Carbamates and crop protection agents containing them

Abstract

Carbamates of the formula I ##STR1## where the substituents have the following meanings: Z is methoxy, NH.sub.2, NHCH.sub.3, N(CH.sub.3).sub.2, CH.sub.3, C.sub.2 H.sub.5, CF.sub.3 or CCl.sub.3,X and Y are identical or different and each is hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may be condensed together to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,R.sup.1 may also be substituted or unsubstituted and is O-alkyl, O-alkenyl, O-alkynyl, O-cycloalkyl, O-cycloalkenyl or O--CO.sub.2 -alkyl,A is --O--, --S--, --CR.sup.2 .dbd.CR.sup.3 --, CHR.sup.2 --O--, --CHR.sup.2 --S--, --CHR.sup.2 --O--N.dbd.C(R.sup.4)--, --CR.sup.2 .dbd.N--O--, --O--N.dbd.C(R.sup.4)--, --C.tbd.C--, --CHR.sup.2 --CHR.sup.3 --, --CHR.sup.2 --O--CO--, --O--CHR.sup.2 -- or a single bond,B is substituted or unsubstituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl, hydrogen, substituted or unsubstituted alkylaryl, substituted or unsubstituted alkylhetaryl, substituted or unsubstituted alkylcycloalkyl, substituted or unsubstituted alkylcycloalkenyl,R.sup.2 and R.sup.3 are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl,R.sup.4 is hydrogen, CN, alkyl, alkenyl, alkynyl, alkoxy or cycloalkyl,R.sup.5 is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl and plant-tolerated acid and base adducts thereof, and fungicides containing them.

Description

DESCRIPTION

The present invention relates to carbamates and crop protection agents, in particular for controlling fungi, insects, nematodes and spider mites.

It is known that aniline derivatives, for example isopropyl N-phenylcarbamate or the corresponding 3-chlorophenyl ester (GB 574 995) or methyl N-3,4-dichloro-phenylcarbamate (BE 612 550) can be used as crop protection agents. However, their fungicidal action is unsatisfactory.

It has now been found, surprisingly, that carbamates of the formula I ##STR2## where the substituents have the following meanings: Z is methoxy, NH.sub.2, NHCH.sub.3, N(CH.sub.3).sub.2, CH.sub.3, C.sub.2 H.sub.5, CF.sub.3 or CCl.sub.3,

X and Y independently of one another are each hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form an unsubstituted or substituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring, R.sup.1 is unsubstituted or substituted alkyl, alkenyl, cyclopropyl, cyclopropylmethyl, cyclobutyl, --CH.sub.2 --CN, --CH.sub.2 OCH.sub.3, --CO.sub.2 CH.sub.3 or --S--R.sup.5, O-alkyl, O-alkenyl, O-alkynyl, O-cycloalkyl, O-cycloalkenyl or O--CO.sub.2 -alkyl, A is --O--, --S--, --CR.sup.2 .dbd.CR.sup.3 --, CHR.sup.2 --O, --CHR.sup.2 --S--, --CHR.sup.2 --O--N.dbd.C(R.sup.4)--, --CR.sup.2 .dbd.N--O--, --O--N.dbd.C(R.sup.4)--, --C.tbd.--C--, --CHR.sup.2 --CHR.sup.3 --, --CHR.sup.2 --O--CO--, --O--CHR.sup.2 -- or a single bond, B can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl, hydrogen, unsubstituted or substituted alkylaryl, unsubstituted or substituted alkylhetaryl, unsubstituted or substituted alkylcycloalkyl or unsubstituted or substituted alkylcycloalkenyl, R.sup.2 and R.sup.3 independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, R.sup.4 is hydrogen, CN, alkyl, alkenyl, alkynyl, alkoxy or cycloalkyl, R.sup.5 is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl, and their plant-tolerated acid addition products and base addition products have a good fungicidal, acaricidal, insecticidal and nematocidal action.

Acids for addition products are, for example, mineral acids, such as hydrochloric acid, hydrobromic acid, phosphoric acid, sulfuric acid or nitric acid, or carboxylic acids, such as formic acid, acetic acid, oxalic acid, malonic acid, lactic acid, malic acid, succinic acid, tartaric acid, citric acid, salicylic acid, p-toluenesulfonic acid or dodecylbenzenesulfonic acid, as well as proton-acidic compounds generally, for example saccharin.

Bases for base addition products are, for example, potassium hydroxide, sodium hydroxide, potassium carbonate, sodium carbonate and ammonium hydroxide.

The novel compounds of the formula I may be obtained in the preparation as mixtures of stereoisomers (E/Z isomers, diastereomers, enantiomers), which can be separated into the individual components in a conventional manner, for example by crystallization or chromatography. Both the individual isomers and mixtures thereof may be used as fungicides, acaricides, nematocides or insecticides, and form the subject of the present invention.

The abovementioned alkyl radicals may be substituted and are of 1 to 6 carbon atoms.

The abovementioned alkenyl and alkynyl radicals may be substituted and are of 2 to 6 carbon atoms.

The abovementioned cycloalkyl radicals are of 3 to 10 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R.sup.6.

The abovementioned aryl radicals are of 6, 10 or 14 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R.sup.6.

The abovementioned hetaryl radicals have 5 to 14 ring atoms, including from 1 to 4 hetero atoms selected from the group consisting of N, O and S, are unsaturated and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R.sup.6.

The above mentioned heterocyclyl radicals have 5 to 14 carbon atoms, including 1 to 4 hetero atoms selected from the group consisting of N, O and S, are saturated or partially unsaturated and are unsubstituted or substituted, for example by 1 to 4 identical or different substitutents R.sup.6.

The abovementioned cycloalkenyl radicals are of 5 to 14 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R.sup.6.

Two adjacent substituents R.sup.6, together with the carbon atoms of which they are substituents, may form a carbocyclic hydrogenated, partially unsaturated or aromatic ring having 3 to 14 carbon atoms or a heterocyclic hydrogenated, partially unsaturated or heteroaromatic ring having 3 to 14 carbon atoms, including 1 to 4 hetero atoms selected from the group consisting of N, O and S.

R.sup.6 may be unsubstituted or substituted, for example by 1 to 4 identical or different substituents R.sup.7, and R.sup.6 is, for example, hydrogen, halogen, cyano, nitro, haloalkyl, alkyl, haloalkoxy, alkenyl, alkynyl, cycloalkyl, aryl, hetaryl, heterocyclyl, cycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, aryloxy, hetaryloxy, heterocyclyloxy, cycloalkenyloxy, alkoximino, alkenyloximino, alkynyloximino, cycloalkoxyimino, cycloalkenyloximino, aryloximino, hetaryloximino, heterocyclyloximino, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkyloxycarbonyl, aryloxycarbonyl, hetaryloxycarbonyl, heterocyclyloxycarbonyl, cycloalkenyloxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkenylaminocarbonyl, dialkenylaminocarbonyl, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, arylthio, hetarylthio, heterocyclylthio, cycloalkenylthio, alkylamino, alkenylamino, alkynylamino, cycloalkylamino, arylamino, hetarylamino, heterocyclylamino, cycloalkenylamino, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, arylcarbonyl, hetarylcarbonyl, heterocyclylcarbonyl, cycloalkenylcarbonyl, alkylsulfoxyl, alkenylsulfoxyl, alkynylsulfoxyl, cycloalkylsulfoxyl, arylsulfoxyl, hetarylsulfoxyl, heterocyclylsulfoxyl, cycloalkenylsulfoxyl, alkylsuifonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, hetarylsulfonyl, heterocyclylsulfonyl, cycloalkenylsulfonyl, alkylsulfinyl, alkenylsulfinyl, alkynylsulfinyl, cycloalkylsulfinyl, arylsulfinyl, hetarylsulfinyl, heterocyclylsulfinyl or cycloalkenylsulfinyl.

R.sup.7 is is any substituent and is, for example, hydrogen, halogen, cyano, nitro, haloalkyl, alkyl, haloalkoxy, alkenyl, alkynyl, cycloalkyl, aryl, hetaryl, heterocyclyl, cycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, aryloxy, hetaryloxy, heterocyclyloxy, cycloalkenyloxy, alkoximino, alkenyloximino, alkynyloximino, cycloalkoximino, cycloalkenyloximino, aryloximino, hetaryloximino, heterocyclyloximino, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkyloxycarbonyl, aryloxycarbonyl, hetaryloxycarbonyl, heterocyclyloxycarbonyl, cycloalkenyloxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkenylaminocarbonyl, dialkenylaminocarbonyl, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, arylthio, hetarylthio, heterocyclylthio, cycloalkenylthio, alkylamino, alkenylamino, alkynylamino, cycloalkylamino, arylamino, hetarylamino, heterocyclylamino, cycloalkenylamino, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, arylcarbonyl, hetarylcarbonyl, heterocyclylcarbonyl, cycloalkenylcarbonyl, alkylsulfoxyl; alkenylsulfoxyl, alkynylsulfoxyl, cycloalkylsulfoxyl, arylsulfoxyl, hetarylsulfoxyl, heterocyclylsulfoxyl, cycloalkenylsulfoxyl, alkylsulfonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, hetarylsulfonyl, heterocyclylsulfonyl, cycloalkenylsulfonyl, alkylsulfinyl, alkenylsulfinyl, alkynylsulfinyl, cycloalkylsulfinyl, arylsulfinyl, hetarylsulfinyl, heterocyclylsulfinyl or cycloalkenylsulfinyl.

The abovementioned alkyl radicals may be substituted, are preferably of 1 to 6 carbon atoms and are, in particular, methyl, ethyl, propyl, such as n-propyl or isopropyl, butyl, such as n-butyl, isobutyl, tert-butyl or sec-butyl, pentyl or hexyl.

The abovementioned alkenyl radicals may be substituted, are preferably of 2 to 6 carbon atoms and are, in particular, ethenyl, propenyl, such as prop-1-enyl, prop-2-enyl or prop-1-en-2-yl, butenyl, such as but-1-enyl, but-2-enyl, but-3-enyl, but-1-en-3-yl, but-2-en-2-yl, but-1-en-2-yl, 2-methyl-1-propenyl or 2-methyl-2-propenyl, pentenyl or hexenyl.

The abovementioned alkynyl radicals may be substituted, are preferably of 2 to 6 carbon atoms and are, in particular, ethynyl, propynyl, such as prop-1-ynyl or prop-3-ynyl, butynyl, such as but-1-ynyl, but-2-ynyl, but-3-ynyl or 1-methylprop-2-ynyl, pentynyl or hexynyl.

The abovementioned halogens are fluorine, chlorine, bromine or iodine.

The abovementioned cycloalkyl radicals are preferably cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, cycloheptyl, cyclooctyl, cyclononyl, cyclodecyl, bornanyl, norbornanyl, dicyclohexyl, bicyclo�3.3.0!octyl, bicyclo�3.2.1!octyl, bicyclo�2.2.2!octyl or bicyclo�3.3.1!nonyl.

The abovementioned cycloalkenyl radicals are preferably cyclopropenyl, cyclobutenyl, cyclopentenyl, cyclohexenyl, cycloheptenyl, cyclooctenyl, cyclononenyl, cyclodecenyl, bornenyl, norbornenyl, bicyclo�3.3.0!octenyl, bicyclo�3.2.1!octenyl, bicyclo�2.2.2!octenyl or bicyclo�3.3.1!nonenyl.

The abovementioned haloalkyl radicals are preferably C.sub.1 -C.sub.4 -haloalkyl, in particular C.sub.1 - or C.sub.2 -haloalkyl, such as chloromethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluoromethyl, dichlorof luoromethyl, chlorodifluoromethyl, 1-fluoroethyl, 2-fluoroethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2-difluoroethyl, 2,2,2-dichloro-2-fluoroethyl, 2,2,2-trichloroethyl or pentafluoroethyl.

The abovementioned haloalkoxy radicals are preferably C.sub.1 -C.sub.4 -haloalkoxy, in particular C.sub.1 - or C.sub.2 -haloalkoxy, such as chloromethoxy, dichloromethoxy, trichloromethoxy, fluoromethoxy, difluoromethoxy, trifluoromethoxy, chlorofluoromethoxy, dichlorofluoromethoxy, chlorodifluoromethoxy, 1-fluoroethoxy, 2-fluoroethoxy, 2,2-difluoroethoxy, 2,2,2-trifluoroethoxy, 2-chloro-2-fluoroethoxy, 2-chloro-2,2-difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy or pentafluoroethoxy.

The abovementioned aryl radicals are preferably phenyl, 1-naphthyl, 2-naphtyl, 1-anthracenyl, 2-anthracenyl or 9-anthracenyl.

The abovementioned hetaryl radicals are preferably furyl, such as 2-furyl or 3-furyl, thienyl, such as 2-thienyl or 3-thienyl, pyrrolyl, such as 1-pyrrolyl, 2-pyrrolyl or 3-pyrrolyl, isoxazolyl, such as 3-isoxazolyl, 4-isoxazolyl or 5-isoxazolyl, isothiazolyl, such as 3-isothiazolyl, 4-isothiazolyl or 5-isothiazolyl, pyrazolyl, such as 1-pyrazolyl, 3-pyrazolyl, 4-pyrazolyl or 5-pyrazolyl, oxazolyl, such as 2-oxazolyl, 4-oxazolyl or 5-oxazolyl, thiazolyl, such as 2-thiazolyl, 4-thiazolyl or 5-thiazolyl, imidazolyl, such as 1-imidazolyl, 2-imidazolyl, 4-imidazolyl or 5-imidazolyl, 1,2,3-thiadiazolyl, 1,2,4-thiadiazolyl, 1,2,5-thiadiazolyl, 1,3,4-thiadiazolyl, tetrazolyl, 1,2,3,4-thiatriazolyl, 1,2,3,4-oxatriazolyl, pyridyl, such as 2-pyridyl or 4-pyridyl, pyridazinyl, such as 3-pyridazinyl or 4-pyridazinyl, pyrimidinyl, such as 2-pyrimidinyl, 4-pyrimidinyl or 5-pyrimidinyl, pyrazinyl, such as 2-pyrazinyl or 3-pyrazinyl, 1,2,4-triazinyl, 1,3,5-triazinyl or 1,2,4,5-tetrazinyl.

Adjacent substituents of the hetero atoms may be condensed to form an aromatic or heteroaromatic ring, so that hetaryl also comprises fused ring systems, eg. benzofuranyl, isobenzofuranyl, 1-benzothienyl, 2-benzothienyl, indolyl, isoindolyl, benzisoxazolyl, benzoxazolyl, benzisothiazolyl, benzothiazolyl, such as 2-benzothiazolyl, 4-benzothiazolyl, 5-benzothiazolyl, 6-benzothiazolyl or 7-benzothiazolyl, indazolyl, benzimidazolyl, benzofurazanyl, dibenzofuranyl, dibenzothienyl, acridinyl, phenanthridinyl, carbazolyl, quinolyl, isoquinolyl, phthalazinyl, quinazolinyl, quinoxalinyl, cinnolinyl, 1,5-naphthyridinyl, 1,6-naphthyridinyl, 1,7-naphthyridinyl, 1,8-naphthyridinyl, pteridinyl, pyrrolopyridinyl, pyrrolopyridazinyl, pyrrolopyrimidinyl, pyrrolopyrazinyl, pyrrolotriazinyl, furopyridyl, furopyridazinyl, furopyrimidinyl, furopyrazinyl, furotriazinyl, thienopyridyl, thienopyridazinyl, thienopyrimidinyl, thienopyrazinyl, thienotriazinyl, imidazopyridazinyl, imidazopyrimidinyl, imidazopyrazinyl, pyrazolopyridyl, pyrazolopyridazinyl, pyrazolopyrimidinyl, pyrazopyrazinyl, isoxazolopyrazinyl, oxazolopyridyl, oxazolopyridazinyl, oxazolopyrimidinyl, oxazolopyrazinyl, thiazolopyridyl, thiazolopyridazinyl, isothiazolopyrazinyl, triazolopyridyl, triazolopyridazinyl, triazolopyrimidinyl or triazolopyrazinyl.

The abovementioned heterocycyl radicals are preferably 2-tetrahydrofuranyl, oxiranyl, 3-tetrahydrofuranyl, 2-tetrahydrothienyl, 3-tetrahydrothienyl, 2-pyrrolidinyl, 3-pyrrolidinyl, 3-isoxazolidinyl, 4-isoxazolidinyl, 5-isoxazolidinyl, 3-isothiazolidinyl, 4-isothiazolidinyl, 5-isothiazolidinyl, 3-pyrazolidinyl, 4-pyrazolidinyl, 5-pyrazolidinyl, 2-oxazolidinyl, 4-oxazolidinyl, 5-oxazolidinyl, 2-thiazolidinyl, 4-thiazolidinyl, 5-thiazolidinyl, 2-imidazolidinyl, 4-imidazolidinyl, 1,2,4-oxadiazolidin-3-yl, 1,2,4-oxadiazolidin-5-yl, 1,2,4-thiadiazolidin-3-yl, 1,2,4-thiadiazolidin-5-yl, 1,2,5-triazolidin-3-yl, 1,3,4-oxadiazolidin-2-yl, 1,3,4-thiadiazolidin-2-yl, 1,3,4-triazolidin-2-yl, 2,3-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,5-dihydrofur-2-yl, 2,5-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,3-dihydrothieno-2-yl, 2,3-dihydrothien-3-yl, 2,5-dihydrothien-2-yl, 2,4-pyrrolin-2-yl, 2,3-pyrrolin-3-yl, 2,5-pyrrolin-2-yl, 2,5-pyrrolin-3-yl, 2,3-isoxazolidin-3-yl, 3,4-isoxazolin-3-yl, 4,5-isoxazolin-2-yl, 2,3-isoxazolin-4-yl, 3,4-isoxazolin-3-yl, 4,5-isoxazolin-4-yl, 2,3-isoxazolin-5-yl, 3,4-isoxazolin-5-yl, 4,5-isoxazolin-5-yl, 2,3-isothiazolin-3-yl, 3,4-isothiazolin-3-yl, 4,5-isothiazolin-3-yl, 2,3-isothiazolin-4-yl, 3,4-isothiazolin-4-yl, 4,5-isothiazolin-4-yl, 2,3-isothiazolin-5-yl, 3,4-isothiazolin-5-yl, 4,5-isothiazolin-5-yl, 2,3-dihydropyrazol-1-yl, 2,3-dihydro-pyrazol-2-yl, 2,3-dihydropyrazol-3-yl, 2,3-dihydropyrazol-4-yl, 2,3-dihydropyrazol-5-yl, 3,4-dihydropyrazol-1-yl, 3,4-dihydropyrazol-2-yl, 3,4-dihydropyrazol-4-yl, 3,4-dihydropyrazol-5-yl, 4,5-dihydropyrazol-1-yl, 4,5-dihydropyrazol-3-yl, 4,5-dihydropyrazol-4-yl, 4,5-dihydropyrazol-5-yl, 3,4-dihydrooxazol-2-yl, 2,3-dihydrooxazol-3-yl, 2,3-dihydrooxazol-4-yl, 2,3-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 3,4-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 2-piperidinyl, 3-piperidinyl, 4-piperidinyl, 3-tetrahydropyridazinyl, 4-tetrahydropyridazinyl, 2-tetrahydropyrimidinyl, 4-tetrahydropyrimidinyl, 5-tetrahydropyrimidinyl, 2-tetrahydropyrazinyl, 1,3,5-tetrahydrotriazin-2-yl, 1,2,4-tetrahydrotriazin-3-yl, 1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, oxazol-2-in-2-yl, 2-tetrahydropyranyl, 1,3-dioxolan-2-yl, thiazol-2-in-2-yl, 3,4,5,6-tetrahydropyridin-2-yl, 4H-1,3-thiazin-2-yl, 4H-3,1-benzothiazin-2-yl, 1,1-dioxo-2,3,4,5-tetrahydrothien-2-yl, 2H-1,4-benzothiazin-3-yl, 2H-1,4-benzoxazin-3-yl, 1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, N-morpholinyl or dihydroquinazolinyl.

The invention furthermore relates to carbamates of the formula I ##STR3## where the substituents have the following meanings: Z is methoxy, NH.sub.2, NHCH.sub.3 or CH.sub.3,

X and Y independently of one another are each hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form a phenyl ring, R.sup.1 is hydrogen, alkyl, alkenyl alkynyl cyclopropyl, cyclopropylmethyl, cyclobutyl, --CH.sub.2 --CN, --CH.sub.2 --O--CH.sub.3, --CO.sub.2 CH.sub.3 or --S--R.sup.5, A is --O--, --CR.sup.2 .dbd.CR.sup.3 --, --C.tbd.C--, --CHR.sup.2 --O--, --CHR.sup.2 --S--, --CHR.sup.2 --O--N.dbd.C(R.sup.4)--, --CR.sup.2 .dbd.N--O-- or --O--N.dbd.C(R.sup.4)--, a) B is substituted phenyl when A is --CR.sup.2 .tbd.--CR.sup.3 --, --C.dbd.C--, --CHR.sup.2 --O--, --CHR.sup.2 --S--, --CHR.sup.2 --O--N.dbd.C(R.sup.4)--, --CR.sup.2 .dbd.N--O-- or --O--N.dbd.C(R.sup.4), b) or B is unsubstituted or substituted cyclolalkyl, unsubstituted or substituted cycloalkenyl, unsubstituted or substituted heterocyclyl, unsubstituted or substituted hetaryl, unsubstituted or substituted naphthyl, unsubstituted or substituted arylalkyl, unsubstituted or substituted hetarylalkyl, unsubstituted or substituted cycloalkylalkyl, unsubstituted or substituted cycloalkenylalkyl or unsubstituted or substituted anthracenyl, R.sup.2 and R.sup.3 independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, R.sup.4 is CN, alkyl, alkenyl, alkynyl or cycloalkyl and R.sup.5 is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl, and their plant-tolerated acid addition products and base addition products.

The invention furthermore relates to carbamates of the formula II ##STR4## where X, Y, R.sup.1 and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula III ##STR5## where X, Y, R.sup.1 and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula I as claimed in claim 2, where A is --CH.dbd.CH-- and X, Y, R.sup.1 and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula VII ##STR6## where the substituents have the following meanings: X and Y independently of one another are each hydrogen, F, Cl, Br, CF.sub.3, CN, NO.sub.2, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form an unsubstituted or substituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

R.sup.1 can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO.sub.2 -alkyl, A is --O--, --S--, --CR.sup.2 .dbd.CR.sup.3 --, CHR.sup.2 --O--, --CHR.sup.2 --S--, --CHR.sup.2 --O--N.dbd.C(R.sup.4)--, --CR.sup.2 .dbd.N--O--, --O--N.dbd.C(R.sup.4)--, --C--.tbd.C--, --CHR.sup.2 --CHR.sup.3 --, --CER.sup.2 --O--CO--, --O--CHR.sup.2 -- or a single bond, B can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl or hydrogen, R.sup.2 and R.sup.3 independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl and R.sup.4 is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy, and their plant-tolerated acid addition products and base addition products.

The invention furthermore relates to carbamates of the formula VIII ##STR7## where A, B and R.sup.1 have the meanings stated in claim 9.

The invention furthermore relates to carbamates of the formula IX ##STR8## where R.sup.1 and B have the meanings stated in claim 1.

The invention furthermore relates to carbamates of the formula X ##STR9## where R.sup.1 and B have the meanings stated in claim 1.

The novel compounds can be prepared, for example, by the following processes:

The nitrobenzenes 1 obtainable by standard processes are reduced to the anilines 2, for example with hydrogen or hydrogen transfer agents, such as ammonium formate, in the presence of suitable catalysts, such as Pd, Pt or Ni, with complex reducing agents, eg. Collman's reagent (Na.sub.2 Fe(CO).sub.4) or by other methods known from the literature (J. March, Advanced Organic Chemistry, 3rd Edition, 1985, page 1103 et seq.). The anilines 2 are reacted under alkaline conditions with methyl chloroformate to give the carbamates 3. The reaction of the carbamates 3 under alkaline conditions with the corresponding alkylating agents, acylating agents or R.sup.5 --S--S(.dbd.O).sub.2 --R.sup.5 gives the derivatives 4 (Scheme 1). ##STR10##

The nitrobenzenes 5 can be converted into the carbamates 6 similarly to Scheme 1. The halogen derivatives 7 (Z=Cl or Br) are obtainable by acidic cleavage 5 of the methyl ether of 6 (Scheme 2). ##STR11##

Alternatively, the halogen derivatives 7 (Z=Cl or Br) are obtainable from the derivatives 9 by free radical halogenation. The carbamates 9 are in turn prepared from the corresponding starting materials 8, similarly to Scheme 1 (Scheme 3). ##STR12##

The halogen derivatives 7 (Z=Cl or Br) can be converted into the active ingredients 10 under alkaline conditions. Alternatively, the compounds 7 are converted into the phosphorus compounds 11a and 11b by reaction with P(C.sub.6 H.sub.5).sub.3 or P(O-Alkyl).sub.3, or into the carbonyl compounds 12 by oxidation (for example with N-methylmorpholine N-oxide) (Scheme 4). ##STR13##

The corresponding stilbenes 13 are obtainable from the phosphonium salts 11a or phosphonates 11b or carbonyl compounds 12 by a Wittig reaction (Scheme 5). ##STR14##

Partial reduction of the nitroaromatics 21 (for example with zinc (similarly to Bamberger et al., Ann. Chem. 316 (1901), 278) or with hydrogen in the presence of suitable catalysts such as platinum (similarly to European Patent 85,890)) gives the hydroxylamines 22, which can be reacted under alkaline conditions with an acylating agent (eg. propionyl chloride) or a carbamoylating agent (eg. methyl isocyanate) to give the compound 23 and then with an electrophile, for example with an alkylating agent, to give the active ingredients 24 (scheme 11). ##STR15##

In addition, the hydroxylamine 25 can be acylated or aminoacylated (for example with methyl isocyanate) (similarly to Bamberger et al., Ann. Chem. 316 (1901), 278; European Patent 85,890) to give the compound 26, which can then be alkylated or alkoxyacylated (for example with chloroformates) to give the hydroxylamine derivative 27. The free radical halogenation of 27, for example with N-bromosuccinamide, bromine, chlorine or So.sub.2 Cl.sub.2 in the presence of free radical initiator, eg. azobisisobutyronitrile, or with exposure to UV light, then gives the halide 28 (Hal=Cl or Br; Scheme 12). ##STR16##

The halides 28 can then be converted into the compounds 29 with the corresponding nucelphiles (Scheme 13). ##STR17##

In addition, the halides 28 can be converted by free radical reaction to the dihalide 30 and then converted with H.sub.2 O/MeOH in the presence of AgNO.sub.3 into the carbonyl compound 31 or reacted directly with N-methylmorpholine N-oxide to give the carbonyl compound 11. Furthermore, the phosphonates, phosphonium salts or phosphine oxides 32 (P is the particular organophosphorus radical) are obtainable from the halides 8 (Scheme 14). ##STR18##

The carbonyl compounds 31 can then be reacted with the corresponding hydroxylamines to give the oximes 33 or can be subjected to a Wittig reaction to give the olefins 34, The olefins 34 are also obtainable by a Wittig reaction starting from the phosphonates, phosphonium salts or phosphine oxides 32 (Scheme 15). ##STR19##

The saturated compounds 35 can be prepared from the olefins 34 by reduction or, where R.sup.2 and R.sup.3 are each H, the acetylenes 36 can be prepared from said olef ins by halogen addition (Hal=Cl, Br or I) and subsequent two-fold elimination of hydrogen halide (Scheme 16). ##STR20##

Alternatively, the ureas 39 can be synthesized by acylation of the hydroxylamines 22 to the compounds 37, subsequent alkylation or acylation to the compounds 38 and substitution of the nucleofugic leaving group V (V is, for example, OCH.sub.3, OCCl.sub.3, CCl.sub.3, O-phenyl or O-p-nitrophenyl) by NH.sub.3, H.sub.2 N--CH.sub.3 or HN(CH.sub.3).sub.2 (Scheme 17). ##STR21##

Alternatively, ureas of the formula 39 can also be obtained by alkylating ureas of the formula 41, which in turn are obtainable from 17 by reacting 17 with the corresponding amines, or directly from 22 by aminocarbonylation (for example with dimethylcarbamoyl chloride or methyl isocyanate) (cf. for example Houben-Weyl, volume E16a, page 208).

Furthermore, ureas of the formula 39 can also be obtained from the N-aryl-O-alkylhydroxylamines of the formula 42 in a similar manner by aminocarbonylation.

The compounds of the formula 42 are in turn obtainable by methods known from the literature, from hydroxylamines of the formula 2 (cf. for example Houben-Weyl, volume E16a, pages 271 and 282-289).

In addition, the hydroxylamines 22 are obtainable from the anilines 43 by formation of the imines 44, oxidation of the compounds 44 with the m-chloroperbenzoic acid and reaction of the oxaziridines 45 with hydroxylamine (Scheme 18; similarly to G. Grundke et al., Synthesis 1987, 1115). ##STR22##

The Examples which follow illustrate the preparation of the novel compounds.

EXAMPLES

Example 1

Methyl N-ethyl-N-(2-(2'-methylphenoxymethyl)-phenyl)-carbamate (Table 7, No. 2)

a) Methyl N-(o-methylphenyl)-carbamate 50 g (0.53 mol) of methyl chloroformate are added dropwise to 53 g (0.5 mol) of o-toluidene in 500 ml of methylene chloride. During this procedure, the reaction solution heats up to the boiling point and a colorless solid is precipitated.

