Nicolaou et al., Nature, vol. 387, May 15, 1997, pp. 268-272.* |
Tolstikov et al., Tetrahedron Letters, No. 12, pp 1857-1858, 1978.* |
Schafer et al , Tetrahedron, vol. 18, No. 22, pp 3299-3308, 1982.* |
Raederstorff et al., The Journal of organic Chemistry, vol. 52, No. 12, pp. 2337-2346, Jun. 1987.* |
Andrade, Rodrigo B. et al., “Solid-Phase Oligosaccharide Synthesis: Preparation of Complex Structures Using a Novel Linker and Different Glycosylating Agents”, Organic Letters 1(11): 1811-1814 (1999). |
Hayashi, Nobuyuki et al., “The Biomimetic Construction of Fused Cyclic Polyethers”, Tetrahedron 53(37): 12425-12468 (1997). |
Jahn, Ullrich et al., “Towards a Tandem-Radical Macrocyclization-Transannular Cyclization Approach to Steroids: Transannular Cyclizations of a Macrocyclic Core”, Tetrahedron Letters 36(49): 8921-8924 (1995). |
Miura, Katsukiyo et al., “Highly Stereoselective Intramolecular Addition of a Hydroxyl Group to Vinylsilanes via 1,2-Silyl Migration”, J. Org. Chem. 62: 8292-8293 (1997). |
Raederstorff, Daniel et al., “Biosynthetic Studies of Marine Lipids. 11. Synthesis, Biosynthesis, and Absolute Configuration of the Internally Branched Demospongic Acid, 22-Methyl-5,9-Octacosadienoic Acid”, Journal of Organic Chemistry 52(12): 2337-2346 (Jun. 12, 1987). |
International Search Report Completed on Apr. 19, 2001 and Mailed on May 4, 2001. |
Arya, P. and Ben, N. R.; Angew. Chem. Int. Ed. Engl. 36 (12): 1280-1282 (1997). |
Boons et al.; “Vinyl Glycosides Oligosaccharide Synthesis: A Strategy for the Preparation of Trisaccharide Libraries Based on Latent-Active Glycosylation **”, Angew. Chem. Int. Ed. Engl. 35 (23/24) : 2845-2847 (1996). |
Ding et al.; “Synthesis and Bilogical Activity of Oligosaccharide Libraries”, Glycoimmunology, Edited by A. Alavi and J. S. Axford; Plenum Press New York, (1965); pp. 261-269. |
Frechet, M. J. and Schuerch, C. “Solid-Phase Synthesis of Oligosaccharides III. Preparation of Some Derivatives of Di- and Tri-Saccharides Via a Simple Alcoholysis Reaction”, Carbohydr. Res. 22 : 399-412 (1972). |
Fraser-Reid et al. ; “n-Pentenyl Glycosides in Organic Chemistry: A Contemporary Example of Serendipity”, Synlett pp. 927-942 ( Dec. 1992 ). |
Izumi, M. and Ichikawa, Y. “Combinatorial Synthesis of Oligosaccharide Library of 2.6-Dideoxysugars”, Tetrahedron Letters 39 : 2079-2082 (1998). |
Johnson et al.; “Vinyl Glycosides in Oligosaccharide Synthesis (Part 5)1: A Latent-Active Glycosylation Strategy for the Preparation of Branched Trisaccharide Libraries” Tetrahedron Letters 39 : 9801-9804 (1998). |
Liang et al.; “Parallel Synthesis and Screening of a Solid Phase Carbohydrate Library”, Science, 274 : 1520-1522 (Nov. 29, 1996). |
Nicolaou, K. C. et al.; “Solid and Solution Phase Synthesis and Biological Evaluation of Combinatorial Sarcodictyin Libraries”, J. Am. Chem. Soc. 120 : 10814-10826 (1998). |
Nicolaou, K.C. et al.; “Solid-Phase Synthesis of Oligosaccharides: Construction of a Dodecasaccharide**”, Angew. Chem. Int. Ed. 37 (11) : 1559-1561 (1998). |
Osborn and Khan; “Recent Developments in Polymer Supported Syntheses of Oligosaccharides and Glycopeptides”, Tetrahedron 55 : 1807-1850 (1999). |
Rademann, J. and Schmidt, R. R. ; “A New Method for the Solid Phase Synthesis of Oligosaccharides1”, Tetrahedron Letters 37 (23) : 3989-3990 (1996). |
Rodebaugh et al. ; “Polymer-Supported Oligosaccharides via n-Pentenyl Glycosides : Methodology for a Carbohydrate Library 1”, J. Org. Chem. 62 : 5660-5661 (1997). |
Scheffler, G. and Schmidt * R. R. “Glycosylation Reactions with a (4-Alkoxypentadienyl)oxy Leaving Group Linking the Glycosyl Donor and the Acceptor Moiety”, J. Org. Chem. 64 : 1319-1325 (1999). |
Schweizer, F. and Hindsgaul, O. “Combinatorial Synthesis of Carbohydrates”, Current Opinion in Chemical Biology 3 (3) : 291-298 (Jun. 1999). |
Sofia, M.J. et al. “Carbohydrate-Based Small-Molecule Scaffolds for the Construction of Universal Pharmacophore Mapping Libraries”, J. Org. Chem. 63: 2802-2803 ( 1998). |
Wang and Hindsgaul ; “Combinatorial Carbohydrate Chemistry”, Glycoimmunology 2, Edited by Axford; Plenum Press, New York, pp. 219-236 (1998). |
Wunberg et al.; “Carbohydrates as Multifunctional Chiral Scaffolds in Combinatorial Synthesis”, Angew. Chem. Int. Ed. 37 (18) : 2503-2505 (1998). |