Claims
- 1. A compound of formula Ia:
- 2. A method for preparing a resin-bound compound of Formula [7]:
- 3. A method of claim 2, which further comprises:
(a) coupling 2-(4-formylphenoxy)acetic acid to a polymeric resin support having a free amino group; and (b) activating the resin-bound 2-(4-formylphenoxy) acetate as an acetal to provide the activated polymeric resin support of Formula [6].
- 4. The method of claim 3 wherein the polymeric resin support is aminomethyl polystyrene uniform beads.
- 5. A method for preparing a resin-bound compound of Formula [4]
- 6. The method of claim 5 wherein the polymeric resin support is aminomethyl polystyrene uniform beads.
- 7. A method for preparing a library of compounds of Formula I
- 8. A library of compounds prepared by the method of claim 7 for screening for inhibiting Mur enzymes.
- 9. A pharmaceutical composition which is comprised of a compound in accordance with claim 1 in combination with a carrier.
- 10. A method of treating a bacterial infection in a mammalian patient in need of such treatment which is comprised of administering to said patient a compound in accordance with claim 1 in an amount which is effective for treating a bacterial infection.
CROSS-REFERENCE TO RELATED APPLICATION
[0001] This application claims the benefit of U.S. Provisional Application No. 60/398,981, filed Jul. 26, 2002.
Provisional Applications (1)
|
Number |
Date |
Country |
|
60398981 |
Jul 2002 |
US |