sub.3); 1.15 (t, 3H, J=8 Hz, CH.sub.3).

Example 2

Methyl N-[2-(2'-methylphenoxymethyl)-phenyl]-N-methylthiocarbamate (Table 7, No. 89)

a) 2-(2'-Methylphenoxymethyl)-nitrobenzene

75 g (0.347 mol) of 2-nitrobenzyl bromide, 37 g (0.342 mol) of o-cresol and 56 g (0.405 mol) of potassium carbonate in 500 ml of dimethylformamide are stirred for 5 hours at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with ether. The ether phase is dried and evaporated down. The crystalline residue is stirred with methanol and filtered off under suction. 73 g (0.300 mol=88%) of the title compound are obtained as a colorless solid.

mp.=83.degree. C.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 8.15 (d, 1H, J=8 Hz, aromatic); 7.95 (d, 1H, J=8 Hz, aromatic); 7.7 (t, 1H, J=8 Hz, aromatic); 7.45 (t, 1H, J=8 Hz, aromatic); 7.15 (m, 2H, aromatic); 6.9 (m, 2H, aromatic); 5.45 (s, 2H, O--CH.sub.2); 2.35 (s, 3H, CH.sub.3).

b) 2-(2'-Methylphenoxymethyl)-aniline

75 g (0.308 mol) of 2-(2'-methylphenoxymethyl)nitrobenzene (Example 2a) and 10 g of 5% strength Pt/C (platinum adsorbed onto active carbon) in 50 ml of methanol are stirred vigorously for two hours under an H.sub.2 atmosphere. Thereafter, a further 2 g of 5% strength Pt/C are added and stirring is continued overnight. The catalyst is then filtered off under suction and is replaced with 10 g of fresh catalyst. Stirring is continued overnight, the mixture is filtered under suction and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography using hexane/ethyl acetate mixtures. 61 g (0.286 mol=93%) of the title compound are obtained as a colorless solid.

mp.=56.degree. C.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.2 (m, 4H, aromatic); 6.95 (d, 1H, J=8 Hz, aromatic); 6.9 (t, 1H, J=6 Hz, aromatic); 6.7 (m, 2H, aromatic); 5.0 (s, 2H, O--CH.sub.2); 4.05 (s, broad, 2H, NH.sub.2); 2.2 (s, 3H, CH.sub.3).

c) Methyl N-(2-(2'-methylphenoxymethyl)-phenyl]-carbamate (Table 7, No. 3)

6 g (63 mmol) of methyl chloroformate are added dropwise to 10 g (47 mmol) of 2-(2'-methylphenoxymethyl)aniline in 500 of methylene chloride at 20-30.degree. C. Stirring is carried out for 3 hours at room temperature, a white solid being precipitated, and the reaction mixture is then stirred with 20 ml of 10% strength sodium hydroxide solution. The organic phase is filtered off under suction over silica gel, the filtrate is evaporated down and the remaining residue is stirred thoroughly with methanol and filtered under suction. 10.5 g (39 mmol=82%) of the title compound are obtained as a colorless solid.

mp.=111.degree. C.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 8.0 (d, broad, 1H, aromatic); 7.7 (s, broad, 1H, aromatic); 7.7 (s, broad, 1H, NH); 6.8-7.5 (m, 6H, aromatic); 5.0 (s, 2H, O--CH.sub.2); 3.75 (s, 3H, O--CH.sub.3); 2.25 (s, 3H, CH.sub.3).

d) Methyl N-[2-(2'-methylphenoxymethyl)-phenyl]-N-methylthiocarbamate (Table 7, No. 89)

0.5 g (20.8 mmol) of sodium hydride is added a little at a time to 4.9 g (17.3 mmol) of methyl N-[2-(2'-methylphenoxymethyl)]-phenylcarbamate (Example 2c) in 80 ml of toluene. After the end of gas evolution, 2.4 g (19 mmol) of methyl methanethiosulfonate are added and stirring is carried out overnight at room temperature. Thereafter, the reaction mixture is extracted with water, dried over MgSO.sub.4 and evaporated down under reduced pressure. The residue is purified by column chromatography with hexane/ethyl acetate mixtures over silica gel. 3 g (9.1 mmol=53%) of the title compound are obtained as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.65 (d, broad, 1H, aromatic); 7.35 (m, 2H, aromatic); 7.15 (m, 3H, aromatic); 6.85 (m, 2H, aromatic); 5.0 (m, 2H, O--CH.sub.2); 3.75 (s, 3H, O--CH.sub.3); 2.55 (s, 3H, S--CH.sub.3); 2.3 (s, 3H, CH.sub.3).

Example 3

Methyl N-allyl-N-[2-(3"-bromophenylmethyliminoxymethyl)phenyl]-carbamate (Table 7, No. 91)

a) o-Methoxymethylnitrobenzene

125 g of 30% strength sodium methylate solution (0.69 mol) in methanol are added dropwise to 130 g (0.6 mol) of o-nitrobenzyl bromide in 200 ml of methanol. During this procedure, the reaction mixture heats up to about 50.degree. C. Stirring is continued for a further 3 hours, the reaction mixture being cooled to room temperature, after which ice water is added to the reaction vessel and the reaction mixture is neutralized by adding dilute hydrochloric acid. The aqueous phase is extracted with three times with ether, and the organic phase is dried over MgSO.sub.4 and evaporated down. 101 g (0.6 mol, quantitative yield) of the title compound are obtained as a residue in the form of a brownish oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 8.1 (d, broad, 1H, aromatic); 7.8 (d, broad, 1H, aromatic); 7.65 (t, broad, 1H, aromatic); 7.45 (t, broad, 1H, aromatic); 4.85 (s, 2H, O--CH.sub.2); 3.5 (s, 3H, OCH.sub.3).

b) Methyl N-(2-methoxymethylphenyl)-carbamate

528 g of 21.8% strength Na.sub.2 [Fe(CO).sub.4 ] solution (0.6 mol; 1 kg of the solution contains 633 g of water, 218 g of Na.sub.2 [Fe(CO).sub.4 ], 108 g of Na.sub.2 CO.sub.3 and 41 g of NaOH) are added dropwise to 101 g (0.6 mol) of o-methoxymethylnitrobenzene (Example 3a) in 1 l of methanol at 20-30.degree. C. Stirring is carried out for 1 hour at room temperature, after which the reaction mixture is diluted with ether. A brown oil separates out in the reaction vessel. The total reaction mixture is poured onto a silica gel column and is eluted with ether. Thereafter, the ether phase is evaporated, the residue is taken up in methylene chloride and the solution is dried over MgSO.sub.4. It is filtered under suction over silica gel and the solvent is then evaporated off under reduced pressure. The residue is purified by column chromatography with hexane and methylene chloride. 83.8 g of o-methoxymethylaniline are obtained as a brown oil, which is directly reacted further.

The resulting crude product is dissolved in 700 ml of methylene chloride, 62.4 g (0.66 mol) of methyl chloroformate are added and 52.2 g (0.66 mol) of pyridine are then added dropwise. Stirring is carried out overnight at room temperature and the reaction mixture is then extracted with dilute hydrochloric acid and water. The organic phase is dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with hexane/ethyl acetate mixtures. 89.4 g (0.41 mol=69%, based on 2-methoxymethylnitrobenzene) of the title compound are obtained as a yellow oil in a purity of about 90%.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm): 8.0 (m, 2H, 1.times.aromatic, NH); 7.35 (t, broad, 1H, aromatic); 7.15 (d, broad, 1H, aromatic); 7.0 (t, broad, 1H, aromatic); 4.5 (s, 2H, OCH.sub.2); 3.8 (s, broad, 3H, OCH.sub.3); 3.4 (s, broad, 3H, OCH.sub.3).

c) Methyl N-(2-bromomethylphenyl)-carbamate

38.6 g (150 mmol) of boron tribromide are added dropwise to 10 g (51 mmol) of methyl N-(2-methoxymethylphenyl)-carbamate (Example 2b) in 100 ml of methylene chloride. Stirring is carried out for 2 hours, after which the vigorously stirred reaction mixture is added dropwise to a solution of 11.8 g (0.17 mol) of NaHCO.sub.3 in water. The organic phase is separated off and the aqueous phase is extracted once with methylene chloride and once with ethyl acetate. The combined organic phases are dried over MgSO.sub.4 and evaporated down. 9.5 g (39 mmol=76%) of the title compound are obtained as a colorless solid.

mp.=132.degree. C.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.85 (d, broad, 1H, aromatic); 7.3 (m, 2H, aromatic); 7.1 (t, broad, 1H, aromatic); 6.9 (s, broad, 1H, NH); 4.5 (s, 2H, CH.sub.2 --Br); 3.8 (s, 3H, OCH.sub.3).

d) Methyl N-[2-(3"-bromophenylmethyliminoxymethyl)-phenyl]-carbamate (Table 7, No. 88)

0.95 g (39 mmol) of sodium hydride is added a little at a time to 7 g (33 mmol) of m-bromoacetophenone oxime in 100 ml of dimethylformamide. When the evolution of gas has ended, 8 g (33 mmol) of methyl N-(2-bromomethylphenyl)-carbamate (Example 3c), dissolved in 10 ml of dimethylformamide, are added dropwise. Stirring is carried out for 3 hours at room temperature, the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The organic phase is washed three times with water, dried and evaporated down. The residue crystallizes and is stirred thoroughly with methanol. 5.1 g (13.5 mmol=41%) of the title compound are obtained as a colorless solid.

mp.=124-125.degree. C.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 8.6 (s, broad, 1H, NH); 7.8-8.1 (m, 2H, aromatic); 7-7.6 (m, 6H, aromatic); 5.2 (s, 2H, O--CH.sub.2); 3.8 (s, 3H, O--CH.sub.3); 2.2 (s, 3H, CH.sub.3).

e) Methyl N-allyl-N-[2-(3"-bromophenylmethyliminoxymethyl)-phenyl]-carbamate (Table 7, No. 91)

0.1 g (4.1 mmol) of sodium hydride is added a little at a time to 1.3 g (3.5 mmol) of methyl N-[2-(3"-bromophenylmethyliminoxymethyl)-phenyl]-carbamate (Example 3d) in 20 ml of dimethylformamide. After gas evolution has ended, 0.5 g (3.8 mmol) of allyl bromide are added and stirring is carried out overnight at room temperature. Thereafter, the reaction mixture is diluted with water and extracted three times with ether. The combined ether phases are washed three times with water, dried over MgSO.sub.4 and evaporated down. 1.5 g (quantitative yield) of the title compound are obtained as a residue in the form of a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)):

7.8 (s, broad, 1H, aromatic); 7.1-7.6 (m, 7H, aromatic); 6.0 (m, 1H, C--CH.dbd.C); 5.1 (m, 4H, O--CH.sub.2 and C.dbd.CH.sub.2); 4.4 (m, 1H, N--CH.sub.A); 4.0 (m, 1H, N--CH.sub.B) 3.6-3.8 (2s, broad, O--CH.sub.3); 2.2 (s, 3H, CH.sub.3).

The compounds described in the Tables below can be prepared in a similar manner.

TABLE 1______________________________________ #STR22## No. X.sub.m______________________________________1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2- Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 ----CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)--CH.sub.3 333 3-C(.dbd.NO-Allyl)--CH.sub.3 334 4-C(.dbd.NO-Allyl)--CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 338 2-C(.dbd.NO-Propargyl)--CH.sub.3 339 3-C(.dbd.NO-Propargyl)--CH.sub.3 340 4-C(.dbd.NO-Propargyl)--CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Proparyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl-C.sub.6 H.sub.4) 396 2-(3'-Cl-C.sub.6 H.sub.4) 397 2-(4'-Cl-C.sub.6 H.sub.4) 398 3-(2'-Cl-C.sub.6 H.sub.4) 399 3-(3'-Cl-C.sub.6 H.sub.4) 400 3-(4'-Cl-C.sub.6 H.sub.4) 401 4-(2'-Cl-C.sub.6 H.sub.4) 402 4-(3'-Cl-C.sub.6 H.sub.4) 403 4-(4'-Cl-C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl-C.sub.6 H.sub.4) 488 2-O-(3'-Cl-C.sub.6 H.sub.4) 489 2-O-(4'-Cl-C.sub.6 H.sub.4) 490 3-O-(2'-Cl-C.sub.6 H.sub.4) 491 3-O-(3'-Cl-C.sub.6 H.sub.4) 492 3-O-(4'-Cl-C.sub.6 H.sub.4) 493 3-O-(4'-Cl-C.sub.6 H.sub.4) 494 4-O-(2'-Cl-C.sub.6 H.sub.4) 495 4-O-(3'-Cl-C.sub.6 H.sub.4) 496 4-O-(4'-Cl-C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 793 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 2______________________________________ #STR23## No. B______________________________________ 1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N--(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N--(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N--(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N--(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N--(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N--(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N--(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N--(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N--(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N--(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N--(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N--(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N--(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N--(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N--(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N--(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N--(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N--(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N--(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N--(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N--(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N--(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N--(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N--(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N--(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N--(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N--(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N--(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N--(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N--(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N--(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N--(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N--(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N--(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N--(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N--(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N--(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N--(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N--(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N--(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N--(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N--(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N--(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N--(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N--(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH.sub.3 -Oxazolyl-4 234 3-C.sub.6 H.sub.5 -Oxazolyl-4 235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 66 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazoly l-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 1-Naphthyl 385 2-Naphthyl______________________________________ TABLE 3______________________________________ #STR24## No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)--CH.sub.3 333 3-C(.dbd.NO-Allyl)--CH.sub.3 334 4-C(.dbd.NO-Allyl)--CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 338 2-C(.dbd.NO-Propargyl)--CH.sub.3 339 3-C(.dbd.NO-Propargyl)--CH.sub.3 340 4-C(.dbd.NO-Propargyl)--CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chlo roallyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Proparyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chl oroallyl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chl oroallyl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 2-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 4______________________________________ #STR25## No. B______________________________________1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4 -)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH.sub.3 -Oxazolyl-4 234 2-C.sub.6 H.sub.5 -Oxazolyl-4 235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 257 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazol yl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazo lyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazo lyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazol yl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl______________________________________ TABLE 5______________________________________ #STR26## No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 C(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 ----CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroall yl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.5) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.5) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.5) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.5) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.5) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.5) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.5) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.5) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.5) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5'______________________________________ TABLE 6______________________________________ #STR27## - No. B______________________________________ 1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-2 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.5 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4 -4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH.sub.3 -Oxazolyl-4 234 2-C.sub.6 H.sub.5 -Oxazolyl-4 235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl- 5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl- 5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2______________________________________ TABLE 7__________________________________________________________________________Selected physical data of some compoundsNo. Compound mp/.degree. C. IR/cm.sup.-1__________________________________________________________________________ 1 #STR28## -- 1707, 1484, 1457 1447, 1303, 1277 - 2 -- 1708, 1495, 1457 1449, 1304, 1241 - 3 111 30## - 4 73 R31## - 5 54 R32## - 6 -- 1706, 1496, 1456 1447, 1294, 1243 - 7 73 R34## - 8 57 R35## - 9 86 R36## - 10 -- 1709, 1599, 1497 1453, 1346, 1241 - 11 -- 1708, 1599, 1497 1455, 1447, 1397 1238 - 12 -- 1740, 1593, 1527 1489, 1456, 1252 1225 - 13 -- 1710, 1603, 1584 1490, 1451, 1364 1254 - 14 -- 1709, 1490, 1456 1447, 1379, 1300 1258 - 15 -- 1712, 1490, 1456 1447, 1378, 1298 1259 - 16 88 R43## - 17 -- 1710, 1511, 1451 1364, 1302, 1238 - 18 -- 1709, 1511, 1456 1447, 1379, 1301 1236 - 19 -- 1712, 1511, 1447 1378, 1298, 1233 - 20 -- 1738, 1723, 1582 1522, 1452, 1223 - 21 -- 1711, 1492, 1480 1447, 1362, 1303 1192, 1159 - 22 -- 1708, 1491, 1479 1446, 1376, 1300 1277, 1150 - 23 -- 1712, 1511, 1447 1378, 1298, 1233 - 24 -- 1736, 1582, 1523 1453, 1221 - 25 -- 1706, 1495, 1485 1363, 1303, 1193 1160 - 26 -- 1706, 1484, 1447 1377, 1301, 1280 1150 - 27 -- 1710, 1495, 1483 1446, 1376, 1299 1233 - 28 92 R55## - 29 -- 1709, 1489, 1447 1362, 1303, 1192 1159 - 30 -- 1706, 1484, 1447 1377, 1301, 1280 1150 - 31 -- 1711, 1488, 1446 1375, 1299, 1232 - 32 132 59## - 33 -- 1709, 1495, 1486 1451, 1366, 1161 1008 - 34 -- 1708, 1487, 1455 1447, 1379, 1300 1009 - 35 -- 1711, 1488, 1447 1378, 1297, 1232 1023, 1008 - 36 -- 1696, 1532, 1515 1453, 1267, 1245 1069 - 37 -- 1712, 1486, 1447 1361, 1303, 1191 1160 - 38 -- 1708, 1485, 1446 1376, 1300, 1274 - 39 -- 1709, 1484, 1446 1374, 1297, 1277 1232 - 40 -- 1712, 1495, 1457 1447, 1378, 1298 1237 - 41 110 68## - 42 -- 1739, 1593, 1528 1511, 1457, 1226 1035 - 43 102 70## - 44 -- 1708, 1513, 1457 1447, 1378, 1302 1246, 1035 - 45 102 72## - 46 74 R73## - 47 -- 1709, 1606, 1512 1364, 1245, 1228 1171, 1162, 1033 1005 - 48 59 R75## - 49 -- 1709, 1447, 1364 1261, 1157, 1034 1007 - 50 -- 1709, 1576, 1446 1379, 1300, 1260 1239, 1156, 1037 - 51 89 R78## - 52 -- 1740, 1593, 1575 1527, 1457, 1316 1300, 1224, 1067 1029 - 53 81 R80## - 54 -- 1711, 1574, 1447 1365, 1322, 1303 1213, 1160, 1033 1008 - 55 -- 1709, 1574, 1446 1378, 1321, 1301 1284, 1213, 1034 - 56 -- 1711, 1505, 1451 1365, 1304, 1245 1160, 1143, 1035 1007 - 57 63 R84## - 58 -- 1710, 1487, 1450 1364, 1301, 1246 1160, 1030, 1006 - 59 -- 1708, 1487, 1449 1378, 1300, 1247 1030, 1009 - 60 -- 1743, 1593, 1528 1502, 1457, 1301 1255, 1190, 1066 1006 - 61 77 R88## - 62 -- 1712, 1503, 1453 1363, 1303, 1259 1244, 1160, 1136 1006 - 63 -- 1711, 1503, 1457 1447, 1380, 1301 1258, 1239, 1136 1015 - 64 92 1743, 1593, 1528 1502, 1457, 1301 1255, 1190, 1066 1006 - 65 90 R92## - 66 70 R93## - 67 75 R94## - 68 108 95## - 69 93 R96## - 70 74 R97## - 71 -- 1712, 1504, 1450 1363, 1303, 1255 1222, 1159, 1134 - 72 -- 1712, 1510, 1498 1450, 1365, 1327 1246, 1150, 1035 1005 - 73 60 R100## - 74 -- 1711, 1509, 1497 1451, 1363, 1302 1264, 1193, 1156 1129 - 75 -- 1710, 1496, 1475 1149, 1365, 1301 1263, 1195, 1159 - 76 66 R103## - 77 86 R104## - 78 91 R105## - 79 100 106## - 80 -- 1710, 1593, 1497 1452, 1364, 1323 1297, 1193, 1165 1153 - 81 -- 1715, 1510, 1447 1367, 1324, 1299 1243, 1149, 1027 996 - 82 -- 1710, 1509, 1456 1446, 1377, 1326 1300, 1241, 1149 1306 - 83 -- 1723, 1509, 1453 1437, 1316, 1292 1241, 1149, 1064 1036 - 84 -- 1738, 1611, 1581 1539, 1446, 1312 1301, 1231, 1201 1067 - 85 -- 1713, 1504, 1447 1375, 1313, 1300 1233, 1143, 1027 - 86 -- 1711, 1486, 1447 1376, 1300, 1281 1150, 1034, 1013 - 87 -- 1714, 1487, 1447 1376, 1300, 1231 1023, 999 - 88 -- 1733, 1594, 1533 1457, 1306, 1231 1013, 984 - 89 -- 1721, 1495, 1453 1437, 1313, 1290 1239, 1123 - 90 -- 1709, 1453, 1366 1303, 1228, 1160 1014 - 91 -- 1708, 1455, 1447 1378, 1299, 1282 1015, 996 - 92 -- 1710, 1447, 1378 1296, 1232, 1045 1023, 995 - 93 108 120## - 94 -- 1717, 1495, 1457 1444, 1376, 1298 1241, 1228, 1193 - 95 -- 1739, 1614, 1603 1542, 1450, 1262 129, 1179 - 96 170 123## - 97 180 124## - 98 173 125## - 99 150 126## - 100 129 127## - 101 112 128## - 102 116 129## - 103 127 130## - 104 108 131## - 105 -- 1710, 1486, 1447 1363, 1307, 1193 1159, 1031, 1006 - 106 -- 1706, 1484, 1447 1376, 1302, 1279 1150, 1031, 1011 923 - 107 -- 1711, 1484, 1446 1376, 1298, 1232 1144, 1024, 995, 922 - 108 147 135## - 109 -- 1716, 1455, 1445 1376, 1297, 1279 1097, 1069, 1017 1008 - 110 -- 1718, 1487, 1447 1394, 1374, 1306 1232, 1025, 1008 - 111 109 138## - 112 -- 1706, 1487, 1450 1387, 1304, 1276 1155, 1022, 1009 769 - 113 -- 1706, 1487, 1453 1383, 1312, 1301 1274, 1155, 1033 1008 - 114 115 141## - 115 167 142## - 116 -- 1729, 1575, 1565 1545, 1523, 1445 1434, 1224, 1060 - 117 110 144## - 118 77 R145## - 119 -- 1712, 1494, 1447 1378, 1298, 1232 1045, 1024, 818, 771 - 120 115 147## - 121 -- 1717, 1455, 1445 1376, 1298, 1278 1097, 1068, 1016 999 - 122 81 R149## - 123 -- 1712, 1493, 1447 1378, 1297, 1232 1047, 1024, 998, 772 - 124 107 151## - 125 -- 1717, 1455, 1445 1376, 1298, 1279 1096, 1068, 1017 999 - 126 128 153## - 127 -- 1712, 1492, 1447 1378, 1298, 1232 1096, 1044, 1023 - 128 119 155## - 129 -- 1717, 1492, 1455 1445, 1376, 1298 1096, 1068, 1012 1000 - 130 133 157## - 131 -- 1712, 1511, 1494 1447, 1378, 1298 1232, 1045, 1024 837 - 132 113 159## - 133 -- 1716, 1511, 1455 1445, 1376, 1298 1228, 1097, 1068 999 - 134 -- 1737, 1592, 1529 1509, 1489, 1455 1303, 1231, 1067 1014 - 135 -- 1712, 1586, 1507 1489, 1454, 1378 1297, 1239, 1023 - 136 148 163## - 137 -- 1716, 1587, 1507 1490, 1455, 1375 1298, 1240, 1068 - 138 90 R165## - 139 -- 1719, 1495, 1464 1446, 1375, 1295 1239, 1104, 1075 1014 - 140 -- 1715, 1495, 1463 1448, 1376, 1298 1239 - 141 134 168## - 142 -- 1744, 1583, 1522 1503, 1458, 1442 1223, 1304, 1035 1004 - 143 -- 1720, 1465, 1446 1372, 1296, 1280 1243, 1144, 1035 1014 - 144 -- 1716, 1505, 1465 1448, 1374, 1298 1279, 1241, 1141 999 - 145 109 172## - 146 158 173## - 147 -- 1718, 1463, 1445 1376, 1294, 1104 1073, 1024, 1010 - 148 -- 1714, 1462, 1447 1377, 1297, 1238 1025, 1009 - 149 140R176##__________________________________________________________________________

