This Application is a provisional of Ser. No. 60/026,945 filed Sep. 24, 1996.
Filing Document | Filing Date | Country | Kind | 102e Date | 371c Date |
---|---|---|---|---|---|
PCT/US97/16624 | WO | 00 | 3/24/1999 | 3/24/1999 |
Publishing Document | Publishing Date | Country | Kind |
---|---|---|---|
WO98/13461 | 4/2/1998 | WO | A |
Number | Name | Date | Kind |
---|---|---|---|
4261868 | Hora et al. | Apr 1981 | |
4318818 | Letton et al. | Mar 1982 | |
4399065 | Bajusz et al. | Aug 1983 | |
4404115 | Tai | Sep 1983 | |
4529525 | Dormal et al. | Jul 1985 | |
4537706 | Severson, Jr. | Aug 1985 | |
4537707 | Severson, Jr. | Aug 1985 | |
4566985 | Bruno et al. | Jan 1986 | |
4652552 | Kettner et al. | Mar 1987 | |
4703036 | Bajusz et al. | Oct 1987 | |
5030378 | Venegas | Jul 1991 | |
5234829 | Brown | Aug 1993 | |
5284829 | McKerrow et al. | Feb 1994 | |
5527487 | Mikkelsen et al. | Jun 1996 |
Number | Date | Country |
---|---|---|
0 130 756 | Jan 1985 | EP |
0 185 390 | Jun 1986 | EP |
0 293 881 | Dec 1988 | EP |
0 376 705 | Jul 1990 | EP |
0 381 262 | Aug 1990 | EP |
0583535 | Mar 1992 | EP |
0 473 502 | Mar 1992 | EP |
0 511 456 | Nov 1992 | EP |
0 583 536 | Feb 1994 | EP |
0 583 534 | Feb 1994 | EP |
0 583 535 | Feb 1994 | EP |
90029670 | Sep 1983 | JP |
9203529 | Mar 1992 | WO |
WO 9203529 | Mar 1992 | WO |
WO 9205239 | Apr 1992 | WO |
WO 9300418 | Jan 1993 | WO |
WO 9313125 | Jul 1993 | WO |
WO 9404651 | Mar 1994 | WO |
WO 9404652 | Mar 1994 | WO |
WO 9524914 | Sep 1995 | WO |
Entry |
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Bajusz et al., “Inhibition of Thrombin and Trypsin by Tripeptide Aldehydes”, Int. J. Peptide Protein Res., vol. 12, pp. 217-221 (1978). |
Nagy et al., “Tripeptide Aldehyde Protease Inhibitors May Depress in Vitro Proclactin and Growth Hormone Release”, Endocrinology, vol. 116, No. 4, pp. 1426-1432, (1985). |
Number | Date | Country | |
---|---|---|---|
60/026945 | Sep 1996 | US |