Claims
- 1. A compound of the formula: ##STR8## where R is an aglycon of from 1 to 10 carbon atoms; and
- X.sub.2 is selected from sulfate and phosphate and pharmaceutical salts thereof.
- 2. The compound according to claim 1 wherein X.sub.2 is sulfate.
- 3. The compound according to claim 1 wherein X.sub.2 is phosphate.
- 4. The compound according to claim 2 wherein R is --(CH.sub.2).sub.8 COOCH.sub.3.
- 5. The compound according to claim 3 wherein R is --(CH.sub.2).sub.8 COOCH.sub.3.
- 6. A pharmaceutical composition suitable for administration to a mammal which composition comprises a pharmaceutically inert carrier and a sufficient amount of a compound of claim 1 so as to provide a dosage range of from about 0.5 mg to about 50 mg/kg of body weight when administered to said mammal.
- 7. The pharmaceutical composition according to claim 6 wherein X.sub.2 is sulfate.
- 8. The pharmaceutical composition according to claim 6 wherein X.sub.2 is phosphate.
- 9. The pharmaceutical composition according to claim 7 wherein R is --(CH.sub.2).sub.8 COOCH.sub.3.
- 10. The pharmaceutical composition according to claim 8 wherein R is --(CH.sub.2).sub.8 COOCH.sub.3.
Parent Case Info
This application is a continuation of application Ser. No. 07/895,930, filed Jun. 9, 1992, now abandoned; which is a continuation in part of application Ser. No. 07/889,017, filed May 26, 1992, now abandoned; which is a continuation-in-part of application Ser. No. 07/714,161, filed Jun. 10, 1991, currently pending. Each of these applications is incorporated herein by reference in its entirety.
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Number |
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895930 |
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Continuation in Parts (2)
|
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889017 |
May 1992 |
|
Parent |
714161 |
Jun 1991 |
|