Stirring is carried out for one hour, after which 200 ml of 10% strength sodium hydroxide solution are added dropwise, the colorless solid going into solution. The organic phase is dried over MgSO.sub.4 and evaporated down under reduced pressure. The remaining solid is stirred with n-hexane and filtered off under suction. 84 g (0.5 mol, quantitative yield) of the title compound are obtained as a colorless solid.

mp.=61.degree.-62.degree. C.; .sup.1 H-NMR (DMSO-d.sub.6 ; .delta. (PPm)): 8.85 (s, 1H, NH); 7.35 (d, broad, 1H, aromatic); 7.1 (m, 3H, aromatic); 3.6 (s, 3H, OCH.sub.3); 2.2 (s, 3H, CH.sub.3)

b) Methyl N-ethyl-N-(o-methylphenyl)-carbamate

5.1 g (0.2 mol) of sodium hydride are added a little at a time to 30 g (0.18 mol) of methyl N-(o-methylphenyl)-carbamate (Example 1a) in 200 ml of dimethylformamide. After the evolution of gas has ceased, 30 g (0.2 mol) of ethyl iodide are added drop-wise, the reaction mixture being lightly cooled in a water bath. A white solid is precipitated. After about 4 hours, the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The organic phase is dried over MgSO.sub.4 and evaporated down. The residue is distilled. 32.5 g (0.17 mol=93%) of the title compound are obtained as a colorless oil. bp..sup.0.5 =74.degree. C.; .sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm): 7.2 (m, 3H, aromatic); 7.1 (m, 1H, aromatic); 3.8 (m, 1H, N--CH.sub.A); 3.6 (s, 3H, OCH.sub.3); 3.5 (m, 1H, N--CH.sub.B); 2.2 (s, 3H, CH.sub.3); 1.1 (t, 3H, CH.sub.3)

c) Methyl N-ethyl-N-(o-bromomethylphenyl)-carbamate

A mixture of 30 g (0.155 mol) of methyl N-ethyl-N-(o-methylphenyl)-carbamate (Example 1b), 33 g (0.185 mol) of N-bromosuccinimide and 0.1 g of azoisobutyronitrile in 300 ml of carbon tetrachloride is exposed to a 300 W UV lamp for 6 hours. During this procedure, the contents of the flask heat up to about 70.degree. C. Thereafter, the reaction mixture is washed four times with water, dried and evaporated down. The residue obtained comprises 41 g of a brown oil which contains the title compound in about 50% purity and is used without further purification in the next reaction.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.2 (m, 4H, aromatic); 4.45 (s, 2H, CH.sub.2 --Br); 3.8 (m, 1H, N--CH.sub.A); 3.6 (s, 3H, OCH.sub.3); 3.5 (m, 1H, N--CH.sub.B); 1.15 (t, 3H, J=8 Hz, CH.sub.3)

d) Methyl N-ethyl-N-(2-(2'-methylphenoxymethyl)-phenyl)-carbamate (Table 7, No. 2)

2.4 g (17 mmol) of sodium hydride are added a little at a time to 8.6 g (80 mmol) of o-cresol in 100 ml of dimethylformamide. Stirring is carried out for 30 minutes at room temperature (20.degree. C.), after which 20.5 g of methylN-ethyl-N-(o-bromomethylphenyl)-carbamate (Example 1c, about 50% purity, about 37 mmol) are added. Stirring is carried out overnight at room temperature, after which the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The combined ether phases are dried over MgSO.sub.4 and evaporated down. The residue is distilled in a kugelrohr (bulb tube) apparatus. 10 g of a yellow oil are obtained at 220.degree. C. and 0.2 mbar, and the oil is then purified by chromatography with cyclohexane/ethyl acetate mixtures over silica gel and then over alumina. The product thus obtained is purified again by kugelrohr distillation. 3.6 g (12 mmol=32%) of the title compound are obtained as a colorless oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.6 (m, 1H, aromatic); 7.35 (m, 2H, aromatic); 7.15 (m, 3H, aromatic); 6.85 (m, 2H, aromatic); 5.0 (dd, broad, 2H, O--CH.sub.2); 3.8 (m, 1H, N--CH.sub.A); 3.6 (s, 3H, O--CH.sub.3); 3.5 (m, 1H, N--CH.sub.B); 2.3 (s, 3H, CH.sub.3); 1.15 (t, 3H, J=8 Hz, CH.sub.3)

Example 2

Methyl N-�2-(2'-methylphenoxymethyl)-phenyl!-N-methyl-thiocarbamate (Table 7, No. 89)

a) 2-(2'-Methylphenoxymethyl)-nitrobenzene

75 g (0.347 mol) of 2-nitrobenzyl bromide, 37 g (0.342 mol) of o-cresol and 56 g (0.405 mol) of potassium carbonate in 500 ml of dimethylformamide are stirred for 5 hours at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with ether. The ether phase is dried and evaporated down. The crystalline residue is stirred with methanol and filtered off under suction. 73 g (0.300 mol=88%) of the title compound are obtained as a colorless solid.

mp.=83.degree. C.; .sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 8.15 (d, 1H, J=8 Hz, aromatic); 7.95 (d, 1H, J=8 Hz, aromatic); 7.7 (t, 1H, J=8 Hz, aromatic); 7.45 (t, 1H, J=8 Hz, aromatic); 7.15 (m, 2H, aromatic); 6.9 (m, 2H, aromatic); 5.45 (s, 2H, O--CH.sub.2); 2.35 (s, 3H, CH.sub.3)

b) 2-(2'-Methylphenoxymethyl)-aniline

75 g (0.308 mol) of 2-(2'-methylphenoxymethyl)-nitrobenzene (Example 2a) and 10 g of 5% strength Pt/C (platinum adsorbed onto active carbon) in 50 ml of methanol are stirred vigorously for two hours under an H.sub.2 atmosphere. Thereafter, a further 2 g of 5% strength Pt/C are added and stirring is continued overnight. The catalyst is then filtered off under suction and is replaced with 10 g of fresh catalyst. Stirring is continued overnight, the mixture is filtered under suction and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography using hexane/ethyl acetate mixtures. 61 g (0.286 mol=93%) of the title compound are obtained as a colorless solid.

mp.=56.degree. C.; .sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.2 (m, 4H, aromatic); 6.95 (d, 1H, J=8 Hz, aromatic); 6.9 (t, 1H, J=6 Hz, aromatic); 6.7 (m, 2H, aromatic); 5.0 (s, 2H, O--CH.sub.2); 4.05 (s, broad, 2H, NH.sub.2); 2.2 (s, 3H, CH.sub.3)

c) Methyl N-�2-(2'-methylphenoxymethyl)-phenyl!-carbamate (Table 7, No. 3)

6 g (63 mmol) of methyl chloroformate are added dropwise to 10 g (47 mmol) of 2-(2'-methylphenoxymethyl)-aniline in 500 of methylene chloride at 20.degree.-30.degree. C. Stirring is carried out for 3 hours at room temperature, a white solid being precipitated, and the reaction mixture is then stirred with 20 ml of 10% strength sodium hydroxide solution. The organic phase is filtered off under suction over silica gel, the filtrate is evaporated down and the remaining residue is stirred thoroughly with methanol and filtered under suction. 10.5 g (39 mmol=82%) of the title compound are obtained as a colorless solid.

mp.=111.degree. C.; .sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 8.0 (d, broad, 1H, aromatic); 7.7 (s, broad, 1H, aromatic); 7.7 (s, broad, 1H, NH); 6.8-7.5 (m, 6H, aromatic); 5.0 (s, 2H, O--CH.sub.2); 3.75 (s, 3H, O--CH.sub.3); 2.25 (s, 3H, CH.sub.3)

d) Methyl N-�2-(2'-methylphenoxymethyl)-phenyl!-N-methylthiocarbamate (Table 7, No. 89)

0.5 g (20.8 mmol) of sodium hydride is added a little at a time to 4.9 g (17.3 mmol) of methyl N-�2-(2'-methylphenoxymethyl)!-phenylcarbamate (Example 2c) in 80 ml of toluene. After the end of gas evolution, 2.4 g (19 mmol) of methyl methanethiosulfonate are added and stirring is carried out overnight at room temperature. Thereafter, the reaction mixture is extracted with water, dried over MgSO.sub.4 and evaporated down under reduced pressure. The residue is purified by column chromatography with hexane/ethyl acetate mixtures over silica gel. 3 g (9.1 mmol=53%) of the title compound are obtained as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.65 (d, broad, 1H, aromatic); 7.35 (m, 2H, aromatic); 7.15 (m, 3H, aromatic); 6.85 (m, 2H, aromatic); 5.0 (m, 2H, O--CH.sub.2); 3.75 (s, 3H, O--CH.sub.3); 2.55 (s, 3H, S--CH.sub.3); 2.3 (s, 3H, CH.sub.3)

Example 3

Methyl N-allyl-N-�2-(3"-bromophenylmethyliminoxymethyl)-phenyl!-carbamate (Table 7, No. 91)

a) o-Methoxymethylnitrobenzene

125 g of 30% strength sodium methylate solution (0.69 mol) in methanol are added dropwise to 130 g (0.6 mol) of o-nitrobenzyl bromide in 200 ml of methanol. During this procedure, the reaction mixture heats up to about 50.degree. C. Stirring is continued for a further 3 hours, the reaction mixture being cooled to room temperature, after which ice water is added to the reaction vessel and the reaction mixture is neutralized by adding dilute hydrochloric acid. The aqueous phase is extracted with three times with ether, and the organic phase is dried over MgSO.sub.4 and evaporated down. 101 g (0.6 mol, quantitative yield) of the title compound are obtained as a residue in the form of a brownish oil. .sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 8.1 (d, broad, 1H, aromatic); 7.8 (d, broad, 1H, aromatic); 7.5 (t, broad, 1H, aromatic); 7.45 (t, broad, 1H, aromatic); 4.85 (s, 2H, O--CH.sub.2); 3.5 (s, 3H, OCH.sub.3)

b) Methyl N-(2-methoxymethylphenyl)-carbamate

528 g of 21.8% strength Na.sub.2 �Fe(CO).sub.4 ! solution (0.6 mol; 1 kg of the solution contains 633 g of water, 218 g of Na.sub.2 �Fe(CO).sub.4 !, 108 g of Na.sub.2 CO.sub.3 and 41 g of NaOH) are added dropwise to 101 g (0.6 mol) of o-methoxymethylnitrobenzene (Example 3a) in 1 l of methanol at 20.degree.-30.degree. C. Stirring is carried out for 1 hour at room temperature, after which the reaction mixture is diluted with ether. A brown oil separates out in the reaction vessel. The total reaction mixture is poured onto a silica gel column and is eluted with ether. Thereafter, the ether phase is evaporated, the residue is taken up in methylene chloride and the solution is dried over MgSO.sub.4. It is filtered under suction over silica gel and the solvent is then evaporated off under reduced pressure. The residue is purified by column chromatography with hexane and methylene chloride. 83.8 g of o-methoxymethylaniline are obtained as a brown oil, which is directly reacted further.

The resulting crude product is dissolved in 700 ml of methylene chloride, 62.4 g (0.66 mol) of methyl chloroformate are added and 52.2 g (0.66 mol) of pyridine are then added dropwise. Stirring is carried out overnight at room temperature and the reaction mixture is then extracted with dilute hydrochloric acid and water. The organic phase is dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with hexane/ethyl acetate mixtures. 89.4 g (0.41 mol=69%, based on 2-methoxymethylnitrobenzene) of the title compound are obtained as a yellow oil in a purity of about 90%.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 8.0 (m, 2H, 1.times. aromatic, NH); 7.35 (t, broad, 1H, aromatic); 7.15 (d, broad, 1H, aromatic); 7.0 (t, broad, 1H, aromatic); 4.5 (s, 2H, OCH.sub.2); 3.8 (s, broad, 3H, OCH.sub.3); 3.4 (s, broad, 3H, OCH.sub.3)

c) Methyl N-(2-bromomethylphenyl)-carbamate

38.6 g (150 mmol) of boron tribromide are added dropwise to 10 g (51 mmol) of methyl N-(2-methoxymethylphenyl)-carbamate (Example 2b) in 100 ml of methylene chloride. Stirring is carried out for 2 hours, after which the vigorously stirred reaction mixture is added dropwise to a solution of 11.8 g (0.17 mol) of NaHCO.sub.3 in water. The organic phase is separated off and the aqueous phase is extracted once with methylene chloride and once with ethyl acetate. The combined organic phases are dried over MgSO.sub.4 and evaporated down. 9.5 g (39 mmol=76%) of the title compound are obtained as a colorless solid.

mp.=132.degree. C.; .sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.85 (d, broad, 1H, aromatic); 7.3 (m, 2H, aromatic); 7.1 (t, broad, 1H, aromatic); 6.9 (s, broad, 1H, NH); 4.5 (s, 2H, CH.sub.2 --Br); 3.8 (s, 3H, OCH.sub.3)

d) Methyl N-�2-(3"-bromophenylmethyliminoxymethyl)-phenyl!-carbamate (Table 7, No. 88)

0.95 g (39 mmol) of sodium hydride is added a little at a time to 7 g (33 mmol) of m-bromoacetophenone oxime in 100 ml of dimethylformamide. When the evolution of gas has ended, 8 g (33 mmol) of methyl N-(2-bromomethylphenyl)-carbamate (Example 3c), dissolved in 10 ml of dimethylformamide, are added dropwise. Stirring is carried out for 3 hours at room temperature, the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The organic phase is washed three times with water, dried and evaporated down. The residue crystallizes and is stirred thoroughly with methanol. 5.1 g (13.5 mmol=41%) of the title compound are obtained as a colorless solid.

mp.=124.degree.-125.degree. C.; .sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 8.6 (s, broad, 1H, NH); 7.8-8.1 (m, 2H, aromatic); 7-7.6 (m, 6H, aromatic); 5.2 (s, 2H, O--CH.sub.2); 3.8 (s, 3H, O--CH.sub.3); 2.2 (s, 3H, CH.sub.3)

e) Methyl N-allyl-N-�2-(3"-bromophenylmethyliminoxy-methyl)-phenyl!-carbamate (Table 7, No. 91)

0.1 g (4.1 mmol) of sodium hydride is added a little at a time to 1.3 g (3.5 mmol) of methyl N-�2-(3"-bromophenylmethyliminoxymethyl)-phenyl!-carbamate (Example 3d) in 20 ml of dimethylformamide. After gas evolution has ended, 0.5 g (3.8 mmol) of allyl bromide are added and stirring is carried out overnight at room temperature. Thereafter, the reaction mixture is diluted with water and extracted three times with ether. The combined ether phases are washed three times with water, dried over MgSO.sub.4 and evaporated down. 1.5 g (quantitative yield) of the title compound are obtained as a residue in the form of a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.8 (s, broad, 1H, aromatic); 7.1-7.6 (m, 7H, aromatic); 6.0 (m, 1H, C--CH.dbd.C); 5.1 (m, 4H, O--CH2 and C.dbd.CH2); 4.4 (m, 1H, N--CH.sub.A); 4.0 (m, 1H, N--CH.sub.B) 3.6-3.8 (2s, broad, O--CH.sub.3); 2.2 (S, 3H, CH.sub.3)

The compounds described in the Tables below can be prepared in a similar manner.

TABLE 1______________________________________ ##STR23##I: R.sup.1 = HII: R.sup.1 = CH.sub.3III: R.sup.1 = AllylIV: R.sup.1 = PropargylV: R.sup.1 = SCH.sub.3VI: R.sup.1 = CH.sub.2 CNVII: R.sup.1 = CH.sub.2 OCH.sub.3VIII: R.sup.1 = COOCH.sub.3No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-C-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2, 5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3) 9644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CN-C-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-C-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 2______________________________________ ##STR24##I: R.sup.1 = HII: R.sup.1 = CH.sub.3III: R.sup.1 = AllylIV: R.sup.1 = PropargylV: R.sup.1 = SCH.sub.3VI: R.sup.1 = CH.sub.2 CNVII: R.sup.1 = CH.sub.2 CCH.sub.3VIII: R.sup.1 = COOCH.sub.3No. B______________________________________ 1 Pyrrolyl-3 2 NCH.sub.3 -Pyrrolyl-3 3 NC.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 NCH.sub.3 -Pyrrolyl-2 21 NC.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CNC.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CNC.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CNC.sub.6 H.sub.4)-Furyl-2 52 5-(4'-ClC.sub.6 H.sub.4)-Furyl-2 53 5-(3'-ClC.sub.6 H.sub.4)-Furyl-2 54 5-(2'-ClC.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CNC.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CNC.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CNC.sub.6 H.sub.4)-Furyl-2 69 4-(4'-ClC.sub.6 H.sub.4)-Furyl-2 70 4-(3'-ClC.sub.6 H.sub.4)-Furyl-2 71 4-(2'-ClC.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3i23 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3i24 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5 (2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 3-CH.sub.3 -Oxazolyl-4234 3-C.sub.6 H.sub.5 -Oxazolyl-4235 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 3-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 3-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 3-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 3-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 3-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 3-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4 66 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 -NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 S-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 S-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-cxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazollyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 1-Naphthyl385 2-Naphthyl______________________________________ TABLE 3______________________________________ ##STR25##I: R.sup.1 = HII: R.sup.1 = CH.sub.3III: R.sup.1 = AllylIV: R.sup.1 = PropargylV: R.sup.1 = SCH.sub.3VI: R.sup.1 = CH.sub.2 CNVII: R.sup.1 = CH.sub.2 OCH.sub.3VIII: R.sup.1 = COOCH.sub.3No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 C(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NCC.sub.2 H.sub.5)CH.sub.3324 3-C(NCC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NC-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NC-CH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3)2-4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3)2-4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3)2-4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAl1yl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-C-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-C-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazo1yl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3) 1644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-C-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-C-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 4______________________________________ ##STR26##I: R.sup.1 = HII: R.sup.1 = CH.sub.3III: R.sup.1 = AllylIV: R.sup.1 = PropargylV: R.sup.1 = SCH.sub.3VI: R.sup.1 = CH.sub.2 CNVII: R.sup.1 = CH.sub.2 OCH.sub.3VIII: R.sup.1 = COOCH.sub.3No. B______________________________________ 1 Pyrrolyl-3 2 N-CH.sub.3 -Pyrrolyl-3 3 N-C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N-CH.sub.3 -Pyrrolyl-2 21 N-C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CNC.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CNC.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CNC.sub.6 H.sub.4)-Furyl-2 52 5-(4'-ClC.sub.6 H.sub.4)-Furyl-2 53 5-(3'-ClC.sub.6 H.sub.4)-Furyl-2 54 5-(2'-ClC.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CNC.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CNC.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CNC.sub.6 H.sub.4)-Furyl-2 69 4-(4'-ClC.sub.6 H.sub.4)-Furyl-2 70 4-(3'-ClC.sub.6 H.sub.4)-Furyl-2 71 4-(2'-ClC.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thieny1-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-PyrazOlyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyraz6lyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 -N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isbthiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-Cl-C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-3365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-3366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-3367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 1-Naphthyl385 2-Naphthyl______________________________________ TABLE 5______________________________________ ##STR27##I: R.sup.1 = HII: R.sup.1 = CH.sub.3III: R.sup.1 = AllylIV: R.sup.1 = PropargylV: R.sup.1 = SCH.sub.3VI: R.sup.1 = CH.sub.2 CNVII: R.sup.1 = CH.sub.2 OCH.sub.3VIII: R.sup.1 = COOCH.sub.3No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 5-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 C(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)OC315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNO-CH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-CH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-CH.sub.2 C.sub.6 H.sub.5) 6383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.5)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.5)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.5)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.5)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.5)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.5)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.5)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.5)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.5)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'______________________________________ TABLE 6______________________________________ ##STR28##I: R.sup.1 = HII: R.sup.1 = CH.sub.3III: R.sup.1 = AllylIV: R.sup.1 = PropargylV: R.sup.1 = SCH.sub.3VI: R.sup.1 = CH.sub.2 CNVII: R.sup.1 = CH.sub.2 OCH.sub.3VIII: R.sup.1 = COOCH.sub.3No. B______________________________________ 1 Pyrrolyl-3 2 N-CH.sub.3 -Pyrrolyl-3 3 N-C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N-CH.sub.3 -Pyrrolyl-2 21 N-C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CNC.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CNC.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CNC.sub.6 H.sub.4)-Furyl-2 52 5-(4'-ClC.sub.6 H.sub.4)-Furyl-2 53 5-(3'-ClC.sub.6 H.sub.4)-Furyl-2 54 5-(2'-ClC.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CNC.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CNC.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CNC.sub.6 H.sub.4)-Furyl-2 69 4-(4'-ClC.sub.6 H.sub.4)-Furyl-2 70 4-(3'-ClC.sub.6 H.sub.4)-Furyl-2 71 4-(2'-ClC.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 N-CH.sub.3 -Pyrazolyl-4127 N-C.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 -N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-I5oxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 N-CH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2______________________________________ TABLE 7__________________________________________________________________________Selected physical data of some compoundsNo. Compound mp/.degree.C. IR/cm.sup.-1__________________________________________________________________________ 1 ##STR29## -- 1707, 1484, 1457, 1447, 1303, 1277 2 ##STR30## -- 1708, 1495, 1457, 1449, 1304, 1241 3 ##STR31## 111 4 ##STR32## 73 5 ##STR33## 54 6 ##STR34## -- 1706, 1496, 1456, 1447, 1294, 1243 7 ##STR35## 73 8 ##STR36## 57 9 ##STR37## 86 10 ##STR38## -- 1709, 1599, 1497, 1453, 1346, 1241 11 ##STR39## -- 1708, 1599, 1497, 1455, 1447, 1397, 1238 12 ##STR40## -- 1740, 1593, 1527, 1489, 1456, 1252, 1225 13 ##STR41## -- 1710, 1603, 1584, 1490, 1451, 1364, 1254 14 ##STR42## -- 1709, 1490, 1456, 1447, 1379, 1300, 1258 15 ##STR43## -- 1712, 1490, 1456, 1447, 1378, 1298, 1259 16 ##STR44## 88 17 ##STR45## -- 1710, 1511, 1451, 1364, 1302, 1238 18 ##STR46## -- 1709, 1511, 1456, 1447, 1379, 1301, 1236 19 ##STR47## -- 1712, 1511, 1447, 1378, 1298, 1233 20 ##STR48## -- 1738, 1723, 1582, 1522, 1452, 1223 21 ##STR49## -- 1711, 1492, 1480, 1447, 1362, 1303, 1192, 1159 22 ##STR50## -- 1708, 1491, 1479, 1446, 1376, 1300, 1277, 1150 23 ##STR51## -- 1712, 1511, 1447, 1378, 1298, 1233 24 ##STR52## -- 1736, 1582, 1523, 1453, 1221 25 ##STR53## -- 1706, 1495, 1485, 1363, 1303, 1193, 1160 26 ##STR54## -- 1706, 1484, 1447, 1377, 1301, 1280, 1150 27 ##STR55## -- 1710, 1495, 1483, 1446, 1376, 1299, 1233 28 ##STR56## 92 29 ##STR57## -- 1709, 1489, 1447, 1362, 1303, 1192, 1159 30 ##STR58## -- 1706, 1484, 1447, 1377, 1301, 1280, 1150 31 ##STR59## -- 1711, 1488, 1446, 1375, 1299, 1232 32 ##STR60## 132 33 ##STR61## -- 1709, 1495, 1486, 1451, 1366, 1161, 1008 34 ##STR62## -- 1708, 1487, 1455, 1447, 1379, 1300, 1009 35 ##STR63## -- 1711, 1488, 1447, 1378, 1297, 1232, 1023, 1008 36 ##STR64## -- 1696, 1532, 1515, 1453, 1267, 1245, 1069 37 ##STR65## -- 1712, 1486, 1447, 1361, 1303, 1191, 1160 38 ##STR66## -- 1708, 1485, 1446, 1376, 1300, 1274 39 ##STR67## -- 1709, 1484, 1446, 1374, 1297, 1277, 1232 40 ##STR68## -- 1712, 1495, 1457, 1447, 1378, 1298, 1237 41 ##STR69## 110 42 ##STR70## -- 1739, 1593, 1528, 1511, 1457, 1226, 1035 43 ##STR71## 102 44 ##STR72## -- 1708, 1513, 1457, 1447, 1378, 1302, 1246, 1035 45 ##STR73## 102 46 ##STR74## 74 47 ##STR75## -- 1709, 1606, 1512, 1364, 1245, 1228, 1171, 1162, 1033, 1005 48 ##STR76## 59 1709, 1447, 1364, 1261, 1157, 1034, 1007 49 ##STR77## -- 1709, 1576, 1446, 1379, 1300, 1260, 1239, 1156, 1037 50 ##STR78## -- 51 ##STR79## 89 52 ##STR80## -- 1740, 1593, 1575, 1527, 1457, 1316, 1300, 1224, 1067, 1029 53 ##STR81## 81 54 ##STR82## -- 1711, 1574, 1447, 1365, 1322, 1303, 1213, 1160, 1033, 1008 55 ##STR83## -- 1709, 1574, 1446, 1378, 1321, 1301, 1284, 1213, 1034 56 ##STR84## -- 1711, 1505, 1451, 1365, 1304, 1245, 1160, 1143, 1035, 1007 57 ##STR85## 63 58 ##STR86## -- 1710, 1487, 1450, 1364, 1301, 1246, 1160, 1030, 1006 59 ##STR87## -- 1708, 1487, 1449, 1378, 1300, 1247, 1030, 1009 60 ##STR88## -- 1743, 1593, 1528, 1502, 1457, 1301, 1255, 1190, 1066, 1006 61 ##STR89## 77 62 ##STR90## -- 1712, 1503, 1453, 1363, 1303, 1259, 1244, 1160, 1136, 1006 63 ##STR91## -- 1711, 1503, 1457, 1447, 1380, 1301, 1258, 1239, 1136, 1015 64 ##STR92## 92 1743, 1593, 1528, 1502, 1457, 1301, 1255, 1190, 1066, 1006 65 ##STR93## 90 66 ##STR94## 70 67 ##STR95## 75 68 ##STR96## 108 69 ##STR97## 93 70 ##STR98## 74 71 ##STR99## -- 1712, 1504, 1450, 1363, 1303, 1255, 1222, 1159, 1134 72 ##STR100## -- 1712, 1510, 1498, 1450, 1365, 1327, 1246, 1150, 1035, 1005 73 ##STR101## 60 74 ##STR102## -- 1711, 1509, 1497, 1451, 1363, 1302, 1264, 1193, 1156, 1129 75 ##STR103## -- 1710, 1496, 1475, 1149, 1365, 1301, 1263, 1195, 1159 76 ##STR104## 66 77 ##STR105## 86 78 ##STR106## 91 79 ##STR107## 100 80 ##STR108## -- 1710, 1593, 1497, 1452, 1364, 1323, 1297, 1193, 1165, 1153 81 ##STR109## -- 1715, 1510, 1447, 1367, 1324, 1299, 1243, 1149, 1027, 996 82 ##STR110## -- 1710, 1509, 1456, 1446, 1377, 1326, 1300, 1241, 1149, 1306 83 ##STR111## -- 1723, 1509, 1453, 1437, 1316, 1292, 1241, 1149, 1064, 1036 84 ##STR112## -- 1738, 1611, 1581, 1539, 1446, 1312, 1301, 1231, 1201, 1067 85 ##STR113## -- 1713, 1504, 1447, 1375, 1313, 1300, 1233, 1143, 1027 86 ##STR114## -- 1711, 1486, 1447, 1376, 1300, 1281, 1150, 1034, 1013 87 ##STR115## -- 1714, 1487, 1447, 1376, 1300, 1231, 1023, 999 88 ##STR116## -- 1733, 1594, 1533, 1457, 1306, 1231, 1013, 984 89 ##STR117## -- 1721, 1495, 1453, 1437, 1313, 1290, 1239, 1123 90 ##STR118## -- 1709, 1453, 1366, 1303, 1228, 1160, 1014 91 ##STR119## -- 1708, 1455, 1447, 1378, 1299, 1282, 1015, 996 92 ##STR120## -- 1710, 1447, 1378, 1296, 1232, 1045, 1023, 995 93 ##STR121## 108 94 ##STR122## -- 1717, 1495, 1457, 1444, 1376, 1298, 1241, 1228, 1193 95 ##STR123## -- 1739, 1614, 1603, 1542, 1450, 1262, 129, 1179 96 ##STR124## 170 97 ##STR125## 180 98 ##STR126## 173 99 ##STR127## 150100 ##STR128## 129101 ##STR129## 112102 ##STR130## 116103 ##STR131## 127104 ##STR132## 108105 ##STR133## -- 1710, 1486, 1447, 1363, 1307, 1193, 1159, 1031, 1006, 919106 ##STR134## -- 1706, 1484, 1447, 1376, 1302, 1279, 1150, 1031, 1011, 923107 ##STR135## -- 1711, 1484, 1446, 1376, 1298, 1232, 1144, 1024, 995, 922108 ##STR136## 147109 ##STR137## 1716, 1455, 1445, 1376, 1297, 1279, 1097, 1069, 1017, 1008110 ##STR138## 1718, 1487, 1447, 1394, 1374, 1306, 1232, 1025, 1008111 ##STR139## 109112 ##STR140## 1706, 1487, 1450, 1387, 1304, 1276, 1155, 1022, 1009, 769113 ##STR141## 1706, 1487, 1453, 1383, 1312, 1301, 1274, 1155, 1033, 1008114 ##STR142## 115115 ##STR143## 167116 ##STR144## 1729, 1575, 1565, 1545, 1523, 1445, 1434, 1224, 1060117 ##STR145## 110118 ##STR146## 77119 ##STR147## 1712, 1494, 1447, 1378, 1298, 1232, 1045, 1024, 818, 771120 ##STR148## 115121 ##STR149## 1717, 1455, 1445, 1376, 1298, 1278, 1097, 1068, 1016, 999122 ##STR150## 81123 ##STR151## 1712, 1493, 1447, 1378, 1297, 1232, 1047, 1024, 998, 772124 ##STR152## 107125 ##STR153## 1717, 1455, 1445, 1376, 1298, 1279, 1096, 1068, 1017, 999126 ##STR154## 128127 ##STR155## 1712, 1492, 1447, 1378, 1298, 1232, 1096, 1044, 1023128 ##STR156## 119129 ##STR157## 1717, 1492, 1455, 1445, 1376, 1298, 1096, 1068, 1012, 1000130 ##STR158## 133131 ##STR159## 1712, 1511, 1494, 1447, 1378, 1298, 1232, 1045, 1024, 837132 ##STR160## 113133 ##STR161## 1716, 1511, 1455, 1445, 1376, 1298, 1228, 1097, 1068, 999134 ##STR162## 1737, 1592, 1529, 1509, 1489, 1455, 1303, 1231, 1067, 1014135 ##STR163## 1712, 1586, 1507, 1489, 1454, 1378, 1297, 1239, 1023136 ##STR164## 148137 ##STR165## 1716, 1587, 1507, 1490, 1455, 1375, 1298, 1240, 1068138 ##STR166## 90139 ##STR167## 1719, 1495, 1464, 1446, 1375, 1295, 1239, 1104, 1075, 1014140 ##STR168## 1715, 1495, 1463, 1448, 1376, 1298, 1239141 ##STR169## 134142 ##STR170## 1744, 1583, 1522, 1503, 1458, 1442, 1223, 1304, 1035, 1004143 ##STR171## 1720, 1465, 1446, 1372, 1296, 1280, 1243, 1144, 1035, 1014144 ##STR172## 1716, 1505, 1465, 1448, 1374, 1298, 1279, 1241, 1141, 999145 ##STR173## 109146 ##STR174## 158147 ##STR175## 1718, 1463, 1445, 1376, 1294, 1104, 1073, 1024, 1010148 ##STR176## 1714, 1462, 1447, 1377, 1297, 1238, 1025, 1009149 ##STR177## 140__________________________________________________________________________

