Claims
- 1. A compound of the formula ##STR8## wherein X is O or S;
- Y is O or S;
- R.sup.1 is hydrogen, halogen, C.sub.1 -C.sub.4 alkyl or C.sub.1 -C.sub.4 alkoxy;
- R.sup.2 is hydrogen, halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.2 -C.sub.4 alkenyl, C.sub.2 -C.sub.4 alkenyloxy, C.sub.2 -C.sub.4 alkynyl, C.sub.2 -C.sub.4 alkynyloxy, mono-, di- or tri-halomethyl, trifluoromethoxy, C.sub.1 -C.sub.4 alkylthio, C.sub.3 -C.sub.4 branched alkylthio, nitro, or cyano;
- R.sup.3 is hydrogen, halogen, methyl, mono-, di- or tri-halomethyl;
- R.sup.4 is
- a) C.sub.3 -C.sub.8 cycloalkyl substituted by one or more C.sub.1 -C.sub.4 alkyl;
- or
- b) ##STR9## wherein R.sup.6 and R.sup.7 are independently, hydrogen or linear or branched, C.sub.1 -C.sub.4 alkyl, C.sub.2 -C.sub.4 alkenyl, or C.sub.2 -C.sub.4 alkynyl, and R.sup.8 is C.sub.3 -C.sub.8 cycloalkyl substituted by one or more C.sub.1 -C.sub.4 alkyl; and
- R.sup.5 is
- a) substituted or unsubstituted, linear or branched C.sub.1 -C.sub.8 alkyl, C.sub.2 -C.sub.8 alkenyl, C.sub.2 -C.sub.8 alkynyl or C.sub.1 -C.sub.8 mono- or di-alkylamino, C.sub.3 -C.sub.7 cycloalkyl, C.sub.3 -C.sub.7 cycloalkylalkoxy, C.sub.3 -C.sub.7 cycloalkenyl, unsubstituted or substituted by C.sub.1 -C.sub.6 alkyl; C.sub.7 -C.sub.10 phenylalkyl, C.sub.1 -C.sub.8 alkoxy, C.sub.1 -C.sub.8 alkoxycarbonyl, C.sub.1 -C.sub.8 mono-, di- or tri-haloalkoxy, C.sub.2 -C.sub.8 alkenyloxy, or C.sub.2 -C.sub.8 alkynyloxy;
- b) aryl, aralkyl, aryloxyalkyl, or cycloalkylaryloxy, wherein the alkyl moiety is C.sub.1 -C.sub.4, the cycloalkyl moiety is C.sub.3 -C.sub.8, and the aryl moiety is naphthyl, phenyl, or phenyl substituted by one or more halogen, carboxy, C.sub.1 -C.sub.8 alkyl, C.sub.1 -C.sub.8 haloalkyl, C.sub.1 -C.sub.8 alkylthio, phenyl, nitro, amino, C.sub.1 -C8 alkoxycarbonylamino, hydroxyl, acetyl, acetyloxy, phenoxy, or C.sub.1 -C.sub.8 alkylcarbonyl;
- or
- c) G--O--
- wherein G is a linear or branched, unsubstituted or halo-substituted, C.sub.1 -C.sub.8 alkyl, C.sub.2 -C.sub.8 alkenyl, or C.sub.2 -C.sub.8 alkynyl; a C.sub.3 -C.sub.7 cycloalkyl or cycloalkenyl, unsubstituted or substituted by C.sub.1 -C.sub.6 alkyl; a phenyl or phenyl substituted by halogen, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy, carboxyl, C.sub.1 -C.sub.8 alkylthio, phenyl, nitro, amino, hydroxyl, acetyl, acetyloxy, phenoxy, C.sub.1 -C.sub.8 alkoxycarbonyl, or C.sub.2 -C.sub.8, alkoxycarbonyl.
- 2. A compound as recited in claim 1 wherein R.sup.4 is
- a) 2,6-dimethylcyclohexyl, 2,5-dimethylcyclo-pentyl, 2,4-dimethylcyclobutyl, 2,3-dimethylcyclopropyl, 1-, 2- or 3-methylcyclopentyl, 1- or 2- methylcyclohexyl, 1-methylcyclobutyl, 1-methylcyclopropyl, or dicyclopropyl;
- or
- b) ##STR10## wherein R.sup.6 and R.sup.7 are independently hydrogen or C.sub.1 -C.sub.4 alkyl and R.sup.8 is 2,6-dimethylcyclohexyl, 2,5-dimethylcyclopentyl, 2,4-O dimethylcyclobutyl, 2,3-dimethylcyclopropyl, 1-, 2- or 3- methylcyclopentyl, 1- or 2- methylcyclohexyl, 1-methylcyclobutyl, 1-methylcyclopropyl, or dicyclopropyl.
- 3. A compound as recited in claim 2 wherein R.sup.1 is hydrogen, R.sup.2 is halogen, R.sup.3 is hydrogen, R.sup.4 is 1-, 2- or 3-methylcyclopentyl, 2,5-dimethylcyclopentyl or 2,6-dimethylcyclohexyl, and R.sup.5 is phenyl, halophenyl, phenylamino, phenylalkylamino, tolyl, or phenylmethoxy, unsubstituted or substituted by C.sub.1 -C.sub.3 alkyl.
- 4. A compound as recited in claim 3 wherein Y is O, R.sup.1 is hydrogen, R.sup.2 is chloro, R.sup.3 is hydrogen, and R.sup.5 is phenyl or 2-fluorophenyl.
- 5. A compound as recited in claim 2 wherein R.sup.1 is hydrogen, R.sup.2 is halogen, R.sup.3 is hydrogen, R.sup.4 is 1-, 2- or 3-methylcyclopentyl, 2,5-dimethylcyclopentyl or 2,6-dimethylcyclohexyl, and R.sup.5 is linear or branched C.sub.3 -C.sub.6 alkyl, C.sub.2 -C.sub.6 alkenyl or alkynyl, C.sub.1 -C.sub.8 alkoxy, C.sub.2 -C.sub.8 alkenyloxy, or C.sub.2 -C.sub.8 alkynyloxy; C.sub.3 -C.sub.7 cycloalkyl or C.sub.3 -C.sub.7 cycloalkenyl, unsubstituted or substituted by C.sub.1 -C.sub.6 alkyl; or C.sub.3 -C.sub.8 cycloalkyloxy.
Parent Case Info
This is a division of application Ser. No. 08/346,811, filed Nov. 30, 1994 now U.S. Pat. No. 5,550,280.
Non-Patent Literature Citations (1)
Entry |
Imagawa, et al., Osaka Kyoiku Diagaku Kiyo, Dia-3-bumon, 40(2) 169-74) ***Abstract***, 1992. |
Divisions (1)
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Number |
Date |
Country |
Parent |
346811 |
Nov 1994 |
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