Number | Name | Date | Kind |
---|---|---|---|
2634293 | Kyrides et al. | Apr 1953 | A |
2876236 | Szabo et al. | Mar 1959 | A |
3145209 | Krapcho | Aug 1964 | A |
3975443 | Harper et al. | Aug 1976 | A |
4738803 | Roques et al. | Apr 1988 | A |
4751306 | Ciganek et al. | Jun 1988 | A |
4757151 | Horwell | Jul 1988 | A |
5039706 | Wilkerson | Aug 1991 | A |
5102667 | Dubroeucq et al. | Apr 1992 | A |
5137873 | Yankner | Aug 1992 | A |
5164372 | Matsuo et al. | Nov 1992 | A |
5187156 | Matsuo et al. | Feb 1993 | A |
5245046 | Youngdale et al. | Sep 1993 | A |
5350852 | Emonds-Alt et al. | Sep 1994 | A |
5530009 | Cho et al. | Jun 1996 | A |
5670499 | Cho et al. | Sep 1997 | A |
5684033 | Cho et al. | Nov 1997 | A |
Number | Date | Country |
---|---|---|
0 135 087 | Mar 1985 | EP |
0 224151 | Jun 1987 | EP |
0 230151 | Jul 1987 | EP |
0 336356 | Oct 1989 | EP |
0 443 132 | Aug 1991 | EP |
0 693 489 | Jan 1996 | EP |
1173833 | Dec 1969 | GB |
WO 9204038 | Mar 1992 | WO |
WO 9301169 | Jan 1993 | WO |
WO 9301170 | Jan 1993 | WO |
WO 9310073 | May 1993 | WO |
WO 9318023 | Sep 1993 | WO |
WO 9322279 | Nov 1993 | WO |
WO 9401402 | Jan 1994 | WO |
Entry |
---|
Kucharczyk et al, J. Med. Chem. 36 p 1654 (1993).* |
Rouissi et al, Biochemical and Biophysical Research Communications, 176, p. 894 (1991).* |
Hampel et al, Glossary of Chemical Terms (2nd Ed.) (Van Nostrand and Reinhold, Publ.) p. 55.* |
Kotelko, et al., Chemical Abstracts, vol. 104, No. 25 (1986), Abstract No. 224680a. |
Kotelko, et al., Chemical Abstracts, vol. 104, No. 25 (1986), Abstract No. 224681b. |
Jerry March, “Advanced Organic Chemistry,” 2nd Edition (1977), published by McGraw-Hill Book Co., pp. 383-384. |
I. Saito, et al., Chem. Ab., 73:110093 (1970), as searched in File CAPLUS. |
B.D. Gitter, et al., “Species Differences in Affinities of Non-Peptide Antagonists for Substance P Receptors”, European Journal of Pharmacology, 197:237-238 (1991). |
D. Jukic, et al., “Neurokinin Receptors Antagonists: Old and New”, Life Sciences, 49:1463-1469 (1991). |
C.A. Maggi, et al., “Tachykinin Receptors and Tachykinin Receptor Antagonists”, Journal of Autonomic Pharmacology, 13:23-93 (1993). |