Example 4

Methyl N-(2-methylphenyl)-N-methoxy-carbamate (Table 14, No. 1)

a) Methyl N-(2-methylphenyl)-N-hydroxy-carbamate

At 25.degree.-30.degree. C., 14.0 g (0.148 mol) of methyl Chloroocarbonate is added dropwise to 16.4 g of N-(2-methylphenyl)-hydroxylamine (crude product, obtained according to Bamberger et al., Ann. Chem. 316 (1901), 278) and 12.9 g (0.163 mol) of pyridine in 100 ml of methylene Chloroide. The mixture is stirred overnight at room temperature (20.degree. C.) and is then extracted with dilute hydroChloroic acid and water. The organic phase is dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 7 g (39 mmol) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 8.6 (s, broad, OH); 7.3 (m, 4H, phenyl); 3.75 (s, 3H, OCH.sub.3); 2.3 (s, 3H, CH.sub.3)

b) Methyl N-(2-methylphenyl)-N-methoxy-carbamate (Table 14, No. 1)

At 20.degree.-30.degree. C., 1.1 g (44.1 mmol) of sodium hydride is added in portions to 6.6 g (36.5 mmol) of the hydroxyl compound from Example 4a in 50 ml of dimethylformamide. Upon conclusion of gas evolution 5.7 g (40.1 mmol) of methyl iodide is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl-t-butyl ether. The combined organic phases are dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 5.2 g (27 mmol=73%) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.25 (m, 4H, phenyl); 3.8; 3.75 (s, 3H, OCH.sub.3 ; 3.75 (s, 3H, OCH.sub.3); 2.3 (s, 3H, CH.sub.3)

Example 5

Methyl N-(2-bromomethylphenyl)-N-methoxy-carbamate (Table 14, No. 2)

2.5 g (12.8 mmol) of the N-methoxycarbamate from Example 4b, 2.5 g (14.1 mmol) of N-bromosuccinimide and a spatula-tip (1 g) of azoisobutyrodinitrile in 20 ml of carbon tetrachloroide were irradiated with a 300 W UV lamp; the reaction mixture heated up to 30.degree.-40.degree. C. After three hours the reaction mixture is extracted twice with water. The organic phase is dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 1.4 g (5.1 mmol=40%) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.5 (m, 1H, phenyl); 7.35 (m, 3H, phenyl); 4.55 (s, 2H, CH.sub.2 --Br); 3.8 (2s, 6H, 2.times. OCH.sub.3)

Example 6

Methyl N-�2-(2'-methylphenoxymethyl)-phenyl!-N-methoxy-carbamate (Table 14, No. 3)

1.2 g (4.4 mmol) of the methyl bromide from Example 5, 0.45 g (4.2 mmol) o-cresol and 0.7 g (4.8 mmol) of K.sub.2 CO.sub.3 in 30 ml of dimethylformamide are stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl-t-butyl ether. The combined organic phases are dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 1.2 g of the title compound containing o-cresol as impurity. The mixture is heated in a furnace at about 1 mbar for about 1 hour at 125.degree. C. The residue obtained is 0.9 g (3 mmol=68%) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 3H, phenyl); 7.15 (m, 2H, phenyl); 6.9 (t, broad, 2H, phenyl); 5.15 (s, 2H, O--CH.sub.2); 3.8 (s, 3H, OCH.sub.3), 3.75 (s, 3H, OCH.sub.3); 2.3 (s, 3H, CH.sub.3)

TABLE 8______________________________________ ##STR178##I: R.sup.1 = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3No. Xm______________________________________1 H2 2-F3 3-F4 4-F5 2,4-F.sub.26 2,4,6-F.sub.37 2,3,4,5,6-F.sub.58 2,3-F.sub.29 2-Cl10 3-Cl11 4-Cl12 2,3-Cl.sub.213 2,4-Cl.sub.214 2,5-Cl.sub.215 2,6-Cl.sub.216 3,4-Cl.sub.217 3,5-Cl.sub.218 2,3,4-Cl.sub.319 2,3,5-Cl.sub.320 2,3,6-Cl.sub.321 2,4,5-Cl.sub.322 2,4,6-Cl.sub.323 3,4,5-Cl.sub.324 2,3,4,6-Cl.sub.425 2,3,5,6-Cl.sub.426 2,3,4,5,6-Cl.sub.527 2-Br28 3-Br29 4-Br30 2,4-Br.sub.231 2,5-Br.sub.232 2,6-Br.sub.233 2,4,6-Br.sub.334 2,3,4,5,6-Br.sub.535 2-I36 3-I37 4-I38 2,4-I.sub.239 2-Cl, 3-F40 2-Cl, 4-F41 2-Cl, 5-F42 2-Cl, 6-F43 2-Cl, 3-Br44 2-Cl, 4-Br45 2-Cl, 5-Br46 2-Cl, 6-Br47 2-Br, 3-Cl48 2-Br, 4-Cl49 2-Br, 5-Cl50 2-Br, 3-F51 2-Br, 4-F52 2-Br, 5-F53 2-Br, 6-F54 2-F, 3-Cl55 2-F, 4-Cl56 2-F, 5-Cl57 3-Cl, 4-F58 3-Cl, 5-F59 3-Cl, 4-Br60 3-Cl, 5-Br61 3-F, 4-Cl62 3-F, 4-Br63 3-Br, 4-Cl64 3-Br, 4-F65 2,6-Cl.sub.2, 4-Br66 2-CH.sub.367 3-CH.sub.368 4-CH.sub.369 2,3-(CH.sub.3).sub.270 2,4-(CH.sub.3).sub.271 2,5-(CH.sub.3).sub.272 2,6-(CH.sub.3).sub.273 3,4-(CH.sub.3).sub.274 3,5-(CH.sub.3).sub.275 2,3,5-(CH.sub.3).sub.376 2,3,4-(CH.sub.3).sub.377 2,3,6-(CH.sub.3).sub.378 2,4,5-(CH.sub.3).sub.379 2,4,6-(CH.sub.3).sub.380 3,4,5-(CH.sub.3).sub.381 2,3,4,6-(CH.sub.3).sub.482 2,3,5,6-(CH.sub.3).sub.483 2,3,4,5,6-(CH.sub.3).sub.584 2-C.sub.2 H.sub.585 3-C.sub.2 H.sub.586 4-C.sub.2 H.sub.587 2,4-(C.sub.2 H.sub.5).sub.288 2,6-(C.sub.2 H.sub.5).sub.289 3,5-(C.sub.2 H.sub.5).sub.290 2,4,6-(C.sub.2 H.sub.5).sub.391 2-n-C.sub.3 H.sub.792 3-n-C.sub.3 H.sub.793 4-n-C.sub.3 H.sub.794 2-i-C.sub.3 H.sub.795 3-i-C.sub.3 H.sub.796 4-i-C.sub.3 H.sub.797 2,4-(i-C.sub.3 H.sub.7).sub.298 2,6-(i-C.sub.3 H.sub.7).sub.299 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O (C.sub.2 H.sub.5)278 3-CH.sub.2 O (C.sub.2 H.sub.5)279 4-CH.sub.2 O (C.sub.2 H.sub.5)280 2-CH.sub.2 O (n-C.sub.3 H.sub.7)281 3-CH.sub.2 O (n-C.sub.3 H.sub.7)282 4-CH.sub.2 O (n-C.sub.3 H.sub.7)283 2-CH.sub.2 O (i-C.sub.3 H.sub.7)284 3-CH.sub.2 O (i-C.sub.3 H.sub.7)285 4-CH.sub.2 O (i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH (CH.sub.3)CH.sub.3299 3-COCH (CH.sub.3)CH.sub.3300 4-COCH (CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH (CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH (CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3) .644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 9______________________________________ ##STR179##I: R.sup.1 = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3No. B______________________________________1 Pyrrolyl-32 NCH.sub.3 -Pyrrolyl-33 NC.sub.6 H.sub.5 -Pyrrolyl-34 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-35 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-36 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-37 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-38 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-39 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-310 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-311 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-312 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-313 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-314 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-315 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-316 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-317 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-318 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-319 Pyrrolyl-220 NCH.sub.3 -Pyrrolyl-221 NC.sub.6 H.sub.5 -Pyrrolyl-222 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-223 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-224 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-225 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-226 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-227 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-228 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-229 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-230 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-231 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-232 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-233 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-234 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-235 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-236 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-237 Furyl-238 5-CH.sub.3 -Furyl-239 5-C.sub.6 H.sub.5 -Furyl-240 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-241 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-242 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-243 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-244 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-245 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-246 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-247 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-248 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-249 5-(4'-CNC.sub.6 H.sub.4)-Furyl-250 5-(3'-CNC.sub.6 H.sub.4)-Furyl-251 5-(2'-CNC.sub.6 H.sub.4)-Furyl-252 5-(4'-ClC.sub.6 H.sub.4)-Furyl-253 5-(3'-ClC.sub.6 H.sub.4)-Furyl-254 5-(2'-ClC.sub.6 H.sub.4)-Furyl-255 4-CH.sub.3 -Furyl-256 4-C.sub.6 H.sub.5 -Furyl-257 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-258 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-259 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-260 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-261 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-262 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-263 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-264 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-265 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-266 4-(4'-CNC.sub.6 H.sub.4)-Furyl-267 4-(3'-CNC.sub.6 H.sub.4)-Furyl-268 4-(2'-CNC.sub.6 H.sub.4)-Furyl-269 4-(4'-ClC.sub.6 H.sub.4)-Furyl-270 4-(3'-ClC.sub.6 H.sub.4)-Furyl-271 4-(2'-ClC.sub.6 H.sub.4)-Furyl-272 Thienyl-273 5-CH.sub.3 -Thienyl-274 5-C.sub.6 H.sub.5 -Thienyl-275 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-276 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-277 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-278 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-279 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-280 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-281 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-282 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-283 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-284 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-285 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-286 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-287 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-288 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-289 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-290 4-CH.sub.3 -Thienyl-291 4-C.sub.6 H.sub.5 -Thienyl-292 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-293 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-294 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-295 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-296 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-297 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-298 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-299 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 Pyridinyl-3385 1-Naphthyl386 2-Naphthyl______________________________________ TABLE 10______________________________________ ##STR180##I: R.sup.1 = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-C-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2 5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NQ-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(-NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propagyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-C-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-C-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 11______________________________________ ##STR181##I: R.sup.1 = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3No. B______________________________________ 1 Pyrrolyl-3 2 NCH.sub.3 -Pyrrolyl-3 3 NC.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 NCH.sub.3 -Pyrrolyl-2 21 NC.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CNC.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CNC.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CNC.sub.6 H.sub.4)-Furyl-2 52 5-(4'-ClC.sub.6 H.sub.4)-Furyl-2 53 5-(3'-ClC.sub.6 H.sub.4)-Furyl-2 54 5-(2'-ClC.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CNC.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CNC.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CNC.sub.6 H.sub.4)-Furyl-2 69 4-(4'-ClC.sub.6 H.sub.4)-Furyl-2 70 4-(3'-ClC.sub.6 H.sub.4)-Furyl-2 71 4-(2'-ClC.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2 ,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazdlyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-axadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 Pyridinyl-3385 1-Naphthyl386 2-Naphthyl______________________________________ TABLE 12______________________________________ ##STR182##I: R.sup.1 = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2, 5-Me.sub.2 -4-CH.sub.3 CO308 2, 5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2, 5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2, 5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)43i 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-C-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'______________________________________ TABLE 13______________________________________ ##STR183##I: R.sup.1 = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3No. B______________________________________ 1 Pyrrolyl-3 2 NCH.sub.3 -Pyrrolyl-3 3 NC.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 NCH.sub.3 -Pyrrolyl-2 21 NC.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CNC.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CNC.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CNC.sub.6 H.sub.4)-Furyl-2 52 5-(4'-ClC.sub.6 H.sub.4)-Furyl-2 53 5-(3'-ClC.sub.6 H.sub.4)-Furyl-2 54 5-(2'-ClC.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CNC.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CNC.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CNC.sub.6 H.sub.4)-Furyl-2 69 4-(4'-ClC.sub.6 H.sub.4)-Furyl-2 70 4-(3'-ClC.sub.6 H.sub.4)-Furyl-2 71 4-(2'-ClC.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 Pyridinyl-3______________________________________ TABLE 14__________________________________________________________________________Selected physical data of some compoundsNo. Compound .sup.1 H-NMR (ppm)__________________________________________________________________________ 1 ##STR184## 3.8 (s, 3H); 3.75 (s, 3H) 2 ##STR185## 3.8 (2s, 2 .times. 3H) 3 ##STR186## 3.8 (s, 3H); 3.75 (s, 3H) 4 ##STR187## 3.95 (q, 2H, I = 7.5 Hz); 3.8 (s, 3H) 5 ##STR188## 4.05 (q, 2H, I = 7.5 Hz); 3.85 (s, 3H) 6 ##STR189## 4.0 (q, 2H, I = 7.5 Hz); 3.8 (s, 3H) 7 ##STR190## 3.8 (s, 3H); 3.75 (s, 3H) 8 ##STR191## 3.8 (s, 3H); 3.75 (s, 3H) 9 ##STR192## 3.85 (s, 3H); 3.8 (s, 3H)10 ##STR193## 4.0 (s, 3H); 3.8 (s, 3H), 3.75 (s, 3H)11 ##STR194## 3.8 (s, 3H); 3.75 (s, 3H)12 ##STR195## 3.8 (s, 3H); 3.75 (s, 3H)13 ##STR196## 3.8 (s, 3H); 3.75 (s, 3H)14 ##STR197## 3.8 (s, 3H); 3.75 (s, 3H) 6615 ##STR198## 3.8 (s, 3H); 3.75 (s, 3H)16 ##STR199## 4.0 (q, 2H, I = 7.5 Hz); 3.8 (s, 3H)17 ##STR200## 3.8 (2s, each 3H)18 ##STR201## 3.8 (2s, each 3H)19 ##STR202## 3.8 (s, 3H); 3.75 (s, 3H)20 ##STR203## 3.8 (s, 3H); 3.75 (s, 3H)21 ##STR204## 3.8 (s, 3H); 3.75 (s, 3H)22 ##STR205## 3.8 (s, 3H); 3.75 (s, 3H)23 ##STR206## 3.8 (s, 3H); 3.75 (s, 3H)24 ##STR207## 3.8 (s, 6H)25 ##STR208## 3.75 (2s, each 3H)26 ##STR209## 3.8 (s, 3H); 3.75 (s, 3H)27 ##STR210## 3.8 (s, 3H); 3.75 (s, 3H)28 ##STR211## 3.8 (s, 3H); 3.75 (s, 3H)29 ##STR212## 3.8 (s, 3H); 3.75 (s, 3H)30 ##STR213## 3.8 (s, 6H)__________________________________________________________________________ TABLE 52______________________________________Selected physical data of some compounds ##STR214## mp .sup.1 H-NMR (ppm) or IRNo. X.sub.m (.degree.C.) (cm.sup.-1)______________________________________ 1 H 3.75 (2s, each 3H) 2 2-CH.sub.3 3.75 (2s, each 3H) 3 3-CH.sub.3 3.75 (2s, each 3H) 4 2,4-(CH.sub.3).sub.2 3.75 (2s, each 3H) 5 4-C.sub.2 H.sub.5 3.75 (2s, each 3H) 6 4-i-C.sub.3 H.sub.7 3.75 (2s, each 3H) 7 4-t-C.sub.4 H.sub.9 3.75 (2s, each 3H) 8 3,4-(CH.sub.3).sub.2 3.75 (2s, each 3H) 9 3-Cl 3.75 (2s, each 3H)10 3-Br 3.75 (2s, each 3H)11 3-CF.sub.3 3.75 (2s, each 3H)12 4-Br 3.75 (2s, each 3H)13 4-F 3.75 (2s, each 3H)14 4-CF.sub.3 3.75 (2s, each 3H)15 4-OCH.sub.3 3.8 (s, 3H); 3.75 (2s, each 3H)16 4-CN 3.75 (2s, each 3H)17 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7 3.75 (2s, each 3H)18 3,4-Cl.sub.2 3.75 (2s, each 3H)19 3-CH.sub.3 -4-OCH.sub.3 3.85 (s, 3H); 3.75 (2s, each 3H)20 4-NO.sub.2 11221 3,5-(CH.sub.3).sub.2 3.75 (2s, each 3H)22 3-CH.sub.3 -4-Cl 3.75 (2s, each 3H)23 3-Cl-4-CH.sub.3 3.75 (2s, each 3H)______________________________________ TABLE 53__________________________________________________________________________Selected physical data of some compounds ##STR215## .sup.1 H-NMR (ppm) or IRNo. X.sub.m mp (.degree.C.) (cm.sup.-1)__________________________________________________________________________ 1 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5 3.8 (s, 3H); 3.75 (s, 3H) 2 2-CH.sub.3 -4-C(CH.sub.3)NO-(trans-CH.sub.2 CHCHCl) 3.8 (s, 3H); 3.75 (s, 3H) 3 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NOCH.sub.3 3.95 (s, 3H); 3.8 (s, 3H); 3.75 (s, 3H) 4 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NOC.sub.2 H.sub.5 3.8 (s, 3H); 3.75 (s, 3H) 5 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-(trans-CH.sub.2 CHCHCl) 3.85 (s, 3H: 3.75 (s, 3H) 6 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NOCH.sub.3 3.95 (s, 3H); 3.8 (s, 3H); 3.75 (s, 3H) 7 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NOC.sub.2 H.sub.5 3.8 (s, 3H); 3.75 (s, 3H) 8 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NO-Allyl 3.8 (s, 3H); 3.75 (s, 3H) 9 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NO-(trans-CH.sub.2 CHCHCl) 3.8 (s, 3H); 3.75 (s, 3H)10 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)NOCH.sub.3 3.95 (s, 3H); 3.8 (s, 3H); 3.75 (s, 3H)11 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)NOC.sub.2 H.sub.5 3.8 (s, 3H); 3.75 (s, 3H)12 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)NO-Allyl 3.8 (s, 3H); 3.75 (s, 3H)13 2-Cl 3.8 (s, 3H); 3.75 (s, 3H)14 4-Cl 3.8 (s, 3H); 3.75 (s, 3H)15 2-CH.sub.3 -4-Cl 3.8 (s, 3H); 3.75 (s, 3H)16 2-Cl-4-CH.sub.3 3.8 (s, 3H); 3.75 (s, 3H)17 2-Cl-5-CH.sub.3 3.8 (s, 3H); 3.75 (s, 3H)18 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl 3.8 (s, 3H); 3.75 (s, 3H)19 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)NO-(trans-CH.sub.2 CHCHCl) 3.8 (s, 3H); 3.75 (s, 3H)__________________________________________________________________________ TABLE 54______________________________________ ##STR216##I: R.sup.1 = CH.sub.3II: R.sup.1 = C.sub.2 H.sub.5No. B______________________________________ 1 2-Pyridyl 2 3-Trifluormethyl-2-pyridyl 3 5-Trifluormethyl-2-pyridyl 4 3,5-Bis-(trifluoromethyl)-2-pyridyl 5 3,5-Dichloro-2-pyridyl 6 3-Chloro-5-trifluoromethyl-2-pyridyl 7 3,5-Dichloro-2-pyridyl 8 2-Chloro-4-trifluoromethylphenyl 9 2-Benzothiazolyl10 5-Chloro-4-methyl-2-benzimidazolyl11 2-Benzoxazolyl12 1-Methyl-5-trifluoromethylimidazo�5,4-a!-pyridin-2-yl13 5-Chloro-2-pyrimidinyl14 4-Methyl-5-phenyl-2-thiazolin-2-yl15 4-Methyl-5-phenyl-2-oxazolin-2-yl16 7-Trifluoromethyl-4-quinolinyl______________________________________ TABLE 55______________________________________Selected physical data of some compounds ##STR217##No. X.sub.m mp (.degree.C.) .sup.1 H-NMR (ppm) or IR (cm.sup.-1)______________________________________1 H 3.75 (s, 3H); 3.65 (s, 3H)2 4-OCH.sub.3 3.8 (s, 3H); 3.75 (s, 3H); 3.65 (s, 3H)3 4-CH.sub.3 3.75 (s, 3H); 3.65 (s, 3H)4 4-Cl 3.75 (s, 3H); 3.65 (s, 3H)5 4-CF.sub.3 3.75 (s, 3H); 3.65 (s, 3H)6 3,5-(CF.sub.3).sub.2 3.75 (s, 3H); 3.65 (s, 3H)7 2,4-Cl.sub.2 3.75 (s, 3H); 3.65 (s, 3H)8 3,4-Cl.sub.2 3.75 (s, 3H); 3.65 (s, 3H)______________________________________

Example 6

O-Methyl-N-(2-methylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 1)

a) N-(2-Methylphenyl)-N-propionyl-hydroxylamine

At 25.degree. to 30.degree. C., 12,5 g (0.135 mol) of propionyl Chloroide and then 10.7 g (0.135 mol) of pyridine are dripped into 30 g of N-(2-methylphenyl)-hydroxylamine (crude product, prepared according to Bamberger et al., Anm. Chem. 316 (1901), 278; content approx. 80% =0.2 mol) in 500 ml of methylene Chloroide. The mixture is stirred for 30 minutes at room temperature, and is then extracted with dilute hydroChloroic acid and water. The organic phase is dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 22.7 g (0.127 mol =63%) of the title compound as a yellow oil.

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 9.4 (s, broad, 1H, OH); 7.2 (m, 4H, phenyl); 2.4 (s, 3H, CH.sub.3); 2.1 (q, broad, 2H, CH.sub.2); 1.1 (t, 3H, I=7 Hz, CH.sub.3)

b) O-Methyl-N-(2-methylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 1)

At 25.degree. to 30.degree. C., a solution of 22.7 g (0.127 mol) (Example 6a) of N-(2-methylphenyl)-N-propionyl-hydroxylamine in 50 ml of dimethylformamide is dripped into a stirred mixture of 3.4 g (0.14 mol) of NaH in 150 ml of dimethylformamide. After completion of gas evolution (15 mins) 18.4 g (0.13 mol) of methyl iodide is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 18 g (0.081 mol =64%) of the title compound as a yellow oil.

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 7.2 (m, 4H, phenyl); 3.7 (s, broad, 3H, OCH.sub.3); 2.6 (s, very broad, 2H, CH.sub.2); 2.3 (s, 3H, CH.sub.3); 1.2 (s, broad, 3H, CH.sub.3)

Example 7

O-Methyl-N-(2-bromomethylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 2)

A mixture of 10 g (51.8 mmol) of the hydroxylamine derivative from Example 1, 11 g (61 mmol) of N-bromosuccinimide and 0.1 g of azoisobutyrodinitrile in 100 ml of CCl.sub.4 is refluxed. One drop of bromine is added and the mixture is refluxed for a further 2.5 hours. The reaction mixture is cooled to room temperature, washed with water, dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained in this sequence 3.4 g (7.9 mmol =15%) of O-methyl-N-(2-bromomethylphenyl)-d-(.alpha., .alpha.-dibromopropionyl)-hydroxylamine, 3.8 g (10.8 mmol =21%) of O-methyl-N-(2-bromomethylphenyl)-N-(.alpha.-bromopropionyl)-hydroxylamine, 2.3 g (8.5 g (8.5 mmol =16%) of the title compound and 3.5 g of starting material, each as brown oils.

a) O-Methyl-N-(2-bromomethylphenyl)-N-(.alpha., .alpha.-dibromopropionyl)-hydroxylamine

7.55 (m, 1H, phenyl); 7.4 (m, 3H, phenyl); 4.5 (s, 2H, CH.sub.2, Br); 3.8 (s, 3H, OCH.sub.3); 2.75 (s, 3H, CH.sub.3)

b) O-Methyl-N-(2-bromomethylphenyl)-N-(.alpha.-bromopropionyl)-hydroxylamine

7.5 (s, broad, 1H, phenyl); 7.4 (s, broad, 3H, phenyl); 5.15 (s, broad, 1H, CH--Br); 4.5 (dd, broad, 2H, CH.sub.2 --Br); 3.8 (s, 3H, OCH.sub.3); 1.85 (s, broad, 3H, CH.sub.3)

c) O-Methyl-N-(2-bromomethylphenyl)-N-propionyl-hydroxylamine

7.5 (m, 1H, phenyl); 7.35 (m, 3H, phenyl); 4.5 (s, broad, 2H, CH.sub.2 --Br); 3.75 (s, 3H, OCH.sub.3); 2.55 (s, very broad, CH.sub.2); 1.2 (t, 3H, I=7 Hz, CH.sub.3)

Example 8

O-Methyl-N-(2-(2'-methylphenyloxymethyl)-phenyl)-N-propionyl-hydroxylamine (Table 21, No. 3)

0.12 g (5 mmol) of sodium hydride is added to a solution of 0.4 g (3.7 mmol) of o-cresol in 5 ml of dimethylformamide. Upon completion of gas evolution, 1 g (3.6 mmol) of the benzyl bromide from Example 2c is added and the mixture is stirred for 2 hours at room temperature. The reaction mixture is diluted with water and extracted three times with methyl tert-butyl ether. The combined organic phases are washed with water, dried over MgSO.sub.4 and evaporated down. The residue is chromatographed with mixtures of cyclohexane and ethyl acetate using Al.sub.2 O.sub.3 and silica gel. There is obtained 0.4 g (1.33 mmol =37%) of the title compound as a yellow oil.

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 7.7 (d, broad, 1H, phenyl); 7.35 (m, 3H, phenyl); 7.1 (m, 2H, phenyl); 6.85 (t, broad, 2H, phenyl); 5.05 (s, 2H, OCH.sub.3); 3.7 (s, 3H, OCH.sub.3); 2.55 (s, very broad, 2H, CH.sub.2); 2.3 (s, 3H, CH.sub.3); 1.2 (t, broad, 3H, CH.sub.3)

Example 9

N-Methyl-N'-methoxy-N'-2-methylphenylurea (Table 21, No. 5)

a) Phenyl N-hydroxy-N-(2-methylphenyl)-carbamate

A mixture of 2.5 g (20 mmol) of N-(2-methylphenyl)-hydroxylamine (crude product, obtained according to Bamberger et al., Anm. Chem. 316 (1901), 278), 3.5 g (25 mmol) of K.sub.2 CO.sub.3 and 3.5 g (22 mmol) of phenyl Chlorooformate in 20 ml of CH.sub.2 Cl.sub.2 is stirred for 2 hours at room temperature. The reaction mixture is then extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 2.0 g (8.2 mmol =42%) of the title compound as a colorless solid (mp=98.degree. C.).

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 7-7.6 (m, 10H, phenyl, OH); 2.35 (s, 3H, CH.sub.3)

b) Phenyl N-methoxy-N-(2-methylphenyl)-carbamate

A mixture of 2.0 g (8.2 mmol) of the phenyl carbamate from Example 4a, 2 g (15 mmol) of K.sub.2 CO.sub.3 and 1.3 g (10 mmol) of dimethyl sulfate in 20 ml of acetone is stirred for 3 hours at room temperature. The reaction mixture is then filtered and evaporated down, and the residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 1.5 g (5.8 mmol =71%) of the title compound as a colorless oil, which slowly crystallizes (mp=60.degree. C.).

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 7.1-7.5 (m, 9H, phenyl); 3.8 (s, 3H, OCH.sub.3); 2.4 (s, 3H, CH.sub.3)

c) N-Methyl-N'-methoxy-N'-2-methylphenylurea (Table 21, No. 5)

1.5 g (5.8 mmol) of the phenyl carbamate from Example 4b in 20 ml of 40% strength aqueous methylamine solution is stirred for 1 hour at 50.degree. C. The reaction mixture is then cooled and extracted with CH.sub.2 Cl.sub.2. The combined organic phases are dried over MgCO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 0.6 g (3.1 mmol =53%) of the title compound as a colorless solid (mp=99.degree. C.).