Example 4

Methyl N-(2-methylphenyl)-N-methoxy-carbamate (Table 14, No. 1)

a) Methyl N-(2-methylphenyl)-N-hydroxy-carbamate

At 25-30.degree. C., 14.0 g (0.148 mol) of methyl Chloroocarbonate is added dropwise to 16.4 g of N-(2-methylphenyl)-hydroxylamine (crude product, obtained according to Bamberger et al., Ann. Chem. 316 (1901), 278) and 12.9 g (0.163 mol) of pyridine in 100 ml of methylene Chloroide. The mixture is stirred overnight at room temperature (20.degree. C.) and is then extracted with dilute hydrochloroic acid and water. The organic phase is dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 7 g (39 mmol) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 8.6 (s, broad, OH); 7.3 (m, 4H, phenyl); 3.75 (s, 3H, OCH.sub.3); 2.3 (s, 3H, CH.sub.3).

b) Methyl N-(2-methylphenyl)-N-methoxy-carbamate (Table 14, No. 1)

At 20-30.degree. C., 1.1 g (44.1 mmol) of sodium hydride is added in portions to 6.6 g (36.5 mmol) of the hydroxyl compound from Example 4a in 50 ml of dimethylformamide. Upon conclusion of gas evolution 5.7 g (40.1 mmol) of methyl iodide is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl-t-butyl ether. The combined organic phases are dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 5.2 g (27mmol=73%) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.25 (m, 4H, phenyl); 3.8; 3.75 (s, 3H, OCH.sub.3 ; 3.75 (s, 3H, OCH.sub.3); 2.3 (s, 3H, CH.sub.3).

Example 5

Methyl N-(2-bromomethylphenyl)-N-methoxy-carbamate (Table 14, No. 2)

2.5 g (12.8 mmol) of the N-methoxycarbamate from Example 4b, 2.5 g (14.1 mmol) of N-bromosuccinimide and a spatula-tip (1 g) of azoisobutyrodinitrile in 20 ml of carbon tetraChloroide were irradiated with a 300 W UV lamp; the reaction mixture heated up to 30-40.degree. C. After three hours the reaction mixture is extracted twice with water. The organic phase is dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 1.4 g (5.1 mmol 40%) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.5 (m, 1H, phenyl); 7.35 (m, 3H, phenyl); 4.55 (s, 2H, CH.sub.2 --Br); 3.8 (2s, 6H, 2.times. OCH.sub.3).

Example 6

Methyl N-[2-(2'-methylphenoxymethyl)-phenyl]-N-methoxy-carbamate (Table 14, No. 3)

1.2 g (4.4 mmol) of the methyl bromide from Example 5, 0.45 g (4.2 mmol) o-cresol and 0.7 g (4.8 mmol) of K.sub.2 CO.sub.3 in 30 ml of dimethylformamide are stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl-t-butyl ether. The combined organic phases are dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 1.2 g of the title compound containing o-cresol as impurity. The mixture is heated in a furnace at about 1 mbar for about 1 hour at 125.degree. C. The residue obtained is 0.9 g (3 mmol=68%) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 3H, phenyl); 7.15 (m, 2H, phenyl); 6.9 (t, broad, 2H, phenyl); 5.15 (s, 2H, O--CH.sub.2); 3.8 (s, 3H, OCH.sub.3), 3.75 (s, 3H, OCH.sub.3); 2.3 (s, 3H, CH.sub.3).

TABLE 8______________________________________ #STR177## No Xm______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl2, 5-NO2 254 2,4-Cl2, 6-NO2 255 2,6-Cl2, 4-NO2 256 2,6-Br2, 4-NO2 257 2,6-I2, 4-NO2 258 2-CH3, 5-i-C3H7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO2CH3 261 4-CO2CH3 262 2-CO2(C2H5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 ----CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)--CH.sub.3 333 3-C(.dbd.NO-Allyl)--CH.sub.3 334 4-C(.dbd.NO-Allyl)--CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 338 2-C(.dbd.NO-Propargyl)--CH.sub.3 339 3-C(.dbd.NO-Propargyl)--CH.sub.3 340 4-C(.dbd.NO-Propargyl)--CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO--(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloro allyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Proparyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH3O2C--C6H4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C6H5 476 4-O--C6H5 478 2-O--(2'-F--C.sub.6 H.sub.4) 479 2-O--(3'-F--C.sub.6 H.sub.4) 480 2-O--(4'-F--C.sub.6 H.sub.4) 481 3-O--(2'-F--C.sub.6 H.sub.4) 482 3-O--(3'-F--C.sub.6 H.sub.4) 483 3-O--(4'-F--C.sub.6 H.sub.4) 484 4-O--(2'-F--C.sub.6 H.sub.4) 485 4-O--(3'-F--C.sub.6 H.sub.4) 486 4-O--(4'-F--C.sub.6 H.sub.4) 487 2-O--(2'-Cl--C.sub.6 H.sub.4) 488 2-O--(3'-Cl--C.sub.6 H.sub.4) 489 2-O--(4'-Cl--C.sub.6 H.sub.4) 490 3-O--(2'-Cl--C.sub.6 H.sub.4) 491 3-O--(3'-Cl--C.sub.6 H.sub.4) 492 3-O--(4'-Cl--C.sub.6 H.sub.4) 493 3-O--(4'-Cl--C.sub.6 H.sub.4) 494 4-O--(2'-Cl--C.sub.6 H.sub.4) 495 4-O--(3'-Cl--C.sub.6 H.sub.4) 496 4-O--(4'-Cl--C.sub.6 H.sub.4) 497 2-O--(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O--(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O--(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O--(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O--(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O--(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O--(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O--(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O--(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O--(4'-CH.sub.3 --CO--C6H4) 509 3-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O--(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 516 2-O--(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 517 2-O--(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 518 3-O--(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 519 3-O--(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 520 3-O--(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 521 4-O--(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 522 4-O--(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 523 4-O--(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 524 2-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O--(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O--(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O--(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O--(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O--(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O--(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O--(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O--(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O--(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O--(2'-NC--C.sub.6 H.sub.4) 552 2-O--(3'-NC--C.sub.6 H.sub.4) 553 2-O--(4'-NC--C.sub.6 H.sub.4) 554 3-O--(2'-NC--C.sub.6 H.sub.4) 555 3-O--(3'-NC--C.sub.6 H.sub.4) 556 3-O--(4'-NC--C.sub.6 H.sub.4) 557 4-O--(2'-NC--C.sub.6 H.sub.4) 558 4-O--(3'-NC--C.sub.6 H.sub.4) 559 4-O--(4'-NC--C.sub.6 H.sub.4) 560 2-O--(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O--(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O--(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O--(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O--(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O--(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O--(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O--(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O--(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 666 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chlor oallyl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chlor oallyl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 9______________________________________ #STR178## No. B______________________________________ 1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N--(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N--(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N--(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N--(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N--(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N--(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N--(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N--(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N--(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N--(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N--(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N--(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N--(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N--(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N--(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N--(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N--(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N--(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N--(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N--(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N--(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N--(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N--(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N--(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N--(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N--(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N--(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N--(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N--(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N--(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N--(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N--(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N--(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N--(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N--(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N--(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N--(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N--(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N--(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N--(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N--(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N--(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N--(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N--(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N--(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH.sub.3 --Oxazolyl-4 234 2-C.sub.6 H.sub.5 --Oxazolyl-4 235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2-4-Triazoly l-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2-4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2-4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2-4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2-4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2-4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl______________________________________ TABLE 10______________________________________ #STR179## No. X.sub.m______________________________________1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C2H5)3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)-CH.sub.3 299 3-CO--CH(CH.sub.3)-CH.sub.3 300 4-CO--CH(CH.sub.3)-CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)-CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)-CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)-CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 ----CH(CH.sub.3)-CO 320 2-C(.dbd.NOCH.sub.3)-CH.sub.3 321 3-C(.dbd.NOCH.sub.3)-CH.sub.3 322 4-C(.dbd.NOCH.sub.3)-CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)-CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)-CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)-CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)-CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)-CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)-CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)-CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)-CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)-CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)-CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)-CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)-CH.sub.3 344 2-C(.dbd.NO--CH.sup.2 --C.sub.6 H.sub.5)-CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)-CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)-CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Proparyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C-C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH3O2C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF3--C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH3--CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O2N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 793 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 11______________________________________ #STR180## No. B______________________________________1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4 -)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH.sub.3 -Oxazolyl-4 234 2-C.sub.6 H.sub.5 -Oxazolyl-4 235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 257 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazol yl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazo lyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazo lyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazol yl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl______________________________________ TABLE 12______________________________________ #STR181## No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C4H9)2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C6H11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 3-CH.sub.3, 4-Cl 199 4-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)--CH.sub.3 333 3-C(.dbd.NO-Allyl)--CH.sub.3 334 4-C(.dbd.NO-Allyl)--CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 338 2-C(.dbd.NO-Propargyl)--CH.sub.3 339 3-C(.dbd.NO-Propargyl)--CH.sub.3 340 4-C(.dbd.NO-Propargyl)--CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chlo roallyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Proparyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C6H5 385 4-C6H5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C6H5 476 4-O--C6H5 478 2-O--(2'-F--C.sub.6 H.sub.4) 479 2-O--(3'-F--C.sub.6 H.sub.4) 480 2-O--(4'-F--C.sub.6 H.sub.4) 481 3-O--(2'-F--C.sub.6 H.sub.4) 482 3-O--(3'-F--C.sub.6 H.sub.4) 483 3-O--(4'-F--C.sub.6 H.sub.4) 484 4-O--(2'-F--C.sub.6 H.sub.4) 485 4-O--(3'-F--C.sub.6 H.sub.4) 486 4-O--(4'-F--C.sub.6 H.sub.4) 487 2-O--(2'-Cl--C.sub.6 H.sub.4) 488 2-O--(3'-Cl--C.sub.6 H.sub.4) 489 2-O--(4'-Cl--C.sub.6 H.sub.4) 490 3-O--(2'-Cl--C.sub.6 H.sub.4) 491 3-O--(3'-Cl--C.sub.6 H.sub.4) 492 3-O--(4'-Cl--C.sub.6 H.sub.4) 493 3-O--(4'-Cl--C.sub.6 H.sub.4) 494 4-O--(2'-Cl--C.sub.6 H.sub.4) 495 4-O--(3'-Cl--C.sub.6 H.sub.4) 496 4-O--(4'-Cl--C.sub.6 H.sub.4) 497 2-O--(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O--(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O--(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O--(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O--(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O--(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O--(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O--(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O--(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O--(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 516 2-O--(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 517 2-O--(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 518 3-O--(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 519 3-O--(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 520 3-O--(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 521 4-O--(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 522 4-O--(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 523 4-O--(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 524 2-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O--(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O--(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O--(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O--(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O--(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O--(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O--(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O--(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O--(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O--(2'-NC--C.sub.6 H.sub.4) 552 2-O--(3'-NC--C.sub.6 H.sub.4) 553 2-O--(4'-NC--C.sub.6 H.sub.4) 554 3-O--(2'-NC--C.sub.6 H.sub.4) 555 3-O--(3'-NC--C.sub.6 H.sub.4) 556 3-O--(4'-NC--C.sub.6 H.sub.4) 557 4-O--(2'-NC--C.sub.6 H.sub.4) 558 4-O--(3'-NC--C.sub.6 H.sub.4) 559 4-O--(4'-NC--C.sub.6 H.sub.4) 560 2-O--(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O--(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O--(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O--(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O--(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O--(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O--(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O--(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O--(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5'______________________________________ TABLE 13______________________________________ #STR182## - No. B______________________________________ 1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH.sub.3 -Oxazolyl-4 234 2-C.sub.6 H.sub.5 -Oxazolyl-4 235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 257 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N-CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 -N-CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 -N-CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3______________________________________ TABLE 14__________________________________________________________________________Selected physical data of some compoundsNo. Compound .sup.1 H-NMR (ppm)__________________________________________________________________________ 1 3.8 (s, 3H); 3.75 (s, 3H) - 2 3.8 (2s, 2 .times. 3H) - 3 3.8 (s, 3H); 3.75 (s, 3H) - 4 3.95 (q, 2H, I = 7.5 Hz); 3.8 (s, 3H) - 5 4.05 (q, 2H, I = 7.5 Hz); 3.85 (s, 3H) - 6 4.0 (q, 2H, I = 7.5 Hz); 3.8 (s, 3H) - 7 3.8 (s, 3H); 3.75 (s, 3H) - 8 3.8 (s, 3H); 3.75 (s, 3H) - 9 3.85 (s, 3H); 3.8 (s, 3H) - 10 4.0 (s, 3H); 3.8 (s, 3H), 3.75 (s, 3H) - 11 3.8 (s, 3H); 3.75 (s, 3H) - 12 3.8 (s, 3H); 3.75 (s, 3H) - 13 3.8 (s, 3H); 3.75 (s, 3H) - 14 3.8 (s, 3H); 3.75 (s, 3H) 66 - 15 3.8 (s, 3H); 3.75 (s, 3H) - 16 4.0 (q, 2H, I = 7.5 Hz); 3.8 (s, 3H) - 17 3.8 (2s, each 3H) - 18 3.8 (2s, each 3H) - 19 3.8 (s, 3H); 3.75 (s, 3H) - 20 3.8 (s, 3H); 3.75 (s, 3H) - 21 3.8 (s, 3H); 3.75 (s, 3H) - 22 3.8 (s, 3H); 3.75 (s, 3H) - 23 3.8 (s, 3H); 3.75 (s, 3H) - 24 3.8 (s, 6H) - 25 3.75 (2s, each 3H) - 26 3.8 (s, 3H); 3.75 (s, 3H) - 27 3.8 (s, 3H); 3.75 (s, 3H) - 28 3.8 (s, 3H); 3.75 (s, 3H) - 29 3.8 (s, 3H); 3.75 (s, 3H) - 30 3.8 (s, 6H)__________________________________________________________________________ TABLE 52______________________________________Selected physical data of some compounds #STR213## .sup.1 H-NMR (ppm) or IR No. X.sub.m mp (.degree. C.) (cm.sup.-1)______________________________________ 1 H 3.75(2s, each 3H) 2 2-CH.sub.3 3.75(2s, each 3H) 3 3-CH.sub.3 3.75(2s, each 3H) 4 2,4-(CH.sub.3).sub.2 3.75(2s, each 3H) 5 4-C.sub.2 H.sub.5 3.75(2s, each 3H) 6 4-i-C.sub.3 H.sub.7 3.75(2s, each 3H) 7 4-t-C.sub.4 H.sub.9 3.75(2s, each 3H) 8 3,4-(CH.sub.3).sub.2 3.75(2s, each 3H) 9 3-Cl 3.75(2s, each 3H) 10 3-Br 3.75(2s, each 3H) 11 3-CF.sub.3 3.75(2s, each 3H) 12 4-Br 3.75(2s, each 3H) 13 4-F 3.75(2s, each 3H) 14 4-CF.sub.3 3.75(2s, each 3H) 15 4-OCH.sub.3 3.8(s, 3H); 3.75(2s, each 3H) 16 4-CN 3.75(2s, each 3H) 17 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 3.75(2s, each 3H) 18 3,4-Cl.sub.2 3.75(2s, each 3H) 19 3-CH.sub.3 -4-OCH.sub.3 3.85(s, 3H); 3.75(2s, each 3H) 20 4-NO.sub.2 112 21 3,5-(CH.sub.3).sub.2 3.75(2s, each 3H) 22 3-CH.sub.3 -4-Cl 3.75(2s, each 3H) 23 3-Cl-4-CH.sub.3 3.75(2s, each 3H)______________________________________ TABLE 53______________________________________Selected physical data of some compounds #STR214## mp .sup.1 H-NMR (ppm) or IR No. X.sub.m (.degree. C.) (cm.sup.-1)______________________________________ 1 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--O-- 3.8(s, 3H); 3.75(s, 3H) C.sub.2 H.sub.5 2 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--O- 3.8(s, 3H); 3.75(s, 3H) (trans-CH.sub.2 --CH.dbd.CHCl) 3 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N-- 3.95(s, 3H); 3.8(s, 3H); OCH.sub.3 3.75(s, 3H) 4 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N-- 3.8(s, 3H); 3.75(s, 3H) OC.sub.2 H.sub.5 5 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--O- 3.85(s, 3H); 3.75(s, 3H) (trans-CH.sub.2 --CH.dbd.CHCl) 6 2-CH.sub.3 -4-C(C.sub.2 H.sub.5).dbd.N--OCH.sub.3 3.95(s, 3H); 3.8(s, 3H); 3.75(s, 3H) 7 2-CH.sub.3 -4-C(C.sub.2 H.sub.5).dbd.N-- 3.8(s, 3H); 3.75(s, 3H) O--C.sub.2 H.sub.5 8 2-CH.sub.3 -4-C(C.sub.2 H.sub.5).dbd.N-- 3.8(s, 3H); 3.75(s, 3H) O-Allyl 9 2-CH.sub.3 -4-C(C.sub.2 H.sub.5).dbd.N-- 3.8(s, 3H); 3.75(s, 3H) O-(trans-CH.sub.2 --CH.dbd.CHCl) 10 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5).dbd. 3.95(S, 3H); 3.8(s, 3H); N--OCH.sub.3 3.75(s, 3H) 11 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5).dbd. 3.8(s, 3H); 3.75(s, 3H) N--O--C.sub.2 H.sub.5 12 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5).dbd. 3.8(s, 3H); 3.75(s, 3H) N--O-Allyl 13 2-Cl 3.8(s, 3H); 3.75(s, 3H) 14 4-Cl 3.8(s, 3H); 3.75(s, 3H) 15 2-CH.sub.3 -4-Cl 3.8(s, 3H); 3.75(s, 3H) 16 2-Cl-4-CH.sub.3 3.8(s, 3H); 3.75(s, 3H) 17 2-Cl-5-CH.sub.3 3.8(s, 3H); 3.75(s, 3H) 18 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd. 3.8(s, 3H); 3.75(s, 3H) N--O-Allyl 19 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5).dbd. 3.8(s, 3H); 3.75(s, 3H) N--O-(trans-CH.sub.2 --CH.dbd.CHCl)______________________________________ TABLE 54______________________________________ #STR215## - No. B______________________________________ 1 2-Pyridyl 2 3-Trifluoromethyl-2-pyridyl 3 5-Trifluoromethyl-2-pyridyl 4 3,5-Bis-(trifluoromethyl)-2-pyridyl 5 3,5-Dichloro-2-pyridyl 6 3-Chloro-5-trifluoromethyl-2-pyridyl 7 3,5-Dichloro-2-pyridyl 8 2-Chloro-4-trifluoromethylphenyl 9 2-Benzothiazolyl 10 5-Chloro-4-methyl-2-benzimidazolyl 11 2-Benzoxazolyl 12 1-Methyl-5-trifluoromethylimi- dazo[5,4-a]-pyridin-2-yl 13 5-Chloro-2-pyrimidinyl 14 4-Methyl-5-phenyl-2-thiazolin-2-yl 15 4-Methyl-5-phenyl-2-oxazolin-2-yl 16 7-Trifluoromethyl-4-quinolinyl______________________________________ TABLE 55______________________________________Selected physical data of some compounds #STR216## -No. X.sub.m mp (.degree. C.) .sup.1 H-NMR (ppm) or IR (cm.sup.-1)______________________________________1 H 3.75(s, 3H); 3.65(s, 3H) 2 4-OCH.sub.3 3.8(s, 3H); 3.75(s, 3H); 3.65(s, 3H) 3 4-CH.sub.3 3.75(s, 3H); 3.65(s, 3H) 4 4-Cl 3.75(s, 3H); 3.65(s, 3H) 5 4-CF.sub.3 3.75(s, 3H); 3.65(s, 3H) 6 3,5-(CF.sub.3).sub.2 3.75(s, 3H); 3.65(s, 3H) 7 2,4-Cl.sub.2 3.75(s, 3H); 3.65(s, 3H) 8 3,4-Cl.sub.2 3.75(s, 3H); 3.65(s, 3H)______________________________________

