Claims
- 1. A compound of the formula: ##STR5## wherein: R.sub.1 is C.sub.1 -C.sub.3 dialkylamino-C.sub.2 -C.sub.5 alkyl;
- R.sub.2 is selected from the group consisting of hydrogen, C.sub.1 -C.sub.3 alkyl and C.sub.1 -C.sub.3 dialkylamino-C.sub.2 -C.sub.5 alkyl;
- R.sub.3 is selected from the group consisting of hydrogen, halogen and methyl; and
- R.sub.4 is selected from the group consisting of hydrogen, methyl, methoxy and chloro
- and pharmaceutically acceptable salts of such compounds.
- 2. The compound of claim 1, which is 1-[N-methyl-N-(2'-dimethylaminoethyl)-amino]-3-phenyl indole or a pharmacologically acceptable salt thereof.
- 3. The compound of claim 2, which is 1-[N-methyl-N-(2'-dimethylaminoethyl)-amino]-3-phenyl indole hydrochloride.
- 4. The compound of claim 1, which is 1-[N-methyl-N-(3'-dimethylaminopropyl)-amino]-3-phenyl indole or a pharmacologically acceptable salt thereof.
- 5. A compound of claim 1, wherein R.sub.2 is methyl.
- 6. A compound of claim 1, wherein said dialkylamino alkyl radical of R.sub.1 and R.sub.2 is C.sub.1 -C.sub.3 dialkylamino-C.sub.2 -C.sub.3 alkyl.
- 7. The compound of claim 1, which is 1-[N-methyl-N-(2'-diethylaminoethyl)-amino]-3-phenyl indole or a pharmacologically acceptable salt thereof.
- 8. The compound of claim 1, which is 1-[N-methyl-N-(2'-dimethylaminoethyl)-amino]-3-(4'-methoxyphenyl)-indole or a pharmacologically acceptable salt thereof.
Priority Claims (1)
Number |
Date |
Country |
Kind |
4339/74 |
Mar 1974 |
CHX |
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Parent Case Info
This application is a continuation of Application Ser. No. 813,856, filed July 8, 1977, which is a continuation of Application Ser. No. 565,739, filed Mar. 31, 1975, both of which are abandoned.
Non-Patent Literature Citations (6)
Entry |
Meyer, J. Chem. Soc. 1965, 3451-3454. |
Arguzov, J. Gen. Chem. USSR (1957) 9, 2341-2354. |
Schatz et al., Chem. Abs. 84, 30886 (1975). |
Jones, J.C.S. Perkins I, 2728-2731 (1972). |
Somei et al., I. Tet Letters 461-462 (1974). |
Somei et al. II Tet Letters 3605-3608 (1974). |
Continuations (2)
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Number |
Date |
Country |
Parent |
813856 |
Jul 1977 |
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Parent |
565739 |
Mar 1975 |
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