.sup.1 H-NMR (COCl.sub.3 ; .delta. in ppm): 7.2 (m, 4H, phenyl); 5.9 (s, broad, 1H, NH); 3.6 (s, 3H, OCH.sub.3); 2.9 (d, 3H, I=approx. 2 Hz, N--CH.sub.3); 2.3 (s, 3H, CH.sub.3)

Example 18

N-Methyl-N'-methoxy-N'-(2-2',5'-dimethylphenoxymethyl)-phenyl)-urea

a) Phenyl N-methoxy-N-(2-bromomethylphenyl)-carbamate

A mixture of 125 g (0.486 mol) of methyl N-methoxy-N-(2-methylphenyl)-carbamate (Example 4b), 88 g (0.494 mol) of N-bromosuccinimide and 1 g of azoisobutyrodinitrile (AIBN) in 800 ml of CCl.sub.4 is refluxed for about 12 hours. 10 g of N-bromosuccinimide is then added and the mixture is refluxed for about 4 hours. The reaction mixture is extracted with water and sodium thiosulfate solution, and the organic phase is dried over MgSO.sub.4 and evaporated down under reduced pressure. The residue crystallizes, is stirred with hexane/methyl tert-butyl ether and suction dried. There is obtained 107 g (63%) of the title compound as a colorless solid.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.1-7.6 (m, 9H, phenyl); 4.5 (s, 2H, CH.sub.2 Br); 3.9 (s, 3H, OCH.sub.3)

b) Phenyl N-methoxy-N-(2-(2',5'-dimethylphenoxymethyl)-phenyl)-carbamate

A mixture of 7 g (20 mmol) of the bromide of Example 5a and 3.3 g (22 mmol) of sodium iodide in 50 ml of acetone is refluxed for 30 minutes. The precipitated solid is then filtered off and the organic phase is evaporated down under reduced pressure. The crude product obtained is the iodide corresponding to Example 5a, which is used in the next reaction without any further purification.

The crude product obtained above is dissolved in 100 ml of dimethylformamide, 3 g (21.6 mmol) of K.sub.2 CO.sub.3 and 7.3 g (60 mmol) of 2,5-dimethylphenol are added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography using methylene chloride/cyclohexane (1:2) over Al.sub.2 O.sub.3. There is obtained 7.3 g (94%) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in PPM): 7.7 (d, broad, 1H, phenyl); 7-7.6 (m, 9H, phenyl); 6.7 (m, 2H, phenyl); 5.2 (s, 2H, OCH.sub.2); 3.85 (s, 3H, OCH.sub.3); 2.3 (s, 6H, 2.times.CH.sub.3).

c) N-Methyl-N'-methoxy-N'-(2-(2', 5'-dimethylphenoxymethyl)-phenyl)-urea (Table 1, No. V. 71)

A mixture of 3.4 g (8.8 mmol) of the phenyl carbamate of Example 5b and 20 ml of 40% strength aqueous methylamine solution is stirred for 2 hours at 50.degree. C. The mixture is allowed to cool and is then extracted with methylene chloride. The organic phase is evaporated down and the residue is purified by column chromatography with mixtures of cyclohexane/ethyl acetate. There is obtained 1 g (36%) of the title compound as a colorless solid (mp=101.degree. C).

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in PPM):

7.75 (m, 1H, phenyl); 6.6-7.4 (m, 6H, phenyl); 6.0 (s, broad, NH); 5.15 (s, 2H, OCH.sub.2); 3.65 (s, 3H, OCH.sub.3); 2.9 (d, 3H, N--CH.sub.3); 2.3 (s, 3H, CH.sub.3); 2.25 (s, 3H, CH.sub.3).

The compounds listed in the tables below may be prepared analogously. Compound I.1 from Table 15 has for instance the following formula ##STR218##

TABLE 15______________________________________I: R.sup.1 = CH.sub.3, Z = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3, Z = CH.sub.3III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5)3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2O (C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NO-CH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NO-CH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NO-CH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 -CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 16______________________________________ ##STR219##I: R.sup.1 = CH.sub.3, Z = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3, Z = CH.sub.3III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3No. B______________________________________1 Pyrrolyl-32 NCH.sub.3 -Pyrrolyl-33 NC.sub.6 H.sub.5 -Pyrrolyl-34 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-35 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-36 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-37 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-38 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-39 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-310 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-311 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-312 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-313 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-314 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-315 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-316 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-317 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-318 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-319 Pyrrolyl-220 NCH.sub.3 -Pyrrolyl-221 NC.sub.6 H.sub.5 -Pyrrolyl-222 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-223 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-224 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-225 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-226 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-227 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-228 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-229 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-230 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-231 N-(4'-CNC.sub.6 H.sub.4 )-Pyrrolyl-232 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-233 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-234 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-235 N-(3'-ClC.sub.6 H.sub.4 )-Pyrrolyl-236 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-237 Furyl-238 5-CH.sub.3 -Furyl-239 5-C.sub.6 H.sub.5 -Furyl-240 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-241 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-242 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-243 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-244 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-245 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-246 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-247 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-248 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-249 5-(4'-CNC.sub.6 H.sub.4)-Furyl-250 5-(3'-CNC.sub.6 H.sub.4)-Furyl-251 5-(2'-CNC.sub.6 H.sub.4)-Furyl-252 5-(4'-ClC.sub.6 H.sub.4)-Furyl-253 5-(3'-ClC.sub.6 H.sub.4)-Furyl-254 5-(2'-ClC.sub.6 H.sub.4)-Furyl-255 4-CH.sub.3 -Furyl-256 4-C.sub.6 H.sub.5 -Furyl-257 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-258 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-259 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-260 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-261 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-262 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-263 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-264 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-265 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-266 4-(4'-CNC.sub.6 H.sub.4)-Furyl-267 4-(3'-CNC.sub.6 H.sub.4)-Furyl-268 4-(2'-CNC.sub.6 H.sub.4)-Furyl-269 4-(4'-ClC.sub.6 H.sub.4)-Furyl-270 4-(3'-ClC.sub.6 H.sub.4)-Furyl-271 4-(2'-ClC.sub.6 H.sub.4)-Furyl-272 Thienyl-273 5-CH.sub.3 -Thienyl-274 5-C.sub.6 H.sub.5 -Thienyl-275 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-276 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-277 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-278 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-279 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-280 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-281 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-282 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-283 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-284 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-285 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-286 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-287 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-288 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-289 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-290 4-CH.sub.3 -Thienyl-291 4-C.sub.6 H.sub.5 -Thienyl-292 4-(4'-,CH.sub.3 C.sub.6 H.sub.4)-Thienyl-293 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-294 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-295 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-296 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-297 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-298 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-299 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 HA)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 -C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 Pyridinyl-3385 1-Naphthyl386 2-Naphthyl______________________________________ TABLE 17______________________________________ ##STR220##I: R.sup.1 = CH.sub.3, Z = CH.sub.3II: R.sup.1 CH.sub.2 CH.sub.3, Z = CH.sub.3III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCHNO. X.sub.m______________________________________1 H2 2-F3 3-F4 4-F5 2,4-F.sub.26 2,4,6-F.sub.37 2,3,4,5,6-F.sub.58 2,3-F.sub.29 2-Cl10 3-Cl11 4-Cl12 2,3-Cl.sub.213 2,4-Cl.sub.214 2,5-Cl.sub.215 2,6-Cl.sub.216 3,4-Cl.sub.217 3,5-Cl.sub.218 2,3,4-Cl.sub.319 2,3,5-Cl.sub.320 2,3,6-Cl.sub.321 2,4,5-Cl.sub.322 2,4,6-Cl.sub.323 3,4,5-Cl.sub.324 2,3,4,6-Cl.sub.425 2,3,5,6-Cl.sub.426 2,3,4,5,6-Cl.sub.527 2-Br28 3-Br29 4-Br30 2,4-Br.sub.231 2,5-Br.sub.232 2,6-Br.sub.233 2,4,6-Br.sub.334 2,3,4,5,6-Br.sub.535 2-I36 3-I37 4-I38 2,4-I.sub.239 2-Cl, 3-F40 2-Cl, 4-F41 2-Cl, 5-F42 2-Cl, 6-F43 2-Cl, 3-Br44 2-Cl, 4-Br45 2-Cl, 5-Br46 2-Cl, 6-Br47 2-Br, 3-Cl48 2-Br, 4-Cl49 2-Br, 5-Cl50 2-Br, 3-F51 2-Br, 4-F52 2-Br, 5-F53 2-Br, 6-F54 2-F, 3-Cl55 2-F, 4-Cl56 2-F, 5-Cl57 3-Cl, 4-F58 3-Cl, 5-F59 3-Cl, 4-Br60 3-Cl, 5-Br61 3-F, 4-Cl62 3-F, 4-Br63 3-Br, 4-Cl64 3-Br, 4-F65 2,6-Cl.sub.2, 4-Br66 2-CH.sub.367 3-CH.sub.368 4-CH.sub.369 2,3-(CH.sub.3).sub.270 2,4-(CH.sub.3).sub.271 2,5-(CH.sub.3).sub.272 2,6-(CH.sub.3).sub.273 3,4-(CH.sub.3).sub.274 3,5-(CH.sub.3).sub.275 2,3,5-(CH.sub.3).sub.376 2,3,4-(CH.sub.3).sub.377 2,3,6-(CH.sub.3).sub.378 2,4,5-(CH.sub.3).sub.379 2,4,6-(CH.sub.3).sub.380 3,4,5-(CH.sub.3).sub.381 2,3,4,6-(CH.sub.3).sub.482 2,3,5,6-(CH.sub.3).sub.483 2,3,4,5,6-(CH.sub.3).sub.584 2-C.sub.2 H.sub.585 3-C.sub.2 H.sub.586 4-C.sub.2 H.sub.587 2,4-(C.sub.2 H.sub.5).sub.288 2,6-(C.sub.2 H.sub.5).sub.289 3,5-(C.sub.2 H.sub.5).sub.290 2,4,6-(C.sub.2 H.sub.5).sub.391 2-n-C.sub.3 H.sub.792 3-n-C.sub.3 H.sub.793 4-n-C.sub.3 H.sub.794 2-i-C.sub.3 H.sub.795 3-i-C.sub.3 H.sub.796 4-i-C.sub.3 H.sub.797 2,4-(i-C.sub.3 H.sub.7).sub.298 2,6-(i-C.sub.3 H.sub.7).sub.299 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(Cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH (CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 -CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-CH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Propargyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4- (CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-CCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 18______________________________________ ##STR221##I: R.sup.1 = CH.sub.3, Z = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3, Z = CH.sub.3III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3No. B______________________________________ 1 Pyrrolyl-3 2 N-CH.sub.3 -Pyrrolyl-3 3 N-C.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 NCH.sub.3 -Pyrrolyl-2 21 NC.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CNC.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CNC.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CNC.sub.6 H.sub.4)-Furyl-2 52 5-(4'-ClC.sub.6 H.sub.4)-Furyl-2 53 5-(3'-ClC.sub.6 H.sub.4)-Furyl-2 54 5-(2'-ClC.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CNC.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CNC.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CNC.sub.6 H.sub.4)-Furyl-2 69 4-(4'-ClC.sub.6 H.sub.4)-Furyl-2 70 4-(3'-ClC.sub.6 H.sub.4)-Furyl-2 71 4-(2'-ClC.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 Pyridinyl-3385 1-Naphthyl386 2-Naphthyl______________________________________ TABLE 19______________________________________ ##STR222##I: R.sup.1 = CH.sub.3, Z = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3, Z = CH.sub.3III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5V: R.sup.1 CH.sub.3, Z = NHCH.sub.3VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2.3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-O-C.sub.2 H.sub.5164 4-O-C.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-O-CH.sub.2 C.sub.6 H.sub.5178 3-O-CH.sub.2 C.sub.6 H.sub.5179 4-O-CH.sub.2 C.sub.6 H.sub.5180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-0-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'______________________________________ TABLE 20______________________________________ ##STR223##I: R.sup.1 = CH.sub.3, Z = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3, Z CH.sub.3III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3No. B______________________________________ 1 Pyrrolyl-3 2 NCH.sub.3 -Pyrrolyl-3 3 NC.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 NCH.sub.3 -Pyrrolyl-2 21 NC.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CNC.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CNC.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CNC.sub.6 H.sub.4)-Furyl-2 52 5-(4'-ClC.sub.6 H.sub.4)-Furyl-2 53 5-(3'-ClC.sub.6 H.sub.4)-Furyl-2 54 5-(2'-ClC.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CNC.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CNC.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CNC.sub.6 H.sub.4)-Furyl-2 69 4-(4'-ClC.sub.6 H.sub.4)-Furyl-2 70 4-(3'-ClC.sub.6 H.sub.4)-Furyl-2 71 4-(2'-ClC.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 Pyridinyl-3______________________________________ TABLE 21__________________________________________________________________________Selected physical data of some compoundsNo. Compound .sup.1 H-NMR (ppm) m.p.__________________________________________________________________________ 1 ##STR224## 3.7 (s, broad, 3H); 1.2 (s, broad, 3H) 2 ##STR225## 3.75 (s, 3H); 1.2 (t, 3H) 3 ##STR226## 3.7 (s, 3H); 1.2 (t, 3H) 4 ##STR227## 3.95 (s, 3H); 3.7 (s, 3H); 1,2 (t, 3H) 5 ##STR228## 3.6 (s, 3H); 2.9 (d, 3H) 6 ##STR229## 123 7 ##STR230## 118 8 ##STR231## 3.7 (s, 3H); 2.55 (s, very__________________________________________________________________________ broad, 2H) TABLE 56______________________________________Selected physical data of some compounds ##STR232## mp .sup.1 H-NMR (ppm) orNo. X.sub.m (.degree.C.) IR (cm.sup.-1)______________________________________1 H 902 2-CH.sub.3 803 2,5-(CH.sub.3).sub.2 1014 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 3.95 (s, 3H); 3.65 (s, 3H); 2.9 (d, 3H)5 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl 3.65 (s, 3H); 2.9 (d, 3H)______________________________________ TABLE 22______________________________________ ##STR233##No. X Z A______________________________________ 1 H CH.sub.3 CH.sub.2 O 2 H CH.sub.3 CH.sub.2 ONC(CH.sub.3) 3 H CH.sub.3 CHCH 4 H NH.sub.2 CH.sub.2 O 5 H NH.sub.2 CH.sub.2 ONC(CH.sub.3) 6 H NH.sub.2 CHCH 7 H N(CH.sub.3).sub.2 CH.sub.2 O 8 H N(CH.sub.3).sub.2 CH.sub.2 ONC(CH.sub.3) 9 H N(CH.sub.3).sub.2 CHCH10 H CCl.sub.3 CH.sub.2 O11 H CCl.sub.3 CH.sub.2 ONC(CH.sub.3)12 H CCl.sub.3 CHCH13 H CF.sub.3 CH.sub.2 O14 H CF.sub.3 CH.sub.2 ONC(CH.sub.3)15 H CF.sub.3 CHCH16 CH.sub.3 CH.sub.3 CH.sub.2 O17 CH.sub.3 CH.sub.3 CH.sub.2 ONC(CH.sub.3)18 CH.sub.3 CH.sub.3 CHCH19 CH.sub.3 NH.sub.2 CH.sub.2 O20 CH.sub.3 NH.sub.2 CH.sub.2 ONC(CH.sub.3)21 CH.sub.3 NH.sub.2 CHCH22 CH.sub.3 N(CH.sub.3).sub.2 CH.sub.2 O23 CH.sub.3 N(CH.sub.3).sub.2 CH.sub.2 ONC(CH.sub.3)24 CH.sub.3 N(CH.sub.3).sub.2 CHCH25 CH.sub.3 CCl.sub.3 CH.sub.2 O26 CH.sub.3 CCl.sub.3 CH.sub.2 ONC(CH.sub.3)27 CH.sub.3 CCl.sub.3 CHCH28 CH.sub.3 CF.sub.3 CH.sub.2 O29 CH.sub.3 CF.sub.3 CH.sub.2 ONC(CH.sub.3)30 CH.sub.3 CF.sub.3 CHCH31 Cl CH.sub.3 CH.sub.2 O32 Cl CH.sub.3 CH.sub.2 ONC(CH.sub.3)33 Cl CH.sub.3 CHCH34 Cl NH.sub.2 CH.sub.2 O35 Cl NH.sub.2 CH.sub.2 ONC(CH.sub.3)36 Cl NH.sub.2 CHCH37 Cl N(CH.sub.3).sub.2 CH.sub.2 O38 Cl N(CH.sub.3).sub.2 CH.sub.2 ONC(CH.sub.3)39 Cl N(CH.sub.3).sub.2 CHCH40 Cl CCl.sub.3 CH.sub.2 O41 Cl CCl.sub.3 CH.sub.2 ONC(CH.sub.3)42 Cl CCl.sub.3 CHCH43 Cl CF.sub.3 CH.sub.2 O44 Cl CF.sub.3 CH.sub.2 ONC(CH.sub.3)45 Cl CF.sub.3 CHCH______________________________________ TABLE 23______________________________________ ##STR234##I: R.sup.1 = CH.sub.3, Z = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3, Z =CH.sub.3III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3No. B______________________________________ 1 2-pyridyl 2 3-Trifluoromethyl-2-pyridyl 3 5-Trifluoromethyl-2-pyridyl 4 3,5-Bis-(trifluoromethyl)-2-pyridyl 5 3,5-Dichloro-2-pyridyl 6 3-Chloro-5-trifluoromethyl-2-pyridyl 7 3,5-Dichloro-2-pyridyl 8 2-Chloro-4-trifluormethylphenyl 9 2-Benzothiazolyl10 5-Chloro-4-methyl-2-benzimidazolyl11 2-Benzoxazolyl12 1-Methyl-5-trifluoromethylimi- dazo�5,4-a!-pyridin-2-yl13 5-Chloro-2-pyrimidinyl14 4-Methyl-5-phenyl-2-thiazolin-2-yl15 4-Methyl-5-phenyl-2-Oxazolin-2-yl16 7-Trifluoromethyl-4-quinolinyl______________________________________

Example 10

N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-O-methyl-hydroxylamine (Table 30, No. 1)

a) N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-hydroxylamine

At 0.degree. to 5.degree. C., 7.0 g (70 mmol) of methyl chloroformate is added dropwise to 11.3 g (80 mmol) of N-2,6-dimethylphenyl-hydroxylamine (prepared analogously to Bamberger et al., Ann. Chem. 316 (1901), 278) and 12.5 g (90 mmol) of K.sub.2 CO.sub.3 in 30 ml of methylene chloride. The mixture is stirred for 30 mins at 0.degree.-5.degree. C., the insoluble solid is filtered off and the filtrate is evaporated down under reduced pressure. The residure is purified by column chromatography with mixtures of cyclohexand and ethyl acetate. There is obtained 1.4 g (7.2 mmol=9%) of the title compound as a dark oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 8.85 (s, broad, 1H, OH); 7.1 (m, 3H, phenyl); 3.75 (s, 3H, OCH.sub.3); 2.3 (s, 6H, 2.times.CH.sub.3)

b) N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-O-methylhydroxylamine (Table 7, No. 1)

A mixture of 1.4 g (7.2 mmol) of N-(2,6-dimethylphenyl)-N-methoxycarbonyl-hydroxylamine (Example 1a), 1.3 g (9 mmol) of K.sub.2 CO.sub.3 and 10 g (8 mmol) of dimethyl sulfate in 10 ml of acetone is stirred overnight at room temperature. The reaction mixture is then diluted with CH.sub.2 Cl.sub.2 and stirred with dilute NH.sub.3 solution. The phases are then separated and the organic phase is extracted another twice with water. The organic phase is dried over MgSO.sub.4 and evaporated down, and the residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 1.2 g (6 mmol=83%) of the title compound as a colorless solid (mp=81.degree. C.).

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.1 (m, 3H, phenyl); 3.75 (s, broad, 6H, 2.times.OCH3); 2.3 (s, 3H, CH.sub.3)

The compounds listed in the following tables may be prepared similarly. Compound I, No. 1 from Table 24, No. 1 has for example the following formula: ##STR235##

TABLE 24______________________________________a I: R.sup.1 = CH.sub.3, X = CH.sub.3b II: R.sup.1 = CH.sub.2 CH.sub.3, X = CH.sub.3c III: R.sup.1 = CH.sub.3, X = Cld IV: R.sup.1 = CH.sub.2 CH.sub.2, X = ClNo. T.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.21I1 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 -CO303 2-Me-4-CH.sub.3 -CH.sub.2 CO304 2-Me-4-CH.sub.3 -CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 -CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 -CO308 2,5-Me.sub.2 -4-CH.sub.3 -CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 -CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 -CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 -CO313 2-Cl-4-CH.sub.3 -CH.sub.2 CO314 2-Cl-4-CH.sub.3 -CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 -CO317 2,5-Cl.sub.2 -4-CH.sub.3 -CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 -CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 -CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)CH.sub.3333 3-C(NO-Allyl)CH.sub.3334 4-C(NO-Allyl)CH.sub.3335 2-C(NO-trans-Chloroallyl)CH.sub.3336 3-C(NO-trans-Chloroallyl)CH.sub.3337 4-C(NO-trans-Chloroallyl)CH.sub.3338 2-C(NO-Propargyl)CH.sub.3339 3-C(NO-Propargyl)CH.sub.3340 4-C(NO-Propargyl)CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 -CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 -CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 -CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 -CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 -CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 -CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 -CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 -CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 -CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 25______________________________________ ##STR236##I: R.sup.1 = CH.sub.3, X = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3, X = CH.sub.3III: R.sup.1 = CH.sub.3, X = ClIV: R.sup.1 = CH.sub.2 CH.sub.3, X = ClNo. B______________________________________ 1 Pyrrolyl-3 2 NCH.sub.3 -Pyrrolyl-3 3 NC.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 NCH.sub.3 -Pyrrolyl-2 21 NC.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CNC.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CNC.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CNC.sub.6 H.sub.4)-Furyl-2 52 5-(4'-ClC.sub.6 H.sub.4)-Furyl-2 53 5-(3'-ClC.sub.6 H.sub.4)-Furyl-2 54 5-(2'-ClC.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CNC.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CNC.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CNC.sub.6 H.sub.4)-Furyl-2 69 4-(4'-ClC.sub.6 H.sub.4)-Furyl-2 70 4-(3'-ClC.sub.6 H.sub.4)-Furyl-2 71 4-(2'-ClC.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(41-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 -N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4 -4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazoiyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 Pyridinyl-3385 1-Naphthyl386 2-Naphthyl______________________________________ TABLE 26______________________________________ ##STR237##I: R.sup.1 = CH.sub.3, X = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3, X = CH.sub.3III: R.sup.1 = CH.sub.3, X = ClIV: R.sup.1 = CH.sub.2 CH.sub.3, X = ClNo. T.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-CH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyI))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 27______________________________________ ##STR238##I: R.sup.1 = CH.sub.3, X = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3, X = CH.sub.3III: R.sup.1 = CH.sub.3, X = ClIV: R.sup.1 = CH.sub.2 CH.sub.3, X = ClNo. B______________________________________ 1 Pyrrolyl-3 2 NCH.sub.3 -Pyrrolyl-3 3 NC.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 N-CH.sub.3 -Pyrrolyl-2 21 N-C.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CNC.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CNC.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CNC.sub.6 H.sub.4)-Furyl-2 52 5-(4'-ClC.sub.6 H.sub.4)-Furyl-2 53 5-(3'-ClC.sub.6 H.sub.4)-Furyl-2 54 5-(2'-ClC.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CNC.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CNC.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CNC.sub.6 H.sub.4)-Furyl-2 69 4-(4'-ClC.sub.6 H.sub.4)-Furyl-2 70 4-(3'-ClC.sub.6 H.sub.4)-Furyl-2 71 4-(2'-ClC.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 -N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 Pyridinyl-3385 1-Naphthyl386 2-Naphthyl______________________________________ TABLE 28______________________________________ ##STR239##I: R.sup.1 = CH.sub.3, X = CH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3, X = CH.sub.3III: R.sup.1 = CH.sub.3, X = ClIV: R.sup.1 = CH.sub.2 CH.sub.3, X = ClNo. T.sub.m______________________________________1 H2 2-F3 3-F4 4-F5 2,4-F.sub.26 2,4,6-F.sub.37 2,3,4,5,6-F.sub.58 2,3-F.sub.29 2-Cl10 3-Cl11 4-Cl12 2,3-Cl.sub.213 2,4-Cl.sub.214 2,5-Cl.sub.215 2,6-Cl.sub.216 3,4-Cl.sub.217 3,5-Cl.sub.218 2,3,4-Cl.sub.319 2,3,5-Cl.sub.320 2,3,6-Cl.sub.321 2,4,5-Cl.sub.322 2,4,6-Cl.sub.323 3,4,5-Cl.sub.324 2,3,4,6-Cl.sub.425 2,3,5,6-Cl.sub.426 2,3,4,5,6-Cl.sub.527 2-Br28 3-Br29 4-Br30 2,4-Br.sub.231 2,5-Br.sub.232 2,6-Br.sub.233 2,4,6-Br.sub.334 2,3,4,5,6-Br.sub.535 2-I36 3-I37 4-I38 2,4-I.sub.239 2-Cl, 3-F40 2-Cl, 4-F41 2-Cl, 5-F42 2-Cl, 6-F43 2-Cl, 3-Br44 2-Cl, 4-Br45 2-Cl, 5-Br46 2-Cl, 6-Br47 2-Br, 3-Cl48 2-Br, 4-Cl49 2-Br, 5-Cl50 2-Br, 3-F51 2-Br, 4-F52 2-Br, 5-F53 2-Br, 6-F54 2-F, 3-Cl55 2-F, 4-Cl56 2-F, 5-Cl57 3-Cl, 4-F58 3-Cl, 5-F59 3-Cl, 4-Br60 3-Cl, 5-Br61 3-F, 4-Cl62 3-F, 4-Br63 3-Br, 4-Cl64 3-Br, 4-F65 2,6-Cl.sub.2, 4-Br66 2-CH.sub.367 3-CH.sub.368 4-CH.sub.369 2,3-(CH.sub.3).sub.270 2,4-(CH.sub.3).sub.271 2,5-(CH.sub.3).sub.272 2,6-(CH.sub.3).sub.273 3,4-(CH.sub.3).sub.274 3,5-(CH.sub.3).sub.275 2,3,5-(CH.sub.3).sub.376 2,3,4-(CH.sub.3).sub.377 2,3,6-(CH.sub.3).sub.378 2,4,5-(CH.sub.3).sub.379 2,4,6-(CH.sub.3).sub.380 3,4,5-(CH.sub.3).sub.381 2,3,4,6-(CH.sub.3).sub.482 2,3,5,6-(CH.sub.3).sub.483 2,3,4,5,6-(CH.sub.3).sub.584 2-C.sub.2 H.sub.585 3-C.sub.2 H.sub.586 4-C.sub.2 H.sub.587 2,4-(C.sub.2 H.sub.5).sub.288 2,6-(C.sub.2 H.sub.5).sub.289 3,5-(C.sub.2 H.sub.5).sub.290 2,4,6-(C.sub.2 H.sub.5).sub.391 2-n-C.sub.3 H.sub.792 3-n-C.sub.3 H.sub.793 4-n-C.sub.3 H.sub.794 2-i-C.sub.3 H.sub.795 3-i-C.sub.3 H.sub.796 4-i-C.sub.3 H.sub.797 2,4-(i-C.sub.3 H.sub.7).sub.298 2,6-(i-C.sub.3 H.sub.7).sub.299 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3,5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7,5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-CCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4, 5-(CH.sub.3).sub.2228 2-Br, 4, 5-(CH.sub.3).sub.2229 2-Cl, 3, 5-(CH.sub.3).sub.2230 2-Br, 3, 5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 214-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 CO-C.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4640 4-Thiazolyl-5'______________________________________ TABLE 29______________________________________ ##STR240##I: R.sup.1 = CH.sub.3, XCH.sub.3II: R.sup.1 = CH.sub.2 CH.sub.3, XCH.sub.3III: R.sup.1 = CH.sub.3, XClIV: R.sup.1 = CH.sub.2 CH.sub.3, XClNo. B______________________________________1 Pyrrolyl-32 NCH.sub.3 -Pyrrolyl-33 NC.sub.6 H.sub.5 -Pyrrolyl-34 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-35 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-36 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-37 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-38 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-39 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-310 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-311 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-312 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-313 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-314 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-315 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-316 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-317 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-318 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-319 Pyrrolyl-220 NCH.sub.3 -Pyrrolyl-221 NC.sub.6 H.sub.5 -Pyrrolyl-222 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-223 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-224 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-225 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-226 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-227 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-228 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-229 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-230 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-231 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-232 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-233 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-234 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-235 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-236 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-237 Furyl-238 5-CH.sub.3 -Furyl-239 5-C.sub.6 H.sub.5 -Furyl-240 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-241 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-242 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-243 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-244 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-245 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-246 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-247 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-248 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-249 5-(4'-CNC.sub.6 H.sub.4)-Furyl-250 5-(3'-CNC.sub.6 H.sub.4)-Furyl-251 5-(2'-CNC.sub.6 H.sub.4)-Furyl-252 5-(4'-ClC.sub.6 H.sub.4)-Furyl-253 5-(3'-ClC.sub.6 H.sub.4)-Furyl-254 5-(2'-ClC.sub.6 H.sub.4)-Furyl-255 4-CH.sub.3 -Furyl-256 4-C.sub.6 H.sub.5 -Furyl-257 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-258 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-259 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-260 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-261 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-262 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-263 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-264 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-265 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-266 4-(4'-CNC.sub.6 H.sub.4)-Furyl-267 4-(3'-CNC.sub.6 H.sub.4)-Furyl-268 4-(2'-CNC.sub.6 H.sub.4)-Furyl-269 4-(4'-ClC.sub.6 H.sub.4)-Furyl-270 4-(3'-ClC.sub.6 H.sub.4)-Furyl-271 4-(2'-ClC.sub.6 H.sub.4)-Furyl-272 Thienyl-273 5-CH.sub.3 -Thienyl-274 5-C.sub.6 H.sub.5 -Thienyl-275 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-276 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-277 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-278 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-279 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-280 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-281 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-282 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-283 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-284 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-285 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-286 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-287 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-288 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-289 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-290 4-CH.sub.3 -Thienyl-291 4-C.sub.6 H.sub.5 -Thienyl-292 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-293 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-294 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-295 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-296 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-297 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-298 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-299 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 Pyridinyl-3______________________________________ TABLE 30__________________________________________________________________________Selected physical data of some compounds IR (cm.sup.-) orNo. Compound .sup.1 H-NMR (ppm) m.p__________________________________________________________________________ ##STR241## 812 ##STR242## 603 ##STR243## 3.85 (s, broad, 3H); 3.7 (s, broad, 3H)4 ##STR244## 3.85 (s, broad, 3H); 3.75 (s, broad, 3H)5 ##STR245## 3.75 (2s, broad, each 3H)6 ##STR246## 917 ##STR247## 3.8 (s, 3H); 3.75 (s, broad, 3H)8 ##STR248## 3.85 (s, 3H); 3.8 (s, broad,__________________________________________________________________________ 3H) TABLE 31______________________________________ ##STR249##I: R.sup.1 = CH.sub.3, X = CH.sub.3II: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3III: R.sup.1 = CH.sub.3, X = ClIV: R.sup.1 = C.sub.2 H.sub.5, X = ClNo. B______________________________________ 1 2-Pyridyl 2 3-Trifluoromethyl-2-Pyridyl 3 5-Trifluoromethyl-2-Pyridyl 4 3,5-Bis-(trifluoromethyl)-2-Pyridyl 5 3,5-Dichloro-2-Pyridyl 6 3-Chloro-5-trifluoromethyl-2-Pyridyl 7 3,5-Dichloro-2-Pyridyl 8 2-Chloro-4-trifluoromethylphenyl 9 2-Benzothiazolyl10 5-Chloro-1-methyl-2-benzimidazolyl11 2-Benzoxazolyl12 1-Methyl-5-trifluoromethylimidazo- �5,4-a!-Pyridin-2-yl13 5-Chloro-2-Pyrimidinyl14 4-Methyl-5-Phenyl-2-thiazolin-2-yl15 4-Methyl-5-Phenyl-2-oxazolin-2-yl16 7-Trifluoromethyl-4-quinolinyl______________________________________ TABLE 57______________________________________Selected physical data of some compounds ##STR250## mp .sup.1 H-NMR (ppm)No. X T.sub.m (.degree.C.) or IR (cm.sup.-1)______________________________________1 Cl 2-CH.sub.3 3.8 (s, broad, 6H)2 Cl 2,5-(CH.sub.3).sub.2 3.8 (s, broad, 6H)3 Cl 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 4.0 (s, 3H); 3.8 (s, broad, 6H)4 Cl 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO- 3.8 (s, broad, 6H) Allyl5 CH.sub.3 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 4.0 (s, 3H); 3.75 (s, broad, 6H)6 CH.sub.3 2-CH.sub.3 3.75 (s, broad, 6H)7 CH.sub.3 2,5-(CH.sub.3).sub.2 3.75 (s, broad, 6H)8 CH.sub.3 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO- 3.75 (s, broad, Allyl 6H)______________________________________

Example 11

2-(2'-Methylphenoxymethyl)-trichloroacetanilide (Table 38, No. 1)

a) 2-(2'-Methylphenoxymethyl)-nitrobenzene

75 g (0.347 mol) of 2-nitrobenzyl bromide, 37 g (0.342 mol) of o-cresol and 56 g (0.405 mol) of potassium carbonate in 500 ml of dimethylformamide is stirred for 5 hours at room temperature (20.degree. C.). The reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The ether phase is dried and evaporated down. The crystalline residue is stirred with methanol and suction filtered. There is obtained 73 g (0.300 mol=88%) of the title compound as a colorless solid.