Example 6

O-Methyl-N-(2-methylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 1)

a) N-(2-Methylphenyl)-N-propionyl-hydroxylamine

At 25 to 30.degree. C., 12,5 g (0.135 mol) of propionyl Chloroide and then 10.7 g (0.135 mol) of pyridine are dripped into 30 g of N-(2-methylphenyl)-hydroxylamine (crude product, prepared according to Bamberger et al., Anm. Chem. 316 (1901), 278; content approx. 80%=0.2 mol) in 500 ml of methylene Chloroide. The mixture is stirred for 30 minutes at room temperature, and is then extracted with dilute hydrochloroic acid and water. The organic phase is dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 22.7 g (0.127 mol=63%) of the title compound as a yellow oil.

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 9.4 (s, broad, 1H, OH); 7.2 (m, 4H, phenyl); 2.4 (s, 3H, CH.sub.3); 2.1 (q, broad, 2H, CH.sub.2); 1.1 (t, 3H, I=7 Hz, CH.sub.3).

b) O-Methyl-N-(2-methylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 1)

At 25 to 30.degree. C., a solution of 22.7 g (0.127 mol) (Example 6a) of N-(2-methylphenyl)-N-propionyl-hydroxylamine in 50 ml of dimethylformamide is dripped into a stirred mixture of 3.4 g (0.14 mol) of NaH in 150 ml of dimethylformamide. After completion of gas evolution (15 mins) 18.4 g (0.13 mol) of methyl iodide is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 18 g (0.081 mol=64%) of the title compound as a yellow oil.

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 7.2 (m, 4H, phenyl); 3.7 (s, broad, 3H, OCH.sub.3); 2.6 (s, very broad, 2H, CH.sub.2); 2.3 (s, 3H, CH.sub.3); 1.2 (s, broad, 3H, CH.sub.3).

Example 7

O-Methyl-N-(2-bromomethylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 2)

A mixture of 10 g (51.8 mmol) of the hydroxylamine derivative from Example 1, 11 g (61 mmol) of N-bromosuccinimide and 0.1 g of azoisobutyrodinitrile in 100 ml of CCl.sub.4 is refluxed. One drop of bromine is added and the mixture is refluxed for a further 2.5 hours. The reaction mixture is cooled to room temperature, washed with water, dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained in this sequence 3.4 g (7.9 mmol=15%) of O-methyl-N-(2-bromomethylphenyl)-d-(.alpha.,.alpha.-dibromopropionyl)-hydroxylamine, 3.8 g (10.8 mmol=21%) of O-methyl-N-(2-bromomethylphenyl)-N-(.alpha.-bromopropionyl)-hydroxylamine, 2.3 g (8.5 g (8.5 mmol=16%) of the title compound and 3.5 g of starting material, each as brown oils.

a) O-Methyl-N-(2-bromomethylphenyl)-N-(.alpha.,.alpha.-dibromopropionyl)-hydroxylamine

7.55 (m, 1H, phenyl); 7.4 (m, 3H, phenyl); 4.5 (s, 2H, CH.sub.2, Br); 3.8 (s, 3H, OCH.sub.3); 2.75 (s, 3H, CH.sub.3).

b) O-Methyl-N-(2-bromomethylphenyl)-N-(.alpha.-bromopropionyl)-hydroxylamine

7.5 (s, broad, 1H, phenyl); 7.4 (s, broad, 3H, phenyl); 5.15 (s, broad, 1H, CH--Br); 4.5 (dd, broad, 2H, CH.sub.2 --Br); 3.8 (s, 3H, OCH.sub.3); 1.85 (s, broad, 3H, CH.sub.3).

c) O-Methyl-N-(2-bromomethylphenyl)-N-propionyl-hydroxylamine

7.5 (m, 1H, phenyl); 7.35 (m, 3H, phenyl); 4.5 (s, broad, 2H, CH.sub.2 --Br); 3.75 (s, 3H, OCH.sub.3); 2.55 (s, very broad, CH.sub.2); 1.2 (t, 3H, I=7 Hz, CH.sub.3).

Example 8

O-Methyl-N-(2-(2'-methylphenyloxymethyl)-phenyl)-N-propionyl-hydroxylamine (Table 21, No. 3)

0.12 g (5 mmol) of sodium hydride is added to a solution of 0.4 g (3.7 mmol) of o-cresol in 5 ml of dimethylformamide. Upon completion of gas evolution, 1 g (3.6 mmol) of the benzyl bromide from Example 2c is added and the mixture is stirred for 2 hours at room temperature. The reaction mixture is diluted with water and extracted three times with methyl tert-butyl ether. The combined organic phases are washed with water, dried over MgSO.sub.4 and evaporated down. The residue is chromatographed with mixtures of cyclohexane and ethyl acetate using Al.sub.2 O.sub.3 and silica gel. There is obtained 0.4 g (1.33 mmol=37%) of the title compound as a yellow oil.

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 7.7 (d, broad, 1H, phenyl); 7.35 (m, 3H, phenyl); 7.1 (m, 2H, phenyl); 6.85 (t, broad, 2H, phenyl); 5.05 (s, 2H, OCH.sub.3); 3.7 (s, 3H, OCH.sub.3); 2.55 (s, very broad, 2H, CH.sub.2); 2.3 (s, 3H, CH.sub.3); 1.2 (t, broad, 3H, CH.sub.3).

Example 9

N-Methyl-N'-methoxy-N'-2-methylphenylurea (Table 21, No. 5)

a) Phenyl N-hydroxy-N-(2-methylphenyl)-carbamate

A mixture of 2.5 g (20 mmol) of N-(2-methylphenyl)-hydroxylamine (crude product, obtained according to Bamberger et al., Anm. Chem. 316 (1901), 278), 3.5 g (25 mmol) of K.sub.2 CO.sub.3 and 3.5 g (22 mmol) of phenyl Chlorooformate in 20 ml of CH.sub.2 Cl.sub.2 is stirred for 2 hours at room temperature. The reaction mixture is then extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 2.0 g (8.2 mmol=42%) of the title compound as a colorless solid (mp=98.degree. C.).

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 7-7.6 (m, 10H, phenyl, OH); 2.35 (s, 3H, CH.sub.3).

b) Phenyl N-methoxy-N-(2-methylphenyl)-carbamate

A mixture of 2.0 g (8.2 mmol) of the phenyl carbamate from Example 4a, 2 g (15 mmol) of K.sub.2 CO.sub.3 and 1.3 g (10 mmol) of dimethyl sulfate in 20 ml of acetone is stirred for 3 hours at room temperature. The reaction mixture is then filtered and evaporated down, and the residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 1.5 g (5.8 mmol=71%) of the title compound as a colorless oil, which slowly crystallizes (mp=60.degree. C.).

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 7.1-7.5 (m, 9H, phenyl); 3.8 (s, 3H, OCH.sub.3); 2.4 (s, 3H, CH.sub.3).

c) N-Methyl-N'-methoxy-N'-2-methylphenylurea (Table 21, No. 5)

1.5 g (5.8 mmol) of the phenyl carbamate from Example 4b in 20 ml of 40% strength aqueous methylamine solution is stirred for 1 hour at 50.degree. C. The reaction mixture is then cooled and extracted with CH.sub.2 Cl.sub.2. The combined organic phases are dried over MgCO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 0.6 g (3.1 mol=53%) of the title compound as a colorless solid (mp 99.degree. C.).

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 7.2 (m, 4H, phenyl); 5.9 (s, broad, 1H, NH); 3.6 (s, 3H, OCH.sub.3); 2.9 (d, 3H, I=approx. 2 Hz, N--CH.sub.3); 2.3 (s, 3H, CH.sub.3).

Example 18

N-Methyl-N'-methoxy-N'-(2-2',5'-dimethylphenoxymethyl)-phenyl)-urea

a) Phenyl N-methoxy-N-(2-bromomethylphenyl)-carbamate

A mixture of 125 g (0.486 mol) of methyl N-methoxy-N-(2-methylphenyl)-carbamate (Example 4b), 88 g (0.494 mol) of N-bromosuccinimide and 1 g of azoisobutyrodinitrile (AIBN) in 800 ml of CCl.sub.4 is refluxed for about 12 hours. 10 g of N-bromosuccinimide is then added and the mixture is refluxed for about 4 hours. The reaction mixture is extracted with water and sodium thiosulfate solution, and the organic phase is dried over MgSO.sub.4 and evaporated down under reduced pressure. The residue crystallizes, is stirred with hexane/methyl tert-butyl ether and suction dried. There is obtained 107 g (63%) of the title compound as a colorless solid.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.1-7.6 (m, 9H, phenyl); 4.65 (s, 2H, CH.sub.2 Br); 3.9 (s, 3H, OCH.sub.3).

b) Phenyl N-methoxy-N-(2-(2',5'-dimethylphenoxymethyl)-phenyl)-carbamate

A mixture of 7 g (20 mmol) of the bromide of Example 5a and 3.3 g (22 mmol) of sodium iodide in 50 ml of acetone is refluxed for 30 minutes. The precipitated solid is then filtered off and the organic phase is evaporated down under reduced pressure. The crude product obtained is the iodide corresponding to Example 5a, which is used in the next reaction without any further purification.

The crude product obtained above is dissolved in 100 ml of dimethylformamide, 3 g (21.6 mmol) of K.sub.2 CO.sub.3 and 7.3 g (60 mmol) of 2,5-dimethylphenol are added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography using methylene chloride/cyclohexane (1:2) over Al.sub.2 O.sub.3. There is obtained 7.3 g (94%) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in PPM): 7.7 (d, broad, 1H, phenyl); 7-7.6 (m, 9H, phenyl); 6.7 (m, 2H, phenyl); 5.2 (s, 2H, OCH.sub.2); 3.85 (s, 3H, OCH.sub.3); 2.3 (s, 6H, 2.times.CH.sub.3).

c) N-Methyl-N'-methoxy-N'-(2-(2',5'-dimethylphenoxymethyl)-phenyl)-urea (Table 1, No. V.71)

A mixture of 3.4 g (8.8 mmol) of the phenyl carbamate of Example 5b and 20 ml of 40% strength aqueous methylamine solution is stirred for 2 hours at 50.degree. C. The mixture is allowed to cool and is then extracted with methylene chloride. The organic phase is evaporated down and the residue is purified by column chromatography with mixtures of cyclohexane/ethyl acetate. There is obtained 1 g (36%) of the title compound as a colorless solid (mp=101.degree. C.).

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in PPM): 7.75 (m, 1H, phenyl); 6.6-7.4 (m, 6H, phenyl); 6.0 (s, broad, NH); 5.15 (s, 2H, OCH.sub.2); 3.65 (s, 3H, OCH.sub.3); 2.9 (d, 3H, N--CH.sub.3); 2.3 (s, 3H, CH.sub.3); 2.25 (s, 3H, CH.sub.3).

The compounds listed in the tables below may be prepared analogously. Compound I.1 from Table 15 has for instance the following formula ##STR217##

TABLE 15______________________________________No. Xm______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3 , 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.2 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C6H13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO2 251 2-NO2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl2, 5-NO2 254 2,3-Cl2, 6-NO2 255 2,6-Cl2, 4-NO2 256 2,6-Br2, 4-NO2 257 2,6-I2, 4-NO2 258 2-CH3, 5-i-C3H7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO2CH3 261 4-CO2CH3 262 2-CO2(C2H5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2O (C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 ----CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH3-4-(CH3-C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH3-4-(C2H5--C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroal- lyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Proparyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH3O2C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C6H5 476 4-O--C6H5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH3--CO--C6H4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O2N--C6H4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 16______________________________________ #STR218## No. B______________________________________1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH.sub.3 -Oxazolyl-4 234 2-C.sub.6 H.sub.5 -Oxazolyl-4 235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl______________________________________ TABLE 17______________________________________ #STR219## No. X.sub.m______________________________________1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroal lyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Proparyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroa llyl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroa llyl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 18______________________________________ #STR220## No. B______________________________________1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH.sub.3 -Oxazolyl-4 234 2-C.sub.6 H.sub.5 -Oxazolyl-4 235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl______________________________________ TABLE 19______________________________________ #STR221## No. X.sub.m______________________________________1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C4H9)2, 4-CH3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C6H11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2 (.sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH3 211 2-Cl, 5-CH3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH2--OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 3-CH3-4-(CH3--C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7 369 2-CH3-4-(C2H5--C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroal lyl 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Proparyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C6H5 385 4-C6H5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C6H4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH3O2C--C6H4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF3--C6H4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C6H5 476 4-O--C6H5 478 2-O-(2'-F--C6H4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C6H4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O2N--C6H4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5'______________________________________ TABLE 20______________________________________ #STR222## No. B______________________________________1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH.sub.3 -Oxazolyl-4 234 2-C.sub.6 H.sub.5 -Oxazolyl-4 235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 257 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadizolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3______________________________________ TABLE 21__________________________________________________________________________Selected physical data of some compoundsNo. Compound .sup.1 H-NMR (ppm) m.p.__________________________________________________________________________ 1 3.7(s, broad, 3H); 1.2(s, broad, 3H) - 2 3.75(s, 3H); 1.2(t, 3H) - 3 3.7(s, 3H); 1.2(t, 3H) - 4 3.95(s, 3H); 3.7(s, 3H); 1.2(t, 3H) - 5 3.6(s, 3H); 2.9(d, 3H) - 6 123 28## - 7 118 29## - 8 3.7(s, 3H); 2.55 (s, very broad, 2H)__________________________________________________________________________ TABLE 56______________________________________Selected physical data of some compounds - #STR231## - .sup.1 H-NMR (ppm) or IR No. X.sub.m mp (.degree. C.) (cm.sup.-1)______________________________________1 H 90 2 2-CH.sub.3 80 3 2,5-(CH.sub.3).sub.2 101 4 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 3.95(s, 3H); 3.65(s, 3H); 2.9(d, 3H) 5 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N-- 3.65(s, 3H); 2.9(d, O-Allyl 3H)______________________________________ TABLE 22______________________________________ #STR232## No. X Z A______________________________________1 H CH.sub.3 --CH.sub.2 O-- 2 H CH.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 3 H CH.sub.3 --CH.dbd.CH-- 4 H NH.sub.2 --CH.sub.2 O-- 5 H NH.sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 6 H NH.sub.2 --CH.dbd.CH-- 7 H N(CH.sub.3).sub.2 --CH.sub.2 O-- 8 H N(CH.sub.3).sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 9 H N(CH.sub.3).sub.2 --CH.dbd.CH-- 10 H CCl.sub.3 --CH.sub.2 O-- 11 H CCl.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 12 H CCl.sub.3 --CH.dbd.CH-- 13 H CF.sub.3 --CH.sub.2 O-- 14 H CF.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 15 H CF.sub.3 --CH.dbd.CH-- 16 CH.sub.3 CH.sub.3 --CH.sub.2 O-- 17 CH.sub.3 CH.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 18 CH.sub.3 CH.sub.3 --CH.dbd.CH-- 19 CH.sub.3 NH.sub.2 --CH.sub.2 O-- 20 CH.sub.3 NH.sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 21 CH.sub.3 NH.sub.2 --CH.dbd.CH-- 22 CH.sub.3 N(CH.sub.3).sub.2 --CH.sub.2 O-- 23 CH.sub.3 N(CH.sub.3).sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 24 CH.sub.3 N(CH.sub.3).sub.2 --CH.dbd.CH-- 25 CH.sub.3 CCl.sub.3 --CH.sub.2 O-- 26 CH.sub.3 CCl.sub.3 --CH.sub.2 O--N.dbd.C(C H.sub.3)-- 27 CH.sub.3 CCl.sub.3 --CH.dbd.CH-- 28 CH.sub.3 CF.sub.3 --CH.sub.2 O-- 29 CH.sub.3 CF.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 30 CH.sub.3 CF.sub.3 --CH.dbd.CH-- 31 Cl CH.sub.3 --CH.sub.2 O-- 32 Cl CH.sub.3 --CH.sub.2 O--N--C(CH.sub.3)-- 33 Cl CH.sub.3 --CH.dbd.CH-- 34 Cl NH.sub.2 --CH.sub.2 O-- 35 Cl NH.sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 36 Cl NH.sub.2 --CH.dbd.CH-- 37 Cl N(CH.sub.3).sub.2 --CH.sub.2 O-- 38 Cl N(CH.sub.3).sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 39 Cl N(CH.sub.3).sub.2 --CH.dbd.CH-- 40 Cl CCl.sub.3 --CH.sub.2 O-- 41 Cl CCl.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 42 Cl CCl.sub.3 --CH.dbd.CH-- 43 Cl CF.sub.3 --CH.sub.2 O-- 44 Cl CF.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 45 Cl CF.sub.3 --CH.dbd.CH--______________________________________ TABLE 23______________________________________ #STR233## No. B______________________________________1 2-Pyridyl 2 3-Trifluoromethyl-2-pyridyl 3 5-Trifluoromethyl-2-pyridyl 4 3,5-Bis-(trifluoromethyl)-2-pyridyl 5 3,5-Dichloro-2-pyridyl 6 3-Chloro-5-trifluoromethyl-2-pyridyl 7 3,5-Dichloro-2-pyridyl 8 2-Chloro-4-trifluormethylphenyl 9 2-Benzothiazolyl 10 5-Chloro-4-methyl-2-benzimidazolyl 11 2-Benzoxazolyl 12 1-Methyl-5-trifluoromethylimi- dazo[5,4-a]-pyridin-2-yl 13 5-Chloro-2-pyrimidinyl 14 4-Methyl-5-phenyl-2-thiazolin-2-yl 15 4-Methyl-5-phenyl-2-oxazolin-2-yl 16 7-Trifluoromethyl-4-quinolinyl______________________________________

Example 10

N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-O-methyl-hydroxylamine (Table 30, No. 1)

a) N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-hydroxylamine

At 0 to 5.degree. C., 7.0 g (70 mmol) of methyl chloroformate is added dropwise to 11.3 g (80 mmol) of N-2,6-dimethylphenyl-hydroxylamine (prepared analogously to Bamberger et al., Ann. Chem. 316 (1901), 278) and 12.5 g (90 mmol) of K.sub.2 CO.sub.3 in 30 ml of methylene chloride. The mixture is stirred for 30 mins at 0-5.degree. C., the insoluble solid is filtered off and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography with mixtures of cyclohexand and ethyl acetate. There is obtained 1.4 g (7.2 mmol 9%) of the title compound as a dark oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 8.85 (s, broad, 1H, OH); 7.1 (m, 3H, phenyl); 3.75 (s, 3H, OCH.sub.3); 2.3 (s, 6H, 2.times.CH.sub.3).

b) N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-O-methylhydroxylamine (Table 7, No. 1)

A mixture of 1.4 g (7.2 mmol) of N-(2,6-dimethylphenyl)-N-methoxycarbonyl-hydroxylamine (Example 1a), 1.3 g (9 mmol) of K.sub.2 CO.sub.3 and 10 g (8 mmol) of dimethyl sulfate in 10 ml of acetone is stirred overnight at room temperature. The reaction mixture is then diluted with CH.sub.2 Cl.sub.2 and stirred with dilute NH.sub.3 solution. The phases are then separated and the organic phase is extracted another twice with water. The organic phase is dried over MgSO.sub.4 and evaporated down, and the residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 1.2 g (6 mmol=83%) of the title compound as a colorless solid (mp=81.degree. C.).

