Claims
- 1. A compound having the formula: ##STR5## Wherein: R.sup.1, R.sup.2, R.sup.3 and R.sup.4 are hydrogen,
- X is --CH.sub.2 -- or --CH.dbd.CH--
- R is ##STR6## and a non-toxic pharmaceutically acceptable salt thereof.
- 2. The compound of claim 1 selected from the group consisting of:
- N-(6-benzoxazolinyl-2-one)-anti-tricyclo[4.2.2.0.sup.2,5 ]-dec-3,9-diene-endo-7,-endo-8-dicarboximide;
- N-(6-benzoxazolinyl-2-one)-anti-tricyclo[3.2.2.0.sup.2,4 ]non-8-ene-endo-6,endo-7-dicarboximide;
- N-(5-benzoxazolinyl-2-one)-anti-tricyclo[4.2.2.0.sup.2,5 ]dec-3,9-diene-endo-7,endo-8-dicarboximide;
- N-(5-benzoxazolinyl-2-one)-anti-tricyclo[3.2.2.0.sup.2,4 ]non-8-ene-endo-6,endo-7-dicarboximide.
- 3. A tranquilizing pharmaceutical composition comprising a therapeutically effective amount in unitary dosage form of a compound having the formula: ##STR7## Wherein: R.sup.1, R.sup.2, R.sup.3 and R.sup.4 are hydrogen,
- X is --CH.sub.2 -- or --CH.dbd.CH--
- R is ##STR8## and a non-toxic pharmaceutically acceptable salt thereof.
- 4. A method of producing a tranquilizing effect comprising administering to a patient in need of such a treatment a therapeutically effective amount in unitary dosage form of a compound having the formula: ##STR9## Wherein: R.sup.1, R.sup.2, R.sup.3 and R.sup.4 are hydrogen,
- X is --CH.sub.2 -- or --CH.dbd.CH--
- R is ##STR10## and a non-toxic pharmaceutically acceptable salt thereof.
Parent Case Info
This is a division of application Ser. No. 713,765 filed Aug. 12, 1976, now U.S. Pat. No. 4,061,763, which is a division of application Ser. No. 575,918 filed May 9, 1975, now U.S. Pat. No. 4,006,233, which in turn is a continuation-in-part of co-pending application Ser. No. 511,961, filed Oct. 4, 1974, now abandoned.
US Referenced Citations (4)
Number |
Name |
Date |
Kind |
3126395 |
Kitahonoki et al. |
Mar 1964 |
|
3476546 |
Roberts et al. |
Nov 1969 |
|
3625946 |
Koch et al. |
Dec 1971 |
|
3770761 |
Bretschneider et al. |
Nov 1973 |
|
Foreign Referenced Citations (2)
Number |
Date |
Country |
1111635 |
Jul 1961 |
DEX |
2226397 |
Nov 1974 |
FRX |
Divisions (2)
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Number |
Date |
Country |
Parent |
713765 |
Aug 1976 |
|
Parent |
575918 |
May 1975 |
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Continuation in Parts (1)
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Number |
Date |
Country |
Parent |
511961 |
Oct 1974 |
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