Mp=83.degree. C. .sup.1 H-NMR, (CDCl.sub.3 ; .delta. (ppm)): 8.15 (d, 1H, I=8 Hz, aromatic); 7.95 (d, 1H, I=8 Hz, aromatic); 7.7 (t, 1H, I=8 Hz, aromatic); 7.45 (t, 1H, I=8 Hz, aromatic); 7.15 (m, 2H, aromatic); 6.9 (m, 2H, aromatic); 5.45 (s, 2H, O--CH.sub.2); 2.35 (s, 3H, CH.sub.3)

b) 2-(2'-Methylphenoxymethyl)-aniline

75 g (0.308 mol) of 2-(2'-methylphenoxymethyl)-nitrobenzene (Example 11a) and 10 g of 5% Pt/C (platinum adsorbed on activated carbon) in 50 ml of methanol are stirred vigorously under a hydrogen blanket for 2 hours. A further 2 g of 5% Pt/C is added and the mixture is stirred overnight. The catalyst is filtered off and replaced by 10 g of fresh catalyst. The mixture is stirred overnight and suction filtered, and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 61 g (0.286 mol=93%) of the title compound as a colorless solid.

Mp=56.degree. C. .sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 7.2 (m, 4H, aromatic); 6.95 (d, 1H, I=8 Hz, aromatic); 6.9 (t, 1H, I=6 Hz, aromatic); 6.7 (m, 2H, aromatic); 5.0 (s, 2H, O--CH.sub.2); 4.05 (s, broad, 2H, NH.sub.2); 2.2 (s, 3H, CH.sub.3)

c) 2-(2'-Methylphenoxymethyl)-trichloroacetanilide (Table 38, No. 1)

At 10.degree.-15.degree. C., a solution of 6 g of 2-(2'-methylphenoxymethyl)-aniline (Example 1b) in 20 ml of CH.sub.2 Cl.sub.2 is added to a mixture of 6.6 g (36 mmol) of trichloroacetyl chloride and 3 g (38 mmol) of pyridine in 50 ml of CH.sub.2 Cl.sub.2. The mixture is stirred for 1 hour at room temperature, and then extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is suction filtered over silica gel and the filtrate which is obtained is evaporated down. The residue crystallizes and is stirred with hexane. There is obtained 7.9 g (22 mmol=78%) of the title compound as a crystalline solid (mp=128.degree. C.).

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm)): 9.6 (s, broad, 1H, NH); 8.1 (d, 1H, I=8 Hz, phenyl); 7.5 (t, broad, 1H, phenyl); 7.4 (d, broad, 1H, phenyl); 7.2 (m, 3H, phenyl); 6.95 (m, 2H, phenyl); 5.1 (s, 2H, OCH.sub.2); 2.2 (s, 3H, CH.sub.3)

Example 12

N-Methyl-N'-(2-(2'-methylphenoxymethyl)-phenyl)-urea (Table 7, No. 2)

In a laboratory autoclave, about 10 ml of methylamine is added to 2 g (5.5 mmol) of the trichloroacetanilide from Example 1c. The autoclave is then closed and the reaction mixture is heated for about 6 hours at 80.degree. C. The reaction mixture is cooled and the autoclave opened. The methylamine is allowed to evaporate off and the solid residue is stirred with methyl tert-butyl ether. The insoluble solid is filtered off and dried under reduced pressure. There is obtained 1.4 g (5.2 mmol=94%) of the title compound as a crystalline solid (mp=144.degree. C.).

.sup.1 H-NMR (DMSO-d.sub.6 ; .delta. (ppm)): 8.05 (s, 1H, NH); 7.8 (d, 1H, I=8 Hz, phenyl); 7.4 (d, 1H, I=8 Hz, phenyl); 6.8-7.3 (m, 6H, phenyl); 6.7 (s, 1H, NH); 5.1 (s, 2H, OCH.sub.2); 2.65 (d, 3H, I=5 Hz, N--CH.sub.3); 2.2 (s, 3H, CH.sub.3)

Example 13

2-(2'-Methylphenoxymethyl)-propionyl anilide (Table 38, No. 3)

A mixture of 3 g (14.1 mmol) of the aniline from Example 11b, 1.35 g (17 mmol) of pyridine and 1.4 g (15.5 mmol) of propionyl chloride in 30 ml of methylene chloride is stirred for 1 hour at room temperature. The reaction mixture is then extracted with diluted hydrochloric acid and water, dried over MgSO.sub.4 and evaporated down. There is obtained 3.8 g (quantitative yield) of the title compound.

.sup.1 H-NMR (COCl.sub.3 ; .delta. (ppm)): 8.25 (s, broad, 1H, NH); 8.15 (d, 1H, I=8 Hz, phenyl); 6.9-7.5 (m, 7H, phenyl); 5.1 (s, 2H, OCH.sub.2); 2.35 (q, 2H, I=8 Hz, CH.sub.2); 2.25 (s, 3H, CH.sub.3); 1.2 (t, 3H, I=8 Hz, CH.sub.3)

Example 14

N-Propionyl-2-(2'-methylphenoxymethyl)-propionyl anilide (Table 38, No. 4)

0.41 g (17.1 mmol) of sodium hydride is added in portions to 3.8 g (14 mmol) of the propionyl anilide from Example 13 in 40 ml of dimethylformamide. Upon completion of gas evolution 1.4 g (15.9 mmol) of propionyl chloride is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 2.6 g (8 mmol=57%) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3): .delta. (ppm): 7.6 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.15 (m, 3H, phenyl); 6.85 (m, 2H, phenyl); 4.85 (m, 2H, OCH.sub.2); 2.6 (m, 4H, 2.times.CH.sub.2); 2.2 (s, 3H, CH.sub.3); 1.1 (t, 6H, I=8 Hz, 2.times.CH.sub.3)

Example 15

N-Methyl-2-(2'-methylphenoxymethyl)-propionyl anilide (Table 38, No. 5)

0.45 g (19 mmol) of sodium hydride is added in portions to 4.0 g (14.8 mmol) of the propionyl anilide from Example 13 in 50 ml of dimethylformamide. Upon completion of gas evolution 3.0 g (21 mmol) of methyl iodide is added and the mixture is stirred for 2 hours at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. The residue crystallizes and is stirred with hexane. There is obtained 3.7 g (11.7 mmol=90%) of the title compound as a colorless solid (mp=80.degree. C.).

.sup.1 H-NMR (CDCl.sub.3 ; .delta. (ppm): 5 7.7 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.2 (m, 3H, phenyl); 6.9 (m, 2H, phenyl); 5.0 (s, 2H, OCH.sub.2); 3.2 (s, 3H, N--CH.sub.3); 2.2 (s, 3H, CH.sub.3); 2.0 (m, 2H, CH.sub.2); 1.0 (t, 3H, I=8 Hz, CH.sub.3)

Example 19

N-Methyl-2-(2'-methylphenoxymethyl)-acetanilide

a) N-Methyl-2-(2'-methylphenoxymethyl)-aniline

A mixture of 5 g (23 mmol) of 2-(2'-methylphenoxymethyl)-aniline (Example 1b), 5 g (36 mmol) of K.sub.2 CO.sub.3 and 3.4 g (24 mmol) of methyl iodide in 50 ml of dimethylformamide is stirred overnight at room temperature. The reaction mixture is diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. The residue is purified chromatographically using mixtures of hexane and methylene chloride. There is obtained 3.0 g (70% purity, about 40% yield) of the title compound as a yellow oil.

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 6.6-7.4 (m, 8H, phenyl); 5.0 (s, 2H, OCH.sub.2); 4.6 (s, broad, 1H, NH); 2.9 (d, 3H, N--CH.sub.3); 2.2 (s, 3H, CH.sub.3).

b) N-Methyl-2-(2'-methylphenoxymethyl)-acetanilide (Table 7, No. 9)

3 g (approx. 9.3 mmol) of N-methyl-2-(2'-methylphenoxymethyl)-aniline (from Example 5a) is added to a mixture of 1.6 g (16 mmol) of acetoanhydride and 1.3 g (16 mmol) of pyridine in 20 ml of methylene chloride. The mixture is stirred for 1 hour at room temperature and is then extracted with dilute hydrochloric acid and water. The organic phase is evaporated down and the residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 2 g (80%) of the title compound as a colorless solid (mp=76.degree. C.).

.sup.1 H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.2 (m, 3H, phenyl); 6.9 (m, 2H, phenyl); 5.0 (s, 2H, OCH.sub.2); 3.25 (s, 3H, CH.sub.3); 2.25 (s, 3H, CH.sub.3); 1.8 (s, 3H, CH.sub.3).

The compounds listed in the tables below may be prepared correspondingly.

Compound I from Table 32, No. 1 has for example the following structural formula: ##STR251##

The compounds described in the following tables may be prepared analogously.

TABLE 32______________________________________ ##STR252##I: R.sup.1 = H, Z = C.sub.2 H.sub.5II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5VI: R.sup.1 = CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5VIII: R.sup.1 = H, Z = NH(CH.sub.3)IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4 -COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-COCH.sub.3303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-COCH.sub.2 CH.sub.2 CH.sub.3305 2-Me-4-COCH(CH.sub.3).sub.2306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-COCH.sub.3308 2,5-Me.sub.2 -4-COCH.sub.2 CH.sub.3309 2,5-Me.sub.2 -4-CH.sub.2 CH.sub.2 COCH.sub.3310 2,5-Me.sub.2 -4-COCH(CH.sub.3).sub.2311 2-Cl-4-CHO312 2-Cl-4-COCH.sub.3313 2-Cl-4-COCH.sub.2 CH.sub.3314 2-Cl-4-COCH(CH.sub.3).sub.2315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-COCH.sub.3317 2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.3318 2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.2 CH.sub.3319 2,5-Cl.sub.2 -4-COCH(CH.sub.3).sub.2320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2 -CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Propargyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-C-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CN-OCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 33______________________________________ ##STR253##I: R.sup.1 = H, Z = C.sub.2 H.sub.5II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5VI: R.sup.1 = CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5VIII: R.sup.1 = H, Z = NH(CH.sub.3)IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C6H5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-COCH.sub.3303 2-Me-4-COCH.sub.2 CH.sub.3304 2-Me-4-COCH.sub.2 CH.sub.2 CH.sub.3305 2-Me-4-COCH(CH.sub.3).sub.2306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-COCH.sub.3308 2,5-Me.sub.2 -4-COCH.sub.2 CH.sub.3309 2,5-Me.sub.2 -4-CH.sub.2 CH.sub.2 COCH.sub.3310 2,5-Me.sub.2 -4-COCH(CH.sub.3).sub.2311 2-Cl-4-CHO312 2-Cl-4-COCH.sub.3313 2-Cl-4-COCH.sub.2 CH.sub.3314 2-Cl-4-COCH(CH.sub.3).sub.2315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-COCH.sub.3317 2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.3318 2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.2 CH.sub.3319 2,5-Cl.sub.2 -4-COCH(CH.sub.3).sub.2320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)CH.sub.3339 3-C(NO-Propargyl)CH.sub.3340 4-C(NO-Propargyl)CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'CH.sub.3 C.sub.6 H.sub.4)406 2-(3'CH.sub.3 C.sub.6 H.sub.4)407 2-(4'CH.sub.3 C.sub.6 H.sub.4)408 3-(2'CH.sub.3 C.sub.6 H.sub.4)409 3-(3'CH.sub.3 C.sub.6 H.sub.4)410 3-(4'CH.sub.3 C.sub.6 H.sub.4)411 4-(2'CH.sub.3 C.sub.6 H.sub.4)412 4-(3'CH.sub.3 C.sub.6 H.sub.4)413 4-(4'CH.sub.3 C.sub.6 H.sub.4)414 2-(2'CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyll))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chlorallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chlorallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 34______________________________________ ##STR254##I: R.sup.1 = H, Z = C.sub.2 H.sub.5II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5VI: R.sup.1 = CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5VIII: R.sup.1 = H, Z, = NH(CH.sub.3)IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = CH.sub.3)XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.3 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-COCH.sub.3303 2-Me-4-COCH.sub.2 CH.sub.3304 2-Me-4-COCH.sub.2 CH.sub.2 CH.sub.3305 2-Me-4-COCH(CH.sub.3).sub.2306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-COCH.sub.3308 2,5-Me.sub.2 -4-COCH.sub.2 CH.sub.3309 2,5-Me.sub.2 -4-CH.sub.2 CH.sub.2 COCH.sub.3310 2, 5-Me.sub.2 -4-COCH(CH.sub.3)2311 2-Cl-4-CHO312 2-Cl-4-COCH.sub.3313 2-Cl-4-COCH.sub.2 CH.sub.3314 2-Cl-4-COCH(CH.sub.3)2315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-COCH.sub.3317 2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.3318 2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.2 CH.sub.3319 2,5-Cl.sub.2 -4-COCH(CH.sub.3)2320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NCC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)CH.sub.3339 3-C(NO-Propargyl)CH.sub.3340 4-C(NO-Propargyl)CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.4)374 2,5-(CH.sub.3).sub.2-4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2-4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2-4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 35______________________________________ ##STR255##I: R.sup.1 = H, Z = C.sub.2 H.sub.5II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5VI: R.sup.1 = CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5VIII: R.sup.1 = H, Z = NH(CH.sub.3)IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-Cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-COCH.sub.2 CH.sub.3304 2-Me-4-COCH.sub.2 CH.sub.2 CH.sub.3305 2-Me-4-COCH(CH.sub.3).sub.2306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-COCH.sub.3308 2,5-Me.sub.2 -4-COCH.sub.2 CH.sub.3309 2,5-Me.sub.2 -4-CH.sub.2 CH.sub.2 COCH.sub.3310 2,5-Me.sub.2 -4-COCH(CH.sub.3).sub.2311 2-Cl-4-CHO312 2-Cl-4-COCH.sub.3313 2-Cl-4-COCH.sub.2 CH.sub.3314 2-Cl-4-COCH(CH.sub.3).sub.2315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-COCH.sub.3317 2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.3318 2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.2 CH.sub.3319 2,5-Cl.sub.2 -4-COCH(CH.sub.3).sub.2320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2;5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Propargyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 36______________________________________ ##STR256##I: R.sup.1 = H, Z = C.sub.2 H.sub.5II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5VI: R.sup.1 = CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5VIII: R.sup.1 = H, Z = NH(CH.sub.3)IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)No. X.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-COCH.sub.2 CH.sub.3304 2-Me-4-COCH.sub.2 CH.sub.2 CH.sub.3305 2-Me-4-COCH(CH.sub.3).sub.2306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-COCH.sub.3308 2,5-Me.sub.2 -4-COCH.sub.2 CH.sub.3309 2,5-Me.sub.2 -4-CH.sub.2 CH.sub.2 COCH.sub.3310 2,5-Me.sub.2 -4-COCH(CH.sub.3).sub.2311 2-Cl-4-CHO312 2-Cl-4-COCH.sub.3313 2-Cl-4-COCH.sub.2 CH.sub.3314 2-Cl-4-COCH(CH.sub.3).sub.2315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-COCH.sub.3317 2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.3318 2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.2 CH.sub.3319 2,5-Cl.sub.2 -4-COCH(CH.sub.3).sub.2320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Propargyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FFC.sub.6 H.sub.4)484 4-O-(2'-Fab,4 C.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'______________________________________ TABLE 37______________________________________ ##STR257##I: R.sup.1 = H, Z = C.sub.2 H.sub.5II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5V: R.sup.1 Propargyl, Z = C.sub.2 H.sub.5VI: R.sup.1 CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5VIII: R.sup.1 = H, Z = NH(CH.sub.3)IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)No. B______________________________________1 Pyrrolyl-32 NCH.sub.3 -Pyrrolyl-33 NC.sub.6 H.sub.5 -Pyrrolyl-34 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-35 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-36 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-37 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-38 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-39 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-310 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-311 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-312 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-313 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-314 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-315 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-316 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-317 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-318 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-319 Pyrrolyl-220 NCH.sub.3 -Pyrrolyl-221 NC.sub.6 H.sub.5 -Pyrrolyl-222 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-223 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-224 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-225 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-226 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-227 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-228 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-229 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-230 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-231 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-232 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-233 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-234 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-235 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-236 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-237 Furyl-238 5-CH.sub.3 -Furyl-239 5-C.sub.6 H.sub.5 -Furyl-240 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-241 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-242 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-243 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-244 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-245 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-246 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-247 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-248 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-249 5-(4'-CNC.sub.6 H.sub.4)-Furyl-250 5-(3'-CNC.sub.6 H.sub.4)-Furyl-251 5-(2'-CNC.sub.6 H.sub.4)-Furyl-252 5-(4'-ClC.sub.6 H.sub.4)-Furyl-253 5-(3'-ClC.sub.6 H.sub.4)-Furyl-254 5-(2'-ClC.sub.6 H.sub.4)-Furyl-255 4-CH.sub.3 -Furyl-256 4-C.sub.6 H.sub.5 -Furyl-257 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-258 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-259 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-260 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-261 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-262 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-263 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-264 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-265 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-266 4-(4'-CNC.sub.6 H.sub.4)-Furyl-267 4-(3'-CNC.sub.6 H.sub.4)-Furyl-268 4-(2'-CNC.sub.6 H.sub.4)-Furyl-269 4-(4'-ClC.sub.6 H.sub.4)-Furyl-270 4-(3'-ClC.sub.6 H.sub.4)-Furyl-271 4-(2'-ClC.sub.6 H.sub.4)-Furyl-272 Thienyl-273 5-CH.sub.3 -Thienyl-274 5-C.sub.6 H.sub.5 -Thienyl-275 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-276 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-277 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-278 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-279 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-280 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-281 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-282 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-283 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-284 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-285 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-286 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-287 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-288 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-289 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-290 4-CH.sub.3 -Thienyl-291 4-C.sub.6 H.sub.5 -Thienyl-292 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-293 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-294 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-295 4-(4'-CH.sub.3 O-C.sub.6 H.sub.4)-Thienyl-296 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-297 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-298 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-299 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4) Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Is6thiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 3-CH.sub.3 -Oxazolyl-4234 3-C.sub.6 H.sub.5 -Oxazolyl-4235 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 3-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 3-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 3-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 3-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 3-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 3-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2______________________________________ TABLE 38______________________________________Selected physical data of some compounds IR (cm.sup.-1) or .sup.1 H-NMR mpNo. Compound (ppm) (.degree.C.)______________________________________ ##STR258## 1282 ##STR259## 1443 ##STR260##4 ##STR261##5 ##STR262## 806 ##STR263## 757 ##STR264## 1888 ##STR265## 1159 ##STR266## 7610 ##STR267## 9611 ##STR268## 3.3 (s, 3H); 2.25 (s, 3H)______________________________________ TABLE 58__________________________________________________________________________Selected physical data of some compounds ##STR269## IR (cm.sup.-1) or .sup.1 H-NMR mpNo. X.sub.m R.sup.1 (ppm) (.degree.C.)__________________________________________________________________________1 2-CH.sub.3 H 1202 2-CH.sub.3 CH.sub.3 oil3 2-CH.sub.3 C.sub.2 H.sub.5 oil4 2-CH.sub.3 Allyl oil5 2-CH.sub.3 Propargyl oil6 2-CH.sub.3 CH.sub.2 OCH.sub.3 oil7 2,5-(CH.sub.3).sub.2 H 1708 2,5-(CH.sub.3).sub.2 CH.sub.3 oil9 2,5-(CH.sub.3).sub.2 C.sub.2 H.sub.5 oil10 2,5-(CH.sub.3).sub.2 Allyl oil11 2,5-(CH.sub.3).sub.2 Propargyl oil12 2,5-(CH.sub.3).sub.2 CH.sub.2 OCH.sub.3 oil13 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 H 12514 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 CH.sub.3 oil15 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 C.sub.2 H.sub.5 oil16 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 Allyl 8717 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 Propargyl oil18 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 CH.sub.2 OCH.sub.3 oil19 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl H 8520 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl CH.sub.3 oil21 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl C.sub.2 H.sub.5 oil22 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl Allyl 8723 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl Propargyl oil24 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl CH.sub.2 OCH.sub.3 oil__________________________________________________________________________ TABLE 59______________________________________Selected physical data of some compounds ##STR270## IR (cm.sup.-1) or .sup.1 H-NMR mpNo. X.sub.m R.sup.1 (ppm) (.degree.C.)______________________________________1 4-CH.sub.3 H 1182 4-CH.sub.3 CH.sub.3 oil3 4-CH.sub.3 C.sub.2 H.sub.5 oil4 4-CH.sub.3 Allyl oil5 4-CH.sub.3 Propargyl oil6 4-CH.sub.3 CH.sub.2 OCH.sub.3 oil7 3,5-Cl.sub.2 H 1608 3,5-Cl.sub.2 CH.sub.3 oil9 3,5-Cl.sub.2 C.sub.2 H.sub.5 oil10 3,5-Cl.sub.2 Allyl 8511 3,5-Cl.sub.2 Propargyl oil12 3,5-Cl.sub.2 CH.sub.2 OCH.sub.3 oil______________________________________ TABLE 39______________________________________ ##STR271##No. X R.sup.1 Z A______________________________________1 H H CH.sub.3 CH.sub.2 O2 H H CH.sub.3 CH.sub.2 ONC (CH.sub.3)3 H H CH.sub.3 CHCH4 H H NH.sub.2 CH.sub.2 O5 H H NH.sub.2 CH.sub.2 ONC(CH.sub.3)6 H H NH.sub.2 CHCH7 H H N(CH.sub.3).sub.2 CH.sub.2 O8 H H N(CH.sub.3).sub.2 CH.sub.2 ONC(CH.sub.3)9 H H N(CH.sub.3).sub.2 CHCH10 H H CCl.sub.3 CH.sub.2 O11 H H CCl.sub.3 CH.sub.2 ONC(CH.sub.3)12 H H CCl.sub.3 CHCH13 H H CF.sub.3 CH.sub.2 O14 H H CF.sub.3 CH.sub.2 ONC(CH.sub.3)15 H H CF.sub.3 CHCH16 H Propargyl CH.sub.3 CH.sub.2 O17 H Propargyl CH.sub.3 CH.sub.2 ONC(CH.sub.3)18 H Propargyl CH.sub.3 CHCH19 H Propargyl NH.sub.2 CH.sub.2 O20 H Propargyl NH.sub.2 CH.sub.2 ONC(CH.sub.3)21 H Propargyl NH.sub.2 CHCH22 H Propargyl N(CH.sub.3).sub.2 CH.sub.2 O23 H Propargyl N(CH.sub.3).sub.2 CH.sub.2 ONC(CH.sub.3)24 H Propargyl N(CH.sub.3).sub.2 CHCH25 H Propargyl CCl.sub.3 CH.sub.2 O26 H Propargyl CCl.sub.3 CH.sub.2 ONC(CH.sub.3)27 H Propargyl CCl.sub.3 CHCH28 H Propargyl CF.sub.3 CH.sub.2 O29 H Propargyl CF.sub.3 CH.sub.2 ONC(CH.sub.3)30 H Propargyl CF.sub.3 CHCH31 CH.sub.3 H CH.sub.3 CH.sub.2 O32 CH.sub.3 H CH.sub.3 CH.sub.2 ONC(CH.sub.3)33 CH.sub.3 H CH.sub.3 CHCH34 CH.sub.3 H NH.sub.2 CH.sub.2 O35 CH.sub.3 H NH.sub.2 CH.sub.2 ONC(CH.sub.3)36 CH.sub.3 H NH.sub.2 CHCH37 CH.sub.3 H N(CH.sub.3).sub.2 CH.sub.2 O38 CH.sub.3 H N(CH.sub.3).sub.2 CH.sub.2 ONC(CH.sub.3)39 CH.sub.3 H N(CH.sub.3).sub.2 CHCH40 CH.sub.3 H CCl.sub.3 CH.sub.2 O41 CH.sub.3 H CCl.sub.3 CH.sub.2 ONC(CH.sub.3)42 CH.sub.3 H CCl.sub.3 CHCH43 CH.sub.3 H CF.sub.3 CH.sub.2 O44 CH.sub.3 H CF.sub.3 CH.sub.2 ONC(CH.sub.3)45 CH.sub.3 H CF.sub.3 CHCH46 CH.sub.3 Propargyl CH.sub.3 CH.sub.2 O47 CH.sub.3 Propargyl CH.sub.3 CH.sub.2 ONC(CH.sub.3)48 CH.sub.3 Propargyl CH.sub.3 CHCH49 CH.sub.3 Propargyl NH.sub.2 CH.sub.2 O50 CH.sub.3 Propargyl NH.sub.2 CH.sub.2 ONC(CH.sub.3)51 CH.sub.3 Propargyl NH.sub.2 CHCH52 CH.sub.3 Propargyl N(CH.sub.3).sub.2 CH.sub.2 O53 CH.sub.3 Propargyl N(CH.sub.3).sub.2 CH.sub.2 ONC(CH.sub.3)54 CH.sub.3 Propargyl N(CH.sub.3).sub.2 CHCH55 CH.sub.3 Propargyl CCl.sub.3 CH.sub.2 O56 CH.sub.3 Propargyl CCl.sub.3 CH.sub.2 ONC(CH.sub.3)57 CH.sub.3 Propargyl CCl.sub.3 CHCH58 CH.sub.3 Propargyl CF.sub.3 CH.sub.2 O59 CH.sub.3 Propargyl CF.sub.3 CH.sub.2 ONC(CH.sub.3)60 CH.sub.3 Propargyl CF.sub.3 CHCH61 Cl H CH.sub.3 CH.sub.2 O62 Cl H CH.sub.3 CH.sub.2 ONC(CH.sub.3)63 Cl H CH.sub.3 CHCH64 Cl H NH.sub.2 CH.sub.2 O65 Cl H NH.sub.2 CH.sub.2 ONC(CH.sub.3)66 Cl H NH.sub.2 CHCH67 Cl H N(CH.sub.3).sub.2 CH.sub.2 O68 Cl H N(CH.sub.3).sub.2 CH.sub.2 ONC(CH.sub.3)69 Cl H N(CH.sub.3).sub.2 CHCH70 Cl H CCl.sub.3 CH.sub.2 O71 Cl H CCl.sub.3 CH.sub.2 ONC(CH.sub.3)72 Cl H CCl.sub.3 CHCH73 Cl H CF.sub.3 CH.sub.2 O74 Cl H CF.sub.3 CH.sub.2 ONC(CH.sub.3)75 Cl H CF.sub.3 CHCH76 Cl Propargyl CH.sub.3 CH.sub.2 O77 Cl Propargyl CH.sub.3 CH.sub.2 ONC(CH.sub.3)78 Cl Propargyl CH.sub.3 CHCH79 Cl Propargyl NH.sub.2 CH.sub.2 O80 CI Propargyl NH.sub.2 CH.sub.2 ONC(CH.sub.3)81 Cl Propargyl NH.sub.2 CHCH82 Cl Propargyl N(CH.sub.3).sub.2 CH.sub.2 O83 Cl Propargyl N(CH.sub.3).sub.2 CH.sub.2 ONC(CH.sub.3)84 Cl Propargyl N(CH.sub.3).sub.2 CHCH85 Cl Propargyl CCl.sub.3 CH.sub.2 O86 Cl Propargyl CCl.sub.3 CH.sub.2 ONC(CH.sub.3)87 Cl Propargyl CCl.sub.3 CHCH88 Cl Propargyl CF.sub.3 CH.sub.2 O89 Cl Propargyl CF.sub.3 CH.sub.2 ONC(CH.sub.3)90 Cl Propargyl CF.sub.3 CHCH______________________________________ TABLE 40______________________________________ ##STR272##I: R.sup.1 = H, Z = C.sub.2 H.sub.5II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5VI: R.sup.1 = CH.sub.2OCH.sub.3, Z = C.sub.2 H.sub.5VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5VIII: R.sup.1 = H, Z = NH(CH.sub.3)IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)No. B______________________________________1 2-Pyridyl2 3-Trifluoromethyl-2-pyridyl3 5-Trifluoromethyl-2-pyridyl4 3,5-Bis-(trifluoromethyl)-2-pyridyl5 3,5-Dichloro-2-pyridyl6 3-chloroo-5-trifluoromethyl-2-pyridyl7 3,5-Dichloro-2-pyridyl8 2-Chloroo-4-trifluoromethylphenyl9 2-Benzothiazolyl10 5-Chloroo-1-methyl-2-benzimidazolyl11 2-Benzoxazolyl12 1-Methyl-5-trifluoromethylimidazo- �5,4-a)!-pyridin-2-yl13 5-Chloroo-2-pyrimidinyl14 4-Methyl-5-phenyl-2-thiazolin-2-yl15 4-Methyl-5-phenyl-2-oxazolin-2-yl16 7-Trifluoromethyl-4-quinolinyl______________________________________

Example 16

Methyl N-�2-(3", 4"-dichlorophenyl-1'-methyliminooxy-methyl-4')-6-methylphenyl!-carbamate (Table 47, No. 2)

a) 2-(Methanesulfonyloxymethyl)-6-methyl-nitrobenzene

At 10.degree.-15.degree. C., 27 g (0.23 mol) of methanesulfonyl chloride dissolved in 20 ml of CH.sub.2 Cl.sub.2 is dripped into a mixture of 34 g (0.2 mol) of 3-methyl-2-nitrobenzyl alcohol and 27 g (0.27 mol) of triethylamine in 100 ml of CH.sub.2 Cl.sub.2. The reaction mixture is stirred for 1 hour at room temperature and is then extracted with water. The organic phase is dried over MgSO.sub.4 and evaporated down. There is obtained as residue 48 g of the title compound as a yellow oil, containing about 10% of the corresponding benzyl chloride as impurity. The crude product is used for the next reaction without any further purification.