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.1 (m, 3H, phenyl); 3.75 (s, broad, 6H, 2.times.OCH.sub.3); 2.3 (s, 3H, CH.sub.3).

The compounds listed in the following tables may be prepared similarly. Compound I, No. 1 from Table 24, No. 1 has for example the following formula: ##STR234##

TABLE 24______________________________________ No. T.sub.m______________________________________1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C2H5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-(C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-(C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-(C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C6H13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO2 251 2-NO2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl2, 5-NO2 254 2,4-Cl2, 6-NO2 255 2,6-Cl2, 4-NO2 256 2,6-Br2, 4-NO2 257 2,6-I2, 4-NO2 258 2-CH3, 5-i-C3H7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO2CH3 261 4-CO2CH3 262 2-CO2(C2H5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2O (C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--Ch.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 -- --CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.6 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH3-4-(CH3--C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH3-4-(C2H5--C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroal lyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Proparyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH3O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroa llyl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroa llyl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 25______________________________________ #STR235## No. B______________________________________1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH.sub.3 -Oxazolyl-4 234 2-C.sub.6 H.sub.5 -Oxazolyl-4 235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 3-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 257 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4,-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1-2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl______________________________________ TABLE 26______________________________________ #STR236## No. T.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C2H5)3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH3 226 3-Br, 4-CH3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.3, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 ----CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)--CH.sub.3 333 3-C(.dbd.NO-Allyl)--CH.sub.3 334 4-C(.dbd.NO-Allyl)--CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 338 2-C(.dbd.NO-Propargyl)--CH.sub.3 339 3-C(.dbd.NO-Propargyl)--CH.sub.3 340 4-C(.dbd.NO-Propargyl)--CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sup.2 --C.sup.6 H.sup.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloro allyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Proparyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C6H5 385 4-C6H5 386 2-(2'-F--C6H4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C6H4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF3--C6H4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C6H5 476 4-O--C6H5 478 2-O--(2'-F--C6H4) 479 2-O--(3'-F--C.sub.6 H.sub.4) 480 2-O--(4'-F--C.sub.6 H.sub.4) 481 3-O--(2'-F--C.sub.6 H.sub.4) 482 3-O--(3'-F--C.sub.6 H.sub.4) 483 3-O--(4'-F--C.sub.6 H.sub.4) 484 4-O--(2'-F--C.sub.6 H.sub.4) 485 4-O--(3'-F--C.sub.6 H.sub.4) 486 4-O--(4'-F--C.sub.6 H.sub.4) 487 2-O--(2'-Cl--C.sub.6 H.sub.4) 488 2-O--(3'-Cl--C.sub.6 H.sub.4) 489 2-O--(4'-Cl--C.sub.6 H.sub.4) 490 3-O--(2'-Cl--C.sub.6 H.sub.4) 491 3-O--(3'-Cl--C.sub.6 H.sub.4) 492 3-O--(4'-Cl--C.sub.6 H.sub.4) 493 3-O--(4'-Cl--C.sub.6 H.sub.4) 494 4-O--(2'-Cl--C.sub.6 H.sub.4) 495 4-O--(3'-Cl--C.sub.6 H.sub.4) 496 4-O--(4'-Cl--C.sub.6 H.sub.4) 497 2-O--(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O--(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O--(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O--(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O--(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O--(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O--(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O--(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O--(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O--(4'-CH.sub.3 --CO--C6H4) 509 3-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O--(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 516 2-O--(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 517 2-O--(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 518 3-O--(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 519 3-O--(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 520 3-O--(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 521 4-O--(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 522 4-O--(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 523 4-O--(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 524 2-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O--(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O--(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O--(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O--(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O--(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O--(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O--(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O--(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O--(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O--(2'-NC--C.sub.6 H.sub.4) 552 2-O--(3'-NC--C.sub.6 H.sub.4) 553 2-O--(4'-NC--C.sub.6 H.sub.4) 554 3-O--(2'-NC--C.sub.6 H.sub.4) 555 3-O--(3'-NC--C.sub.6 H.sub.4) 556 3-O--(4'-NC--C.sub.6 H.sub.4) 557 4-O--(2'-NC--C.sub.6 H.sub.4) 558 4-O--(3'-NC--C.sub.6 H.sub.4) 559 4-O--(4'-NC--C.sub.6 H.sub.4) 560 2-O--(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O--(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O--(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O--(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O--(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O--(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O--(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O--(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O--(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chlor oallyl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chlor oallyl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 27______________________________________ #STR237## I: R.sup.1 = CH.sub.3, X = CH.sub.3 II: R.sup.1 = CH.sub.2 --CH.sub.3, X = CH.sub.3 III: R.sup.1 = CH.sub.3, X = Cl IV: R.sup.1 = CH.sub.2 --CH.sub.3, X = Cl -No. B______________________________________ 1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH.sub.3 -Oxazolyl-4 234 3-C.sub.6 H.sub.5 -Oxazolyl-4 235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl______________________________________ TABLE 28______________________________________ #STR238## I: R.sup.1 = CH.sub.3, X = CH.sub.3 II: R.sup.1 = CH.sub.2 --CH.sub.3, X = CH.sub.3 III: R.sup.1 = CH.sub.3, X = Cl IV: R.sup.1 = CH.sub.2 --CH.sub.3, X = Cl -No. T.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,5-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroa llyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-Cl--C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5'______________________________________ TABLE 29______________________________________ #STR239## I: R.sup.1 = CH.sub.3, X = CH.sub.3 II: R.sup.1 = CH.sub.2 --CH.sub.3, X = CH.sub.3 III: R.sup.1 = CH.sub.3, X = Cl IV: R.sup.1 = CH.sub.2 --CH.sub.3, X = Cl -No. B______________________________________ 1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH.sub.3 -Oxazolyl-4 234 3-C.sub.6 H.sub.5 -Oxazolyl-4 235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3______________________________________ TABLE 30______________________________________Selected physical data of some compounds IR (cm.sup.-1) or .sup.1 H-NMR No. Compound (ppm) m.p______________________________________ 1 81 240## - 2 60 241## - 3 3.85(s, broad, 3H); 3.7(s, broad, 3H) - 4 3.85(s, broad, 3H); 3.75(s, broad, 3H) - 5 3.75(2s, broad, each 3H) - 6 91 245## - 7 3.8(s, 3H); 3.75(s, broad, 3H) - 8 3.85(s, 3H); 3.8(s, broad,______________________________________ 3H) TABLE 31______________________________________ #STR248## I: R.sup.1 = CH.sub.3, X = CH.sub.3 II: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3 III: R.sup.1 = CH.sub.3, X = Cl IV: R.sup.1 = C.sub.2 H.sub.5, X = Cl -No. B______________________________________ 1 2-Pyridyl 2 3-Trifluoromethyl-2-pyridyl 3 5-Trifluoromethyl-2-pyridyl 4 3,5-Bis-(trifluoromethyl)-2-pyridyl 5 3,5-Dichloro-2-pyridyl 6 3-Chloro-5-trifluoromethyl-2-pyridyl 7 3,5-Dichloro-2-pyridyl 8 2-Chloro-4-trifluoromethylphenyl 9 2-Benzothiazolyl 10 5-Chloro-1-methyl-2-benzimidazolyl 11 2-Benzoxazolyl 12 1-Methyl-5-trifluoromethylimidazo- [5,4-a]-pyridin-2-yl 13 5-Chloro-2-pyrimidinyl 14 4-Methyl-5-phenyl-2-thiazolin-2-yl 15 4-Methyl-5-phenyl-2-oxazolin-2-yl 16 7-Trifluoromethyl-4-quinolinyl______________________________________ TABLE 57______________________________________Selected physical data of some compounds #STR249## mp .sup.1 H-NMR (ppm) No. X T.sub.m (.degree. C.) or IR (cm.sup.-1)______________________________________1 Cl 2-CH.sub.3 3.8(s, broad, 6H) 2 Cl 2,5-(CH.sub.3).sub.2 3.8(s, broad, 6H) 3 Cl 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 4.0(s, 3H); 3.8 (s, broad, 6H) 4 Cl 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--O-- 3.8(s, broad, 6H) Allyl 5 CH.sub.3 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 4.0(s, 3H); 3.75 (s, broad, 6H) 6 CH.sub.3 2-CH.sub.3 3.75(s, broad, 6H) 7 CH.sub.3 2,5-(CH.sub.3).sub.2 3.75(s, broad, 6H) 8 CH.sub.3 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--O-- 3.75(s, broad, Allyl 6H)______________________________________

Example 11

2-(2'-Methylphenoxymethyl)-trichloroacetanilide (Table 38, No. 1)

a) 2-(2'-Methylphenoxymethyl)-nitrobenzene

75 g (0.347 mol) of 2-nitrobenzyl bromide, 37 g (0.342 mol) of o-cresol and 56 g (0.405 mol) of potassium carbonate in 500 ml of dimethylformamide is stirred for 5 hours at room temperature (20.degree. C.). The reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The ether phase is dried and evaporated down. The crystalline residue is stirred with methanol and suction filtered. There is obtained 73 g (0.300 mol=88%) of the title compound as a colorless solid.

Mp=83.degree. C.

.sup.1 H-NMR, (CDCl.sub.3 ; .delta. (ppm)): 8.15 (d, 1H, I=8 Hz, aromatic); 7.95 (d, 1H, I=8 Hz, 1H, I=8 Hz, aromatic); 7.15 (m, 2H, aromatic); 6.9 (m, 2H, aromatic); 5.45 (s, 2H, O--CH.sub.2); 2.35 (s, 3H, CH.sub.3).

b) 2-(2'-Methylphenoxymethyl)-aniline

75 g (0.308 mol) of 2-(2'-methylphenoxymethyl)-nitrobenzene (Example 11a) and 10 g of 5% Pt/C (platinum adsorbed on activated carbon) in 50 ml of methanol are stirred vigorously under a hydrogen blanket for 2 hours. A further 2 g of 5% Pt/C is added and the mixture is stirred overnight. The catalyst is filtered off and replaced by 10 g of fresh catalyst. The mixture is stirred overnight and suction filtered, and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 61 g (0.286 mol=93%) of the title compound as a colorless solid.

Mp=56.degree. C.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.2 (m, 4H, aromatic); 6.95 (d, 1H, I=8 Hz, aromatic); 6,9 (t, 1H, I=6 Hz, aromatic); 6.7 (m, 2H, aromatic); 5.0 (s, 2H, O--CH.sub.2); 4.05 (s, broad, 2H, NH.sub.2); 2.2 (s, 3H, CH.sub.3).

c) 2-(2'-Methylphenoxymethyl)-trichloroacetanilide (Table 38, No. 1)

At 10-15.degree. C., a solution of 6 g of 2-(2'-methylphenoxymethyl)-aniline (Example 1b) in 20 ml of CH.sub.2 Cl.sub.2 is added to a mixture of 6.6 g (36 mmol) of trichloroacetyl chloride and 3 g (38 mmol) of pyridine in 50 ml of CH.sub.2 Cl.sub.2. The mixture is stirred for 1 hour at room temperature, and then extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is suction filtered over silica gel and the filtrate which is obtained is evaporated down. The residue crystallizes and is stirred with hexane. There is obtained 7.9 g (22 mmol=78%) of the title compound as a crystalline solid (mp=128.degree. C.).

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 9.6 (s, broad, 1H, NH); 8.1 (d, 1H, I=8 Hz, phenyl); 7.5 (t, broad, 1H, phenyl); 7.4 (d, broad, 1H, phenyl); 7.2 (m, 3H, phenyl); 6.95 (m, 2H, phenyl); 5.1 (s, 2H, OCH.sub.2); 2.2 (s, 3H, CH.sub.3).

Example 12

N-Methyl-N'-(2-(2'-methylphenoxymethyl)-phenyl)-urea (Table 7, No. 2)

In a laboratory autoclave, about 10 ml of methylamine is added to 2 g (5.5 mmol) of the trichloroacetanilide from Example 1c. The autoclave is then closed and the reaction mixture is heated for about 6 hours at 80.degree. C. The reaction mixture is cooled and the autoclave opened. The methylamine is allowed to evaporate off and the solid residue is stirred with methyl tert-butyl ether. The insoluble solid is filtered off and dried under reduced pressure. There is obtained 1.4 g (5.2 mmol=94%) of the title compound as a crystalline solid (mp=144.degree. C.).

.sup.1 H-NMR (DMSO-d.sub.6 ; .delta. (ppm)): 8.05 (s, 1H, NH); 7.8 (d, 1H, I=8 Hz, phenyl); 7.4 (d, 1H, I=8 Hz, phenyl); 6.8-7.3 (m, 6H, phenyl); 6.7 (s, 1H, NH); 5.1 (S, 2H, OCH.sub.2); 2.65 (d, 3H, I=5 Hz, N--CH.sub.3); 2.2 (s, 3H, CH.sub.3).

Example 13

2-(2'-Methylphenoxymethyl)-propionyl anilide (Table 38, No. 3)

A mixture of 3 g (14.1 mmol) of the aniline from Example 11b, 1.35 g (17 mmol) of pyridine and 1.4 g (15.5 mmol) of propionyl chloride in 30 ml of methylene chloride is stirred for 1 hour at room temperature. The reaction mixture is then extracted with diluted hydrochloric acid and water, dried over MgSO.sub.4 and evaporated down. There is obtained 3.8 g (quantitative yield) of the title compound.

.sup.1 H-NMR (COCl.sub.3 ; .delta. (ppm)): 8.25 (s, broad, 1H, NH); 8.15 (d, 1H, I=8 Hz, phenyl); 6.9-7.5 (m, 7H, phenyl); 5.1 (s, 2H, OCH.sub.2); 2.35 (q, 2H, I=8 Hz, CH.sub.2); 2.25 (s, 3H, CH.sub.3); 1.2 (t, 3H, I=8 Hz, CH.sub.3).

Example 14

N-Propionyl-2-(2'-methylphenoxymethyl)-propionyl anilide (Table 38, No. 4)

0.41 g (17.1 mmol) of sodium hydride is added in portions to 3.8 g (14 mmol) of the propionyl anilide from Example 13 in 40 ml of dimethylformamide. Upon completion of gas evolution 1.4 g (15.9 mmol) of propionyl chloride is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 2.6 g (8 mmol=57%) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3): .delta. (ppm): 7.6 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.15 (m, 3H, phenyl); 6.85 (m, 2H, phenyl); 4.85 (m, 2H, OCH.sub.2); 2.6 (m, 4H, 2.times.CH.sub.2); 2.2 (s, 3H, CH.sub.3); 1.1 (t, 6H, I=8 Hz, 2.times.CH.sub.3).

Example 15

N-Methyl-2-(2'-methylphenoxymethyl)-propionyl anilide (Table 38, No. 5)

0.45 g (19 mmol) of sodium hydride is added in portions to 4.0 g (14.8 mmol) of the propionyl anilide from Example 13 in 50 ml of dimethylformamide. Upon completion of gas evolution 3.0 g (21 mmol) of methyl iodide is added and the mixture is stirred for 2 hours at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. The residue crystallizes and is stirred with hexane. There is obtained 3.7 g (11.7 mmol=90%) of the title compound as a colorless solid (mp=80.degree. C.).

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.2 (m, 3H, phenyl); 6.9 (m, 2H, phenyl); 5.0 (s, 2H, OCH.sub.2); 3.2 (s, 3H, N--CH.sub.3); 2.2 (s, 3H, CH.sub.3); 2.0 (m, 2H, CH.sub.2); 1.0 (t, 3H, I=8 Hz, CH.sub.3).

Example 19

N-Methyl-2-(2'-methylphenoxymethyl)-acetanilide

a) N-Methyl-2-(2'-methylphenoxymethyl)-aniline

A mixture of 5 g (23 mmol) of 2-(2'-methylphenoxymethyl)-aniline (Example 1b), 5 g (36 mmol) of K.sub.2 CO.sub.3 and 3.4 g (24 mmol) of methyl iodide in 50 ml of dimethylformamide is stirred overnight at room temperature. The reaction mixture is diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is purified chromatographically using mixtures of hexane and methylene chloride. There is obtained 3.0 g (70% purity, about 40% yield) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 6.6-7.4 (m, 8H, phenyl); 5.0 (s, 2H, OCH.sub.2); 4.6 (s, broad, 1H, NH); 2.9 (d, 3H, N--CH.sub.3); 2.2 (s, 3H, CH.sub.3).

b) N-Methyl-2-(2'-methylphenoxymethyl)-acetanilide (Table 7, No. 9)

3 g (approx. 9.3 mmol) of N-methyl-2-(2'-methylphenoxymethyl)-aniline (from Example 5a) is added to a mixture of 1.6 g (16 mmol) of acetoanhydride and 1.3 g (16 mmol) of pyridine in 20 ml of methylene chloride. The mixture is stirred for 1 hour at room temperature and is then extracted with dilute hydrochloric acid and water. The organic phase is evaporated down and the residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 2 g (80%) of the title compound as a colorless solid (mp=76.degree. C.).

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.2 (m, 3H, phenyl); 6.9 (m, 2H, phenyl); 5.0 (s, 2H, OCH.sub.2); 3.25 (s, 3H, CH.sub.3); 2.25 (s, 3H, CH.sub.3); 1.8 (s, 3H, CH.sub.3).

The compounds listed in the tables below may be prepared correspondingly.

Compound I from Table 32, No. 1 has for example the following structural formula: ##STR250##

The compounds described in the following tables may be prepared analogously.

TABLE 32______________________________________ #STR251## I: R.sup.1 = H, Z = C.sub.2 H.sub.5 II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 VI: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = C.sub.2 H.sub.5 VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 VIII: R.sup.1 = H, Z = NH(CH.sub.3) IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3) X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3) XI: R.sup.1 = Allyl, Z = NH(CH.sub.3) XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3) XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = NH(CH.sub.3) XIV: R.sup.1 = CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3) -No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,5-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 305 2-Me-4-CO--CH(CH.sub.3).sub.2 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CO--CH.sub.3 308 2,5-Me.sub.2 -4-CO--CH.sub.2 --CH.sub.3 309 2,5-Me.sub.2 -4-CH.sub.2 --CH.sub.2 --CO--CH.sub.3 310 2,5-Me.sub.2 -4-CO--CH(CH.sub.3).sub.2 311 2-Cl-4-CHO 312 2-Cl-4-CO--CH.sub.3 313 2-Cl-4-CO--CH.sub.2 --CH.sub.3 314 2-Cl-4-CO--CH(CH.sub.3).sub.2 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CO--CH.sub.3 317 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.3 318 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 319 2,5-Cl.sub.2 -4-CO--CH(CH.sub.3).sub.2 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 33______________________________________ #STR252## I: R.sup.1 = H, Z = C.sub.2 H.sub.5 II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 VI: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = C.sub.2 H.sub.5 VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 VIII: R.sup.1 = H, Z = NH(CH.sub.3) IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3) X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3) XI: R.sup.1 = Allyl, Z = NH(CH.sub.3) XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3) XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = NH(CH.sub.3) XIV: R.sup.1 = CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3) -No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,5-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CO--CH.sub.2 --CH.sub.3 304 2-Me-4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 305 2-Me-4-CO--CH(CH.sub.3).sub.2 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CO--CH.sub.3 308 2,5-Me.sub.2 -4-CO--CH.sub.2 --CH.sub.3 309 2,5-Me.sub.2 -4-CH.sub.2 --CH.sub.2 --CO--CH.sub.3 310 2,5-Me.sub.2 -4-CO--CH(CH.sub.3).sub.2 311 2-Cl-4-CHO 312 2-Cl-4-CO--CH.sub.3 313 2-Cl-4-CO--CH.sub.2 --CH.sub.3 314 2-Cl-4-CO--CH(CH.sub.3).sub.2 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CO--CH.sub.3 317 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.3 318 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 319 2,5-Cl.sub.2 -4-CO--CH(CH.sub.3).sub.2 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 34______________________________________ #STR253## I: R.sup.1 = H, Z = C.sub.2 H.sub.5 II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 VI: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = C.sub.2 H.sub.5 VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 VIII: R.sup.1 = H, Z = NH(CH.sub.3) IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3) X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3) XI: R.sup.1 = Allyl, Z = NH(CH.sub.3) XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3) XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = NH(CH.sub.3) XIV: R.sup.1 = CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3) -No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,5-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CO--CH.sub.3 303 2-Me-4-CO--CH.sub.2 --CH.sub.3 304 2-Me-4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 305 2-Me-4-CO--CH(CH.sub.3).sub.2 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CO--CH.sub.3 308 2,5-Me.sub.2 -4-CO--CH.sub.2 --CH.sub.3 309 2,5-Me.sub.2 -4-CH.sub.2 --CH.sub.2 --CO--CH.sub.3 310 2,5-Me.sub.2 -4-CO--CH(CH.sub.3).sub.2 311 2-Cl-4-CHO 312 2-Cl-4-CO--CH.sub.3 313 2-Cl-4-CO--CH.sub.2 --CH.sub.3 314 2-Cl-4-CO--CH(CH.sub.3).sub.2 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CO--CH.sub.3 317 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.3 318 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 319 2,5-Cl.sub.2 -4-CO--CH(CH.sub.3).sub.2 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 35______________________________________ #STR254## I: R.sup.1 = H, Z = C.sub.2 H.sub.5 II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 VI: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = C.sub.2 H.sub.5 VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 VIII: R.sup.1 = H, Z = NH(CH.sub.3) IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3) X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3) XI: R.sup.1 = Allyl, Z = NH(CH.sub.3) XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3) XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = NH(CH.sub.3) XIV: R.sup.1 = CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3) -No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CO--CH.sub.2 --CH.sub.3 304 2-Me-4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 305 2-Me-4-CO--CH(CH.sub.3).sub.2 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CO--CH.sub.3 308 2,5-Me.sub.2 -4-CO--CH.sub.2 --CH.sub.3 309 2,5-Me.sub.2 -4-CH.sub.2 --CH.sub.2 --CO--CH.sub.3 310 2,5-Me.sub.2 -4-CO--CH(CH.sub.3).sub.2 311 2-Cl-4-CHO 312 2-Cl-4-CO--CH.sub.3 313 2-Cl-4-CO--CH.sub.2 --CH.sub.3 314 2-Cl-4-CO--CH(CH.sub.3).sub.2 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CO--CH.sub.3 317 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.3 318 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 319 2,5-Cl.sub.2 -4-CO--CH(CH.sub.3).sub.2 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroall yl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 36______________________________________ #STR255## I: R.sup.1 = H, Z = C.sub.2 H.sub.5 II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 VI: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = C.sub.2 H.sub.5 VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 VIII: R.sup.1 = H, Z = NH(CH.sub.3) IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3) X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3) XI: R.sup.1 = Allyl, Z = NH(CH.sub.3) XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3) XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = NH(CH.sub.3) XIV: R.sup.1 = CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3) -No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CO--CH.sub.2 --CH.sub.3 304 2-Me-4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 305 2-Me-4-CO--CH(CH.sub.3).sub.2 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CO--CH.sub.3 308 2,5-Me.sub.2 -4-CO--CH.sub.2 --CH.sub.3 309 2,5-Me.sub.2 -4-CH.sub.2 --CH.sub.2 --CO--CH.sub.3 310 2,5-Me.sub.2 -4-CO--CH(CH.sub.3).sub.2 311 2-Cl-4-CHO 312 2-Cl-4-CO--CH.sub.3 313 2-Cl-4-CO--CH.sub.2 --CH.sub.3 314 2-Cl-4-CO--CH(CH.sub.3).sub.2 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CO--CH.sub.3 317 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.3 318 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 319 2,5-Cl.sub.2 -4-CO--CH(CH.sub.3).sub.2 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroa llyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5'______________________________________ TABLE 37______________________________________ #STR256## I: R.sup.1 = H, Z = C.sub.2 H.sub.5 II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 VI: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = C.sub.2 H.sub.5 VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 VIII: R.sup.1 = H, Z = NH(CH.sub.3) IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3) X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3) XI: R.sup.1 = Allyl, Z = NH(CH.sub.3) XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3) XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = NH(CH.sub.3) XIV: R.sup.1 = CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3) -No. B______________________________________ 1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH.sub.3 -Oxazolyl-4 234 3-C.sub.6 H.sub.5 -Oxazolyl-4 235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2______________________________________ TABLE 38______________________________________Selected physical data of some compounds IR (cm.sup.-1) or .sup.1 H-NMR mp No. Compound (ppm) (.degree. C.)______________________________________ 1 128 57## - 2 144 58## - 3 #STR259## - 4 #STR260## - 5 80 61## - 6 75 62## - 7 188 63## - 8 115 64## - 9 76 65## - 10 96 66## - 11 3.3 (s, 3H); 2.25(s, 3H)______________________________________ TABLE 58______________________________________Selected physical data of some compounds #STR268## IR (cm.sup.-1) or .sup.1 H- NMR mp No. X.sub.m R.sup.1 (ppm) (.degree. C.)______________________________________ 1 2-CH.sub.3 H 120 2 2-CH.sub.3 CH.sub.3 oil 3 2-CH.sub.3 C.sub.2 H.sub.5 oil 4 2-CH.sub.3 Allyl oil 5 2-CH.sub.3 Propargyl oil 6 2-CH.sub.3 CH.sub.2 --OCH.sub.3 oil 7 2,5-(CH.sub.3).sub.2 H 170 8 2,5-(CH.sub.3).sub.2 CH.sub.3 oil 9 2,5-(CH.sub.3).sub.2 C.sub.2 H.sub.5 oil 10 2,5-(CH.sub.3).sub.2 Allyl oil 11 2,5-(CH.sub.3).sub.2 Propargyl oil 12 2,5-(CH.sub.3).sub.2 CH.sub.2 --OCH.sub.3 oil 13 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 H 125 14 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 CH.sub.3 oil 15 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 C.sub.2 H.sub.5 oil 16 2-CH.sub.3 -4-C(CH.sub.3).dbd. N--OCH.sub.3 Allyl 87 17 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 Propargyl oil 18 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 CH.sub.2 --OCH.sub.3 oil 19 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--O-Allyl H 85 20 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--O-Allyl CH.sub.3 oil 21 2,5-(CH.sub.3).sub.2 -4-C(CH.s ub.3).dbd.N--O-Allyl C.sub.2 H.sub.5 oil 22 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--O-Allyl Allyl 87 23 2,5-(CH.sub.3).sub.2 -4-C(CH.s ub.3).dbd.N--O-Allyl Propargyl oil 24 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--O-Allyl CH.sub.2 --OCH.sub .3 oil______________________________________ TABLE 59______________________________________Selected physical data of some compounds #STR269## IR (cm.sup.-1) or .sup.1 H-NMR No. X.sub.m R.sup.1 (ppm) mp (.degree. C.)______________________________________1 4-CH.sub.3 H 118 2 4-CH.sub.3 CH.sub.3 oil 3 4-CH.sub.3 C.sub.2 H.sub.5 oil 4 4-CH.sub.3 Allyl oil 5 4-CH.sub.3 Propargyl oil 6 4-CH.sub.3 CH.sub.2 --OCH.sub.3 oil 7 3,5-Cl.sub.2 H 160 8 3,5-Cl.sub.2 CH.sub.3 oil 9 3,5-Cl.sub.2 C.sub.2 H.sub.5 oil 10 3,5-Cl.sub.2 Allyl 85 11 3,5-Cl.sub.2 Propargyl oil 12 3,5-Cl.sub.2 CH.sub.2 --OCH.sub.3 oil______________________________________ TABLE 39______________________________________ #STR270## No. X R.sup.1 X A______________________________________ 1 H H CH.sub.3 --CH.sub.2 O-- 2 H H CH.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 3 H H CH.sub.3 --CH.dbd.CH-- 4 H H NH.sub.2 --CH.sub.2 O-- 5 H H NH.sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 6 H H NH.sub.2 --CH.dbd.CH-- 7 H H N(CH.sub.3).sub.2 --CH.sub.2 O-- 8 H H N(CH.sub.3).sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 9 H H N(CH.sub.3).sub.2 --CH.dbd.CH-- 10 H H CCl.sub.3 --CH.sub.2 O-- 11 H H CCl.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 12 H H CCl.sub.3 --CH.dbd.CH-- 13 H H CF.sub.3 --CH.sub.2 O-- 14 H H CF.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 15 H H CF.sub.3 --CH.dbd.CH-- 16 H Propargyl CH.sub.3 --CH.sub.2 O-- 17 H Propargyl CH.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 18 H Propargyl CH.sub.3 --CH.dbd.CH-- 19 H Propargyl NH.sub.2 --CH.sub.2 O-- 20 H Propargyl NH.sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 21 H Propargyl NH.sub.2 --CH.dbd.CH-- 22 H Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O-- 23 H Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O--N--.dbd.C(CH.sub.3)-- 24 H Propargyl N(CH.sub.3).sub.2 --CH.dbd.C H-- 25 H Propargyl CCl.sub.3 --CH.sub.2 O-- 26 H Propargyl CCl.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 27 H Propargyl CCl.sub.3 --CH.dbd.CH-- 28 H Propargyl CF.sub.3 --CH.sub.2 O-- 29 H Propargyl CF.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 30 H Propargyl CF.sub.3 --CH.dbd.CH-- 31 CH.sub.3 H CH.sub.3 --CH.sub.2 O-- 32 CH.sub.3 H CH.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 33 CH.sub.3 H CH.sub.3 --CH.dbd.CH-- 34 CH.sub.3 H NH.sub.2 --CH.sub.2 O-- 35 CH.sub.3 H NH.sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 36 CH.sub.3 H NH.sub.2 --CH.dbd.CH-- 37 CH.sub.3 H N(CH.sub.3).sub.2 --CH.sub.2 O-- 38 CH.sub.3 H N(CH.sub.3).sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 39 CH.sub.3 H N(CH.sub.3).sub.2 --CH.dbd.CH -- 40 CH.sub.3 H CCl.sub.3 --CH.sub.2 O-- 41 CH.sub.3 H CCl.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 42 CH.sub.3 H CCl.sub.3 --CH.dbd.CH-- 43 CH.sub.3 H CF.sub.3 --CH.sub.2 O-- 44 CH.sub.3 H CF.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 45 CH.sub.3 H CF.sub.3 --CH.dbd.CH-- 46 CH.sub.3 Propargyl CH.sub.3 --CH.sub.2 O-- 47 CH.sub.3 Propargyl CH.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 48 CH.sub.3 Propargyl CH.sub.3 --CH.dbd.CH- - 49 CH.sub.3 Propargyl NH.sub.2 --CH.sub.2 O-- 50 CH.sub.3 Propargyl NH.sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 51 CH.sub.3 Propargyl NH.sub.2 --CH.dbd.CH- - 52 CH.sub.3 Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O-- 53 CH.sub.3 Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)- - 54 CH.sub.3 Propargyl N(CH.sub.3).sub.2 --CH.dbd.CH-- 55 CH.sub.3 Propargyl CCl.sub.3 --CH.sub.2 O-- 56 CH.sub.3 Propargyl CCl.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 57 CH.sub.3 Propargyl CCl.sub.3 --CH.dbd.CH -- 58 CH.sub.3 Propargyl CF.sub.3 --CH.sub.2 O-- 59 CH.sub.3 Propargyl CF.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 60 CH.sub.3 Propargyl CF.sub.3 --CH.dbd.CH- - 61 Cl H CH.sub.3 --CH.sub.2 O-- 62 Cl H CH.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 63 Cl H CH.sub.3 --CH.dbd.CH-- 64 Cl H NH.sub.2 --CH.sub.2 O-- 65 Cl H NH.sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 66 Cl H NH.sub.2 --CH.dbd.CH-- 67 Cl H N(CH.sub.3).sub.2 --CH.sub.2 O-- 68 Cl H N(CH.sub.3).sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 69 Cl H N(CH.sub.3).sub.2 --CH.dbd.CH-- 70 Cl H CCl.sub.3 --CH.sub.2 O-- 71 Cl H CCl.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 72 Cl H CCl.sub.3 --CH.dbd.CH-- 73 Cl H CF.sub.3 --CH.sub.2 O-- 74 Cl H CF.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 75 Cl H CF.sub.3 --CH.dbd.CH-- 76 Cl Propargyl CH.sub.3 --CH.sub.2 O-- 77 Cl Propargyl CH.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 78 Cl Propargyl CH.sub.3 --CH.dbd.CH-- 79 Cl Propargyl NH.sub.2 --CH.sub.2 O-- 80 Cl Propargyl NH.sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 81 Cl Propargyl NH.sub.2 --CH.dbd.CH-- 82 Cl Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O-- 83 Cl Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 84 Cl Propargyl N(CH.sub.3).sub.2 --CH.dbd. CH-- 85 Cl Propargyl CCl.sub.3 --CH.sub.2 O-- 86 Cl Propargyl CCl.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 87 Cl Propargyl CCl.sub.3 --CH.dbd.CH-- 88 Cl Propargyl CF.sub.3 --CH.sub.2 O-- 89 Cl Propargyl CF.sub.3 --CH.sub.2 O--N.dbd.C(CH.sub.3)-- 90 Cl Propargyl CF.sub.3 --CH.dbd.CH--______________________________________ TABLE 40______________________________________ #STR271## I: R.sup.1 = H, Z = C.sub.2 H.sub.5 II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 VI: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = C.sub.2 H.sub.5 VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 VIII: R.sup.1 = H, Z = NH(CH.sub.3) IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3) X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3) XI: R.sup.1 = Allyl, Z = NH(CH.sub.3) XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3) XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = NH(CH.sub.3) XIV: R.sup.1 = CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3) -No. B______________________________________ 1 2-Pyridyl 2 3-Trifluoromethyl-2-pyridyl 3 5-Trifluoromethyl-2-pyridyl 4 3,5-Bis-(trifluoromethyl)-2-pyridyl 5 3,5-Dichloro-2-pyridyl 6 3-Chloroo-5-trifluoromethyl-2-pyridyl 7 3,5-Dichloro-2-pyridyl 8 2-Chloroo-4-trifluoromethylphenyl 9 2-Benzothiazolyl 10 5-Chloroo-1-methyl-2-benzimidazolyl 11 2-Benzoxazolyl 12 1-Methyl-5-trifluoromethylimidazo- [5,4-a]-pyridin-2-yl 13 5-Chloroo-2-pyrimidinyl 14 4-Methyl-5-phenyl-2-thiazolin-2-yl 15 4-Methyl-5-phenyl-2-oxazolin-2-yl 16 7-Trifluoromethyl-4-quinolinyl______________________________________

Example 16

Methyl N-[2-(3",4"-dichlorophenyl-1'-methyliminooxymethyl-4')-6-methylphenyl]-carbamate (Table 47, No. 2)

a) 2-(Methanesulfonyloxymethyl)-6-methyl-nitrobenzene

At 10-15.degree. C., 27 g (0.23 mol) of methanesulfonyl chloride dissolved in 20 ml of CH.sub.2 Cl.sub.2 is dripped into a mixture of 34 g (0.2 mol) of 3-methyl-2-nitrobenzyl alcohol and 27 g (0.27 mol) of triethylamine in 100 ml of CH.sub.2 Cl.sub.2. The reaction mixture is stirred for 1 hour at room temperature and is then extracted with water. The organic phase is dried over MgSO.sub.4 and evaporated down. There is obtained as residue 48 g of the title compound as a yellow oil, containing about 10% of the corresponding benzyl chloride as impurity. The crude product is used for the next reaction without any further purification.

.sup.1 H-NMR(COCl.sub.3 ; .delta. in ppm): 7.3-7.6 (m, 3H, phenyl); 5.3 (S, 2H, OCH.sub.2); 3.0 (S, 3H, CH.sub.3 --SO.sub.3); 2.4 (S, 3H, CH.sub.3).

b) 2-(3",4"-Dichlorophenyl-1'-methyl-iminooxymethyl-4')-6-methyl-nitrobenzene

At room temperature, 1.8 g (75 mmol) of sodium hydride is added in portions to a solution of 13 g (64 mmol) of 3,4-dichloroacetophenonoxime in 100 ml of dimethylformamide. Upon conclusion of gas evolution, a solution of 16 g (65 mmol) of the mesylate from Example 1a in 30 ml of dimethylformamide is dripped in at 25-30.degree. C., and the mixture is then stirred for 1 hour at room temperature. The reaction mixture is diluted with water and the aqueous phase is then extracted three times with methyl tert-butyl ether. The combined organic phases are washed with water, dried over MGSO.sub.4 and evaporated down. The residue crystallizes and is stirred with methanol. The mother liquor is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained a total of 20.4 g (58 mmol=90%) of the title compound as pale yellow crystals.

.sup.1 H-NMR(CDCl.sub.3 ; .delta. in ppm): 7.7 (S, broad, 1H, phenyl); 7.2-7.6 (m, 5H, phenyl); 5.3 (S, 2H, OCH.sub.2); 2.4 (S, 3H, CH.sub.3); 2.2 (S, 3H, CH.sub.3).

c) 2-(3",4"-Dichlorophenyl-1'-methyl-iminooxymethyl-4')-6-methyl-aniline

At 20-30.degree. C., 53 g of 21.8% strength Na.sub.2 [Fe(CO).sub.4 ] solution (1 kg of the solution contains 633 g of water, 218 g of Na.sub.2 [Fe(CO).sub.4 ], 108 g of Na.sub.2 CO.sub.3 and 41 g of NaOH) is added dropwise to 19 g (52.8 mmol) of the nitrobenzene from Example 16b in 150 ml of methanol. The brown suspension is stirred for 2 hours at room temperature, and the reaction mixture is then diluted with methylene chloride and the mixture is suction filtered using kieselguhr. The residue is again washed with CH.sub.2 Cl.sub.2 and the combined extracts are extracted with water, dried over MgSO.sub.4 and evaporated down. The brown residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 14.3 g (44.3 mmol=82%) of the title compound as a beige solid.