.sup.1 H-NMR(COCl.sub.3 ; .delta. bin ppm): 7.3-7.6 (m, 3H, phenyl); 5.3 (S, 2H, OCH.sub.2); 3.0 (S, 3H, CH.sub.3 -SO.sub.3); 2.4 (S, 3H, CH.sub.3)

b) 2-(3", 4"-Dichlorophenyl-1'-methyl-iminooxymethyl-4')-6-methyl-nitrobenzene

At room temperature, 1.8 g (75 mmol) of sodium hydride is added in portions to a solution of 13 g (64 mmol) of 3,4-dichloroacetophenonoxime in 100 ml of dimethylformamide. Upon conclusion of gas evolution, a solution of 16 g (65 mmol) of the mesylate from Example 1a in 30 ml of dimethylformamide is dripped in at 25.degree.-30.degree. C., and the mixture is then stirred for 1 hour at room temperature. The reaction mixture is diluted with water and the aqueous phase is then extracted three times with methyl tert-butyl ether. The combined organic phases are washed with water, dried over MGSO.sub.4 and evaporated down. The residue crystallizes and is stirred with methanol. The mother liquor is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained a total of 20.4 g (58 mmol=90%) of the title compound as pale yellow crystals.

.sup.1 H-NMR(CDCl.sub.3 ; .delta. in ppm): 7.7 (S, broad, 1H, phenyl); 7.2-7.6 (m, 5H, phenyl); 5.3 (S, 2H, OCH.sub.2); 2.4 (S, 3H, CH.sub.3); 2.2 (S, 3H, CH.sub.3)

c) 2-(3", 4"-Dichlorophenyl-1-methyl-iminooxymethyl-4')-6-methyl-aniline

At 20.degree.-30.degree. C., 53 g of 21.8% strength Na.sub.2 �Fe(CO).sub.4 ! solution (1 kg of the solution contains 633 g of water, 218 g of Na.sub.2 �Fe(CO).sub.4 !, 108 g of Na.sub.2 CO.sub.3 and 41 g of NaOH) is added dropwise to 19 g (52.8 mmol) of the nitrobenzene from Example 16b in 150 ml of methanol. The brown suspension is stirred for 2 hours at room temperature, and the reaction mixture is then diluted with methylene chloride and the mixture is suction filtered using kieselguhr. The residue is again washed with CH.sub.2 Cl.sub.2 and the combined extracts are extracted with water, dried over MgSO.sub.4 and evaporated down. The brown residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 14.3 g (44.3 inmol=82%) of the title compound as a beige solid.

1H-NMR(CDCl.sub.3 ; .delta. in ppm): 7.7 (S, 1H, phenyl); 7.5 (m, 2H, phenyl); 7.1 (t, broad, 2H, phenyl); 6.7 (t, 1H, I=8 Hz, phenyl); 5.2 (S, 2H, OCH.sub.2); 4.15 (S, 2H, NH.sub.2 ; 2.2 (S, 3H, CH.sub.3)

d) Methyl N-�2-(3", 4"-dichlorophenyl-1'-methyl-iminooxymethyl-4'-6-methylphenyl!-carbamate (Table 47, No. 2)

At 20.degree.-30.degree. C., 4.8 g (50 mmol) of methyl chloroformate and subsequently 4.8 g (60 mmol) of pyridine are dripped into a solution of 14.3 g (44 mmol) of the aniline from Example 1c in 150 ml of CH.sub.2 Cl.sub.2. The mixture is stirred overnight at room temperature and is then extracted with dilute hydrochloric acid and water. The reaction mixture is suction filtered using silica gel, dried over MgSO.sub.4 and evaporated down. The residue crystallizes and is stirred with cyclohexane. There is obtained 13.8 g (36 mmol=82%) of the title compound as a colorless solid (mp=109.degree. C.).

.sup.1 H-NMR(CDCl.sub.3 ; .delta. in ppm): 7.8 (S, 1H, phenyl); 7.6 (S, broad, 1H, NH); 7.4 (S, 2H, phenyl); 7.2 (m, 3H, phenyl); 5.2 (S, 2H, OCH.sub.2); 3.8 (S, 3H, OCH.sub.3); 2.3 (S, 3H, CH.sub.3); 2.2 (S, 3H, CH.sub.3)

Example 17

Methyl N-�2-(3", 4"-dichlorophenyl-1'-methyl-iminooxymethyl-4')-6-methylphenyl!-N-propargyl-carbamate (Table 47, No. 13)

At 25.degree.-30.degree. C., 0.15 g (6.3 mmol) of sodium hydride is added in portions to a solution of 1.9 g (5 mmol) of the carbamate from Example 16d in 20 ml of dimethylformamide. When no more gas evolves, 0.75 g (6.3 mmol) of propargyl bromide is added and the whole is stirred overnight at room temperature. The reaction mixture is diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO.sub.4 and evaporated down. There is obtained 1.4 g (3.3 mmol=67%) of the title compound as a yellow oil.

1H-NMR (CDCl.sub.3 ; .delta. in ppm): 7.75 (S, broad, 1H, phenyl); 7.2-7.6 (m, 5H, phenyl); 5.2 (dd, 2H, I=12 Hz, OCH.sub.2); 4.4 (dd, broad, I=16 Hz, NCH.sub.2); (S, 3H, OCH.sub.3); 2.3 (S, 3H, CH.sub.3); 2.25 (S, broad, 1H, C.tbd.CH); 2.2 (S, 3H, CH.sub.3); the .sup.1 H-NMR spectrum also contains signals of about 20% of the amide rotamer.

The compounds described in the following tables may be prepared analogously.

TABLE 41______________________________________ ##STR273##I: R.sup.1 = H, X = CH.sub.3II: R.sup.1 = CH.sub.3, X = CH.sub.3III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3IV: R.sup.1 = Allyl, X = CH.sub.3V: R.sup.1 = Propargyl, X = CH.sub.3VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3VIII: R.sup.1 = H, X = ClIX: R.sup.1 = CH.sub.3, X = ClX: R.sup.1 = C.sub.2 H.sub.5, X = ClXI: R.sup.1 = Allyl, X = ClXII: R.sup.1 = Propargyl, X = ClXIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = ClXIV: R.sup.1 = CO.sub.2 CH.sub.3, X = ClCompound I from Table 41 has for instance the followingstructural formula: ##STR274##No. T.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOn-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOn-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 5-Cl-6-OCH.sub.3______________________________________ TABLE 42______________________________________ ##STR275##I: R.sup.1 = H, X = CH.sub.3II: R.sup.1 = CH.sub.3, X = CH.sub.3III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3IV: R.sup.1 = Allyl, X = CH.sub.3V: R.sup.1 = Propargyl, X = CH.sub.3VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3VIII: R.sup.1 = H, X = ClIX: R.sup.1 = CH.sub.3, X = ClX: R.sup.1 = C.sub.2 H.sub.5, X = ClXI: R.sup.1 = Allyl, X = ClXII: R.sup.1 = Propargyl, X = ClXIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = ClXIV: R.sup.1 = CO.sub.2 CH.sub.3, X = ClNo. B______________________________________ 1 Pyrrolyl-3 2 NCH.sub.3 -Pyrrolyl-3 3 NC.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 NCH.sub.3 -Pyrrolyl-2 21 NC.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CNC.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CNC.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CNC.sub.6 H.sub.4)-Furyl-2 52 5-(4'-ClC.sub.6 H.sub.4)-Furyl-2 53 5-(3'-ClC.sub.6 H.sub.4)-Furyl-2 54 5-(2'-ClC.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CNC.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CNC.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CNC.sub.6 H.sub.4)-Furyl-2 69 4-(4'-ClC.sub.6 H.sub.4)-Furyl-2 70 4-(3'-ClC.sub.6 H.sub.4)-Furyl-2 71 4-(2'-ClC.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-pyrazolyl-4143 3-CH.sub.3 -N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C6H4 -4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazqlyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 3-CH.sub.3 -Oxazolyl-4234 3-C.sub.6 H.sub.5 -Oxazolyl-4235 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 3-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 3-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 3-(2'-CNC.sub.6 H.sub.4)-oxazolyl-4247 3-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 3-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 3-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 1-Naphthyl385 2-Naphthyl______________________________________ TABLE 43______________________________________ ##STR276##I: R.sup.1 = H, X = CH.sub.3II: R.sup.1 = CH.sub.3, X = CH.sub.3III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3IV: R.sup.1 = Allyl, X = CH.sub.3V: R.sup.1 = Propargyl, X = CH.sub.3VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3VIII: R.sup.1 = H, X = ClIX: R.sup.1 = CH.sub.3, X = ClX: R.sup.1 = C.sub.2 H.sub.5, X = ClXI: R.sup.1 = Allyl, X = ClXII: R.sup.1 = Propargyl, X = ClXIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = ClXIV: R.sup.1 = CO.sub.2 CH.sub.3, X = ClNo. T.sub.m______________________________________ 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F.sub.2 6 2,4,6-F.sub.3 7 2,3,4,5,6-F.sub.5 8 2,3-F.sub.2 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl.sub.2 13 2,4-Cl.sub.2 14 2,5-Cl.sub.2 15 2,6-Cl.sub.2 16 3,4-Cl.sub.2 17 3,5-Cl.sub.2 18 2,3,4-Cl.sub.3 19 2,3,5-Cl.sub.3 20 2,3,6-Cl.sub.3 21 2,4,5-Cl.sub.3 22 2,4,6-Cl.sub.3 23 3,4,5-Cl.sub.3 24 2,3,4,6-Cl.sub.4 25 2,3,5,6-Cl.sub.4 26 2,3,4,5,6-Cl.sub.5 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br.sub.2 31 2,5-Br.sub.2 32 2,6-Br.sub.2 33 2,4,6-Br.sub.3 34 2,3,4,5,6-Br.sub.5 35 2-I 36 3-I 37 4-I 38 2,4-I.sub.2 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl.sub.2, 4-Br 66 2-CH.sub.3 67 3-CH.sub.3 68 4-CH.sub.3 69 2,3-(CH.sub.3).sub.2 70 2,4-(CH.sub.3).sub.2 71 2,5-(CH.sub.3).sub.2 72 2,6-(CH.sub.3).sub.2 73 3,4-(CH.sub.3).sub.2 74 3,5-(CH.sub.3).sub.2 75 2,3,5-(CH.sub.3).sub.3 76 2,3,4-(CH.sub.3).sub.3 77 2,3,6-(CH.sub.3).sub.3 78 2,4,5-(CH.sub.3).sub.3 79 2,4,6-(CH.sub.3).sub.3 80 3,4,5-(CH.sub.3).sub.3 81 2,3,4,6-(CH.sub.3).sub.4 82 2,3,5,6-(CH.sub.3).sub.4 83 2,3,4,5,6-(CH.sub.3).sub.5 84 2-C.sub.2 H.sub.5 85 3-C.sub.2 H.sub.5 86 4-C.sub.2 H.sub.5 87 2,4-(C.sub.2 H.sub.5).sub.2 88 2,6-(C.sub.2 H.sub.5).sub.2 89 3,5-(C.sub.2 H.sub.5).sub.2 90 2,4,6-(C.sub.2 H.sub.5).sub.3 91 2-n-C.sub.3 H.sub.7 92 3-n-C.sub.3 H.sub.7 93 4-n-C.sub.3 H.sub.7 94 2-i-C.sub.3 H.sub.7 95 3-i-C.sub.3 H.sub.7 96 4-i-C.sub.3 H.sub.7 97 2,4-(i-C.sub.3 H.sub.7).sub.2 98 2,6-(i-C.sub.3 H.sub.7).sub.2 99 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.4, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-O-CH.sub.2 C.sub.6 H.sub.5178 3-O-CH.sub.2 C.sub.6 H.sub.5179 4-O-CH.sub.2 C.sub.6 H.sub.5180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-NO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-CL242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CB.sub.3).sub.2, 6-F247 2,4-(CB.sub.3).sub.2, 6-Cl248 2,4-(CB.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Propargyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'641 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNOCH.sub.3)645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNOC.sub.2 H.sub.5)646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-n-C.sub.3 H.sub.7)647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-i-C.sub.3 H.sub.7)648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-Allyl)649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-trans-Chloroallyl)650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-Propargyl)651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-n-C.sub.4 H.sub.9)652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNOCH.sub.2 C.sub.6 H.sub.5)653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNOCH.sub.3)654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNOC.sub.2 H.sub.5)655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-n-C.sub.3 H.sub.7)656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-i-C.sub.3 H.sub.7)657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-Allyl)658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-trans-Chloroallyl)659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-Propargyl)660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-n-C.sub.4 H.sub.9)661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNOCH.sub.2 C.sub.6 H.sub.5)662 2-O-n-C.sub.4 H.sub.9663 2-O-i-C.sub.4 H.sub.9664 2-O-s-C.sub.4 H.sub.9665 2-O-t-C.sub.4 H.sub.9666 2-Neopentyloxy667 3-O-n-C.sub.4 H.sub.9668 3-O-i-C.sub.4 H.sub.9669 3-O-s-C.sub.4 H.sub.9670 3-O-t-C.sub.4 H.sub.9671 3-Neopentyloxy672 4-O-n-C.sub.4 H.sub.9673 4-O-i-C.sub.4 H.sub.9674 4-O-s-C.sub.4 H.sub.9675 4-O-t-C.sub.4 H.sub.9676 4-Neopentyloxy677 3-CH.sub.3 -4-OCH.sub.3678 3-CH.sub.3 -4-OC.sub.2 H.sub.5679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9684 3-CH.sub.3 -4-Neopentyloxy685 2-CH.sub.3 -3-OCH.sub.3686 2-CH.sub.3 -4-OCH.sub.3687 2-CH.sub.3 -5-OCH.sub.3688 2-CH.sub.3 -6-OCH.sub.3689 3-CH.sub.3 -4-OCH.sub.3690 3-CH.sub.3 -5-OCH.sub.3691 3-CH.sub.3 -6-OCH.sub.3692 4-CH.sub.3 -5-OCH.sub.3693 4-CH.sub.3 -6-OCH.sub.3694 4-CH.sub.3 -6-OCH.sub.3695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7705 2-Cl-3-OCH.sub.3706 2-Cl-4-OCH.sub.3707 2-Cl-5-OCH.sub.3708 2-Cl-6-OCH.sub.3709 3-Cl-4-OCH.sub.3710 3-Cl-5-OCH.sub.3711 3-Cl-6-OCH.sub.3712 4-Cl-5-OCH.sub.3713 4-Cl-6-OCH.sub.3714 4-Cl-6-OCH.sub.3______________________________________ TABLE 44______________________________________ ##STR277##I: R.sup.1 = H, X = CH.sub.3II: R.sup.1 = CH.sub.3, X = CH.sub.3III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3IV: R.sup.1 = Allyl, X = CH.sub.3V: R.sup.1 = Propargyl, X = CH.sub.3VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3VIII: R.sup.1 = H, X = ClIX: R.sup.1 = CH.sub.3, X = ClX: R.sup.1 = C.sub.2 H.sub.5, X = ClXI: R.sup.1 = Allyl, X = ClXII: R.sup.1 = Propargyl, X = ClXIII: R.sup.1 = CH.sub.2OCH.sub.3, X = ClXIV: R.sup.1 = CO.sub.2 CH.sub.3, X = ClNo. B______________________________________ 1 Pyrrolyl-3 2 NCH.sub.3 -Pyrrolyl-3 3 NC.sub.6 H.sub.5 -Pyrrolyl-3 4 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 5 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 6 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3 7 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 8 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 9 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3 10 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 11 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 12 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3 13 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 14 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 15 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3 16 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 17 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 18 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3 19 Pyrrolyl-2 20 NCH.sub.3 -Pyrrolyl-2 21 NC.sub.6 H.sub.5 -Pyrrolyl-2 22 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 23 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 24 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2 25 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 26 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 27 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2 28 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 29 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 30 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2 31 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 32 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 33 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2 34 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 35 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 36 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2 37 Furyl-2 38 5-CH.sub.3 -Furyl-2 39 5-C.sub.6 H.sub.5 -Furyl-2 40 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 41 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 42 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 43 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 44 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 45 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 46 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 47 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 48 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 49 5-(4'-CNC.sub.6 H.sub.4)-Furyl-2 50 5-(3'-CNC.sub.6 H.sub.4)-Furyl-2 51 5-(2'-CNC.sub.6 H.sub.4)-Furyl-2 52 5-(4'-ClC.sub.6 H.sub.4)-Furyl-2 53 5-(3'-ClC.sub.6 H.sub.4)-Furyl-2 54 5-(2'-ClC.sub.6 H.sub.4)-Furyl-2 55 4-CH.sub.3 -Furyl-2 56 4-C.sub.6 H.sub.5 -Furyl-2 57 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 58 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 59 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2 60 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 61 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 62 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2 63 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 64 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 65 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2 66 4-(4'-CN-C.sub.6 H.sub.4)-Furyl-2 67 4-(3'-CN-C.sub.6 H.sub.4)-Furyl-2 68 4-(2'-CN-C.sub.6 H.sub.4)-Furyl-2 69 4-(4'-ClC.sub.6 H.sub.4)-Furyl-2 70 4-(3'-ClC.sub.6 H.sub.4)-Furyl-2 71 4-(2'-ClC.sub.6 H.sub.4)-Furyl-2 72 Thienyl-2 73 5-CH.sub.3 -Thienyl-2 74 5-C.sub.6 H.sub.5 -Thienyl-2 75 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 76 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 77 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 78 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 79 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 80 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 81 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 82 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 83 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 84 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2 85 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2 86 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2 87 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2 88 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2 89 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2 90 4-CH.sub.3 -Thienyl-2 91 4-C.sub.6 H.sub.5 -Thienyl-2 92 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 93 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 94 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2 95 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 96 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 97 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2 98 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2 99 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CN-C.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CN-C.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CN-C.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Chloroisoxazolyl-5190 3-(4'-CN-C.sub.6 H.sub.4)-Chloroisoxazolyl-5191 3-(3'-CN-C.sub.6 H.sub.4)-Chloroisoxazolyl-5192 3-(2'-CN-C.sub.6 H.sub.4)-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 3-CH.sub.3 -Oxazolyl-5234 3-C.sub.6 H.sub.5 -Oxazolyl-5235 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-5236 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-5237 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-5238 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-5239 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-5240 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-5241 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-5242 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-5243 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-5244 3-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-5245 3-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-5246 3-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-5247 3-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-5248 3-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-5249 3-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-5250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4257 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3248 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3249 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2384 1-Naphthyl385 2-Naphthyl______________________________________ TABLE 45______________________________________ ##STR278##I: R.sup.1 = H, X = CH.sub.3II: R.sup.1 = CH.sub.3, X = CH.sub.3III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3IV: R.sup.1 = Allyl, X = CH.sub.3V: R.sup.1 = Propargyl, X = CH.sub.3VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3VIII: R.sup.1 = H, X = ClIX: R.sup.1 = CH.sub.3, X = ClX: R.sup.1 = C.sub.2 H.sub.5, X = ClXI: R.sup.1 = Allyl, X = ClXII: R.sup.1 = Propargyl, X = ClXIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = ClXIV: R.sup.1 = CO.sub.2 CH.sub.3, X = ClNo. T.sub.m______________________________________1 H2 2-F3 3-F4 4-F5 2,4-F.sub.26 2,4,6-F.sub.37 2,3,4,5,6,-F.sub.58 2,3-F.sub.29 2-Cl10 3-Cl11 4-Cl12 2,3,-Cl.sub.213 2,4-Cl.sub.214 2,5-Cl.sub.215 2,6-Cl.sub.216 3,4-Cl.sub.217 3,5-Cl.sub.218 2,3,4-Cl.sub.319 2,3,5-Cl.sub.320 2,3,6-Cl.sub.321 2,4,5-Cl.sub.322 2,4,6-Cl.sub.323 3,4,5-Cl.sub.324 2,3,4,6-Cl.sub.425 2,3,5,6-Cl.sub.426 2,3,4,5,6-Cl.sub.527 2-Br28 3-Br29 4-Br30 2,4-Br.sub.231 2,5-Br.sub.232 2,6-Br.sub.233 2,4,6-Br.sub.334 2,3,4,5,6-Br.sub.535 2-I36 3-I37 4-I38 2,4-I.sub.239 2-Cl, 3-F40 2-Cl, 4-F41 2-Cl, 5-F42 2-Cl, 6-F43 2-Cl, 3-Br44 2-Cl, 4-Br45 2-Cl, 5-Br46 2-Cl, 6-Br47 2-Br, 3-Cl48 2-Br, 4-Cl49 2-Br, 5-Cl50 2-Br, 3-F51 2-Br, 4-F52 2-Br, 5-F53 2-Br, 6-F54 2-F, 3-Cl55 2-F, 4-Cl56 2-F, 5-Cl57 3-Cl, 4-F58 3-Cl, 5-F59 3-Cl, 4-Br60 3-Cl, 5-Br61 3-F, 4-Cl62 3-F, 4-Br63 3-Br, 4-Cl64 3-Br, 4-F65 2,6-Cl.sub.2, 4-Br66 2-CH.sub.367 3-CH.sub.368 4-CH.sub.369 2,3-(CH.sub.3).sub.270 2,4-(CH.sub.3).sub.271 2,5-(CH.sub.3).sub.272 2,6-(CH.sub.3).sub.273 3,4-(CH.sub.3).sub.274 3,5-(CH.sub.3).sub.275 2,3,5-(CH.sub.3).sub.376 2,3,4-(CH.sub.3).sub.377 2,3,6-(CH.sub.3).sub.378 2,4,5-(CH.sub.3).sub.379 2,4,6-(CH.sub.3).sub.380 3,4,5-(CH.sub.3).sub.381 2,3,4,6-(CH.sub.3).sub.482 2,3,5,6-(CH.sub.3).sub.483 2,3,4,5,6-(CH.sub.3).sub.584 2-C.sub.2 H.sub.585 3-C.sub.2 H.sub.586 4-C.sub.2 H.sub.587 2,4-(C.sub.2 H.sub.5).sub.288 2,6-(C.sub.2 H.sub.5).sub.289 3,5-(C.sub.2 H.sub.5).sub.290 2,4,6-(C.sub.2 H.sub.5).sub.391 2-n-C.sub.3 H.sub.792 3-n-C.sub.3 H.sub.793 4-n-C.sub.3 H.sub.794 2-i-C.sub.3 H.sub.795 3-i-C.sub.3 H.sub.796 4-i-C.sub.3 H.sub.797 2,4-(i-C.sub.3 H.sub.7).sub.298 2,6-(i-C.sub.3 H.sub.7).sub.299 3,5-(i-C.sub.3 H.sub.7).sub.2100 2,4,6-(i-C.sub.3 H.sub.7).sub.3101 2-s-C.sub.4 H.sub.9102 3-s-C.sub.4 H.sub.9103 4-s-C.sub.4 H.sub.9104 2-t-C.sub.4 H.sub.9105 3-t-C.sub.4 H.sub.9106 4-t-C.sub.4 H.sub.9107 2,3-(t-C.sub.4 H.sub.9).sub.2108 2,4-(t-C.sub.4 H.sub.9).sub.2109 2,5-(t-C.sub.4 H.sub.9).sub.2110 2,6-(t-C.sub.4 H.sub.9).sub.2111 3,4-(t-C.sub.4 H.sub.9).sub.2112 2,4,6-(t-C.sub.4 H.sub.9).sub.3113 4-n-C.sub.9 H.sub.19114 4-n-C.sub.12 H.sub.25115 4-n-C.sub.15 H.sub.31116 4-(1,1,3,3-Tetramethylbutyl)117 4-(2,4,4-Trimethylpropyl)118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7128 2-Allyl129 3-Allyl130 4-Allyl131 2-Allyl, 6-CH.sub.3132 2-cyclo-C.sub.6 H.sub.11133 3-cyclo-C.sub.6 H.sub.11134 4-cyclo-C.sub.6 H.sub.11135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11137 2-CH.sub.2 C.sub.6 H.sub.5138 3-CH.sub.2 C.sub.6 H.sub.5139 4-CH.sub.2 C.sub.6 H.sub.5140 2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3141 2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5142 2-C.sub.6 H.sub.5143 3-C.sub.6 H.sub.5144 4-C.sub.6 H.sub.5145 4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2147 2-Cl, 4-C.sub.6 H.sub.5148 2-Br, 4-C.sub.6 H.sub.5149 2-C.sub.6 H.sub.5, 4-Cl150 2-C.sub.6 H.sub.5, 4-Br151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5155 2-cyclo-C.sub.6 H.sub.11, 4-Cl156 2-cyclo-C.sub.6 H.sub.11, 4-Br157 2-Cl, 4-cyclo-C.sub.6 H.sub.11158 2-Br, 4-cyclo-C.sub.6 H.sub.11159 2-OCH.sub.3160 3-OCH.sub.3161 4-OCH.sub.3162 2-OC.sub.2 H.sub.5163 3-OC.sub.2 H.sub.5164 4-OC.sub.2 H.sub.5165 2-O-n-C.sub.3 H.sub.7166 3-O-n-C.sub.3 H.sub.7167 4-O-n-C.sub.3 H.sub.7168 2-O-i-C.sub.3 H.sub.7169 3-O-i-C.sub.3 H.sub.7170 4-O-i-C.sub.3 H.sub.7171 2-O-n-C.sub.6 H.sub.13172 3-O-n-C.sub.6 H.sub.13173 4-O-n-C.sub.6 H.sub.13174 2-O-n-C.sub.8 H.sub.17175 3-O-n-C.sub.8 H.sub.17176 4-O-n-C.sub.8 H.sub.17177 2-OCH.sub.2 C.sub.6 H.sub.5178 3-OCH.sub.2 C.sub.6 H.sub.5179 4-OCH.sub.2 C.sub.6 H.sub.5180 2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5181 3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5182 4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5183 2,4-(OCH.sub.3).sub.2184 2-CF.sub.3185 3-CF.sub.3186 4-CF.sub.3187 2-OCF.sub.3188 3-OCF.sub.3189 4-OCF.sub.3190 3-OCH.sub.2 CHF.sub.2191 2-CO.sub.2192 3-NO.sub.2193 4-NO.sub.2194 2-CN195 3-CN196 4-CN197 2-CH.sub.3, 3-Cl198 2-CH.sub.3, 4-Cl199 2-CH.sub.3, 5-Cl200 2-CH.sub.3, 6-Cl201 2-CH.sub.3, 3-F202 2-CH.sub.3, 4-F203 2-CH.sub.3, 5-F204 2-CH.sub.3, 6-F205 2-CH.sub.3, 3-Br206 2-CH.sub.3, 4-Br207 2-CH.sub.3, 5-Br208 2-CH.sub.3, 6-Br209 2-Cl, 3-CH.sub.3210 2-Cl, 4-CH.sub.3211 2-Cl, 5-CH.sub.3212 2-F, 3-CH.sub.3213 2-F, 4-CH.sub.3214 2-F, 5-CH.sub.3215 2-Br, 3-CH.sub.3216 2-Br, 4-CH.sub.3217 2-Br, 5-CH.sub.3218 3-CH.sub.3, 4-Cl219 3-CH.sub.3, 5-Cl220 3-CH.sub.3, 4-F221 3-CH.sub.3, 5-F222 3-CH.sub.3, 4-Br223 3-CH.sub.3, 5-Br224 3-F, 4-CH.sub.3225 3-Cl, 4-CH.sub.3226 3-Br, 4-CH.sub.3227 2-Cl, 4,5-(CH.sub.3).sub.2228 2-Br, 4,5-(CH.sub.3).sub.2229 2-Cl, 3,5-(CH.sub.3).sub.2230 2-Br, 3,5-(CH.sub.3).sub.2231 2,6-Cl.sub.2, 4-CH.sub.3232 2,6-F.sub.2, 4-CH.sub.3233 2,6-Br.sub.2, 4-CH.sub.3234 2,4-Br.sub.2, 6-CH.sub.3235 2,4-F.sub.2, 6-CH.sub.3236 2,4-Br.sub.2, 6-CH.sub.3237 2,6-(CH.sub.3).sub.2, 4-F238 2,6-(CH.sub.3).sub.2, 4-Cl239 2,6-(CH.sub.3).sub.2, 4-Br240 3,5-(CH.sub.3).sub.2, 4-F241 3,5-(CH.sub.3).sub.2, 4-Cl242 3,5-(CH.sub.3).sub.2, 4-Br243 2,3,6-(CH.sub.3).sub.3, 4-F244 2,3,6-(CH.sub.3).sub.3, 4-Cl245 2,3,6-(CH.sub.3).sub.3, 4-Br246 2,4-(CH.sub.3).sub.2, 6-F247 2,4-(CH.sub.3).sub.2, 6-Cl248 2,4-(CH.sub.3).sub.2, 6-Br249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3250 2-Cl, 4-NO.sub.2251 2-NO.sub.2, 4-Cl252 2-OCH.sub.3, 5-NO.sub.2253 2,4-Cl.sub.2, 5-NO.sub.2254 2,4-Cl.sub.2, 6-NO.sub.2255 2,6-Cl.sub.2, 4-NO.sub.2256 2,6-Br.sub.2, 4-NO.sub.2257 2,6-I.sub.2, 4-NO.sub.2258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl259 2-CO.sub.2 CH.sub.3260 3-CO.sub.2 CH.sub.3261 4-CO.sub.2 CH.sub.3262 2-CO.sub.2 (C.sub.2 H.sub.5)263 3-CO.sub.2 (C.sub.2 H.sub.5)264 4-CO.sub.2 (C.sub.2 H.sub.5)265 2-CO.sub.2 (n-C.sub.3 H.sub.7)266 3-CO.sub.2 (n-C.sub.3 H.sub.7)267 4-CO.sub.2 (n-C.sub.3 H.sub.7)268 2-CO.sub.2 (i-C.sub.3 H.sub.7)269 3-CO.sub.2 (i-C.sub.3 H.sub.7)270 4-CO.sub.2 (i-C.sub.3 H.sub.7)271 2-CO.sub.2 (n-C.sub.6 H.sub.13)272 3-CO.sub.2 (n-C.sub.6 H.sub.13)273 4-CO.sub.2 (n-C.sub.6 H.sub.13)274 2-CH.sub.2 OCH.sub.3275 3-CH.sub.2 OCH.sub.3276 4-CH.sub.2 OCH.sub.3277 2-CH.sub.2 O(C.sub.2 H.sub.5)278 3-CH.sub.2 O(C.sub.2 H.sub.5)279 4-CH.sub.2 O(C.sub.2 H.sub.5)280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)286 2-CHO287 3-CHO288 4-CHO289 2-COCH.sub.3290 3-COCH.sub.3291 4-COCH.sub.3292 2-COCH.sub.2 CH.sub.3293 3-COCH.sub.2 CH.sub.3294 4-COCH.sub.2 CH.sub.3295 2-COCH.sub.2 CH.sub.2 CH.sub.3296 3-COCH.sub.2 CH.sub.2 CH.sub.3297 4-COCH.sub.2 CH.sub.2 CH.sub.3298 2-COCH(CH.sub.3)CH.sub.3299 3-COCH(CH.sub.3)CH.sub.3300 4-COCH(CH.sub.3)CH.sub.3301 2-Me-4-CHO302 2-Me-4-CH.sub.3 CO303 2-Me-4-CH.sub.3 CH.sub.2 CO304 2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO305 2-Me-4-CH.sub.3 CH(CH.sub.3)CO306 2,5-Me.sub.2 -4-CHO307 2,5-Me.sub.2 -4-CH.sub.3 CO308 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO309 2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO310 2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO311 2-Cl-4-CHO312 2-Cl-4-CH.sub.3 CO313 2-Cl-4-CH.sub.3 CH.sub.2 CO314 2-Cl-4-CH.sub.3 CH(CH.sub.3)CO315 2,5-Cl.sub.2 -4-CHO316 2,5-Cl.sub.2 -4-CH.sub.3 CO317 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO318 2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO319 2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO320 2-C(NOCH.sub.3)CH.sub.3321 3-C(NOCH.sub.3)CH.sub.3322 4-C(NOCH.sub.3)CH.sub.3323 2-C(NOC.sub.2 H.sub.5)CH.sub.3324 3-C(NOC.sub.2 H.sub.5)CH.sub.3325 4-C(NOC.sub.2 H.sub.5)CH.sub.3326 2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3327 3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3328 4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3329 2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3330 3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3331 4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3332 2-C(NO-Allyl)-CH.sub.3333 3-C(NO-Allyl)-CH.sub.3334 4-C(NO-Allyl)-CH.sub.3335 2-C(NO-trans-Chloroallyl)-CH.sub.3336 3-C(NO-trans-Chloroallyl)-CH.sub.3337 4-C(NO-trans-Chloroallyl)-CH.sub.3338 2-C(NO-Propargyl)-CH.sub.3339 3-C(NO-Propargyl)-CH.sub.3340 4-C(NO-Propargyl)-CH.sub.3341 2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3342 3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3343 4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3344 2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3345 3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3346 4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3347 2-CH.sub.3 -4-CHNOCH.sub.3348 2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5349 2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7350 2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7351 2-CH.sub.3 -4-CHNO-Allyl352 2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)353 2-CH.sub.3 -4-CHNO-Propargyl354 2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9355 2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5356 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)357 2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)358 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)359 2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)360 2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)361 2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)362 2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)363 2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)364 2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)383 2-C.sub.6 H.sub.5384 3-C.sub.6 H.sub.5385 4-C.sub.6 H.sub.5386 2-(2'-FC.sub.6 H.sub.4)387 2-(3'-FC.sub.6 H.sub.4)388 2-(4'-FC.sub.6 H.sub.4)389 3-(2'-FC.sub.6 H.sub.4)390 3-(3'-FC.sub.6 H.sub.4)391 3-(4'-FC.sub.6 H.sub.4)392 4-(2'-FC.sub.6 H.sub.4)393 4-(3'-FC.sub.6 H.sub.4)394 4-(4'-FC.sub.6 H.sub.4)395 2-(2'-ClC.sub.6 H.sub.4)396 2-(3'-ClC.sub.6 H.sub.4)397 2-(4'-ClC.sub.6 H.sub.4)398 3-(2'-ClC.sub.6 H.sub.4)399 3-(3'-ClC.sub.6 H.sub.4)400 3-(4'-ClC.sub.6 H.sub.4)401 4-(2'-ClC.sub.6 H.sub.4)402 4-(3'-ClC.sub.6 H.sub.4)403 4-(4'-ClC.sub.6 H.sub.4)405 2-(2'-CH.sub.3 C.sub.6 H.sub.4)406 2-(3'-CH.sub.3 C.sub.6 H.sub.4)407 2-(4'-CH.sub.3 C.sub.6 H.sub.4)408 3-(2'-CH.sub.3 C.sub.6 H.sub.4)409 3-(3'-CH.sub.3 C.sub.6 H.sub.4)410 3-(4'-CH.sub.3 C.sub.6 H.sub.4)411 4-(2'-CH.sub.3 C.sub.6 H.sub.4)412 4-(3'-CH.sub.3 C.sub.6 H.sub.4)413 4-(4'-CH.sub.3 C.sub.6 H.sub.4)414 2-(2'-CH.sub.3 COC.sub.6 H.sub.4)415 2-(3'-CH.sub.3 COC.sub.6 H.sub.4)416 2-(4'-CH.sub.3 COC.sub.6 H.sub.4)417 3-(2'-CH.sub.3 COC.sub.6 H.sub.4)418 3-(3'-CH.sub.3 COC.sub.6 H.sub.4)419 3-(4'-CH.sub.3 COC.sub.6 H.sub.4)420 4-(2'-CH.sub.3 COC.sub.6 H.sub.4)421 4-(3'-CH.sub.3 COC.sub.6 H.sub.4)422 4-(4'-CH.sub.3 COC.sub.6 H.sub.4)423 2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)424 2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)425 2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)426 3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)427 3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)428 3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)429 4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)430 4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)431 4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)432 2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)433 2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)434 2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)435 3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)436 3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)437 3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)438 4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)439 4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)440 4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)441 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)442 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)443 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)444 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)445 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)446 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)447 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)448 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)449 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)450 2-(2'-O.sub.2 NC.sub.6 H.sub.4)451 2-(3'-O.sub.2 NC.sub.6 H.sub.4)452 2-(4'-O.sub.2 NC.sub.6 H.sub.4)453 3-(2'-O.sub.2 NC.sub.6 H.sub.4)454 3-(3'-O.sub.2 NC.sub.6 H.sub.4)455 3-(4'-O.sub.2 NC.sub.6 H.sub.4)456 4-(2'-O.sub.2 NC.sub.6 H.sub.4)457 4-(3'-O.sub.2 NC.sub.6 H.sub.4)458 4-(4'-O.sub.2 NC.sub.6 H.sub.4)459 2-(2'-NCC.sub.6 H.sub.4)460 2-(3'-NCC.sub.6 H.sub.4)461 2-(4'-NCC.sub.6 H.sub.4)462 3-(2'-NCC.sub.6 H.sub.4)463 3-(3'-NCC.sub.6 H.sub.4)464 3-(4'-NCC.sub.6 H.sub.4)465 4-(2'-NCC.sub.6 H.sub.4)466 4-(3'-NCC.sub.6 H.sub.4)467 4-(4'-NCC.sub.6 H.sub.4)468 2-(2'-CF.sub.3 C.sub.6 H.sub.4)469 2-(3'-CF.sub.3 C.sub.6 H.sub.4)470 2-(4'-CF.sub.3 C.sub.6 H.sub.4)471 3-(2'-CF.sub.3 C.sub.6 H.sub.4)472 3-(3'-CF.sub.3 C.sub.6 H.sub.4)473 3-(4'-CF.sub.3 C.sub.6 H.sub.4)474 4-(2'-CF.sub.3 C.sub.6 H.sub.4)475 4-(3'-CF.sub.3 C.sub.6 H.sub.4)476 4-(4'-CF.sub.3 C.sub.6 H.sub.4)477 2-OC.sub.6 H.sub.5475 3-OC.sub.6 H.sub.5476 4-OC.sub.6 H.sub.5478 2-O-(2'-FC.sub.6 H.sub.4)479 2-O-(3'-FC.sub.6 H.sub.4)480 2-O-(4'-FC.sub.6 H.sub.4)481 3-O-(2'-FC.sub.6 H.sub.4)482 3-O-(3'-FC.sub.6 H.sub.4)483 3-O-(4'-FC.sub.6 H.sub.4)484 4-O-(2'-FC.sub.6 H.sub.4)485 4-O-(3'-FC.sub.6 H.sub.4)486 4-O-(4'-FC.sub.6 H.sub.4)487 2-O-(2'-ClC.sub.6 H.sub.4)488 2-O-(3'-ClC.sub.6 H.sub.4)489 2-O-(4'-ClC.sub.6 H.sub.4)490 3-O-(2'-ClC.sub.6 H.sub.4)491 3-O-(3'-ClC.sub.6 H.sub.4)492 3-O-(4'-ClC.sub.6 H.sub.4)493 3-O-(4'-ClC.sub.6 H.sub.4)494 4-O-(2'-ClC.sub.6 H.sub.4)495 4-O-(3'-ClC.sub.6 H.sub.4)496 4-O-(4'-ClC.sub.6 H.sub.4)497 2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)498 2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)499 2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)500 3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)501 3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)502 3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)503 4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)504 4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)505 4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)506 2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)507 2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)508 2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)509 3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)510 3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)511 3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)512 4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)513 4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)514 4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)515 2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)516 2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)517 2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)518 3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)519 3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)520 3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)521 4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)522 4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)523 4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)524 2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)525 2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)526 2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)527 3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)528 3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)529 3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)530 4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)531 4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)532 4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)533 2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)534 2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)535 2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)536 3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)537 3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)538 3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)539 4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)540 4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)541 4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)542 2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)543 2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)544 2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)545 3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)546 3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)547 3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)548 4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)549 4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)550 4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)551 2-O-(2'-NCC.sub.6 H.sub.4)552 2-O-(3'-NCC.sub.6 H.sub.4)553 2-O-(4'-NCC.sub.6 H.sub.4)554 3-O-(2'-NCC.sub.6 H.sub.4)555 3-O-(3'-NCC.sub.6 H.sub.4)556 3-O-(4'-NCC.sub.6 H.sub.4)557 4-O-(2'-NCC.sub.6 H.sub.4)558 4-O-(3'-NCC.sub.6 H.sub.4)559 4-O-(4'-NCC.sub.6 H.sub.4)560 2-O-(2'-CF.sub.3 C.sub.6 H.sub.5)561 2-O-(3'-CF.sub.3 C.sub.6 H.sub.5)562 2-O-(4'-CF.sub.3 C.sub.6 H.sub.5)563 3-O-(2'-CF.sub.3 C.sub.6 H.sub.5)564 3-O-(3'-CF.sub.3 C.sub.6 H.sub.5)565 3-O-(4'-CF.sub.3 C.sub.6 H.sub.5)566 4-O-(2'-CF.sub.3 C.sub.6 H.sub.5)567 4-O-(3'-CF.sub.3 C.sub.6 H.sub.5)568 4-O-(4'-CF.sub.3 C.sub.6 H.sub.5)569 2-Pyridinyl-2'570 2-Pyridinyl-3'571 2-Pyridinyl-4'572 3-Pyridinyl-2'573 3-Pyridinyl-3'574 3-Pyridinyl-4'575 4-Pyridinyl-2'576 4-Pyridinyl-3'577 4-Pyridinyl-4'578 2-Pyrimidinyl-2'579 2-Pyrimidinyl-3'580 2-Pyrimidinyl-4'581 3-Pyrimidinyl-2'582 3-Pyrimidinyl-3'583 3-Pyrimidinyl-4'584 4-Pyrimidinyl-2'585 4-Pyrimidinyl-3'586 4-Pyrimidinyl-4'587 2-Pyrazolyl-1'588 2-Pyrazolyl-3'589 2-Pyrazolyl-4'590 3-Pyrazolyl-1'591 3-Pyrazolyl-3'592 3-Pyrazolyl-4'593 4-Pyrazolyl-1'594 4-Pyrazolyl-3'595 4-Pyrazolyl-4'596 2-Isoxazolyl-3'597 2-Isoxazolyl-4'598 2-Isoxazolyl-5'599 3-Isoxazolyl-3'600 3-Isoxazolyl-4'601 3-Isoxazolyl-5'602 4-Isoxazolyl-3'603 4-Isoxazolyl-4'604 4-Isoxazolyl-5'605 2-Isothiazolyl-3'606 2-Isothiazolyl-4'607 2-Isothiazolyl-5'608 3-Isothiazolyl-3'609 3-Isothiazolyl-4'610 3-Isothiazolyl-5'611 4-Isothiazolyl-3'612 4-Isothiazolyl-4'613 4-Isothiazolyl-5'614 2-Imidazolyl-1'615 2-Imidazolyl-2'616 2-Imidazolyl-4'617 3-Imidazolyl-1'618 3-Imidazolyl-2'619 3-Imidazolyl-4'620 4-Imidazolyl-1'621 4-Imidazolyl-2'622 4-Imidazolyl-4'623 2-Oxazolyl-2'624 2-Oxazolyl-4'625 2-Oxazolyl-5'626 3-Oxazolyl-2'627 3-Oxazolyl-4'628 3-Oxazolyl-5'629 4-Oxazolyl-2'630 4-Oxazolyl-4'631 4-Oxazolyl-5'632 2-Thiazolyl-2'633 2-Thiazolyl-4'634 2-Thiazolyl-5'635 3-Thiazolyl-2'636 3-Thiazolyl-4'637 3-Thiazolyl-5'638 4-Thiazolyl-2'639 4-Thiazolyl-4'640 4-Thiazolyl-5'______________________________________ TABLE 46______________________________________ ##STR279##I: R.sup.1 = H, X = CH.sub.3II: R.sup.1 = CH.sub.3, X = CH.sub.3III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3IV: R.sup.1 = Allyl, X = CH.sub.3V: R.sup.1 = Propargyl, X = CH.sub.3VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3VIII: R.sup.1 = H, X = ClIX: R.sup.1 = CH.sub.3, X = ClX: R.sup.1 = C.sub.2 H.sub.5, X = ClXI: R.sup.1 = Allyl, X = ClXII: R.sup.1 = Propargyl, X = ClXIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = ClXIV: R.sup.1 = CO.sub.2 CH.sub.3, X = ClV: R.sup.1 =No. B______________________________________1 Pyrrolyl-32 NCH.sub.3 -Pyrrolyl-33 NC.sub.6 H.sub.5 -Pyrrolyl-34 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-35 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-36 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-37 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-38 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-39 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-310 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-311 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-312 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-313 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-314 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-315 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-316 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-317 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-318 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-319 Pyrrolyl-220 NCH.sub.3 -Pyrrolyl-221 NC.sub.6 H.sub.5 -Pyrrolyl-222 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-223 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-224 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-225 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-226 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-227 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-228 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-229 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-230 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-231 N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-232 N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-233 N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-234 N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-235 N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-236 N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-237 Furyl-238 5-CH.sub.3 -Furyl-239 5-C.sub.6 H.sub.5 -Furyl-240 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-241 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-242 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-243 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-244 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-245 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-246 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-247 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-248 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-249 5-(4'-CNC.sub.6 H.sub.4)-Furyl-250 5-(3'-CNC.sub.6 H.sub.4)-Furyl-251 5-(2'-CNC.sub.6 H.sub.4)-Furyl-252 5-(4'-ClC.sub.6 H.sub.4)-Furyl-253 5-(3'-ClC.sub.6 H.sub.4)-Furyl-254 5-(2'-ClC.sub.6 H.sub.4)-Furyl-255 4-CH.sub.3 -Furyl-256 4-C.sub.6 H.sub.5 -Furyl-257 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-258 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-259 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-260 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-261 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-262 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-263 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-264 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-265 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-266 4-(4'-CNC.sub.6 H.sub.4)-Furyl-267 4-(3'-CNC.sub.6 H.sub.4)-Furyl-268 4-(2'-CNC.sub.6 H.sub.4)-Furyl-269 4-(4'-ClC.sub.6 H.sub.4)-Furyl-270 4-(3'-ClC.sub.6 H.sub.4)-Furyl-271 4-(2'-ClC.sub.6 H.sub.4)-Furyl-272 Thienyl-273 5-CH.sub.3 -Thienyl-274 5-C.sub.6 H.sub.5 -Thienyl-275 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-276 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-277 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-278 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-279 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-280 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-281 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-282 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-283 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-284 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-285 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-286 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-287 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-288 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-289 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-290 4-CH.sub.3 -Thienyl-291 4-C.sub.6 H.sub.5 -Thienyl-292 4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-293 4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-294 4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-295 4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-296 4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-297 4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-298 4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-299 4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2100 4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2101 4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2102 4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2103 4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2104 4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2105 4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2106 4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2107 Thienyl-3108 5-CH.sub.3 -Thienyl-3109 5-C.sub.6 H.sub.5 -Thienyl-3110 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3111 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3112 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3113 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3114 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3115 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3116 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3117 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3118 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3119 5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3120 5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3121 5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3122 5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3123 5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3124 5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3125 Pyrazolyl-4126 NCH.sub.3 -Pyrazolyl-4127 NC.sub.6 H.sub.5 -Pyrazolyl-4128 N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4129 N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4130 N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4131 N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4132 N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4133 N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4134 N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4135 N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4136 N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4137 N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4138 N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4139 N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4140 N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4141 N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4142 N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4143 3-CH.sub.3 N-Methylpyrazolyl-4144 3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4145 3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4146 3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4147 3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4148 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4149 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4150 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4151 3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4152 3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4153 3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4154 3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4155 3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4156 3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4157 3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4158 3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4159 3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4160 Isoxazolyl-5161 3-CH.sub.3 -Isoxazolyl-5162 3-C.sub.6 H.sub.5 -Isoxazolyl-5163 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5164 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5165 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5166 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5167 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5168 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5169 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5170 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5171 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5172 3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5173 3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5174 3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5175 3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5176 3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5177 3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5178 4-Chloroisoxazolyl-5179 3-CH.sub.3 -4-Chloroisoxazolyl-5180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5181 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5182 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5183 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5184 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5185 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5186 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5187 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5188 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5189 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5190 3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5191 3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5192 3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5193 3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5194 3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5195 3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5196 Isoxazolyl-3197 5-CH.sub.3 -Isoxazolyl-3198 5-C.sub.6 H.sub.5 -Isoxazolyl-3199 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3200 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3201 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3202 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3203 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3204 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3205 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3206 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3207 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3208 5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3209 5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3210 5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3211 5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3212 5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3213 5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3214 Isothiazolyl-5215 3-CH.sub.3 -Isothiazolyl-5216 3-C.sub.6 H.sub.5 -Isothiazolyl-5217 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5218 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5219 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5220 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5221 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5222 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5223 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5224 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5225 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5226 3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5227 3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5228 3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5229 3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5230 3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5231 3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5232 Oxazolyl-4233 2-CH.sub.3 -Oxazolyl-4234 2-C.sub.6 H.sub.5 -Oxazolyl-4235 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4236 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4237 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4238 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4239 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4240 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4241 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4242 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4243 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4244 2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4245 2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4246 2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4247 2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4248 2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4249 2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4250 Thiazolyl-4251 2-CH.sub.3 -Thiazolyl-4252 2-C.sub.6 H.sub.5 -Thiazolyl-4253 2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4254 2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4255 2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4256 2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4267 2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4258 2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4259 2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4260 2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4261 2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4262 2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4263 2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4264 2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4265 2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4266 2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4267 2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4268 NCH.sub.3 -1,2,4-Triazolyl-5269 3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5270 3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5271 3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5272 3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5273 3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5274 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5275 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5276 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5277 3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5278 3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5279 3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5280 3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5281 3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5282 3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5283 3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5284 3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5285 3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5286 1,3,4-Oxadiazolyl-2287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2289 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2290 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2291 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2292 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2293 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2294 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2295 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2296 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2297 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2298 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2299 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2300 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2301 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2302 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2303 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2304 1,2,4-Oxadiazolyl-3305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3307 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3308 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3309 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3310 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3311 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3312 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3313 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3314 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3315 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3316 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3317 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3318 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3319 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3320 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3321 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3322 1,2,4-Oxadiazolyl-5323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5325 3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5326 3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5327 3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5328 3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5329 3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5330 3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5331 3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5332 3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5333 3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5334 3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5335 3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5336 3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5337 3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5338 3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5339 3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5340 1,2,4-Thiadiazolyl-3341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3343 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3344 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3345 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3346 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3347 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3348 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3349 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3350 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3351 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3352 5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3353 5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3354 5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3355 5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3356 5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3357 5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3358 1,3,4-Thiadiazolyl-2359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2361 5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2362 5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2363 5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2364 5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2365 5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2366 5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2367 5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2368 5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2369 5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2370 5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2371 5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2372 5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2373 5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2374 5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2375 5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2376 Pyridinyl-2377 Pyridinyl-4378 Pyridazinyl-3379 Pyridazinyl-4380 Pyridazinyl-2381 Pyrimidinyl-4382 Pyrimidinyl-5383 Pyrimidinyl-2______________________________________ TABLE 47______________________________________Selected physical data of some compounds ##STR280## IR (cm.sup.-1) orNo. X.sub.m R.sup.1 .sup.1 h-NMR (ppm) mp______________________________________1 4-Cl H 1332 3,4-Cl.sub.2 H 1093 4-t-C.sub.4 H.sub.9 H 864 4-CH.sub.3 H 1175 4-CF.sub.3 H 1036 3-Br H 997 3-Cl H 938 3-CF.sub.3 H 889 3,5-Cl.sub.2 H 10010 3,4-(CH.sub.3).sub.2 H 12711 3,4-Cl.sub.2 CH.sub.3 7412 3,4-Cl.sub.2 Allyl 3.65(S, 3H); 2.2(S, 6H)13 3,4-Cl.sub.2 Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H)14 3,4-Cl.sub.2 CH.sub.2 OCH.sub.3 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H)15 3,4-Cl.sub.2 COOCH.sub.3 13716 4-t-C.sub.4 H.sub.9 CH.sub.3 3.65(S, 3H); 2.25(S, 3H); 2.2(S, 3H)17 4-t-C.sub.4 H.sub.9 Allyl 6918 4-t-C.sub.4 H.sub.9 Propargyl 11719 4-t-C.sub.4 H.sub.9 CH.sub.2 OCH.sub.3 3.65(S, 3H); 2.25(S, 3H); 117 2.2(S, 3H)20 4-t-C.sub.4 H.sub.9 COOCH.sub.3 3.65, 2.1 11921 4-CH.sub.3 CH.sub.3 6922 4-CH.sub.3 Allyl 3.65(S, 3H); 2.25(S, 3H); 2.2(S, 3H)23 4-CH.sub.3 Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H)24 4-CH.sub.3 CH.sub.2 OCH.sub.3 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H)25 4-CH.sub.3 COOCH.sub.3 9726 4-CF.sub.3 CH.sub.3 7627 4-CF.sub.3 Allyl 3.65(S, 3H); 2.3(S, 3H); 2.25(S, 3H)28 4-CF.sub.3 Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.25(S, 3H)29 4-CF.sub.3 CH.sub.2 OCH.sub.3 3.65(S, 3H); 2.25(S, 3H);30 4-CF.sub.3 COOCH.sub.3 10331 4-Cl CH.sub.3 10632 4-Cl Allyl 3.65(S, 3H); 2.2(2S, each 3H)33 4-Cl Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H)34 4-Cl CH.sub.2 OCH.sub.3 3.65(S, 3H); 2.25(S, 3H); 2.2(S, 3H)35 4-Cl COOCH.sub.3 10936 3-Br CH.sub.3 7537 3-Br Allyl 3.65(S, 3H); 2.2(2S, each 3H38 3-Br Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H)39 3-Br CH.sub.2 OCH.sub.3 7240 3-Br COOCH.sub.3 13141 3-Cl CH.sub.3 8442 3-Cl Allyl 3.65(S, 3H); 2.25(S, 3H); 2.2(S, 3H)43 3-Cl Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H)44 3-Cl CH.sub.2 OCH.sub.3 6645 3-Cl COOCH.sub.3 12346 3-CF.sub.3 CH.sub.3 6347 3-CF.sub.3 Allyl 6448 3-CF.sub.3 Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.25(S, 3H)49 3-CF.sub.3 CH.sub.2 OCH.sub.3 8950 3-CF.sub.3 COOCH.sub.3 13651 4-Br COOCH.sub.3 10352 4-Br H 10853 4-Br Propargyl 1710,1486,1469,1447,1376, 1299,1252,1026,1008,77454 4-Br CH.sub.2 OCH.sub.3 1715,1468,1445,1370,1301, 1274,1090,1059,1008,77555 3,4-(CH.sub.3).sub.2 CH.sub.3 oil56 3,4-(CH.sub.3).sub.2 Allyl oil57 3,4-(CH.sub.3).sub.2 Propargyl oil58 3,4-(CH.sub.3).sub.2 CH.sub.2 OCH.sub.3 oil59 3,4-(CH.sub.3).sub.2 COOCH.sub.3 13560 3,5-Cl.sub.2 CH.sub.3 9561 3,5-Cl.sub.2 Allyl 9762 3,5-Cl.sub.2 Propargyl 10063 3,5-Cl.sub.2 CH.sub.2 OCH.sub.3 11264 3,5-Cl.sub.2 COOCH.sub.3 160______________________________________ TABLE 48__________________________________________________________________________Selected physical data of some compounds ##STR281## IR (cm.sup.-1) orNo. X.sub.m R.sup.1 .sup.1 h-NMR (ppm) mp__________________________________________________________________________1 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 H 822 2,4-(CH.sub.3).sub.2 H 1313 2,5-(CH.sub.3).sub.2 H 1244 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5 H 1025 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NOC.sub.2 H.sub.5 H 1166 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 H 1227 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 CH.sub.3 4.0(S, 3H); 3.65(S, 3H)8 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 Allyl 1019 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 Propargyl 4.0(S, 3H); 3.65(S, 3H)10 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 CH.sub.2 OCH.sub.3 4.0(S, 3H); 3.65(S, 3H)11 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3 COOCH.sub.3 12212 2,4-(CH.sub.3).sub.2 CH.sub.3 3.65(S, 3H); 2.25(2s, each 3H)13 2,4-(CH.sub.3).sub.2 Allyl 5914 2,4-(CH.sub.3).sub.2 Propargyl 3.65(S, 3H); 2.25(3s, each 3H)15 2,4-(CH.sub.3).sub.2 CH.sub.2 OCH.sub.3 7616 2,4-(CH.sub.3).sub.2 COOCH.sub.3 13317 2,5-(CH.sub.3).sub.2 CH.sub.3 3.65(S, 3H); 2.3(S, 3H)18 2,5-(CH.sub.3).sub.2 Allyl 5619 2,5-(CH.sub.3).sub.2 Propargyl 8020 2,5-(CH.sub.3).sub.2 CH.sub.2 OCH.sub.3 3.65(S, 3H); 2.3(S, 3H) 8021 2,5-(CH.sub.3).sub.2 CH.sub.2 OCH.sub.3 14022 2-CH.sub.3 H 10723 2-CH.sub.3 Propargyl oil24 2-CH.sub.3 COOCH.sub.3 13525 2-CH.sub.3 CH.sub.2 OCH.sub.3 oil26 2-CH.sub.3 -4-C(CH.sub.3)NO-Allyl H 9727 2-CH.sub.3 -4-C(CH.sub.3)NO-Allyl Propargyl oil28 2-CH.sub.3 -4-C(CH.sub.3)NO-Allyl COOCH.sub.3 13029 2-CH.sub.3 -4-C(CH.sub.3)NO-Allyl HC.sub.2 OCH.sub.3 oil30 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5 CH.sub.3 oil31 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5 Allyl 7532 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5 Propargyl 7733 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5 CH.sub.2 OCH.sub.3 oil34 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5 COOCH.sub.3 oil35 2-CH.sub.3 -4-C(CH.sub.3)NOOCH.sub.3 CH.sub.3 oil36 2-CH.sub.3 -4-C(CH.sub.3)NOOCH.sub.3 Allyl 10437 2-CH.sub.3 -4-C(CH.sub.3)NOOCH.sub.3 Propargyl oil38 2-CH.sub.3 -4-C(CH.sub.3)NOOCH.sub.3 CH.sub.2 OCH.sub.3 oil39 2-CH.sub.3 -4-C(CH.sub.3)NOOCH.sub.3 COOCH.sub.3 15840 2-CH.sub.3 -4-C(CH.sub.3)NOOC.sub.2 H.sub.5 CH.sub.3 oil41 2-CH.sub.3 -4-C(CH.sub.3)NOOC.sub.2 H.sub.5 Allyl 7142 2-CH.sub.3 -4-C(CH.sub.3)NOOC.sub.2 H.sub.5 Propargyl oil43 2-CH.sub.3 -4-C(CH.sub.3)NOOC.sub.2 H.sub.5 CH.sub.2 OCH.sub.3 oil44 2-CH.sub.3 -4-C(CH.sub.3)NOOC.sub.2 H.sub.5 COOCH.sub.3 128__________________________________________________________________________ TABLE 49______________________________________ ##STR282##I: R.sup.1 = H, X = CH.sub.3II: R.sup.1 = CH.sub.3, X = CH.sub.3III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3IV: R.sup.1 = Allyl, X = CH.sub.3V: R.sup.1 = Propargyl, X = CH.sub.3VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3VIII: R.sup.1 = H, X = ClIX: R.sup.1 = CH.sub.3, X = ClX: R.sup.1 = C.sub.2 H.sub.5, X = ClXI: R.sup.1 = Allyl, X = ClXII: R.sup.1 = Propargyl, X = ClXIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = ClXIV: R.sup.1 = CO.sub.2 CH.sub.3, X = ClNo. B______________________________________1 2-Pyridyl2 3-Trifluoromethyl-2-pyridyl3 5-Trifluoromethyl-2-pyridyl4 3,5-Bis-(trifluoromethyl-2-pyridyl5 3,5-Dichloro-2-pyridyl6 3-Chloro-5-trifluoromethyl-2-pyridyl7 3,5-Dichloro-2-pyridyl8 2-Chloro-4-trifluoromethylphenyl9 2-Benzothiazolyl10 5-Chloro-1-methyl-2-benzimidazolyl11 2-Benzoxazolyl12 1-Methyl-5-trifluoromethylimide-azo�5,4-a!-pyridin-2-yl13 5-Chloro-2-pyrimidinyl14 4-Methyl-5-phenyl-2-thiazolin-2-yl15 4-Methyl-5-phenyl-2-oxazolin-2-yl16 7-Trifluoromethyl-4-quinolinyl______________________________________ TABLE 50______________________________________Selected physical data of some compounds ##STR283##No. X.sub.m IR (cm.sup.-1) or .sup.1 H-NMR (ppm) mp______________________________________1 4-NO.sub.2 1122 3,4-Cl.sub.2 3.8(s, 3H); 3.75(s, 3H)3 2,4-(CH.sub.3).sub.2 3.75(s, 3H); 3.7(s, 3H)4 H 3.75(2s, each 3H)5 4-i-C.sub.3 H.sub.7 3.8(s, 3H); 3.75(s, 3H)6 3,4-(CH.sub.3).sub.2 3.8(s, 3H); 3.75(s, 3H)7 3-CH.sub.3 -4-OCH.sub.3 3.85(s, 3H); 3.8(s, 3H); 3.75(s, 3H)8 3-CH.sub.3 -4-O- 3.8(2s, each 3H) I-C.sub.3 H.sub.79 4-CF.sub.3 3.8(s, 3H); 3.75(s, 3H)10 3-CH.sub.3 3.8(2s, each 3H)11 3-CF.sub.3 3.8(s, 3H); 3.75(s, 3H)12 4-F 3.8(s, 3H); 3.75(s, 3H)13 4-Br 3.8(s, 3H); 3.75(s, 3H)14 3-Br 3.8(s, 3H); 3.75(s, 3H)15 4-t-Bu 3.8(s, 3H); 3.75(s, 3H)16 4-OCH.sub.3 3.85(s, 3H); 3.8(s, 3H); 3.75(s, 3H)17 2-CH.sub.3 3.8(s, 3H); 3.75(s, 3H)18 3-Cl 3.8(s, 3H); 3.75(s, 3H)19 4-CN 3.8(s, 3H); 3.75(s, 3H)20 4-C.sub.2 H.sub.5 3.8(s, 3H); 3.75(s, 3H)______________________________________ TABLE 51______________________________________Selected physical data of some comounds ##STR284##No. X.sub.m IR (cm.sup.-1) or .sup.1 H-NMR (ppm) mp______________________________________1 4-Cl 3.8(s, 3H); 3.75(s, 3H)2 2-Cl 3.8(s, 3H); 3.75(s, 3H)3 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5) 3.8(s, 3H); 3.75(s, 3H) N-Allyl4 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5) 3.9(s, 3H); 3.8(s, 3H); NOCH.sub.3 3.75(s, 3H)5 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NO- 3.8(s, 3H); 3.75(s, 3H) trans-Cl-Allyl6 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NO- 3.8(s, 3H); 3.75(s, 3H) Allyl7 2-CH.sub.3 -4-Cl 3.8(s, 3H); 3.75(s, 3H)8 2-Cl-4-CH.sub.3 3.8(s, 3H); 3.75(s, 3H)9 2-Cl-5-CH.sub.3 3.8(s, 3H); 3.75(s, 3H)10 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)N 4.2(z, 2H); 3.8(s, 3H); OC.sub.2 H.sub.5 3.75(s, 3H)11 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)N 3.95(s, 3H); 3.8(s, 3H); OCH.sub.3 3.75(s, 3H)12 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3) 3.8(s, 3H); 3.75(s, 3H) NO-trans-Cl-Allyl13 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3) 4.2(t, 2H); 3.8(s, 3H); NOC.sub.2 H.sub.5 3.75(s, 3H)14 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3) 3.95(s, 3H); 3.8(s, 3H); NOCH.sub.3 3.75(s, 3H)15 2-CH.sub.3 -4-C(CH.sub.3)NO- 3.8(s, 3H); 3.75(s, 3H) trans-Cl-Allyl16 2-CH.sub.3 -4-C(CH.sub.3)N- 4.2(t, 2H); 3.8(s, 3H); OC.sub.2 H.sub.5 3.75(s, 3H)17 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5) 4.2(t, 2H); 3.8(s, 3H); NOC.sub.2 H.sub.5 3.75(s, 3H)______________________________________ TABLE 60______________________________________ ##STR285##No. B______________________________________1 Phenyl2 3-Phenoxyphenyl3 3-(2-Cyanophenoxy)-phenyl4 4-Chlorophenyl5 3-Trifluoromethylphenyl6 3-tert.-Butoxyphenyl7 3,5-Dichlorophenyl8 3,5-Diethylphenyl9 2-Pyridyl10 4-Pyrimidinyl11 6-Phenoxy-pyrimidin-4-yl12 6-Chloropyrimidin-4-yl13 6-(2-Fluorophenoxy)-pyrimidin-4-yl14 6-(2-Methylphenoxy)-pyrimidin-4-yl15 6-(2-Cyanophenoxy)-pyrimdin-4-yl16 6-(2,6-Difluorophenoxy)-pyrimidin-4-yl______________________________________