.sup.1 H-NMR(CDCl.sub.3 ; .delta. in ppm): 7.7 (S, 1H, phenyl); 7.5 (m, 2H, phenyl); 7.1 (t, broad, 2H, phenyl); 6.7 (t, 1H, I=8 Hz, phenyl); 5.2 (S, 2H, OCH.sub.2); 4.15 (S, 2H, NH.sub.2 ; 2.2 (S, 3H, CH.sub.3).

d) Methyl N-[2-(3",4"-dichlorophenyl-1'-methyl-iminooxymethyl-4'-6-methylphenyl]-carbamate (Table 47, No. 2)

At 20-30.degree. C., 4.8 g (50 mmol) of methyl chloroformate and subsequently 4.8 g (60 mmol) of pyridine are dripped into a solution of 14.3 g (44 mmol) of the aniline from Example 1c in 150 ml of CH.sub.2 Cl.sub.2. The mixture is stirred overnight at room temperature and is then extracted with dilute hydrochloric acid and water. The reaction mixture is suction filtered using silica gel, dried over MgSO.sub.4 and evaporated down. The residue crystallizes and is stirred with cyclohexane. There is obtained 13.8 g (36 mmol=82%) of the title compound as a colorless solid (mp=109.degree. C.).

.sup.1 H-NMR(CDCl.sub.3 ; .delta. in ppm): 7.8 (S, 1H, phenyl); 7.6 (S, broad, 1H, NH); 7.4 (S, 2H, phenyl); 7.2 (m, 3H, phenyl); 5.2 (S, 2H, OCH.sub.2); 3.8 (S, 3H, OCH.sub.3); 2.3 (S, 3H, CH.sub.3); 2.2 (S, 3H, CH.sub.3).

Example 17

Methyl N-[2-(3",4"-dichlorophenyl-1'-methyl-iminooxymethyl-4')-6-methylphenyl]-N-propargyl-carbamate (Table 47, No. 13)

At 25-30.degree. C., 0.15 g (6.3 mmol) of sodium hydride is added in portions to a solution of 1.9 g (5 mmol) of the carbamate from Example 16d in 20 ml of dimethylformamide. When no more gas evolves, 0.75 g (6.3 mmol) of propargyl bromide is added and the whole is stirred overnight at room temperature. The reaction mixture is diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. There is obtained 1.4 g (3.3 mmol=67%) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.75 (S, broad, 1H, phenyl); 7.2-7.6 (m, 5H, phenyl); 5.2 (dd, 2H, I=12 Hz, OCH.sub.2); 4.4 (dd, broad, I=16 Hz, NCH.sub.2); (S, 3H, OCH.sub.3); 2.3 (S, 3H, CH.sub.3); 2.25 (S, broad, 1H, C.tbd.CH); 2.2 (S, 3H, CH.sub.3); the .sup.1 H-NMR spectrum also contains signals of about 20% of the amide rotamer.

The compounds described in the following tables may be prepared analogously.

TABLE 41______________________________________ #STR272## I: R.sup.1 = H, CH.sub.3 II: R.sup.1 = CH.sub.3, X = CH.sub.3 III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3 IV: R.sup.1 = Allyl, X = CH.sub.3 V: R.sup.1 = Propargyl, X = CH.sub.3 VI: R.sup.1 = CH.sub.2 --OCH.sub.3, X = CH.sub.3 VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3 VIII: R.sup.1 = H, X = Cl IX: R.sup.1 = CH.sub.3, X = Cl X: R.sup.1 = C.sub.2 H.sub.5, X = Cl XI: R.sup.1 = Allyl, X = Cl XII: R.sup.1 = Propargyl, X = Cl XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, X = Cl XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl -Compound I from Table 41 has for instance the following structural formula: #STR273## No. T.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7) 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloro allyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-Cl--C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chlor oallyl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chlor oallyl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 42______________________________________ #STR274## No. B______________________________________ 1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.2 H.sub.6 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N-CH.sub.3 -Pyrrolyl-2 21 N-C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N-CH.sub.3 -Pyrazolyl-4 127 N-C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 -N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazol yl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH.sub.3 -Oxazolyl-4 234 3-C.sub.6 H.sub.5 -Oxazolyl-4 235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 257 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Thiazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Thiazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiaz olyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazol yl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazol yl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazoly l-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazolyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazol yl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Thiazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazol yl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazo lyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazol yl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazo lyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazol yl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiaz olyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazo lyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiaz olyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazo lyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 1-Naphthyl 385 2-Naphthyl______________________________________ TABLE 43______________________________________ #STR275## No. T.sub.m______________________________________1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4,-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 ----CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)-CH.sub.3 333 3-C(.dbd.NO-Allyl)-CH.sub.3 334 4-C(.dbd.NO-Allyl)-CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)-CH.sub.3 338 2-C(.dbd.NO-Propargyl)-CH.sub.3 339 3-C(.dbd.NO-Propargyl)-CH.sub.3 340 4-C(.dbd.NO-Propargyl)-CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chloroallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroal lyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5' 641 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub. 3) 642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.N--O--CH.sub.2 --CH.sub.2 --OCH.sub.3) 644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroa llyl) 650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.3 H.sub.5) 653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OCH.sub.3) 654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--OC.sub.2 H.sub.5) 655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.3 H.sub.7) 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-i-C.sub.3 H.sub.7) 657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Allyl) 658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-trans-Chloroa llyl) 659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-Propargyl) 660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O-n-C.sub.4 H.sub.9) 661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C.dbd.N--O--CH.sub.2 --C.sub.6 H.sub.5) 662 2-O-n-C.sub.4 H.sub.9 663 2-O-i-C.sub.4 H.sub.9 664 2-O-s-C.sub.4 H.sub.9 665 2-O-t-C.sub.4 H.sub.9 666 2-Neopentyloxy 667 3-O-n-C.sub.4 H.sub.9 668 3-O-i-C.sub.4 H.sub.9 669 3-O-s-C.sub.4 H.sub.9 670 3-O-t-C.sub.4 H.sub.9 671 3-Neopentyloxy 672 4-O-n-C.sub.4 H.sub.9 673 4-O-i-C.sub.4 H.sub.9 674 4-O-s-C.sub.4 H.sub.9 675 4-O-t-C.sub.4 H.sub.9 676 4-Neopentyloxy 677 3-CH.sub.3 -4-OCH.sub.3 678 3-CH.sub.3 -4-OC.sub.2 H.sub.5 679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7 680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9 681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9 682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9 683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9 684 3-CH.sub.3 -4-Neopentyloxy 685 2-CH.sub.3 -3-OCH.sub.3 686 2-CH.sub.3 -4-OCH.sub.3 687 2-CH.sub.3 -5-OCH.sub.3 688 2-CH.sub.3 -6-OCH.sub.3 689 3-CH.sub.3 -4-OCH.sub.3 690 3-CH.sub.3 -5-OCH.sub.3 691 3-CH.sub.3 -6-OCH.sub.3 692 4-CH.sub.3 -5-O--CH.sub.3 693 4-CH.sub.3 -6-O--CH.sub.3 694 4-CH.sub.3 -6-OCH.sub.3 695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7 696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7 703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7 705 2-Cl-3-OCH.sub.3 706 2-Cl-4-OCH.sub.3 707 2-Cl-5-OCH.sub.3 708 2-Cl-6-OCH.sub.3 709 3-Cl-4-OCH.sub.3 710 3-Cl-5-OCH.sub.3 711 3-Cl-6-OCH.sub.3 712 4-Cl-5-OCH.sub.3 713 4-Cl-6-OCH.sub.3 714 5-Cl-6-OCH.sub.3______________________________________ TABLE 44______________________________________ #STR276## No. B______________________________________1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N--CH.sub.3 -Pyrazolyl-4 127 N--C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH.sub.3 -Oxazolyl-4 234 3-C.sub.6 H.sub.5 -Oxazolyl-4 235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 257 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria zolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz olyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 1-Naphthyl 385 2-Naphthyl______________________________________ TABLE 45______________________________________ #STR277## No. T.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2 100 2,4,6-(i-C.sub.3 H.sub.7).sub.3 101 2-s-C.sub.4 H.sub.9 102 3-s-C.sub.4 H.sub.9 103 4-s-C.sub.4 H.sub.9 104 2-t-C.sub.4 H.sub.9 105 3-t-C.sub.4 H.sub.9 106 4-t-C.sub.4 H.sub.9 107 2,3-(t-C.sub.4 H.sub.9).sub.2 108 2,4-(t-C.sub.4 H.sub.9).sub.2 109 2,5-(t-C.sub.4 H.sub.9).sub.2 110 2,6-(t-C.sub.4 H.sub.9).sub.2 111 3,4-(t-C.sub.4 H.sub.9).sub.2 112 2,4,6-(t-C.sub.4 H.sub.9).sub.3 113 4-n-C.sub.9 H.sub.19 114 4-n-C.sub.12 H.sub.25 115 4-n-C.sub.15 H.sub.31 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3 119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3 120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3 121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9 122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9 123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7 124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7 125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7 126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3 127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH.sub.3 132 2-cyclo-C.sub.6 H.sub.11 133 3-cyclo-C.sub.6 H.sub.11 134 4-cyclo-C.sub.6 H.sub.11 135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3 136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11 137 2-CH.sub.2 --C.sub.6 H.sub.5 138 3-CH.sub.2 --C.sub.6 H.sub.5 139 4-CH.sub.2 --C.sub.6 H.sub.5 140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3 141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5 142 2-C.sub.6 H.sub.5 143 3-C.sub.6 H.sub.5 144 4-C.sub.6 H.sub.5 145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4) 146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2 147 2-Cl, 4-C.sub.6 H.sub.5 148 2-Br, 4-C.sub.6 H.sub.5 149 2-C.sub.6 H.sub.5, 4-Cl 150 2-C.sub.6 H.sub.5, 4-Br 151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl 152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br 153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5 154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5 155 2-cyclo-C.sub.6 H.sub.11, 4-Cl 156 2-cyclo-C.sub.6 H.sub.11, 4-Br 157 2-Cl, 4-cyclo-C.sub.6 H.sub.11 158 2-Br, 4-cyclo-C.sub.6 H.sub.11 159 2-OCH.sub.3 160 3-OCH.sub.3 161 4-OCH.sub.3 162 2-OC.sub.2 H.sub.5 163 3-O--C.sub.2 H.sub.5 164 4-O--C.sub.2 H.sub.5 165 2-O-n-C.sub.3 H.sub.7 166 3-O-n-C.sub.3 H.sub.7 167 4-O-n-C.sub.3 H.sub.7 168 2-O-i-C.sub.3 H.sub.7 169 3-O-i-C.sub.3 H.sub.7 170 4-O-i-C.sub.3 H.sub.7 171 2-O-n-C.sub.6 H.sub.13 172 3-O-n-C.sub.6 H.sub.13 173 4-O-n-C.sub.6 H.sub.13 174 2-O-n-C.sub.8 H.sub.17 175 3-O-n-C.sub.8 H.sub.17 176 4-O-n-C.sub.8 H.sub.17 177 2-O--CH.sub.2 C.sub.6 H.sub.5 178 3-O--CH.sub.2 C.sub.6 H.sub.5 179 4-O--CH.sub.2 C.sub.6 H.sub.5 180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5 183 2,4-(OCH.sub.3).sub.2 184 2-CF.sub.3 185 3-CF.sub.3 186 4-CF.sub.3 187 2-OCF.sub.3 188 3-OCF.sub.3 189 4-OCF.sub.3 190 3-OCH.sub.2 CHF.sub.2 191 2-NO.sub.2 192 3-NO.sub.2 193 4-NO.sub.2 194 2-CN 195 3-CN 196 4-CN 197 2-CH.sub.3, 3-Cl 198 2-CH.sub.3, 4-Cl 199 2-CH.sub.3, 5-Cl 200 2-CH.sub.3, 6-Cl 201 2-CH.sub.3, 3-F 202 2-CH.sub.3, 4-F 203 2-CH.sub.3, 5-F 204 2-CH.sub.3, 6-F 205 2-CH.sub.3, 3-Br 206 2-CH.sub.3, 4-Br 207 2-CH.sub.3, 5-Br 208 2-CH.sub.3, 6-Br 209 2-Cl, 3-CH.sub.3 210 2-Cl, 4-CH.sub.3 211 2-Cl, 5-CH.sub.3 212 2-F, 3-CH.sub.3 213 2-F, 4-CH.sub.3 214 2-F, 5-CH.sub.3 215 2-Br, 3-CH.sub.3 216 2-Br, 4-CH.sub.3 217 2-Br, 5-CH.sub.3 218 3-CH.sub.3, 4-Cl 219 3-CH.sub.3, 5-Cl 220 3-CH.sub.3, 4-F 221 3-CH.sub.3, 5-F 222 3-CH.sub.3, 4-Br 223 3-CH.sub.3, 5-Br 224 3-F, 4-CH.sub.3 225 3-Cl, 4-CH.sub.3 226 3-Br, 4-CH.sub.3 227 2-Cl, 4,5-(CH.sub.3).sub.2 228 2-Br, 4,5-(CH.sub.3).sub.2 229 2-Cl, 3,5-(CH.sub.3).sub.2 230 2-Br, 3,5-(CH.sub.3).sub.2 231 2,6-Cl.sub.2, 4-CH.sub.3 232 2,6-F.sub.2, 4-CH.sub.3 233 2,6-Br.sub.2, 4-CH.sub.3 234 2,4-Br.sub.2, 6-CH.sub.3 235 2,4-F.sub.2, 6-CH.sub.3 236 2,4-Br.sub.2, 6-CH.sub.3 237 2,6-(CH.sub.3).sub.2, 4-F 238 2,6-(CH.sub.3).sub.2, 4-Cl 239 2,6-(CH.sub.3).sub.2, 4-Br 240 3,5-(CH.sub.3).sub.2, 4-F 241 3,5-(CH.sub.3).sub.2, 4-Cl 242 3,5-(CH.sub.3).sub.2, 4-Br 243 2,3,6-(CH.sub.3).sub.3, 4-F 244 2,3,6-(CH.sub.3).sub.3, 4-Cl 245 2,3,6-(CH.sub.3).sub.3, 4-Br 246 2,4-(CH.sub.3).sub.2, 6-F 247 2,4-(CH.sub.3).sub.2, 6-Cl 248 2,4-(CH.sub.3).sub.2, 6-Br 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3 250 2-Cl, 4-NO.sub.2 251 2-NO.sub.2, 4-Cl 252 2-OCH.sub.3, 5-NO.sub.2 253 2,4-Cl.sub.2, 5-NO.sub.2 254 2,4-Cl.sub.2, 6-NO.sub.2 255 2,6-Cl.sub.2, 4-NO.sub.2 256 2,6-Br.sub.2, 4-NO.sub.2 257 2,6-I.sub.2, 4-NO.sub.2 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl 259 2-CO.sub.2 CH.sub.3 260 3-CO.sub.2 CH.sub.3 261 4-CO.sub.2 CH.sub.3 262 2-CO.sub.2 (C.sub.2 H.sub.5) 263 3-CO.sub.2 (C.sub.2 H.sub.5) 264 4-CO.sub.2 (C.sub.2 H.sub.5) 265 2-CO.sub.2 (n-C.sub.3 H.sub.7) 266 3-CO.sub.2 (n-C.sub.3 H.sub.7) 267 4-CO.sub.2 (n-C.sub.3 H.sub.7) 268 2-CO.sub.2 (i-C.sub.3 H.sub.7) 269 3-CO.sub.2 (i-C.sub.3 H.sub.7) 270 4-CO.sub.2 (i-C.sub.3 H.sub.7) 271 2-CO.sub.2 (n-C.sub.6 H.sub.13) 272 3-CO.sub.2 (n-C.sub.6 H.sub.13) 273 4-CO.sub.2 (n-C.sub.6 H.sub.13) 274 2-CH.sub.2 --OCH.sub.3 275 3-CH.sub.2 --OCH.sub.3 276 4-CH.sub.2 --OCH.sub.3 277 2-CH.sub.2 O(C.sub.2 H.sub.5) 278 3-CH.sub.2 O(C.sub.2 H.sub.5) 279 4-CH.sub.2 O(C.sub.2 H.sub.5) 280 2-CH.sub.2 O(n-C.sub.3 H.sub.7) 281 3-CH.sub.2 O(n-C.sub.3 H.sub.7) 282 4-CH.sub.2 O(n-C.sub.3 H.sub.7) 283 2-CH.sub.2 O(i-C.sub.3 H.sub.7) 284 3-CH.sub.2 O(i-C.sub.3 H.sub.7) 285 4-CH.sub.2 O(i-C.sub.3 H.sub.7) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO--CH.sub.3 290 3-CO--CH.sub.3 291 4-CO--CH.sub.3 292 2-CO--CH.sub.2 --CH.sub.3 293 3-CO--CH.sub.2 --CH.sub.3 294 4-CO--CH.sub.2 --CH.sub.3 295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3 298 2-CO--CH(CH.sub.3)--CH.sub.3 299 3-CO--CH(CH.sub.3)--CH.sub.3 300 4-CO--CH(CH.sub.3)--CH.sub.3 301 2-Me-4-CHO 302 2-Me-4-CH.sub.3 --CO 303 2-Me-4-CH.sub.3 --CH.sub.2 --CO 304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO 306 2,5-Me.sub.2 -4-CHO 307 2,5-Me.sub.2 -4-CH.sub.3 --CO 308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 311 2-Cl-4-CHO 312 2-Cl-4-CH.sub.3 --CO 313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO 314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO 315 2,5-Cl.sub.2 -4-CHO 316 2,5-Cl.sub.2 -4-CH.sub.3 --CO 317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO 318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO 319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO 320 2-C(.dbd.NOCH.sub.3)--CH.sub.3 321 3-C(.dbd.NOCH.sub.3)--CH.sub.3 322 4-C(.dbd.NOCH.sub.3)--CH.sub.3 323 2-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 324 3-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 325 4-C(.dbd.NOC.sub.2 H.sub.5)--CH.sub.3 326 2-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 327 3-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 328 4-C(.dbd.NO-n-C.sub.3 H.sub.7)--CH.sub.3 329 2-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 330 3-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 331 4-C(.dbd.NO-i-C.sub.3 H.sub.7)--CH.sub.3 332 2-C(.dbd.NO-Allyl)--CH.sub.3 333 3-C(.dbd.NO-Allyl)--CH.sub.3 334 4-C(.dbd.NO-Allyl)--CH.sub.3 335 2-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 336 3-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 337 4-C(.dbd.NO-trans-Chloroallyl)--CH.sub.3 338 2-C(.dbd.NO-Propargyl)--CH.sub.3 339 3-C(.dbd.NO-Propargyl)--CH.sub.3 340 4-C(.dbd.NO-Propargyl)--CH.sub.3 341 2-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 342 3-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 343 4-C(.dbd.NO-n-C.sub.4 H.sub.9)--CH.sub.3 344 2-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 345 3-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 346 4-C(.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3 347 2-CH.sub.3 -4-CH.dbd.NOCH.sub.3 348 2-CH.sub.3 -4-CH.dbd.NOC.sub.2 H.sub.5 349 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.3 H.sub.7 350 2-CH.sub.3 -4-CH.dbd.NO-i-C.sub.3 H.sub.7 351 2-CH.sub.3 -4-CH.dbd.NO-Allyl 352 2-CH.sub.3 -4-CH.dbd.NO-(trans-Chloroallyl) 353 2-CH.sub.3 -4-CH.dbd.NO-Propargyl 354 2-CH.sub.3 -4-CH.dbd.NO-n-C.sub.4 H.sub.9 355 2-CH.sub.3 -4-CH.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5 356 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 357 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 358 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.3 H.sub.7) 359 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 360 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Allyl) 361 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-trans-Chloroallyl) 362 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-Propargyl) 363 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 364 2-CH.sub.3 -4-(CH.sub.3 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.3) 366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--C.sub.2 H.sub.5) 367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.3 H.sub.7) 368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-i-C.sub.3 H.sub.7 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Allyl) 370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-trans-Chlor oallyl) 371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-Propargyl) 372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO-n-C.sub.4 H.sub.9) 373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C.dbd.NO--CH.sub.2 --C.sub.6 H.sub.5) 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOCH.sub.3) 375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NOC.sub.2 H.sub.5) 376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub. 3 H.sub.7) 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-i-C.sub.3 H.sub.7) 378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Allyl) 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-trans-Ch loroallyl) 380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-Proparyl) 381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO-n-C.sub.4 H.sub.9) 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C.dbd.NO--CH.sub. 2 --C.sub.6 H.sub.5) 383 2-C.sub.6 H.sub.5 384 3-C.sub.6 H.sub.5 385 4-C.sub.6 H.sub.5 386 2-(2'-F--C.sub.6 H.sub.4) 387 2-(3'-F--C.sub.6 H.sub.4) 388 2-(4'-F--C.sub.6 H.sub.4) 389 3-(2'-F--C.sub.6 H.sub.4) 390 3-(3'-F--C.sub.6 H.sub.4) 391 3-(4'-F--C.sub.6 H.sub.4) 392 4-(2'-F--C.sub.6 H.sub.4) 393 4-(3'-F--C.sub.6 H.sub.4) 394 4-(4'-F--C.sub.6 H.sub.4) 395 2-(2'-Cl--C.sub.6 H.sub.4) 396 2-(3'-Cl--C.sub.6 H.sub.4) 397 2-(4'-Cl--C.sub.6 H.sub.4) 398 3-(2'-Cl--C.sub.6 H.sub.4) 399 3-(3'-Cl--C.sub.6 H.sub.4) 400 3-(4'-Cl--C.sub.6 H.sub.4) 401 4-(2'-Cl--C.sub.6 H.sub.4) 402 4-(3'-Cl--C.sub.6 H.sub.4) 403 4-(4'-Cl--C.sub.6 H.sub.4) 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4) 406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4) 407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4) 408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4) 409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4) 410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4) 411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4) 412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4) 413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4) 414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 423 2-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 424 2-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 425 2-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 426 3-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 427 3-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 428 3-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 429 4-(2'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 430 4-(3'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 431 4-(4'-(CH.sub.3 --C(.dbd.NOAllyl))-C.sub.6 H.sub.4) 432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4) 451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4) 452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4) 453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4) 454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4) 455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4) 456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4) 457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4) 458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4) 459 2-(2'-NC--C.sub.6 H.sub.4) 460 2-(3'-NC--C.sub.6 H.sub.4) 461 2-(4'-NC--C.sub.6 H.sub.4) 462 3-(2'-NC--C.sub.6 H.sub.4) 463 3-(3'-NC--C.sub.6 H.sub.4) 464 3-(4'-NC--C.sub.6 H.sub.4) 465 4-(2'-NC--C.sub.6 H.sub.4) 466 4-(3'-NC--C.sub.6 H.sub.4) 467 4-(4'-NC--C.sub.6 H.sub.4) 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4) 469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4) 470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4) 471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4) 472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4) 473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4) 474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4) 475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4) 476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4) 477 2-O--C.sub.6 H.sub.5 475 3-O--C.sub.6 H.sub.5 476 4-O--C.sub.6 H.sub.5 478 2-O-(2'-F--C.sub.6 H.sub.4) 479 2-O-(3'-F--C.sub.6 H.sub.4) 480 2-O-(4'-F--C.sub.6 H.sub.4) 481 3-O-(2'-F--C.sub.6 H.sub.4) 482 3-O-(3'-F--C.sub.6 H.sub.4) 483 3-O-(4'-F--C.sub.6 H.sub.4) 484 4-O-(2'-F--C.sub.6 H.sub.4) 485 4-O-(3'-F--C.sub.6 H.sub.4) 486 4-O-(4'-F--C.sub.6 H.sub.4) 487 2-O-(2'-Cl--C.sub.6 H.sub.4) 488 2-O-(3'-Cl--C.sub.6 H.sub.4) 489 2-O-(4'-Cl--C.sub.6 H.sub.4) 490 3-O-(2'-Cl--C.sub.6 H.sub.4) 491 3-O-(3'-Cl--C.sub.6 H.sub.4) 492 3-O-(4'-Cl--C.sub.6 H.sub.4) 493 3-O-(4'-Cl--C.sub.6 H.sub.4) 494 4-O-(2'-Cl--C.sub.6 H.sub.4) 495 4-O-(3'-Cl--C.sub.6 H.sub.4) 496 4-O-(4'-Cl--C.sub.6 H.sub.4) 497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4) 504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4) 505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4) 506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4) 513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4) 514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4) 515 2-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 516 2-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 517 2-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 518 3-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 519 3-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 520 3-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 521 4-O-(2'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 522 4-O-(3'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 523 4-O-(4'-(CH.sub.3 --C(.dbd.NOAllyl))--C.sub.6 H.sub.4) 524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4) 533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4) 540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4) 541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4) 542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4) 549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4) 550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4) 551 2-O-(2'-NC--C.sub.6 H.sub.4) 552 2-O-(3'-NC--C.sub.6 H.sub.4) 553 2-O-(4'-NC--C.sub.6 H.sub.4) 554 3-O-(2'-NC--C.sub.6 H.sub.4) 555 3-O-(3'-NC--C.sub.6 H.sub.4) 556 3-O-(4'-NC--C.sub.6 H.sub.4) 557 4-O-(2'-NC--C.sub.6 H.sub.4) 558 4-O-(3'-NC--C.sub.6 H.sub.4) 559 4-O-(4'-NC--C.sub.6 H.sub.4) 560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.5) 561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.5) 562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.5) 563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.5) 564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.5) 565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.5) 566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.5) 567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.5) 568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.5) 569 2-Pyridinyl-2' 570 2-Pyridinyl-3' 571 2-Pyridinyl-4' 572 3-Pyridinyl-2' 573 3-Pyridinyl-3' 574 3-Pyridinyl-4' 575 4-Pyridinyl-2' 576 4-Pyridinyl-3' 577 4-Pyridinyl-4' 578 2-Pyrimidinyl-2' 579 2-Pyrimidinyl-3' 580 2-Pyrimidinyl-4' 581 3-Pyrimidinyl-2' 582 3-Pyrimidinyl-3' 583 3-Pyrimidinyl-4' 584 4-Pyrimidinyl-2' 585 4-Pyrimidinyl-3' 586 4-Pyrimidinyl-4' 587 2-Pyrazolyl-1' 588 2-Pyrazolyl-3' 589 2-Pyrazolyl-4' 590 3-Pyrazolyl-1' 591 3-Pyrazolyl-3' 592 3-Pyrazolyl-4' 593 4-Pyrazolyl-1' 594 4-Pyrazolyl-3' 595 4-Pyrazolyl-4' 596 2-Isoxazolyl-3' 597 2-Isoxazolyl-4' 598 2-Isoxazolyl-5' 599 3-Isoxazolyl-3' 600 3-Isoxazolyl-4' 601 3-Isoxazolyl-5' 602 4-Isoxazolyl-3' 603 4-Isoxazolyl-4' 604 4-Isoxazolyl-5' 605 2-Isothiazolyl-3' 606 2-Isothiazolyl-4' 607 2-Isothiazolyl-5' 608 3-Isothiazolyl-3' 609 3-Isothiazolyl-4' 610 3-Isothiazolyl-5' 611 4-Isothiazolyl-3' 612 4-Isothiazolyl-4' 613 4-Isothiazolyl-5' 614 2-Imidazolyl-1' 615 2-Imidazolyl-2' 616 2-Imidazolyl-4' 617 3-Imidazolyl-1' 618 3-Imidazolyl-2' 619 3-Imidazolyl-4' 620 4-Imidazolyl-1' 621 4-Imidazolyl-2' 622 4-Imidazolyl-4' 623 2-Oxazolyl-2' 624 2-Oxazolyl-4' 625 2-Oxazolyl-5' 626 3-Oxazolyl-2' 627 3-Oxazolyl-4' 628 3-Oxazolyl-5' 629 4-Oxazolyl-2' 630 4-Oxazolyl-4' 631 4-Oxazolyl-5' 632 2-Thiazolyl-2' 633 2-Thiazolyl-4' 634 2-Thiazolyl-5' 635 3-Thiazolyl-2' 636 3-Thiazolyl-4' 637 3-Thiazolyl-5' 638 4-Thiazolyl-2' 639 4-Thiazolyl-4' 640 4-Thiazolyl-5'______________________________________ TABLE 46______________________________________ #STR278## No. B______________________________________ 1 Pyrrolyl-3 2 N--CH.sub.3 -Pyrrolyl-3 3 N--C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N--CH.sub.3 -Pyrrolyl-2 21 N--C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2 70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2 71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2 101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2 102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2 103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2 104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2 105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2 106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2 107 Thienyl-3 108 5-CH.sub.3 -Thienyl-3 109 5-C.sub.6 H.sub.5 -Thienyl-3 110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3 113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3 116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3 119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3 120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3 121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3 122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3 123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3 124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3 125 Pyrazolyl-4 126 N-CH.sub.3 -Pyrazolyl-4 127 N-C.sub.6 H.sub.5 -Pyrazolyl-4 128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4 131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4 134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4 137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4 140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4 143 3-CH.sub.3 --N-Methylpyrazolyl-4 144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4 145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH.sub.3 -Isoxazolyl-5 162 3-C.sub.6 H.sub.5 -Isoxazolyl-5 163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5 166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5 169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5 172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5 175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH.sub.3 -4-Chloroisoxazolyl-5 180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5 181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH.sub.3 -Isoxazolyl-3 198 5-C.sub.6 H.sub.5 -Isoxazolyl-3 199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3 202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3 205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3 208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3 211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH.sub.3 -Isothiazolyl-5 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5 217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5 220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5 223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5 226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5 229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH.sub.3 -Oxazolyl-4 234 3-C.sub.6 H.sub.5 -Oxazolyl-4 235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4 238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4 241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4 244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4 247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH.sub.3 -Thiazolyl-4 252 2-C.sub.6 H.sub.5 -Thiazolyl-4 253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4 256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 257 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4 259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4 262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4 265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4 268 N--CH.sub.3 -1,2,4-Triazolyl-5 269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5 270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5 271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazoly l-5 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2 288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2 289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3 306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3 307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5 324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5 325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3 342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3 343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2 360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2 361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2______________________________________ TABLE 47______________________________________Selected physical data of some compounds #STR279## IR (cm.sup.-1) or No. X.sub.m R.sup.1 .sup.1 H-NMR (ppm) mp______________________________________ 1 4-Cl H 133 2 3,4-Cl.sub.2 H 109 3 4-t-C.sub.4 H.sub.9 H 86 4 4-CH.sub.3 H 117 5 4-CF.sub.3 H 103 6 3-Br H 99 7 3-Cl H 93 8 3-CF.sub.3 H 88 9 3,5-Cl.sub.2 H 100 10 3,4-(CH.sub.3).sub.2 H 127 11 3,4-Cl.sub.2 CH.sub.3 74 12 3,4-Cl.sub.2 Allyl 3.65(S, 3H); 2.2(S, 6H) 13 3,4-Cl.sub.2 Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 14 3,4-Cl.sub.2 CH.sub.2 --OCH.sub.3 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 15 3,4-Cl.sub.2 CO--OCH.sub.3 137 16 4-t-C.sub.4 H.sub.9 CH.sub.3 3.65(S, 3H); 2.25(S, 3H); 2.2(S, 3H) 17 4-t-C.sub.4 H.sub.9 Allyl 69 18 4-t-C.sub.4 H.sub.9 Propargyl 117 19 4-t-C.sub.4 H.sub.9 CH.sub.2 --OCH.sub.3 3.65(S, 3H); 2.25(S, 3H); 117 2.2(S, 3H) 20 4-t-C.sub.4 H.sub.9 CO--OCH.sub.3 3.65; 2.1 119 21 4-CH.sub.3 CH.sub.3 69 22 4-CH.sub.3 Allyl 3.65(S, 3H); 2.25(S, 3H); 2.2(S, 3H) 23 4-CH.sub.3 Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 24 4-CH.sub.3 CH.sub.2 --OCH.sub.3 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 25 4-CH.sub.3 CO--OCH.sub.3 97 26 4-CF.sub.3 CH.sub.3 76 27 4-CF.sub.3 Allyl 3.65(S, 3H); 2.3(S, 3H); 2.25(S, 3H) 28 4-CF.sub.3 Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.25(S, 3H) 29 4-CF.sub.3 CH.sub.2 --OCH.sub.3 3.65(S, 3H); 2.25(S, 6H) 30 4-CF.sub.3 CO--OCH.sub.3 103 31 4-Cl CH.sub.3 106 32 4-Cl Allyl 3.65(S, 3H); 2.2(2S, each 3H) 33 4-Cl Propargyl 3.65(S, 3H); 2.3(S, 3H; 2.2(S, 3H) 34 4-Cl CH.sub.2 --OCH.sub.3 3.65(S, 3H); 2.25(S, 3H; 2.2(S, 3H) 35 4-Cl CO--OCH.sub.3 109 36 3-Br CH.sub.3 75 37 3-Br Allyl 3.65(S, 3H); 2.2(2S, each 3H 38 3-Br Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 39 3-Br CH.sub.2 --OCH.sub.3 72 40 3-Br CO--OCH.sub.3 131 41 3-Cl CH.sub.3 84 42 3-Cl Allyl 3.65(S, 3H); 2.25(S, 3H); 2.2(S, 3H) 43 3-Cl Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 44 3-Cl CH.sub.2 --OCH.sub.3 66 45 3-Cl CO--OCH.sub.3 123 46 3-CF.sub.3 CH.sub.3 63 47 3-CF.sub.3 Allyl 64 48 3-CF.sub.3 Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.25(S, 3H) 49 3-CF.sub.3 CH.sub.2 --OCH.sub.3 89 50 3-CF.sub.3 CO--OCH.sub.3 136 51 4-Br CO--OCH.sub.3 103 52 4-Br H 108 53 4-Br Propargyl 1710, 1486, 1469, 1447, 1376, 1299, 1252, 1026, 1008, 774 54 4-Br CH.sub.2 --OCH.sub.3 1715, 1468, 1445, 1370, 1301, 1274, 1090, 1059, 1008, 775 55 3,4-(CH.sub.3).sub.2 CH.sub.3 oil 56 3,4-(CH.sub.3).sub.2 Allyl oil 57 3,4-(CH.sub.3).sub.2 Propargyl oil 58 3,4-(CH.sub.3).sub.2 CH.sub.2 --OCH.sub.3 oil 59 3,4-(CH.sub.3).sub.2 CO--OCH.sub.3 135 60 3,5-Cl.sub.2 CH.sub.3 95 61 3,5-Cl.sub.2 Allyl 97 62 3,5-Cl.sub.2 Propargyl 100 63 3,5-Cl.sub.2 CH.sub.2 --OCH.sub.3 112 64 3,5-Cl.sub.2 CO--OCH.sub.3 160______________________________________ TABLE 48__________________________________________________________________________Selected physical data of some compounds #STR280## IR (cm.sup.-1) or No. X.sub.m R.sup.1 .sup.1 H-NMR (ppm) mp__________________________________________________________________________ 1 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 H 82 2 2,4-(CH.sub.3).sub.2 H 131 3 2,5-(CH.sub.3).sub.2 H 124 4 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OC.sub.2 H.sub.5 H 102 5 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--OC.sub.2 H.sub.5 H 116 6 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3) .dbd.N--OCH.sub.3 H 122 7 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 CH.sub.3 4.0(S, 3H); 3.65(S, 3H) 8 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 Allyl 101 9 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 Propargyl 4.0(S, 3H); 3.65(S, 3H) 10 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 CH.sub.2 --OCH.sub.3 4.0(S, 3H); 3.65(S, 3H) 11 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--OCH.sub.3 CO--OCH.sub.3 122 12 2,4-(CH.sub.3).sub.2 CH.sub.3 3.65(S, 3H); 2.25(2s, each 3H) 13 2,4-(CH.sub.3).sub.2 Allyl 59 14 2,4-(CH.sub.3).sub.2 Propargyl 3.65(S, 3H); 2.25(3s, each 3H) 15 2,4-(CH.sub.3).sub.2 CH.sub.2 --OCH.sub.3 76 16 2,4-(CH.sub.3).sub.2 CO--OCH.sub.3 133 17 2,5-(CH.sub.3).sub.2 CH.sub.3 3.65(S, 3H); 2.3(S, 3H) 18 2,5-(CH.sub.3).sub.2 Allyl 56 19 2,5-(CH.sub.3).sub.2 Propargyl 80 20 2,5-(CH.sub.3).sub.2 CH.sub.2 --OCH.sub.3 3.65(S, 3H); 2.3(S, 3H) 80 21 2,5-(CH.sub.3).sub.2 CH.sub.2 --OCH.sub.3 140 22 2-CH.sub.3 H 107 23 2-CH.sub.3 Propargyl oil 24 2-CH.sub.3 CO--OCH.sub.3 135 25 2-CH.sub.3 CH.sub.2 --OCH.sub.3 oil 26 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--O-- H 97 Allyl 27 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--O-- Propargyl oil Allyl 28 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--O-- CO--OCH.sub.3 130 Allyl 29 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--O-- CH.sub.2 --OCH.sub.3 oil Allyl 30 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--O--C.sub.2 H.sub.5 CH.sub.3 oil 31 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--O- -C.sub.2 H.sub.5 Allyl 75 32 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--O--C.sub.2 H.sub.5 Propargyl 77 33 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--O- -C.sub.2 H.sub.5 CH.sub.2 --OCH.sub.3 oil 34 2-CH.sub.3 -4-C(CH.sub.3).dbd.N--O--C.sub.2 H.sub.5 CO--OCH.sub.3 oil 35 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--OCH.sub.3 CH.sub.3 oil 36 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3) .dbd.N--OCH.sub.3 Allyl 104 37 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--OCH.sub.3 Propargyl oil 38 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3) .dbd.N--OCH.sub.3 CH.sub.2 --OCH.sub.3 oil 39 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--OCH.sub.3 CO--OCH.sub.3 158 40 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--OC.sub.2 H.sub.5 CH.sub.3 oil 41 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--OC.sub.2 H.sub.5 Allyl 71 42 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--OC.sub.2 H.sub.5 Propargyl oil 43 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--OC.sub.2 H.sub.5 CH.sub.2 --OCH.sub.3 oil 44 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd.N--OC.sub.2 H.sub.5 CO--OCH.s ub.3 128__________________________________________________________________________ TABLE 49______________________________________ #STR281## No. B______________________________________ 1 2-Pyridyl 2 3-Trifluoromethyl-2-pyridyl 3 5-Trifluoromethyl-2-pyridyl 4 3,5-Bis-(trifluoromethyl)-2-pyridyl 5 3,5-Dichloro-2-pyridyl 6 3-Chloro-5-trifluoromethyl-2-pyridyl 7 3,5-Dichloro-2-pyridyl 8 2-Chloro-4-trifluoromethylphenyl 9 2-Benzothiazolyl 10 5-Chloro-1-methyl-2-benzimidazolyl 11 2-Benzoxazolyl 12 1-Methyl-5-trifluoromethylimide-azo[5,4-a]- pyridin-2-yl 13 5-Chloro-2-pyrimidinyl 14 4-Methyl-5-phenyl-2-thiazolin-2-yl 15 4-Methyl-5-phenyl-2-oxazolin-2-yl 16 7-Trifluoromethyl-4-quinolinyl______________________________________ TABLE 50______________________________________Selected physical data of some compounds - #STR282## No. X.sub.m IR (cm.sup.-1) or .sup.1 H-NMR (ppm) mp______________________________________1 4-NO.sub.2 112 2 3,4-Cl.sub.2 3.8(s, 3H); 3.75(s, 3H) 3 2,4-(CH.sub.3).sub.2 3.75(s, 3H); 3.7(s, 3H) 4 H 3.75(2s, each 3H) 5 4-i-C.sub.3 H.sub.7 3.8(s, 3H); 3.75(s, 3H) 6 3,4-(CH.sub.3).sub.2 3.8(s, 3H); 3.75(s, 3H) 7 3-CH.sub.3 -4-OCH.sub.3 3.85(s, 3H); 3.8(s, 3H); 3.75(s, 3H) 8 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 3.8(2s, each 3H) 9 4-CF.sub.3 3.8(s, 3H); 3.75(s, 3H) 10 3-CH.sub.3 3.8(2s, each 3H) 11 3-CF.sub.3 3.8(s, 3H); 3.75(s, 3H) 12 4-F 3.8(s, 3H); 3.75(s, 3H) 13 4-Br 3.8(s, 3H); 3.75(s, 3H) 14 3-Br 3.8(s, 3H); 3.75(s, 3H) 15 4-t-Bu 3.8(s, 3H); 3.75(s, 3H) 16 4-OCH.sub.3 3.85(s, 3H); 3.8(s, 3H); 3.75(s, 3H) 17 2-CH.sub.3 3.8(s, 3H); 3.75(s, 3H) 18 3-Cl 3.8(s, 3H); 3.75(s, 3H) 19 4-CN 3.8(s, 3H); 3.75(s, 3H) 20 4-C.sub.2 H.sub.5 3.8(s, 3H); 3.75(s, 3H)______________________________________ TABLE 51______________________________________Selected physical data of some compounds - #STR283## No. X.sub.m IR(cm.sup.-1) or .sup.1 H-NMR (ppm) mp______________________________________1 4-Cl 3.8(s, 3H); 3.75(s, 3H) 2 2-Cl 3.8(s, 3H); 3.75(s, 3H) 3 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5).dbd. 3.8(s, 3H); 3.75(s, 3H) N--O-Allyl 4 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5).dbd. 3.9(s, 3H); 3.8(s, 3H); N--O--CH.sub.3 3.75(s, 3H) 5 2-CH.sub.3 -4-C(C.sub.2 H.sub.5).dbd.N--O- 3.8(s, 3H); 3.75(s, 3H) trans-Cl-Allyl 6 2-CH.sub.3 -4-C(C.sub.2 H.sub.5).dbd.N--O- 3.8(s, 3H); 3.75(s, 3H) Allyl 7 2-CH.sub.3 -4-Cl 3.8(s, 3H); 3.75(s, 3H) 8 2-Cl-4-CH.sub.3 3.8(s, 3H); 3.75(s, 3H) 9 2-Cl-5-CH.sub.3 3.8(s, 3H); 3.75(s, 3H) 10 2-CH.sub.3 -4-C(C.sub.2 H.sub.5).dbd.N-- 4.2(q, 2H); 3.8(s, 3H); O-C.sub.2 H.sub.5 3.75(s, 3H) 11 2-CH.sub.3 -4-C(C.sub.2 H.sub.5).dbd.N-- 3.95(s, 3H); 3.8(s, 3H); O--CH.sub.3 3.75(s, 3H) 12 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd. 3.8(s, 3H); 3.75(s, 3H) N--O-trans-Cl-Allyl 13 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd. 4.2(t, 2H); 3.8(s, 3H); --N--O--C.sub.2 H.sub.5 3.75(s, 3H) 14 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3).dbd. 3.95(s, 3H); 3.8(s, 3H); N--O--CH.sub.3 3.75(s, 3H) 15 2-CH.sub.3 -4-C(CH.sub.3).dbd.N --O- 3.8(s, 3H); 3.75(s, 3H) trans-Cl-Allyl 16 2-CH.sub.3 -4-C(CH.sub.3).dbd.N-- 4.2(t, 2H); 3.8(s, 3H); O--C.sub.2 H.sub.5 3.75(s, 3H) 17 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5).dbd. 4.2(t, 2H); 3.8(s, 3H); N--O--C.sub.2 H.sub.5 3.75(s, 3H)______________________________________ TABLE 60______________________________________ #STR284## No. B______________________________________1 Phenyl 2 3-Phenoxyphenyl 3 3-(2-Cyanophenoxy)-phenyl 4 4-Chlorophenyl 5 3-Trifluoromethylphenyl 6 3-tert.-Butoxyphenyl 7 3,5-Dichlorophenyl 8 3,5-Diethylphenyl 9 2-Pyridyl 10 4-Pyrimidinyl 11 6-Phenoxy-pyrimidin-4-yl 12 6-Chloropyrimidin-4-yl 13 6-(2-Fluorophenoxy)-pyrimidin-4-yl 14 6-(2-Methylphenoxy)-pyrimidin-4-yl 15 6-(2-Cyanophenoxy)-pyrimidin-4-yl 16 6-(2,6-Difluorophenoxy)-pyrimidin-4-yl______________________________________