The novel compounds are suitable as fungicides.

The fungicidal compounds according to the invention, or agents containing them, may be applied for instance in the form of directly sprayable solutions, powders, suspensions (including high-percentage aqueous, oily or other suspen- sions), dispersions, emulsions, oil dispersions, pastes, dusts, broadcasting agents, or granules by spraying, atomizing, d usting, broadcasting or watering. The forms of application depend entirely on the purpose for which the agents are being used, but they must ensure as fine a distribution of the active ingredients according to the invention as possible. Normally, the plants are sprayed or dusted with the active ingredients, or the seeds of the plants are treated with the active ingredients.

The formulations are produced in known manner, for example by extending the active ingredient with solvents and/or carriers, with or without the use of emulsifiers and dispersants; if water is used as solvent, it is also possible to employ other organic solvents as auxiliary solvents. Suitable auxiliaries for this purpose are solvents such as aromatics (e.g., xylene), chlorinated aromatics (e.g., chlorobenzenes), paraffins (e.g., crude oil fractions), alcohols (e.g., methanol, butanol), ketones (e.g., cyclohexanone), amines (e.g., ethanolamine, dimethylformamide), and water; carriers such as ground natural minerals (e.g., kaolins, aluminas, talc and chalk) and ground synthetic minerals (e.g., highly disperse silica and silicates); emulsifiers such as nonionic and anionic emulsifiers (e.g., polyoxyethylene fatty alcohol ethers, alkyl sulfonates and aryl sulfonates); and dispersants such as lignin-sulfite waste liquors and methylcellulose.

Examples of surfactants are: alkali metal, alkaline earth metal and ammonium salts of aromatic sulfonic acids, e.g., ligninsulfonic acid, phenolsulfonic acid, naphthalenesulfonic acid and dibutylnaphthalenesulfonic acid, and of fatty acids, alkyl and alkylaryl sulfonates, and alkyl, lauryl ether and fatty alcohol sulfates, and salts of sulfated hexadecanols, heptadecanols, and octadecanols, salts of fatty alcohol glycol ethers, condensation products of sulfonated naphthalene and naphthalene derivatives with formaldehyde, condensation products of naphthalene or naphthalenesulfonic acids with phenol and formaldehyde, polyoxyethylene octylphenol ethers, ethoxylated isooctylphenol, ethoxylated octylphenol and ethoxylated nonylphenol, alkylphenol polyglycol ethers, tributylphenyl polyglycol ethers, alkylaryl polyether alcohols, isotridecyl alcohol, fatty alcohol ethylene oxide condensates, ethoxylated castor oil, polyoxyethylene alkyl ethers, ethoxylated polyoxypropylene, lauryl alcohol polyglycol ether acetal, sorbitol esters, lignin-sulfite waste liquors and methyl cellulose.

Powders, dusts and broadcasting agents may be prepared by mixing or grinding the active ingredients with a solid carrier.

Granules, e.g., coated, impregnated or homogeneous granules, may be prepared by bonding the active ingredients to solid carriers. Examples of solid carriers are mineral earths such as silicic acids, silica gels, silicates, talc, kaolin, attapulgus clay, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate, magnesium sulfate, magnesium oxide, ground plastics, fertilizers such as ammonium sulfate, ammonium phosphate, ammonium nitrate, and ureas, and vegetable products such as grain meals, bark meal, wood meal, and nutshell meal, cellulosic powders, etc.

Examples of formulations are given below.

I. A solution of 90 parts by weight of the compound from Table 7, No. 1 (7/1) and 10 parts by weight of N-methyl-.alpha.-pyrrolidone, which is suitable for application in the form of very fine drops.

II. A mixture of 20 parts by weight of compound 7/2, 80 parts by weight of xylene, 10 parts by weight of the adduct of 8 to 10 moles of ethylene oxide and 1 mole of oleic acid-N-monoethanolamide, 5 parts by weight of the calcium salt of dodecylbenzenesulfonic acid, and 5 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil. By finely dispersing the mixture in water, a dispersion is obtained.

III. An aqueous dispersion of 20 parts by weight of compound 7/3, 40 parts by weight of cyclohexanone, 30 parts by weight of isobutanol, 20 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil.

IV. An aqueous dispersion of 20 parts by weight of compound 7/4, 25 parts by weight of cyclohexanol, 65 parts by weight of a mineral oil fraction having a boiling point between 210.degree. and 280.degree. C., and 10 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil.

V. A hammer-milled mixture of 80 parts by weight of compound 7/5, 3 parts by weight of the sodium salt of diisobutylnaphthalene-.alpha.-sulfonic acid, 10 parts by weight of the sodium salt of a lignin-sulfonic acid obtained from a sulfite waste liquor, and 7 parts by weight of powdered silica gel. By finely dispersing the mixture in water, a spray liquor is obtained.

VI. An intimate mixture of 3 parts by weight of compound 7/6 and 97 parts by weight of particulate kaolin. The dust contains 3wt % of the active ingredient.

VII. An intimate mixture of 30 parts by weight of compound 7/7, 92 parts by weight of powdered silica gel and 8 parts by weight of paraffin oil sprayed onto the surface of this silica gel. This formulation of the active ingredient exhibits good adherence.

VIII. A stable aqueous dispersion of 40 parts by weight of compound 7/8, 10 parts of the sodium salt of a phenolsulfonic acid-urea-formaldehyde condensate, 2 parts of silica gel and 48 parts of water, which dispersion can be further diluted.

IX. A stable oily dispersion of 20 parts by weight of compound 7/9, 2 parts by weight of the calcium salt of dodecylbenzenesulfonic acid, 8 parts by weight of a fatty alcohol polyglycol ether, 2 parts by weight of the sodium salt of a phenolsulfonic acid-urea-formaldehyde condensate and 68 parts by weight of a paraffinic mineral oil.

The novel compounds are extremely effective on a broad spectrum of phytopathogenic fungi, in particular those from the class consisting of the Ascomycetes and Basidiomycetes. Some of them have a systemic action and can be used as foliar and soil fungicides.

The fungicidal compounds are of particular interest for controlling a large number of fungi in various crops or their seeds, especially wheat, rye, barley, oats, rice, Indian corn, lawns, cotton, soybeans, coffee, sugar cane, fruit and ornamentals in horticulture and viticulture, and in vegetables such as cucumbers, beans and cucurbits.

The compounds are applied by treating the fungi, or the seeds, plants, materials or soil to be protected against fungus attack with a fungicidally effective amount of the active ingredients.

The agents may be applied before or after infection of the materials, plants or seed by the fungi.

The compounds I are particularly useful for controlling the following plant diseases:

Erysiphe graminis in cereals, Erysiphe cichoracearum and Sphaerotheca fuliginea in cucurbits, Podosphaera leucotricha in apples, Uncinula necator in vines, Puccinia species in cereals, Rhizoctonia solani in cotton, Ustilago species in cereals and sugar cane, Venturia inaequalis (scab) in apples, Helminthosporium species in cereals, Septoria nodorum in wheat, Botrytis cinerea (gray mold) in strawberries and grapes, Cercospora arachidicola in groundnuts, Pseudocercosporella herpotrichoides in wheat and barley, Pyricularia oryzae in rice, Phytophthora infestans in potatoes and tomatoes, Fusarium and Verticillium species in various plants, Plasmopara viticola in grapes, Alternaria species in fruit and vegetables.

The novel compounds may also be used for protecting materials (timber), for instance against Paecilomyces variotii.

The fungicidal agents generally contain from 0.1 to 95, an preferably from 0.5 to 90, wt % of active ingredient.

The application rates depend on the effect desired, and are from 0.02 to 3 kg of active ingredient per hectare.

When the active ingredients are used for treating seed, amounts of from 0.001 to 50, and preferably from 0.01 to 10, g per kg of seed are generally needed.

When the agents according to the invention are used as fungicides, they may be present together with other active ingredients, e.g., herbicides, insecticides, growth regulators, other fungicides, and fertilizers.

When they are mixed with other fungicides, the spectrum of fungicidal action is in many cases increased.

USE EXAMPLES

The active ingredients used for comparison purposes were isopropyl N-phenylcarbamate (A)--known from GB 574 995--, isopropyl N-3-chlorophenylcarbamate (B)--known from GB 574 995 --and methyl N-3,4-dichlorophenylcarbamate (C)--known from BE 612 550.

Example 1

Action on wheat mildew

Leaves of pot-grown wheat seedlings of the "Fruhgold" variety were sprayed with aqueous liquors containing (dry basis) 80% of active ingredient and 20% of emulsifier, and dusted, 24 hours after the sprayed-on layer had dried, with spores of wheat mildew (Erysiphe graminis var. tritici). The plants were then set up in the greenhouse at from 20.degree. to 22.degree. C. and a relative humidity of from 75 to 80%. The extent of mildew spread was assessed after 7 days.

The results show that active ingredients nos. 1, 2, 3, 4, 8, 9, 20, 23, 31, 33, 34, 35, 36, 42, 43, 44, 47, 48, 52, 53, 54, 55, 56, 57, 60, 61, 62, 63, 64, 67, 69, 70, 71, 72, 74, 78, 79, 85, 87, 89, 90, 91, 92, 93, 94, 95, 104, 105, 106 and 107 from Table 7 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (95%) than prior art comparative agents A (45%), B (45%) and C (45%).

Example 2

Action on Pyricularia oryzae (protective)

Leaves of pot-grown rice seedlings of the "Bahia" variety were sprayed to runoff with aqueous emulsions containing (dry basis) 80% of active ingredient and 20% of emulsifier, and inoculated 24 hours later with an aqueous spore suspension of Pyricularia oryzae. The plants were then set up in climatic cabinets at 22.degree. to 24.degree. C. and 95 to 99% relative humidity. The extent of fungus attack was assessed after 6 days.

The results show that active ingredients nos. 1, 2, 12, 18, 19, 22, 29, 39, 40, 42, 47, 49, 50, 52, 53, 54, 60, 61, 62, 63, 69, 70, 71, 72, 73, 74, 81, 83, 85, 87, 89, 90, 91, 92, 94, 95, 104, 105, 106 and 107 from Table 7 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (95%) than prior art comparative agents A (30%), B (30%) and C (30%).

Example 3

Action on wheat mildew

Leaves of pot-grown wheat seedlings of the "Fruhgold" variety were sprayed with aqueous liquors containing (dry basis) 80% of active ingredient and 20% of emulsifier, and dusted, 24 hours after the sprayed-on layer had dried, with spores of wheat mildew (Erysiphe graminis var. tritici). The plants were then set up in the greenhouse at from 20.degree. to 22.degree. C. and a relative humidity of from 75 to 80%. The extent of mildew spread was assessed after 7 days.

The results show that active ingredient no. 3 from Table 14, nos. 3 and 4 from Table 21, nos. 1, 3, 4, 5, 6, 7, 8, 9, 10, 11, 15, 17, 18, 19, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 31, 32, 33, 34, 35, 36, 37, 38, 39, 40 41, 42, 43 and 44 from Table 48, nos. 7, 8, 9, 10, 11, 13, 14, 15, 16, 17, 18, 20 and 23 from Table 14, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18 and 19 from Table 52, and nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16 and 17 from Table 53 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (100%) than prior art comparative agents A, B and C (15%).

Example 4

Action on Pyricularia oryzae (protective)

Leaves of pot-grown rice seedlings of the "Bahia" variety were sprayed to runoff with aqueous emulsions containing (dry basis) 80% of active ingredient and 20% of emulsifier, and inoculated 24 hours later with an aqueous spore suspension of Pyricularia oryzae. The plants were then set up in climatic cabinets at 22.degree. to 24.degree. C. and 95 to 99% relative humidity. The extent of fungus attack was assessed after 6 days.

The results show that active ingredient nos. 3, 7, 8, 9, 10, 11, 13, 14, 15, 16, 17, 18, 20, 21, 22 and 24 from Table 14, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18, 19 and 20 from Table 52, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16 and 17 from Table 53, nos. 3 and 4 from Table 21, nos. 4 and 5 from Table 38, nos. 4, 7, 10, 16, 20, 21, 22, 23, 24, 25, 41, 42, 55, 56, 57, 58 and 59 from Table 47, and nos. 1, 4, 5, 6, 7, 8, 11, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 31, 32, 33, 34, 35, 36, 37, 38, 39, 40, 41, 42, 43 and 44 from Table 48 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (100%) than prior art comparative agents A, B and C (0%).

Use Example 5

Action on Botrytis cinerea

Paprika seedlings of the "Neusiedler Ideal Elite" variety were sprayed, after 4 to 5 leaves were well developed, to runoff with aqueous suspensions containing (dry basis) 80% of active ingredient and 20% of emulsifier. After the sprayed-on layer had dried, the plants were sprinkled with a conidial suspension of the fungus Botrytis cinerea, and placed at 22.degree. to 24.degree. C. in a chamber of high humidity. After 5 days, the disease had spread to such a great extent on the untreated plants that the necroses covered the major portion of the leaves.

______________________________________ Percentage leaf attack after spraying with aqueous formu- lations containing 500 ppmActive ingredient of active ingredient______________________________________Table 30, active ingr. no. 2 5Comparative substance A 100Comparative substance B 100Comparative substance C 100Untreated 100______________________________________

Use Example 6

Action on Plasmopara viticola

Leaves of potted vines of the Muller-Thurgau variety were sprayed with aqueous suspensions containing (dry basis) 80% of active ingredient and 20% of emulsifier. To assess the duration of action, the plants were set up, after the sprayed-on layer had dried, for 8 days in the greenhouse. Then the leaves were infected with a zoospore suspension of Plasmopara viticola. The plants were first placed for 48 hours in a water vapor-saturated chamber at 24.degree. C. and then in a greenhouse for 5 days at from 20.degree. to 30.degree. C. To accelerate and intensify the sporangiophore discharge, the plants were then again placed in the moist chamber for 16 hours. The extent of fungus attack was then assessed on the undersides of the leaves.

______________________________________ Percentage leaf attack after applying aqueous formu- lations containing 500 ppmActive ingredient of active ingredient______________________________________Table 21, active ingr. no. 3 5Table 21, active ingr. no. 4 0Table 30, active ingr. no. 1 15Comparative substance A 65______________________________________ ______________________________________ Percentage leaf attack after applying aqueous formula- tions containing 500 ppm ofActive ingredient active ingredient______________________________________Comparative substance B 40Comparative substance C 25Untreated 65______________________________________

Claims

1. A compound of the formula I ##STR286## where Z is a trifluoromethyl, trichloromethyl, methoxy, amino, methylamino or dimethylamino;

X,Y are hydrogen, fluoro, chloro, bromo, trifluoromethyl, cyano, nitro, alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, or

X,Y together form a substituted aromatic, alicyclic, partially or completely hydrogenated ring;

R.sup.1 is alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, cycloalkenyloxy, or alkoxycarbonyloxy;

A is a single bond, O, S, CR.sup.2 .dbd.CR.sup.3, CHR.sup.2 O, CHR.sup.2 S, CHR.sup.2 --ON.dbd.CR.sup.4, CR.sup.2 .dbd.NO, ON.dbd.CR.sup.4, C.tbd.C, CHR.sup.2 --CHR.sup.3, CHR.sup.2 O--CO, or OCHR.sup.2 ;

B is hydrogen, optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, arylalkyl, cycloalkylalkyl, or cycloalkenylalkyl;

R.sup.2,R.sup.3 are hydrogen, alkyl, alkenyl, alkynyl, or cycloalkyl;

R.sup.4 is hydrogen, cyano, alkyl, alkenyl, alkynyl, alkoxy, or cycloalkyl;

provided that B is not hydrogen when A denotes a single bond.

2. The compound of claim 1, wherein X and/or Y denote hydrogen.

3. The compound of claim 1, where

X,Y are hydrogen, fluoro, chloro, bromo, trifluoromethyl, cyano, nitro, C.sub.1 -C.sub.6 -alkylalkyl, C.sub.2 -C.sub.6 -alkenyl, C.sub.2 -C.sub.6 -alkynyl, C.sub.1 -C.sub.6 -alkoxy, C.sub.2 -C.sub.6 -alkenyloxy, C.sub.2 -C.sub.6 -alkynyloxy, or

X,Y together form a substituted aromatic or alicyclic partially or completely hydrogenated ring.

4. The compound of claim 1, where

R.sup.2 -R.sup.3 are hydrogen, C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.6 -alkenyl, C.sub.2 -C.sub.6 -alkynyl, or C.sub.3 -C.sub.10 -cycloalkyl; and

R.sup.4 is hydrogen, cyano, C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.6 -alkenyl, C.sub.2 -C.sub.6 -alkynyl, C.sub.1 -C.sub.6 -alkoxy, or C.sub.3 -C.sub.10 -cycloalkyl.

5. The compound of claim 1, where

R.sup.1 is C.sub.1 -C.sub.6 -alkoxy, C.sub.2 -C.sub.6 -alkenyloxy, C.sub.2 -C.sub.6 -alkynyloxy, C.sub.3 -C.sub.10 -cycloalkoxy, C.sub.3 -C.sub.10 -cycloalkenyloxy, or C.sub.1 -C.sub.6 -alkoxycarbonyloxy.

6. A compound of formula ##STR287## where Z is methoxy;

X,Y are hydrogen, fluoro, bromo, trifluoromethyl, cyano, nitro, alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, or

X,Y together form a substituted aromatic, alicyclic, partially or completely hydrogenated ring;

R.sup.1 is alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, cycloalkenyloxy, or alkoxycarbonyloxy;

A is a single bond, O, S, CR.sup.2 .dbd.CR.sup.3, CHR.sup.2 O, CHR.sup.2 S, CHR.sup.2 --ON.dbd.CR.sup.4, CR.sup.2 .dbd.NO, ON.dbd.CR.sup.4, C.tbd.C, CHR.sup.2 -CHR.sup.3, CHR.sup.2 --O--CO, or OCHR.sup.2 ;

B is hydrogen, optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, arylalkyl, cycloalkylalkyl, or cycloalkenylalkyl;

R.sup.2,R.sup.3 are hydrogen, alkyl, alkenyl, alkynyl, or cycloalkyl;

R.sup.4 is hydrogen, cyano, alkyl, alkenyl, alkynyl, alkoxy, or cycloalkyl; provided that B is not hydrogen when A denotes a single bond.

7. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 1, or a plant tolerated acid or base adduct thereof.

8. A process for combating fungi comprising the step of treating fungi, plants, seeds, soil or material threatened by fungal attack with a fungicidally effective amount of a compound of the compound of claim 1, or a plant-tolerated acid or base adduct thereof.

9. The compound of claim 1, wherein

B denotes hydrogen, or optional substituted C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.6 -alkenyl, C.sub.3 -C.sub.10 -cycloalkyl, C.sub.3 -C.sub.10 -cycloalkenyl, C.sub.3 -C.sub.10 -cycloalkynyl, aryl, aryl C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.10 -cycloalkyl-C.sub.1 -C.sub.6 -alkyl, or C.sub.3 -C.sub.10 -cycloalkenyl-C.sub.1 -C.sub.6 -alkyl .

10. The compound of claim 1, where R.sup.1 is C.sub.1 - or C.sub.2 -alkoxy.

11. The compound of claim 1, where Z is methoxy.

12. The compound of claim 1, where A is O, CH.dbd.CH, CH.sub.2 --O, CH.sub.2 --ON.dbd.CR.sup.4, or O--CH.sub.2, and R.sup.4 is hydrogen, cyano, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, or C.sub.3 -C.sub.6 -cycloalkyl.

13. The compound of claim 1, where B is unsubstituted or substituted aryl.

14. The compound of claim 1, where

R.sup.1 is C.sub.1- or C.sub.2 -alkoxy,

Z is methoxy,

A is O, CH.dbd.CH, CH.sub.2 --O, CH.sub.2 --ON.dbd.CR4, or O--CH.sub.2, and

R.sup.4 is hydrogen, cyano, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, or C.sub.3 -C.sub.6 -cycloalkyl, and

B is unsubstituted or substituted aryl.

15. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 10 or a plant tolerated acid or base adduct thereof.

16. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 11 or a plant tolerated acid or base adduct thereof.

17. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 12 or a plant tolerated acid or base adduct thereof.

18. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 13 or a plant tolerated acid or base adduct thereof.

19. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 14 or a plant tolerated acid or base adduct thereof.