The novel compounds are suitable as fungicides. The fungicidal compounds according to the invention, or agents containing them, may be applied for instance in the form of directly sprayable solutions, powders, suspensions (including high-percentage aqueous, oily or other suspensions), dispersions, emulsions, oil dispersions, pastes, dusts, broadcasting agents, or granules by spraying, atomizing, dusting, broadcasting or watering. The forms of application depend entirely on the purpose for which the agents are being used, but they must ensure as fine a distribution of the active ingredients according to the invention as possible.

Normally, the plants are sprayed or dusted with the active ingredients, or the seeds of the plants are treated with the active ingredients.

The formulations are produced in known manner, for example by extending the active ingredient with solvents and/or carriers, with or without the use of emulsifiers and dispersants; if water is used as solvent, it is also possible to employ other organic solvents as auxiliary solvents. Suitable auxiliaries for this purpose are solvents such as aromatics (e.g., xylene), chlorinated aromatics (e.g., chlorobenzenes), paraffins (e.g., crude oil fractions), alcohols (e.g., methanol, butanol), ketones (e.g., cyclohexanone), amines (e.g., ethanolamine, dimethylformamide), and water; carriers such as ground natural minerals (e.g., kaolins, aluminas, talc and chalk) and ground synthetic minerals (e.g., highly disperse silica and silicates); emulsifiers such as nonionic and anionic emulsifiers (e.g., polyoxyethylene fatty alcohol ethers, alkyl sulfonates and aryl sulfonates); and dispersants such as lignin-sulfite waste liquors and methylcellulose.

Examples of surfactants are: alkali metal, alkaline earth metal and ammonium salts of aromatic sulfonic acids, e.g., ligninsulfonic acid, phenolsulfonic acid, naphthalenesulfonic acid and dibutylnaphthalenesulfonic acid, and of fatty acids, alkyl and alkylaryl sulfonates, and alkyl, lauryl ether and fatty alcohol sulfates, and salts of sulfated hexadecanols, heptadecanols, and octadecanols, salts of fatty alcohol glycol ethers, condensation products of sulfonated naphthalene and naphthalene derivatives with formaldehyde, condensation products of naphthalene or naphthalenesulfonic acids with phenol and formaldehyde, polyoxyethylene octylphenol ethers, ethoxylated isooctylphenol, ethoxylated octylphenol and ethoxylated nonylphenol, alkylphenol polyglycol ethers, tributylphenyl polyglycol ethers, alkylaryl polyether alcohols, isotridecyl alcohol, fatty alcohol ethylene oxide condensates, ethoxylated castor oil, polyoxyethylene alkyl ethers, ethoxylated polyoxypropylene, lauryl alcohol polyglycol ether acetal, sorbitol esters, lignin-sulfite waste liquors and methyl cellulose.

Powders, dusts and broadcasting agents may be prepared by mixing or grinding the active ingredients with a solid carrier.

Granules, e.g., coated, impregnated or homogeneous granules, may be prepared by bonding the active ingredients to solid carriers. Examples of solid carriers are mineral earths such as silicic acids, silica gels, silicates, talc, kaolin, attapulgus clay, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate, magnesium sulfate, magnesium oxide, ground plastics, fertilizers such as ammonium sulfate, ammonium phosphate, ammonium nitrate, and ureas, and vegetable products such as grain meals, bark meal, wood meal, and nutshell meal, cellulosic powders, etc.

Examples of formulations are given below.

I. A solution of 90 parts by weight of the compound from Table 7, No. 1 (7/1) and 10 parts by weight of N-methyl-.alpha.-pyrrolidone, which is suitable for application in the form of very fine drops. II. A mixture of 20 parts by weight of compound 7/2, 80 parts by weight of xylene, 10 parts by weight of the adduct of 8 to 10 moles of ethylene oxide and 1 mole of oleic acid-N-monoethanolamide, 5 parts by weight of the calcium salt of dodecylbenzenesulfonic acid, and 5 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil. By finely dispersing the mixture in water, a dispersion is obtained. III. An aqueous dispersion of 20 parts by weight of compound 7/3, 40 parts by weight of cyclohexanone, 30 parts by weight of isobutanol, 20 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil. IV. An aqueous dispersion of 20 parts by weight of compound 7/4, 25 parts by weight of cyclohexanol, 65 parts by weight of a mineral oil fraction having a boiling point between 210 and 280.degree. C., and 10 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil. V. A hammer-milled mixture of 80 parts by weight of compound 7/5, 3 parts by weight of the sodium salt of diisobutylnaphthalene-.alpha.-sulfonic acid, 10 parts by weight of the sodium salt of a lignin-sulfonic acid obtained from a sulfite waste liquor, and 7 parts by weight of powdered silica gel. By finely dispersing the mixture in water, a spray liquor is obtained. VI. An intimate mixture of 3 parts by weight of compound 7/6 and 97 parts by weight of particulate kaolin. The dust contains 3 wt % of the active ingredient. VII. An intimate mixture of 30 parts by weight of compound 7/7, 92 parts by weight of powdered silica gel and 8 parts by weight of paraffin oil sprayed onto the surface of this silica gel. This formulation of the active ingredient exhibits good adherence. VIII. A stable aqueous dispersion of 40 parts by weight of compound 7/8, 10 parts of the sodium salt of a phenolsulfonic acid-urea-formaldehyde condensate, 2 parts of silica gel and 48 parts of water, which dispersion can be further diluted. IX. A stable oily dispersion of 20 parts by weight of compound 7/9, 2 parts by weight of the calcium salt of dodecylbenzenesulfonic acid, 8 parts by weight of a fatty alcohol polyglycol ether, 2 parts by weight of the sodium salt of a phenolsulfonic acid-urea-formaldehyde condensate and 68 parts by weight of a paraffinic mineral oil.

The novel compounds are extremely effective on a broad spectrum of phytopathogenic fungi, in particular those from the class consisting of the Ascomycetes and Basidiomycetes. Some of them have a systemic action and can be used as foliar and soil fungicides.

The fungicidal compounds are of particular interest for controlling a large number of fungi in various crops or their seeds, especially wheat, rye, barley, oats, rice, Indian corn, lawns, cotton, soybeans, coffee, sugar cane, fruit and ornamentals in horticulture and viticulture, and in vegetables such as cucumbers, beans and cucurbits.

The compounds are applied by treating the fungi, or the seeds, plants, materials or soil to be protected against fungus attack with a fungicidally effective amount of the active ingredients.

The agents may be applied before or after infection of the materials, plants or seed by the fungi.

The compounds I are particularly useful for controlling the following plant diseases:

Erysiphe graminis in cereals, Erysiphe cichoracearum and Sphaerotheca fuliginea in cucurbits, Podosphaera leucotricha in apples, Uncinula necator in vines, Puccinia species in cereals, Rhizoctonia solani in cotton, Ustilago species in cereals and sugar cane, Venturia inaequalis (scab) in apples, Helminthosporium species in cereals, Septoria nodorum in wheat, Botrytis cinerea (gray mold) in strawberries and grapes, Cercospora arachidicola in groundnuts, Pseudocercosporella herpotrichoides in wheat and barley, Pyricularia oryzae in rice, Phytophthora infestans in potatoes and tomatoes, Fusarium and Verticillium species in various plants, Plasmopara viticola in grapes, Alternaria species in fruit and vegetables.

The novel compounds may also be used for protecting materials (timber), for instance against Paecilomyces variotii.

The fungicidal agents generally contain from 0.1 to 95, an preferably from 0.5 to 90, wt % of active ingredient.

The application rates depend on the effect desired, and are from 0.02 to 3 kg of active ingredient per hectare.

When the active ingredients are used for treating seed, amounts of from 0.001 to 50, and preferably from 0.01 to 10, g per kg of seed are generally needed.

When the agents according to the invention are used as fungicides, they may be present together with other active ingredients, e.g., herbicides, insecticides, growth regulators, other fungicides, and fertilizers.

When they are mixed with other fungicides, the spectrum of fungicidal action is in many cases increased.

USE EXAMPLES

The active ingredients used for comparison purposes were isopropyl N-phenylcarbamate (A)--known from GB 574 995 isopropyl N-3-chlorophenylcarbamate (B)--known from GB 574 995--and methyl N-3,4-dichlorophenylcarbamate (C)--known from BE 612 550.

Example 1

Action on Wheat Mildew

Leaves of pot-grown wheat seedlings of the "Fruhgold" variety were sprayed with aqueous liquors containing (dry basis) 80% of active ingredient and 20% of emulsifier, and dusted, 24 hours after the sprayed-on layer had dried, with spores of wheat mildew (Erysiphe graminis var. tritici). The plants were then set up in the greenhouse at from 20 to 22.degree. C. and a relative humidity of from 75 to 80%. The extent of mildew spread was assessed after 7 days.

The results show that active ingredients nos. 1, 2, 3, 4, 8, 9, 20, 23, 31, 33, 34, 35, 36, 42, 43, 44, 47, 48, 52, 53, 54, 55, 56, 57, 60, 61, 62, 63, 64, 67, 69, 70, 71, 72, 74, 78, 79, 85, 87, 89, 90, 91, 92, 93, 94, 95, 104, 105, 106 and 107 from Table 7 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (95%) than prior art comparative agents A (45%), B (45%) and C (45%).

Example 2

Action on Pyricularia oryzae (Protective)

Leaves of pot-grown rice seedlings of the "Bahia" variety were sprayed to runoff with aqueous emulsions containing (dry basis) 80% of active ingredient and 20% of emulsifier, and inoculated 24 hours later with an aqueous spore suspension of Pyricularia oryzae. The plants were then set up in climatic cabinets at 22 to 24.degree. C. and 95 to 99% relative humidity. The extent of fungus attack was assessed after 6 days.

The results show that active ingredients nos. 1, 2, 12, 18, 19, 22, 29, 39, 40, 42, 47, 49, 50, 52, 53, 54, 60, 61, 62, 63, 69, 70, 71, 72, 73, 74, 81, 83, 85, 87, 89, 90, 91, 92, 94, 95, 104, 105, 106 and 107 from Table 7 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (95%) than prior art comparative agents A (30%), B (30%) and C (30%).

Example 3

Action on Wheat Mildew

Leaves of pot-grown wheat seedlings of the "Fruhgold" variety were sprayed with aqueous liquors containing (dry basis) 80% of active ingredient and 20% of emulsifier, and dusted, 24 hours after the sprayed-on layer had dried, with spores of wheat mildew (Erysiphe graminis var. tritici). The plants were then set up in the greenhouse at from 20 to 22.degree. C. and a relative humidity of from 75 to 80%. The extent of mildew spread was assessed after 7 days.

The results show that active ingredient no. 3 from Table 14, nos. 3 and 4 from Table 21, nos. 1, 3, 4, 5, 6, 7, 8, 9, 10, 11, 15, 17, 18, 19, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 31, 32, 33, 34, 35, 36, 37, 38, 39, 40 41, 42, 43 and 44 from Table 48, nos. 7, 8, 9, 10, 11, 13, 14, 15, 16, 17, 18, 20 and 23 from Table 14, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18 and 19 from Table 52, and nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16 and 17 from Table 53 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (100%) than prior art comparative agents A, B and C (15%).

Example 4

Action on Pyricularia oryzae (Protective)

Leaves of pot-grown rice seedlings of the "Bahia" variety were sprayed to runoff with aqueous emulsions containing (dry basis) 80% of active ingredient and 20% of emulsifier, and inoculated 24 hours later with an aqueous spore suspension of Pyricularia oryzae. The plants were then set up in climatic cabinets at 22 to 24.degree. C. and 95 to 99% relative humidity. The extent of fungus attack was assessed after 6 days.

The results show that active ingredient nos. 3, 7, 8, 9, 10, 11, 13, 14, 15, 16, 17, 18, 20, 21, 22 and 24 from Table 14, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18, 19 and 20 from Table 52, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16 and 17 from Table 53, nos. 3 and 4 from Table 21, nos. 4 and 5 from Table 38, nos. 4, 7, 10, 16, 20, 21, 22, 23, 24, 25, 41, 42, 55, 56, 57, 58 and 59 from Table 47, and nos. 1, 4, 5, 6, 7, 8, 11, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 31, 32, 33, 34, 35, 36, 37, 38, 39, 40, 41, 42, 43 and 44 from Table 48 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (100%) than prior art comparative agents A, B and C (0%).

Use Example 5

Action on Botrytis cinerea

Paprika seedlings of the "Neusiedler Ideal Elite" variety were sprayed, after 4 to 5 leaves were well developed, to runoff with aqueous suspensions containing (dry basis) 80% of active ingredient and 20% of emulsifier. After the sprayed-on layer had dried, the plants were sprinkled with a conidial suspension of the fungus Botrytis cinerea, and placed at 22 to 24.degree. C. in a chamber of high humidity. After 5 days, the disease had spread to such a great extent on the untreated plants that the necroses covered the major portion of the leaves.

______________________________________ Percentage leaf attack after spraying with aqueous for- mulations containing 500 ppm Active ingredient of active ingredient______________________________________Table 30, active ingr. no. 2 5 Comparative substance A 100 Comparative substance B 100 Comparative substance C 100 Untreated 100______________________________________

Use Example 6

Action on Plasmopara viticola

Leaves of potted vines of the Muller-Thurgau variety were sprayed with aqueous suspensions containing (dry basis) 80% of active ingredient and 20% of emulsifier. To assess the duration of action, the plants were set up, after the sprayed-on layer had dried, for 8 days in the greenhouse. Then the leaves were infected with a zoospore suspension of Plasmopara viticola. The plants were first placed for 48 hours in a water vapor-saturated chamber at 24.degree. C. and then in a greenhouse for 5 days at from 20 to 30.degree. C. To accelerate and intensify the sporangiophore discharge, the plants were then again placed in the moist chamber for 16 hours. The extent of fungus attack was then assessed on the undersides of the leaves.

______________________________________ Percentage leaf attack after applying aqueous formula- tions containing 500 ppm of Active ingredient active ingredient______________________________________Table 21, active ingr. no. 3 5 Table 21, active ingr. no. 4 0 Table 30, active ingr. no. 1 15 Comparative substance A 65 Comparative substance B 40 Comparative substance C 25 Untreated 65______________________________________

Claims

1. An intermediate of the formula VI ##STR285## where X and Y are identical or different and each is hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may be condensed together to form a phenyl ring,

R.sup.1 is hydrogen, alkyl, alkenyl, alkynyl, cyclopropyl, cyclopropylmethyl, cyclobutyl, --CH.sub.2 --CN, --CH.sub.2 --O--CH.sub.3, --CO.sub.2 CH.sub.3 or --S--R.sup.5, wherein R.sup.5 is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl,

Z is O--(C.sub.1 -C.sub.4)-alkyl.

2. An intermediate of the formula XI ##STR286## where X and Y are identical or different and each is hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may together be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

R.sup.1 is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO.sub.2 -alkyl,

R.sup.2 is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, and

Hal is halogen.

3. An intermediate of the formula XII ##STR287## where X and Y are identical or different and each is hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may together be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

R.sup.1 is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO.sub.2 -alkyl, and

R.sup.2 is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl.

4. An intermediate of the formula XIII ##STR288## where X and Y are identical or different and each is hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may together be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

A is --O--, --S--, --CR.sup.2 .dbd.CR.sup.3 --, CHR.sup.2 --O--, --CHR.sup.2 --S--, --CHR.sup.2 --O--N.dbd.C(R.sup.4)--, --CR.sup.2 .dbd.N--O--, --O--N.dbd.C(R.sup.4)--, --C.tbd.C--, --CHR.sup.2 --CHR.sup.3 --, --CHR.sup.2 --O--CO--, --O--CHR.sup.2 -- or a single bond,

B is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl or hydrogen, and

R.sup.2 and R.sup.3 are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, and R.sup.4 is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy,

wherein B is not hydrogen when A is a single bond.

5. An intermediate of the formula XXXI ##STR289## where X and Y are identical or different and each is F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may together be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring, or Y is hydrogen,

R.sup.1 is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO.sub.2 -alkyl,

R.sup.2 is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, and

Hal is halogen.

6. An intermediate of the formula XXXII ##STR290## where X and Y are identical or different and each is F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may together be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring, or Y is hydrogen,

R.sup.1 is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO.sub.2 -alkyl, and

R.sup.2 is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl.

7. An intermediate of the formula XXXIII ##STR291## where X and Y are identical or different and each is F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may together be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring, or Y is hydrogen,

A is --O--, --S--, --CR.sup.2 .dbd.CR.sup.3 --, --CHR.sup.2 --O--, --CHR.sup.2 --S--, --CHR.sup.2 --O--N.dbd.C(R.sup.4)--, --CR.sup.2 .dbd.N--O--, --O--N.dbd.C(R.sup.4)--, --C.tbd.C--, --CHR.sup.2 --CHR.sup.3 --, --CHR.sup.2 --O--CO--, --O--CHR.sup.2 -- or a single bond,

B is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl or hydrogen, and

R.sup.2 and R.sup.3 are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, and R.sup.4 is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy.