Phosphoric benzoyl derivatives and their use as herbicides

The present invention relates to phosphorus-containing benzoyl derivatives of the formula I

in which:

X is oxygen or sulfur;

R

1

,R

2

are hydrogen, C

1

-C

6

-alkyl, C

2

-C

6

-alkenyl, C

2

-C

6

-alkynyl, hydroxyl, C

1

-C

6

-alkoxy, C

3

-C

6

-alkenyloxy, C

3

-C

6

-alkynyloxy, mercapto, C

1

-C

6

-alkylthio, C

3

-C

6

-alkenylthio, C

3

-C

6

-alkynylthio, amino, C

1

-C

6

-alkylamino, di(C

1

-C

6

-alkyl)amino, (C

1

-C

6

-alkoxy)(C

1

-C

6

-alkyl)amino, (C

3

-C

6

-alkenyl)(C

1

-C

6

-alkyl)amino, (C

3

-C

6

-alkynyl)(C

1

-C

6

-alkyl)amino, di(C

3

-C

6

-alkenyl)amino or di(C

3

-C

6

-alkynyl)amino, where the abovementioned alkyl, alkenyl or alkynyl radicals may be partially or fully halogenated and/or may carry one to three of the following groups: nitro, cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio, C

1

-C

4

-alkylsulfinyl, C

1

-C

4

-alkylsulfonyl, di(C

1

-C

4

-alkyl)amino, C

1

-C

4

-alkylcarbonyl, C

1

-C

4

-alkoxycarbonyl, phenyl or heterocyclyl, where the the two last-mentioned radicals for their part may be partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl;

are phenyl or phenoxy which may be partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl; or

R

1

and R

2

together form an —O—(CH

2

)

m

—O—, —O—(CH

2

)

m

—S—, —S—(CH

2

)

m

—S—, —NR

5

—(CH

2

)

m

—NR

5

—, —O—(CH

2

)

m

—NR

5

—, —S—(CH

2

)

m

—NR

5

—, —(CH

2

)

n

—O—, —(CH

2

)

n

—S— or —(CH

2

)

n

—NR

5

chain which may carry one to three radicals from the following group:

halogen, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-alkoxycarbonyl or phenyl which is unsubstituted or partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl; or

R

1

and R

2

together form a —(CH

2

)

p

chain which may be interrupted by oxygen, sulfur or NR

5

and/or may carry one to three radicals from the following group:

halogen, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-alkoxycarbonyl or phenyl which is unsubstituted or partially or fully halogenated and/or may carry one to three of the following groups: nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl;

R

3

is hydrogen, nitro, cyano, halogen, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, C

1

-C

6

-alkoxy-C

1

-C

6

-alkyl, C

1

-C

6

-haloalkoxy-C

1

-C

6

-alkyl, C

1

-C

6

-alkylthio-C

1

-C

6

-alkyl, C

1

-C

6

-alkylsulfinyl-C

1

-C

6

-alkyl, C

1

-C

6

-alkylsulfonyl-C

1

-C

6

-alkyl, C

1

-C

6

-alkylcarbonyl, C

1

-C

6

-alkoxycarbonyl, C

1

-C

6

-alkoxy, C

1

-C

6

-haloalkoxy, C

1

-C

6

-alkylthio, C

1

-C

6

-haloalkylthio, C

1

-C

6

-alkylsulfinyl, C

1

-C

6

-haloalkylsulfinyl, C

1

-C

6

-alkylsulfonyl, C

1

-C

6

-haloalkylsulfonyl, aminosulfonyl, C

1

-C

6

-alkylaminosulfonyl, di(C

1

-C

6

-alkyl)aminosulfonyl, (C

1

-C

6

-alkylsulfonyl)amino, (C

1

-C

6

-haloalkylsulfonyl)amino, N—(C

1

-C

6

-alkyl)—N—(C

1

-C

6

-alkylsulfonyl)amino, N—(C

1

-C

6

-alkyl)—N—(C

1

-C

6

-haloalkylsulfonyl)amino, —P(═X)R

1

R

2

, phenyl or heterocyclyl, where the two last-mentioned radicals may be partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl;

R

4

is nitro, cyano, halogen, C

1

-C

6

-alkyl, C

1

-C

6

-alkoxy, C

1

-C

6

-alkylthio, C

1

-C

6

-alkylsulfinyl or C

1

-C

6

-alkylsulfonyl;

R

5

is hydrogen, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl or C

1

-C

6

-alkoxy;

l is 0, 1 or 2;

m is 2, 3 or 4;

n is 3, 4 or 5;

p is 4, 5 or 6;

Q is a radical of the formula Q

1

, Q

2

, Q

3

or Q

4

R

6

is hydroxyl, mercapto, halogen, OR

13

, SR

13

, SOR

14

, SO

2

R

14

, OSO

2

R

14

, POR

15

R

16

, OPR

15

R

16

, OPOR

15

R

16

, OPSR

15

R

16

, NR

17

R

18

, ONR

18

R

19

, N-bonded heterocyclyl or O—(N-bonded heterocyclyl), where the heterocyclyl radical of the two last-mentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

7

,R

9

,R

11

are hydrogen, nitro, halogen, cyano, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, di(C

1

-C

6

-alkoxy)methyl, di(C

1

-C

6

-alkylthio)methyl, (C

1

-C

6

-alkoxy)(C

1

-C

6

-alkylthio)methyl, hydroxyl, C

1

-C

6

-alkoxy, C

1

-C

6

-haloalkoxy, C

1

-C

6

-alkoxycarbonyloxy, C

1

-C

6

-alkylthio, C

1

-C

6

-haloalkylthio, C

1

-C

6

-alkylsulfinyl, C

1

-C

6

-haloalkylsulfinyl, C

1

-C

6

-alkylsulfonyl, C

1

-C

6

-haloalkylsulfonyl, C

1

-C

6

-alkylcarbonyl, C

1

-C

6

-haloalkylcarbonyl, C

1

-C

6

-alkoxycarbonyl or C

1

-C

6

-haloalkoxycarbonyl;

R

8

,R

10

,R

12

are hydrogen, C

1

-C

6

-alkyl, C

1

-C

6

-alkoxy, C

1

-C

6

-alkylthio or C

1

-C

6

-alkoxycarbonyl; or

R

7

and R

8

or R

9

and R

10

or R

11

and R

12

together form an —O—(CH

2

)

u

—O—, —O—(CH

2

)

u

—S—, —S—(CH

2

)

u

—S—, —O—(CH

2

)

v

— or —S—(CH

2

)

v

chain which may be substituted by one to three radicals from the following group:

halogen, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl or C

1

-C

4

-alkoxycarbonyl; or

R

7

and R

8

or R

9

and R

10

or R

11

and R

12

together form a —(CH

2

)

w

chain which may be interrupted by oxygen or sulfur and/or may be substituted by one to four radicals from the following group:

halogen, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl or C

1

-C

4

-alkoxycarbonyl; or

R

7

and R

8

or R

9

and R

10

or R

11

and R

12

together form a methylidene group which may be substituted by one to two radicals from the following group:

halogen, hydroxyl, formyl, cyano, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, C

1

-C

6

-alkoxy, C

1

-C

6

-haloalkoxy, C

1

-C

6

-alkylthio, C

1

-C

6

-haloalkylthio, C

1

-C

6

-alkylsulfinyl, C

1

-C

6

-haloalkylsulfinyl, C

1

-C

6

-alkylsulfonyl or C

1

-C

6

-haloalkylsulfonyl; or

R

7

and R

8

or R

9

and R

10

or R

11

and R

12

together with the carbon atom to which they are attached form a carbonyl group; or

R

7

and R

9

or R

9

and R

11

or R

7

and R

11

together form a —(CH

2

)

v

chain which may be substituted by one to three radicals from the following group:

halogen, C

1

-C

6

-alkyl, C

1

-C

6

-alkoxy, hydroxyl or C

1

-C

6

-alkoxycarbonyl;

R

13

is C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-alkynyl, C

3

-C

6

-haloalkynyl, C

3

-C

6

-cycloalkyl, C

1

-C

20

-alkylcarbonyl, C

2

-C

6

-alkenylcarbonyl, C

2

-C

6

-alkynylcarbonyl, C

3

-C

6

-cycloalkylcarbonyl, C

1

-C

6

-alkylaminocarbonyl, C

1

-C

6

-alkylcarbonyl-C

1

-C

6

-alkyl or C

1

-C

6

-alkoxyimino-C

1

-C

6

-alkyl, where the abovementioned alkyl and cycloalkyl radicals may be partially or fully halogenated and/or may carry one to three of the following groups:

cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio, di(C

1

-C

4

-alkyl)amino, C

1

-C

4

-alkylcarbonyl, C

1

-C

4

-alkoxycarbonyl, C

1

-C

4

-alkoxy-C

1

-C

4

-alkoxycarbonyl, di(C

1

-C

4

-alkyl)amino-C

1

-C

4

-alkoxycarbonyl, hydroxycarbonyl, C

1

-C

4

-alkylaminocarbonyl, di(C

1

-C

4

-alkyl)aminocarbonyl, aminocarbonyl, C

1

-C

4

-alkylcarbonyloxy or C

3

-C

6

-cycloalkyl;

is phenyl, heterocyclyl, phenyl-C

1

-C

6

-alkyl, heterocyclyl-C

1

-C

6

-alkyl, phenylcarbonyl, heterocyclylcarbonyl, phenylaminocarbonyl or heterocyclylaminocarbonyl, where the phenyl and the heterocyclyl radical of the 8 last-mentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

14

,R

15

, R

16

are C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-alkynyl, C

3

-C

6

-haloalkynyl, C

3

-C

6

-cycloalkyl, hydroxyl, C

1

-C

6

-alkoxy, amino, C

1

-C

6

-alkylamino, C

1

-C

6

-haloalkylamino, di(C

1

-C

6

-alkyl)amino or di(C

1

-C

6

-haloalkyl)amino, where the abovementioned alkyl, cycloalkyl and alkoxy radicals may be partially or fully halogenated and/or may carry one to three of the following groups:

cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio, di(C

1

-C

4

-alkyl)amino, C

1

-C

4

-alkylcarbonyl or C

1

-C

4

-alkoxycarbonyl;

are phenyl, heterocyclyl, phenoxy or heterocyclyloxy, where the phenyl and the heterocyclyl radical of the last-mentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

17

is C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-alkynyl, C

3

-C

6

-halogenalkynyl, C

3

-C

6

-cycloalkyl, hydroxyl, C

1

-C

6

-alkoxy, C

3

-C

6

-alkenyloxy or C

3

-C

6

-alkynyloxy, where the abovementioned alkyl, cycloalkyl and alkoxy radicals may be partially or fully halogenated and/or may carry one to three radicals from the following groups:

cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio or di(C

1

-C

4

-alkyl)amino;

is phenyl, heterocyclyl, phenyl-C

1

-C

6

-alkyl or heterocyclyl-C

1

-C

6

-alkyl, where the phenyl or heterocyclyl radical of the four last-mentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

18

, R

19

are C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-alkynyl or C

1

-C

6

-alkylcarbonyl;

u is 2 to 4;

v is 1 to 5;

w is 2 to 5;

R

20

is a radical as mentioned under R

6

;

R

21

is hydrogen, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, hydroxyl, C

1

-C

6

-alkoxy or C

1

-C

6

-haloalkoxy;

R

22

is hydrogen, halogen, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, hydroxyl, C

1

-C

6

-alkoxy, C

1

-C

6

-haloalkoxy, C

1

-C

6

-alkylthio or C

1

-C

6

-haloalkylthio;

R

23

is hydrogen, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, C

3

-C

6

-cycloalkyl or C

3

-C

6

-halocycloalkyl;

R

24

is hydrogen, C

1

-C

6

-alkoxycarbonyl, C

1

-C

6

-haloalkoxycarbonyl, hydroxycarbonyl or cyano;

R

25

is C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, C

3

-C

6

-cycloalkyl or C

3

-C

6

-halocycloalkyl;

and their agriculturally useful salts.

Moreover, the invention relates to the processes and intermediates for preparing compounds of the formula I, compositions comprising them and to the use of the compounds of the formula I and of the compositions comprising them for controlling pests.

Herbicidally effective phosphorothionoamidates are disclosed in the literature, for example in DE-A 22 60 705 and DE-A 21 66 729. Furtheermore, U.S. Pat. No. 3,775,057 describes pyridinylphosphonates.

Likewise, substituted benzoylisoxazoles or -pyrazoles and substituted 2-phenylcyclohexane-1,3-diones or 1-phenyl-2-cyanoalkane-1,3-diones are disclosed, for example, in EP-A 418 175, EP-A 609 797, WO 96/26 192, WO 96/26 206, EP-A 203 428, U.S. Pat. No. 4,780,127, EP-A 315 075 and EP-A 625 505.

However, the herbicidal properties of the prior art compounds and their compatibility with crop plants are not entirely satisfactory. It is an object of the present invention to provide novel, in particular herbicidally effective compounds having improved properties.

We have found that this object is achieved by the phosphorus-containing benzoyl derivatives of the formula I and their herbicidal action.

Furthermore, we have found herbicidal compositions comprising the compounds I and having very good herbicidal action. Moreover, we have found processes for preparing these compositions and methods for controlling undesirable vegetation using the compounds I.

Depending on the substitution pattern, the compounds of the formula I can contain one or more chiral centers, in which case they exist in the form of enantiomers or diastereomer mixtures.

The invention provides both the pure enantiomers or diastereomers and mixtures thereof.

The compounds of the formula I can also be present in the form of their agriculturally useful salts, the type of salt generally being immaterial. In general, the salts of those cations or the acid addition salts of those acids are suitable whose cations and anions, respectively, do not affect the herbicidal action of the compounds I negatively.

Suitable cations are, in particular, ions of the alkali metals, preferably lithium, sodium and potassium, the alkaline earth metals, preferably calcium and magnesium, and the transition metals, preferably manganese, copper, zinc and iron, and also ammonium, where, if desired, one to four hydrogen atoms may be replaced by C

1

-C

4

-alkyl, hydroxy-C

1

-C

4

-alkyl, C

1

-C

4

-alkoxy-C

1

-C

4

-alkyl, hydroxy-C

1

-C

4

-alkoxy-C

1

-C

4

-alkyl, phenyl or benzyl, preferably ammonium, dimethylammonium, diisopropylammonium, tetramethylammonium, tetrabutylammonium, 2-(2-hydroxyeth-1-oxy)eth-1-ylammonium, di(2-hydroxyeth-1-yl)ammonium, trimethylbenzylammonium, furthermore phosphonium ions, sulfonium ions, preferably tri(C

1

-C

4

-alkyl)sulfonium and sulfoxonium ions, preferably tri(C

1

-C

4

-alkyl)sulfoxonium.

Anions of useful acid addition salts are primarily chloride, bromide, fluoride, hydrogen sulfate, sulfate, dihydrogen phosphate, hydrogen phosphate, nitrate, hydrogen carbonate, carbonate, hexafluorosilicate, hexafluorophosphate, benzoate and the anions of C

1

-C

4

-alkanoic acids, preferably formate, acetate, propionate and butyrate.

The organic molecular moieties mentioned for the substituents R

1

-R

25

or as radicals on phenyl and heterocyclyl radicals are collective terms for individual lists of the individual group members. All hydrocarbon chains, i.e. all alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl, alkylamino, dialkylamino, haloalkylamino, di(haloalkyl)amino, N-alkoxy-N-alkylamino, N-alkylsulfonylamino, N-haloalkylsulfonylamino, N-alkyl-N-alkylsulfonylamino, N-alkyl-N-haloalkylsulfonylamino, alkylcarbonyl, haloalkylcarbonyl, alkoxycarbonyl, haloalkoxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoxyalkyl, haloalkoxyalkyl, alkylthioalkyl, alkylsulfinylalkyl, alkylsulfonylalkyl, dialkoxymethyl, dialkylthiomethyl, (alkoxy)(alkylthio)methyl, alkylcarbonylalkyl, alkoxyiminoalkyl, alkoxycarbonyloxy, phenylalkyl, heterocyclylalkyl, dialkylaminoalkoxycarbonyl, alkoxyalkoxycarbonyl, alkenylcarbonyl, N-alkenyl-N-alkylamino, dialkenylamino, alkynylcarbonyl, N-alkynyl-N-alkylamino, dialkynylamino, alkenyl, alkynyl, haloalkenyl, haloalkynyl, alkenyloxy, alkenylthio, alkynyloxy and alkynylthio moieties can be straight-chain or branched. Unless indicated otherwise, halogenated substituents preferably carry one to five identical or different halogen atoms. The term halogen represents in each case fluorine, chlorine, bromine or iodine.

Examples of other meanings are:

C

1

-C

4

-alkyl: for example methyl, ethyl, propyl, 1-methylethyl, butyl, 1-methylpropyl, 2-methylpropyl or 1,1-dimethylethyl;

C

1

-C

6

-alkyl, and the alkyl moieties of C

1

-C

6

-alkylcarbonyl-C

1

-C

6

-alkyl, C

1

-C

6

-alkoxyimino-C

1

-C

6

-alkyl, N—(C

3

-C

6

-alkenyl)-N—(C

1

-C

6

-alkyl)amino, N—(C

3

-C

6

-alkynyl)-N—(C

1

-C

6

-alkyl)amino, phenyl-C

1

-C

6

-alkyl, N—(C

1

-C

6

-alkyl)-N—(C

1

-C

6

-alkylsulfonyl)amino, N—(C

1

-C

6

-alkyl)-N—(C

1

-C

6

-haloalkylsulfonyl)amino, heterocyclyl-C

1

-C

6

-alkyl: C

1

-C

4

-alkyl as mentioned above, and also, for example, pentyl, 1-methylbutyl, 2-methylbutyl, 3-methylbutyl, 2,2-dimethylpropyl, 1-ethylpropyl, hexyl, 1,1-dimethylpropyl, 1,2-dimethylpropyl, 1-methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1,1-dimethylbutyl, 1,2-dimethylbutyl, 1,3-dimethylbutyl, 2,2-dimethylbutyl, 2,3-dimethylbutyl, 3,3-dimethylbutyl, 1-ethylbutyl, 2-ethylbutyl, 1,1,2-trimethylpropyl, 1-ethyl-1-methylpropyl or 1-ethyl-3-methylpropyl;

C

1

-C

4

-haloalkyl: a C

1

-C

4

-alkyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example, chloromethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluorpmethyl, dichlorofluoromethyl, chlorodifluoromethyl, 2-fluoroethyl, 2-chloroethyl, 2-bromoethyl, 2-iodoethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2-difluoroethyl, 2,2-dichloro-2-fluoroethyl, 2,2,2-trichloroethyl, pentafluoroethyl, 2-fluoropropyl, 3-fluoropropyl, 2,2-difluoropropyl, 2,3-difluoropropyl, 2-chloropropyl, 3-chloropropyl, 2,3-dichloropropyl, 2-bromopropyl, 3-bromopropyl, 3,3,3-trifluoropropyl, 3,3,3-trichloropropyl, 2,2,3,3,3-pentafluoropropyl, heptafluoropropyl, 1-(fluoromethyl)-2-fluoroethyl, 1-(chloromethyl)-2-chloroethyl, 1-(bromomethyl)-2-bromoethyl, 4-fluorobutyl, 4-chlorobutyl, 4-bromobutyl or nonafluorobutyl;

C

1

-C

6

-haloalkyl, and the haloalkyl moieties of C

1

-C

6

-haloalkylamino, di(C

1

-C

6

-haloalkyl)amino: C

1

-C

4

-haloalkyl, as mentioned above, and also, for example, 5-fluoropentyl, 5-chloropentyl, 5-bromopentyl, 5-iodopentyl, undecafluoropentyl, 6-fluorohexyl, 6-chlorohexyl, 6-bromohexyl, 6-iodohexyl or dodecafluorohexyl;

C

1

-C

4

-alkoxy: for example methoxy, ethoxy, propoxy, 1-methylethoxy, butoxy, 1-methylpropoxy, 2-methylpropoxy or 1,1-dimethylethoxy;

C

1

-C

6

-alkoxy, and the alkoxy moieties of di(C

1

-C

6

-alkoxy)methyl, (C

1

-C

6

-alkoxy)(C

1

-C

6

-alkylthio)methyl, C

1

-C

6

-alkoxyimino-C

1

-C

6

-alkyl and N—(C

1

-C

6

-alkoxy)-N—(C

1

-C

6

-alkyl)amino: C

1

-C

4

-alkoxy as mentioned above, and also, for example, pentoxy, 1-methylbutoxy, 2-methylbutoxy, 3-methylbutoxy, 1,1-dimethylpropoxy, 1,2-dimethylpropoxy, 2,2-dimethylpropoxy, 1-ethylpropoxy, hexoxy, 1-methylpentoxy, 2-methylpentoxy, 3-methylpentoxy, 4-methylpentoxy, 1,1-dimethylbutoxy, 1,2-dimethylbutoxy, 1,3-dimethylbutoxy, 2,2-dimethylbutoxy, 2,3-dimethylbutoxy, 3,3-dimethylbutoxy, 1-ethylbutoxy, 2-ethylbutoxy, 1,1,2-trimethylpropoxy, 1,2,2-trimethylpropoxy, 1-ethyl-1-methylpropoxy or 1-ethyl-2-methylpropoxy;

C

1

-C

4

-haloalkoxy: a C

1

-C

4

-alkoxy radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example, fluoromethoxy, difluoromethoxy, trifluoromethoxy, chlorodifluoromethoxy, bromodifluoromethoxy, 2-fluoroethoxy, 2-chloroethoxy, 2-bromomethoxy, 2-iodoethoxy, 2,2-difluoroethoxy, 2,2,2-trifluoroethoxy, 2-chloro-2-fluoroethoxy, 2-chloro-2,2-difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy, pentafluoroethoxy, 2-fluoropropoxy, 3-fluoropropoxy, 2-chloropropoxy, 3-chloropropoxy, 2-bromopropoxy, 3-bromopropoxy, 2,2-difluoropropoxy, 2,3-difluoropropoxy, 2,3-dichloropropoxy, 3,3,3-trifluoropropoxy, 3,3,3-trichloropropoxy, 2,2,3,3,3-pentafluoropropoxy, heptafluoropropoxy, 1-(fluoromethyl)-2-fluoroethoxy, 1-(chloromethyl)-2-chloroethoxy, 1-(bromomethyl)-2-bromoethoxy, 4-fluorobutoxy, 4-chlorobutoxy, 4-bromobutoxy or nonafluorobutoxy;

C

1

-C

6

-haloalkoxy, and the haloalkoxy moieties of C

1

-C

6

-haloalkoxy-C

1

-C

6

-alkyl: C

1

-C

4

-haloalkoxy as mentioned above, and also, for example, 5-fluoropentoxy, 5-chloropentoxy, 5-bromopentoxy, 5-iodopentoxy, undecafluoropentoxy, 6-fluorohexoxy, 6-chlorohexoxy, 6-bromohexoxy, 6-iodohexoxy or dodecafluorohexoxy;

C

1

-C

4

-alkylthio: for example methylthio, ethylthio, propylthio, 1-methylethylthio, butylthio, 1-methylpropylthio, 2-methylpropylthio or 1,1-dimethylethylthio;

C

1

-C

6

-alkylthio, and the alkylthio moieties of C

1

-C

6

-alkylthio-C

1

-C

6

-alkyl, di(C

1

-C

6

-alkylthio)methyl and (C

1

-C

6

-alkoxy)(C

1

-C

6

-alkylthio)methyl: C

1

-C

4

-alkylthio as mentioned above, and also, for example, pentylthio, 1-methylbutylthio, 2-methylbutylthio, 3-methylbutylthio, 2,2-dimethylpropylthio, 1-ethylpropylthio, hexylthio, 1,1-dimethylpropylthio, 1,2-dimethylpropylthio, 1-methylpentylthio, 2-methylpentylthio, 3-methylpentylthio, 4-methylpentylthio, 1,1-dimethylbutylthio, 1,2-dimethylbutylthio, 1,3-dimethylbutylthio, 2,2-dimethylbutylthio, 2,3-dimethylbutylthio, 3,3-dimethylbutylthio, 1-ethylbutylthio, 2-ethylbutylthio, 1,1,2-trimethylpropylthio, 1,2,2-trimethylpropylthio, 1-ethyl-1-methylpropylthio or 1-ethyl-2-methylpropylthio;

C

1

-C

6

-haloalkylthio: a C

1

-C

6

-alkylthio radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example, fluoromethylthio, difluoromethylthio, trifluoromethylthio, chlorodifluoromethylthio, bromodifluoromethylthio, 2-fluoroethylthio, 2-chloroethylthio, 2-bromoethylthio, 2-iodoethylthio, 2,2-difluoroethylthio, 2,2,2-trifluoroethylthio, 2,2,2-trichloroethylthio, 2-chloro-2-fluoroethylthio, 2-chloro-2,2-difluoroethylthio, 2,2-dichloro-2-fluoroethylthio, pentafluoroethylthio, 2-fluoropropylthio, 3-fluoropropylthio, 2-chloropropylthio, 3-chloropropylthio, 2-bromopropylthio, 3-bromopropylthio, 2,2-difluoropropylthio, 2,3-difluoropropylthio, 2,3-dichloropropylthio, 3,3,3-trifluoropropylthio, 3,3,3-trichloropropylthio, 2,2,3,3,3-pentafluoropropylthio, heptafluoropropylthio, 1-(fluoromethyl)-2-fluoroethylthio, 1-(chloromethyl)-2-chloroethylthio, 1-(bromomethyl)-2-bromoethylthio, 4-fluorobutylthio, 4-chlorobutylthio, 4-bromobutylthio, nonafluorobutylthio, 5-fluoropentylthio, 5-chloropentylthio, 5-bromopentylthio, 5-iodopentylthio, undecafluoropentylthio, 6-fluorohexylthio, 6-chlorohexylthio, 6-bromohexylthio, 6-iodohexylthio or dodecafluorohexylthio;

C

1

-C

4

-alkylsulfinyl (C

1

-C

4

-alkyl-S(═O)—): for example methylsulfinyl, ethylsulfinyl, propylsulfinyl, 1-methylethylsulfinyl, butylsulfinyl, 1-methylpropylsulfinyl, 2-methylpropylsulfinyl or 1,1-dimethylethylsulfinyl;

C

1

-C

6

-alkylsulfinyl and the alkylsulfinyl radicals of C

1

-C

6

-alkylsulfinyl-C

1

-C

6

-alkyl: C

1

-C

4

-alkylsulfinyl, as mentioned above, and also, for example, pentylsulfinyl, 1-methylbutylsulfinyl, 2-methylbutylsulfinyl, 3-methylbutylsulfinyl, 2,2-dimethylpropylsulfinyl, 1-ethylpropylsulfinyl, 1,1-dimethylpropylsulfinyl, 1,2-dimethylpropylsulfinyl, hexylsulfinyl, 1-methylpentylsulfinyl, 2-methylpentylsulfinyl, 3-methylpentylsulfinyl, 4-methylpentylsulfinyl, 1,1-dimethylbutylsulfinyl, 1,2-dimethylbutylsulfinyl, 1,3-dimethylbutylsulfinyl, 2,2-dimethylbutylsulfinyl, 2,3-dimethylbutylsulfinyl, 3,3-dimethylbutylsulfinyl, 1-ethylbutylsulfinyl, 2-ethylbutylsulfinyl, 1,1,2-trimethylpropylsulfinyl, 1,2,2-trimethyl propylsulfinyl, 1-ethyl-1-methylpropylsulfinyl or 1-ethyl-2-methylpropylsulfinyl;

C

1

-C

6

-haloalkylsulfinyl: a C

1

-C

6

-alkylsulfinyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example, fluoromethylsulfinyl, difluoromethylsulfinyl, trifluoromethylsulfinyl, chlorodifluoromethylsulfinyl, bromodifluoromethylsulfinyl, 2-fluoroethylsulfinyl, 2-chloroethylsulfinyl, 2-bromoethylsulfinyl, 2-iodoethylsulfinyl, 2,2-difluoroethylsulfinyl, 2,2,2-trifluoroethylsulfinyl, 2,2,2-trichloroethylsulfinyl, 2-chloro-2-fluoroethylsulfinyl, 2-chloro-2,2-difluoroethylsulfinyl, 2,2-dichloro-2-fluoroethylsulfinyl, pentafluoroethylsulfinyl, 2-fluoropropylsulfinyl, 3-fluoropropylsulfinyl, 2-chloropropylsulfinyl, 3-chloropropylsulfinyl, 2-bromopropylsulfinyl, 3-bromopropylsulfinyl, 2,2-difluoropropylsulfinyl, 2,3-difluoropropylsulfinyl, 2,3-dichloropropylsulfinyl, 3,3,3-trifluoropropylsulfinyl, 3,3,3-trichloropropylsulfinyl, 2,2,3,3,3-pentafluoropropylsulfinyl, heptafluoropropylsulfinyl, 1-(fluoromethyl)-2-fluoroethylsulfinyl, 1-(chloromethyl)-2-chloroethylsulfinyl, 1-(bromomethyl)-2-bromoethylsulfinyl, 4-fluorobutylsulfinyl, 4-chlorobutylsulfinyl, 4-bromobutylsulfinyl, nonafluorobutylsulfinyl, 5-fluoropentylsulfinyl, 5-chloropentylsulfinyl, 5-bromopentylsulfinyl, 5-iodopentylsulfinyl, undecafluoropentylsulfinyl, 6-fluorohexylsulfinyl, 6-chaorohexylsulfinyl, 6-bromohexylsulfinyl, 6-iodohexylsulfinyl or dodecafluorohexylsulfinyl;

C

1

-C

4

-alkylsulfonyl (C

1

-C

4

-alkyl-S(═O)

2

—): for example methylsulfonyl, ethylsulfonyl, propylsulfonyl, 1-methylethylsulfonyl, butylsulfonyl, 1-methylpropylsulfonyl, 2-methylpropyl sulfonyl or 1,1-dimethylethylsulfonyl;

C

1

-C

6

-alkylsulfonyl, and the alkylsulfonyl radicals of C

1

-C

6

-alkylsulfonyl-C

3

-C

6

-alkyl, C

1

-C

6

-alkylsulfonylamino and N—(C

4

-C

6

-alkyl)-N—(C

1

-C

6

-alkylsulfonyl)amino: C

1

-C

4

-alkylsulfonyl as mentioned above, and also pentylsulfonyl, 1-methylbutylsulfonyl, 2-methylbutylsulfonyl, 3-methylbutylsulfonyl, 1,1-dimethylpropylsulfonyl, 1,2-dimethylpropylsulfonyl, 2,2-dimethylpropylsulfonyl, 1-ethylpropylsulfonyl, hexylsulfonyl, 1-methylpentylsulfonyl, 2-methylpentylsulfonyl, 3-methylpentylsulfonyl, 4-methylpentylsulfonyl, 1,1-dimethylbutylsulfonyl, 1,2-dimethylbutylsulfonyl, 1,3-dimethylbutylsulfonyl, 2,2-dimethylbutylsulfonyl, 2,3-dimethylbutylsulfonyl, 3,3-dimethylbutylsulfonyl, 1-ethylbutylsulfonyl, 2-ethylbutylsulfonyl, 1,1,2-trimethylpropylsulfonyl, 1,2,2-trimethylpropylsulfonyl, 1-ethyl-1-methylpropylsulfonyl or 1-ethyl-2-methylpropylsulfonyl;

C

1

-C

6

-haloalkylsulfonyl, and the haloalkylsulfonyl radicals of N—(C

1

-C

6

-haloalkylsulfonyl)amino and N—(C

1

-C

6

-alkyl)-N—(C

1

-C

6

-haloalkylsulfonyl)amino: a C

1

-

6

-alkylsulfonyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example, fluoromethylsulfonyl, difluoromethylsulfonyl, trifluoromethylsulfonyl, chlorodifluoromethylsulfonyl, bromodifluoromethylsulfonyl, 2-fluoroethylsulfonyl, 2-chloroethylsulfonyl, 2-bromoethylsulfonyl, 2-iodoethylsulfonyl, 2,2-difluoroethylsulfonyl, 2,2,2-trifluoroethylsulfonyl, 2-chloro-2-fluoroethylsulfonyl, 2-chloro-2,2-difluoroethylsulfonyl, 2,2-dichloro-2-fluoroethylsulfonyl, 2,2,2-trichloroethylsulfonyl, pentafluoroethylsulfonyl, 2-fluoropropylsulfonyl, 3-fluoropropylsulfonyl, 2-chloropropylsulfonyl, 3-chloropropylsulfonyl, 2-bromopropylsulfonyl, 3-bromopropylsulfonyl, 2,2-difluoropropylsulfonyl, 2,3-difluoropropylsulfonyl, 2,3-dichloropropylsulfonyl, 3,3,3-trifluoropropylsulfonyl, 3,3,3-trichloropropylsulfonyl, 2,2,3,3,3-pentafluoropropylsulfonyl, heptafluoropropylsulfonyl, 1-(fluoromethyl)-2-fluoroethylsulfonyl, 1-(chloromethyl)-2-chloroethylsulfonyl, 1-(bromomethyl)-2-bromoethylsulfonyl, 4-fluorobutylsulfonyl, 4-chlorobutylsulfonyl, 4-bromobutylsulfonyl, nonafluorobutylsulfonyl, 5-fluoropentylsulfonyl, 5-chloropentylsulfonyl, 5-bromopentylsulfonyl, 5-iodopentylsulfonyl, 6-fluorohexylsulfonyl, 6-bromohexylsulfonyl, 6-iodohexylsulfonyl or dodecafluorohexylsulfonyl;

C

1

-C

6

-alkylamino, and the alkylamino radicals of (C

1

-C

6

-alkoxy)(C

1

-C

6

-alkyl)amino: for example methylamino, ethylamino, propylamino, 1-methylethylamino, butylamino, 1-methylpropylamino, 2-methylpropylamino, 1,1-dimethylethylamino, pentylamino, 1-methylbutylamino, 2-methylbutylamino, 3-methylbutylamino, 2,2-dimethylpropylamino, 1-ethylpropylamino, hexylamino, 1,1-dimethylpropylamino, 1,2-dimethylpropylamino, 1-methylpentylamino, 2-methylpentylamino, 3-methylpentylamino, 4-methylpentylamino, 1,1-dimethylbutylamino, 1,2-dimethylbutylamino, 1,3-dimethylbutylamino, 2,2-dimethylbutylamino, 2,3-dimethylbutylamino, 3,3-dimethylbutylamino, 1-ethylbutylamino, 2-ethylbutylamino, 1,1,2-trimethylpropylamino, 1,2,2-trimethylpropylamino, 1-ethyl-1-methylpropylamino or 1-ethyl-2-methylpropylamino;

(C

1

-C

6

-alkylamino)sulfonyl: for example methylaminosulfonyl, ethylaminosulfonyl, propylaminosulfonyl, 1-methylethylaminosulfonyl, butylaminosulfonyl, 1-methylpropylaminosulfonyl, 2-methylpropylaminosulfonyl, 1,1-dimethylethylaminosulfonyl, pentylaminosulfonyl, 1-methylbutylaminosulfonyl, 2-methylbutylaminosulfonyl, 3-methylbutylaminosulfonyl, 2,2-dimethylpropylaminosulfonyl, 1-ethylpropylaminosulfonyl, hexylaminosulfonyl, 1,1-dimethylpropylaminosulfonyl, 1,2-dimethylpropylaminosulfonyl, 1-methylpentylaminosulfonyl, 2-methylpentylaminosulfonyl, 3-methylpentylaminosulfonyl, 4-methylpentylaminosulfonyl, 1,1-dimethylbutylaminosulfonyl, 1,2-dimethylbutylaminosulfonyl, 1,3-dimethylbutylaminosulfonyl, 2,2-dimethylbutylaminosulfonyl, 2,3-dimethylbutylaminosulfonyl, 3,3-dimethylbutylaminosulfonyl, 1-ethylbutylaminosulfonyl, 2-ethylbutylaminosulfonyl, 1,1,2-trimethylpropylaminosulfonyl, 1,2,2-trimethylpropylaminosulfonyl, 1-ethyl-1-methylpropylaminosulfonyl or 1-ethyl-2-methylpropylaminosulfonyl;

di(C

1

-C

6

-alkyl)aminosulfonyl: for example N,N-dimethylaminosulfonyl, N,N-diethylaminosulfonyl, N,N-di(1-methylethyl)aminosulfonyl, N,N-dipropylaminosulfonyl, N,N-dibutylaminosulfonyl, N,N-di(1-methylpropyl)aminosulfonyl, N,N-di(2-methylpropyl)aminosulfonyl, N,N-di(1,1-dimethylethyl)aminosulfonyl, N-ethyl-N-methylaminosulfonyl, N-methyl-N-propylaminosulfonyl, N-methyl-N-(1-methylethyl)aminosulfonyl, N-butyl-N-methylaminosulfonyl, N-methyl-N-(1-methylpropyl)aminosulfonyl, N-methyl-N-(2-methylpropyl)aminosulfonyl, N-(1,1-dimethylethyl)-N-methylaminosulfonyl, N-ethyl-N-propylaminosulfonyl, N-ethyl-N-(1-methylethyl)aminosulfonyl, N-butyl-N-ethylaminosulfonyl, N-ethyl-N-(1-methylpropyl)aminosulfonyl, N-ethyl-N-(2-methylpropyl)aminosulfonyl, N-ethyl-N-(1,1-dimethylethyl)aminosulfonyl, N-(1-methylethyl)-N-propylaminosulfonyl, N-butyl-N-propylaminosulfonyl, N-(1-methylpropyl)-N-propylaminosulfonyl, N-(2-methylpropyl)-N-propylaminosulfonyl, N-(1,1-dimethylethyl)-N-propylaminosulfonyl, N-butyl-N-(1-methylethyl)aminosulfonyl, N-(1-methylethyl)-N-(1-methylpropyl)aminosulfonyl, N-(1-methylethyl)-N-(2-methylpropyl)aminosulfonyl, N-(1,1-dimethylethyl)-N-(1-methylethyl)aminosulfonyl, N-butyl-N-(1-methylpropyl)aminosulfonyl, N-butyl-N-(2-methylpropyl)aminosulfonyl, N-butyl-N-(1,1-dimethylethyl)aminosulfonyl, N-(1-methylpropyl)-N-(2-methylpropyl)aminosulfonyl, N-(1,1-dimethylethyl)-N-(1-methylpropyl)aminosulfonyl, N-(1,1-dimethylethyl)-N-(2-methylpropyl)aminosulfonyl, N-methyl-N-pentylaminosulfonyl, N-methyl-N-(1-methylbutyl)aminosulfonyl, N-methyl-N-(2-methylbutyl)aminosulfonyl, N-methyl-N-(3-methylbutyl)aminosulfonyl, N-methyl-N-(2,2-dimethylpropyl)aminosulfonyl, N-methyl-N-(1-ethylpropyl)aminosulfonyl, N-methyl-N-hexylaminosulfonyl, N-methyl-N-(1,1-dimethylpropyl)aminosulfonyl, N-methyl-N-(1,2-dimethylpropyl)aminosulfonyl, N-methyl-N-(1-methylpentyl)aminosulfonyl, N-methyl-N-(2-methylpentyl)aminosulfonyl, N-methyl-N-(3-methylpentyl)aminosulfonyl, N-methyl-N-(4-methylpentyl)aminosulfonyl, N-methyl-N-(1,1-dimethylbutyl)aminosulfonyl, N-methyl-N-(1,2-dimethylbutyl)aminosulfonyl, N-methyl-N-(1,3-dimethylbutyl)aminosulfonyl, N-methyl-N-(2,2-dimethylbutyl)aminosulfonyl, N-methyl-N-(2,3-dimethylbutyl)aminosulfonyl, N-methyl-N-(3,3-dimethylbutyl)aminosulfonyl, N-methyl-N-(1-ethylbutyl)aminosulfonyl, N-methyl-N-(2-ethylbutyl)aminosulfonyl, N-methyl-N-(1,1,2-trimethylpropyl)aminosulfonyl, N-methyl-N-(1,2,2-trimethylpropyl)aminosulfonyl, N-methyl-N-(1-ethyl-1-methylpropyl)aminosulfonyl, N-methyl-N-(1-ethyl-2-methylpropyl)aminosulfonyl, N-ethyl-N-pentylaminosulfonyl, N-ethyl-N-(1-methylbutyl)aminosulfonyl, N-ethyl-N-(2-methylbutyl)aminosulfonyl, N-ethyl-N-(3-methylbutyl)aminosulfonyl, N-ethyl-N-(2,2-dimethylpropyl)aminosulfonyl, N-ethyl-N-(1-ethylpropyl)aminosulfonyl, N-ethyl-N-hexylaminosulfonyl, N-ethyl-N-(1,1-dimethylpropyl)aminosulfonyl, N-ethyl-N-(1,2-dimethylpropyl)aminosulfonyl, N-ethyl-N-(1-methylpentyl )aminosulfonyl, N-ethyl-N-(2-methylpentyl)aminosulfonyl, N-ethyl-N-(3-methylpentyl)aminosulfonyl, N-ethyl-N-(4-methylpentyl)aminosulfonyl, N-ethyl-N-(1,1-dimethyl butyl)aminosulfonyl, N-ethyl-N-(1,2-dimethylbutyl)aminosulfonyl, N-ethyl-N-(1,3-dimethylbutyl)aminosulfonyl, N-ethyl-N-(2,2-dimethylbutyl)aminosulfonyl, N-ethyl-N-(2,3-dimethylbutyl)aminosulfonyl, N-ethyl-N-(3,3-dimethylbutyl)aminosulfonyl, N-ethyl-N-(1-ethylbutyl)aminosulfonyl, N-ethyl-N-(2-ethylbutyl)aminosulfonyl, N-ethyl-N-(1,1,2-trimethylpropyl)aminosulfonyl, N-ethyl-N-(1,2,2-trimethylpropyl)aminosulfonyl, N-ethyl-N-(1-ethyl-1-methylpropyl)aminosulfonyl, N-ethyl-N-(1-ethyl-2-methylpropyl)aminosulfonyl, N-propyl-N-pentylaminosulfonyl, N-butyl-N-pentylaminosulfonyl, N,N-dipentylaminosulfonyl, N-propyl-N-hexylaminosulfonyl, N-butyl-N-hexylaminosulfonyl, N-pentyl-N-hexylaminosulfonyl or N,N-dihexylaminosulfonyl;

di(C

1

-C

4

-alkyl)amino, and the dialkylamino radicals of di(C

1

-C

4

-alkyl)amino-C

1

-C

4

-alkoxycarbonyl: for example N,N-dimethylamino, N,N-diethylamino, N,N-dipropylamino, N,N-di(1-methylethyl)amino, N,N-dibutylamino, N,N-di(1-methylpropyl)amino, N,N-di(2-methylpropyl)amino, N,N-di(1,1-dimethylethyl)amino, N-ethyl-N-methylamino, N-methyl-N-propylamino, N-methyl-N-(1-methylethyl)amino, N-butyl-N-methylamino, N-methyl-N-(1-methylpropyl)amino, N-methyl-N-(2-methylpropyl)amino, N-(1,1-dimethylethyl)-N-methylamino, N-ethyl-N-propylamino, N-ethyl-N-(1-methylethyl)amino, N-butyl-N-ethylamino, N-ethyl-N-(1-methylpropyl)amino, N-ethyl-N-(2-methylpropyl)amino, N-ethyl-N-(1,1-dimethylethyl)amino, N-(1-methylethyl)-N-propylamino, N-butyl-N-propylamino, N-(1-methylpropyl)-N-propylamino, N-(2-methylpropyl)-N-propylamino, N-(1,1-dimethylethyl)-N-propylamino, N-butyl-N-(1-methylethyl)amino, N-(1-methylethyl)-N-(1-methylpropyl)amino, N-(1-methylethyl)-N-(2-methylpropyl)amino, N-(1,1-dimethylethyl)-N-(1-methylethyl)amino, N-butyl-N-(1-methylpropyl)amino, N-butyl-N-(2-methylpropyl)amino, N-butyl-N-(1,1-dimethylethyl)amino, N-(1-methylpropyl)-N-(2-methylpropyl)amino, N-(1,1-dimethylethyl)-N-(1-methylpropyl)amino or N-(1,1-dimethylethyl)-N-(2-methylpropyl)amino;

di(C

1

-C

6

-alkyl)amino: di(C

1

-C

4

-alkyl)amino as mentioned above, and also N,N-dipentylamino, N,N-dihexylamino, N-methyl-N-pentylamino, N-ethyl-N-pentylamino, N-methyl-N-hexylamino or N-ethyl-N-hexylamino;

C

1

-C

4

-alkylcarbonyl: for example methylcarbonyl, ethylcarbonyl, propylcarbonyl, 1-methylethylcarbonyl, butylcarbonyl, 1-methylpropylcarbonyl, 2-methylpropylcarbonyl or 1,1-dimethylethylcarbonyl;

C

1

-C

6

-alkylcarbonyl, and the alkylcarbonyl radicals of C

1

-C

6

-alkylcarbonyl-C

1

-C

6

-alkyl: C

1

-C

4

-alkylcarbonyl as mentioned above, and also, for example, pentylcarbonyl, 1-methylbutylcarbonyl, 2-methylbutylcarbonyl, 3-methylbutylcarbonyl, 2,2-dimethylpropylcarbonyl, 1-ethylpropylcarbonyl, hexylcarbonyl, 1,1-dimethylpropylcarbonyl, 1,2-dimethylpropylcarbonyl, 1-methylpentylcarbonyl, 2-methylpentylcarbonyl, 3-methylpentylcarbonyl, 4-methylpentylcarbonyl, 1,1-dimethylbutylcarbonyl, 1,2-dimethylbutylcarbonyl, 1,3-dimethylbutylcarbonyl, 2,2-dimethylbutylcarbonyl, 2,3-dimethylbutylcarbonyl, 3,3-dimethylbutylcarbonyl, 1-ethylbutylcarbonyl, 2-ethylbutylcarbonyl, 1,1,2-trimethylpropylcarbonyl, 1,2,2-trimethylpropylcarbonyl, 1-ethyl-1-methylpropylcarbonyl or 1-ethyl-2-methylpropylcarbonyl;

C

1

-C

20

-alkylcarbonyl: C

1

-C

6

-alkylcarbonyl as mentioned above, and also heptylcarbonyl, octylcarbonyl, pentadecylcarbonyl or heptadecylcarbonyl;

C

1

-C

6

-haloalkylcarbonyl: a C

1

-C

6

-alkylcarbonyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example, chloroacetyl, dichloroacetyl, trichloroacetyl, fluoroacetyl, difluoroacetyl, trifluoroacetyl, chlorofluoroacetyl, dichlorofluoroacetyl, chlorodifluoroacetyl, 2-fluoroethylcarbonyl, 2-chloroethylcarbonyl, 2-bromoethylcarbonyl, 2-iodoethylcarbonyl, 2,2-difluoroethylcarbonyl, 2,2,2-trifluoroethylcarbonyl, 2-chloro-2-fluoroethylcarbonyl, 2-chloro-2,2-difluoroethylcarbonyl, 2,2-dichloro-2-fluoroethylcarbonyl, 2,2,2-trichloroethylcarbonyl, pentafluoroethylcarbonyl, 2-fluoropropylcarbonyl, 3-fluoropropylcarbonyl, 2,2-difluoropropylcarbonyl, 2,3-difluoropropylcarbonyl, 2-chloropropylcarbonyl, 3-chloropropylcarbonyl, 2,3-dichloropropylcarbonyl, 2-bromopropylcarbonyl, 3-bromopropylcarbonyl, 3,3,3-trifluoropropylcarbonyl, 3,3,3-trichloropropylcarbonyl, 2,2,3,3,3-pentafluoropropylcarbonyl, heptafluoropropylcarbonyl, 1-(fluoromethyl)-2-fluoroethylcarbonyl, 1-(chloromethyl)-2-chloroethylcarbonyl, 1-(bromomethyl)-2-bromoethylcarbonyl, 4-fluorobutylcarbonyl, 4-chlorobutylcarbonyl, 4-bromobutylcarbonyl, nonafluorobutylcarbonyl, 5-fluoropentylcarbonyl, 5-chloropentylcarbonyl, 5-bromopentylcarbonyl, perfluoropentylcarbonyl, 6-fluorohexylcarbonyl, 6-chlorohexylcarbonyl, 6-bromohexylcarbonyl or perfluorohexylcarbonyl;

C

1

-C

4

-alkoxycarbonyl, and the alkoxycarbonyl moieties of di(C

1

-C

4

-alkyl)amino-C

1

-C

4

-alkoxycarbonyl: for example methoxycarbonyl, ethoxycarbonyl, propoxycarbonyl, 1-methylethoxycarbonyl, butoxycarbonyl, 1-methylpropoxycarbonyl, 2-methylpropoxycarbonyl or 1,1-dimethylethoxycarbonyl;

(C

1

-C

6

-alkoxy)carbonyl, and the alkoxycarbonyl moieties of C

1

-C

6

-alkoxycarbonyloxy: (C

1

-C

4

-alkoxy)carbonyl as mentioned above, and also, for example, pentoxycarbonyl, 1-methylbutoxycarbonyl, 2-methylbutoxycarbonyl, 3-methylbutoxycarbonyl, 2,2-dimethylpropoxycarbonyl, 1-ethylpropoxycarbonyl, hexoxycarbonyl, 1,1-dimethylpropoxycarbonyl, 1,2-dimethylpropoxycarbonyl, 1-methylpentoxycarbonyl, 2-methylpentoxycarbonyl, 3-methylpentoxycarbonyl, 4-methylpentoxycarbonyl, 1,1-dimethylbutoxycarbonyl, 1,2-dimethylbutoxycarbonyl, 1,3-dimethylbutoxycarbonyl, 2,2-dimethylbutoxycarbonyl, 2,3-dimethylbutoxycarbonyl, 3,3-dimethylbutoxycarbonyl, 1-ethylbutoxycarbonyl, 2-ethylbutoxycarbonyl, 1,1,2-trimethylpropoxycarbonyl, 1,2,2-trimethylpropoxycarbonyl, 1-ethyl-1-methylpropoxycarbonyl or 1-ethyl-2-methylpropoxycarbonyl;

C

1

-C

6

-haloalkoxycarbonyl: a C

1

-C

6

-alkoxycarbonyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example, fluoromethoxycarbonyl, difluoromethoxycarbonyl, trifluoromethoxycarbonyl, chlorodifluoromethoxycarbonyl, bromodifluoromethoxycarbonyl, 2-fluoroethoxycarbonyl, 2-chloroethoxycarbonyl, 2-bromoethoxycarbonyl, 2-iodoethoxycarbonyl, 2,2-difluoroethoxycarbonyl, 2,2,2-trifluoroethoxycarbonyl, 2-chloro-2-fluoroethoxycarbonyl, 2-chloro-2,2-difluoroethoxycarbonyl, 2,2-dichloro-2-fluoroethoxycarbonyl, 2,2,2-trichloroethoxycarbonyl, pentafluoroethoxycarbonyl, 2-fluoropropoxycarbonyl, 3-fluoropropoxycarbonyl, 2-chloropropoxycarbonyl, 3-chloropropoxycarbonyl, 2-bromopropoxycarbonyl, 3-bromopropoxycarbonyl, 2,2-difluoropropoxycarbonyl, 2,3-difluoropropoxycarbonyl, 2,3-dichloropropoxycarbonyl, 3,3,3-trifluoropropoxycarbonyl, 3,3,3-trichloropropoxycarbonyl, 2,2,3,3,3-pentafluoropropoxycarbonyl, heptafluoropropoxycarbonyl, 1-(2fluoromethyl)-2-fluoroethoxycarbonyl, 1-(chloromethyl)-2-chloroethoxycarbonyl, 1-(bromomethyl)-2-bromoethoxycarbonyl, 4-fluorobutoxycarbonyl, 4-chlorobutoxycarbonyl, 4-bromobutoxycarbonyl, 4-iodobutoxycarbonyl, 5-fluoropentoxycarbonyl, 5-chloropentoxycarbonyl, 5-bromopentoxycarbonyl, 6-fluorohexoxycarbonyl, 6-chlorohexoxycarbonyl or 6-bromohexoxycarbonyl;

(C

1

-C

4

-alkylamino)carbonyl: for example methylaminocarbonyl, ethylaminocarbonyl, propylaminocarbonyl, 1-methylethylaminocarbonyl, butylaminocarbonyl, 1-methylpropylaminocarbonyl, 2-methylpropylaminocarbonyl or 1,1-dimethylethylaminocarbonyl;

(C

1

-C

6

-alkylamino)carbonyl: (C

1

-C

4

-alkylamino)carbonyl as mentioned above, and also, for example, pentylaminocarbonyl, 1-methylbutylaminocarbonyl, 2-methylbutylaminocarbonyl, 3-methylbutylaminocarbonyl, 2,2-dimethylpropylaminocarbonyl, 1-ethylpropylaminocarbonyl, hexylaminocarbonyl, 1,1-dimethylpropylaminocarbonyl, 1,2-dimethylpropylaminocarbonyl, 1-methylpentylaminocarbonyl, 2-methylpentylaminocarbonyl, 3-methylpentylaminocarbonyl, 4-methylpentylaminocarbonyl, 1,1-dimethylbutylaminocarbonyl, 1,2-dimethylbutylaminocarbonyl, 1,3-dimethylbutylaminocarbonyl, 2,2-dimethylbutylaminocarbonyl, 2,3-dimethylbutylaminocarbonyl, 3,3-dimethylbutylaminocarbonyl, 1-ethylbutylaminocarbonyl, 2-ethylbutylaminocarbonyl, 1,1,2-trimethylpropylaminocarbonyl, 1,2,2-trimethylpropylaminocarbonyl, 1-ethyl-1-methylpropylaminocarbonyl or 1-ethyl-2-methylpropylaminocarbonyl;

di(C

1

-C

4

-alkyl)aminocarbonyl: for example N,N-dimethylaminocarbonyl, N,N-diethylaminocarbonyl, N,N-di(1-methylethyl)aminocarbonyl, N,N-dipropylaminocarbonyl, N,N-dibutylaminocarbonyl, N,N-di(1-methylpropyl)aminocarbonyl, N,N-di(2-methylpropyl)aminocarbonyl, N,N-di(1,1-dimethylethyl)aminocarbonyl, N-ethyl-N-methylaminocarbonyl, N-methyl-N-propylaminocarbonyl, N-methyl-N-(1-methylethyl)aminocarbonyl, N-butyl-N-methylaminocarbonyl, N-methyl-N-(1-methylpropyl)aminocarbonyl, N-methyl-N-(2-methylpropyl)aminocarbonyl, N-(1,1-dimethylethyl)-N-methylaminocarbonyl, N-ethyl-N-propylaminocarbonyl, N-ethyl-N-(1-methylethyl)aminocarbonyl, N-butyl-N-ethylaminocarbonyl, N-ethyl-N-(1-methylpropyl)aminocarbonyl, N-ethyl-N-(2-methylpropyl)aminocarbonyl, N-ethyl-N-(1,1-dimethylethyl)aminocarbonyl, N-(1-methylethyl)-N-propylaminocarbonyl, N-butyl-N-propylaminocarbonyl, N-(1-methylpropyl)-N-propylaminocarbonyl, N-(2-methylpropyl)-N-propylaminocarbonyl, N-(1,1-dimethylethyl)-N-propylaminocarbonyl, N-butyl-N-(1-methylethyl)aminocarbonyl, N-(-methylethyl)-N-(1-methylpropyl)aminocarbonyl, N-(1-methylethyl)-N-(2-methylpropyl)aminocarbonyl, N-(1,1-dimethylethyl)-N-(2-methylethyl)aminocarbonyl, N-butyl-N-(1-methylpropyl)aminocarbonyl, N-butyl-N-(2-methylpropyl)aminocarbonyl, N-butyl-N-(1,1-dimethylethyl)aminocarbonyl, N-(1-methylpropyl)-N-(2-methylpropyl)aminocarbonyl, N-(1,1-dimethylethyl)-N-(1-methylpropyl)aminocarbonyl or N-(1,1-dimethylethyl)-N-(2-methylpropyl)aminocarbonyl;

C

1

-C

6

-alkoxy-C

1

-C

6

-alkyl: C

1

-C

6

-alkyl which is substituted by C

1

-C

6

-alkoxy as mentioned above, i.e., for example, methoxymethyl, ethoxymethyl, propoxymethyl, (1-methylethoxy)methyl, butoxymethyl, (1-methylpropoxy)methyl, (2-methylpropoxy)methyl, (1,1-dimethylethoxy)methyl, 2-(methoxy)ethyl, 2-(ethoxy)ethyl, 2-(propoxy)ethyl, 2-(1-methylethoxy)ethyl, 2-(butoxy)ethyl, 2-(1-methylpropoxy)ethyl, 2-(2-methylpropoxy)ethyl, 2-(1,1-dimethylethoxy)ethyl, 2-(methoxy)propyl, 2-(ethoxy)propyl, 2-(propoxy)propyl, 2-(1-methylethoxy)propyl, 2-(butoxy)propyl, 2-(1-methylpropoxy)propyl, 2-(2-methylpropoxy)propyl, 2-(1,1-dimethylethoxy)propyl, 3-(methoxy)propyl, 3-(ethoxy)propyl, 3-(propoxy)propyl, 3-(1-methylethoxy)propyl, 3-(butoxy)propyl, 3-(1-methylpropoxy)propyl, 3-(2-methylpropoxy)propyl, 3-(1,1-dimethylethoxy)propyl, 2-(methoxy)butyl, 2-(ethoxy)butyl, 2-(propoxy)butyl, 2-(1-methylethoxy)butyl, 2-(butoxy)butyl, 2-(1-methylpropoxy)butyl, 2-(2-methylpropoxy)butyl, 2-(1,1-dimethylethoxy)butyl, 3-(methoxy)butyl, 3-(ethoxy)butyl, 3-(propoxy)butyl, 3-(1-methylethoxy)butyl, 3-(butoxy)butyl, 3-(1-methylpropoxy)butyl, 3-(2-methylpropoxy)butyl, 3-(1,1-dimethylethoxy)butyl, 4-(methoxy)butyl, 4-(ethoxy)butyl, 4-(propoxy)butyl, 4-(1-methylethoxy)butyl, 4-(butoxy)butyl, 4-(1-methylpropoxy)butyl, 4-(2-methylpropoxy)butyl, 4-(1,1-dimethylethoxy)butyl, 5-methoxypentyl, 5-ethoxypentyl, 6-methoxyhexyl or 6-ethoxyhexyl;

the C

1

-C

4

-alkoxy-C

1

-C

4

-alkoxy radical of C

1

-C

4

-alkoxy-C

1

-C

4

-alkoxycarbonyl: C

1

-C

4

-alkoxy which is substituted by C

1

-C

4

-alkoxy as mentioned above, i.e., for example, methoxymethoxy, ethoxymethoxy, propoxymethoxy, (1-methylethoxy)methoxy, butoxymethoxy, (1-methylpropoxy)methoxy, (2-methylpropoxy)methoxy, (1,1-dimethylethoxy)methoxy, 2-(methoxy)ethoxy, 2-(ethoxy)ethoxy, 2-(propoxy)ethoxy, 2-(1-methylethoxy)ethoxy, 2-(butoxy)ethoxy, 2-(1-methylpropoxy)ethoxy, 2-(2-methylpropoxy)ethoxy, 2-(1,1-dimethylethoxy)ethoxy, 2-(methoxy)propoxy, 2-(ethoxy)propoxy, 2-(propoxy)propoxy, 2-(1-methylethoxy)propoxy, 2-(butoxy)propoxy, 2-(1-methylpropoxy)propoxy, 2-(2-methylpropoxy)propoxy, 2-(1,1-dimethylethoxy)propoxy, 3-(methoxy)propoxy, 3-(ethoxy)propoxy, 3-(propoxy)propoxy, 3-(1-methylethoxy)propoxy, 3-(butoxy)propoxy, 3-(1-methylpropoxy)propoxy, 3-(2-methylpropoxy)propoxy, 3-(1,1-dimethylethoxy)propoxy, 2-(methoxy)butoxy, 2-(ethoxy)butoxy, 2-(propoxy)butoxy, 2-(1-methylethoxy)butoxy, 2-(butoxy)butoxy, 2-(1-methylpropoxy)butoxy, 2-(2-methylpropoxy)butoxy, 2-(1,1-dimethylethoxy)butoxy, 3-(methoxy)butoxy, 3-(ethoxy)butoxy, 3-(propoxy)butoxy, 3-(1-methylethoxy)butoxy, 3-(butoxy)butoxy, 3-(1-methylpropoxy)butoxy, 3-(2-methylpropoxy)butoxy, 3-(1,1-dimethylethoxy)butoxy, 4-(methoxy)butoxy, 4-(ethoxy)-butoxy, 4-(propoxy)butoxy, 4-(1-methylethoxy)butoxy, 4-(butoxy)butoxy, 4-(1-methylpropoxy)butoxy, 4-(2-methylpropoxy)butoxy or 4-(1,1-dimethylethoxy)butoxy;

C

3

-C

6

-alkenyl, and the alkenyl moieties of C

3

-C

6

-alkenylcarbonyl, C

3

-C

6

-alkenyloxy, C

3

-C

6

-alkenylthio, N—(C

3

-C

6

-alkenyl)-N—(C

1

-C

6

-alkyl)amino and di(C

3

-C

6

-alkenyl)amino: for example prop-2-en-1-yl, but-1-en-4-yl, 1-methylprop-2-en-1-yl, 2-methylprop-2-en-1-yl, 2-buten-1-yl, 1-penten-3-yl, 1-penten-4-yl, 2-penten-4-yl, 1-methylbut-2-en-1-yl, 2-methylbut-2-en-1-yl, 3-methylbut-2-en-1-yl, 1-methylbut-3-en-1-yl, 2-methylbut-3-en-1-yl, 3-methylbut-3-en-1-yl, 1,1-dimethylprop-2-en-1-yl, 1,2-dimethylprop-2-en-1-yl, 1-ethylprop-2-en-1-yl, hex-3-en-1-yl, hex-4-en-1-yl, hex-5-en-1-yl, 1-methylpent-3-en-1-yl, 2-methylpent-3-en-1-yl, 3-methylpent-3-en-1-yl, 4-methylpent-3-en-1-yl, 1-methylpent-4-en-1-yl, 2-methylpent-4-en-1-yl, 3-methylpent-4-en-1-yl, 4-methylpent-4-en-1-yl, 1,1-dimethylbut-2-en-1-yl, 1,1-dimethylbut-3-en-1-yl, 1,2-dimethylbut-2-en-1-yl, 1,2-dimethylbut-3-en-1-yl, 1,3-dimethylbut-2-en-1-yl, 1,3-dimethylbut-3-en-1-yl, 2,2-dimethylbut-3-en-1-yl, 2,3-dimethylbut-2-en-1-yl, 2,3-dimethylbut-3-en-1-yl, 3,3-dimethylbut-2-en-1-yl, 1-ethylbut-2-en-1-yl, 1-ethylbut-3-en-1-yl, 2-ethylbut-2-en-1-yl, 2-ethylbut-3-en-1-yl, 1,1,2-trimethylprop-2-en-1-yl, 1-ethyl-1-methylprop-2-en-1-yl or 1-ethyl-2-methylprop-2-en-1-yl;

C

2

-C

6

-alkenyl, and the alkenyl moieties of C

2

-C

6

-alkenylcarbonyl: C

3

-C

6

-alkenyl as mentioned above, and also ethenyl;

C

3

-C

6

-haloalkenyl: a C

3

-C

6

-alkenyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example, 2-chloroallyl, 3-chloroallyl, 2,3-dichloroallyl, 3,3-dichloroallyl, 2,3,3-trichloroallyl, 2,3-dichlorobut-2-enyl, 2-bromoallyl, 3-bromoallyl, 2,3-dibromoallyl, 3,3-dibromoallyl, 2,3,3-tribromoallyl or 2,3-dibromobut-2-enyl;

C

3

-C

6

-alkynyl, and the alkynyl moieties of C

3

-C

6

-alkynylcarbonyl, C

3

-C

6

-alkynyloxy, C

3

-C

6

-alkynylthio, N—(C

3

-C

6

-alkynyl)-N—(C

1

-C

6

-alkyl)amino and di(C

3

-C

6

-alkynyl)amino: for example propargyl, but-1-yn-3-yl, but-1-yn-4-yl, but-2-yn-1-yl, pent-1-yn-3-yl, pent-1-yn-4-yl, pent-1-yn-5-yl, pent-2-yn-1-yl, pent-2-yn-4-yl, pent-2-yn-5-yl, 3-methylbut-1-yn-3-yl, 3-methylbut-1-yn-4-yl, hex-1-yn-3-yl, hex-1-yn-4-yl, hex-1-yn-5-yl, hex-1-yn-6-yl, hex-2-yn-1-yl, hex-2-yn-4-yl, hex-2-yn-5-yl, hex-2-yn-6-yl, hex-3-yn-1-yl, hex-3-yn-2-yl, 3-methylpent-1-yn-3-yl, 3-methylpent-1-yn-4-yl, 3-methylpent-1-yn-5-yl, 4-methylpent-2-yn-4-yl or 4-methylpent-2-yn-5-yl;

C

2

-C

6

-alkynyl, and the alkynyl moieties of C

2

-C

6

-alkynylcarbonyl: C

3

-C

6

-alkynyl as mentioned above, and also ethynyl;

C

3

-C

6

-haloalkynyl: a C

3

-C

6

-alkynyl radical as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example, 1,1-difluoroprop-2-yn-1-yl, 3-iodoprop-2-yn-1-yl, 4-fluorobut-2-yn-1-yl, 4-chlorobut-2-yn-1-yl, 1,1-difluorobut-2-yn-1-yl, 4-iodobut-3-yn-1-yl, 5-fluoropent-3-yn-1-yl, 5-iodopent-4-yn-1-yl, 6-fluorohex-4-yn-1-yl or 6-iodohex-5-yn-1-yl;

C

3

-C

6

-cycloalkyl, and the cycloalkyl moieties of C

3

-C

6

-cycloalkylcarbonyl: for example cyclopropyl, cyclobutyl, cyclopentyl or cyclohexyl;

C

3

-C

6

-halocycloalkyl: a C

3

-C

6

-cycloalkyl radical as mentioned above which may be partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., for example, 2,2-dichlorocycloprop-1-yl, 2,2-difluorocycloprop-1-yl, 3-chlorocyclopent-1-yl, 3-fluorocyclopent-1-yl, 3-bromocyclopent-1-yl, 3,3-dichlorocyclopent-1-yl, 3,3-difluorocyclopent-1-yl, 4-chlorocyclohex-1-yl, 4-fluorocyclohex-1-yl, 4-bromocyclohex-1-yl, 4,4-dichlorocyclohex-1-yl or 4,4-difluorocyclohex-1-yl;

heterocyclyl, and the heterocyclyl moieties of heterocyclylcarbonyl, heterocyclyl-C

1

-C

6

-alkyl, heterocyclyloxy, heterocyclylaminocarbonyl: a saturated, partially saturated or unsaturated 5- or 6-membered heterocyclic ring which is attached via carbon and contains one to four identical or different heteroatoms selected from the following group: oxygen, sulfur and nitrogen, i.e., for example, 5-membered rings such as:

tetrahydrofuran-2-yl, tetrahydrofuran-3-yl, tetrahydrothien-2-yl, tetrahydrothien-3-yl, tetrahydropyrrol-2-yl, tetrahydropyrrol-3-yl, 2,3-dihydrofuran-2-yl, 2,3-dihydrofuran-3-yl, 2,5-dihydrofuran-2-yl, 2,5-dihydrofuran-3-yl, 4,5-dihydrofuran-2-yl, 4,5-dihydrofuran-3-yl, 2,3-dihydrothien-2-yl, 2,3-dihydrothien-3-yl, 2,5-dihydrothien-2-yl, 2,5-dihydrothien-3-yl, 4,5-dihydrothien-2-yl, 4,5-dihydrothien-3-yl, 2,3-dihydro-1H-pyrrol-2-yl, 2,3-dihydro-1H-pyrrol-3-yl, 2,5-dihydro-1H-pyrrol-2-yl, 2,5-dihydro-1H-pyrrol-3-yl, 4,5-dihydro-1H-pyrrol-2-yl, 4,5-dihydro-1H-pyrrol-3-yl, 3,4-dihydro-2H-pyrrol-2-yl, 3,4-dihydro-2H-pyrrol-3-yl, 3,4-dihydro-5H-pyrrol-2-yl, 3,4-dihydro-5H-pyrrol-3-yl, 2-furyl, 3-furyl, 2-thienyl, 3-thienyl, pyrrol-2-yl, pyrrol-3-yl, tetrahydropyrazol-3-yl, tetrahydropyrazol-4-yl, tetrahydroisoxazol-3-yl, tetrahydroisoxazol-4-yl, tetrahydroisoxazol-5-yl, 1,2-oxathiolan-3-yl, 1,2-oxathiolan-4-yl, 1,2-oxathiolan-5-yl, tetrahydroisothiazol-3-yl, tetrahydroisothiazol-4-yl, tetrahydroisothiazol-5-yl, 1,2-dithiolan-3-yl, 1,2-dithiolan-4-yl, tetrahydroimidazol-2-yl, tetrahydroimidazol-4-yl, tetrahydrooxazol-2-yl, tetrahydrooxazol-4-yl, tetrahydrooxazol-5-yl, tetrahydrothiazol-2-yl, tetrahydrothiazol-4-yl, tetrahydrothiazol-5-yl, 1,3-dioxolan-2-yl, 1,3-dioxolan-4-yl, 1,3-oxathiolan-2-yl, 1,3-oxathiolan-4-yl, 1,3-oxathiolan-5-yl, 1,3-dithiolan-2-yl, 1,3-dithiolan-4-yl, 4,5-dihydro-1H-pyrazol-3-yl, 4,5-dihydro-1H-pyrazol-4-yl, 4,5-dihydro-1H-pyrazol-5-yl, 2,5-dihydro-1H-pyrazol-3-yl, 2,5-dihydro-1H-pyrazol-4-yl, 2,5-dihydro-1H-pyrazol-5-yl, 4,5-dihydroisoxazol-3-yl, 4,5-dihydroisoxazol-4-yl, 4,5-dihydroisoxazol-5-yl, 2,5-dihydroisoxazol-3-yl, 2,5-dihydroisoxazol-4-yl, 2,5-dihydroisoxazol-5-yl, 2,3-dihydroisoxazol-3-yl, 2,3-dihydroisoxazol-4-yl, 2,3-dihydroisoxazol-5-yl, 4,5-dihydroisothiazol-3-yl, 4,5-dihydroisothiazol-4-yl, 4,5-dihydroisothiazol-5-yl, 2,5-dihydroisothiazol-3-yl, 2,5-dihydroisothiazol-4-yl, 2,5-dihydroisothiazol-5-yl, 2,3-dihydroisothiazol-3-yl, 2,3-dihydroisothiazol-4-yl, 2,3-dihydroisothiazol-5-yl, Δ

3

-1,2-dithiol-3-yl, Δ

3

-1,2-dithiol-4-yl, Δ

3

-1,2-dithiol-5-yl, 4,5-dihydro-1H-imidazol-2-yl, 4,5-dihydro-1H-imidazol-4-yl, 4,5-dihydro-1H-imidazol-5-yl, 2,5-dihydro-1H-imidazol-2-yl, 2,5-dihydro-1H-imidazol-4-yl, 2,5-dihydro-1H-imidazol-5-yl, 2,3-dihydro-1H-imidazol-2-yl, 2,3-dihydro-1H-imidazol-4-yl, 4,5-dihydrooxazol-2-yl, 4,5-dihydrooxazol-4-yl, 4,5-dihydrooxazol-5-yl, 2,5-dihydrooxazol-2-yl, 2,5-dihydrooxazol-4-yl, 2,5-dihydrooxazol-5-yl, 2,3-dihydrooxazol-2-yl, 2,3-dihydrooxazol-4-yl, 2,3-dihydrooxazol-5-yl, 4,5-dihydrothiazol-2-yl, 4,5-dihydrothiazol-4-yl, 4,5-dihydrothiazol-5-yl, 2,5-dihydrothiazol-2-yl, 2,5-dihydrothiazol-4-yl, 2,5-dihydrothiazol-5-yl, 2,3-dihydrothiazol-2-yl, 2,3-dihydrothiazol-4-yl, 2,3-dihydrothiazol-5-yl, 1,3-dioxol-2-yl, 1,3-dioxol-4-yl, 1,3-dithiol-2-yl, 1,3-dithiol-4-yl, 1,3-oxathiol-2-yl, 1,3-oxathiol-4-yl, 1,3-oxathiol-5-yl, pyrazol-3-yl, pyrazol-4-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl, isothiazol-3-yl, isothiazol-4-yl, isothiazol-5-yl, imidazol-2-yl, imidazol-4-yl, oxazol-2-yl, oxazol-4-yl, oxazol-5-yl, thiazol-2-yl, thiazol-4-yl, thiazol-5-yl, 1,2,3-Δ

2

-oxadiazolin-4-yl, 1,2,3-Δ

2

-oxadiazolin-5-yl, 1,2,4-Δ

4

-oxadiazolin-3-yl, 1,2,4-Δ

4

-oxadiazolin-5-yl, 1,2,4-Δ

2

-oxadiazolin-3-yl, 1,2,4-Δ

2

-oxadiazolin-5-yl, 1,2,4-Δ

3

-oxadiazolin-3-yl, 1,2,4-Δ

3

-oxadiazolin-5-yl, 1,3,4-Δ

2

-oxadiazolin-2-yl, 1,3,4-Δ

2

-oxadiazolin-5-yl, 1,3,4-Δ

3

-oxadiazolin-2-yl, 1,3,4-oxadiazolin-2-yl, 1,2,4-Δ

4

-thiadiazolin-3-yl, 1,2,4-Δ

4

-thiadiazolin-5-yl, 1,2,4-Δ

3

-thiadiazolin-3-yl, 1,2,4-Δ

3

-thiadiazolin-5-yl, 1,2,4-Δ

2

-thiadiazolin-3-yl, 1,2,4-Δ

2

-thiadiazolin-5-yl, 1,3,4-Δ

2

-thiadiazolin-2-yl, 1,3,4-Δ

2

-thiadiazolin-5-yl, 1,3,4-Δ

3

-thiadiazolin-2-yl, 1,3,4-thiadiazolin-2-yl, 1,3,2-dioxathiolan-4-yl, 1,2,3-Δ

2

-triazolin-4-yl, 1,2,3-Δ

2

-triazolin-5-yl, 1,2,4-Δ

2

-triazolin-3-yl, 1,2,4-Δ

2

-triazolin-5-yl, 1,2,4-Δ

3

-triazolin-3-yl, 1,2,4-Δ

3

-triazolin-5-yl, 1,2,4-Δ

1

-triazolin-2-yl, 1,2,4-triazolin-3-yl, 3H-1,2,4-dithiazol-5-yl, 2H-1,3,4-dithiazol-5-yl, 2H-1,3,4-oxathiazol-5-yl, 1,2,3-oxadiazol-4-yl, 1,2,3-oxadiazol-5-yl, 1,2,4-oxadiazol-3-yl, 1,2,4,-oxadiazol-5-yl, 1,3,4-oxadiazol-2-yl, 1,2,3-thiadiazol-4-yl, 1,2,3-thiadiazol-5-yl, 1,2,4-thiadiazol-3-yl, 1,2,4-thiadiazol-5-yl, 1,3,4-thiadiazolyl-2-yl, 1,2,3-triazol-4-yl, 1,2,4-triazol-3-yl, tetrazol-5-yl,

6-membered rings such as:

tetrahydropyran-2-yl, tetrahydropyran-3-yl, tetrahydropyran-4-yl, piperidin-2-yl, piperidin-3-yl, piperidin-4-yl, tetrahydrothiopyran-2-yl, tetrahydrothiopyran-3-yl, tetrahydrothiopyran-4-yl, 2H-3,4-dihydropyran-6-yl, 2H-3,4-dihydropyran-5-yl, 2H-3,4-dihydropyran-4-yl, 2H-3,4-dihydropyran-3-yl, 2H-3,4-dihydropyran-2-yl, 2H-3,4-dihydropyran-6-yl, 2H-3,4-dihydrothiopyran-5-yl, 2H-3,4-dihydrothiopyran-4-yl, 2H-3,4-dihydropyran-3-yl, 2H-3,4-dihydropyran-2-yl, 1,2,3,4-tetrahydropyridin-6-yl, 1,2,3,4-tetrahydropyridin-5-yl, 1,2,3,4-tetrahydropyridin-4-yl, 1,2,3,4-tetrahydropyridin-3-yl, 1,2,3,4-tetrahydropyridin-2-yl, 2H-5,6-dihydropyran-2-yl, 2H-5,6-dihydropyran-3-yl, 2H-5,6-dihydropyran-4-yl, 2H-5,6-dihydropyran-5-yl, 2H-5,6-dihydropyran-6-yl, 2H-5,6-dihydrothiopyran-2-yl, 2H-5,6-dihydrothiopyran-3-yl, 2H-5,6-dihydrothiopyran-4-yl, 2H-5,6-dihydrothiopyran-5-yl, 2H-5,6-dihydrothiopyran-6-yl, 1,2,5,6-tetrahydropyridin-2-yl, 1,2,5,6-tetrahydropyridin-3-yl, 1,2,5,6-tetrahydropyridin-4-yl, 1,2,5,6-tetrahydropyridin-5-yl, 1,2,5,6-tetrahydropyridin-6-yl, 2,3,4,5-tetrahydropyridin-2-yl, 2,3,4,5-tetrahydropyridin-3-yl, 2,3,4,5-tetrahydropyridin-4-yl, 2,3,4,5-tetrahydropyridin-5-yl, 2,3,4,5-tetrahydropyridin-6-yl, 4H-pyran-2-yl, 4H-pyran-3-yl, 4H-pyran-4-yl, 4H-thiopyran-2-yl, 4H-thiopyran-3-yl, 4H-thiopyran-4-yl, 1,4-dihydropyridin-2-yl, 1,4-dihydropyridin-3-yl, 1,4-dihydropyridin-4-yl, 2H-pyran-2-yl, 2H-pyran-3-yl, 2H-pyran-4-yl, 2H-pyran-5-yl, 2H-pyran-6-yl, 2H-thiopyran-2-yl, 2H-thiopyran-3-yl, 2H-thiopyran-4-yl, 2H-thiopyran-5-yl, 2H-thiopyran-6-yl, 1,2-dihydropyridin-2-yl, 1,2-dihydropyridin-3-yl, 1,2-dihydropyridin-4-yl, 1,2-dihydropyridin-5-yl, 1,2-dihydropyridin-6-yl, 3,4-dihydropyridin-2-yl, 3,1-dihydropyridin-3-yl, 3,4-dihydropyridin-4-yl, 3,4-dihydropyridin-5-yl, 3,4-dihydropyridin-6-yl, 2,5-dihydropyridin-2-yl, 2,5-dihydropyridin-3-yl, 2,5-dihydropyridin-4-yl, 2,5-dihydropyridin-5-yl, 2,5-dihydropyridin-6-yl, 2,3-dihydropyridin-2-yl, 2,3-dihydropyridin-3-yl, 2,3-dihydropyridin-4-yl, 2,3-dihydropyridin-5-yl, 2,3-dihydropyridin-6-yl, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, 1,3-dioxan-2-yl, 1,3-dioxan-4-yl, 1,3-dioxan-5-yl, 1,4-dioxan-2-yl, 1,3-dithian-2-yl, 1,3-dithian-4-yl, 1,3-dithian-5-yl, 1,4-dithian-2-yl, 1,3-oxathian-2-yl, 1,3-oxathian-4-yl, 1,3-oxathian-5-yl, 1,3-oxathian-6-yl, 1,4-oxathian-2-yl, 1,4-oxathian-3-yl, 1,2-dithian-3-yl, 1,2-dithian-4-yl, hexahydropyrimidin-2-yl, hexahydropyrimidin-4-yl, hexahydropyrimidin-5-yl, hexahydropyrazin-2-yl, hexahydropyridazin-3-yl, hexahydropyridazin-4-yl, tetrahydro-1,3-oxazin-2-yl, tetrahydro-1,3-oxazin-4-yl, tetrahydro-1,3-oxazin-5-yl, tetrahydro-1,3-oxazin-6-yl, tetrahydro-1,3-thiazin-2-yl, tetrahydro-1,3-thiazin-4-yl, tetrahydro-1,3-thiazin-5-yl, tetrahydro-1,3-thiazin-6-yl, tetrahydro-1,4-thiazin-2-yl, tetrahydro-1,4-thiazin-3-yl, tetrahydro-1,4-oxazin-2-yl, tetrahydro-1,4-oxazin-3-yl, tetrahydro-1,2-oxazin-3-yl, tetrahydro-1,2-oxazin-4-yl, tetrahydro-1,2-oxazin-5-yl, tetrahydro-1,2-oxazin-6-yl, 2H-5,6-dihydro-1,2-oxazin-3-yl, 2H-5,6-dihydro-1,2-oxazin-4-yl, 2H-5,6-dihydro-1,2-oxazin-5-yl, 2H-5,6-dihydro-1,2-oxazin-6-yl, 2H-5,6-dihydro-1,2-thiazin-3-yl, 2H-5,6-dihydro-1,2-thiazin-4-yl, 2H-5,6-dihydro-1,2-thiazin-5-yl, 2H-5,6-dihydro-1,2-thiazin-6-yl, 4H-5,6-dihydro-1,2-oxazin-3-yl, 4H-5,6-dihydro-1,2-oxazin-4-yl, 4H-5,6-dihydro-1,2-oxazin-5-yl, 4H-5,6-dihydro-1,2-oxazin-6-yl, 4H-5,6-dihydro-1,2-thiazin-3-yl, 4H-5,6-dihydro-1,2-thiazin-4-yl, 4H-5,6-dihydro-1,2-thiazin-5-yl, 4H-5,6-dihydro-1,2-thiazin-6-yl, 2H-3,6-dihydro-1,2-oxazin-3-yl, 2H-3,6-dihydro-1,2-oxazin-4-yl, 2H-3,6-dihydro-1,2-oxazin-5-yl, 2H-3,6-dihydro-1,2-oxazin-6-yl, 2H-3,6-dihydro-1,2-thiazin-3-yl, 2H-3,6-dihydro-1,2-thiazin-4-yl, 2H-3,6-dihydro-1,2-thiazin-5-yl, 2H-3,6-dihydro-1,2-thiazin-6-yl, 2H-3,4-dihydro-1,2-oxazin-3-yl, 2H-3,4-dihydro-1,2-oxazin-4-yl, 2H-3,4-dihydro-1,2-oxazin-5-yl, 2H-3,4-dihydro-1,2-oxazin-6-yl, 2H-3,4-dihydro-1,2-thiazin-3-yl, 2H-3,4-dihydro-1,2-thiazin-4-yl, 2H-3,4-dihydro-1,2-thiazin-5-yl, 2H-3,4-dihydro-1,2-thiazin-6-yl, 2,3,4,5-tetrahydropyridazin-3-yl, 2,3,4,5-tetrahydropyridazin-4-yl, 2,3,4,5-tetrahydropyridazin-5-yl, 2,3,4,5-tetrahydropyridazin-6-yl, 3,4,5,6-tetrahydropyridazin-3-yl, 3,4,5,6-tetrahydropyridazin-4-yl, 1,2,5,6-tetrahydropyridazin-3-yl, 1,2,5,6-tetrahydropyridazin-4-yl, 1,2,5,6-tetrahydropyridazin-5-yl, 1,2,5,6-tetrahydropyridazin-6-yl, 1,2,3,6-tetrahydropyridazin-3-yl, 1,2,3,6-tetrahydropyridazin-4-yl, 4H-5,6-dihydro-1,3-oxazin-2-yl, 4H-5,6-dihydro-1,3-oxazin-4-yl, 4H-5,6-dihydro-1,3-oxazin-5-yl, 4H-5,6-dihydro-1,3-oxazin-6-yl, 4H-5,6-dihydro-1,3-thiazin-2-yl, 4H-5,6-dihydro-1,3-thiazin-4-yl, 4H-5,6-dihydro-1,3-thiazin-5-yl, 4H-5,6-dihydro-1,3-thiazin-6-yl, 3,4,5-6-tetrahydropyrimidin-2-yl, 3,4,5,6-tetrahydropyrimidin-4-yl, 3,4,5,6-tetrahydropyrimidin-5-yl, 3,4,5,6-tetrahydropyrimidin-6-yl, 1,2,3,4-tetrahydropyrazin-2-yl, 1,2,3,4-tetrahydropyrazin-5-yl, 1,2,3,4-tetrahydropyrimidin-2-yl, 1,2,3,4-tetrahydropyrimidin-4-yl, 1,2,3,4-tetrahydropyrimidin-5-yl, 1,2,3,4-tetrahydropyrimidin-6-yl, 2,3-dihydro-1,4-thiazin-2-yl, 2,3-dihydro-1,4-thiazin-3-yl, 2,3-dihydro-1,4-thiazin-5-yl, 2,3-dihydro-1,4-thiazin-6-yl, 2H-1,2-oxazin-3-yl, 2H-1,2-oxazin-4-yl, 2H-1,2-oxazin-5-yl, 2H-1,2-oxazin-6-yl, 2H-1,2-thiazin-3-yl, 2H-1,2-thiazin-4-yl, 2H-1,2-thiazin-5-yl, 2H-1,2-thiazin-6-yl, 4H-1,2-oxazin-3-yl, 4H-1,2-oxazin-4-yl, 4H-1,2-oxazin-5-yl, 4H-1,2-oxazin-6-yl, 4H-1,2-thiazin-3-yl, 4H-1,2-thiazin-4-yl, 4H-1,2-thiazin-5-yl, 4H-1,2-thiazin-6-yl, 6H-1,2-oxazin-3-yl, 6H-1,2-oxazin-4-yl, 6H-1,2-oxazin-5-yl, 6H-1,2-oxazin-6-yl, 6H-1,2-thiazin-3-yl, 6H-1,2-thiazin-4-yl, 6H-1,2-thiazin-5-yl, 6H-1,2-thiazin-6-yl, 2H-1,3-oxazin-2-yl, 2H-1,3-oxazin-4-yl, 2H-1,3-oxazin-5-yl, 2H-1,3-oxazin-6-yl, 2H-1,3-thiazin-2-yl, 2H-1,3-thiazin-4-yl, 2H-1,3-thiazin-5-yl, 2H-1,3-thiazin-6-yl, 4H-1,3-oxazin-2-yl, 4H-1,3-oxazin-4-yl, 4H-1,3-oxazin-5-yl, 4H-1,3-oxazin-6-yl, 4H-1,3-thiazin-2-yl, 4H-1,3-thiazin-4-yl, 4H-1,3-thiazin-5-yl, 4H-1,3-thiazin-6-yl, 6H-1,3-oxazin-2-yl, 6H-1,3-oxazin-4-yl, 6H-1,3-oxazin-5-yl, 6H-1,3-oxazin-6-yl, 6H-1,3-thiazin-2-yl, 6H-1,3-oxazin-4-yl, 6H-1,3-oxazin-5-yl, 6H-1,3-thiazin-6-yl, 2H-1,4-oxazin-2-yl, 2H-1,4-oxazin-3-yl, 2H-1,4-oxazin-5-yl, 2H-1,4-oxazin-6-yl, 2H-1,4-thiazin-2-yl, 2H-1,4-thiazin-3-yl, 2H-1,4-thiazin-5-yl, 2H-1,4-thiazin-6-yl, 4H-1,4-oxazin-2-yl, 4H-1,4-oxazin-3-yl, 4H-1,4-thiazin-2-yl, 4H-1,4-thiazin-3-yl, 1,4-dihydropyridazin-3-yl, 1,4-dihydropyridazin-4-yl, 1,4-dihydropyridazin-5-yl, 1,4-dihydropyridazin-6-yl, 1,4-dihydropyrazin-2-yl, 1,2-dihydropyrazin-2-yl, 1,2-dihydropyrazin-3-yl, 1,2-dihydropyrazin-5-yl, 1,2-dihydropyrazin-6-yl, 1,4-dihydropyrimidin-2-yl, 1,4-dihydropyrimidin-4-yl, 1,4-dihydropyrimidin-5-yl, 1,4-dihydropyrimidin-6-yl, 3,4-dihydropyrimidin-2-yl, 3,4-dihydropyrimidin-4-yl, 3,4-dihydropyrimidin-5-yl or 3,4-dihydropyrimidin-6-yl, pyridazin-3-yl, pyridazin-4-yl, pyrimidin-2-yl, pyrimidin-4-yl, pyrimidin-5-yl, pyrazin-2-yl, 1,3,5-triazin-2-yl, 1,2,4-triazin-3-yl, 1,2,4-triazin-5-yl, 1,2,4-triazin-6-yl, 1,2,4,5-tetrazin-3-yl;

where, if appropriate, the sulfur of the abovementioned heterocycles can oxidized to S═O or S(═O)

2

;

and where a bicyclic ring system may be formed with a fused-on phenyl ring or a C

3

-C

6

-carbocycle or with a further 5- to 6-membered heterocycle.

N-bonded heterocyclyl: a saturated, partially saturated or unsaturated 5- or 6-membered heterocyclic ring which is attached via nitrogen and contains at least one nitrogen and, if appropriate, one to three identical or different heteroatoms selected from the following group: oxygen, sulfur or nitrogen, i.e., for example

N-bonded 5-membered rings such as:

tetrahydropyrrol-1-yl, 2,3-dihydro-1H-pyrrol-1-yl, 2,5-dihydro-1H-pyrrol-1-yl, pyrrol-1-yl, tetrahydropyrazol-1-yl, tetrahydroisoxazol-2-yl, tetrahydroisothiazol-2-yl, tetrahydroimidazol-1-yl, tetrahydrooxazol-3-yl, tetrahydrothiazol-3-yl, 4,5-dihydro-1H-pyrazol-1-yl, 2,5-dihydro-1H-pyrazol-1-yl, 2,3-dihydro-1H-pyrazol-1-yl, 2,5-dihydroisoxazol-2-yl, 2,3-dihydroisoxazol-2-yl, 2,5-dihydroisothiazol-2-yl, 2,3-dihydroisoxazol-2-yl, 4,5-dihydro-1H-imidazol-1-yl, 2,5-dihydro-1H-imidazol-1-yl, 2,3-dihydro-1H-imidazol-1-yl, 2,3-dihydrooxazol-3-yl, 2,3-dihydrothiazol-3-yl, pyrazol-1-yl, imidazol-1-yl, 1,2,4-Δ

4

-oxadiazolin-2-yl, 1,2,4-Δ

2

-oxadiazolin-4-yl, 1,2,4-Δ

3

-oxadiazolin-2-yl, 1,3,4-Δ

2

-oxadiazolin-4-yl, 1,2,4-Δ

5

-thiadiazolin-2-yl, 1,2,4-Δ

3

-thiadiazolin-2-yl, 1,2,4-Δ

2

-thiadiazolin-4-yl, 1,3,4-Δ

2

-thiadiazolin-4-yl, 1,2,3-Δ

2

-triazolin-1-yl, 1,2,4-Δ

2

-triazolin-1-yl, 1,2,4-Δ

2

-triazolin-4-yl, 1,2,4-Δ

3

-triazolin-1-yl, 1,2,4-Δ

1

-triazolin-4-yl, 1,2,3-triazol-1-yl, 1,2,4-triazol-1-yl, tetrazol-1-yl;

and N-bonded 6-membered rings such as:

piperidin-1-yl, 1,2,3,4-tetrahydropyridin-1-yl, 1,2,5,6-tetrahydropyridin-1-yl, 1,4-dihydropyridin-1-yl, 1,2-dihydropyridin-1-yl, hexahydropyrimidin-1-yl, hexahydropyrazin-1-yl, hexahydropyridazin-1-yl, tetrahydro-1,3-oxazin-3-yl, tetrahydro-1,3-thiazin-3-yl, tetrahydro-1,4-thiazin-4-yl, tetrahydro-1,4-oxazin-4-yl, tetrahydro-1,2-oxazin-2-yl, 2H-5,6-dihydro-1,2-oxazin-2-yl, 2H-5,6-dihydro-1,2-thiazin-2-yl, 2H-3,6-dihydro-1,2-oxazin-2-yl, 2H-3,6-dihydro-1,2-thiazin-oxazin-2-yl, 2H-3,4-dihydro-1,2-thiazin-2-yl, 2,3,4,5-tetrahydropyridazin-2-yl, 1,2,5,6-tetrahydropyridazin-1-yl, 1,2,5,6-tetrahydropyridazin-2-yl, 1,2, 3,6-tetrahydropyridazin-1-yl, 3,4,5,6-tetrahydropyrimidin-3-yl, 1,2,3,4-tetrahydropyrazin-1-yl, 1,2,3,4-tetrahydropyrimidin-1-yl, 1,2,3,4-tetrahydropyrimidin-3-yl, 2,3-dihydro-1,4-thiazin-4-yl, 2H-1,2-oxazin-2-yl, 2H-1,2-thiazin-2-yl, 4H-1,4-oxazin-4-yl, 4H-1,4-thiazin-4-yl, 1,4-dihydropyridazin-1-yl, 1,4-dihydropyrazin-1-yl, 1,2-dihydropyrazin-1-yl, 1,4-dihydropyrimidin-1-yl or 3,4-dihydropyrimidin-3-yl, and

N-bonded cyclic imides such as:

phthalimide, tetrahydrophthalimide, succinimide, maleimide or glutarimide, and also 4-oxo-1,4-dihydropyridin-1-yl.

All phenyl rings or heterocyclyl radicals and all phenyl components in phenyl-C

1

-C

6

-alkyl, phenoxy, phenylcarbonyl and phenylaminocarbonyl or heterocyclyl components in heterocyclyl-C

1

-C

6

-alkyl, heterocyclyloxy, heterocyclylcarbonyl and heterocyclylaminocarbonyl are, unless stated otherwise, preferably unsubstituted or they carry one to three halogen atoms and/or one nitro group, one cyano radical and/or one or two methyl, trifluoromethyl, methoxy or trifluoromethoxy substituents.

Suitable heterocycyl radicals are, in particular, 5-membered aromatic heterocycles, for example 2-furyl, 3-furyl, 2-thienyl, 3-thienyl, pyrrol-2-yl, pyrrol-3-yl, pyrazol-3-yl, pyrazol-4-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl, isothiazol-3-yl, isothiazol-4-yl, isothiazol-5-yl, imidazol-2-yl, imidazol-4-yl, oxazol-2-yl, oxazol-4-yl, oxazol-5-yl, thiazol-2-yl, thiazol-4-yl, thiazol-5-yl, 1,2,4-triazol-3-yl or tetrazol-5-yl;

5-membered partially unsaturated heterocycles, for example 4,5-dihydro-1H-pyrazol-3-yl, 4,5-dihydro-1H-pyrazol-4-yl, 4,5-dihydro-1H-pyrazol-5-yl, 4,5-dihydroisoxazol-3-yl, 4,5-dihydroisoxazol-4-yl, 4,5-dihydroisoxazol-5-yl, 4,5-dihydrooxazol-2-yl, 4,5-dihydrooxazol-2-yl, 4,5-dihydrothiazol-2-yl or 4,5-dihydroimidazol-2-yl;

5-membered saturated heterocycles, for example tetrahydrofuran-2-yl, tetrahydrofuran-3-yl, tetrahydrothien-2-yl, tetrahydrothien-3-yl, tetrahydropyrrol-2-yl, tetrahydropyrrol-3-yl, 1,3-dioxolan-2-yl, 1,3-dioxolan-4-yl, 1,3-oxathiolan-2-yl, 1,3-oxathiolan-4-yl, 1,3-oxathiolan-5-yl, 1,3-dithiolan-2-yl or 1,3-dithiolan-4-yl;

6-membered aromatic heterocycles, for example pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyrimidin-2-yl, pyrimidin-4-yl, pyrimidin-5-yl, pyrazin-2-yl, 1,3,5-triazin-2-yl, 1,2,4-triazin-3-yl, 1,2,4-triazin-5-yl or 1,2,4-triazin-6-yl;

6-membered partially unsaturated heterocycles, for example 2H-3,4-dihydropyran-6-yl, 2H-3,4-dihydropyran-5-yl, 2H-3,4-dihydropyran-4-yl, 2H-3,4-dihydropyran-3-yl, 2H-3,4-dihydropyran-2-yl, 2H-3,4-dihydrothiopyran-6-yl, 2H-3,4-dihydrothiopyran-5-yl, 2H-3,4-dihydrothiopyran-4-yl, 2H-3,4-dihydrothiopyran-3-yl, 2H-3,4-dihydrothiopyran-2-yl, 4H-5,6-dihydro-1,3-oxazin-2-yl, 4H-5,6-dihydro-1,3-thiazin-2-yl or 3,4,5,6-tetrahydropyrimidin-2-yl;

6-membered saturated heterocycles, for example tetrahydropyran-2-yl, tetrahydropyran-3-yl, tetrahydropyran-4-yl, piperidin-2-yl, piperidin-3-yl, piperidin-4-yl, tetrahydrothiopyran-2-yl, tetrahydrothiopyran-3-yl, tetrahydrothiopyran-4-yl, 1,3-dioxan-2-yl, 1,3-dioxan-4-yl, 1,3-dioxan-5-yl, 1,3-dithian-2-yl, 1,3-dithian-4-yl, 1,3-dithian-5-yl, 1,3-oxathian-2-yl, 1,3-oxathian-4-yl, 1,3-oxathian-5-yl, tetrahydro-1,4-oxazin-2-yl, tetrahydro-1,4-oxazin-3-yl, tetrahydro-1,4-thiazin-2-yl or tetrahydro-1,4-thiazin-3-yl.

The compounds of the formula I according to the invention where Q=Q

1

are referred to as compounds of the formula Ia, compounds of the formula I where Q=Q

2

are referred to as Ib, compounds of the formula I where Q=Q

3

are referred to as Ic and compounds of the formula I where Q=Q

4

are referred to as Id.

With respect to the use of the compounds of the formula I according to invention as herbicides, the variables preferably have the following meaning, in each case on their own or in combination:

X is oxygen or sulfur;

in particular oxygen;

R

1

, R

2

are hydrogen, C

1

-C

6

-alkyl, hydroxyl, C

1

-C

6

-alkoxy, C

1

-C

6

-alkylthio, di(C

1

-C

6

-alkyl)amino, where the alkyl radicals of the five last-mentioned substituents may be partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylsulfonyl or C

1

-C

4

-alkoxycarbonyl;

in particular hydrogen, C

1

-C

4

-alkyl such as methyl, ethyl, propyl, 1-methylethyl, butyl, 1-methylbutyl or 2-methylbutyl, hydroxyl, C

1

-C

4

-alkoxy such as methoxy, ethoxy, propoxy, 1-methylethoxy, butoxy or 2-methylbutoxy, C

1

-C

4

-alkylthio such as methylthio, ethylthio, propylthio or 1-methylethylthio, or di(C

1

-C

4

-alkyl)amino such as dimethylamino, diethylamino, dipropylamino, dibutylamino, N-methyl-N-ethylamino, N-methyl-N-propylamino, N-methyl-N-butylamino, N-ethyl-N-propylamino or N-ethyl-N-butylamino; or

R

1

and R

2

together form a O—O(CH

2

)

m

—O—, —O—(CH

2

)

m

—S—, —S—(CH

2

)

m

—S—, —NR

5

—(CH

2

)

m

—NR

5

—, —O—(CH

2

)

m

—NR

5

—, —S—(CH

2

)

m

—NR

5

— or —(CH

2

)

p

chain which may carry one to three radicals from the following group: halogen, cyano, C

1

-C

4

-alkyl or C

1

-C

4

-alkoxycarbonyl; in particular, R

1

and R

2

together form a —O—(CH

2

)

m

—O, —O—(CH

2

)

m

—S—, —S—(CH

2

)

m

—S or —(CH

2

)

p

chain;

R

3

is hydrogen, nitro, cyano, halogen, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, C

1

-C

6

-alkoxy, C

1

-C

6

-haloalkoxy, C

1

-C

6

-alkylthio, C

1

-C

6

-haloalkylthio, C

1

-C

6

-alkylsulfinyl, C

1

-C

6

-haloalkylsulfinyl, C

1

-C

6

-alkylsulfonyl, C

1

-C

6

-haloalkylsulfonyl, —P(═O)(C

1

-C

4

-alkyl)

2

or —P(═O)(C

1

-C

4

-alkoxy)

2

; in particular nitro, halogen, C

1

-C

4

-alkyl such as methyl or ethyl, C

1

-C

4

-haloalkyl such as difluoromethyl or trifluoromethyl, C

1

-C

4

-alkoxy such as methoxy or ethoxy, C

1

-C

4

-haloalkoxy such as difluoromethoxy, trifluoromethoxy or chlorodifluoromethoxy, C

1

-C

4

-alkylthio such as methylthio or ethylthio, C

1

-C

4

-alkylsulfonyl such as methylsulfonyl or ethylsulfonyl, C

1

-C

4

-haloalkylsulfonyl such as difluoromethylsulfonyl, trifluoromethylsulfonyl or chlorodifluoromethylsulfonyl, —P(═O)(CH

3

)

2

, —P(═O)(CH

2

CH

3

)

2

, —P(═O)(OCH

3

)

2

or —P(═O)(OCH

2

CH

3

)

2

;

R

4

is halogen, such as chlorine or bromine, or C

1

-C

4

-alkyl, such as methyl or ethyl;

R

5

is hydrogen or C

1

-C

4

-alkyl, such as methyl or ethyl;

l is 0 or 1;

m is 2, 3 or 4;

p is 4 or 5;

Q is a radical of the formula Q

1

, Q

2

, Q

3

or Q

4

;

R

6

is hydroxyl, mercapto, halogen, OR

13

, SR

13

, SO

2

R

14

, OSO

2

R

14

, OPOR

15

R

16

, OPR

15

R

16

, OPSR

15

R

16

, NR

17

R

18

, ONR

18

R

19

, N-bonded heterocyclyl or O—(N-bonded heterocyclyl), where the heterocyclyl radical of the two last-mentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

7

,R

9

,R

11

are hydrogen, halogen, cyano, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, di(C

1

-C

6

-alkoxy)methyl, di(C

1

-C

6

-alkylthio)methyl, (C

1

-C

6

-alkoxy)(C

1

-C

6

-alkylthio)methyl, hydroxyl, C

1

-C

6

-alkoxy, C

1

-C

6

-haloalkoxy, C

1

-C

6

-alkoxycarbonyloxy, C

1

-C

6

-alkylthio, C

1

-C

6

-haloalkylthio, C

1

-C

6

-alkylsulfonyl, C

1

-C

6

-haloalkylsulfonyl, C

1

-C

6

-alkylcarbonyl, C

1

-C

6

-haloalkylcarbonyl, C

1

-C

6

-alkoxycarbonyl or C

1

-C

6

-haloalkoxycarbonyl;

R

8

,R

10

,R

12

are hydrogen or C

1

-C

6

-alkyl;

in particular hydrogen or C

1

-C

4

-alkyl, such as methyl or ethyl; or

R

7

and R

8

or R

9

and R

10

or R

11

and R

12

together form a —O—(CH

2

)

u

—O—, —O—(CH

2

)

u

—S—, —S—(CH

2

)

u

—S—, —O—(CH

2

)

v

— or —S—(CH

2

)

v

chain which may be substituted by one to three radicals from the following group:

halogen, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl or C

1

-C

4

-alkoxycarbonyl; or

R

7

and R

8

or R

9

and R

10

or R

11

and R

12

together form a —(CH

2

)

w

chain which may be interrupted by oxygen or sulfur and/or substituted by one to four radicals from the following group:

halogen, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl or C

1

-C

4

-alkoxycarbonyl; or

R

7

and R

8

or R

9

and R

10

or R

11

and R

12

together with the carbon atoms to which they are attached form a carbonyl group; or

R

7

and R

9

or R

9

and R

11

or R

7

and R

11

together form a —(CH

2

)

v

chain which may be substituted by one to three radicals from the following group: halogen, C

1

-C

6

-alkyl, C

1

-C

6

-alkoxy, hydroxyl or C

1

-C

6

-alkoxycarbonyl;

R

13

is C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-alkynyl, C

1

-C

6

-alkylcarbonyl, C

2

-C

6

-alkenylcarbonyl, C

3

-C

6

-cycloalkylcarbonyl, C

1

-C

6

-alkylaminocarbonyl, C

1

-C

6

-alkylcarbonyl-C

1

-C

6

-alkyl or C

1

-C

6

-alkoxyimino-C

1

-C

6

-alkyl, where the abovementioned alkyl and cycloalkyl radicals may be partially or fully halogenated and/or may carry one to three of the following groups:

cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio, C

1

-C

4

-alkylcarbonyl, C

1

-C

4

-alkoxycarbonyl, hydroxycarbonyl, di(C

1

-C

4

-alkyl)aminocarbonyl, C

1

-C

4

-alkylcarbonyloxy or C

3

-C

6

-cycloalkyl;

is phenyl, heterocyclyl, phenyl-C

1

-C

6

-alkyl, heterocyclyl-C

1

-C

6

-alkyl, phenylcarbonyl or heterocyclylcarbonyl, where the phenyl and the heterocyclyl radical of the 6 last-mentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

14

,R

15

, R

16

are C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-cycloalkyl, hydroxyl, C

1

-C

6

-alkoxy, di(C

1

-C

6

-alkyl)amino or di(C

1

-C

6

-haloalkyl)amino, where the abovementioned alkyl, cycloalkyl and alkoxy radicals may be partially or fully halogenated and/or may carry one to three of the following groups: cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio, C

1

-C

4

-alkylcarbonyl or C

1

-C

4

-alkoxycarbonyl;

are phenyl, heterocyclyl, phenoxy or heterocyclyloxy, where the phenyl and the heterocyclyl radical of the last-mentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

17

is C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-cycloalkyl, C

1

-C

6

-alkoxy or C

3

-C

6

-alkenyloxy, where the abovementioned alkyl, cycloalkyl and alkoxy radicals may be partially or fully halogenated and/or may carry one to three radicals from the following group:

cyano, C

1

-C

4

-alkoxy or C

1

-C

4

-alkylthio;

is phenyl, heterocyclyl, phenyl-C

1

-C

6

-alkyl or heterocyclyl-C

1

-C

6

-alkyl, where the phenyl or heterocyclyl radical of the four last-mentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

18

, R

19

are C

1

-C

6

-alkyl or C

3

-C

6

-alkenyl;

u is from 2 to 4;

v is from 1 to 5;

w is from 2 to 5;

R

20

is a radical as mentioned under R

6

;

R

21

is hydrogen, C

1

-C

6

-alkyl or C

1

-C

6

-haloalkyl; in particular hydrogen or C

1

-C

4

-alkyl such as methyl, ethyl, propyl, 1-methyleth-1-yl or 1,1-dimethyleth-1-yl;

R

22

is hydrogen or C

1

-C

6

-alkyl; in particular hydrogen or C

1

-C

4

-alkyl, such as methyl or ethyl;

R

23

is C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, C

3

-C

6

-cycloalkyl or C

3

-C

6

-halocycloalkyl; in particular C

1

-C

6

-alkyl or C

3

-C

6

-cycloalkyl; very preferably cyclopropyl;

R

24

is hydrogen;

R

25

is C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, C

3

-C

6

-cycloalkyl or C

3

-C

6

-halocycloalkyl; in particular C

1

-C

6

-alkyl or C

3

-C

6

-cycloalkyl.

Particular preference is given to the compounds Ia especially the compounds Ia where the variables have the following meanings, in each case on their own or in combination:

R

6

is hydroxyl, mercapto, halogen, OR

13

, SR

13

, SO

2

R

14

, OSO

2

R

14

, NR

17

R

18

, ONR

18

R

19

or N-bonded heterocyclyl, where the heterocyclyl radical of the last-mentioned substituent may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

7

,R

9

,R

11

are hydrogen, halogen, cyano, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, di(C

1

-C

6

-alkoxy)methyl, di(C

1

-C

6

-alkylthio)methyl, (C

1

-C

6

-alkoxy)(C

1

-C

6

-alkylthio)methyl, hydroxyl, C

1

-C

6

-alkoxy, C

1

-C

6

-haloalkoxy, C

1

-C

6

-alkoxycarbonyloxy, C

1

-C

6

-alkylthio or C

1

-C

6

-haloalkylthio;

R

8

,R

10

,R

12

are hydrogen or C

1

-C

6

-alkyl;

in particular hydrogen or C

1

-C

4

-alkyl, such as methyl or ethyl; or

R

9

and R

10

together with the carbon to which they are attached form a carbonyl group; or

R

7

and R

11

together form a —(CH

2

)

v

chain which may be substituted by one to three C

1

-C

4

-alkyl radicals;

R

13

is C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-alkynyl, C

1

-C

6

-alkylcarbonyl, C

3

-C

6

-cycloalkylcarbonyl, C

1

-C

6

-alkylaminocarbonyl or C

1

-C

6

-alkylcarbonyl-C

1

-C

6

-alkyl, where the abovementioned alkyl or cycloalkyl radicals may be partially or fully halogenated and/or may carry one to three of the following groups:

cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio, C

1

-C

4

-alkylcarbonyl, C

1

-C

4

-alkoxycarbonyl, hydroxycarbonyl, di(C

1

-C

4

-alkyl)aminocarbonyl, C

1

-C

4

-alkylcarbonyloxy or C

3

-C

6

-cycloalkyl;

is phenyl, heterocyclyl, phenyl-C

1

-C

6

-alkyl, heterocyclyl-C

1

-C

6

-alkyl, phenylcarbonyl or heterocyclylcarbonyl, where the phenyl and the heterocyclyl radical of the 6 last-mentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

14

is C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-cycloalkyl, hydroxyl, C

1

-C

6

-alkoxy, di(C

1

-C

6

-alkyl)amino or di(C

1

-C

6

-haloalkyl)amino, where the abovementioned alkyl, cycloalkyl and alkoxy radicals may be partially or fully halogenated and/or may carry one to three of the following groups:

cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio, C

1

-C

4

-alkylcarbonyl or C

1

-C

4

-alkoxycarbonyl;

are phenyl, heterocyclyl, phenoxy or heterocyclyloxy, where the phenyl and the heterocyclyl radical of the last-mentioned substituents may be partially or fully halogenated and/or carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

17

is C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-cycloalkyl, C

1

-C

6

-alkoxy or C

3

-C

6

-alkenyloxy, where the abovementioned alkyl, cycloalkyl and alkoxy radicals may be partially or fully halogenated and/or may carry one to three radicals from the following group:

cyano, C

1

-C

4

-alkoxy or C

1

-C

4

-alkylthio;

is phenyl, heterocyclyl, phenyl-C

1

-C

6

-alkyl or heterocyclyl-C

1

-C

6

-alkyl, where the phenyl or heterocyclyl radical of the four last-mentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

18

, R

19

are C

1

-C

6

-alkyl or C

3

-C

6

-alkenyl;

v is 1 or 2;

in particular 2.

Particular preference is also given to compounds of the formula Ia where

R

6

is hydroxyl, mercapto, phenylcarbonyloxy, C

1

-C

6

-alkylthio, phenylthio, N—(C

1

-C

6

-alkoxy)-N—(C

1

-C

6

-alkyl)amino, 1-tetrahydropyrrolyl or 2-tetrahydroisoxazolyl, where the phenyl radicals of the abovementioned radicals may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

in particular hydroxyl, phenylcarbonyloxy, C

1

-C

4

-alkylthio, phenylthio, N—(C

1

-C

4

-alkoxy)-N—(C

1

-C

4

-alkyl)amino, 1-tetrahydropyrrolyl or 2-tetrahydroisoxazolyl;

R

7

,R

8

,R

9

,R

10

,R

11

,R

12

are hydrogen or C

1

-C

4

-alkyl, such as methyl or ethyl;

in particular hydrogen or methyl; or

R

9

and R

10

together with the carbon to which they are attached form a carbonyl group; or

R

7

and R

11

together form a —(CH

2

)— or —(CH

2

)

2

— chain.

Extraordinary preference is given to the compounds of the formula Ia where

R

6

is hydroxyl, mercapto, phenylcarbonyloxy, C

1

-C

6

-alkylthio, phenylthio, where the phenyl radicals of the abovementioned radicals may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

in particular hydroxyl or phenylthio, where the phenyl radical may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy.

Preference is also given to compounds Ib, especially compounds Ib where the variables have the following meanings:

R

20

is a radical as mentioned under R

6

;

R

21

is hydrogen, C

1

-C

6

-alkyl or C

1

-C

6

-haloalkyl; in particular C

1

-C

4

-alkyl, such as methyl, ethyl, 1-methyleth-1-yl or 1,1-dimethyleth-1-yl, or C

1

-C

4

-haloalkyl, such as 2-fluoroethyl or 2,2,2-trifluoroethyl;

R

22

is hydrogen, C

1

-C

6

-alkyl or C

1

-C

6

-haloalkyl, in particular hydrogen, C

1

-C

4

-alkyl, such as methyl or ethyl, or C

1

-C

4

-haloalkyl, such as trifluoromethyl; in particular hydrogen, methyl or trifluoromethyl.

Preference is also given to the compounds Ib where the variables have the following meanings:

R

20

is hydroxyl, mercapto, halogen, OR

13

, SR

13

, SO

2

R

14

, OSO

2

R

14

, NR

17

R

18

, ONR

18

R

19

or N-bonded heterocyclyl, where the heterocyclyl radical of the lastmentioned substituent may be partially or fully halogenated and/or may carry one to three of the following radicals: nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

13

is C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-alkynyl, C

1

-C

6

-alkylcarbonyl, C

3

-C

6

-cycloalkylcarbonyl, C

1

-C

6

-alkylaminocarbonyl, N,N-di-(C

1

-C

6

-alkyl) or C

1

-C

6

-alkylcarbonyl-C

1

-C

6

-alkyl, where the alkyl or cycloalkyl radicals mentioned may be partially or fully halogenated and/or may carry one to three of the following groups:

cyano, C

1 4

-alkoxy, C

1

-C

4

-alkylthio, C

1

-C

4

-alkylcarbonyl, C

1

-C

4

-alkoxycarbonyl, hydroxycarbonyl, di-(C

1

-C

4

-alkyl)aminocarbonyl, C

1

-C

4

-alkylcarbonyloxy or C

3

-C

6

-cycloalkyl;

is phenyl, heterocyclyl, phenyl-C

1

-C

6

-alkyl, heterocyclyl-C

1

-C

6

-alkyl, phenylcarbonyl or heterocyclylcarbonyl, where the phenyl and the heterocyclyl radical of the 6 lastmentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

14

is C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-cycloalkyl, hydroxyl, C

1

-C

6

-alkoxy, di-(C

1

-C

6

-alkyl)amino or di-(C

1

-C

6

-haloalkyl)amino, where the alkyl, cycloalkyl and alkoxy radicals mentioned may be partially or fully halogenated and/or may carry one to three of the following groups:

cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio, C

1

-C

4

-alkylcarbonyl or C

1

-C

4

-alkoxycarbonyl;

is phenyl, heterocyclyl, phenoxy or heterocyclyloxy, where the phenyl and the heterocyclyl radical of the lastmentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

17

is C

1

-C

6

-alkyl, C

3

-C

6

-alkenyl, C

3

-C

6

-haloalkenyl, C

3

-C

6

-cycloalkyl, C

1

-C

6

-alkoxy or C

3

-C

6

-alkenyloxy, where the alkyl, cycloalkyl and alkoxy radicals mentioned may be partially or fully halogenated and/or may carry one to three radicals from the group below:

cyano, C

1

-C

4

-alkoxy or C

1

-C

4

-alkylthio;

is phenyl, heterocyclyl, phenyl-C

1

-C

6

-alkyl or heterocyclyl-C

1

-C

6

-alkyl, where the phenyl or heterocyclyl radical of the four lastmentioned substituents may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

18

, R

19

are C

1

-C

6

-alkyl or C

3

-C

6

-alkenyl;

R

21

is C

1

-C

6

-alkyl, such as methyl, ethyl, 1-methyleth-1-yl, or 1,1-dimethyleth-1-yl;

R

22

is hydrogen or C

1

-C

6

-alkyl such as methyl or ethyl; in particular hydrogen or methyl.

Extraordinary preference is given to the compounds Ib where the variables have the following meaning:

R

20

is hydroxyl.

Preference is also given to compounds of the formula Ic, especially compounds Ic where the variables have the following meanings:

R

23

is C

1

-C

6

-alkyl or C

3

-C

6

-cycloalkyl; in particular cyclopropyl;

R

24

is hydrogen.

Preference is also given to compounds of the formula Id, especially compounds Id where the variables have the following meanings:

R

25

is C

1

-C

6

-alkyl or C

3

-C

6

-cycloalkyl.

Preference is furthermore given to the compounds I1 (≡I where X═O, R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position)

With respect to the variables R

1

to R

4

and Q, what is said above applies.

Particular preference is given to the compounds I1 where the variables have the following meanings:

R

3

is nitro, cyano, halogen, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

6

-alkoxy, C

1

-C

4

-haloalkoxy, C

1

-C

4

-alkylsulfonyl or C

1

-C

4

-haloalkylsulfonyl;

R

4

is halogen, such as chlorine or bromine, or C

1

-C

4

-alkyl, such as methyl or ethyl;

l is 0 or 1.

Furthermore, preference is also given to the compounds I2 (≡I where X═O, R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position)

With respect to the variables R

1

to R

4

and Q, what was said above applies.

Particular preference is given to the compounds I2 where the variables have the following meanings:

R

3

is nitro, cyano, halogen, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy, C

1

-C

4

-alkylthio, C

1

-C

4

-haloalkylthio, C

1

-C

4

-alkylsulfonyl or C

1

-C

4

-haloalkylsulfonyl;

R

4

is halogen, such as chlorine or bromine, or C

1

-C

4

-alkyl, such as methyl or ethyl;

l is 0 or 1.

Preference is furthermore given to the compounds I, in particular the compounds Ia, Ib, I1 or I2, where the variables have the following meanings:

R

1

,R

2

are hydrogen, hydroxyl, C

1

-C

6

-alkyl or C

1

-C

6

-alkoxy, where the alkyl radicals of the two lastmentioned substituents may be partially or fully halogenated and/or may carry one to three of the following groups: nitro, cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylsulfonyl or C

1

-C

4

-alkoxycarbonyl;

particularly preferably hydrogen, C

1

-C

4

-alkyl or C

1

-C

4

-alkoxy.

Preference is furthermore given to the compounds I1a (≡I where X═O, R

3

is attached in position 4, R

4

l

is attached in position 5 and “P(═X)R

1

R

2

” is attached in position 2 and Q=Q

1

).

Particular preference is given to the compounds I1a (≡I where X═O, R

3

is in position 4, R

4

l

is in position 5 and “P(═X)R

1

R

2

” is in position 2), where the variables have the following meanings:

R

1

,R

2

are C

1

-C

4

-alkyl or C

1

-C

4

-alkoxy;

in particular C

1

-C

4

-alkyl;

R

3

is halogen;

l is 0;

R

6

is hydroxyl;

R

7

,R

8

,R

9

,R

10

,R

11

,R

12

are hydrogen or C

1

-C

4

-alkyl,

or R

9

and R

10

together with the carbon to which they are attached form a carbonyl group.

Preference is furthermore given to the compounds I2a (≡I where X═O, R

3

is attached in position 2, R

4

l

is attached in position 5 and “P(═X)R

1

R

2

” is attached in position 4 and Q=Q

1

).

Particular preference is given to the compounds I2a (≡I where X═O, R

3

is attached in position 2, R

4

l

is attached in position 5 and “P(═X)R

1

R

2

” is attached in position 4 and Q=Q

1

), where the variables have the following meanings:

R

1

,R

2

are C

1

-C

4

-alkyl or C

1

-C

4

-alkoxy;

R

3

is halogen;

l is 0;

R

6

is hydroxyl or phenylthio, where the phenyl radical may be partially or fully halogenated and/or may carry one to three of the following radicals:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy or C

1

-C

4

-haloalkoxy;

R

7

,R

8

,R

9

,R

10

,R

11

,R

12

are hydrogen or C

1

-C

4

-alkyl; or R

9

and R

10

together with the carbon to which they are attached form a carbonyl group;

or R

7

and R

11

together form a —(CH

2

)— or —(CH

2

)

2

— chain, in particular a —(CH

2

)

2

— chain.

Preference is furthermore given to the compounds I2b (≡I where X═O, R

3

is in position 2, R

4

l

is in position 5 and “P(═X)R

1

R

2

” is in position 4).

Particular preference is given to the compounds I2b (≡I where X═O, R

3

is in position 2, R

4

l

is in position 5 and “P(═X)R

1

R

2

” is in position 4), where the variables have the following meanings:

R

1

,R

2

are C

1

-C

4

-alkyl or C

1

-C

4

-alkoxy; in particular C

1

-C

4

-alkoxy;

R

3

is halogen;

l is 0;

R

20

is hydroxyl;

R

21

is C

1

-C

4

-alkyl;

R

22

is hydrogen or C

1

-C

4

-alkyl; in particular hydrogen.

Extraordinary preference is given to the compounds I1a1 (≡I where X═O, R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position, Q=Q

1

, R

7

to R

12

=hydrogen), in particular to the compounds I1a1.n where the variables R

1

to R

4

and R

6

are as defined in Table 1.

The given radical definitions X, R

1

to R

12

, Q and l are preferred for the compounds according to the invention not only in combination with one another, but in each case also on their own.

TABLE 1

I1a1

n

R

1

R

2

R

3

R

4

R

6

1

H

H

H

H(l = O)

OH

2

CH

3

CH

3

H

H(l = O)

OH

3

CH

2

CH

3

CH

2

CH

3

H

H(l = O)

OH

4

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

H(l = O)

OH

5

OCH

3

OCH

3

H

H(l = O)

OH

6

OCH

2

CH

3

OCH

2

CH

3

H

H(l = O)

OH

7

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

H(l = O)

OH

8

SCH

3

SCH

3

H

H(l = O)

OH

9

SCH

2

CH

3

SCH

2

CH

3

H

H(l = O)

OH

10

N(CH

3

)

2

N(CH

3

)

2

H

H(l = O)

OH

11

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

H(l = O)

OH

12

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

H(l = O)

OH

13

O—(CH

2

CH

2

)—O

H

H(l = O)

OH

14

O—(CH

2

CH

2

CH

2

)—O

H

H(l = O)

OH

15

S—(CH

2

CH

2

)—S

H

H(l = O)

OH

16

S—(CH

2

CH

2

CH

2

)—S

H

H(l = O)

OH

17

—(CH

2

)

4

—

H

H(l = O)

OH

18

—(CH

2

)

5

—

H

H(l = O)

OH

19

H

H

NO

2

H(l = O)

OH

20

CH

3

CH

3

NO

2

H(l = O)

OH

21

CH

2

CH

3

CH

2

CH

3

NO

2

H(l = O)

OH

22

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

H(l = O)

OH

23

OCH

3

OCH

3

NO

2

H(l = O)

OH

24

OCH

2

CH

3

OCH

2

CH

3

NO

2

H(l = O)

OH

25

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

H(l = O)

OH

26

SCH

3

SCH

3

NO

2

H(l = O)

OH

27

SCH

2

CH

3

SCH

2

CH

3

NO

2

H(l = O)

OH

28

N(CH

3

)

2

N(CH

3

)

2

NO

2

H(l = O)

OH

29

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

H(l = O)

OH

30

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

H(l = O)

OH

31

O—(CH

2

CH

2

)—O

NO

2

H(l = O)

OH

32

O—(CH

2

CH

2

CH

2

)—O

NO

2

H(l = O)

OH

33

S—(CH

2

CH

2

)—S

NO

2

H(l = O)

OH

34

S—(CH

2

CH

2

CH

2

)—S

NO

2

H(l = O)

OH

35

—(CH

2

)

4

—

NO

2

H(l = O)

OH

36

—(CH

2

)

5

—

NO

2

H(l = O)

OH

37

H

H

CN

H(l = O)

OH

38

CH

3

CH

3

CN

H(l = O)

OH

39

CH

2

CH

3

CH

2

CH

3

CN

H(l = O)

OH

40

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

H(l = O)

OH

41

OCH

3

OCH

3

CN

H(l = O)

OH

42

OCH

2

CH

3

OCH

2

CH

3

CN

H(l = O)

OH

43

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

H(l = O)

OH

44

SCH

3

SCH

3

CN

H(l = O)

OH

45

SCH

2

CH

3

SCH

2

CH

3

CN

H(l = O)

OH

46

N(CH

3

)

2

N(CH

3

)

2

CN

H(l = O)

OH

47

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

H(l = O)

OH

48

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

H(l = O)

OH

49

O—(CH

2

CH

2

)—O

CN

H(l = O)

OH

50

O—(CH

2

CH

2

CH

2

)—O

CN

H(l = O)

OH

51

S—(CH

2

CH

2

)—S

CN

H(l = O)

OH

52

S—(CH

2

CH

2

CH

2

)—S

CN

H(l = O)

OH

53

—(CH

2

)

4

—

CN

H(l = O)

OH

54

—(CH

2

)

5

—

CN

H(l = O)

OH

55

H

H

F

H(l = O)

OH

56

CH

3

CH

3

F

H(l = O)

OH

57

CH

2

CH

3

CH

2

CH

3

F

H(l = O)

OH

58

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

H(l = O)

OH

59

OCH

3

OCH

3

F

H(l = O)

OH

60

OCH

2

CH

3

OCH

2

CH

3

F

H(l = O)

OH

61

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

H(l = O)

OH

62

SCH

3

SCH

3

F

H(l = O)

OH

63

SCH

2

CH

3

SCH

2

CH

3

F

H(l = O)

OH

64

N(CH

3

)

2

N(CH

3

)

2

F

H(l = O)

OH

65

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

H(l = O)

OH

66

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

H(l = O)

OH

67

O—(CH

2

CH

2

)—O

F

H(l = O)

OH

68

O—(CH

2

CH

2

CH

2

)—O

F

H(l = O)

OH

69

S—(CH

2

CH

2

)—S

F

H(l = O)

OH

70

S—(CH

2

CH

2

CH

2

)—S

F

H(l = O)

OH

71

—(CH

2

)

4

—

F

H(l = O)

OH

72

—(CH

2

)

5

—

F

H(l = O)

OH

73

H

H

Cl

H(l = O)

OH

74

CH

3

CH

3

Cl

H(l = O)

OH

75

CH

2

CH

3

CH

2

CH

3

Cl

H(l = O)

OH

76

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

H(l = O)

OH

77

OCH

3

OCH

3

Cl

H(l = O)

OH

78

OCH

2

CH

3

OCH

2

CH

3

Cl

H(l = O)

OH

79

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

H(l = O)

OH

80

SCH

3

SCH

3

Cl

H(l = O)

OH

81

SCH

2

CH

3

SCH

2

CH

3

Cl

H(l = O)

OH

82

N(CH

3

)

2

N(CH

3

)

2

Cl

H(l = O)

OH

83

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

H(l = O)

OH

84

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

H(l = O)

OH

85

O—(CH

2

CH

2

)—O

Cl

H(l = O)

OH

86

O—(CH

2

CH

2

CH

2

)—O

Cl

H(l = O)

OH

87

S—(CH

2

CH

2

)—S

Cl

H(l = O)

OH

88

S—(CH

2

CH

2

CH

2

)—S

Cl

H(l = O)

OH

89

—(CH

2

)

4

—

Cl

H(l = O)

OH

90

—(CH

2

)

5

—

Cl

H(l = O)

OH

91

H

H

Br

H(l = O)

OH

92

CH

3

CH

3

Br

H(l = O)

OH

93

CH

2

CH

3

CH

2

CH

3

Br

H(l = O)

OH

94

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

H(l = O)

OH

95

OCH

3

OCH

3

Br

H(l = O)

OH

96

OCH

2

CH

3

OCH

2

CH

3

Br

H(l = O)

OH

97

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

H(l = O)

OH

98

SCH

3

SCH

3

Br

H(l = O)

OH

99

SCH

2

CH

3

SCH

2

CH

3

Br

H(l = O)

OH

100

N(CH

3

)

2

N(CH

3

)

2

Br

H(l = O)

OH

101

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

H(l = O)

OH

102

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

H(l = O)

OH

103

O—(CH

2

CH

2

)—O

Br

H(l = O)

OH

104

O—(CH

2

CH

2

CH

2

)—O

Br

H(l = O)

OH

105

S—(CH

2

CH

2

)—S

Br

H(l = O)

OH

106

S—(CH

2

CH

2

CH

2

)—S

Br

H(l = O)

OH

107

—(CH

2

)

4

—

Br

H(l = O)

OH

108

—(CH

2

)

5

—

Br

H(l = O)

OH

109

H

H

CH

3

H(l = O)

OH

110

CH

3

CH

3

CH

3

H(l = O)

OH

111

CH

2

CH

3

CH

2

CH

3

CH

3

H(l = O)

OH

112

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

H(l = O)

OH

113

OCH

3

OCH

3

CH

3

H(l = O)

OH

114

OCH

2

CH

3

OCH

2

CH

3

CH

3

H(l = O)

OH

115

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

H(l = O)

OH

116

SCH

3

SCH

3

CH

3

H(l = O)

OH

117

SCH

2

CH

3

SCH

2

CH

3

CH

3

H(l = O)

OH

118

N(CH

3

)

2

N(CH

3

)

2

CH

3

H(l = O)

OH

119

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

H(l = O)

OH

120

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

H(l = O)

OH

121

O—(CH

2

CH

2

)—O

CH

3

H(l = O)

OH

122

O—(CH

2

CH

2

CH

2

)—O

CH

3

H(l = O)

OH

123

S—(CH

2

CH

2

)—S

CH

3

H(l = O)

OH

124

S—(CH

2

CH

2

CH

2

)—S

CH

3

H(l = O)

OH

125

—(CH

2

)

4

—

CH

3

H(l = O)

OH

126

—(CH

2

)

5

—

CH

3

H(l = O)

OH

127

H

H

CH

2

CH

3

H(l = O)

OH

128

CH

3

CH

3

CH

2

CH

3

H(l = O)

OH

129

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

H(l = O)

OH

130

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

OH

131

OCH

3

OCH

3

CH

2

CH

3

H(l = O)

OH

132

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

H(l = O)

OH

133

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

OH

134

SCH

3

SCH

3

CH

2

CH

3

H(l = O)

OH

135

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

H(l = O)

OH

136

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

H(l = O)

OH

137

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

H(l = O)

OH

138

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

H(l = O)

OH

139

O—(CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

OH

140

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

OH

141

S—(CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

OH

142

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

OH

143

—(CH

2

)

4

—

CH

2

CH

3

H(l = O)

OH

144

—(CH

2

)

5

—

CH

2

CH

3

H(l = O)

OH

145

H

H

CF

3

H(l = O)

OH

146

CH

3

CH

3

CF

3

H(l = O)

OH

147

CH

2

CH

3

CH

2

CH

3

CF

3

H(l = O)

OH

148

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

H(l = O)

OH

149

OCH

3

OCH

3

CF

3

H(l = O)

OH

150

OCH

2

CH

3

OCH

2

CH

3

CF

3

H(l = O)

OH

151

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

H(l = O)

OH

152

SCH

3

SCH

3

CF

3

H(l = O)

OH

153

SCH

2

CH

3

SCH

2

CH

3

CF

3

H(l = O)

OH

154

N(CH

3

)

2

N(CH

3

)

2

CF

3

H(l = O)

OH

155

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

H(l = O)

OH

156

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

H(l = O)

OH

157

O—(CH

2

CH

2

)—O

CF

3

H(l = O)

OH

158

O—(CH

2

CH

2

CH

2

)—O

CF

3

H(l = O)

OH

159

S—(CH

2

CH

2

)—S

CF

3

H(l = O)

OH

160

S—(CH

2

CH

2

CH

2

)—S

CF

3

H(l = O)

OH

161

—(CH

2

)

4

—

CF

3

H(l = O)

OH

162

—(CH

2

)

5

—

CF

3

H(l = O)

OH

163

H

H

OCH

3

H(l = O)

OH

164

CH

3

CH

3

OCH

3

H(l = O)

OH

165

CH

2

CH

3

CH

2

CH

3

OCH

3

H(l = O)

OH

166

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

H(l = O)

OH

167

OCH

3

OCH

3

OCH

3

H(l = O)

OH

168

OCH

2

CH

3

OCH

2

CH

3

OCH

3

H(l = O)

OH

169

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

H(l = O)

OH

170

SCH

3

SCH

3

OCH

3

H(l = O)

OH

171

SCH

2

CH

3

SCH

2

CH

3

OCH

3

H(l = O)

OH

172

N(CH

3

)

2

N(CH

3

)

2

OCH

3

H(l = O)

OH

173

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

H(l = O)

OH

174

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

H(l = O)

OH

175

O—(CH

2

CH

2

)—O

OCH

3

H(l = O)

OH

176

O—(CH

2

CH

2

CH

2

)—O

OCH

3

H(l = O)

OH

177

S—(CH

2

CH

2

)—S

OCH

3

H(l = O)

OH

178

S—(CH

2

CH

2

CH

2

)—S

OCH

3

H(l = O)

OH

179

—(CH

2

)

4

—

OCH

3

H(l = O)

OH

180

—(CH

2

)

5

—

OCH

3

H(l = O)

OH

181

H

H

OCH

2

CH

3

H(l = O)

OH

182

CH

3

CH

3

OCH

2

CH

3

H(l = O)

OH

183

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

H(l = O)

OH

184

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

OH

185

OCH

3

OCH

3

OCH

2

CH

3

H(l = O)

OH

186

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

H(l = O)

OH

187

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

OH

188

SCH

3

SCH

3

OCH

2

CH

3

H(l = O)

OH

189

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

H(l = O)

OH

190

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

H(l = O)

OH

191

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

H(l = O)

OH

192

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

H(l = O)

OH

193

O—(CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

OH

194

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

OH

195

S—(CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

OH

196

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

OH

197

—(CH

2

)

4

—

OCH

2

CH

3

H(l = O)

OH

198

—(CH

2

)

5

—

OCH

2

CH

3

H(l = O)

OH

199

H

H

SCH

3

H(l = O)

OH

200

CH

3

CH

3

SCH

3

H(l = O)

OH

201

CH

2

CH

3

CH

2

CH

3

SCH

3

H(l = O)

OH

202

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

H(l = O)

OH

203

OCH

3

OCH

3

SCH

3

H(l = O)

OH

204

OCH

2

CH

3

OCH

2

CH

3

SCH

3

H(l = O)

OH

205

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

H(l = O)

OH

206

SCH

3

SCH

3

SCH

3

H(l = O)

OH

207

SCH

2

CH

3

SCH

2

CH

3

SCH

3

H(l = O)

OH

208

N(CH

3

)

2

N(CH

3

)

2

SCH

3

H(l = O)

OH

209

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

H(l = O)

OH

210

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

H(l = O)

OH

211

O—(CH

2

CH

2

)—O

SCH

3

H(l = O)

OH

212

O—(CH

2

CH

2

CH

2

)—O

SCH

3

H(l = O)

OH

213

S—(CH

2

CH

2

)—S

SCH

3

H(l = O)

OH

214

S—(CH

2

CH

2

CH

2

)—S

SCH

3

H(l = O)

OH

215

—(CH

2

)

4

—

SCH

3

H(l = O)

OH

216

—(CH

2

)

5

—

SCH

3

H(l = O)

OH

217

H

H

SO

2

CH

3

H(l = O)

OH

218

CH

3

CH

3

SO

2

CH

3

H(l = O)

OH

219

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

H(l = O)

OH

220

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

OH

221

OCH

3

OCH

3

SO

2

CH

3

H(l = O)

OH

222

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

H(l = O)

OH

223

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

OH

224

SCH

3

SCH

3

SO

2

CH

3

H(l = O)

OH

225

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

H(l = O)

OH

226

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

H(l = O)

OH

227

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

H(l = O)

OH

228

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

H(l = O)

OH

229

O—(CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

OH

230

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

OH

231

S—(CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

OH

232

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

OH

233

—(CH

2

)

4

—

SO

2

CH

3

H(l = O)

OH

234

—(CH

2

)

5

—

SO

2

CH

3

H(l = O)

OH

235

H

H

PO(OCH

3

)

2

H(l = O)

OH

236

CH

3

CH

3

PO(OCH

3

)

2

H(l = O)

OH

237

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

OH

238

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

OH

239

OCH

3

OCH

3

PO(OCH

3

)

2

H(l = O)

OH

240

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

OH

241

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

OH

242

SCH

3

SCH

3

PO(OCH

3

)

2

H(l = O)

OH

243

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

OH

244

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

H(l = O)

OH

245

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

H(l = O)

OH

246

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

H(l = O)

OH

247

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

OH

248

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

OH

249

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

OH

250

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

OH

251

—(CH

2

)

4

—

PO(OCH

3

)

2

H(l = O)

OH

252

—(CH

2

)

5

—

PO(OCH

3

)

2

H(l = O)

OH

253

H

H

PO(OCH

2

CH

3

)

2

H(l = O)

OH

254

CH

3

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OH

255

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OH

256

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OH

257

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OH

258

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OH

259

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OH

260

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OH

261

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OH

262

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

OH

263

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

OH

264

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

H(l = O)

OH

265

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

OH

266

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

OH

267

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

OH

268

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

OH

269

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

H(l = O)

OH

270

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

H(l = O)

OH

271

H

H

PO(CH

3

)

2

H(l = O)

OH

272

CH

3

CH

3

PO(CH

3

)

2

H(l = O)

OH

273

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

OH

274

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

OH

275

OCH

3

OCH

3

PO(CH

3

)

2

H(l = O)

OH

276

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

H(l = O)

OH

277

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

OH

278

SCH

3

SCH

3

PO(CH

3

)

2

H(l = O)

OH

279

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

H(l = O)

OH

280

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

H(l = O)

OH

281

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

H(l = O)

OH

282

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

H(l = O)

OH

283

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

OH

284

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

OH

285

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

OH

286

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

OH

287

—(CH

2

)

4

—

PO(CH

3

)

2

H(l = O)

OH

288

—(CH

2

)

5

—

PO(CH

3

)

2

H(l = O)

OH

289

H

H

PO(CH

2

CH

3

)

2

H(l = O)

OH

290

CH

3

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OH

291

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OH

292

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OH

293

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

H(l = O)

OH

294

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OH

295

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OH

296

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

H(l = O)

OH

297

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OH

298

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

OH

299

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

OH

300

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

H(l = O)

OH

301

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

OH

302

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

OH

303

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

OH

304

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

OH

305

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

H(l = O)

OH

306

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

H(l = O)

OH

307

H

H

H

H(l = O)

OCOC

6

H

5

308

CH

3

CH

3

H

H(l = O)

OCOC

6

H

5

309

CH

2

CH

3

CH

2

CH

3

H

H(l = O)

OCOC

6

H

5

310

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

H(l = O)

OCOC

6

H

5

311

OCH

3

OCH

3

H

H(l = O)

OCOC

6

H

5

312

OCH

2

CH

3

OCH

2

CH

3

H

H(l = O)

OCOC

6

H

5

313

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

H(l = O)

OCOC

6

H

5

314

SCH

3

SCH

3

H

H(l = O)

OCOC

6

H

5

315

SCH

2

CH

3

SCH

2

CH

3

H

H(l = O)

OCOC

6

H

5

316

N(CH

3

)

2

N(CH

3

)

2

H

H(l = O)

OCOC

6

H

5

317

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

H(l = O)

OCOC

6

H

5

318

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

H(l = O)

OCOC

6

H

5

319

O—(CH

2

CH

2

)—O

H

H(l = O)

OCOC

6

H

5

320

O—(CH

2

CH

2

CH

2

)—O

H

H(l = O)

OCOC

6

H

5

321

S—(CH

2

CH

2

)—S

H

H(l = O)

OCOC

6

H

5

322

S—(CH

2

CH

2

CH

2

)—S

H

H(l = O)

OCOC

6

H

5

323

—(CH

2

)

4

—

H

H(l = O)

OCOC

6

H

5

324

—(CH

2

)

5

—

H

H(l = O)

OCOC

6

H

5

325

H

H

NO

2

H(l = O)

OCOC

6

H

5

326

CH

3

CH

3

NO

2

H(l = O)

OCOC

6

H

5

327

CH

2

CH

3

CH

2

CH

3

NO

2

H(l = O)

OCOC

6

H

5

328

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

H(l = O)

OCOC

6

H

5

329

OCH

3

OCH

3

NO

2

H(l = O)

OCOC

6

H

5

330

OCH

2

CH

3

OCH

2

CH

3

NO

2

H(l = O)

OCOC

6

H

5

331

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

H(l = O)

OCOC

6

H

5

332

SCH

3

SCH

3

NO

2

H(l = O)

OCOC

6

H

5

333

SCH

2

CH

3

SCH

2

CH

3

NO

2

H(l = O)

OCOC

6

H

5

334

N(CH

3

)

2

N(CH

3

)

2

NO

2

H(l = O)

OCOC

6

H

5

335

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

H(l = O)

OCOC

6

H

5

336

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

H(l = O)

OCOC

6

H

5

337

O—(CH

2

CH

2

)—O

NO

2

H(l = O)

OCOC

6

H

5

338

O—(CH

2

CH

2

CH

2

)—O

NO

2

H(l = O)

OCOC

6

H

5

339

S—(CH

2

CH

2

)—S

NO

2

H(l = O)

OCOC

6

H

5

340

S—(CH

2

CH

2

CH

2

)—S

NO

2

H(l = O)

OCOC

6

H

5

341

—(CH

2

)

4

—

NO

2

H(l = O)

OCOC

6

H

5

342

—(CH

2

)

5

—

NO

2

H(l = O)

OCOC

6

H

5

343

H

H

CN

H(l = O)

OCOC

6

H

5

344

CH

3

CH

3

CN

H(l = O)

OCOC

6

H

5

345

CH

2

CH

3

CH

2

CH

3

CN

H(l = O)

OCOC

6

H

5

346

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

H(l = O)

OCOC

6

H

5

347

OCH

3

OCH

3

CN

H(l = O)

OCOC

6

H

5

348

OCH

2

CH

3

OCH

2

CH

3

CN

H(l = O)

OCOC

6

H

5

349

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

H(l = O)

OCOC

6

H

5

350

SCH

3

SCH

3

CN

H(l = O)

OCOC

6

H

5

351

SCH

2

CH

3

SCH

2

CH

3

CN

H(l = O)

OCOC

6

H

5

352

N(CH

3

)

2

N(CH

3

)

2

CN

H(l = O)

OCOC

6

H

5

353

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

H(l = O)

OCOC

6

H

5

354

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

H(l = O)

OCOC

6

H

5

355

O—(CH

2

CH

2

)—O

CN

H(l = O)

OCOC

6

H

5

356

O—(CH

2

CH

2

CH

2

)—O

CN

H(l = O)

OCOC

6

H

5

357

S—(CH

2

CH

2

)—S

CN

H(l = O)

OCOC

6

H

5

358

S—(CH

2

CH

2

CH

2

)—S

CN

H(l = O)

OCOC

6

H

5

359

—(CH

2

)

4

—

CN

H(l = O)

OCOC

6

H

5

360

—(CH

2

)

5

—

CN

H(l = O)

OCOC

6

H

5

361

H

H

F

H(l = O)

OCOC

6

H

5

362

CH

3

CH

3

F

H(l = O)

OCOC

6

H

5

363

CH

2

CH

3

CH

2

CH

3

F

H(l = O)

OCOC

6

H

5

364

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

H(l = O)

OCOC

6

H

5

365

OCH

3

OCH

3

F

H(l = O)

OCOC

6

H

5

366

OCH

2

CH

3

OCH

2

CH

3

F

H(l = O)

OCOC

6

H

5

367

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

H(l = O)

OCOC

6

H

5

368

SCH

3

SCH

3

F

H(l = O)

OCOC

6

H

5

369

SCH

2

CH

3

SCH

2

CH

3

F

H(l = O)

OCOC

6

H

5

370

N(CH

3

)

2

N(CH

3

)

2

F

H(l = O)

OCOC

6

H

5

371

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

H(l = O)

OCOC

6

H

5

372

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

H(l = O)

OCOC

6

H

5

373

O—(CH

2

CH

2

)—O

F

H(l = O)

OCOC

6

H

5

374

O—(CH

2

CH

2

CH

2

)—O

F

H(l = O)

OCOC

6

H

5

375

S—(CH

2

CH

2

)—S

F

H(l = O)

OCOC

6

H

5

376

S—(CH

2

CH

2

CH

2

)—S

F

H(l = O)

OCOC

6

H

5

377

—(CH

2

)

4

—

F

H(l = O)

OCOC

6

H

5

378

—(CH

2

)

5

—

F

H(l = O)

OCOC

6

H

5

379

H

H

Cl

H(l = O)

OCOC

6

H

5

380

CH

3

CH

3

Cl

H(l = O)

OCOC

6

H

5

381

CH

2

CH

3

CH

2

CH

3

Cl

H(l = O)

OCOC

6

H

5

382

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

H(l = O)

OCOC

6

H

5

383

OCH

3

OCH

3

Cl

H(l = O)

OCOC

6

H

5

384

OCH

2

CH

3

OCH

2

CH

3

Cl

H(l = O)

OCOC

6

H

5

385

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

H(l = O)

OCOC

6

H

5

386

SCH

3

SCH

3

Cl

H(l = O)

OCOC

6

H

5

387

SCH

2

CH

3

SCH

2

CH

3

Cl

H(l = O)

OCOC

6

H

5

388

N(CH

3

)

2

N(CH

3

)

2

Cl

H(l = O)

OCOC

6

H

5

389

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

H(l = O)

OCOC

6

H

5

390

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

H(l = O)

OCOC

6

H

5

391

O—(CH

2

CH

2

)—O

Cl

H(l = O)

OCOC

6

H

5

392

O—(CH

2

CH

2

CH

2

)—O

Cl

H(l = O)

OCOC

6

H

5

393

S—(CH

2

CH

2

)—S

Cl

H(l = O)

OCOC

6

H

5

394

S—(CH

2

CH

2

CH

2

)—S

Cl

H(l = O)

OCOC

6

H

5

395

—(CH

2

)

4

—

Cl

H(l = O)

OCOC

6

H

5

396

—(CH

2

)

5

—

Cl

H(l = O)

OCOC

6

H

5

397

H

H

Br

H(l = O)

OCOC

6

H

5

398

CH

3

CH

3

Br

H(l = O)

OCOC

6

H

5

399

CH

2

CH

3

CH

2

CH

3

Br

H(l = O)

OCOC

6

H

5

400

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

H(l = O)

OCOC

6

H

5

401

OCH

3

OCH

3

Br

H(l = O)

OCOC

6

H

5

402

OCH

2

CH

3

OCH

2

CH

3

Br

H(l = O)

OCOC

6

H

5

403

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

H(l = O)

OCOC

6

H

5

404

SCH

3

SCH

3

Br

H(l = O)

OCOC

6

H

5

405

SCH

2

CH

3

SCH

2

CH

3

Br

H(l = O)

OCOC

6

H

5

406

N(CH

3

)

2

N(CH

3

)

2

Br

H(l = O)

OCOC

6

H

5

407

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

H(l = O)

OCOC

6

H

5

408

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

H(l = O)

OCOC

6

H

5

409

O—(CH

2

CH

2

)—O

Br

H(l = O)

OCOC

6

H

5

410

O—(CH

2

CH

2

CH

2

)—O

Br

H(l = O)

OCOC

6

H

5

411

S—(CH

2

CH

2

)—S

Br

H(l = O)

OCOC

6

H

5

412

S—(CH

2

CH

2

CH

2

)—S

Br

H(l = O)

OCOC

6

H

5

413

—(CH

2

)

4

—

Br

H(l = O)

OCOC

6

H

5

414

—(CH

2

)

5

—

Br

H(l = O)

OCOC

6

H

5

415

H

H

CH

3

H(l = O)

OCOC

6

H

5

416

CH

3

CH

3

CH

3

H(l = O)

OCOC

6

H

5

417

CH

2

CH

3

CH

2

CH

3

CH

3

H(l = O)

OCOC

6

H

5

418

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

H(l = O)

OCOC

6

H

5

419

OCH

3

OCH

3

CH

3

H(l = O)

OCOC

6

H

5

420

OCH

2

CH

3

OCH

2

CH

3

CH

3

H(l = O)

OCOC

6

H

5

421

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

H(l = O)

OCOC

6

H

5

422

SCH

3

SCH

3

CH

3

H(l = O)

OCOC

6

H

5

423

SCH

2

CH

3

SCH

2

CH

3

CH

3

H(l = O)

OCOC

6

H

5

424

N(CH

3

)

2

N(CH

3

)

2

CH

3

H(l = O)

OCOC

6

H

5

425

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

H(l = O)

OCOC

6

H

5

426

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

H(l = O)

OCOC

6

H

5

427

O—(CH

2

CH

2

)—O

CH

3

H(l = O)

OCOC

6

H

5

428

O—(CH

2

CH

2

CH

2

)—O

CH

3

H(l = O)

OCOC

6

H

5

429

S—(CH

2

CH

2

)—S

CH

3

H(l = O)

OCOC

6

H

5

430

S—(CH

2

CH

2

CH

2

)—S

CH

3

H(l = O)

OCOC

6

H

5

431

—(CH

2

)

4

—

CH

3

H(l = O)

OCOC

6

H

5

432

—(CH

2

)

5

—

CH

3

H(l = O)

OCOC

6

H

5

433

H

H

CH

2

CH

3

H(l = O)

OCOC

6

H

5

434

CH

3

CH

3

CH

2

CH

3

H(l = O)

OCOC

6

H

5

435

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

H(l = O)

OCOC

6

H

5

436

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

OCOC

6

H

5

437

OCH

3

OCH

3

CH

2

CH

3

H(l = O)

OCOC

6

H

5

438

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

H(l = O)

OCOC

6

H

5

439

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

OCOC

6

H

5

440

SCH

3

SCH

3

CH

2

CH

3

H(l = O)

OCOC

6

H

5

441

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

H(l = O)

OCOC

6

H

5

442

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

H(l = O)

OCOC

6

H

5

443

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

H(l = O)

OCOC

6

H

5

444

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

H(l = O)

OCOC

6

H

5

445

O—(CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

OCOC

6

H

5

446

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

OCOC

6

H

5

447

S—(CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

OCOC

6

H

5

448

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

OCOC

6

H

5

449

—(CH

2

)

4

—

CH

2

CH

3

H(l = O)

OCOC

6

H

5

450

—(CH

2

)

5

—

CH

2

CH

3

H(l = O)

OCOC

6

H

5

451

H

H

CF

3

H(l = O)

OCOC

6

H

5

452

CH

3

CH

3

CF

3

H(l = O)

OCOC

6

H

5

453

CH

2

CH

3

CH

2

CH

3

CF

3

H(l = O)

OCOC

6

H

5

454

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

H(l = O)

OCOC

6

H

5

455

OCH

3

OCH

3

CF

3

H(l = O)

OCOC

6

H

5

456

OCH

2

CH

3

OCH

2

CH

3

CF

3

H(l = O)

OCOC

6

H

5

457

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

H(l = O)

OCOC

6

H

5

458

SCH

3

SCH

3

CF

3

H(l = O)

OCOC

6

H

5

459

SCH

2

CH

3

SCH

2

CH

3

CF

3

H(l = O)

OCOC

6

H

5

460

N(CH

3

)

2

N(CH

3

)

2

CF

3

H(l = O)

OCOC

6

H

5

461

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

H(l = O)

OCOC

6

H

5

462

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

H(l = O)

OCOC

6

H

5

463

O—(CH

2

CH

2

)—O

CF

3

H(l = O)

OCOC

6

H

5

464

O—(CH

2

CH

2

CH

2

)—O

CF

3

H(l = O)

OCOC

6

H

5

465

S—(CH

2

CH

2

)—S

CF

3

H(l = O)

OCOC

6

H

5

466

S—(CH

2

CH

2

CH

2

)—S

CF

3

H(l = O)

OCOC

6

H

5

467

—(CH

2

)

4

—

CF

3

H(l = O)

OCOC

6

H

5

468

—(CH

2

)

5

—

CF

3

H(l = O)

OCOC

6

H

5

469

H

H

OCH

3

H(l = O)

OCOC

6

H

5

470

CH

3

CH

3

OCH

3

H(l = O)

OCOC

6

H

5

471

CH

2

CH

3

CH

2

CH

3

OCH

3

H(l = O)

OCOC

6

H

5

472

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

H(l = O)

OCOC

6

H

5

473

OCH

3

OCH

3

OCH

3

H(l = O)

OCOC

6

H

5

474

OCH

2

CH

3

OCH

2

CH

3

OCH

3

H(l = O)

OCOC

6

H

5

475

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

H(l = O)

OCOC

6

H

5

476

SCH

3

SCH

3

OCH

3

H(l = O)

OCOC

6

H

5

477

SCH

2

CH

3

SCH

2

CH

3

OCH

3

H(l = O)

OCOC

6

H

5

478

N(CH

3

)

2

N(CH

3

)

2

OCH

3

H(l = O)

OCOC

6

H

5

479

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

H(l = O)

OCOC

6

H

5

480

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

H(l = O)

OCOC

6

H

5

481

O—(CH

2

CH

2

)—O

OCH

3

H(l = O)

OCOC

6

H

5

482

O—(CH

2

CH

2

CH

2

)—O

OCH

3

H(l = O)

OCOC

6

H

5

483

S—(CH

2

CH

2

)—S

OCH

3

H(l = O)

OCOC

6

H

5

484

S—(CH

2

CH

2

CH

2

)—S

OCH

3

H(l = O)

OCOC

6

H

5

485

—(CH

2

)

4

—

OCH

3

H(l = O)

OCOC

6

H

5

486

—(CH

2

)

5

—

OCH

3

H(l = O)

OCOC

6

H

5

487

H

H

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

488

CH

3

CH

3

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

489

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

490

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

491

OCH

3

OCH

3

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

492

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

493

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

494

SCH

3

SCH

3

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

495

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

496

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

497

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

498

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

499

O—(CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

500

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

501

S—(CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

502

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

503

—(CH

2

)

4

—

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

504

—(CH

2

)

5

—

OCH

2

CH

3

H(l = O)

OCOC

6

H

5

505

H

H

SCH

3

H(l = O)

OCOC

6

H

5

506

CH

3

CH

3

SCH

3

H(l = O)

OCOC

6

H

5

507

CH

2

CH

3

CH

2

CH

3

SCH

3

H(l = O)

OCOC

6

H

5

508

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

H(l = O)

OCOC

6

H

5

509

OCH

3

OCH

3

SCH

3

H(l = O)

OCOC

6

H

5

510

OCH

2

CH

3

OCH

2

CH

3

SCH

3

H(l = O)

OCOC

6

H

5

511

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

H(l = O)

OCOC

6

H

5

512

SCH

3

SCH

3

SCH

3

H(l = O)

OCOC

6

H

5

513

SCH

2

CH

3

SCH

2

CH

3

SCH

3

H(l = O)

OCOC

6

H

5

514

N(CH

3

)

2

N(CH

3

)

2

SCH

3

H(l = O)

OCOC

6

H

5

515

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

H(l = O)

OCOC

6

H

5

516

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

H(l = O)

OCOC

6

H

5

517

O—(CH

2

CH

2

)—O

SCH

3

H(l = O)

OCOC

6

H

5

518

O—(CH

2

CH

2

CH

2

)—O

SCH

3

H(l = O)

OCOC

6

H

5

519

S—(CH

2

CH

2

)—S

SCH

3

H(l = O)

OCOC

6

H

5

520

—(CH

2

)

4

—

SCH

3

H(l = O)

OCOC

6

H

5

521

—(CH

2

)

5

—

SCH

3

H(l = O)

OCOC

6

H

5

522

S—(CH

2

CH

2

CH

2

)—S

SCH

3

H(l = O)

OCOC

6

H

5

523

—(CH

2

)

4

—

SCH

3

H(l = O)

OCOC

6

H

5

524

—(CH

2

)

5

—

SCH

3

H(l = O)

OCOC

6

H

5

525

H

H

SO

2

CH

3

H(l = O)

OCOC

6

H

5

526

CH

3

CH

3

SO

2

CH

3

H(l = O)

OCOC

6

H

5

527

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

H(l = O)

OCOC

6

H

5

528

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

OCOC

6

H

5

529

OCH

3

OCH

3

SO

2

CH

3

H(l = O)

OCOC

6

H

5

530

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

H(l = O)

OCOC

6

H

5

531

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

OCOC

6

H

5

532

SCH

3

SCH

3

SO

2

CH

3

H(l = O)

OCOC

6

H

5

533

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

H(l = O)

OCOC

6

H

5

534

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

H(l = O)

OCOC

6

H

5

535

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

H(l = O)

OCOC

6

H

5

536

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

H(l = O)

OCOC

6

H

5

537

O—(CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

OCOC

6

H

5

538

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

OCOC

6

H

5

539

S—(CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

OCOC

6

H

5

540

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

OCOC

6

H

5

541

—(CH

2

)

4

—

SO

2

CH

3

H(l = O)

OCOC

6

H

5

542

—(CH

2

)

5

—

SO

2

CH

3

H(l = O)

OCOC

6

H

5

543

H

H

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

544

CH

3

CH

3

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

545

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

546

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

547

OCH

3

OCH

3

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

548

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

549

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

550

SCH

3

SCH

3

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

551

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

552

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

553

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

554

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

555

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

556

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

557

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

558

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

559

—(CH

2

)

4

—

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

560

—(CH

2

)

5

—

PO(OCH

3

)

2

H(l = O)

OCOC

6

H

5

561

H

H

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

562

CH

3

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

563

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

564

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

565

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

566

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

567

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

568

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

569

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

570

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

571

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

572

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

573

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

574

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

575

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

576

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

577

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

578

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

579

H

H

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

580

CH

3

CH

3

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

581

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

582

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

583

OCH

3

OCH

3

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

584

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

585

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

586

SCH

3

SCH

3

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

587

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

588

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

589

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

590

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

591

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

592

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

593

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

594

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

595

—(CH

2

)

4

—

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

596

—(CH

2

)

5

—

PO(CH

3

)

2

H(l = O)

OCOC

6

H

5

597

H

H

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

598

CH

3

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

599

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

600

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

601

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

602

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

603

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

604

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

605

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

606

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

607

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

608

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

609

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

610

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

611

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

612

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

613

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

614

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

H(l = O)

OCOC

6

H

5

615

H

H

H

H(l = O)

SCH

3

616

CH

3

CH

3

H

H(l = O)

SCH

3

617

CH

2

CH

3

CH

2

CH

3

H

H(l = O)

SCH

3

618

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

H(l = O)

SCH

3

619

OCH

3

OCH

3

H

H(l = O)

SCH

3

620

OCH

2

CH

3

OCH

2

CH

3

H

H(l = O)

SCH

3

621

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

H(l = O)

SCH

3

622

SCH

3

SCH

3

H

H(l = O)

SCH

3

623

SCH

2

CH

3

SCH

2

CH

3

H

H(l = O)

SCH

3

624

N(CH

3

)

2

N(CH

3

)

2

H

H(l = O)

SCH

3

625

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

H(l = O)

SCH

3

626

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

H(l = O)

SCH

3

627

O—(CH

2

CH

2

)—O

H

H(l = O)

SCH

3

628

O—(CH

2

CH

2

CH

2

)—O

H

H(l = O)

SCH

3

629

S—(CH

2

CH

2

)—S

H

H(l = O)

SCH

3

630

S—(CH

2

CH

2

CH

2

)—S

H

H(l = O)

SCH

3

631

—(CH

2

)

4

—

H

H(l = O)

SCH

3

632

—(CH

2

)

5

—

H

H(l = O)

SCH

3

633

H

H

NO

2

H(l = O)

SCH

3

634

CH

3

CH

3

NO

2

H(l = O)

SCH

3

635

CH

2

CH

3

CH

2

CH

3

NO

2

H(l = O)

SCH

3

636

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

H(l = O)

SCH

3

637

OCH

3

OCH

3

NO

2

H(l = O)

SCH

3

638

OCH

2

CH

3

OCH

2

CH

3

NO

2

H(l = O)

SCH

3

639

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

H(l = O)

SCH

3

640

SCH

3

SCH

3

NO

2

H(l = O)

SCH

3

641

SCH

2

CH

3

SCH

2

CH

3

NO

2

H(l = O)

SCH

3

642

N(CH

3

)

2

N(CH

3

)

2

NO

2

H(l = O)

SCH

3

643

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

H(l = O)

SCH

3

644

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

H(l = O)

SCH

3

645

O—(CH

2

CH

2

)—O

NO

2

H(l = O)

SCH

3

646

O—(CH

2

CH

2

CH

2

)—O

NO

2

H(l = O)

SCH

3

647

S—(CH

2

CH

2

)—S

NO

2

H(l = O)

SCH

3

648

S—(CH

2

CH

2

CH

2

)—S

NO

2

H(l = O)

SCH

3

649

—(CH

2

)

4

—

NO

2

H(l = O)

SCH

3

650

—(CH

2

)

5

—

NO

2

H(l = O)

SCH

3

651

H

H

CN

H(l = O)

SCH

3

652

CH

3

CH

3

CN

H(l = O)

SCH

3

653

CH

2

CH

3

CH

2

CH

3

CN

H(l = O)

SCH

3

654

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

H(l = O)

SCH

3

655

OCH

3

OCH

3

CN

H(l = O)

SCH

3

656

OCH

2

CH

3

OCH

2

CH

3

CN

H(l = O)

SCH

3

657

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

H(l = O)

SCH

3

658

SCH

3

SCH

3

CN

H(l = O)

SCH

3

659

SCH

2

CH

3

SCH

2

CH

3

CN

H(l = O)

SCH

3

660

N(CH

3

)

2

N(CH

3

)

2

CN

H(l = O)

SCH

3

661

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

H(l = O)

SCH

3

662

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

H(l = O)

SCH

3

663

O—(CH

2

CH

2

)—O

CN

H(l = O)

SCH

3

664

O—(CH

2

CH

2

CH

2

)—O

CN

H(l = O)

SCH

3

665

S—(CH

2

CH

2

)—S

CN

H(l = O)

SCH

3

666

S—(CH

2

CH

2

CH

2

)—S

CN

H(l = O)

SCH

3

667

—(CH

2

)

4

—

CN

H(l = O)

SCH

3

668

—(CH

2

)

5

—

CN

H(l = O)

SCH

3

669

H

H

F

H(l = O)

SCH

3

670

CH

3

CH

3

F

H(l = O)

SCH

3

671

CH

2

CH

3

CH

2

CH

3

F

H(l = O)

SCH

3

672

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

H(l = O)

SCH

3

673

OCH

3

OCH

3

F

H(l = O)

SCH

3

674

OCH

2

CH

3

OCH

2

CH

3

F

H(l = O)

SCH

3

675

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

H(l = O)

SCH

3

676

SCH

3

SCH

3

F

H(l = O)

SCH

3

677

SCH

2

CH

3

SCH

2

CH

3

F

H(l = O)

SCH

3

678

N(CH

3

)

2

N(CH

3

)

2

F

H(l = O)

SCH

3

679

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

H(l = O)

SCH

3

680

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

H(l = O)

SCH

3

681

O—(CH

2

CH

2

)—O

F

H(l = O)

SCH

3

682

O—(CH

2

CH

2

CH

2

)—O

F

H(l = O)

SCH

3

683

S—(CH

2

CH

2

)—S

F

H(l = O)

SCH

3

684

S—(CH

2

CH

2

CH

2

)—S

F

H(l = O)

SCH

3

685

—(CH

2

)

4

—

F

H(l = O)

SCH

3

686

—(CH

2

)

5

—

F

H(l = O)

SCH

3

687

H

H

Cl

H(l = O)

SCH

3

688

CH

3

CH

3

Cl

H(l = O)

SCH

3

689

CH

2

CH

3

CH

2

CH

3

Cl

H(l = O)

SCH

3

690

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

H(l = O)

SCH

3

691

OCH

3

OCH

3

Cl

H(l = O)

SCH

3

692

OCH

2

CH

3

OCH

2

CH

3

Cl

H(l = O)

SCH

3

693

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

H(l = O)

SCH

3

694

SCH

3

SCH

3

Cl

H(l = O)

SCH

3

695

SCH

2

CH

3

SCH

2

CH

3

Cl

H(l = O)

SCH

3

696

N(CH

3

)

2

N(CH

3

)

2

Cl

H(l = O)

SCH

3

697

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

H(l = O)

SCH

3

698

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

H(l = O)

SCH

3

699

O—(CH

2

CH

2

)—O

Cl

H(l = O)

SCH

3

700

O—(CH

2

CH

2

CH

2

)—O

Cl

H(l = O)

SCH

3

701

S—(CH

2

CH

2

)—S

Cl

H(l = O)

SCH

3

702

S—(CH

2

CH

2

CH

2

)—S

Cl

H(l = O)

SCH

3

703

—(CH

2

)

4

—

Cl

H(l = O)

SCH

3

704

—(CH

2

)

5

—

Cl

H(l = O)

SCH

3

705

H

H

Br

H(l = O)

SCH

3

706

CH

3

CH

3

Br

H(l = O)

SCH

3

707

CH

2

CH

3

CH

2

CH

3

Br

H(l = O)

SCH

3

708

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

H(l = O)

SCH

3

709

OCH

3

OCH

3

Br

H(l = O)

SCH

3

710

OCH

2

CH

3

OCH

2

CH

3

Br

H(l = O)

SCH

3

711

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

H(l = O)

SCH

3

712

SCH

3

SCH

3

Br

H(l = O)

SCH

3

713

SCH

2

CH

3

SCH

2

CH

3

Br

H(l = O)

SCH

3

714

N(CH

3

)

2

N(CH

3

)

2

Br

H(l = O)

SCH

3

715

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

H(l = O)

SCH

3

716

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

H(l = O)

SCH

3

717

O—(CH

2

CH

2

)—O

Br

H(l = O)

SCH

3

718

O—(CH

2

CH

2

CH

2

)—O

Br

H(l = O)

SCH

3

719

S—(CH

2

CH

2

)—S

Br

H(l = O)

SCH

3

720

S—(CH

2

CH

2

CH

2

)—S

Br

H(l = O)

SCH

3

721

—(CH

2

)

4

—

Br

H(l = O)

SCH

3

722

—(CH

2

)

5

—

Br

H(l = O)

SCH

3

723

H

H

CH

3

H(l = O)

SCH

3

724

CH

3

CH

3

CH

3

H(l = O)

SCH

3

725

CH

2

CH

3

CH

2

CH

3

CH

3

H(l = O)

SCH

3

726

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

H(l = O)

SCH

3

727

OCH

3

OCH

3

CH

3

H(l = O)

SCH

3

728

OCH

2

CH

3

OCH

2

CH

3

CH

3

H(l = O)

SCH

3

729

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

H(l = O)

SCH

3

730

SCH

3

SCH

3

CH

3

H(l = O)

SCH

3

731

SCH

2

CH

3

SCH

2

CH

3

CH

3

H(l = O)

SCH

3

732

N(CH

3

)

2

N(CH

3

)

2

CH

3

H(l = O)

SCH

3

733

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

H(l = O)

SCH

3

734

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

H(l = O)

SCH

3

735

O—(CH

2

CH

2

)—O

CH

3

H(l = O)

SCH

3

736

O—(CH

2

CH

2

CH

2

)—O

CH

3

H(l = O)

SCH

3

737

S—(CH

2

CH

2

)—S

CH

3

H(l = O)

SCH

3

738

S—(CH

2

CH

2

CH

2

)—S

CH

3

H(l = O)

SCH

3

739

—(CH

2

)

4

—

CH

3

H(l = O)

SCH

3

740

—(CH

2

)

5

—

CH

3

H(l = O)

SCH

3

741

H

H

CH

2

CH

3

H(l = O)

SCH

3

742

CH

3

CH

3

CH

2

CH

3

H(l = O)

SCH

3

743

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

H(l = O)

SCH

3

744

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

SCH

3

745

OCH

3

OCH

3

CH

2

CH

3

H(l = O)

SCH

3

746

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

H(l = O)

SCH

3

747

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

SCH

3

748

SCH

3

SCH

3

CH

2

CH

3

H(l = O)

SCH

3

749

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

H(l = O)

SCH

3

750

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

H(l = O)

SCH

3

751

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

H(l = O)

SCH

3

752

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

H(l = O)

SCH

3

753

O—(CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

SCH

3

754

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

SCH

3

755

S—(CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

SCH

3

756

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

SCH

3

757

—(CH

2

)

4

—

CH

2

CH

3

H(l = O)

SCH

3

758

—(CH

2

)

5

—

CH

2

CH

3

H(l = O)

SCH

3

759

H

H

CF

3

H(l = O)

SCH

3

760

CH

3

CH

3

CF

3

H(l = O)

SCH

3

761

CH

2

CH

3

CH

2

CH

3

CF

3

H(l = O)

SCH

3

762

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

H(l = O)

SCH

3

763

OCH

3

OCH

3

CF

3

H(l = O)

SCH

3

764

OCH

2

CH

3

OCH

2

CH

3

CF

3

H(l = O)

SCH

3

765

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

H(l = O)

SCH

3

766

SCH

3

SCH

3

CF

3

H(l = O)

SCH

3

767

SCH

2

CH

3

SCH

2

CH

3

CF

3

H(l = O)

SCH

3

768

N(CH

3

)

2

N(CH

3

)

2

CF

3

H(l = O)

SCH

3

769

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

H(l = O)

SCH

3

770

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

H(l = O)

SCH

3

771

O—(CH

2

CH

2

)—O

CF

3

H(l = O)

SCH

3

772

O—(CH

2

CH

2

CH

2

)—O

CF

3

H(l = O)

SCH

3

773

S—(CH

2

CH

2

)—S

CF

3

H(l = O)

SCH

3

774

S—(CH

2

CH

2

CH

2

)—S

CF

3

H(l = O)

SCH

3

775

—(CH

2

)

4

—

CF

3

H(l = O)

SCH

3

776

—(CH

2

)

5

—

CF

3

H(l = O)

SCH

3

777

H

H

OCH

3

H(l = O)

SCH

3

778

CH

3

CH

3

OCH

3

H(l = O)

SCH

3

779

CH

2

CH

3

CH

2

CH

3

OCH

3

H(l = O)

SCH

3

780

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

H(l = O)

SCH

3

781

OCH

3

OCH

3

OCH

3

H(l = O)

SCH

3

782

OCH

2

CH

3

OCH

2

CH

3

OCH

3

H(l = O)

SCH

3

783

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

H(l = O)

SCH

3

784

SCH

3

SCH

3

OCH

3

H(l = O)

SCH

3

785

SCH

2

CH

3

SCH

2

CH

3

OCH

3

H(l = O)

SCH

3

786

N(CH

3

)

2

N(CH

3

)

2

OCH

3

H(l = O)

SCH

3

787

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

H(l = O)

SCH

3

788

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

H(l = O)

SCH

3

789

O—(CH

2

CH

2

)—O

OCH

3

H(l = O)

SCH

3

790

O—(CH

2

CH

2

CH

2

)—O

OCH

3

H(l = O)

SCH

3

791

S—(CH

2

CH

2

)—S

OCH

3

H(l = O)

SCH

3

792

S—(CH

2

CH

2

CH

2

)—S

OCH

3

H(l = O)

SCH

3

793

—(CH

2

)

4

—

OCH

3

H(l = O)

SCH

3

794

—(CH

2

)

5

—

OCH

3

H(l = O)

SCH

3

795

H

H

OCH

2

CH

3

H(l = O)

SCH

3

796

CH

3

CH

3

OCH

2

CH

3

H(l = O)

SCH

3

797

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

H(l = O)

SCH

3

798

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

SCH

3

799

OCH

3

OCH

3

OCH

2

CH

3

H(l = O)

SCH

3

800

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

H(l = O)

SCH

3

801

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

SCH

3

802

SCH

3

SCH

3

OCH

2

CH

3

H(l = O)

SCH

3

803

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

H(l = O)

SCH

3

804

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

H(l = O)

SCH

3

805

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

H(l = O)

SCH

3

806

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

H(l = O)

SCH

3

807

O—(CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

SCH

3

808

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

SCH

3

809

S—(CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

SCH

3

810

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

SCH

3

811

—(CH

2

)

4

—

OCH

2

CH

3

H(l = O)

SCH

3

812

—(CH

2

)

5

—

OCH

2

CH

3

H(l = O)

SCH

3

813

H

H

SCH

3

H(l = O)

SCH

3

814

CH

3

CH

3

SCH

3

H(l = O)

SCH

3

815

CH

2

CH

3

CH

2

CH

3

SCH

3

H(l = O)

SCH

3

816

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

H(l = O)

SCH

3

817

OCH

3

OCH

3

SCH

3

H(l = O)

SCH

3

818

OCH

2

CH

3

OCH

2

CH

3

SCH

3

H(l = O)

SCH

3

819

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

H(l = O)

SCH

3

820

SCH

3

SCH

3

SCH

3

H(l = O)

SCH

3

821

SCH

2

CH

3

SCH

2

CH

3

SCH

3

H(l = O)

SCH

3

822

N(CH

3

)

2

N(CH

3

)

2

SCH

3

H(l = O)

SCH

3

823

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

H(l = O)

SCH

3

824

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

H(l = O)

SCH

3

825

O—(CH

2

CH

2

)—O

SCH

3

H(l = O)

SCH

3

826

O—(CH

2

CH

2

CH

2

)—O

SCH

3

H(l = O)

SCH

3

827

S—(CH

2

CH

2

)—S

SCH

3

H(l = O)

SCH

3

828

S—(CH

2

CH

2

CH

2

)—S

SCH

3

H(l = O)

SCH

3

829

—(CH

2

)

4

—

SCH

3

H(l = O)

SCH

3

830

—(CH

2

)

5

—

SCH

3

H(l = O)

SCH

3

831

H

H

SO

2

CH

3

H(l = O)

SCH

3

832

CH

3

CH

3

SO

2

CH

3

H(l = O)

SCH

3

833

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

H(l = O)

SCH

3

834

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

SCH

3

835

OCH

3

OCH

3

SO

2

CH

3

H(l = O)

SCH

3

836

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

H(l = O)

SCH

3

837

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

SCH

3

838

SCH

3

SCH

3

SO

2

CH

3

H(l = O)

SCH

3

839

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

H(l = O)

SCH

3

840

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

H(l = O)

SCH

3

841

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

H(l = O)

SCH

3

842

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

H(l = O)

SCH

3

843

O—(CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

SCH

3

844

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

SCH

3

845

S—(CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

SCH

3

846

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

SCH

3

847

—(CH

2

)

4

—

SO

2

CH

3

H(l = O)

SCH

3

848

—(CH

2

)

5

—

SO

2

CH

3

H(l = O)

SCH

3

849

H

H

PO(OCH

3

)

2

H(l = O)

SCH

3

850

CH

3

CH

3

PO(OCH

3

)

2

H(l = O)

SCH

3

851

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

SCH

3

852

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

SCH

3

853

OCH

3

OCH

3

PO(OCH

3

)

2

H(l = O)

SCH

3

854

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

SCH

3

855

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

SCH

3

856

SCH

3

SCH

3

PO(OCH

3

)

2

H(l = O)

SCH

3

857

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

SCH

3

858

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

H(l = O)

SCH

3

859

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

H(l = O)

SCH

3

860

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

H(l = O)

SCH

3

861

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

SCH

3

862

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

SCH

3

863

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

SCH

3

864

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

SCH

3

865

—(CH

2

)

4

—

PO(OCH

3

)

2

H(l = O)

SCH

3

866

—(CH

2

)

5

—

PO(OCH

3

)

2

H(l = O)

SCH

3

867

H

H

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

868

CH

3

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

869

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

870

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

871

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

872

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

873

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

874

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

875

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

876

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

877

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

878

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

879

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

880

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

881

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

882

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

883

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

884

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

H(l = O)

SCH

3

885

H

H

PO(CH

3

)

2

H(l = O)

SCH

3

886

CH

3

CH

3

PO(CH

3

)

2

H(l = O)

SCH

3

887

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

SCH

3

888

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

SCH

3

889

OCH

3

OCH

3

PO(CH

3

)

2

H(l = O)

SCH

3

890

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

H(l = O)

SCH

3

891

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

SCH

3

892

SCH

3

SCH

3

PO(CH

3

)

2

H(l = O)

SCH

3

893

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

H(l = O)

SCH

3

894

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

H(l = O)

SCH

3

895

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

H(l = O)

SCH

3

896

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

H(l = O)

SCH

3

897

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

SCH

3

898

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

SCH

3

899

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

SCH

3

900

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

SCH

3

901

—(CH

2

)

4

—

PO(CH

3

)

2

H(l = O)

SCH

3

902

—(CH

2

)

5

—

PO(CH

3

)

2

H(l = O)

SCH

3

903

H

H

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

904

CH

3

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

905

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

906

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

907

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

908

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

909

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

910

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

911

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

912

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

913

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

914

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

915

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

916

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

917

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

918

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

919

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

920

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

H(l = O)

SCH

3

921

H

H

H

H(l = O)

SC

6

H

5

922

CH

3

CH

3

H

H(l = O)

SC

6

H

5

923

CH

2

CH

3

CH

2

CH

3

H

H(l = O)

SC

6

H

5

924

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

H(l = O)

SC

6

H

5

925

OCH

3

OCH

3

H

H(l = O)

SC

6

H

5

926

OCH

2

CH

3

OCH

2

CH

3

H

H(l = O)

SC

6

H

5

927

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

H(l = O)

SC

6

H

5

928

SCH

3

SCH

3

H

H(l = O)

SC

6

H

5

929

SCH

2

CH

3

SCH

2

CH

3

H

H(l = O)

SC

6

H

5

930

N(CH

3

)

2

N(CH

3

)

2

H

H(l = O)

SC

6

H

5

931

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

H(l = O)

SC

6

H

5

932

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

H(l = O)

SC

6

H

5

933

O—(CH

2

CH

2

)—O

H

H(l = O)

SC

6

H

5

934

O—(CH

2

CH

2

CH

2

)—O

H

H(l = O)

SC

6

H

5

935

S—(CH

2

CH

2

)—S

H

H(l = O)

SC

6

H

5

936

S—(CH

2

CH

2

CH

2

)—S

H

H(l = O)

SC

6

H

5

937

—(CH

2

)

4

—

H

H(l = O)

SC

6

H

5

938

—(CH

2

)

5

—

H

H(l = O)

SC

6

H

5

939

H

H

NO

2

H(l = O)

SC

6

H

5

940

CH

3

CH

3

NO

2

H(l = O)

SC

6

H

5

941

CH

2

CH

3

CH

2

CH

3

NO

2

H(l = O)

SC

6

H

5

942

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

H(l = O)

SC

6

H

5

943

OCH

3

OCH

3

NO

2

H(l = O)

SC

6

H

5

944

OCH

2

CH

3

OCH

2

CH

3

NO

2

H(l = O)

SC

6

H

5

945

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

H(l = O)

SC

6

H

5

946

SCH

3

SCH

3

NO

2

H(l = O)

SC

6

H

5

947

SCH

2

CH

3

SCH

2

CH

3

NO

2

H(l = O)

SC

6

H

5

948

N(CH

3

)

2

N(CH

3

)

2

NO

2

H(l = O)

SC

6

H

5

949

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

H(l = O)

SC

6

H

5

950

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

H(l = O)

SC

6

H

5

951

O—(CH

2

CH

2

)—O

NO

2

H(l = O)

SC

6

H

5

952

O—(CH

2

CH

2

CH

2

)—O

NO

2

H(l = O)

SC

6

H

5

953

S—(CH

2

CH

2

)—S

NO

2

H(l = O)

SC

6

H

5

954

S—(CH

2

CH

2

CH

2

)—S

NO

2

H(l = O)

SC

6

H

5

955

—(CH

2

)

4

—

NO

2

H(l = O)

SC

6

H

5

956

—(CH

2

)

5

—

NO

2

H(l = O)

SC

6

H

5

957

H

H

CN

H(l = O)

SC

6

H

5

958

CH

3

CH

3

CN

H(l = O)

SC

6

H

5

959

CH

2

CH

3

CH

2

CH

3

CN

H(l = O)

SC

6

H

5

960

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

H(l = O)

SC

6

H

5

961

OCH

3

OCH

3

CN

H(l = O)

SC

6

H

5

962

OCH

2

CH

3

OCH

2

CH

3

CN

H(l = O)

SC

6

H

5

963

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

H(l = O)

SC

6

H

5

964

SCH

3

SCH

3

CN

H(l = O)

SC

6

H

5

965

SCH

2

CH

3

SCH

2

CH

3

CN

H(l = O)

SC

6

H

5

966

N(CH

3

)

2

N(CH

3

)

2

CN

H(l = O)

SC

6

H

5

967

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

H(l = O)

SC

6

H

5

968

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

H(l = O)

SC

6

H

5

969

O—(CH

2

CH

2

)—O

CN

H(l = O)

SC

6

H

5

970

O—(CH

2

CH

2

CH

2

)—O

CN

H(l = O)

SC

6

H

5

971

S—(CH

2

CH

2

)—S

CN

H(l = O)

SC

6

H

5

972

S—(CH

2

CH

2

CH

2

)—S

CN

H(l = O)

SC

6

H

5

973

—(CH

2

)

4

—

CN

H(l = O)

SC

6

H

5

974

—(CH

2

)

5

—

CN

H(l = O)

SC

6

H

5

975

H

H

F

H(l = O)

SC

6

H

5

976

CH

3

CH

3

F

H(l = O)

SC

6

H

5

977

CH

2

CH

3

CH

2

CH

3

F

H(l = O)

SC

6

H

5

978

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

H(l = O)

SC

6

H

5

979

OCH

3

OCH

3

F

H(l = O)

SC

6

H

5

980

OCH

2

CH

3

OCH

2

CH

3

F

H(l = O)

SC

6

H

5

981

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

H(l = O)

SC

6

H

5

982

SCH

3

SCH

3

F

H(l = O)

SC

6

H

5

983

SCH

2

CH

3

SCH

2

CH

3

F

H(l = O)

SC

6

H

5

984

N(CH

3

)

2

N(CH

3

)

2

F

H(l = O)

SC

6

H

5

985

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

H(l = O)

SC

6

H

5

986

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

H(l = O)

SC

6

H

5

987

O—(CH

2

CH

2

)—O

F

H(l = O)

SC

6

H

5

988

O—(CH

2

CH

2

CH

2

)—O

F

H(l = O)

SC

6

H

5

989

S—(CH

2

CH

2

)—S

F

H(l = O)

SC

6

H

5

990

S—(CH

2

CH

2

CH

2

)—S

F

H(l = O)

SC

6

H

5

991

—(CH

2

)

4

—

F

H(l = O)

SC

6

H

5

992

—(CH

2

)

5

—

F

H(l = O)

SC

6

H

5

993

H

H

Cl

H(l = O)

SC

6

H

5

994

CH

3

CH

3

Cl

H(l = O)

SC

6

H

5

995

CH

2

CH

3

CH

2

CH

3

Cl

H(l = O)

SC

6

H

5

996

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

H(l = O)

SC

6

H

5

997

OCH

3

OCH

3

Cl

H(l = O)

SC

6

H

5

998

OCH

2

CH

3

OCH

2

CH

3

Cl

H(l = O)

SC

6

H

5

999

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

H(l = O)

SC

6

H

5

1000

SCH

3

SCH

3

Cl

H(l = O)

SC

6

H

5

1001

SCH

2

CH

3

SCH

2

CH

3

Cl

H(l = O)

SC

6

H

5

1002

N(CH

3

)

2

N(CH

3

)

2

Cl

H(l = O)

SC

6

H

5

1003

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

H(l = O)

SC

6

H

5

1004

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

H(l = O)

SC

6

H

5

1005

O—(CH

2

CH

2

)—O

Cl

H(l = O)

SC

6

H

5

1006

O—(CH

2

CH

2

CH

2

)—O

Cl

H(l = O)

SC

6

H

5

1007

S—(CH

2

CH

2

)—S

Cl

H(l = O)

SC

6

H

5

1008

S—(CH

2

CH

2

CH

2

)—S

Cl

H(l = O)

SC

6

H

5

1009

—(CH

2

)

4

—

Cl

H(l = O)

SC

6

H

5

1010

—(CH

2

)

5

—

Cl

H(l = O)

SC

6

H

5

1011

H

H

Br

H(l = O)

SC

6

H

5

1012

CH

3

CH

3

Br

H(l = O)

SC

6

H

5

1013

CH

2

CH

3

CH

2

CH

3

Br

H(l = O)

SC

6

H

5

1014

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

H(l = O)

SC

6

H

5

1015

OCH

3

OCH

3

Br

H(l = O)

SC

6

H

5

1016

OCH

2

CH

3

OCH

2

CH

3

Br

H(l = O)

SC

6

H

5

1017

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

H(l = O)

SC

6

H

5

1018

SCH

3

SCH

3

Br

H(l = O)

SC

6

H

5

1019

SCH

2

CH

3

SCH

2

CH

3

Br

H(l = O)

SC

6

H

5

1020

N(CH

3

)

2

N(CH

3

)

2

Br

H(l = O)

SC

6

H

5

1021

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

H(l = O)

SC

6

H

5

1022

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

H(l = O)

SC

6

H

5

1023

O—(CH

2

CH

2

)—O

Br

H(l = O)

SC

6

H

5

1024

O—(CH

2

CH

2

CH

2

)—O

Br

H(l = O)

SC

6

H

5

1025

S—(CH

2

CH

2

)—S

Br

H(l = O)

SC

6

H

5

1026

S—(CH

2

CH

2

CH

2

)—S

Br

H(l = O)

SC

6

H

5

1027

—(CH

2

)

4

—

Br

H(l = O)

SC

6

H

5

1028

—(CH

2

)

5

—

Br

H(l = O)

SC

6

H

5

1029

H

H

CH

3

H(l = O)

SC

6

H

5

1030

CH

3

CH

3

CH

3

H(l = O)

SC

6

H

5

1031

CH

2

CH

3

CH

2

CH

3

CH

3

H(l = O)

SC

6

H

5

1032

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

H(l = O)

SC

6

H

5

1033

OCH

3

OCH

3

CH

3

H(l = O)

SC

6

H

5

1034

OCH

2

CH

3

OCH

2

CH

3

CH

3

H(l = O)

SC

6

H

5

1035

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

H(l = O)

SC

6

H

5

1036

SCH

3

SCH

3

CH

3

H(l = O)

SC

6

H

5

1037

SCH

2

CH

3

SCH

2

CH

3

CH

3

H(l = O)

SC

6

H

5

1038

N(CH

3

)

2

N(CH

3

)

2

CH

3

H(l = O)

SC

6

H

5

1039

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

H(l = O)

SC

6

H

5

1040

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

H(l = O)

SC

6

H

5

1041

O—(CH

2

CH

2

)—O

CH

3

H(l = O)

SC

6

H

5

1042

O—(CH

2

CH

2

CH

2

)—O

CH

3

H(l = O)

SC

6

H

5

1043

S—(CH

2

CH

2

)—S

CH

3

H(l = O)

SC

6

H

5

1044

S—(CH

2

CH

2

CH

2

)—S

CH

3

H(l = O)

SC

6

H

5

1045

—(CH

2

)

4

—

CH

3

H(l = O)

SC

6

H

5

1046

—(CH

2

)

5

—

CH

3

H(l = O)

SC

6

H

5

1047

H

H

CH

2

CH

3

H(l = O)

SC

6

H

5

1048

CH

3

CH

3

CH

2

CH

3

H(l = O)

SC

6

H

5

1049

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

H(l = O)

SC

6

H

5

1050

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

SC

6

H

5

1051

OCH

3

OCH

3

CH

2

CH

3

H(l = O)

SC

6

H

5

1052

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

H(l = O)

SC

6

H

5

1053

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

SC

6

H

5

1054

SCH

3

SCH

3

CH

2

CH

3

H(l = O)

SC

6

H

5

1055

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

H(l = O)

SC

6

H

5

1056

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

H(l = O)

SC

6

H

5

1057

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

H(l = O)

SC

6

H

5

1058

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

H(l = O)

SC

6

H

5

1059

O—(CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

SC

6

H

5

1060

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

SC

6

H

5

1061

S—(CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

SC

6

H

5

1062

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

SC

6

H

5

1063

—(CH

2

)

4

—

CH

2

CH

3

H(l = O)

SC

6

H

5

1064

—(CH

2

)

5

—

CH

2

CH

3

H(l = O)

SC

6

H

5

1065

H

H

CF

3

H(l = O)

SC

6

H

5

1066

CH

3

CH

3

CF

3

H(l = O)

SC

6

H

5

1067

CH

2

CH

3

CH

2

CH

3

CF

3

H(l = O)

SC

6

H

5

1068

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

H(l = O)

SC

6

H

5

1069

OCH

3

OCH

3

CF

3

H(l = O)

SC

6

H

5

1070

OCH

2

CH

3

OCH

2

CH

3

CF

3

H(l = O)

SC

6

H

5

1071

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

H(l = O)

SC

6

H

5

1072

SCH

3

SCH

3

CF

3

H(l = O)

SC

6

H

5

1073

SCH

2

CH

3

SCH

2

CH

3

CF

3

H(l = O)

SC

6

H

5

1074

N(CH

3

)

2

N(CH

3

)

2

CF

3

H(l = O)

SC

6

H

5

1075

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

H(l = O)

SC

6

H

5

1076

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

H(l = O)

SC

6

H

5

1077

O—(CH

2

CH

2

)—O

CF

3

H(l = O)

SC

6

H

5

1078

O—(CH

2

CH

2

CH

2

)—O

CF

3

H(l = O)

SC

6

H

5

1079

S—(CH

2

CH

2

)—S

CF

3

H(l = O)

SC

6

H

5

1080

S—(CH

2

CH

2

CH

2

)—S

CF

3

H(l = O)

SC

6

H

5

1081

—(CH

2

)

4

—

CF

3

H(l = O)

SC

6

H

5

1082

—(CH

2

)

5

—

CF

3

H(l = O)

SC

6

H

5

1083

H

H

OCH

3

H(l = O)

SC

6

H

5

1084

CH

3

CH

3

OCH

3

H(l = O)

SC

6

H

5

1085

CH

2

CH

3

CH

2

CH

3

OCH

3

H(l = O)

SC

6

H

5

1086

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

H(l = O)

SC

6

H

5

1087

OCH

3

OCH

3

OCH

3

H(l = O)

SC

6

H

5

1088

OCH

2

CH

3

OCH

2

CH

3

OCH

3

H(l = O)

SC

6

H

5

1089

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

H(l = O)

SC

6

H

5

1090

SCH

3

SCH

3

OCH

3

H(l = O)

SC

6

H

5

1091

SCH

2

CH

3

SCH

2

CH

3

OCH

3

H(l = O)

SC

6

H

5

1092

N(CH

3

)

2

N(CH

3

)

2

OCH

3

H(l = O)

SC

6

H

5

1093

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

H(l = O)

SC

6

H

5

1094

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

H(l = O)

SC

6

H

5

1095

O—(CH

2

CH

2

)—O

OCH

3

H(l = O)

SC

6

H

5

1096

O—(CH

2

CH

2

CH

2

)—O

OCH

3

H(l = O)

SC

6

H

5

1097

S—(CH

2

CH

2

)—S

OCH

3

H(l = O)

SC

6

H

5

1098

S—(CH

2

CH

2

CH

2

)—S

OCH

3

H(l = O)

SC

6

H

5

1099

—(CH

2

)

4

—

OCH

3

H(l = O)

SC

6

H

5

1100

—(CH

2

)

5

—

OCH

3

H(l = O)

SC

6

H

5

1101

H

H

OCH

2

CH

3

H(l = O)

SC

6

H

5

1102

CH

3

CH

3

OCH

2

CH

3

H(l = O)

SC

6

H

5

1103

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

H(l = O)

SC

6

H

5

1104

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

SC

6

H

5

1105

OCH

3

OCH

3

OCH

2

CH

3

H(l = O)

SC

6

H

5

1106

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

H(l = O)

SC

6

H

5

1107

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

SC

6

H

5

1108

SCH

3

SCH

3

OCH

2

CH

3

H(l = O)

SC

6

H

5

1109

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

H(l = O)

SC

6

H

5

1110

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

H(l = O)

SC

6

H

5

1111

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

H(l = O)

SC

6

H

5

1112

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

H(l = O)

SC

6

H

5

1113

O—(CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

SC

6

H

5

1114

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

SC

6

H

5

1115

S—(CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

SC

6

H

5

1116

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

SC

6

H

5

1117

—(CH

2

)

4

—

OCH

2

CH

3

H(l = O)

SC

6

H

5

1118

—(CH

2

)

5

—

OCH

2

CH

3

H(l = O)

SC

6

H

5

1119

H

H

SCH

3

H(l = O)

SC

6

H

5

1120

CH

3

CH

3

SCH

3

H(l = O)

SC

6

H

5

1121

CH

2

CH

3

CH

2

CH

3

SCH

3

H(l = O)

SC

6

H

5

1122

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

H(l = O)

SC

6

H

5

1123

OCH

3

OCH

3

SCH

3

H(l = O)

SC

6

H

5

1124

OCH

2

CH

3

OCH

2

CH

3

SCH

3

H(l = O)

SC

6

H

5

1125

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

H(l = O)

SC

6

H

5

1126

SCH

3

SCH

3

SCH

3

H(l = O)

SC

6

H

5

1127

SCH

2

CH

3

SCH

2

CH

3

SCH

3

H(l = O)

SC

6

H

5

1128

N(CH

3

)

2

N(CH

3

)

2

SCH

3

H(l = O)

SC

6

H

5

1129

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

H(l = O)

SC

6

H

5

1130

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

H(l = O)

SC

6

H

5

1131

O—(CH

2

CH

2

)—O

SCH

3

H(l = O)

SC

6

H

5

1132

O—(CH

2

CH

2

CH

2

)—O

SCH

3

H(l = O)

SC

6

H

5

1133

S—(CH

2

CH

2

)—S

SCH

3

H(l = O)

SC

6

H

5

1134

S—(CH

2

CH

2

CH

2

)—S

SCH

3

H(l = O)

SC

6

H

5

1135

—(CH

2

)

4

—

SCH

3

H(l = O)

SC

6

H

5

1136

—(CH

2

)

5

—

SCH

3

H(l = O)

SC

6

H

5

1137

H

H

SO

2

CH

3

H(l = O)

SC

6

H

5

1138

CH

3

CH

3

SO

2

CH

3

H(l = O)

SC

6

H

5

1139

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

H(l = O)

SC

6

H

5

1140

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

SC

6

H

5

1141

OCH

3

OCH

3

SO

2

CH

3

H(l = O)

SC

6

H

5

1142

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

H(l = O)

SC

6

H

5

1143

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

SC

6

H

5

1144

SCH

3

SCH

3

SO

2

CH

3

H(l = O)

SC

6

H

5

1145

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

H(l = O)

SC

6

H

5

1146

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

H(l = O)

SC

6

H

5

1147

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

H(l = O)

SC

6

H

5

1148

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

H(l = O)

SC

6

H

5

1149

O—(CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

SC

6

H

5

1150

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

SC

6

H

5

1151

S—(CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

SC

6

H

5

1152

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

SC

6

H

5

1153

—(CH

2

)

4

—

SO

2

CH

3

H(l = O)

SC

6

H

5

1154

—(CH

2

)

5

—

SO

2

CH

3

H(l = O)

SC

6

H

5

1155

H

H

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1156

CH

3

CH

3

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1157

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1158

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1159

OCH

3

OCH

3

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1160

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1161

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1162

SCH

3

SCH

3

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1163

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1164

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1165

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1166

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1167

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1168

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1169

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1170

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1171

—(CH

2

)

4

—

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1172

—(CH

2

)

5

—

PO(OCH

3

)

2

H(l = O)

SC

6

H

5

1173

H

H

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1174

CH

3

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1175

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1176

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1177

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1178

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1179

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1180

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1181

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1182

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1183

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1184

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1185

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1186

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1187

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1188

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1189

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1190

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1191

H

H

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1192

CH

3

CH

3

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1193

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1194

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1195

OCH

3

OCH

3

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1196

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1197

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1198

SCH

3

SCH

3

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1199

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1200

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1201

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1202

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1203

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1204

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1205

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1206

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1207

—(CH

2

)

4

—

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1208

—(CH

2

)

5

—

PO(CH

3

)

2

H(l = O)

SC

6

H

5

1209

H

H

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1210

CH

3

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1211

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1212

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1213

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1214

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1215

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1216

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1217

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1218

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1219

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1220

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1221

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1222

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1223

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1224

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1225

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1226

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

H(l = O)

SC

6

H

5

1227

H

H

H

H(l = O)

Het1

1228

CH

3

CH

3

H

H(l = O)

Het1

1229

CH

2

CH

3

CH

2

CH

3

H

H(l = O)

Het1

1230

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

H(l = O)

Het1

1231

OCH

3

OCH

3

H

H(l = O)

Het1

1232

OCH

2

CH

3

OCH

2

CH

3

H

H(l = O)

Het1

1233

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

H(l = O)

Het1

1234

SCH

3

SCH

3

H

H(l = O)

Het1

1235

SCH

2

CH

3

SCH

2

CH

3

H

H(l = O)

Het1

1236

N(CH

3

)

2

N(CH

3

)

2

H

H(l = O)

Het1

1237

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

H(l = O)

Het1

1238

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

H(l = O)

Het1

1239

O—(CH

2

CH

2

)—O

H

H(l = O)

Het1

1240

O—(CH

2

CH

2

CH

2

)—O

H

H(l = O)

Het1

1241

S—(CH

2

CH

2

)—S

H

H(l = O)

Het1

1242

S—(CH

2

CH

2

CH

2

)—S

H

H(l = O)

Het1

1243

—(CH

2

)

4

—

H

H(l = O)

Het1

1244

—(CH

2

)

5

—

H

H(l = O)

Het1

1245

H

H

NO

2

H(l = O)

Het1

1246

CH

3

CH

3

NO

2

H(l = O)

Het1

1247

CH

2

CH

3

CH

2

CH

3

NO

2

H(l = O)

Het1

1248

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

H(l = O)

Het1

1249

OCH

3

OCH

3

NO

2

H(l = O)

Het1

1250

OCH

2

CH

3

OCH

2

CH

3

NO

2

H(l = O)

Het1

1251

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

H(l = O)

Het1

1252

SCH

3

SCH

3

NO

2

H(l = O)

Het1

1253

SCH

2

CH

3

SCH

2

CH

3

NO

2

H(l = O)

Het1

1254

N(CH

3

)

2

N(CH

3

)

2

NO

2

H(l = O)

Het1

1255

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

H(l = O)

Het1

1256

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

H(l = O)

Het1

1257

O—(CH

2

CH

2

)—O

NO

2

H(l = O)

Het1

1258

O—(CH

2

CH

2

CH

2

)—O

NO

2

H(l = O)

Het1

1259

S—(CH

2

CH

2

)—S

NO

2

H(l = O)

Het1

1260

S—(CH

2

CH

2

CH

2

)—S

NO

2

H(l = O)

Het1

1261

—(CH

2

)

4

—

NO

2

H(l = O)

Het1

1262

—(CH

2

)

5

—

NO

2

H(l = O)

Het1

1263

H

H

CN

H(l = O)

Het1

1264

CH

3

CH

3

CN

H(l = O)

Het1

1265

CH

2

CH

3

CH

2

CH

3

CN

H(l = O)

Het1

1266

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

H(l = O)

Het1

1267

OCH

3

OCH

3

CN

H(l = O)

Het1

1268

OCH

2

CH

3

OCH

2

CH

3

CN

H(l = O)

Het1

1269

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

H(l = O)

Het1

1270

SCH

3

SCH

3

CN

H(l = O)

Het1

1271

SCH

2

CH

3

SCH

2

CH

3

CN

H(l = O)

Het1

1272

N(CH

3

)

2

N(CH

3

)

2

CN

H(l = O)

Het1

1273

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

H(l = O)

Het1

1274

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

H(l = O)

Het1

1275

O—(CH

2

CH

2

)—O

CN

H(l = O)

Het1

1276

O—(CH

2

CH

2

CH

2

)—O

CN

H(l = O)

Het1

1277

S—(CH

2

CH

2

)—S

CN

H(l = O)

Het1

1278

S—(CH

2

CH

2

CH

2

)—S

CN

H(l = O)

Het1

1279

—(CH

2

)

4

—

CN

H(l = O)

Het1

1280

—(CH

2

)

5

—

CN

H(l = O)

Het1

1281

H

H

F

H(l = O)

Het1

1282

CH

3

CH

3

F

H(l = O)

Het1

1283

CH

2

CH

3

CH

2

CH

3

F

H(l = O)

Het1

1284

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

H(l = O)

Het1

1285

OCH

3

OCH

3

F

H(l = O)

Het1

1286

OCH

2

CH

3

OCH

2

CH

3

F

H(l = O)

Het1

1287

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

H(l = O)

Het1

1288

SCH

3

SCH

3

F

H(l = O)

Het1

1289

SCH

2

CH

3

SCH

2

CH

3

F

H(l = O)

Het1

1290

N(CH

3

)

2

N(CH

3

)

2

F

H(l = O)

Het1

1291

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

H(l = O)

Het1

1292

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

H(l = O)

Het1

1293

O—(CH

2

CH

2

)—O

F

H(l = O)

Het1

1294

O—(CH

2

CH

2

CH

2

)—O

F

H(l = O)

Het1

1295

S—(CH

2

CH

2

)—S

F

H(l = O)

Het1

1296

S—(CH

2

CH

2

CH

2

)—S

F

H(l = O)

Het1

1297

—(CH

2

)

4

—

F

H(l = O)

Het1

1298

—(CH

2

)

5

—

F

H(l = O)

Het1

1299

H

H

Cl

H(l = O)

Het1

1300

CH

3

CH

3

Cl

H(l = O)

Het1

1301

CH

2

CH

3

CH

2

CH

3

Cl

H(l = O)

Het1

1302

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

H(l = O)

Het1

1303

OCH

3

OCH

3

Cl

H(l = O)

Het1

1304

OCH

2

CH

3

OCH

2

CH

3

Cl

H(l = O)

Het1

1305

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

H(l = O)

Het1

1306

SCH

3

SCH

3

Cl

H(l = O)

Het1

1307

SCH

2

CH

3

SCH

2

CH

3

Cl

H(l = O)

Het1

1308

N(CH

3

)

2

N(CH

3

)

2

Cl

H(l = O)

Het1

1309

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

H(l = O)

Het1

1310

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

H(l = O)

Het1

1311

O—(CH

2

CH

2

)—O

Cl

H(l = O)

Het1

1312

O—(CH

2

CH

2

CH

2

)—O

Cl

H(l = O)

Het1

1313

S—(CH

2

CH

2

)—S

Cl

H(l = O)

Het1

1314

S—(CH

2

CH

2

CH

2

)—S

H(l = O)

Het1

1315

—(CH

2

)

4

—

Cl

H(l = O)

Het1

1316

—(CH

2

)

5

—

Cl

H(l = O)

Het1

1317

H

H

Br

H(l = O)

Het1

1318

CH

3

CH

3

Br

H(l = O)

Het1

1319

CH

2

CH

3

CH

2

CH

3

Br

H(l = O)

Het1

1320

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

H(l = O)

Het1

1321

OCH

3

OCH

3

Br

H(l = O)

Het1

1322

OCH

2

CH

3

OCH

2

CH

3

Br

H(l = O)

Het1

1323

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

H(l = O)

Het1

1324

SCH

3

SCH

3

Br

H(l = O)

Het1

1325

SCH

2

CH

3

SCH

2

CH

3

Br

H(l = O)

Het1

1326

N(CH

3

)

2

N(CH

3

)

2

Br

H(l = O)

Het1

1327

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

H(l = O)

Het1

1328

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

H(l = O)

Het1

1329

O—(CH

2

CH

2

)—O

Br

H(l = O)

Het1

1330

O—(CH

2

CH

2

CH

2

)—O

Br

H(l = O)

Het1

1331

S—(CH

2

CH

2

)—S

Br

H(l = O)

Het1

1332

S—(CH

2

CH

2

CH

2

)—S

Br

H(l = O)

Het1

1333

—(CH

2

)

4

—

Br

H(l = O)

Het1

1334

—(CH

2

)

5

—

Br

H(l = O)

Het1

1335

H

H

CH

3

H(l = O)

Het1

1336

CH

3

CH

3

CH

3

H(l = O)

Het1

1337

CH

2

CH

3

CH

2

CH

3

CH

3

H(l = O)

Het1

1338

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

H(l = O)

Het1

1339

OCH

3

OCH

3

CH

3

H(l = O)

Het1

1340

OCH

2

CH

3

OCH

2

CH

3

CH

3

H(l = O)

Het1

1341

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

H(l = O)

Het1

1342

SCH

3

SCH

3

CH

3

H(l = O)

Het1

1343

SCH

2

CH

3

SCH

2

CH

3

CH

3

H(l = O)

Het1

1344

N(CH

3

)

2

N(CH

3

)

2

CH

3

H(l = O)

Het1

1345

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

H(l = O)

Het1

1346

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

H(l = O)

Het1

1347

O—(CH

2

CH

2

)—O

CH

3

H(l = O)

Het1

1348

O—(CH

2

CH

2

CH

2

)—O

CH

3

H(l = O)

Het1

1349

S—(CH

2

CH

2

)—S

CH

3

H(l = O)

Het1

1350

S—(CH

2

CH

2

CH

2

)—S

CH

3

H(l = O)

Het1

1351

—(CH

2

)

4

—

CH

3

H(l = O)

Het1

1352

—(CH

2

)

5

—

CH

3

H(l = O)

Het1

1353

H

H

CH

2

CH

3

H(l = O)

Het1

1354

CH

3

CH

3

CH

2

CH

3

H(l = O)

Het1

1355

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

H(l = O)

Het1

1356

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

Het1

1357

OCH

3

OCH

3

CH

2

CH

3

H(l = O)

Het1

1358

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

H(l = O)

Het1

1359

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

Het1

1360

SCH

3

SCH

3

CH

2

CH

3

H(l = O)

Het1

1361

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

H(l = O)

Het1

1362

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

H(l = O)

Het1

1363

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

H(l = O)

Het1

1364

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

H(l = O)

Het1

1365

O—(CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

Het1

1366

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

Het1

1367

S—(CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

Het1

1368

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

Het1

1369

—(CH

2

)

4

—

CH

2

CH

3

H(l = O)

Het1

1370

—(CH

2

)

5

—

CH

2

CH

3

H(l = O)

Het1

1371

H

H

CF

3

H(l = O)

Het1

1372

CH

3

CH

3

CF

3

H(l = O)

Het1

1373

CH

2

CH

3

CH

2

CH

3

CF

3

H(l = O)

Het1

1374

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

H(l = O)

Het1

1375

OCH

3

OCH

3

CF

3

H(l = O)

Het1

1376

OCH

2

CH

3

OCH

2

CH

3

CF

3

H(l = O)

Het1

1377

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

H(l = O)

Het1

1378

SCH

3

SCH

3

CF

3

H(l = O)

Het1

1379

SCH

2

CH

3

SCH

2

CH

3

CF

3

H(l = O)

Het1

1380

N(CH

3

)

2

N(CH

3

)

2

CF

3

H(l = O)

Het1

1381

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

H(l = O)

Het1

1382

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

H(l = O)

Het1

1383

O—(CH

2

CH

2

)—O

CF

3

H(l = O)

Het1

1384

O—(CH

2

CH

2

CH

2

)—O

CF

3

H(l = O)

Het1

1385

S—(CH

2

CH

2

)—S

CF

3

H(l = O)

Het1

1386

S—(CH

2

CH

2

CH

2

)—S

CF

3

H(l = O)

Het1

1387

—(CH

2

)

4

—

CF

3

H(l = O)

Het1

1388

—(CH

2

)

5

—

CF

3

H(l = O)

Het1

1389

H

H

OCH

3

H(l = O)

Het1

1390

CH

3

CH

3

OCH

3

H(l = O)

Het1

1391

CH

2

CH

3

CH

2

CH

3

OCH

3

H(l = O)

Het1

1392

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

H(l = O)

Het1

1393

OCH

3

OCH

3

OCH

3

H(l = O)

Het1

1394

OCH

2

CH

3

OCH

2

CH

3

OCH

3

H(l = O)

Het1

1395

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

H(l = O)

Het1

1396

SCH

3

SCH

3

OCH

3

H(l = O)

Het1

1397

SCH

2

CH

3

SCH

2

CH

3

OCH

3

H(l = O)

Het1

1398

N(CH

3

)

2

N(CH

3

)

2

OCH

3

H(l = O)

Het1

1399

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

H(l = O)

Het1

1400

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

H(l = O)

Het1

1401

O—(CH

2

CH

2

)—O

OCH

3

H(l = O)

Het1

1402

O—(CH

2

CH

2

CH

2

)—O

OCH

3

H(l = O)

Het1

1403

S—(CH

2

CH

2

)—S

OCH

3

H(l = O)

Het1

1404

S—(CH

2

CH

2

CH

2

)—S

OCH

3

H(l = O)

Het1

1405

—(CH

2

)

4

—

OCH

3

H(l = O)

Het1

1406

—(CH

2

)

5

—

OCH

3

H(l = O)

Het1

1407

H

H

OCH

2

CH

3

H(l = O)

Het1

1408

CH

3

CH

3

OCH

2

CH

3

H(l = O)

Het1

1409

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

H(l = O)

Het1

1410

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

Het1

1411

OCH

3

OCH

3

OCH

2

CH

3

H(l = O)

Het1

1412

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

H(l = O)

Het1

1413

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

Het1

1414

SCH

3

SCH

3

OCH

2

CH

3

H(l = O)

Het1

1415

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

H(l = O)

Het1

1416

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

H(l = O)

Het1

1417

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

H(l = O)

Het1

1418

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

H(l = O)

Het1

1419

O—(CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

Het1

1420

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

Het1

1421

S—(CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

Het1

1422

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

Het1

1423

—(CH

2

)

4

—

OCH

2

CH

3

H(l = O)

Het1

1424

—(CH

2

)

5

—

OCH

2

CH

3

H(l = O)

Het1

1425

H

H

SCH

3

H(l = O)

Het1

1426

CH

3

CH

3

SCH

3

H(l = O)

Het1

1427

CH

2

CH

3

CH

2

CH

3

SCH

3

H(l = O)

Het1

1428

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

H(l = O)

Het1

1429

OCH

3

OCH

3

SCH

3

H(l = O)

Het1

1430

OCH

2

CH

3

OCH

2

CH

3

SCH

3

H(l = O)

Het1

1431

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

H(l = O)

Het1

1432

SCH

3

SCH

3

SCH

3

H(l = O)

Het1

1433

SCH

2

CH

3

SCH

2

CH

3

SCH

3

H(l = O)

Het1

1434

N(CH

3

)

2

N(CH

3

)

2

SCH

3

H(l = O)

Het1

1435

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

H(l = O)

Het1

1436

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

H(l = O)

Het1

1437

O—(CH

2

CH

2

)—O

SCH

3

H(l = O)

Het1

1438

O—(CH

2

CH

2

CH

2

)—O

SCH

3

H(l = O)

Het1

1439

S—(CH

2

CH

2

)—S

SCH

3

H(l = O)

Het1

1440

S—(CH

2

CH

2

CH

2

)—S

H(l = O)

Het1

1441

—(CH

2

)

4

—

SCH

3

H(l = O)

Het1

1442

—(CH

2

)

5

—

SCH

3

H(l = O)

Het1

1443

H

H

SO

2

CH

3

H(l = O)

Het1

1444

CH

3

CH

3

SO

2

CH

3

H(l = O)

Het1

1445

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

H(l = O)

Het1

1446

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

Het1

1447

OCH

3

OCH

3

SO

2

CH

3

H(l = O)

Het1

1448

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

H(l = O)

Het1

1449

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

Het1

1450

SCH

3

SCH

3

SO

2

CH

3

H(l = O)

Het1

1451

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

H(l = O)

Het1

1452

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

H(l = O)

Het1

1453

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

H(l = O)

Het1

1454

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

H(l = O)

Het1

1455

O—(CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

Het1

1456

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

Het1

1457

S—(CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

Het1

1458

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

Het1

1459

—(CH

2

)

4

—

SO

2

CH

3

H(l = O)

Het1

1460

—(CH

2

)

5

—

SO

2

CH

3

H(l = O)

Het1

1461

H

H

PO(OCH

3

)

2

H(l = O)

Het1

1462

CH

3

CH

3

PO(OCH

3

)

2

H(l = O)

Het1

1463

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het1

1464

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het1

1465

OCH

3

OCH

3

PO(OCH

3

)

2

H(l = O)

Het1

1466

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het1

1467

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het1

1468

SCH

3

SCH

3

PO(OCH

3

)

2

H(l = O)

Het1

1469

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het1

1470

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

H(l = O)

Het1

1471

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

H(l = O)

Het1

1472

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

H(l = O)

Het1

1473

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

Het1

1474

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

Het1

1475

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

Het1

1476

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

Het1

1477

—(CH

2

)

4

—

PO(OCH

3

)

2

H(l = O)

Het1

1478

—(CH

2

)

5

—

PO(OCH

3

)

2

H(l = O)

Het1

1479

H

H

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1480

CH

3

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1481

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1482

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1483

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1484

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1485

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1486

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1487

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1488

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1489

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1490

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1491

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1492

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1493

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1494

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1495

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1496

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

H(l = O)

Het1

1497

H

H

PO(CH

3

)

2

H(l = O)

Het1

1498

CH

3

CH

3

PO(CH

3

)

2

H(l = O)

Het1

1499

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het1

1500

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het1

1501

OCH

3

OCH

3

PO(CH

3

)

2

H(l = O)

Het1

1502

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het1

1503

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het1

1504

SCH

3

SCH

3

PO(CH

3

)

2

H(l = O)

Het1

1505

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het1

1506

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

H(l = O)

Het1

1507

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

H(l = O)

Het1

1508

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

H(l = O)

Het1

1509

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

Het1

1510

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

Het1

1511

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

Het1

1512

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

Het1

1513

—(CH

2

)

4

—

PO(CH

3

)

2

H(l = O)

Het1

1514

—(CH

2

)

5

—

PO(CH

3

)

2

H(l = O)

Het1

1515

H

H

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1516

CH

3

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1517

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1518

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1519

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1520

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1521

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1522

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1523

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1524

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1525

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1526

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1527

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1528

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1529

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1530

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1531

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1532

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

H(l = O)

Het1

1533

H

H

H

H(l = O)

Het2

1534

CH

3

CH

3

H

H(l = O)

Het2

1535

CH

2

CH

3

CH

2

CH

3

H

H(l = O)

Het2

1536

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

H(l = O)

Het2

1537

OCH

3

OCH

3

H

H(l = O)

Het2

1538

OCH

2

CH

3

OCH

2

CH

3

H

H(l = O)

Het2

1539

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

H(l = O)

Het2

1540

SCH

3

SCH

3

H

H(l = O)

Het2

1541

SCH

2

CH

3

SCH

2

CH

3

H

H(l = O)

Het2

1542

N(CH

3

)

2

N(CH

3

)

2

H

H(l = O)

Het2

1543

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

H(l = O)

Het2

1544

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

H(l = O)

Het2

1545

O—(CH

2

CH

2

)—O

H

H(l = O)

Het2

1546

O—(CH

2

CH

2

CH

2

)—O

H

H(l = O)

Het2

1547

S—(CH

2

CH

2

)—S

H

H(l = O)

Het2

1548

S—(CH

2

CH

2

CH

2

)—S

H

H(l = O)

Het2

1549

—(CH

2

)

4

—

H

H(l = O)

Het2

1550

—(CH

2

)

5

—

H

H(l = O)

Het2

1551

H

H

NO

2

H(l = O)

Het2

1552

CH

3

CH

3

NO

2

H(l = O)

Het2

1553

CH

2

CH

3

CH

2

CH

3

NO

2

H(l = O)

Het2

1554

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

H(l = O)

Het2

1555

OCH

3

OCH

3

NO

2

H(l = O)

Het2

1556

OCH

2

CH

3

OCH

2

CH

3

NO

2

H(l = O)

Het2

1557

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

H(l = O)

Het2

1558

SCH

3

SCH

3

NO

2

H(l = O)

Het2

1559

SCH

2

CH

3

SCH

2

CH

3

NO

2

H(l = O)

Het2

1560

N(CH

3

)

2

N(CH

3

)

2

NO

2

H(l = O)

Het2

1561

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

H(l = O)

Het2

1562

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

H(l = O)

Het2

1563

O—(CH

2

CH

2

)—O

NO

2

H(l = O)

Het2

1564

O—(CH

2

CH

2

CH

2

)—O

NO

2

H(l = O)

Het2

1565

S—(CH

2

CH

2

)—S

NO

2

H(l = O)

Het2

1566

S—(CH

2

CH

2

CH

2

)—S

NO

2

H(l = O)

Het2

1567

—(CH

2

)

4

—

NO

2

H(l = O)

Het2

1568

—(CH

2

)

5

—

NO

2

H(l = O)

Het2

1569

H

H

CN

H(l = O)

Het2

1570

CH

3

CH

3

CN

H(l = O)

Het2

1571

CH

2

CH

3

CH

2

CH

3

CN

H(l = O)

Het2

1572

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

H(l = O)

Het2

1573

OCH

3

OCH

3

CN

H(l = O)

Het2

1574

OCH

2

CH

3

OCH

2

CH

3

CN

H(l = O)

Het2

1575

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

H(l = O)

Het2

1576

SCH

3

SCH

3

CN

H(l = O)

Het2

1577

SCH

2

CH

3

SCH

2

CH

3

CN

H(l = O)

Het2

1578

N(CH

3

)

2

N(CH

3

)

2

CN

H(l = O)

Het2

1579

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

H(l = O)

Het2

1580

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

H(l = O)

Het2

1581

O—(CH

2

CH

2

)—O

CN

H(l = O)

Het2

1582

O—(CH

2

CH

2

CH

2

)—O

CN

H(l = O)

Het2

1583

S—(CH

2

CH

2

)—S

CN

H(l = O)

Het2

1584

S—(CH

2

CH

2

CH

2

)—S

CN

H(l = O)

Het2

1585

—(CH

2

)

4

—

CN

H(l = O)

Het2

1586

—(CH

2

)

5

—

CN

H(l = O)

Het2

1587

H

H

F

H(l = O)

Het2

1588

CH

3

CH

3

F

H(l = O)

Het2

1589

CH

2

CH

3

CH

2

CH

3

F

H(l = O)

Het2

1590

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

H(l = O)

Het2

1591

OCH

3

OCH

3

F

H(l = O)

Het2

1592

OCH

2

CH

3

OCH

2

CH

3

F

H(l = O)

Het2

1593

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

H(l = O)

Het2

1594

SCH

3

SCH

3

F

H(l = O)

Het2

1595

SCH

2

CH

3

SCH

2

CH

3

F

H(l = O)

Het2

1596

N(CH

3

)

2

N(CH

3

)

2

F

H(l = O)

Het2

1597

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

H(l = O)

Het2

1598

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

H(l = O)

Het2

1599

O—(CH

2

CH

2

)—O

F

H(l = O)

Het2

1600

O—(CH

2

CH

2

CH

2

)—O

F

H(l = O)

Het2

1601

S—(CH

2

CH

2

)—S

F

H(l = O)

Het2

1602

S—(CH

2

CH

2

CH

2

)—S

F

H(l = O)

Het2

1603

—(CH

2

)

4

—

F

H(l = O)

Het2

1604

—(CH

2

)

5

—

F

H(l = O)

Het2

1605

H

H

Cl

H(l = O)

Het2

1606

CH

3

CH

3

Cl

H(l = O)

Het2

1607

CH

2

CH

3

CH

2

CH

3

Cl

H(l = O)

Het2

1608

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

H(l = O)

Het2

1609

OCH

3

OCH

3

Cl

H(l = O)

Het2

1610

OCH

2

CH

3

OCH

2

CH

3

Cl

H(l = O)

Het2

1611

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

H(l = O)

Het2

1612

SCH

3

SCH

3

Cl

H(l = O)

Het2

1613

SCH

2

CH

3

SCH

2

CH

3

Cl

H(l = O)

Het2

1614

N(CH

3

)

2

N(CH

3

)

2

Cl

H(l = O)

Het2

1615

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

H(l = O)

Het2

1616

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

H(l = O)

Het2

1617

O—(CH

2

CH

2

)—O

Cl

H(l = O)

Het2

1618

O—(CH

2

CH

2

CH

2

)—O

Cl

H(l = O)

Het2

1619

S—(CH

2

CH

2

)—S

Cl

H(l = O)

Het2

1620

S—(CH

2

CH

2

CH

2

)—S

Cl

H(l = O)

Het2

1621

—(CH

2

)

4

—

Cl

H(l = O)

Het2

1622

—(CH

2

)

5

—

Cl

H(l = O)

Het2

1623

H

H

Br

H(l = O)

Het2

1624

CH

3

CH

3

Br

H(l = O)

Het2

1625

CH

2

CH

3

CH

2

CH

3

Br

H(l = O)

Het2

1626

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

H(l = O)

Het2

1627

OCH

3

OCH

3

Br

H(l = O)

Het2

1628

OCH

2

CH

3

OCH

2

CH

3

Br

H(l = O)

Het2

1629

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

H(l = O)

Het2

1630

SCH

3

SCH

3

Br

H(l = O)

Het2

1631

SCH

2

CH

3

SCH

2

CH

3

Br

H(l = O)

Het2

1632

N(CH

3

)

2

N(CH

3

)

2

Br

H(l = O)

Het2

1633

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

H(l = O)

Het2

1634

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

H(l = O)

Het2

1635

O—(CH

2

CH

2

)—O

Br

H(l = O)

Het2

1636

O—(CH

2

CH

2

CH

2

)—O

Br

H(l = O)

Het2

1637

S—(CH

2

CH

2

)—S

Br

H(l = O)

Het2

1638

S—(CH

2

CH

2

CH

2

)—S

Br

H(l = O)

Het2

1639

—(CH

2

)

4

—

Br

H(l = O)

Het2

1640

—(CH

2

)

5

—

Br

H(l = O)

Het2

1641

H

H

CH

3

H(l = O)

Het2

1642

CH

3

CH

3

CH

3

H(l = O)

Het2

1643

CH

2

CH

3

CH

2

CH

3

CH

3

H(l = O)

Het2

1644

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

H(l = O)

Het2

1645

OCH

3

OCH

3

CH

3

H(l = O)

Het2

1646

OCH

2

CH

3

OCH

2

CH

3

CH

3

H(l = O)

Het2

1647

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

H(l = O)

Het2

1648

SCH

3

SCH

3

CH

3

H(l = O)

Het2

1649

SCH

2

CH

3

SCH

2

CH

3

CH

3

H(l = O)

Het2

1650

N(CH

3

)

2

N(CH

3

)

2

CH

3

H(l = O)

Het2

1651

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

H(l = O)

Het2

1652

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

H(l = O)

Het2

1653

O—(CH

2

CH

2

)—O

CH

3

H(l = O)

Het2

1654

O—(CH

2

CH

2

CH

2

)—O

CH

3

H(l = O)

Het2

1655

S—(CH

2

CH

2

)—S

CH

3

H(l = O)

Het2

1656

S—(CH

2

CH

2

CH

2

)—S

CH

3

H(l = O)

Het2

1657

—(CH

2

)

4

—

CH

3

H(l = O)

Het2

1658

—(CH

2

)

5

—

CH

3

H(l = O)

Het2

1659

H

H

CH

2

CH

3

H(l = O)

Het2

1660

CH

3

CH

3

CH

2

CH

3

H(l = O)

Het2

1661

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

H(l = O)

Het2

1662

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

Het2

1663

OCH

3

OCH

3

CH

2

CH

3

H(l = O)

Het2

1664

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

H(l = O)

Het2

1665

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

Het2

1666

SCH

3

SCH

3

CH

2

CH

3

H(l = O)

Het2

1667

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

H(l = O)

Het2

1668

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

H(l = O)

Het2

1669

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

H(l = O)

Het2

1670

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

H(l = O)

Het2

1671

O—(CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

Het2

1672

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

Het2

1673

S—(CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

Het2

1674

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

Het2

1675

—(CH

2

)

4

—

CH

2

CH

3

H(l = O)

Het2

1676

—(CH

2

)

5

—

CH

2

CH

3

H(l = O)

Het2

1677

H

H

CF

3

H(l = O)

Het2

1678

CH

3

CH

3

CF

3

H(l = O)

Het2

1679

CH

2

CH

3

CH

2

CH

3

CF

3

H(l = O)

Het2

1680

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

H(l = O)

Het2

1681

OCH

3

OCH

3

CF

3

H(l = O)

Het2

1682

OCH

2

CH

3

OCH

2

CH

3

CF

3

H(l = O)

Het2

1683

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

H(l = O)

Het2

1684

SCH

3

SCH

3

CF

3

H(l = O)

Het2

1685

SCH

2

CH

3

SCH

2

CH

3

CF

3

H(l = O)

Het2

1686

N(CH

3

)

2

N(CH

3

)

2

CF

3

H(l = O)

Het2

1687

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

H(l = O)

Het2

1688

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

H(l = O)

Het2

1689

O—(CH

2

CH

2

)—O

CF

3

H(l = O)

Het2

1690

O—(CH

2

CH

2

CH

2

)—O

CF

3

H(l = O)

Het2

1691

S—(CH

2

CH

2

)—S

CF

3

H(l = O)

Het2

1692

S—(CH

2

CH

2

CH

2

)—S

CF

3

H(l = O)

Het2

1693

—(CH

2

)

4

—

CF

3

H(l = O)

Het2

1694

—(CH

2

)

5

—

CF

3

H(l = O)

Het2

1695

H

H

OCH

3

H(l = O)

Het2

1696

CH

3

CH

3

OCH

3

H(l = O)

Het2

1697

CH

2

CH

3

CH

2

CH

3

OCH

3

H(l = O)

Het2

1698

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

H(l = O)

Het2

1699

OCH

3

OCH

3

OCH

3

H(l = O)

Het2

1700

OCH

2

CH

3

OCH

2

CH

3

OCH

3

H(l = O)

Het2

1701

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

H(l = O)

Het2

1702

SCH

3

SCH

3

OCH

3

H(l = O)

Het2

1703

SCH

2

CH

3

SCH

2

CH

3

OCH

3

H(l = O)

Het2

1704

N(CH

3

)

2

N(CH

3

)

2

OCH

3

H(l = O)

Het2

1705

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

H(l = O)

Het2

1706

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

H(l = O)

Het2

1707

O—(CH

2

CH

2

)—O

OCH

3

H(l = O)

Het2

1708

O—(CH

2

CH

2

CH

2

)—O

OCH

3

H(l = O)

Het2

1709

S—(CH

2

CH

2

)—S

OCH

3

H(l = O)

Het2

1710

S—(CH

2

CH

2

CH

2

)—S

OCH

3

H(l = O)

Het2

1711

—(CH

2

)

4

—

OCH

3

H(l = O)

Het2

1712

—(CH

2

)

5

—

OCH

3

H(l = O)

Het2

1713

H

H

OCH

2

CH

3

H(l = O)

Het2

1714

CH

3

CH

3

OCH

2

CH

3

H(l = O)

Het2

1715

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

H(l = O)

Het2

1716

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

Het2

1717

OCH

3

OCH

3

OCH

2

CH

3

H(l = O)

Het2

1718

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

H(l = O)

Het2

1719

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

Het2

1720

SCH

3

SCH

3

OCH

2

CH

3

H(l = O)

Het2

1721

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

H(l = O)

Het2

1722

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

H(l = O)

Het2

1723

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

H(l = O)

Het2

1724

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

H(l = O)

Het2

1725

O—(CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

Het2

1726

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

Het2

1727

S—(CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

Het2

1728

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

Het2

1729

—(CH

2

)

4

—

OCH

2

CH

3

H(l = O)

Het2

1730

—(CH

2

)

5

—

OCH

2

CH

3

H(l = O)

Het2

1731

H

H

SCH

3

H(l = O)

Het2

1732

CH

3

CH

3

SCH

3

H(l = O)

Het2

1733

CH

2

CH

3

CH

2

CH

3

SCH

3

H(l = O)

Het2

1734

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

H(l = O)

Het2

1735

OCH

3

OCH

3

SCH

3

H(l = O)

Het2

1736

OCH

2

CH

3

OCH

2

CH

3

SCH

3

H(l = O)

Het2

1737

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

H(l = O)

Het2

1738

SCH

3

SCH

3

SCH

3

H(l = O)

Het2

1739

SCH

2

CH

3

SCH

2

CH

3

SCH

3

H(l = O)

Het2

1740

N(CH

3

)

2

N(CH

3

)

2

SCH

3

H(l = O)

Het2

1741

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

H(l = O)

Het2

1742

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

H(l = O)

Het2

1743

O—(CH

2

CH

2

)—O

SCH

3

H(l = O)

Het2

1744

O—(CH

2

CH

2

CH

2

)—O

SCH

3

H(l = O)

Het2

1745

S—(CH

2

CH

2

)—S

SCH

3

H(l = O)

Het2

1746

S—(CH

2

CH

2

CH

2

)—S

SCH

3

H(l = O)

Het2

1747

—(CH

2

)

4

—

SCH

3

H(l = O)

Het2

1748

—(CH

2

)

5

—

SCH

3

H(l = O)

Het2

1749

H

H

SO

2

CH

3

H(l = O)

Het2

1750

CH

3

CH

3

SO

2

CH

3

H(l = O)

Het2

1751

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

H(l = O)

Het2

1752

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

Het2

1753

OCH

3

OCH

3

SO

2

CH

3

H(l = O)

Het2

1754

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

H(l = O)

Het2

1755

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

Het2

1756

SCH

3

SCH

3

SO

2

CH

3

H(l = O)

Het2

1757

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

H(l = O)

Het2

1758

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

H(l = O)

Het2

1759

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

H(l = O)

Het2

1760

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

H(l = O)

Het2

1761

O—(CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

Het2

1762

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

Het2

1763

S—(CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

Het2

1764

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

Het2

1765

—(CH

2

)

4

—

SO

2

CH

3

H(l = O)

Het2

1766

—(CH

2

)

5

—

SO

2

CH

3

H(l = O)

Het2

1767

H

H

PO(OCH

3

)

2

H(l = O)

Het2

1768

CH

3

CH

3

PO(OCH

3

)

2

H(l = O)

Het2

1769

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het2

1770

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het2

1771

OCH

3

OCH

3

PO(OCH

3

)

2

H(l = O)

Het2

1772

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het2

1773

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het2

1774

SCH

3

SCH

3

PO(OCH

3

)

2

H(l = O)

Het2

1775

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het2

1776

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

H(l = O)

Het2

1777

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

H(l = O)

Het2

1778

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

H(l = O)

Het2

1779

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

Het2

1780

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

Het2

1781

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

Het2

1782

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

Het2

1783

—(CH

2

)

4

—

PO(OCH

3

)

2

H(l = O)

Het2

1784

—(CH

2

)

5

—

PO(OCH

3

)

2

H(l = O)

Het2

1785

H

H

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1786

CH

3

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1787

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1788

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1789

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1790

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1791

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1792

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1793

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1794

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1795

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1796

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1797

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1798

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1799

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1800

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1801

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1802

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

H(l = O)

Het2

1803

H

H

PO(CH

3

)

2

H(l = O)

Het2

1804

CH

3

CH

3

PO(CH

3

)

2

H(l = O)

Het2

1805

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het2

1806

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het2

1807

OCH

3

OCH

3

PO(CH

3

)

2

H(l = O)

Het2

1808

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het2

1809

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het2

1810

SCH

3

SCH

3

PO(CH

3

)

2

H(l = O)

Het2

1811

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het2

1812

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

H(l = O)

Het2

1813

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

H(l = O)

Het2

1814

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

H(l = O)

Het2

1815

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

Het2

1816

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

Het2

1817

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

Het2

1818

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

Het2

1819

—(CH

2

)

4

—

PO(CH

3

)

2

H(l = O)

Het2

1820

—(CH

2

)

5

—

PO(CH

3

)

2

H(l = O)

Het2

1821

H

H

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1822

CH

3

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1823

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1824

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1825

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1826

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1827

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1828

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1829

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1830

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1831

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1832

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1833

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1834

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1835

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1836

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1837

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1838

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

H(l = O)

Het2

1839

H

H

H

H(l = O)

Het3

1840

CH

3

CH

3

H

H(l = O)

Het3

1841

CH

2

CH

3

CH

2

CH

3

H

H(l = O)

Het3

1842

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

H(l = O)

Het3

1843

OCH

3

OCH

3

H

H(l = O)

Het3

1844

OCH

2

CH

3

OCH

2

CH

3

H

H(l = O)

Het3

1845

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

H(l = O)

Het3

1846

SCH

3

SCH

3

H

H(l = O)

Het3

1847

SCH

2

CH

3

SCH

2

CH

3

H

H(l = O)

Het3

1848

N(CH

3

)

2

N(CH

3

)

2

H

H(l = O)

Het3

1849

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

H(l = O)

Het3

1850

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

H(l = O)

Het3

1851

O—(CH

2

CH

2

)—O

H

H(l = O)

Het3

1852

O—(CH

2

CH

2

CH

2

)—O

H

H(l = O)

Het3

1853

S—(CH

2

CH

2

)—S

H

H(l = O)

Het3

1854

S—(CH

2

CH

2

CH

2

)—S

H

H(l = O)

Het3

1855

—(CH

2

)

4

—

H

H(l = O)

Het3

1856

—(CH

2

)

5

—

H

H(l = O)

Het3

1857

H

H

NO

2

H(l = O)

Het3

1858

CH

3

CH

3

NO

2

H(l = O)

Het3

1859

CH

2

CH

3

CH

2

CH

3

NO

2

H(l = O)

Het3

1860

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

H(l = O)

Het3

1861

OCH

3

OCH

3

NO

2

H(l = O)

Het3

1862

OCH

2

CH

3

OCH

2

CH

3

NO

2

H(l = O)

Het3

1863

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

H(l = O)

Het3

1864

SCH

3

SCH

3

NO

2

H(l = O)

Het3

1865

SCH

2

CH

3

SCH

2

CH

3

NO

2

H(l = O)

Het3

1866

N(CH

3

)

2

N(CH

3

)

2

NO

2

H(l = O)

Het3

1867

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

H(l = O)

Het3

1868

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

H(l = O)

Het3

1869

O—(CH

2

CH

2

)—O

NO

2

H(l = O)

Het3

1870

O—(CH

2

CH

2

CH

2

)—O

NO

2

H(l = O)

Het3

1871

S—(CH

2

CH

2

)—S

NO

2

H(l = O)

Het3

1872

S—(CH

2

CH

2

CH

2

)—S

NO

2

H(l = O)

Het3

1873

—(CH

2

)

4

—

NO

2

H(l = O)

Het3

1874

—(CH

2

)

5

—

NO

2

H(l = O)

Het3

1875

H

H

CN

H(l = O)

Het3

1876

CH

3

CH

3

CN

H(l = O)

Het3

1877

CH

2

CH

3

CH

2

CH

3

CN

H(l = O)

Het3

1878

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

H(l = O)

Het3

1879

OCH

3

OCH

3

CN

H(l = O)

Het3

1880

OCH

2

CH

3

OCH

2

CH

3

CN

H(l = O)

Het3

1881

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

H(l = O)

Het3

1882

SCH

3

SCH

3

CN

H(l = O)

Het3

1883

SCH

2

CH

3

SCH

2

CH

3

CN

H(l = O)

Het3

1884

N(CH

3

)

2

N(CH

3

)

2

CN

H(l = O)

Het3

1885

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

H(l = O)

Het3

1886

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

H(l = O)

Het3

1887

O—(CH

2

CH

2

)—O

CN

H(l = O)

Het3

1888

O—(CH

2

CH

2

CH

2

)—O

CN

H(l = O)

Het3

1889

S—(CH

2

CH

2

)—S

CN

H(l = O)

Het3

1890

S—(CH

2

CH

2

CH

2

)—S

CN

H(l = O)

Het3

1891

—(CH

2

)

4

—

CN

H(l = O)

Het3

1892

—(CH

2

)

5

—

CN

H(l = O)

Het3

1893

H

H

F

H(l = O)

Het3

1894

CH

3

CH

3

F

H(l = O)

Het3

1895

CH

2

CH

3

CH

2

CH

3

F

H(l = O)

Het3

1896

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

H(l = O)

Het3

1897

OCH

3

OCH

3

F

H(l = O)

Het3

1898

OCH

2

CH

3

OCH

2

CH

3

F

H(l = O)

Het3

1899

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

H(l = O)

Het3

1900

SCH

3

SCH

3

F

H(l = O)

Het3

1901

SCH

2

CH

3

SCH

2

CH

3

F

H(l = O)

Het3

1902

N(CH

3

)

2

N(CH

3

)

2

F

H(l = O)

Het3

1903

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

H(l = O)

Het3

1904

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

H(l = O)

Het3

1905

O—(CH

2

CH

2

)—O

F

H(l = O)

Het3

1906

O—(CH

2

CH

2

CH

2

)—O

F

H(l = O)

Het3

1907

S—(CH

2

CH

2

)—S

F

H(l = O)

Het3

1908

S—(CH

2

CH

2

CH

2

)—S

F

H(l = O)

Het3

1909

—(CH

2

)

4

—

F

H(l = O)

Het3

1910

—(CH

2

)

5

—

F

H(l = O)

Het3

1911

H

H

Cl

H(l = O)

Het3

1912

CH

3

CH

3

Cl

H(l = O)

Het3

1913

CH

2

CH

3

CH

2

CH

3

Cl

H(l = O)

Het3

1914

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

H(l = O)

Het3

1915

OCH

3

OCH

3

Cl

H(l = O)

Het3

1916

OCH

2

CH

3

OCH

2

CH

3

Cl

H(l = O)

Het3

1917

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

H(l = O)

Het3

1918

SCH

3

SCH

3

Cl

H(l = O)

Het3

1919

SCH

2

CH

3

SCH

2

CH

3

Cl

H(l = O)

Het3

1920

N(CH

3

)

2

N(CH

3

)

2

Cl

H(l = O)

Het3

1921

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

H(l = O)

Het3

1922

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

H(l = O)

Het3

1923

O—(CH

2

CH

2

)—O

Cl

H(l = O)

Het3

1924

O—(CH

2

CH

2

CH

2

)—O

Cl

H(l = O)

Het3

1925

S—(CH

2

CH

2

)—S

Cl

H(l = O)

Het3

1926

S—(CH

2

CH

2

CH

2

)—S

Cl

H(l = O)

Het3

1927

—(CH

2

)

4

—

Cl

H(l = O)

Het3

1928

—(CH

2

)

5

—

Cl

H(l = O)

Het3

1929

H

H

Br

H(l = O)

Het3

1930

CH

3

CH

3

Br

H(l = O)

Het3

1931

CH

2

CH

3

CH

2

CH

3

Br

H(l = O)

Het3

1932

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

H(l = O)

Het3

1933

OCH

3

OCH

3

Br

H(l = O)

Het3

1934

OCH

2

CH

3

OCH

2

CH

3

Br

H(l = O)

Het3

1935

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

H(l = O)

Het3

1936

SCH

3

SCH

3

Br

H(l = O)

Het3

1937

SCH

2

CH

3

SCH

2

CH

3

Br

H(l = O)

Het3

1938

N(CH

3

)

2

N(CH

3

)

2

Br

H(l = O)

Het3

1939

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

H(l = O)

Het3

1940

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

H(l = O)

Het3

1941

O—(CH

2

CH

2

)—O

Br

H(l = O)

Het3

1942

O—(CH

2

CH

2

CH

2

)—O

Br

H(l = O)

Het3

1943

S—(CH

2

CH

2

)—S

Br

H(l = O)

Het3

1944

S—(CH

2

CH

2

CH

2

)—S

Br

H(l = O)

Het3

1945

—(CH

2

)

4

—

Br

H(l = O)

Het3

1946

—(CH

2

)

5

—

Br

H(l = O)

Het3

1947

H

H

CH

3

H(l = O)

Het3

1948

CH

3

CH

3

CH

3

H(l = O)

Het3

1949

CH

2

CH

3

CH

2

CH

3

CH

3

H(l = O)

Het3

1950

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

H(l = O)

Het3

1951

OCH

3

OCH

3

CH

3

H(l = O)

Het3

1952

OCH

2

CH

3

OCH

2

CH

3

CH

3

H(l = O)

Het3

1953

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

H(l = O)

Het3

1954

SCH

3

SCH

3

CH

3

H(l = O)

Het3

1955

SCH

2

CH

3

SCH

2

CH

3

CH

3

H(l = O)

Het3

1956

N(CH

3

)

2

N(CH

3

)

2

CH

3

H(l = O)

Het3

1957

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

H(l = O)

Het3

1958

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

H(l = O)

Het3

1959

O—(CH

2

CH

2

)—O

CH

3

H(l = O)

Het3

1960

O—(CH

2

CH

2

CH

2

)—O

CH

3

H(l = O)

Het3

1961

S—(CH

2

CH

2

)—S

CH

3

H(l = O)

Het3

1962

S—(CH

2

CH

2

CH

2

)—S

CH

3

H(l = O)

Het3

1963

—(CH

2

)

4

—

CH

3

H(l = O)

Het3

1964

—(CH

2

)

5

—

CH

3

H(l = O)

Het3

1965

H

H

CH

2

CH

3

H(l = O)

Het3

1966

CH

3

CH

3

CH

2

CH

3

H(l = O)

Het3

1967

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

H(l = O)

Het3

1968

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

Het3

1969

OCH

3

OCH

3

CH

2

CH

3

H(l = O)

Het3

1970

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

H(l = O)

Het3

1971

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

H(l = O)

Het3

1972

SCH

3

SCH

3

CH

2

CH

3

H(l = O)

Het3

1973

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

H(l = O)

Het3

1974

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

H(l = O)

Het3

1975

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

H(l = O)

Het3

1976

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

H(l = O)

Het3

1977

O—(CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

Het3

1978

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

H(l = O)

Het3

1979

S—(CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

Het3

1980

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

H(l = O)

Het3

1981

—(CH

2

)

4

—

CH

2

CH

3

H(l = O)

Het3

1982

—(CH

2

)

5

—

CH

2

CH

3

H(l = O)

Het3

1983

H

H

CF

3

H(l = O)

Het3

1984

CH

3

CH

3

CF

3

H(l = O)

Het3

1985

CH

2

CH

3

CH

2

CH

3

CF

3

H(l = O)

Het3

1986

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

H(l = O)

Het3

1987

OCH

3

OCH

3

CF

3

H(l = O)

Het3

1988

OCH

2

CH

3

OCH

2

CH

3

CF

3

H(l = O)

Het3

1989

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

H(l = O)

Het3

1990

SCH

3

SCH

3

CF

3

H(l = O)

Het3

1991

SCH

2

CH

3

SCH

2

CH

3

CF

3

H(l = O)

Het3

1992

N(CH

3

)

2

N(CH

3

)

2

CF

3

H(l = O)

Het3

1993

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

H(l = O)

Het3

1994

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

H(l = O)

Het3

1995

O—(CH

2

CH

2

)—O

CF

3

H(l = O)

Het3

1996

O—(CH

2

CH

2

CH

2

)—O

CF

3

H(l = O)

Het3

1997

S—(CH

2

CH

2

)—S

CF

3

H(l = O)

Het3

1998

S—(CH

2

CH

2

CH

2

)—S

CF

3

H(l = O)

Het3

1999

—(CH

2

)

4

—

CF

3

H(l = O)

Het3

2000

—(CH

2

)

5

—

CF

3

H(l = O)

Het3

2001

H

H

OCH

3

H(l = O)

Het3

2002

CH

3

CH

3

OCH

3

H(l = O)

Het3

2003

CH

2

CH

3

CH

2

CH

3

OCH

3

H(l = O)

Het3

2004

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

H(l = O)

Het3

2005

OCH

3

OCH

3

OCH

3

H(l = O)

Het3

2006

OCH

2

CH

3

OCH

2

CH

3

OCH

3

H(l = O)

Het3

2007

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

H(l = O)

Het3

2008

SCH

3

SCH

3

OCH

3

H(l = O)

Het3

2009

SCH

2

CH

3

SCH

2

CH

3

OCH

3

H(l = O)

Het3

2010

N(CH

3

)

2

N(CH

3

)

2

OCH

3

H(l = O)

Het3

2011

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

H(l = O)

Het3

2012

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

H(l = O)

Het3

2013

O—(CH

2

CH

2

)—O

OCH

3

H(l = O)

Het3

2014

O—(CH

2

CH

2

CH

2

)—O

OCH

3

H(l = O)

Het3

2015

S—(CH

2

CH

2

)—S

OCH

3

H(l = O)

Het3

2016

S—(CH

2

CH

2

CH

2

)—S

OCH

3

H(l = O)

Het3

2017

—(CH

2

)

4

—

OCH

3

H(l = O)

Het3

2018

—(CH

2

)

5

—

OCH

3

H(l = O)

Het3

2019

H

H

OCH

2

CH

3

H(l = O)

Het3

2020

CH

3

CH

3

OCH

2

CH

3

H(l = O)

Het3

2021

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

H(l = O)

Het3

2022

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

Het3

2023

OCH

3

OCH

3

OCH

2

CH

3

H(l = O)

Het3

2024

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

H(l = O)

Het3

2025

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

H(l = O)

Het3

2026

SCH

3

SCH

3

OCH

2

CH

3

H(l = O)

Het3

2027

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

H(l = O)

Het3

2028

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

H(l = O)

Het3

2029

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

H(l = O)

Het3

2030

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

H(l = O)

Het3

2031

O—(CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

Het3

2032

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

H(l = O)

Het3

2033

S—(CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

Het3

2034

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

H(l = O)

Het3

2035

—(CH

2

)

4

—

OCH

2

CH

3

H(l = O)

Het3

2036

—(CH

2

)

5

—

OCH

2

CH

3

H(l = O)

Het3

2037

H

H

SCH

3

H(l = O)

Het3

2038

CH

3

CH

3

SCH

3

H(l = O)

Het3

2039

CH

2

CH

3

CH

2

CH

3

SCH

3

H(l = O)

Het3

2040

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

H(l = O)

Het3

2041

OCH

3

OCH

3

SCH

3

H(l = O)

Het3

2042

OCH

2

CH

3

OCH

2

CH

3

SCH

3

H(l = O)

Het3

2043

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

H(l = O)

Het3

2044

SCH

3

SCH

3

SCH

3

H(l = O)

Het3

2045

SCH

2

CH

3

SCH

2

CH

3

SCH

3

H(l = O)

Het3

2046

N(CH

3

)

2

N(CH

3

)

2

SCH

3

H(l = O)

Het3

2047

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

H(l = O)

Het3

2048

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

H(l = O)

Het3

2049

O—(CH

2

CH

2

)—O

SCH

3

H(l = O)

Het3

2050

O—(CH

2

CH

2

CH

2

)—O

SCH

3

H(l = O)

Het3

2051

S—(CH

2

CH

2

)—S

SCH

3

H(l = O)

Het3

2052

S—(CH

2

CH

2

CH

2

)—S

SCH

3

H(l = O)

Het3

2053

—(CH

2

)

4

—

SCH

3

H(l = O)

Het3

2054

—(CH

2

)

5

—

SCH

3

H(l = O)

Het3

2055

H

H

SO

2

CH

3

H(l = O)

Het3

2056

CH

3

CH

3

SO

2

CH

3

H(l = O)

Het3

2057

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

H(l = O)

Het3

2058

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

Het3

2059

OCH

3

OCH

3

SO

2

CH

3

H(l = O)

Het3

2060

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

H(l = O)

Het3

2061

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

H(l = O)

Het3

2062

SCH

3

SCH

3

SO

2

CH

3

H(l = O)

Het3

2063

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

H(l = O)

Het3

2064

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

H(l = O)

Het3

2065

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

H(l = O)

Het3

2066

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

H(l = O)

Het3

2067

O—(CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

Het3

2068

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

H(l = O)

Het3

2069

S—(CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

Het3

2070

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

H(l = O)

Het3

2071

—(CH

2

)

4

—

SO

2

CH

3

H(l = O)

Het3

2072

—(CH

2

)

5

—

SO

2

CH

3

H(l = O)

Het3

2073

H

H

PO(OCH

3

)

2

H(l = O)

Het3

2074

CH

3

CH

3

PO(OCH

3

)

2

H(l = O)

Het3

2075

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het3

2076

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het3

2077

OCH

3

OCH

3

PO(OCH

3

)

2

H(l = O)

Het3

2078

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het3

2079

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het3

2080

SCH

3

SCH

3

PO(OCH

3

)

2

H(l = O)

Het3

2081

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

H(l = O)

Het3

2082

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

H(l = O)

Het3

2083

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

H(l = O)

Het3

2084

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

H(l = O)

Het3

2085

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

Het3

2086

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

H(l = O)

Het3

2087

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

Het3

2088

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

H(l = O)

Het3

2089

—(CH

2

)

4

—

PO(OCH

3

)

2

H(l = O)

Het3

2090

—(CH

2

)

5

—

PO(OCH

3

)

2

H(l = O)

Het3

2091

H

H

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2092

CH

3

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2093

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2094

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2095

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2096

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2097

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2098

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2099

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2100

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2101

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2102

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2103

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2104

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2105

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2106

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2107

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2108

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

H(l = O)

Het3

2109

H

H

PO(CH

3

)

2

H(l = O)

Het3

2110

CH

3

CH

3

PO(CH

3

)

2

H(l = O)

Het3

2111

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het3

2112

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het3

2113

OCH

3

OCH

3

PO(CH

3

)

2

H(l = O)

Het3

2114

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het3

2115

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het3

2116

SCH

3

SCH

3

PO(CH

3

)

2

H(l = O)

Het3

2117

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

H(l = O)

Het3

2118

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

H(l = O)

Het3

2119

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

H(l = O)

Het3

2120

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

H(l = O)

Het3

2121

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

Het3

2122

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

H(l = O)

Het3

2123

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

Het3

2124

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

H(l = O)

Het3

2125

—(CH

2

)

4

—

PO(CH

3

)

2

H(l = O)

Het3

2126

—(CH

2

)

5

—

PO(CH

3

)

2

H(l = O)

Het3

2127

H

H

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2128

CH

3

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2129

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2130

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2131

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2132

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2133

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2134

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2135

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2136

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2137

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2138

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2139

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2140

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2141

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2142

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2143

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2144

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

H(l = O)

Het3

2145

H

H

H

CH

3

OH

2146

CH

3

CH

3

H

CH

3

OH

2147

CH

2

CH

3

CH

2

CH

3

H

CH

3

OH

2148

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

CH

3

OH

2149

OCH

3

OCH

3

H

CH

3

OH

2150

OCH

2

CH

3

OCH

2

CH

3

H

CH

3

OH

2151

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

CH

3

OH

2152

SCH

3

SCH

3

H

CH

3

OH

2153

SCH

2

CH

3

SCH

2

CH

3

H

CH

3

OH

2154

N(CH

3

)

2

N(CH

3

)

2

H

CH

3

OH

2155

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

CH

3

OH

2156

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

CH

3

OH

2157

O—(CH

2

CH

2

)—O

H

CH

3

OH

2158

O—(CH

2

CH

2

CH

2

)—O

H

CH

3

OH

2159

S—(CH

2

CH

2

)—S

H

CH

3

OH

2160

S—(CH

2

CH

2

CH

2

)—S

H

CH

3

OH

2161

—(CH

2

)

4

—

H

CH

3

OH

2162

—(CH

2

)

5

—

H

CH

3

OH

2163

H

H

NO

2

CH

3

OH

2164

CH

3

CH

3

NO

2

CH

3

OH

2165

CH

2

CH

3

CH

2

CH

3

NO

2

CH

3

OH

2166

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

CH

3

OH

2167

OCH

3

OCH

3

NO

2

CH

3

OH

2168

OCH

2

CH

3

OCH

2

CH

3

NO

2

CH

3

OH

2169

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

CH

3

OH

2170

SCH

3

SCH

3

NO

2

CH

3

OH

2171

SCH

2

CH

3

SCH

2

CH

3

NO

2

CH

3

OH

2172

N(CH

3

)

2

N(CH

3

)

2

NO

2

CH

3

OH

2173

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

CH

3

OH

2174

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

CH

3

OH

2175

O—(CH

2

CH

2

)—O

NO

2

CH

3

OH

2176

O—(CH

2

CH

2

CH

2

)—O

NO

2

CH

3

OH

2177

S—(CH

2

CH

2

)—S

NO

2

CH

3

OH

2178

S—(CH

2

CH

2

CH

2

)—S

NO

2

CH

3

OH

2179

—(CH

2

)

4

—

NO

2

CH

3

OH

2180

—(CH

2

)

5

—

NO

2

CH

3

OH

2181

H

H

CN

CH

3

OH

2182

CH

3

CH

3

CN

CH

3

OH

2183

CH

2

CH

3

CH

2

CH

3

CN

CH

3

OH

2184

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

CH

3

OH

2185

OCH

3

OCH

3

CN

CH

3

OH

2186

OCH

2

CH

3

OCH

2

CH

3

CN

CH

3

OH

2187

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

CH

3

OH

2188

SCH

3

SCH

3

CN

CH

3

OH

2189

SCH

2

CH

3

SCH

2

CH

3

CN

CH

3

OH

2190

N(CH

3

)

2

N(CH

3

)

2

CN

CH

3

OH

2191

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

CH

3

OH

2192

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

CH

3

OH

2193

O—(CH

2

CH

2

)—O

CN

CH

3

OH

2194

O—(CH

2

CH

2

CH

2

)—O

CN

CH

3

OH

2195

S—(CH

2

CH

2

)—S

CN

CH

3

OH

2196

S—(CH

2

CH

2

CH

2

)—S

CN

CH

3

OH

2197

—(CH

2

)

4

—

CN

CH

3

OH

2198

—(CH

2

)

5

—

CN

CH

3

OH

2199

H

H

F

CH

3

OH

2200

CH

3

CH

3

F

CH

3

OH

2201

CH

2

CH

3

CH

2

CH

3

F

CH

3

OH

2202

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

CH

3

OH

2203

OCH

3

OCH

3

F

CH

3

OH

2204

OCH

2

CH

3

OCH

2

CH

3

F

CH

3

OH

2205

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

CH

3

OH

2206

SCH

3

SCH

3

F

CH

3

OH

2207

SCH

2

CH

3

SCH

2

CH

3

F

CH

3

OH

2208

N(CH

3

)

2

N(CH

3

)

2

F

CH

3

OH

2209

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

CH

3

OH

2210

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

CH

3

OH

2211

O—(CH

2

CH

2

)—O

F

CH

3

OH

2212

O—(CH

2

CH

2

CH

2

)—O

F

CH

3

OH

2213

S—(CH

2

CH

2

)—S

F

CH

3

OH

2214

S—(CH

2

CH

2

CH

2

)—S

F

CH

3

OH

2215

—(CH

2

)

4

—

F

CH

3

OH

2216

—(CH

2

)

5

—

F

CH

3

OH

2217

H

H

Cl

CH

3

OH

2218

CH

3

CH

3

Cl

CH

3

OH

2219

CH

2

CH

3

CH

2

CH

3

Cl

CH

3

OH

2220

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

CH

3

OH

2221

OCH

3

OCH

3

Cl

CH

3

OH

2222

OCH

2

CH

3

OCH

2

CH

3

Cl

CH

3

OH

2223

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

CH

3

OH

2224

SCH

3

SCH

3

Cl

CH

3

OH

2225

SCH

2

CH

3

SCH

2

CH

3

Cl

CH

3

OH

2226

N(CH

3

)

2

N(CH

3

)

2

Cl

CH

3

OH

2227

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

CH

3

OH

2228

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

CH

3

OH

2229

O—(CH

2

CH

2

)—O

Cl

CH

3

OH

2230

O—(CH

2

CH

2

CH

2

)—O

Cl

CH

3

OH

2231

S—(CH

2

CH

2

)—S

Cl

CH

3

OH

2232

S—(CH

2

CH

2

CH

2

)—S

Cl

CH

3

OH

2233

—(CH

2

)

4

—

Cl

CH

3

OH

2234

—(CH

2

)

5

—

Cl

CH

3

OH

2235

H

H

Br

CH

3

OH

2236

CH

3

CH

3

Br

CH

3

OH

2237

CH

2

CH

3

CH

2

CH

3

Br

CH

3

OH

2238

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

CH

3

OH

2239

OCH

3

OCH

3

Br

CH

3

OH

2240

OCH

2

CH

3

OCH

2

CH

3

Br

CH

3

OH

2241

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

CH

3

OH

2242

SCH

3

SCH

3

Br

CH

3

OH

2243

SCH

2

CH

3

SCH

2

CH

3

Br

CH

3

OH

2244

N(CH

3

)

2

N(CH

3

)

2

Br

CH

3

OH

2245

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

CH

3

OH

2246

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

CH

3

OH

2247

O—(CH

2

CH

2

)—O

Br

CH

3

OH

2248

O—(CH

2

CH

2

CH

2

)—O

Br

CH

3

OH

2249

S—(CH

2

CH

2

)—S

Br

CH

3

OH

2250

S—(CH

2

CH

2

CH

2

)—S

Br

CH

3

OH

2251

—(CH

2

)

4

—

Br

CH

3

OH

2252

—(CH

2

)

5

—

Br

CH

3

OH

2253

H

H

CH

3

CH

3

OH

2254

CH

3

CH

3

CH

3

CH

3

OH

2255

CH

2

CH

3

CH

2

CH

3

CH

3

CH

3

OH

2256

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

CH

3

OH

2257

OCH

3

OCH

3

CH

3

CH

3

OH

2258

OCH

2

CH

3

OCH

2

CH

3

CH

3

CH

3

OH

2259

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

CH

3

OH

2260

SCH

3

SCH

3

CH

3

CH

3

OH

2261

SCH

2

CH

3

SCH

2

CH

3

CH

3

CH

3

OH

2262

N(CH

3

)

2

N(CH

3

)

2

CH

3

CH

3

OH

2263

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

CH

3

OH

2264

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

CH

3

OH

2265

O—(CH

2

CH

2

)—O

CH

3

CH

3

OH

2266

O—(CH

2

CH

2

CH

2

)—O

CH

3

CH

3

OH

2267

S—(CH

2

CH

2

)—S

CH

3

CH

3

OH

2268

S—(CH

2

CH

2

CH

2

)—S

CH

3

CH

3

OH

2269

—(CH

2

)

4

—

CH

3

CH

3

OH

2270

—(CH

2

)

5

—

CH

3

CH

3

OH

2271

H

H

CH

2

CH

3

CH

3

OH

2272

CH

3

CH

3

CH

2

CH

3

CH

3

OH

2273

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

CH

3

OH

2274

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

CH

3

OH

2275

OCH

3

OCH

3

CH

2

CH

3

CH

3

OH

2276

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

CH

3

OH

2277

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

CH

3

OH

2278

SCH

3

SCH

3

CH

2

CH

3

CH

3

OH

2279

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

CH

3

OH

2280

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

CH

3

OH

2281

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

CH

3

OH

2282

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

CH

3

OH

2283

O—(CH

2

CH

2

)—O

CH

2

CH

3

CH

3

OH

2284

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

CH

3

OH

2285

S—(CH

2

CH

2

)—S

CH

2

CH

3

CH

3

OH

2286

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

CH

3

OH

2287

—(CH

2

)

4

—

CH

2

CH

3

CH

3

OH

2288

—(CH

2

)

5

—

CH

2

CH

3

CH

3

OH

2289

H

H

CF

3

CH

3

OH

2290

CH

3

CH

3

CF

3

CH

3

OH

2291

CH

2

CH

3

CH

2

CH

3

CF

3

CH

3

OH

2292

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

CH

3

OH

2293

OCH

3

OCH

3

CF

3

CH

3

OH

2294

OCH

2

CH

3

OCH

2

CH

3

CF

3

CH

3

OH

2295

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

CH

3

OH

2296

SCH

3

SCH

3

CF

3

CH

3

OH

2297

SCH

2

CH

3

SCH

2

CH

3

CF

3

CH

3

OH

2298

N(CH

3

)

2

N(CH

3

)

2

CF

3

CH

3

OH

2299

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

CH

3

OH

2300

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

CH

3

OH

2301

O—(CH

2

CH

2

)—O

CF

3

CH

3

OH

2302

O—(CH

2

CH

2

CH

2

)—O

CF

3

CH

3

OH

2303

S—(CH

2

CH

2

)—S

CF

3

CH

3

OH

2304

S—(CH

2

CH

2

CH

2

)—S

CF

3

CH

3

OH

2305

—(CH

2

)

4

—

CF

3

CH

3

OH

2306

—(CH

2

)

5

—

CF

3

CH

3

OH

2307

H

H

OCH

3

CH

3

OH

2308

CH

3

CH

3

OCH

3

CH

3

OH

2309

CH

2

CH

3

CH

2

CH

3

OCH

3

CH

3

OH

2310

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

CH

3

OH

2311

OCH

3

OCH

3

OCH

3

CH

3

OH

2312

OCH

2

CH

3

OCH

2

CH

3

OCH

3

CH

3

OH

2313

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

CH

3

OH

2314

SCH

3

SCH

3

OCH

3

CH

3

OH

2315

SCH

2

CH

3

SCH

2

CH

3

OCH

3

CH

3

OH

2316

N(CH

3

)

2

N(CH

3

)

2

OCH

3

CH

3

OH

2317

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

CH

3

OH

2318

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

CH

3

OH

2319

O—(CH

2

CH

2

)—O

OCH

3

CH

3

OH

2320

O—(CH

2

CH

2

CH

2

)—O

OCH

3

CH

3

OH

2321

S—(CH

2

CH

2

)—S

OCH

3

CH

3

OH

2322

S—(CH

2

CH

2

CH

2

)—S

OCH

3

CH

3

OH

2323

—(CH

2

)

4

—

OCH

3

CH

3

OH

2324

—(CH

2

)

5

—

OCH

3

CH

3

OH

2325

H

H

OCH

2

CH

3

CH

3

OH

2326

CH

3

CH

3

OCH

2

CH

3

CH

3

OH

2327

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

CH

3

OH

2328

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

CH

3

OH

2329

OCH

3

OCH

3

OCH

2

CH

3

CH

3

OH

2330

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

CH

3

OH

2331

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

CH

3

OH

2332

SCH

3

SCH

3

OCH

2

CH

3

CH

3

OH

2333

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

CH

3

OH

2334

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

CH

3

OH

2335

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

CH

3

OH

2336

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

CH

3

OH

2337

O—(CH

2

CH

2

)—O

OCH

2

CH

3

CH

3

OH

2338

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

CH

3

OH

2339

S—(CH

2

CH

2

)—S

OCH

2

CH

3

CH

3

OH

2340

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

CH

3

OH

2341

—(CH

2

)

4

—

OCH

2

CH

3

CH

3

OH

2342

—(CH

2

)

5

—

OCH

2

CH

3

CH

3

OH

2343

H

H

SCH

3

CH

3

OH

2344

CH

3

CH

3

SCH

3

CH

3

OH

2345

CH

2

CH

3

CH

2

CH

3

SCH

3

CH

3

OH

2346

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

CH

3

OH

2347

OCH

3

OCH

3

SCH

3

CH

3

OH

2348

OCH

2

CH

3

OCH

2

CH

3

SCH

3

CH

3

OH

2349

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

CH

3

OH

2350

SCH

3

SCH

3

SCH

3

CH

3

OH

2351

SCH

2

CH

3

SCH

2

CH

3

SCH

3

CH

3

OH

2352

N(CH

3

)

2

N(CH

3

)

2

SCH

3

CH

3

OH

2353

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

CH

3

OH

2354

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

CH

3

OH

2355

O—(CH

2

CH

2

)—O

SCH

3

CH

3

OH

2356

O—(CH

2

CH

2

CH

2

)—O

SCH

3

CH

3

OH

2357

S—(CH

2

CH

2

)—S

SCH

3

CH

3

OH

2358

S—(CH

2

CH

2

CH

2

)—S

SCH

3

CH

3

OH

2359

—(CH

2

)

4

—

SCH

3

CH

3

OH

2360

—(CH

2

)

5

—

SCH

3

CH

3

OH

2361

H

H

SO

2

CH

3

CH

3

OH

2362

CH

3

CH

3

SO

2

CH

3

CH

3

OH

2363

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

CH

3

OH

2364

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

CH

3

OH

2365

OCH

3

OCH

3

SO

2

CH

3

CH

3

OH

2366

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

CH

3

OH

2367

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

CH

3

OH

2368

SCH

3

SCH

3

SO

2

CH

3

CH

3

OH

2369

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

CH

3

OH

2370

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

CH

3

OH

2371

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

CH

3

OH

2372

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

CH

3

OH

2373

O—(CH

2

CH

2

)—O

SO

2

CH

3

CH

3

OH

2374

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

CH

3

OH

2375

S—(CH

2

CH

2

)—S

SO

2

CH

3

CH

3

OH

2376

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

CH

3

OH

2377

—(CH

2

)

4

—

SO

2

CH

3

CH

3

OH

2378

—(CH

2

)

5

—

SO

2

CH

3

CH

3

OH

2379

H

H

PO(OCH

3

)

2

CH

3

OH

2380

CH

3

CH

3

PO(OCH

3

)

2

CH

3

OH

2381

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

CH

3

OH

2382

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

CH

3

OH

2383

OCH

3

OCH

3

PO(OCH

3

)

2

CH

3

OH

2384

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

CH

3

OH

2385

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

CH

3

OH

2386

SCH

3

SCH

3

PO(OCH

3

)

2

CH

3

OH

2387

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

CH

3

OH

2388

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

CH

3

OH

2389

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

CH

3

OH

2390

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

CH

3

OH

2391

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

CH

3

OH

2392

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

CH

3

OH

2393

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

CH

3

OH

2394

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

CH

3

OH

2395

—(CH

2

)

4

—

PO(OCH

3

)

2

CH

3

OH

2396

—(CH

2

)

5

—

PO(OCH

3

)

2

CH

3

OH

2397

H

H

PO(OCH

2

CH

3

)

2

CH

3

OH

2398

CH

3

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OH

2399

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OH

2400

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OH

2401

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

CH

3

OH

2402

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OH

2403

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OH

2404

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

CH

3

OH

2405

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OH

2406

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

CH

3

OH

2407

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

CH

3

OH

2408

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

CH

3

OH

2409

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

CH

3

OH

2410

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

CH

3

OH

2411

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

CH

3

OH

2412

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

CH

3

OH

2413

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

CH

3

OH

2414

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

CH

3

OH

2415

H

H

PO(CH

3

)

2

CH

3

OH

2416

CH

3

CH

3

PO(CH

3

)

2

CH

3

OH

2417

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

CH

3

OH

2418

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

CH

3

OH

2419

OCH

3

OCH

3

PO(CH

3

)

2

CH

3

OH

2420

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

CH

3

OH

2421

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

CH

3

OH

2422

SCH

3

SCH

3

PO(CH

3

)

2

CH

3

OH

2423

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

CH

3

OH

2424

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

CH

3

OH

2425

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

CH

3

OH

2426

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

CH

3

OH

2427

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

CH

3

OH

2428

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

CH

3

OH

2429

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

CH

3

OH

2430

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

CH

3

OH

2431

—(CH

2

)

4

—

PO(CH

3

)

2

CH

3

OH

2432

—(CH

2

)

5

—

PO(CH

3

)

2

CH

3

OH

2433

H

H

PO(CH

2

CH

3

)

2

CH

3

OH

2434

CH

3

CH

3

PO(CH

2

CH

3

)

2

CH

3

OH

2435

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

OH

2436

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

OH

2437

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

CH

3

OH

2438

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

OH

2439

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

OH

2440

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

CH

3

OH

2441

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

OH

2442

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

CH

3

OH

2443

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

CH

3

OH

2444

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

CH

3

OH

2445

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

CH

3

OH

2446

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

CH

3

OH

2447

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

CH

3

OH

2448

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

CH

3

OH

2449

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

CH

3

OH

2450

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

CH

3

OH

2451

H

H

H

CH

3

OCOC

6

H

5

2452

CH

3

CH

3

H

CH

3

OCOC

6

H

5

2453

CH

2

CH

3

CH

2

CH

3

H

CH

3

OCOC

6

H

5

2454

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

CH

3

OCOC

6

H

5

2455

OCH

3

OCH

3

H

CH

3

OCOC

6

H

5

2456

OCH

2

CH

3

OCH

2

CH

3

H

CH

3

OCOC

6

H

5

2457

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

CH

3

OCOC

6

H

5

2458

SCH

3

SCH

3

H

CH

3

OCOC

6

H

5

2459

SCH

2

CH

3

SCH

2

CH

3

H

CH

3

OCOC

6

H

5

2460

N(CH

3

)

2

N(CH

3

)

2

H

CH

3

OCOC

6

H

5

2461

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

CH

3

OCOC

6

H

5

2462

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

CH

3

OCOC

6

H

5

2463

O—(CH

2

CH

2

)—O

H

CH

3

OCOC

6

H

5

2464

O—(CH

2

CH

2

CH

2

)—O

H

CH

3

OCOC

6

H

5

2465

S—(CH

2

CH

2

)—S

H

CH

3

OCOC

6

H

5

2466

S—(CH

2

CH

2

CH

2

)—S

H

CH

3

OCOC

6

H

5

2467

—(CH

2

)

4

—

H

CH

3

OCOC

6

H

5

2468

—(CH

2

)

5

—

H

CH

3

OCOC

6

H

5

2469

H

H

NO

2

CH

3

OCOC

6

H

5

2470

CH

3

CH

3

NO

2

CH

3

OCOC

6

H

5

2471

CH

2

CH

3

CH

2

CH

3

NO

2

CH

3

OCOC

6

H

5

2472

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

CH

3

OCOC

6

H

5

2473

OCH

3

OCH

3

NO

2

CH

3

OCOC

6

H

5

2474

OCH

2

CH

3

OCH

2

CH

3

NO

2

CH

3

OCOC

6

H

5

2475

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

CH

3

OCOC

6

H

5

2476

SCH

3

SCH

3

NO

2

CH

3

OCOC

6

H

5

2477

SCH

2

CH

3

SCH

2

CH

3

NO

2

CH

3

OCOC

6

H

5

2478

N(CH

3

)

2

N(CH

3

)

2

NO

2

CH

3

OCOC

6

H

5

2479

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

CH

3

OCOC

6

H

5

2480

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

CH

3

OCOC

6

H

5

2481

O—(CH

2

CH

2

)—O

NO

2

CH

3

OCOC

6

H

5

2482

O—(CH

2

CH

2

CH

2

)—O

NO

2

CH

3

OCOC

6

H

5

2483

S—(CH

2

CH

2

)—S

NO

2

CH

3

OCOC

6

H

5

2484

S—(CH

2

CH

2

CH

2

)—S

NO

2

CH

3

OCOC

6

H

5

2485

—(CH

2

)

4

—

NO

2

CH

3

OCOC

6

H

5

2486

—(CH

2

)

5

—

NO

2

CH

3

OCOC

6

H

5

2487

H

H

CN

CH

3

OCOC

6

H

5

2488

CH

3

CH

3

CN

CH

3

OCOC

6

H

5

2489

CH

2

CH

3

CH

2

CH

3

CN

CH

3

OCOC

6

H

5

2490

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

CH

3

OCOC

6

H

5

2491

OCH

3

OCH

3

CN

CH

3

OCOC

6

H

5

2492

OCH

2

CH

3

OCH

2

CH

3

CN

CH

3

OCOC

6

H

5

2493

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

CH

3

OCOC

6

H

5

2494

SCH

3

SCH

3

CN

CH

3

OCOC

6

H

5

2495

SCH

2

CH

3

SCH

2

CH

3

CN

CH

3

OCOC

6

H

5

2496

N(CH

3

)

2

N(CH

3

)

2

CN

CH

3

OCOC

6

H

5

2497

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

CH

3

OCOC

6

H

5

2498

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

CH

3

OCOC

6

H

5

2499

O—(CH

2

CH

2

)—O

CN

CH

3

OCOC

6

H

5

2500

O—(CH

2

CH

2

CH

2

)—O

CN

CH

3

OCOC

6

H

5

2501

S—(CH

2

CH

2

)—S

CN

CH

3

OCOC

6

H

5

2502

S—(CH

2

CH

2

CH

2

)—S

CN

CH

3

OCOC

6

H

5

2503

—(CH

2

)

4

—

CN

CH

3

OCOC

6

H

5

2504

—(CH

2

)

5

—

CN

CH

3

OCOC

6

H

5

2505

H

H

F

CH

3

OCOC

6

H

5

2506

CH

3

CH

3

F

CH

3

OCOC

6

H

5

2507

CH

2

CH

3

CH

2

CH

3

F

CH

3

OCOC

6

H

5

2508

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

CH

3

OCOC

6

H

5

2509

OCH

3

OCH

3

F

CH

3

OCOC

6

H

5

2510

OCH

2

CH

3

OCH

2

CH

3

F

CH

3

OCOC

6

H

5

2511

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

CH

3

OCOC

6

H

5

2512

SCH

3

SCH

3

F

CH

3

OCOC

6

H

5

2513

SCH

2

CH

3

SCH

2

CH

3

F

CH

3

OCOC

6

H

5

2514

N(CH

3

)

2

N(CH

3

)

2

F

CH

3

OCOC

6

H

5

2515

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

CH

3

OCOC

6

H

5

2516

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

CH

3

OCOC

6

H

5

2517

O—(CH

2

CH

2

)—O

F

CH

3

OCOC

6

H

5

2518

O—(CH

2

CH

2

CH

2

)—O

F

CH

3

OCOC

6

H

5

2519

S—(CH

2

CH

2

)—S

F

CH

3

OCOC

6

H

5

2520

S—(CH

2

CH

2

CH

2

)—S

F

CH

3

OCOC

6

H

5

2521

—(CH

2

)

4

—

F

CH

3

OCOC

6

H

5

2522

—(CH

2

)

5

—

F

CH

3

OCOC

6

H

5

2523

H

H

Cl

CH

3

OCOC

6

H

5

2524

CH

3

CH

3

Cl

CH

3

OCOC

6

H

5

2525

CH

2

CH

3

CH

2

CH

3

Cl

CH

3

OCOC

6

H

5

2526

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

CH

3

OCOC

6

H

5

2527

OCH

3

OCH

3

Cl

CH

3

OCOC

6

H

5

2528

OCH

2

CH

3

OCH

2

CH

3

Cl

CH

3

OCOC

6

H

5

2529

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

CH

3

OCOC

6

H

5

2530

SCH

3

SCH

3

Cl

CH

3

OCOC

6

H

5

2531

SCH

2

CH

3

SCH

2

CH

3

Cl

CH

3

OCOC

6

H

5

2532

N(CH

3

)

2

N(CH

3

)

2

Cl

CH

3

OCOC

6

H

5

2533

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

CH

3

OCOC

6

H

5

2534

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

CH

3

OCOC

6

H

5

2535

O—(CH

2

CH

2

)—O

Cl

CH

3

OCOC

6

H

5

2536

O—(CH

2

CH

2

CH

2

)—O

Cl

CH

3

OCOC

6

H

5

2537

S—(CH

2

CH

2

)—S

Cl

CH

3

OCOC

6

H

5

2538

S—(CH

2

CH

2

CH

2

)—S

Cl

CH

3

OCOC

6

H

5

2539

—(CH

2

)

4

—

Cl

CH

3

OCOC

6

H

5

2540

—(CH

2

)

5

—

Cl

CH

3

OCOC

6

H

5

2541

H

H

Br

CH

3

OCOC

6

H

5

2542

CH

3

CH

3

Br

CH

3

OCOC

6

H

5

2543

CH

2

CH

3

CH

2

CH

3

Br

CH

3

OCOC

6

H

5

2544

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

CH

3

OCOC

6

H

5

2545

OCH

3

OCH

3

Br

CH

3

OCOC

6

H

5

2546

OCH

2

CH

3

OCH

2

CH

3

Br

CH

3

OCOC

6

H

5

2547

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

CH

3

OCOC

6

H

5

2548

SCH

3

SCH

3

Br

CH

3

OCOC

6

H

5

2549

SCH

2

CH

3

SCH

2

CH

3

Br

CH

3

OCOC

6

H

5

2550

N(CH

3

)

2

N(CH

3

)

2

Br

CH

3

OCOC

6

H

5

2551

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

CH

3

OCOC

6

H

5

2552

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

CH

3

OCOC

6

H

5

2553

O—(CH

2

CH

2

)—O

Br

CH

3

OCOC

6

H

5

2554

O—(CH

2

CH

2

CH

2

)—O

Br

CH

3

OCOC

6

H

5

2555

S—(CH

2

CH

2

)—S

Br

CH

3

OCOC

6

H

5

2556

S—(CH

2

CH

2

CH

2

)—S

Br

CH

3

OCOC

6

H

5

2557

—(CH

2

)

4

—

Br

CH

3

OCOC

6

H

5

2558

—(CH

2

)

5

—

Br

CH

3

OCOC

6

H

5

2559

H

H

CH

3

CH

3

OCOC

6

H

5

2560

CH

3

CH

3

CH

3

CH

3

OCOC

6

H

5

2561

CH

2

CH

3

CH

2

CH

3

CH

3

CH

3

OCOC

6

H

5

2562

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

CH

3

OCOC

6

H

5

2563

OCH

3

OCH

3

CH

3

CH

3

OCOC

6

H

5

2564

OCH

2

CH

3

OCH

2

CH

3

CH

3

CH

3

OCOC

6

H

5

2565

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

CH

3

OCOC

6

H

5

2566

SCH

3

SCH

3

CH

3

CH

3

OCOC

6

H

5

2567

SCH

2

CH

3

SCH

2

CH

3

CH

3

CH

3

OCOC

6

H

5

2568

N(CH

3

)

2

N(CH

3

)

2

CH

3

CH

3

OCOC

6

H

5

2569

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

CH

3

OCOC

6

H

5

2570

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

CH

3

OCOC

6

H

5

2571

O—(CH

2

CH

2

)—O

CH

3

CH

3

OCOC

6

H

5

2572

O—(CH

2

CH

2

CH

2

)—O

CH

3

CH

3

OCOC

6

H

5

2573

S—(CH

2

CH

2

)—S

CH

3

CH

3

OCOC

6

H

5

2574

S—(CH

2

CH

2

CH

2

)—S

CH

3

CH

3

OCOC

6

H

5

2575

—(CH

2

)

4

—

CH

3

CH

3

OCOC

6

H

5

2576

—(CH

2

)

5

—

CH

3

CH

3

OCOC

6

H

5

2577

H

H

CH

2

CH

3

CH

3

OCOC

6

H

5

2578

CH

3

CH

3

CH

2

CH

3

CH

3

OCOC

6

H

5

2579

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

CH

3

OCOC

6

H

5

2580

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

CH

3

OCOC

6

H

5

2581

OCH

3

OCH

3

CH

2

CH

3

CH

3

OCOC

6

H

5

2582

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

CH

3

OCOC

6

H

5

2583

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

CH

3

OCOC

6

H

5

2584

SCH

3

SCH

3

CH

2

CH

3

CH

3

OCOC

6

H

5

2585

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

CH

3

OCOC

6

H

5

2586

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

CH

3

OCOC

6

H

5

2587

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

CH

3

OCOC

6

H

5

2588

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

CH

3

OCOC

6

H

5

2589

O—(CH

2

CH

2

)—O

CH

2

CH

3

CH

3

OCOC

6

H

5

2590

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

CH

3

OCOC

6

H

5

2591

S—(CH

2

CH

2

)—S

CH

2

CH

3

CH

3

OCOC

6

H

5

2592

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

CH

3

OCOC

6

H

5

2593

—(CH

2

)

4

—

CH

2

CH

3

CH

3

OCOC

6

H

5

2594

—(CH

2

)

5

—

CH

2

CH

3

CH

3

OCOC

6

H

5

2595

H

H

CF

3

CH

3

OCOC

6

H

5

2596

CH

3

CH

3

CF

3

CH

3

OCOC

6

H

5

2597

CH

2

CH

3

CH

2

CH

3

CF

3

CH

3

OCOC

6

H

5

2598

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

CH

3

OCOC

6

H

5

2599

OCH

3

OCH

3

CF

3

CH

3

OCOC

6

H

5

2600

OCH

2

CH

3

OCH

2

CH

3

CF

3

CH

3

OCOC

6

H

5

2601

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

CH

3

OCOC

6

H

5

2602

SCH

3

SCH

3

CF

3

CH

3

OCOC

6

H

5

2603

SCH

2

CH

3

SCH

2

CH

3

CF

3

CH

3

OCOC

6

H

5

2604

N(CH

3

)

2

N(CH

3

)

2

CF

3

CH

3

OCOC

6

H

5

2605

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

CH

3

OCOC

6

H

5

2606

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

CH

3

OCOC

6

H

5

2607

O—(CH

2

CH

2

)—O

CF

3

CH

3

OCOC

6

H

5

2608

O—(CH

2

CH

2

CH

2

)—O

CF

3

CH

3

OCOC

6

H

5

2609

S—(CH

2

CH

2

)—S

CF

3

CH

3

OCOC

6

H

5

2610

S—(CH

2

CH

2

CH

2

)—S

CF

3

CH

3

OCOC

6

H

5

2611

—(CH

2

)

4

—

CF

3

CH

3

OCOC

6

H

5

2612

—(CH

2

)

5

—

CF

3

CH

3

OCOC

6

H

5

2613

H

H

OCH

3

CH

3

OCOC

6

H

5

2614

CH

3

CH

3

OCH

3

CH

3

OCOC

6

H

5

2615

CH

2

CH

3

CH

2

CH

3

OCH

3

CH

3

OCOC

6

H

5

2616

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

CH

3

OCOC

6

H

5

2617

OCH

3

OCH

3

OCH

3

CH

3

OCOC

6

H

5

2618

OCH

2

CH

3

OCH

2

CH

3

OCH

3

CH

3

OCOC

6

H

5

2619

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

CH

3

OCOC

6

H

5

2620

SCH

3

SCH

3

OCH

3

CH

3

OCOC

6

H

5

2621

SCH

2

CH

3

SCH

2

CH

3

OCH

3

CH

3

OCOC

6

H

5

2622

N(CH

3

)

2

N(CH

3

)

2

OCH

3

CH

3

OCOC

6

H

5

2623

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

CH

3

OCOC

6

H

5

2624

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

CH

3

OCOC

6

H

5

2625

O—(CH

2

CH

2

)—O

OCH

3

CH

3

OCOC

6

H

5

2626

O—(CH

2

CH

2

CH

2

)—O

OCH

3

CH

3

OCOC

6

H

5

2627

S—(CH

2

CH

2

)—S

OCH

3

CH

3

OCOC

6

H

5

2628

S—(CH

2

CH

2

CH

2

)—S

OCH

3

CH

3

OCOC

6

H

5

2629

—(CH

2

)

4

—

OCH

3

CH

3

OCOC

6

H

5

2630

—(CH

2

)

5

—

OCH

3

CH

3

OCOC

6

H

5

2631

H

H

OCH

2

CH

3

CH

3

OCOC

6

H

5

2632

CH

3

CH

3

OCH

2

CH

3

CH

3

OCOC

6

H

5

2633

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

CH

3

OCOC

6

H

5

2634

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

CH

3

OCOC

6

H

5

2635

OCH

3

OCH

3

OCH

2

CH

3

CH

3

OCOC

6

H

5

2636

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

CH

3

OCOC

6

H

5

2637

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

CH

3

OCOC

6

H

5

2638

SCH

3

SCH

3

OCH

2

CH

3

CH

3

OCOC

6

H

5

2639

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

CH

3

OCOC

6

H

5

2640

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

CH

3

OCOC

6

H

5

2641

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

CH

3

OCOC

6

H

5

2642

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

CH

3

OCOC

6

H

5

2643

O—(CH

2

CH

2

)—O

OCH

2

CH

3

CH

3

OCOC

6

H

5

2644

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

CH

3

OCOC

6

H

5

2645

S—(CH

2

CH

2

)—S

OCH

2

CH

3

CH

3

OCOC

6

H

5

2646

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

CH

3

OCOC

6

H

5

2647

—(CH

2

)

4

—

OCH

2

CH

3

CH

3

OCOC

6

H

5

2648

—(CH

2

)

5

—

OCH

2

CH

3

CH

3

OCOC

6

H

5

2649

H

H

SCH

3

CH

3

OCOC

6

H

5

2650

CH

3

CH

3

SCH

3

CH

3

OCOC

6

H

5

2651

CH

2

CH

3

CH

2

CH

3

SCH

3

CH

3

OCOC

6

H

5

2652

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

CH

3

OCOC

6

H

5

2653

OCH

3

OCH

3

SCH

3

CH

3

OCOC

6

H

5

2654

OCH

2

CH

3

OCH

2

CH

3

SCH

3

CH

3

OCOC

6

H

5

2655

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

CH

3

OCOC

6

H

5

2656

SCH

3

SCH

3

SCH

3

CH

3

OCOC

6

H

5

2657

SCH

2

CH

3

SCH

2

CH

3

SCH

3

CH

3

OCOC

6

H

5

2658

N(CH

3

)

2

N(CH

3

)

2

SCH

3

CH

3

OCOC

6

H

5

2659

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

CH

3

OCOC

6

H

5

2660

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

CH

3

OCOC

6

H

5

2661

O—(CH

2

CH

2

)—O

SCH

3

CH

3

OCOC

6

H

5

2662

O—(CH

2

CH

2

CH

2

)—O

SCH

3

CH

3

OCOC

6

H

5

2663

S—(CH

2

CH

2

)—S

SCH

3

CH

3

OCOC

6

H

5

2664

S—(CH

2

CH

2

CH

2

)—S

SCH

3

CH

3

OCOC

6

H

5

2665

—(CH

2

)

4

—

SCH

3

CH

3

OCOC

6

H

5

2666

—(CH

2

)

5

—

SCH

3

CH

3

OCOC

6

H

5

2667

H

H

SO

2

CH

3

CH

3

OCOC

6

H

5

2668

CH

3

CH

3

SO

2

CH

3

CH

3

OCOC

6

H

5

2669

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

CH

3

OCOC

6

H

5

2670

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

CH

3

OCOC

6

H

5

2671

OCH

3

OCH

3

SO

2

CH

3

CH

3

OCOC

6

H

5

2672

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

CH

3

OCOC

6

H

5

2673

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

CH

3

OCOC

6

H

5

2674

SCH

3

SCH

3

SO

2

CH

3

CH

3

OCOC

6

H

5

2675

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

CH

3

OCOC

6

H

5

2676

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

CH

3

OCOC

6

H

5

2677

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

CH

3

OCOC

6

H

5

2678

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

CH

3

OCOC

6

H

5

2679

O—(CH

2

CH

2

)—O

SO

2

CH

3

CH

3

OCOC

6

H

5

2680

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

CH

3

OCOC

6

H

5

2681

S—(CH

2

CH

2

)—S

SO

2

CH

3

CH

3

OCOC

6

H

5

2682

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

CH

3

OCOC

6

H

5

2683

—(CH

2

)

4

—

SO

2

CH

3

CH

3

OCOC

6

H

5

2684

—(CH

2

)

5

—

SO

2

CH

3

CH

3

OCOC

6

H

5

2685

H

H

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2686

CH

3

CH

3

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2687

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2688

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2689

OCH

3

OCH

3

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2690

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2691

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2692

SCH

3

SCH

3

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2693

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2694

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2695

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2696

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2697

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2698

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2699

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2700

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2701

—(CH

2

)

4

—

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2702

—(CH

2

)

5

—

PO(OCH

3

)

2

CH

3

OCOC

6

H

5

2703

H

H

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2704

CH

3

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2705

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2706

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2707

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2708

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2709

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2710

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2711

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2712

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2713

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2714

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2715

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2716

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2717

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2718

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2719

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2720

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2721

H

H

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2722

CH

3

CH

3

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2723

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2724

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2725

OCH

3

OCH

3

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2726

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2727

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2728

SCH

3

SCH

3

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2729

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2730

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2731

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2732

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2733

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2734

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2735

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2736

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2737

—(CH

2

)

4

—

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2738

—(CH

2

)

5

—

PO(CH

3

)

2

CH

3

OCOC

6

H

5

2739

H

H

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2740

CH

3

CH

3

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2741

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2742

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2743

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2744

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2745

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2746

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2747

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2748

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2749

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2750

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2751

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2752

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2753

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2754

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2755

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2756

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

CH

3

OCOC

6

H

5

2757

H

H

H

CH

3

SCH

3

2758

CH

3

CH

3

H

CH

3

SCH

3

2759

CH

2

CH

3

CH

2

CH

3

H

CH

3

SCH

3

2760

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

CH

3

SCH

3

2761

OCH

3

OCH

3

H

CH

3

SCH

3

2762

OCH

2

CH

3

OCH

2

CH

3

H

CH

3

SCH

3

2763

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

CH

3

SCH

3

2764

SCH

3

SCH

3

H

CH

3

SCH

3

2765

SCH

2

CH

3

SCH

2

CH

3

H

CH

3

SCH

3

2766

N(CH

3

)

2

N(CH

3

)

2

H

CH

3

SCH

3

2767

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

CH

3

SCH

3

2768

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

CH

3

SCH

3

2769

O—(CH

2

CH

2

)—O

H

CH

3

SCH

3

2770

O—(CH

2

CH

2

CH

2

)—O

H

CH

3

SCH

3

2771

S—(CH

2

CH

2

)—S

H

CH

3

SCH

3

2772

S—(CH

2

CH

2

CH

2

)—S

H

CH

3

SCH

3

2773

—(CH

2

)

4

—

H

CH

3

SCH

3

2774

—(CH

2

)

5

—

H

CH

3

SCH

3

2775

H

H

NO

2

CH

3

SCH

3

2776

CH

3

CH

3

NO

2

CH

3

SCH

3

2777

CH

2

CH

3

CH

2

CH

3

NO

2

CH

3

SCH

3

2778

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

CH

3

SCH

3

2779

OCH

3

OCH

3

NO

2

CH

3

SCH

3

2780

OCH

2

CH

3

OCH

2

CH

3

NO

2

CH

3

SCH

3

2781

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

CH

3

SCH

3

2782

SCH

3

SCH

3

NO

2

CH

3

SCH

3

2783

SCH

2

CH

3

SCH

2

CH

3

NO

2

CH

3

SCH

3

2784

N(CH

3

)

2

N(CH

3

)

2

NO

2

CH

3

SCH

3

2785

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

CH

3

SCH

3

2786

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

CH

3

SCH

3

2787

O—(CH

2

CH

2

)—O

NO

2

CH

3

SCH

3

2788

O—(CH

2

CH

2

CH

2

)—O

NO

2

CH

3

SCH

3

2789

S—(CH

2

CH

2

)—S

NO

2

CH

3

SCH

3

2790

S—(CH

2

CH

2

CH

2

)—S

NO

2

CH

3

SCH

3

2791

—(CH

2

)

4

—

NO

2

CH

3

SCH

3

2792

—(CH

2

)

5

—

NO

2

CH

3

SCH

3

2793

H

H

CN

CH

3

SCH

3

2794

CH

3

CH

3

CN

CH

3

SCH

3

2795

CH

2

CH

3

CH

2

CH

3

CN

CH

3

SCH

3

2796

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

CH

3

SCH

3

2797

OCH

3

OCH

3

CN

CH

3

SCH

3

2798

OCH

2

CH

3

OCH

2

CH

3

CN

CH

3

SCH

3

2799

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

CH

3

SCH

3

2800

SCH

3

SCH

3

CN

CH

3

SCH

3

2801

SCH

2

CH

3

SCH

2

CH

3

CN

CH

3

SCH

3

2802

N(CH

3

)

2

N(CH

3

)

2

CN

CH

3

SCH

3

2803

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

CH

3

SCH

3

2804

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

CH

3

SCH

3

2805

O—(CH

2

CH

2

)—O

CN

CH

3

SCH

3

2806

O—(CH

2

CH

2

CH

2

)—O

CN

CH

3

SCH

3

2807

S—(CH

2

CH

2

)—S

CN

CH

3

SCH

3

2808

S—(CH

2

CH

2

CH

2

)—S

CN

CH

3

SCH

3

2809

—(CH

2

)

4

—

CN

CH

3

SCH

3

2810

—(CH

2

)

5

—

CN

CH

3

SCH

3

2811

H

H

F

CH

3

SCH

3

2812

CH

3

CH

3

F

CH

3

SCH

3

2813

CH

2

CH

3

CH

2

CH

3

F

CH

3

SCH

3

2814

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

CH

3

SCH

3

2815

OCH

3

OCH

3

F

CH

3

SCH

3

2816

OCH

2

CH

3

OCH

2

CH

3

F

CH

3

SCH

3

2817

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

CH

3

SCH

3

2818

SCH

3

SCH

3

F

CH

3

SCH

3

2819

SCH

2

CH

3

SCH

2

CH

3

F

CH

3

SCH

3

2820

N(CH

3

)

2

N(CH

3

)

2

F

CH

3

SCH

3

2821

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

CH

3

SCH

3

2822

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

CH

3

SCH

3

2823

O—(CH

2

CH

2

)—O

F

CH

3

SCH

3

2824

O—(CH

2

CH

2

CH

2

)—O

F

CH

3

SCH

3

2825

S—(CH

2

CH

2

)—S

F

CH

3

SCH

3

2826

S—(CH

2

CH

2

CH

2

)—S

F

CH

3

SCH

3

2827

—(CH

2

)

4

—

F

CH

3

SCH

3

2828

—(CH

2

)

5

—

F

CH

3

SCH

3

2829

H

H

Cl

CH

3

SCH

3

2830

CH

3

CH

3

Cl

CH

3

SCH

3

2831

CH

2

CH

3

CH

2

CH

3

Cl

CH

3

SCH

3

2832

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

CH

3

SCH

3

2833

OCH

3

OCH

3

Cl

CH

3

SCH

3

2834

OCH

2

CH

3

OCH

2

CH

3

Cl

CH

3

SCH

3

2835

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

CH

3

SCH

3

2836

SCH

3

SCH

3

Cl

CH

3

SCH

3

2837

SCH

2

CH

3

SCH

2

CH

3

Cl

CH

3

SCH

3

2838

N(CH

3

)

2

N(CH

3

)

2

Cl

CH

3

SCH

3

2839

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

CH

3

SCH

3

2840

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

CH

3

SCH

3

2841

O—(CH

2

CH

2

)—O

Cl

CH

3

SCH

3

2842

O—(CH

2

CH

2

CH

2

)—O

Cl

CH

3

SCH

3

2843

S—(CH

2

CH

2

)—S

Cl

CH

3

SCH

3

2844

S—(CH

2

CH

2

CH

2

)—S

Cl

CH

3

SCH

3

2845

—(CH

2

)

4

—

Cl

CH

3

SCH

3

2846

—(CH

2

)

5

—

Cl

CH

3

SCH

3

2847

H

H

Br

CH

3

SCH

3

2848

CH

3

CH

3

Br

CH

3

SCH

3

2849

CH

2

CH

3

CH

2

CH

3

Br

CH

3

SCH

3

2850

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

CH

3

SCH

3

2851

OCH

3

OCH

3

Br

CH

3

SCH

3

2852

OCH

2

CH

3

OCH

2

CH

3

Br

CH

3

SCH

3

2853

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

CH

3

SCH

3

2854

SCH

3

SCH

3

Br

CH

3

SCH

3

2855

SCH

2

CH

3

SCH

2

CH

3

Br

CH

3

SCH

3

2856

N(CH

3

)

2

N(CH

3

)

2

Br

CH

3

SCH

3

2857

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

CH

3

SCH

3

2858

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

CH

3

SCH

3

2859

O—(CH

2

CH

2

)—O

Br

CH

3

SCH

3

2860

O—(CH

2

CH

2

CH

2

)—O

Br

CH

3

SCH

3

2861

S—(CH

2

CH

2

)—S

Br

CH

3

SCH

3

2862

S—(CH

2

CH

2

CH

2

)—S

Br

CH

3

SCH

3

2863

—(CH

2

)

4

—

Br

CH

3

SCH

3

2864

—(CH

2

)

5

—

Br

CH

3

SCH

3

2865

H

H

CH

3

CH

3

SCH

3

2866

CH

3

CH

3

CH

3

CH

3

SCH

3

2867

CH

2

CH

3

CH

2

CH

3

CH

3

CH

3

SCH

3

2868

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

CH

3

SCH

3

2869

OCH

3

OCH

3

CH

3

CH

3

SCH

3

2870

OCH

2

CH

3

OCH

2

CH

3

CH

3

CH

3

SCH

3

2871

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

CH

3

SCH

3

2872

SCH

3

SCH

3

CH

3

CH

3

SCH

3

2873

SCH

2

CH

3

SCH

2

CH

3

CH

3

CH

3

SCH

3

2874

N(CH

3

)

2

N(CH

3

)

2

CH

3

CH

3

SCH

3

2875

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

CH

3

SCH

3

2876

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

CH

3

SCH

3

2877

O—(CH

2

CH

2

)—O

CH

3

CH

3

SCH

3

2878

O—(CH

2

CH

2

CH

2

)—O

CH

3

CH

3

SCH

3

2879

S—(CH

2

CH

2

)—S

CH

3

CH

3

SCH

3

2880

S—(CH

2

CH

2

CH

2

)—S

CH

3

CH

3

SCH

3

2881

—(CH

2

)

4

—

CH

3

CH

3

SCH

3

2882

—(CH

2

)

5

—

CH

3

CH

3

SCH

3

2883

H

H

CH

2

CH

3

CH

3

SCH

3

2884

CH

3

CH

3

CH

2

CH

3

CH

3

SCH

3

2885

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

CH

3

SCH

3

2886

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

CH

3

SCH

3

2887

OCH

3

OCH

3

CH

2

CH

3

CH

3

SCH

3

2888

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

CH

3

SCH

3

2889

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

CH

3

SCH

3

2890

SCH

3

SCH

3

CH

2

CH

3

CH

3

SCH

3

2891

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

CH

3

SCH

3

2892

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

CH

3

SCH

3

2893

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

CH

3

SCH

3

2894

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

CH

3

SCH

3

2895

O—(CH

2

CH

2

)—O

CH

2

CH

3

CH

3

SCH

3

2896

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

CH

3

SCH

3

2897

S—(CH

2

CH

2

)—S

CH

2

CH

3

CH

3

SCH

3

2898

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

CH

3

SCH

3

2899

—(CH

2

)

4

—

CH

2

CH

3

CH

3

SCH

3

2900

—(CH

2

)

5

—

CH

2

CH

3

CH

3

SCH

3

2901

H

H

CF

3

CH

3

SCH

3

2902

CH

3

CH

3

CF

3

CH

3

SCH

3

2903

CH

2

CH

3

CH

2

CH

3

CF

3

CH

3

SCH

3

2904

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

CH

3

SCH

3

2905

OCH

3

OCH

3

CF

3

CH

3

SCH

3

2906

OCH

2

CH

3

OCH

2

CH

3

CF

3

CH

3

SCH

3

2907

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

CH

3

SCH

3

2908

SCH

3

SCH

3

CF

3

CH

3

SCH

3

2909

SCH

2

CH

3

SCH

2

CH

3

CF

3

CH

3

SCH

3

2910

N(CH

3

)

2

N(CH

3

)

2

CF

3

CH

3

SCH

3

2911

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

CH

3

SCH

3

2912

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

CH

3

SCH

3

2913

O—(CH

2

CH

2

)—O

CF

3

CH

3

SCH

3

2914

O—(CH

2

CH

2

CH

2

)—O

CF

3

CH

3

SCH

3

2915

S—(CH

2

CH

2

)—S

CF

3

CH

3

SCH

3

2916

S—(CH

2

CH

2

CH

2

)—S

CF

3

CH

3

SCH

3

2917

—(CH

2

)

4

—

CF

3

CH

3

SCH

3

2918

—(CH

2

)

5

—

CF

3

CH

3

SCH

3

2919

H

H

OCH

3

CH

3

SCH

3

2920

CH

3

CH

3

OCH

3

CH

3

SCH

3

2921

CH

2

CH

3

CH

2

CH

3

OCH

3

CH

3

SCH

3

2922

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

CH

3

SCH

3

2923

OCH

3

OCH

3

OCH

3

CH

3

SCH

3

2924

OCH

2

CH

3

OCH

2

CH

3

OCH

3

CH

3

SCH

3

2925

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

CH

3

SCH

3

2926

SCH

3

SCH

3

OCH

3

CH

3

SCH

3

2927

SCH

2

CH

3

SCH

2

CH

3

OCH

3

CH

3

SCH

3

2928

N(CH

3

)

2

N(CH

3

)

2

OCH

3

CH

3

SCH

3

2929

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

CH

3

SCH

3

2930

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

CH

3

SCH

3

2931

O—(CH

2

CH

2

)—O

OCH

3

CH

3

SCH

3

2932

O—(CH

2

CH

2

CH

2

)—O

OCH

3

CH

3

SCH

3

2933

S—(CH

2

CH

2

)—S

OCH

3

CH

3

SCH

3

2934

S—(CH

2

CH

2

CH

2

)—S

OCH

3

CH

3

SCH

3

2935

—(CH

2

)

4

—

OCH

3

CH

3

SCH

3

2936

—(CH

2

)

5

—

OCH

3

CH

3

SCH

3

2937

H

H

OCH

2

CH

3

CH

3

SCH

3

2938

CH

3

CH

3

OCH

2

CH

3

CH

3

SCH

3

2939

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

CH

3

SCH

3

2940

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

CH

3

SCH

3

2941

OCH

3

OCH

3

OCH

2

CH

3

CH

3

SCH

3

2942

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

CH

3

SCH

3

2943

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

CH

3

SCH

3

2944

SCH

3

SCH

3

OCH

2

CH

3

CH

3

SCH

3

2945

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

CH

3

SCH

3

2946

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

CH

3

SCH

3

2947

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

CH

3

SCH

3

2948

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

CH

3

SCH

3

2949

O—(CH

2

CH

2

)—O

OCH

2

CH

3

CH

3

SCH

3

2950

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

CH

3

SCH

3

2951

S—(CH

2

CH

2

)—S

OCH

2

CH

3

CH

3

SCH

3

2952

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

CH

3

SCH

3

2953

—(CH

2

)

4

—

OCH

2

CH

3

CH

3

SCH

3

2954

—(CH

2

)

5

—

OCH

2

CH

3

CH

3

SCH

3

2955

H

H

SCH

3

CH

3

SCH

3

2956

CH

3

CH

3

SCH

3

CH

3

SCH

3

2957

CH

2

CH

3

CH

2

CH

3

SCH

3

CH

3

SCH

3

2958

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

CH

3

SCH

3

2959

OCH

3

OCH

3

SCH

3

CH

3

SCH

3

2960

OCH

2

CH

3

OCH

2

CH

3

SCH

3

CH

3

SCH

3

2961

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

CH

3

SCH

3

2962

SCH

3

SCH

3

SCH

3

CH

3

SCH

3

2963

SCH

2

CH

3

SCH

2

CH

3

SCH

3

CH

3

SCH

3

2964

N(CH

3

)

2

N(CH

3

)

2

SCH

3

CH

3

SCH

3

2965

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

CH

3

SCH

3

2966

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

CH

3

SCH

3

2967

O—(CH

2

CH

2

)—O

SCH

3

CH

3

SCH

3

2968

O—(CH

2

CH

2

CH

2

)—O

SCH

3

CH

3

SCH

3

2969

S—(CH

2

CH

2

)—S

SCH

3

CH

3

SCH

3

2970

S—(CH

2

CH

2

CH

2

)—S

SCH

3

CH

3

SCH

3

2971

—(CH

2

)

4

—

SCH

3

CH

3

SCH

3

2972

—(CH

2

)

5

—

SCH

3

CH

3

SCH

3

2973

H

H

SO

2

CH

3

CH

3

SCH

3

2974

CH

3

CH

3

SO

2

CH

3

CH

3

SCH

3

2975

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

CH

3

SCH

3

2976

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

CH

3

SCH

3

2977

OCH

3

OCH

3

SO

2

CH

3

CH

3

SCH

3

2978

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

CH

3

SCH

3

2979

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

CH

3

SCH

3

2980

SCH

3

SCH

3

SO

2

CH

3

CH

3

SCH

3

2981

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

CH

3

SCH

3

2982

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

CH

3

SCH

3

2983

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

CH

3

SCH

3

2984

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

CH

3

SCH

3

2985

O—(CH

2

CH

2

)—O

SO

2

CH

3

CH

3

SCH

3

2986

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

CH

3

SCH

3

2987

S—(CH

2

CH

2

)—S

SO

2

CH

3

CH

3

SCH

3

2988

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

CH

3

SCH

3

2989

—(CH

2

)

4

—

SO

2

CH

3

CH

3

SCH

3

2990

—(CH

2

)

5

—

SO

2

CH

3

CH

3

SCH

3

2991

H

H

PO(OCH

3

)

2

CH

3

SCH

3

2992

CH

3

CH

3

PO(OCH

3

)

2

CH

3

SCH

3

2993

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

CH

3

SCH

3

2994

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

CH

3

SCH

3

2995

OCH

3

OCH

3

PO(OCH

3

)

2

CH

3

SCH

3

2996

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

CH

3

SCH

3

2997

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

CH

3

SCH

3

2998

SCH

3

SCH

3

PO(OCH

3

)

2

CH

3

SCH

3

2999

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

CH

3

SCH

3

3000

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

CH

3

SCH

3

3001

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

CH

3

SCH

3

3002

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

CH

3

SCH

3

3003

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

CH

3

SCH

3

3004

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

CH

3

SCH

3

3005

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

CH

3

SCH

3

3006

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

CH

3

SCH

3

3007

—(CH

2

)

4

—

PO(OCH

3

)

2

CH

3

SCH

3

3008

—(CH

2

)

5

—

PO(OCH

3

)

2

CH

3

SCH

3

3009

H

H

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3010

CH

3

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3011

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3012

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3013

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3014

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3015

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3016

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3017

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3018

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3019

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3020

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3021

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3022

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3023

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3024

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3025

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3026

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

CH

3

SCH

3

3027

H

H

PO(CH

3

)

2

CH

3

SCH

3

3028

CH

3

CH

3

PO(CH

3

)

2

CH

3

SCH

3

3029

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

CH

3

SCH

3

3030

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

CH

3

SCH

3

3031

OCH

3

OCH

3

PO(CH

3

)

2

CH

3

SCH

3

3032

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

CH

3

SCH

3

3033

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

CH

3

SCH

3

3034

SCH

3

SCH

3

PO(CH

3

)

2

CH

3

SCH

3

3035

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

CH

3

SCH

3

3036

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

CH

3

SCH

3

3037

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

CH

3

SCH

3

3038

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

CH

3

SCH

3

3039

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

CH

3

SCH

3

3040

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

CH

3

SCH

3

3041

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

CH

3

SCH

3

3042

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

CH

3

SCH

3

3043

—(CH

2

)

4

—

PO(CH

3

)

2

CH

3

SCH

3

3044

—(CH

2

)

5

—

PO(CH

3

)

2

CH

3

SCH

3

3045

H

H

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3046

CH

3

CH

3

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3047

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3048

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3049

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3050

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3051

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3052

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3053

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3054

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3055

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3056

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3057

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3058

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3059

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3060

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3061

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3062

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

CH

3

SCH

3

3063

H

H

H

CH

3

SC

6

H

5

3064

CH

3

CH

3

H

CH

3

SC

6

H

5

3065

CH

2

CH

3

CH

2

CH

3

H

CH

3

SC

6

H

5

3066

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

CH

3

SC

6

H

5

3067

OCH

3

OCH

3

H

CH

3

SC

6

H

5

3068

OCH

2

CH

3

OCH

2

CH

3

H

CH

3

SC

6

H

5

3069

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

CH

3

SC

6

H

5

3070

SCH

3

SCH

3

H

CH

3

SC

6

H

5

3071

SCH

2

CH

3

SCH

2

CH

3

H

CH

3

SC

6

H

5

3072

N(CH

3

)

2

N(CH

3

)

2

H

CH

3

SC

6

H

5

3073

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

CH

3

SC

6

H

5

3074

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

CH

3

SC

6

H

5

3075

O—(CH

2

CH

2

)—O

H

CH

3

SC

6

H

5

3076

O—(CH

2

CH

2

CH

2

)—O

H

CH

3

SC

6

H

5

3077

S—(CH

2

CH

2

)—S

H

CH

3

SC

6

H

5

3078

S—(CH

2

CH

2

CH

2

)—S

H

CH

3

SC

6

H

5

3079

—(CH

2

)

4

—

H

CH

3

SC

6

H

5

3080

—(CH

2

)

5

—

H

CH

3

SC

6

H

5

3081

H

H

NO

2

CH

3

SC

6

H

5

3082

CH

3

CH

3

NO

2

CH

3

SC

6

H

5

3083

CH

2

CH

3

CH

2

CH

3

NO

2

CH

3

SC

6

H

5

3084

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

CH

3

SC

6

H

5

3085

OCH

3

OCH

3

NO

2

CH

3

SC

6

H

5

3086

OCH

2

CH

3

OCH

2

CH

3

NO

2

CH

3

SC

6

H

5

3087

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

CH

3

SC

6

H

5

3088

SCH

3

SCH

3

NO

2

CH

3

SC

6

H

5

3089

SCH

2

CH

3

SCH

2

CH

3

NO

2

CH

3

SC

6

H

5

3090

N(CH

3

)

2

N(CH

3

)

2

NO

2

CH

3

SC

6

H

5

3091

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

CH

3

SC

6

H

5

3092

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

CH

3

SC

6

H

5

3093

O—(CH

2

CH

2

)—O

NO

2

CH

3

SC

6

H

5

3094

O—(CH

2

CH

2

CH

2

)—O

NO

2

CH

3

SC

6

H

5

3095

S—(CH

2

CH

2

)—S

NO

2

CH

3

SC

6

H

5

3096

S—(CH

2

CH

2

CH

2

)—S

NO

2

CH

3

SC

6

H

5

3097

—(CH

2

)

4

—

NO

2

CH

3

SC

6

H

5

3098

—(CH

2

)

5

—

NO

2

CH

3

SC

6

H

5

3099

H

H

CN

CH

3

SC

6

H

5

3100

CH

3

CH

3

CN

CH

3

SC

6

H

5

3101

CH

2

CH

3

CH

2

CH

3

CN

CH

3

SC

6

H

5

3102

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

CH

3

SC

6

H

5

3103

OCH

3

OCH

3

CN

CH

3

SC

6

H

5

3104

OCH

2

CH

3

OCH

2

CH

3

CN

CH

3

SC

6

H

5

3105

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

CH

3

SC

6

H

5

3106

SCH

3

SCH

3

CN

CH

3

SC

6

H

5

3107

SCH

2

CH

3

SCH

2

CH

3

CN

CH

3

SC

6

H

5

3108

N(CH

3

)

2

N(CH

3

)

2

CN

CH

3

SC

6

H

5

3109

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

CH

3

SC

6

H

5

3110

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

CH

3

SC

6

H

5

3111

O—(CH

2

CH

2

)—O

CN

CH

3

SC

6

H

5

3112

O—(CH

2

CH

2

CH

2

)—O

CN

CH

3

SC

6

H

5

3113

S—(CH

2

CH

2

)—S

CN

CH

3

SC

6

H

5

3114

S—(CH

2

CH

2

CH

2

)—S

CN

CH

3

SC

6

H

5

3115

—(CH

2

)

4

—

CN

CH

3

SC

6

H

5

3116

—(CH

2

)

5

—

CN

CH

3

SC

6

H

5

3117

H

H

F

CH

3

SC

6

H

5

3118

CH

3

CH

3

F

CH

3

SC

6

H

5

3119

CH

2

CH

3

CH

2

CH

3

F

CH

3

SC

6

H

5

3120

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

CH

3

SC

6

H

5

3121

OCH

3

OCH

3

F

CH

3

SC

6

H

5

3122

OCH

2

CH

3

OCH

2

CH

3

F

CH

3

SC

6

H

5

3123

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

CH

3

SC

6

H

5

3124

SCH

3

SCH

3

F

CH

3

SC

6

H

5

3125

SCH

2

CH

3

SCH

2

CH

3

F

CH

3

SC

6

H

5

3126

N(CH

3

)

2

N(CH

3

)

2

F

CH

3

SC

6

H

5

3127

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

CH

3

SC

6

H

5

3128

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

CH

3

SC

6

H

5

3129

O—(CH

2

CH

2

)—O

F

CH

3

SC

6

H

5

3130

O—(CH

2

CH

2

CH

2

)—O

F

CH

3

SC

6

H

5

3131

S—(CH

2

CH

2

)—S

F

CH

3

SC

6

H

5

3132

S—(CH

2

CH

2

CH

2

)—S

F

CH

3

SC

6

H

5

3133

—(CH

2

)

4

—

F

CH

3

SC

6

H

5

3134

—(CH

2

)

5

—

F

CH

3

SC

6

H

5

3135

H

H

Cl

CH

3

SC

6

H

5

3136

CH

3

CH

3

Cl

CH

3

SC

6

H

5

3137

CH

2

CH

3

CH

2

CH

3

Cl

CH

3

SC

6

H

5

3138

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

CH

3

SC

6

H

5

3139

OCH

3

OCH

3

Cl

CH

3

SC

6

H

5

3140

OCH

2

CH

3

OCH

2

CH

3

Cl

CH

3

SC

6

H

5

3141

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

CH

3

SC

6

H

5

3142

SCH

3

SCH

3

Cl

CH

3

SC

6

H

5

3143

SCH

2

CH

3

SCH

2

CH

3

Cl

CH

3

SC

6

H

5

3144

N(CH

3

)

2

N(CH

3

)

2

Cl

CH

3

SC

6

H

5

3145

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

CH

3

SC

6

H

5

3146

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

CH

3

SC

6

H

5

3147

O—(CH

2

CH

2

)—O

Cl

CH

3

SC

6

H

5

3148

O—(CH

2

CH

2

CH

2

)—O

Cl

CH

3

SC

6

H

5

3149

S—(CH

2

CH

2

)—S

Cl

CH

3

SC

6

H

5

3150

S—(CH

2

CH

2

CH

2

)—S

Cl

CH

3

SC

6

H

5

3151

—(CH

2

)

4

—

Cl

CH

3

SC

6

H

5

3152

—(CH

2

)

5

—

Cl

CH

3

SC

6

H

5

3153

H

H

Br

CH

3

SC

6

H

5

3154

CH

3

CH

3

Br

CH

3

SC

6

H

5

3155

CH

2

CH

3

CH

2

CH

3

Br

CH

3

SC

6

H

5

3156

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

CH

3

SC

6

H

5

3157

OCH

3

OCH

3

Br

CH

3

SC

6

H

5

3158

OCH

2

CH

3

OCH

2

CH

3

Br

CH

3

SC

6

H

5

3159

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

CH

3

SC

6

H

5

3160

SCH

3

SCH

3

Br

CH

3

SC

6

H

5

3161

SCH

2

CH

3

SCH

2

CH

3

Br

CH

3

SC

6

H

5

3162

N(CH

3

)

2

N(CH

3

)

2

Br

CH

3

SC

6

H

5

3163

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

CH

3

SC

6

H

5

3164

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

CH

3

SC

6

H

5

3165

O—(CH

2

CH

2

)—O

Br

CH

3

SC

6

H

5

3166

O—(CH

2

CH

2

CH

2

)—O

Br

CH

3

SC

6

H

5

3167

S—(CH

2

CH

2

)—S

Br

CH

3

SC

6

H

5

3168

S—(CH

2

CH

2

CH

2

)—S

Br

CH

3

SC

6

H

5

3169

—(CH

2

)

4

—

Br

CH

3

SC

6

H

5

3170

—(CH

2

)

5

—

Br

CH

3

SC

6

H

5

3171

H

H

CH

3

CH

3

SC

6

H

5

3172

CH

3

CH

3

CH

3

CH

3

SC

6

H

5

3173

CH

2

CH

3

CH

2

CH

3

CH

3

CH

3

SC

6

H

5

3174

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

CH

3

SC

6

H

5

3175

OCH

3

OCH

3

CH

3

CH

3

SC

6

H

5

3176

OCH

2

CH

3

OCH

2

CH

3

CH

3

CH

3

SC

6

H

5

3177

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

CH

3

SC

6

H

5

3178

SCH

3

SCH

3

CH

3

CH

3

SC

6

H

5

3179

SCH

2

CH

3

SCH

2

CH

3

CH

3

CH

3

SC

6

H

5

3180

N(CH

3

)

2

N(CH

3

)

2

CH

3

CH

3

SC

6

H

5

3181

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

CH

3

SC

6

H

5

3182

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

CH

3

SC

6

H

5

3183

O—(CH

2

CH

2

)—O

CH

3

CH

3

SC

6

H

5

3184

O—(CH

2

CH

2

CH

2

)—O

CH

3

CH

3

SC

6

H

5

3185

S—(CH

2

CH

2

)—S

CH

3

CH

3

SC

6

H

5

3186

S—(CH

2

CH

2

CH

2

)—S

CH

3

CH

3

SC

6

H

5

3187

—(CH

2

)

4

—

CH

3

CH

3

SC

6

H

5

3188

—(CH

2

)

5

—

CH

3

CH

3

SC

6

H

5

3189

H

H

CH

2

CH

3

CH

3

SC

6

H

5

3190

CH

3

CH

3

CH

2

CH

3

CH

3

SC

6

H

5

3191

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

CH

3

SC

6

H

5

3192

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

CH

3

SC

6

H

5

3193

OCH

3

OCH

3

CH

2

CH

3

CH

3

SC

6

H

5

3194

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

CH

3

SC

6

H

5

3195

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

CH

3

SC

6

H

5

3196

SCH

3

SCH

3

CH

2

CH

3

CH

3

SC

6

H

5

3197

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

CH

3

SC

6

H

5

3198

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

CH

3

SC

6

H

5

3199

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

CH

3

SC

6

H

5

3200

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

CH

3

SC

6

H

5

3201

O—(CH

2

CH

2

)—O

CH

2

CH

3

CH

3

SC

6

H

5

3202

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

CH

3

SC

6

H

5

3203

S—(CH

2

CH

2

)—S

CH

2

CH

3

CH

3

SC

6

H

5

3204

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

CH

3

SC

6

H

5

3205

—(CH

2

)

4

—

CH

2

CH

3

CH

3

SC

6

H

5

3206

—(CH

2

)

5

—

CH

2

CH

3

CH

3

SC

6

H

5

3207

H

H

CF

3

CH

3

SC

6

H

5

3208

CH

3

CH

3

CF

3

CH

3

SC

6

H

5

3209

CH

2

CH

3

CH

2

CH

3

CF

3

CH

3

SC

6

H

5

3210

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

CH

3

SC

6

H

5

3211

OCH

3

OCH

3

CF

3

CH

3

SC

6

H

5

3212

OCH

2

CH

3

OCH

2

CH

3

CF

3

CH

3

SC

6

H

5

3213

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

CH

3

SC

6

H

5

3214

SCH

3

SCH

3

CF

3

CH

3

SC

6

H

5

3215

SCH

2

CH

3

SCH

2

CH

3

CF

3

CH

3

SC

6

H

5

3216

N(CH

3

)

2

N(CH

3

)

2

CF

3

CH

3

SC

6

H

5

3217

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

CH

3

SC

6

H

5

3218

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

CH

3

SC

6

H

5

3219

O—(CH

2

CH

2

)—O

CF

3

CH

3

SC

6

H

5

3220

O—(CH

2

CH

2

CH

2

)—O

CF

3

CH

3

SC

6

H

5

3221

S—(CH

2

CH

2

)—S

CF

3

CH

3

SC

6

H

5

3222

S—(CH

2

CH

2

CH

2

)—S

CF

3

CH

3

SC

6

H

5

3223

—(CH

2

)

4

—

CF

3

CH

3

SC

6

H

5

3224

—(CH

2

)

5

—

CF

3

CH

3

SC

6

H

5

3225

H

H

OCH

3

CH

3

SC

6

H

5

3226

CH

3

CH

3

OCH

3

CH

3

SC

6

H

5

3227

CH

2

CH

3

CH

2

CH

3

OCH

3

CH

3

SC

6

H

5

3228

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

CH

3

SC

6

H

5

3229

OCH

3

OCH

3

OCH

3

CH

3

SC

6

H

5

3230

OCH

2

CH

3

OCH

2

CH

3

OCH

3

CH

3

SC

6

H

5

3231

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

CH

3

SC

6

H

5

3232

SCH

3

SCH

3

OCH

3

CH

3

SC

6

H

5

3233

SCH

2

CH

3

SCH

2

CH

3

OCH

3

CH

3

SC

6

H

5

3234

N(CH

3

)

2

N(CH

3

)

2

OCH

3

CH

3

SC

6

H

5

3235

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

CH

3

SC

6

H

5

3236

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

CH

3

SC

6

H

5

3237

O—(CH

2

CH

2

)—O

OCH

3

CH

3

SC

6

H

5

3238

O—(CH

2

CH

2

CH

2

)—O

OCH

3

CH

3

SC

6

H

5

3239

S—(CH

2

CH

2

)—S

OCH

3

CH

3

SC

6

H

5

3240

S—(CH

2

CH

2

CH

2

)—S

OCH

3

CH

3

SC

6

H

5

3241

—(CH

2

)

4

—

OCH

3

CH

3

SC

6

H

5

3242

—(CH

2

)

5

—

OCH

3

CH

3

SC

6

H

5

3243

H

H

OCH

2

CH

3

CH

3

SC

6

H

5

3244

CH

3

CH

3

OCH

2

CH

3

CH

3

SC

6

H

5

3245

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

CH

3

SC

6

H

5

3246

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

CH

3

SC

6

H

5

3247

OCH

3

OCH

3

OCH

2

CH

3

CH

3

SC

6

H

5

3248

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

CH

3

SC

6

H

5

3249

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

CH

3

SC

6

H

5

3250

SCH

3

SCH

3

OCH

2

CH

3

CH

3

SC

6

H

5

3251

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

CH

3

SC

6

H

5

3252

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

CH

3

SC

6

H

5

3253

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

CH

3

SC

6

H

5

3254

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

CH

3

SC

6

H

5

3255

O—(CH

2

CH

2

)—O

OCH

2

CH

3

CH

3

SC

6

H

5

3256

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

CH

3

SC

6

H

5

3257

S—(CH

2

CH

2

)—S

OCH

2

CH

3

CH

3

SC

6

H

5

3258

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

CH

3

SC

6

H

5

3259

—(CH

2

)

4

—

OCH

2

CH

3

CH

3

SC

6

H

5

3260

—(CH

2

)

5

—

OCH

2

CH

3

CH

3

SC

6

H

5

3261

H

H

SCH

3

CH

3

SC

6

H

5

3262

CH

3

CH

3

SCH

3

CH

3

SC

6

H

5

3263

CH

2

CH

3

CH

2

CH

3

SCH

3

CH

3

SC

6

H

5

3264

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

CH

3

SC

6

H

5

3265

OCH

3

OCH

3

SCH

3

CH

3

SC

6

H

5

3266

OCH

2

CH

3

OCH

2

CH

3

SCH

3

CH

3

SC

6

H

5

3267

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

CH

3

SC

6

H

5

3268

SCH

3

SCH

3

SCH

3

CH

3

SC

6

H

5

3269

SCH

2

CH

3

SCH

2

CH

3

SCH

3

CH

3

SC

6

H

5

3270

N(CH

3

)

2

N(CH

3

)

2

SCH

3

CH

3

SC

6

H

5

3271

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

CH

3

SC

6

H

5

3272

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

CH

3

SC

6

H

5

3273

O—(CH

2

CH

2

)—O

SCH

3

CH

3

SC

6

H

5

3274

O—(CH

2

CH

2

CH

2

)—O

SCH

3

CH

3

SC

6

H

5

3275

S—(CH

2

CH

2

)—S

SCH

3

CH

3

SC

6

H

5

3276

S—(CH

2

CH

2

CH

2

)—S

SCH

3

CH

3

SC

6

H

5

3277

—(CH

2

)

4

—

SCH

3

CH

3

SC

6

H

5

3278

—(CH

2

)

5

—

SCH

3

CH

3

SC

6

H

5

3279

H

H

SO

2

CH

3

CH

3

SC

6

H

5

3280

CH

3

CH

3

SO

2

CH

3

CH

3

SC

6

H

5

3281

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

CH

3

SC

6

H

5

3282

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

CH

3

SC

6

H

5

3283

OCH

3

OCH

3

SO

2

CH

3

CH

3

SC

6

H

5

3284

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

CH

3

SC

6

H

5

3285

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

CH

3

SC

6

H

5

3286

SCH

3

SCH

3

SO

2

CH

3

CH

3

SC

6

H

5

3287

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

CH

3

SC

6

H

5

3288

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

CH

3

SC

6

H

5

3289

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

CH

3

SC

6

H

5

3290

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

CH

3

SC

6

H

5

3291

O—(CH

2

CH

2

)—O

SO

2

CH

3

CH

3

SC

6

H

5

3292

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

CH

3

SC

6

H

5

3293

S—(CH

2

CH

2

)—S

SO

2

CH

3

CH

3

SC

6

H

5

3294

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

CH

3

SC

6

H

5

3295

—(CH

2

)

4

—

SO

2

CH

3

CH

3

SC

6

H

5

3296

—(CH

2

)

5

—

SO

2

CH

3

CH

3

SC

6

H

5

3297

H

H

PO(OCH

3

)

2

CH

3

SC

6

H

5

3298

CH

3

CH

3

PO(OCH

3

)

2

CH

3

SC

6

H

5

3299

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

CH

3

SC

6

H

5

3300

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

CH

3

SC

6

H

5

3301

OCH

3

OCH

3

PO(OCH

3

)

2

CH

3

SC

6

H

5

3302

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

CH

3

SC

6

H

5

3303

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

CH

3

SC

6

H

5

3304

SCH

3

SCH

3

PO(OCH

3

)

2

CH

3

SC

6

H

5

3305

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

CH

3

SC

6

H

5

3306

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

CH

3

SC

6

H

5

3307

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

CH

3

SC

6

H

5

3308

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

CH

3

SC

6

H

5

3309

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

CH

3

SC

6

H

5

3310

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

CH

3

SC

6

H

5

3311

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

CH

3

SC

6

H

5

3312

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

CH

3

SC

6

H

5

3313

—(CH

2

)

4

—

PO(OCH

3

)

2

CH

3

SC

6

H

5

3314

—(CH

2

)

5

—

PO(OCH

3

)

2

CH

3

SC

6

H

5

3315

H

H

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3316

CH

3

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3317

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3318

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3319

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3320

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3321

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3322

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3323

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3324

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3325

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3326

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3327

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3328

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3329

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3330

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3331

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3332

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

CH

3

SC

6

H

5

3333

H

H

PO(CH

3

)

2

CH

3

SC

6

H

5

3334

CH

3

CH

3

PO(CH

3

)

2

CH

3

SC

6

H

5

3335

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

CH

3

SC

6

H

5

3336

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

CH

3

SC

6

H

5

3337

OCH

3

OCH

3

PO(CH

3

)

2

CH

3

SC

6

H

5

3338

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

CH

3

SC

6

H

5

3339

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

CH

3

SC

6

H

5

3340

SCH

3

SCH

3

PO(CH

3

)

2

CH

3

SC

6

H

5

3341

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

CH

3

SC

6

H

5

3342

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

CH

3

SC

6

H

5

3343

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

CH

3

SC

6

H

5

3344

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

CH

3

SC

6

H

5

3345

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

CH

3

SC

6

H

5

3346

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

CH

3

SC

6

H

5

3347

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

CH

3

SC

6

H

5

3348

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

CH

3

SC

6

H

5

3349

—(CH

2

)

4

—

PO(CH

3

)

2

CH

3

SC

6

H

5

3350

—(CH

2

)

5

—

PO(CH

3

)

2

CH

3

SC

6

H

5

3351

H

H

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3352

CH

3

CH

3

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3353

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3354

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3355

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3356

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3357

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3358

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3359

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3360

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3361

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3362

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3363

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3364

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3365

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3366

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3367

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3368

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

CH

3

SC

6

H

5

3369

H

H

H

CH

3

Het1

3370

CH

3

CH

3

H

CH

3

Het1

3371

CH

2

CH

3

CH

2

CH

3

H

CH

3

Het1

3372

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

CH

3

Het1

3373

OCH

3

OCH

3

H

CH

3

Het1

3374

OCH

2

CH

3

OCH

2

CH

3

H

CH

3

Het1

3375

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

CH

3

Het1

3376

SCH

3

SCH

3

H

CH

3

Het1

3377

SCH

2

CH

3

SCH

2

CH

3

H

CH

3

Het1

3378

N(CH

3

)

2

N(CH

3

)

2

H

CH

3

Het1

3379

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

CH

3

Het1

3380

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

CH

3

Het1

3381

O—(CH

2

CH

2

)—O

H

CH

3

Het1

3382

O—(CH

2

CH

2

CH

2

)—O

H

CH

3

Het1

3383

S—(CH

2

CH

2

)—S

H

CH

3

Het1

3384

S—(CH

2

CH

2

CH

2

)—S

H

CH

3

Het1

3385

—(CH

2

)

4

—

H

CH

3

Het1

3386

—(CH

2

)

5

—

H

CH

3

Het1

3387

H

H

NO

2

CH

3

Het1

3388

CH

3

CH

3

NO

2

CH

3

Het1

3389

CH

2

CH

3

CH

2

CH

3

NO

2

CH

3

Het1

3390

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

CH

3

Het1

3391

OCH

3

OCH

3

NO

2

CH

3

Het1

3392

OCH

2

CH

3

OCH

2

CH

3

NO

2

CH

3

Het1

3393

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

CH

3

Het1

3394

SCH

3

SCH

3

NO

2

CH

3

Het1

3395

SCH

2

CH

3

SCH

2

CH

3

NO

2

CH

3

Het1

3396

N(CH

3

)

2

N(CH

3

)

2

NO

2

CH

3

Het1

3397

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

CH

3

Het1

3398

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

CH

3

Het1

3399

O—(CH

2

CH

2

)—O

NO

2

CH

3

Het1

3400

O—(CH

2

CH

2

CH

2

)—O

NO

2

CH

3

Het1

3401

S—(CH

2

CH

2

)—S

NO

2

CH

3

Het1

3402

S—(CH

2

CH

2

CH

2

)—S

NO

2

CH

3

Het1

3403

—(CH

2

)

4

—

NO

2

CH

3

Het1

3404

—(CH

2

)

5

—

NO

2

CH

3

Het1

3405

H

H

CN

CH

3

Het1

3406

CH

3

CH

3

CN

CH

3

Het1

3407

CH

2

CH

3

CH

2

CH

3

CN

CH

3

Het1

3408

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

CH

3

Het1

3409

OCH

3

OCH

3

CN

CH

3

Het1

3410

OCH

2

CH

3

OCH

2

CH

3

CN

CH

3

Het1

3411

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

CH

3

Het1

3412

SCH

3

SCH

3

CN

CH

3

Het1

3413

SCH

2

CH

3

SCH

2

CH

3

CN

CH

3

Het1

3414

N(CH

3

)

2

N(CH

3

)

2

CN

CH

3

Het1

3415

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

CH

3

Het1

3416

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

CH

3

Het1

3417

O—(CH

2

CH

2

)—O

CN

CH

3

Het1

3418

O—(CH

2

CH

2

CH

2

)—O

CN

CH

3

Het1

3419

S—(CH

2

CH

2

)—S

CN

CH

3

Het1

3420

S—(CH

2

CH

2

CH

2

)—S

CN

CH

3

Het1

3421

—(CH

2

)

4

—

CN

CH

3

Het1

3422

—(CH

2

)

5

—

CN

CH

3

Het1

3423

H

H

F

CH

3

Het1

3424

CH

3

CH

3

F

CH

3

Het1

3425

CH

2

CH

3

CH

2

CH

3

F

CH

3

Het1

3426

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

CH

3

Het1

3427

OCH

3

OCH

3

F

CH

3

Het1

3428

OCH

2

CH

3

OCH

2

CH

3

F

CH

3

Het1

3429

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

CH

3

Het1

3430

SCH

3

SCH

3

F

CH

3

Het1

3431

SCH

2

CH

3

SCH

2

CH

3

F

CH

3

Het1

3432

N(CH

3

)

2

N(CH

3

)

2

F

CH

3

Het1

3433

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

CH

3

Het1

3434

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

CH

3

Het1

3435

O—(CH

2

CH

2

)—O

F

CH

3

Het1

3436

O—(CH

2

CH

2

CH

2

)—O

F

CH

3

Het1

3437

S—(CH

2

CH

2

)—S

F

CH

3

Het1

3438

S—(CH

2

CH

2

CH

2

)—S

F

CH

3

Het1

3439

—(CH

2

)

4

—

F

CH

3

Het1

3440

—(CH

2

)

5

—

F

CH

3

Het1

3441

H

H

Cl

CH

3

Het1

3442

CH

3

CH

3

Cl

CH

3

Het1

3443

CH

2

CH

3

CH

2

CH

3

Cl

CH

3

Het1

3444

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

CH

3

Het1

3445

OCH

3

OCH

3

Cl

CH

3

Het1

3446

OCH

2

CH

3

OCH

2

CH

3

Cl

CH

3

Het1

3447

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

CH

3

Het1

3448

SCH

3

SCH

3

Cl

CH

3

Het1

3449

SCH

2

CH

3

SCH

2

CH

3

Cl

CH

3

Het1

3450

N(CH

3

)

2

N(CH

3

)

2

Cl

CH

3

Het1

3451

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

CH

3

Het1

3452

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

CH

3

Het1

3453

O—(CH

2

CH

2

)—O

Cl

CH

3

Het1

3454

O—(CH

2

CH

2

CH

2

)—O

Cl

CH

3

Het1

3455

S—(CH

2

CH

2

)—S

Cl

CH

3

Het1

3456

S—(CH

2

CH

2

CH

2

)—S

Cl

CH

3

Het1

3457

—(CH

2

)

4

—

Cl

CH

3

Het1

3458

—(CH

2

)

5

—

Cl

CH

3

Het1

3459

H

H

Br

CH

3

Het1

3460

CH

3

CH

3

Br

CH

3

Het1

3461

CH

2

CH

3

CH

2

CH

3

Br

CH

3

Het1

3462

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

CH

3

Het1

3463

OCH

3

OCH

3

Br

CH

3

Het1

3464

OCH

2

CH

3

OCH

2

CH

3

Br

CH

3

Het1

3465

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

CH

3

Het1

3466

SCH

3

SCH

3

Br

CH

3

Het1

3467

SCH

2

CH

3

SCH

2

CH

3

Br

CH

3

Het1

3468

N(CH

3

)

2

N(CH

3

)

2

Br

CH

3

Het1

3469

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

CH

3

Het1

3470

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

CH

3

Het1

3471

O—(CH

2

CH

2

)—O

Br

CH

3

Het1

3472

O—(CH

2

CH

2

CH

2

)—O

Br

CH

3

Het1

3473

S—(CH

2

CH

2

)—S

Br

CH

3

Het1

3474

S—(CH

2

CH

2

CH

2

)—S

Br

CH

3

Het1

3475

—(CH

2

)

4

—

Br

CH

3

Het1

3476

—(CH

2

)

5

—

Br

CH

3

Het1

3477

H

H

CH

3

CH

3

Het1

3478

CH

3

CH

3

CH

3

CH

3

Het1

3479

CH

2

CH

3

CH

2

CH

3

CH

3

CH

3

Het1

3480

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

CH

3

Het1

3481

OCH

3

OCH

3

CH

3

CH

3

Het1

3482

OCH

2

CH

3

OCH

2

CH

3

CH

3

CH

3

Het1

3483

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

CH

3

Het1

3484

SCH

3

SCH

3

CH

3

CH

3

Het1

3485

SCH

2

CH

3

SCH

2

CH

3

CH

3

CH

3

Het1

3486

N(CH

3

)

2

N(CH

3

)

2

CH

3

CH

3

Het1

3487

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

CH

3

Het1

3488

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

CH

3

Het1

3489

O—(CH

2

CH

2

)—O

CH

3

CH

3

Het1

3490

O—(CH

2

CH

2

CH

2

)—O

CH

3

CH

3

Het1

3491

S—(CH

2

CH

2

)—S

CH

3

CH

3

Het1

3492

S—(CH

2

CH

2

CH

2

)—S

CH

3

CH

3

Het1

3493

—(CH

2

)

4

—

CH

3

CH

3

Het1

3494

—(CH

2

)

5

—

CH

3

CH

3

Het1

3495

H

H

CH

2

CH

3

CH

3

Het1

3496

CH

3

CH

3

CH

2

CH

3

CH

3

Het1

3497

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

CH

3

Het1

3498

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

CH

3

Het1

3499

OCH

3

OCH

3

CH

2

CH

3

CH

3

Het1

3500

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

CH

3

Het1

3501

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

CH

3

Het1

3502

SCH

3

SCH

3

CH

2

CH

3

CH

3

Het1

3503

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

CH

3

Het1

3504

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

CH

3

Het1

3505

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

CH

3

Het1

3506

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

CH

3

Het1

3507

O—(CH

2

CH

2

)—O

CH

2

CH

3

CH

3

Het1

3508

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

CH

3

Het1

3509

S—(CH

2

CH

2

)—S

CH

2

CH

3

CH

3

Het1

3510

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

CH

3

Het1

3511

—(CH

2

)

4

—

CH

2

CH

3

CH

3

Het1

3512

—(CH

2

)

5

—

CH

2

CH

3

CH

3

Het1

3513

H

H

CF

3

CH

3

Het1

3514

CH

3

CH

3

CF

3

CH

3

Het1

3515

CH

2

CH

3

CH

2

CH

3

CF

3

CH

3

Het1

3516

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

CH

3

Het1

3517

OCH

3

OCH

3

CF

3

CH

3

Het1

3518

OCH

2

CH

3

OCH

2

CH

3

CF

3

CH

3

Het1

3519

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

CH

3

Het1

3520

SCH

3

SCH

3

CF

3

CH

3

Het1

3521

SCH

2

CH

3

SCH

2

CH

3

CF

3

CH

3

Het1

3522

N(CH

3

)

2

N(CH

3

)

2

CF

3

CH

3

Het1

3523

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

CH

3

Het1

3524

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

CH

3

Het1

3525

O—(CH

2

CH

2

)—O

CF

3

CH

3

Het1

3526

O—(CH

2

CH

2

CH

2

)—O

CF

3

CH

3

Het1

3527

S—(CH

2

CH

2

)—S

CF

3

CH

3

Het1

3528

S—(CH

2

CH

2

CH

2

)—S

CF

3

CH

3

Het1

3529

—(CH

2

)

4

—

CF

3

CH

3

Het1

3530

—(CH

2

)

5

—

CF

3

CH

3

Het1

3531

H

H

OCH

3

CH

3

Het1

3532

CH

3

CH

3

OCH

3

CH

3

Het1

3533

CH

2

CH

3

CH

2

CH

3

OCH

3

CH

3

Het1

3534

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

CH

3

Het1

3535

OCH

3

OCH

3

OCH

3

CH

3

Het1

3536

OCH

2

CH

3

OCH

2

CH

3

OCH

3

CH

3

Het1

3537

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

CH

3

Het1

3538

SCH

3

SCH

3

OCH

3

CH

3

Het1

3539

SCH

2

CH

3

SCH

2

CH

3

OCH

3

CH

3

Het1

3540

N(CH

3

)

2

N(CH

3

)

2

OCH

3

CH

3

Het1

3541

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

CH

3

Het1

3542

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

CH

3

Het1

3543

O—(CH

2

CH

2

)—O

OCH

3

CH

3

Het1

3544

O—(CH

2

CH

2

CH

2

)—O

OCH

3

CH

3

Het1

3545

S—(CH

2

CH

2

)—S

OCH

3

CH

3

Het1

3546

S—(CH

2

CH

2

CH

2

)—S

OCH

3

CH

3

Het1

4044

N(CH

3

)

2

N(CH

3

)

2

F

CH

3

Het3

4045

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

CH

3

Het3

4046

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

CH

3

Het3

4047

O—(CH

2

CH

2

)—O

F

CH

3

Het3

4048

O—(CH

2

CH

2

CH

2

)—O

F

CH

3

Het3

4049

S—(CH

2

CH

2

)—S

F

CH

3

Het3

4050

S—(CH

2

CH

2

CH

2

)—S

F

CH

3

Het3

4051

—(CH

2

)

4

—

F

CH

3

Het3

4052

—(CH

2

)

5

—

F

CH

3

Het3

4053

H

H

Cl

CH

3

Het3

4054

CH

3

CH

3

Cl

CH

3

Het3

4055

CH

2

CH

3

CH

2

CH

3

Cl

CH

3

Het3

4056

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

CH

3

Het3

4057

OCH

3

OCH

3

Cl

CH

3

Het3

4058

OCH

2

CH

3

OCH

2

CH

3

Cl

CH

3

Het3

4059

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

CH

3

Het3

4060

SCH

3

SCH

3

Cl

CH

3

Het3

4061

SCH

2

CH

3

SCH

2

CH

3

Cl

CH

3

Het3

4062

N(CH

3

)

2

N(CH

3

)

2

Cl

CH

3

Het3

4063

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

CH

3

Het3

4064

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

CH

3

Het3

4065

O—(CH

2

CH

2

)—O

Cl

CH

3

Het3

4066

O—(CH

2

CH

2

CH

2

)—O

Cl

CH

3

Het3

4067

S—(CH

2

CH

2

)—S

Cl

CH

3

Het3

4068

S—(CH

2

CH

2

CH

2

)—S

Cl

CH

3

Het3

4069

—(CH

2

)

4

—

Cl

CH

3

Het3

4070

—(CH

2

)

5

—

Cl

CH

3

Het3

4071

H

H

Br

CH

3

Het3

4072

CH

3

CH

3

Br

CH

3

Het3

4073

CH

2

CH

3

CH

2

CH

3

Br

CH

3

Het3

4074

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

CH

3

Het3

4075

OCH

3

OCH

3

Br

CH

3

Het3

4076

OCH

2

CH

3

OCH

2

CH

3

Br

CH

3

Het3

4077

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

CH

3

Het3

4078

SCH

3

SCH

3

Br

CH

3

Het3

4079

SCH

2

CH

3

SCH

2

CH

3

Br

CH

3

Het3

4080

N(CH

3

)

2

N(CH

3

)

2

Br

CH

3

Het3

4081

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

CH

3

Het3

4082

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

CH

3

Het3

4083

O—(CH

2

CH

2

)—O

Br

CH

3

Het3

4084

O—(CH

2

CH

2

CH

2

)—O

Br

CH

3

Het3

4085

S—(CH

2

CH

2

)—S

Br

CH

3

Het3

4086

S—(CH

2

CH

2

CH

2

)—S

Br

CH

3

Het3

4087

—(CH

2

)

4

—

Br

CH

3

Het3

4088

—(CH

2

)

5

—

Br

CH

3

Het3

4089

H

H

CH

3

CH

3

Het3

4090

CH

3

CH

3

CH

3

CH

3

Het3

4091

CH

2

CH

3

CH

2

CH

3

CH

3

CH

3

Het3

4092

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

CH

3

Het3

4093

OCH

3

OCH

3

CH

3

CH

3

Het3

4094

OCH

2

CH

3

OCH

2

CH

3

CH

3

CH

3

Het3

4095

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

CH

3

Het3

4096

SCH

3

SCH

3

CH

3

CH

3

Het3

4097

SCH

2

CH

3

SCH

2

CH

3

CH

3

CH

3

Het3

4098

N(CH

3

)

2

N(CH

3

)

2

CH

3

CH

3

Het3

4099

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

CH

3

Het3

4100

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

CH

3

Het3

4101

O—(CH

2

CH

2

)—O

CH

3

CH

3

Het3

4102

O—(CH

2

CH

2

CH

2

)—O

CH

3

CH

3

Het3

4103

S—(CH

2

CH

2

)—S

CH

3

CH

3

Het3

4104

S—(CH

2

CH

2

CH

2

)—S

CH

3

CH

3

Het3

4105

—(CH

2

)

4

—

CH

3

CH

3

Het3

4106

—(CH

2

)

5

—

CH

3

CH

3

Het3

4107

H

H

CH

2

CH

3

CH

3

Het3

4108

CH

3

CH

3

CH

2

CH

3

CH

3

Het3

4109

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

CH

3

Het3

4110

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

CH

3

Het3

4111

OCH

3

OCH

3

CH

2

CH

3

CH

3

Het3

4112

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

CH

3

Het3

4113

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

CH

3

Het3

4114

SCH

3

SCH

3

CH

2

CH

3

CH

3

Het3

4115

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

CH

3

Het3

4116

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

CH

3

Het3

4117

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

CH

3

Het3

4118

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

CH

3

Het3

4119

O—(CH

2

CH

2

)—O

CH

2

CH

3

CH

3

Het3

4120

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

CH

3

Het3

4121

S—(CH

2

CH

2

)—S

CH

2

CH

3

CH

3

Het3

4122

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

CH

3

Het3

4123

—(CH

2

)

4

—

CH

2

CH

3

CH

3

Het3

4124

—(CH

2

)

5

—

CH

2

CH

3

CH

3

Het3

4125

H

H

CF

3

CH

3

Het3

4126

CH

3

CH

3

CF

3

CH

3

Het3

4127

CH

2

CH

3

CH

2

CH

3

CF

3

CH

3

Het3

4128

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

CH

3

Het3

4129

OCH

3

OCH

3

CF

3

CH

3

Het3

4130

OCH

2

CH

3

OCH

2

CH

3

CF

3

CH

3

Het3

4131

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

CH

3

Het3

4132

SCH

3

SCH

3

CF

3

CH

3

Het3

4133

SCH

2

CH

3

SCH

2

CH

3

CF

3

CH

3

Het3

4134

N(CH

3

)

2

N(CH

3

)

2

CF

3

CH

3

Het3

4135

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

CH

3

Het3

4136

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

CH

3

Het3

4137

O—(CH

2

CH

2

)—O

CF

3

CH

3

Het3

4138

O—(CH

2

CH

2

CH

2

)—O

CF

3

CH

3

Het3

4139

S—(CH

2

CH

2

)—S

CF

3

CH

3

Het3

4140

S—(CH

2

CH

2

CH

2

)—S

CF

3

CH

3

Het3

4141

—(CH

2

)

4

—

CF

3

CH

3

Het3

4142

—(CH

2

)

5

—

CF

3

CH

3

Het3

4143

H

H

OCH

3

CH

3

Het3

4144

CH

3

CH

3

OCH

3

CH

3

Het3

4145

CH

2

CH

3

CH

2

CH

3

OCH

3

CH

3

Het3

4146

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

CH

3

Het3

4147

OCH

3

OCH

3

OCH

3

CH

3

Het3

4148

OCH

2

CH

3

OCH

2

CH

3

OCH

3

CH

3

Het3

4149

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

CH

3

Het3

4150

SCH

3

SCH

3

OCH

3

CH

3

Het3

4151

SCH

2

CH

3

SCH

2

CH

3

OCH

3

CH

3

Het3

4152

N(CH

3

)

2

N(CH

3

)

2

OCH

3

CH

3

Het3

4153

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

CH

3

Het3

4154

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

CH

3

Het3

4155

O—(CH

2

CH

2

)—O

OCH

3

CH

3

Het3

4156

O—(CH

2

CH

2

CH

2

)—O

OCH

3

CH

3

Het3

4157

S—(CH

2

CH

2

)—S

OCH

3

CH

3

Het3

4158

S—(CH

2

CH

2

CH

2

)—S

OCH

3

CH

3

Het3

4159

—(CH

2

)

4

—

OCH

3

CH

3

Het3

4160

—(CH

2

)

5

—

OCH

3

CH

3

Het3

4161

H

H

OCH

2

CH

3

CH

3

Het3

4162

CH

3

CH

3

OCH

2

CH

3

CH

3

Het3

4163

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

CH

3

Het3

4164

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

CH

3

Het3

4165

OCH

3

OCH

3

OCH

2

CH

3

CH

3

Het3

4166

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

CH

3

Het3

4167

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

CH

3

Het3

4168

SCH

3

SCH

3

OCH

2

CH

3

CH

3

Het3

4169

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

CH

3

Het3

4170

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

CH

3

Het3

4171

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

CH

3

Het3

4172

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

CH

3

Het3

4173

O—(CH

2

CH

2

)—O

OCH

2

CH

3

CH

3

Het3

4174

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

CH

3

Het3

4175

S—(CH

2

CH

2

)—S

OCH

2

CH

3

CH

3

Het3

4176

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

CH

3

Het3

4177

—(CH

2

)

4

—

OCH

2

CH

3

CH

3

Het3

4178

—(CH

2

)

5

—

OCH

2

CH

3

CH

3

Het3

4179

H

H

SCH

3

CH

3

Het3

4180

CH

3

CH

3

SCH

3

CH

3

Het3

4181

CH

2

CH

3

CH

2

CH

3

SCH

3

CH

3

Het3

4182

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

CH

3

Het3

4183

OCH

3

OCH

3

SCH

3

CH

3

Het3

4184

OCH

2

CH

3

OCH

2

CH

3

SCH

3

CH

3

Het3

4185

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

CH

3

Het3

4186

SCH

3

SCH

3

SCH

3

CH

3

Het3

4187

SCH

2

CH

3

SCH

2

CH

3

SCH

3

CH

3

Het3

4188

N(CH

3

)

2

N(CH

3

)

2

SCH

3

CH

3

Het3

4189

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

CH

3

Het3

4190

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

CH

3

Het3

4191

O—(CH

2

CH

2

)—O

SCH

3

CH

3

Het3

4192

O—(CH

2

CH

2

CH

2

)—O

SCH

3

CH

3

Het3

4193

S—(CH

2

CH

2

)—S

SCH

3

CH

3

Het3

4194

S—(CH

2

CH

2

CH

2

)—S

SCH

3

CH

3

Het3

4195

—(CH

2

)

4

—

SCH

3

CH

3

Het3

4196

—(CH

2

)

5

—

SCH

3

CH

3

Het3

4197

H

H

SO

2

CH

3

CH

3

Het3

4198

CH

3

CH

3

SO

2

CH

3

CH

3

Het3

4199

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

CH

3

Het3

4200

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

CH

3

Het3

4201

OCH

3

OCH

3

SO

2

CH

3

CH

3

Het3

4202

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

CH

3

Het3

4203

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

CH

3

Het3

4204

SCH

3

SCH

3

SO

2

CH

3

CH

3

Het3

4205

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

CH

3

Het3

4206

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

CH

3

Het3

4207

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

CH

3

Het3

4208

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

CH

3

Het3

4209

O—(CH

2

CH

2

)—O

SO

2

CH

3

CH

3

Het3

4210

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

CH

3

Het3

4211

S—(CH

2

CH

2

)—S

SO

2

CH

3

CH

3

Het3

4212

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

CH

3

Het3

4213

—(CH

2

)

4

—

SO

2

CH

3

CH

3

Het3

4214

—(CH

2

)

5

—

SO

2

CH

3

CH

3

Het3

4215

H

H

PO(OCH

3

)

2

CH

3

Het3

4216

CH

3

CH

3

PO(OCH

3

)

2

CH

3

Het3

4217

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

CH

3

Het3

4218

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

CH

3

Het3

4219

OCH

3

OCH

3

PO(OCH

3

)

2

CH

3

Het3

4220

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

CH

3

Het3

4221

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

CH

3

Het3

4222

SCH

3

SCH

3

PO(OCH

3

)

2

CH

3

Het3

4223

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

CH

3

Het3

4224

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

CH

3

Het3

4225

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

CH

3

Het3

4226

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

CH

3

Het3

4227

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

CH

3

Het3

4228

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

CH

3

Het3

4229

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

CH

3

Het3

4230

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

CH

3

Het3

4231

—(CH

2

)

4

—

PO(OCH

3

)

2

CH

3

Het3

4232

—(CH

2

)

5

—

PO(OCH

3

)

2

CH

3

Het3

4233

H

H

PO(OCH

2

CH

3

)

2

CH

3

Het3

4234

CH

3

CH

3

PO(OCH

2

CH

3

)

2

CH

3

Het3

4235

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

Het3

4236

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

Het3

4237

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

CH

3

Het3

4238

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

Het3

4239

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

Het3

4240

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

CH

3

Het3

4241

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

CH

3

Het3

4242

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

CH

3

Het3

4243

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

CH

3

Het3

4244

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

CH

3

Het3

4245

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

CH

3

Het3

4246

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

CH

3

Het3

4247

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

CH

3

Het3

4248

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

CH

3

Het3

4249

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

CH

3

Het3

4250

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

CH

3

Het3

4251

H

H

PO(CH

3

)

2

CH

3

Het3

4252

CH

3

CH

3

PO(CH

3

)

2

CH

3

Het3

4253

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

CH

3

Het3

4254

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

CH

3

Het3

4255

OCH

3

OCH

3

PO(CH

3

)

2

CH

3

Het3

4256

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

CH

3

Het3

4257

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

CH

3

Het3

4258

SCH

3

SCH

3

PO(CH

3

)

2

CH

3

Het3

4259

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

CH

3

Het3

4260

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

CH

3

Het3

4261

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

CH

3

Het3

4262

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

CH

3

Het3

4263

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

CH

3

Het3

4264

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

CH

3

Het3

4265

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

CH

3

Het3

4266

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

CH

3

Het3

4267

—(CH

2

)

4

—

PO(CH

3

)

2

CH

3

Het3

4268

—(CH

2

)

5

—

PO(CH

3

)

2

CH

3

Het3

4269

H

H

PO(CH

2

CH

3

)

2

CH

3

Het3

4270

CH

3

CH

3

PO(CH

2

CH

3

)

2

CH

3

Het3

4271

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

Het3

4272

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

Het3

4273

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

CH

3

Het3

4274

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

Het3

4275

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

Het3

4276

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

CH

3

Het3

4277

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

CH

3

Het3

4278

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

CH

3

Het3

4279

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

CH

3

Het3

4280

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

CH

3

Het3

4281

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

CH

3

Het3

4282

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

CH

3

Het3

4283

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

CH

3

Het3

4284

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

CH

3

Het3

4285

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

CH

3

Het3

4286

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

CH

3

Het3

4287

H

H

H

Cl

OH

4288

CH

3

CH

3

H

Cl

OH

4289

CH

2

CH

3

CH

2

CH

3

H

Cl

OH

4290

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Cl

OH

4291

OCH

3

OCH

3

H

Cl

OH

4292

OCH

2

CH

3

OCH

2

CH

3

H

Cl

OH

4293

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Cl

OH

4294

SCH

3

SCH

3

H

Cl

OH

4295

SCH

2

CH

3

SCH

2

CH

3

H

Cl

OH

4296

N(CH

3

)

2

N(CH

3

)

2

H

Cl

OH

4297

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Cl

OH

4298

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Cl

OH

4299

O—(CH

2

CH

2

)—O

H

Cl

OH

4300

O—(CH

2

CH

2

CH

2

)—O

H

Cl

OH

4301

S—(CH

2

CH

2

)—S

H

Cl

OH

4302

S—(CH

2

CH

2

CH

2

)—S

H

Cl

OH

4303

—(CH

2

)

4

—

H

Cl

OH

4304

—(CH

2

)

5

—

H

Cl

OH

4305

H

H

NO

2

Cl

OH

4306

CH

3

CH

3

NO

2

Cl

OH

4307

CH

2

CH

3

CH

2

CH

3

NO

2

Cl

OH

4308

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Cl

OH

4309

OCH

3

OCH

3

NO

2

Cl

OH

4310

OCH

2

CH

3

OCH

2

CH

3

NO

2

Cl

OH

4311

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Cl

OH

4312

SCH

3

SCH

3

NO

2

Cl

OH

4313

SCH

2

CH

3

SCH

2

CH

3

NO

2

Cl

OH

4314

N(CH

3

)

2

N(CH

3

)

2

NO

2

Cl

OH

4315

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Cl

OH

4316

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Cl

OH

4317

O—(CH

2

CH

2

)—O

NO

2

Cl

OH

4318

O—(CH

2

CH

2

CH

2

)—O

NO

2

Cl

OH

4319

S—(CH

2

CH

2

)—S

NO

2

Cl

OH

4320

S—(CH

2

CH

2

CH

2

)—S

NO

2

Cl

OH

4321

—(CH

2

)

4

—

NO

2

Cl

OH

4322

—(CH

2

)

5

—

NO

2

Cl

OH

4323

H

H

CN

Cl

OH

4324

CH

3

CH

3

CN

Cl

OH

4325

CH

2

CH

3

CH

2

CH

3

CN

Cl

OH

4326

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Cl

OH

4327

OCH

3

OCH

3

CN

Cl

OH

4328

OCH

2

CH

3

OCH

2

CH

3

CN

Cl

OH

4329

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Cl

OH

4330

SCH

3

SCH

3

CN

Cl

OH

4331

SCH

2

CH

3

SCH

2

CH

3

CN

Cl

OH

4332

N(CH

3

)

2

N(CH

3

)

2

CN

Cl

OH

4333

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Cl

OH

4334

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Cl

OH

4335

O—(CH

2

CH

2

)—O

CN

Cl

OH

4336

O—(CH

2

CH

2

CH

2

)—O

CN

Cl

OH

4337

S—(CH

2

CH

2

)—S

CN

Cl

OH

4338

S—(CH

2

CH

2

CH

2

)—S

CN

Cl

OH

4339

—(CH

2

)

4

—

CN

Cl

OH

4340

—(CH

2

)

5

—

CN

Cl

OH

4341

H

H

F

Cl

OH

4342

CH

3

CH

3

F

Cl

OH

4343

CH

2

CH

3

CH

2

CH

3

F

Cl

OH

4344

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Cl

OH

4345

OCH

3

OCH

3

F

Cl

OH

4346

OCH

2

CH

3

OCH

2

CH

3

F

Cl

OH

4347

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Cl

OH

4348

SCH

3

SCH

3

F

Cl

OH

4349

SCH

2

CH

3

SCH

2

CH

3

F

Cl

OH

4350

N(CH

3

)

2

N(CH

3

)

2

F

Cl

OH

4351

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Cl

OH

4352

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Cl

OH

4353

O—(CH

2

CH

2

)—O

F

Cl

OH

4354

O—(CH

2

CH

2

CH

2

)—O

F

Cl

OH

4355

S—(CH

2

CH

2

)—S

F

Cl

OH

4356

S—(CH

2

CH

2

CH

2

)—S

F

Cl

OH

4357

—(CH

2

)

4

—

F

Cl

OH

4358

—(CH

2

)

5

—

F

Cl

OH

4359

H

H

Cl

Cl

OH

4360

CH

3

CH

3

Cl

Cl

OH

4361

CH

2

CH

3

CH

2

CH

3

Cl

Cl

OH

4362

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Cl

OH

4363

OCH

3

OCH

3

Cl

Cl

OH

4364

OCH

2

CH

3

OCH

2

CH

3

Cl

Cl

OH

4365

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Cl

OH

4366

SCH

3

SCH

3

Cl

Cl

OH

4367

SCH

2

CH

3

SCH

2

CH

3

Cl

Cl

OH

4368

N(CH

3

)

2

N(CH

3

)

2

Cl

Cl

OH

4369

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Cl

OH

4370

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Cl

OH

4371

O—(CH

2

CH

2

)—O

Cl

Cl

OH

4372

O—(CH

2

CH

2

CH

2

)—O

Cl

Cl

OH

4373

S—(CH

2

CH

2

)—S

Cl

Cl

OH

4374

S—(CH

2

CH

2

CH

2

)—S

Cl

Cl

OH

4375

—(CH

2

)

4

—

Cl

Cl

OH

4376

—(CH

2

)

5

—

Cl

Cl

OH

4377

H

H

Br

Cl

OH

4378

CH

3

CH

3

Br

Cl

OH

4379

CH

2

CH

3

CH

2

CH

3

Br

Cl

OH

4380

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Cl

OH

4381

OCH

3

OCH

3

Br

Cl

OH

4382

OCH

2

CH

3

OCH

2

CH

3

Br

Cl

OH

4383

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Cl

OH

4384

SCH

3

SCH

3

Br

Cl

OH

4385

SCH

2

CH

3

SCH

2

CH

3

Br

Cl

OH

4386

N(CH

3

)

2

N(CH

3

)

2

Br

Cl

OH

4387

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Cl

OH

4388

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Cl

OH

4389

O—(CH

2

CH

2

)—O

Br

Cl

OH

4390

O—(CH

2

CH

2

CH

2

)—O

Br

Cl

OH

4391

S—(CH

2

CH

2

)—S

Br

Cl

OH

4392

S—(CH

2

CH

2

CH

2

)—S

Br

Cl

OH

4393

—(CH

2

)

4

—

Br

Cl

OH

4394

—(CH

2

)

5

—

Br

Cl

OH

4395

H

H

CH

3

Cl

OH

4396

CH

3

CH

3

CH

3

Cl

OH

4397

CH

2

CH

3

CH

2

CH

3

CH

3

Cl

OH

4398

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Cl

OH

4399

OCH

3

OCH

3

CH

3

Cl

OH

4400

OCH

2

CH

3

OCH

2

CH

3

CH

3

Cl

OH

4401

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Cl

OH

4402

SCH

3

SCH

3

CH

3

Cl

OH

4403

SCH

2

CH

3

SCH

2

CH

3

CH

3

Cl

OH

4404

N(CH

3

)

2

N(CH

3

)

2

CH

3

Cl

OH

4405

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Cl

OH

4406

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Cl

OH

4407

O—(CH

2

CH

2

)—O

CH

3

Cl

OH

4408

O—(CH

2

CH

2

CH

2

)—O

CH

3

Cl

OH

4409

S—(CH

2

CH

2

)—S

CH

3

Cl

OH

4410

S—(CH

2

CH

2

CH

2

)—S

CH

3

Cl

OH

4411

—(CH

2

)

4

—

CH

3

Cl

OH

4412

—(CH

2

)

5

—

CH

3

Cl

OH

4413

H

H

CH

2

CH

3

Cl

OH

4414

CH

3

CH

3

CH

2

CH

3

Cl

OH

4415

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Cl

OH

4416

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Cl

OH

4417

OCH

3

OCH

3

CH

2

CH

3

Cl

OH

4418

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Cl

OH

4419

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Cl

OH

4420

SCH

3

SCH

3

CH

2

CH

3

Cl

OH

4421

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Cl

OH

4422

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Cl

OH

4423

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Cl

OH

4424

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Cl

OH

4425

O—(CH

2

CH

2

)—O

CH

2

CH

3

Cl

OH

4426

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Cl

OH

4427

S—(CH

2

CH

2

)—S

CH

2

CH

3

Cl

OH

4428

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Cl

OH

4429

—(CH

2

)

4

—

CH

2

CH

3

Cl

OH

4430

—(CH

2

)

5

—

CH

2

CH

3

Cl

OH

4431

H

H

CF

3

Cl

OH

4432

CH

3

CH

3

CF

3

Cl

OH

4433

CH

2

CH

3

CH

2

CH

3

CF

3

Cl

OH

4434

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Cl

OH

4435

OCH

3

OCH

3

CF

3

Cl

OH

4436

OCH

2

CH

3

OCH

2

CH

3

CF

3

Cl

OH

4437

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Cl

OH

4438

SCH

3

SCH

3

CF

3

Cl

OH

4439

SCH

2

CH

3

SCH

2

CH

3

CF

3

Cl

OH

4440

N(CH

3

)

2

N(CH

3

)

2

CF

3

Cl

OH

4441

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Cl

OH

4442

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Cl

OH

4443

O—(CH

2

CH

2

)—O

CF

3

Cl

OH

4444

O—(CH

2

CH

2

CH

2

)—O

CF

3

Cl

OH

4445

S—(CH

2

CH

2

)—S

CF

3

Cl

OH

4446

S—(CH

2

CH

2

CH

2

)—S

CF

3

Cl

OH

4447

—(CH

2

)

4

—

CF

3

Cl

OH

4448

—(CH

2

)

5

—

CF

3

Cl

OH

4449

H

H

OCH

3

Cl

OH

4450

CH

3

CH

3

OCH

3

Cl

OH

4451

CH

2

CH

3

CH

2

CH

3

OCH

3

Cl

OH

4452

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Cl

OH

4453

OCH

3

OCH

3

OCH

3

Cl

OH

4454

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Cl

OH

4455

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Cl

OH

4456

SCH

3

SCH

3

OCH

3

Cl

OH

4457

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Cl

OH

4458

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Cl

OH

4459

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Cl

OH

4460

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Cl

OH

4461

O—(CH

2

CH

2

)—O

OCH

3

Cl

OH

4462

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Cl

OH

4463

S—(CH

2

CH

2

)—S

OCH

3

Cl

OH

4464

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Cl

OH

4465

—(CH

2

)

4

—

OCH

3

Cl

OH

4466

—(CH

2

)

5

—

OCH

3

Cl

OH

4467

H

H

OCH

2

CH

3

Cl

OH

4468

CH

3

CH

3

OCH

2

CH

3

Cl

OH

4469

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Cl

OH

4470

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Cl

OH

4471

OCH

3

OCH

3

OCH

2

CH

3

Cl

OH

4472

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Cl

OH

4473

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Cl

OH

4474

SCH

3

SCH

3

OCH

2

CH

3

Cl

OH

4475

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Cl

OH

4476

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Cl

OH

4477

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Cl

OH

4478

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Cl

OH

4479

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Cl

OH

4480

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Cl

OH

4481

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Cl

OH

4482

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Cl

OH

4483

—(CH

2

)

4

—

OCH

2

CH

3

Cl

OH

4484

—(CH

2

)

5

—

OCH

2

CH

3

Cl

OH

4485

H

H

SCH

3

Cl

OH

4486

CH

3

CH

3

SCH

3

Cl

OH

4487

CH

2

CH

3

CH

2

CH

3

SCH

3

Cl

OH

4488

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Cl

OH

4489

OCH

3

OCH

3

SCH

3

Cl

OH

4490

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Cl

OH

4491

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Cl

OH

4492

SCH

3

SCH

3

SCH

3

Cl

OH

4493

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Cl

OH

4494

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Cl

OH

4495

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Cl

OH

4496

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Cl

OH

4497

O—(CH

2

CH

2

)—O

SCH

3

Cl

OH

4498

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Cl

OH

4499

S—(CH

2

CH

2

)—S

SCH

3

Cl

OH

4500

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Cl

OH

4501

—(CH

2

)

4

—

SCH

3

Cl

OH

4502

—(CH

2

)

5

—

SCH

3

Cl

OH

4503

H

H

SO

2

CH

3

Cl

OH

4504

CH

3

CH

3

SO

2

CH

3

Cl

OH

4505

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Cl

OH

4506

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Cl

OH

4507

OCH

3

OCH

3

SO

2

CH

3

Cl

OH

4508

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Cl

OH

4509

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Cl

OH

4510

SCH

3

SCH

3

SO

2

CH

3

Cl

OH

4511

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Cl

OH

4512

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Cl

OH

4513

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Cl

OH

4514

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Cl

OH

4515

O—(CH

2

CH

2

)—O

SO

2

CH

3

Cl

OH

4516

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Cl

OH

4517

S—(CH

2

CH

2

)—S

SO

2

CH

3

Cl

OH

4518

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Cl

OH

4519

—(CH

2

)

4

—

SO

2

CH

3

Cl

OH

4520

—(CH

2

)

5

—

SO

2

CH

3

Cl

OH

4521

H

H

PO(OCH

3

)

2

Cl

OH

4522

CH

3

CH

3

PO(OCH

3

)

2

Cl

OH

4523

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Cl

OH

4524

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

OH

4525

OCH

3

OCH

3

PO(OCH

3

)

2

Cl

OH

4526

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Cl

OH

4527

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

OH

4528

SCH

3

SCH

3

PO(OCH

3

)

2

Cl

OH

4529

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Cl

OH

4530

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Cl

OH

4531

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Cl

OH

4532

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Cl

OH

4533

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

OH

4534

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

OH

4535

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

OH

4536

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

OH

4537

—(CH

2

)

4

—

PO(OCH

3

)

2

Cl

OH

4538

—(CH

2

)

5

—

PO(OCH

3

)

2

Cl

OH

4539

H

H

PO(OCH

2

CH

3

)

2

Cl

OH

4540

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Cl

OH

4541

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

OH

4542

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

OH

4543

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Cl

OH

4544

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

OH

4545

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

OH

4546

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Cl

OH

4547

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

OH

4548

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

OH

4549

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

OH

4550

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Cl

OH

4551

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

OH

4552

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

OH

4553

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

OH

4554

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

OH

4555

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Cl

OH

4556

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Cl

OH

4557

H

H

PO(CH

3

)

2

Cl

OH

4558

CH

3

CH

3

PO(CH

3

)

2

Cl

OH

4559

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Cl

OH

4560

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

OH

4561

OCH

3

OCH

3

PO(CH

3

)

2

Cl

OH

4562

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Cl

OH

4563

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

OH

4564

SCH

3

SCH

3

PO(CH

3

)

2

Cl

OH

4565

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Cl

OH

4566

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Cl

OH

4567

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Cl

OH

4568

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Cl

OH

4569

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

OH

4570

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

OH

4571

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

OH

4572

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

OH

4573

—(CH

2

)

4

—

PO(CH

3

)

2

Cl

OH

4574

—(CH

2

)

5

—

PO(CH

3

)

2

Cl

OH

4575

H

H

PO(CH

2

CH

3

)

2

Cl

OH

4576

CH

3

CH

3

PO(CH

2

CH

3

)

2

Cl

OH

4577

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

OH

4578

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

OH

4579

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

Cl

OH

4580

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

OH

4581

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

OH

4582

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

Cl

OH

4583

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

OH

4584

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

Cl

OH

4585

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

Cl

OH

4586

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

Cl

OH

4587

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

Cl

OH

4588

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

Cl

OH

4589

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

Cl

OH

4590

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

Cl

OH

4591

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

Cl

OH

4592

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

Cl

OH

4593

H

H

H

Cl

OCOC

6

H

5

4594

CH

3

CH

3

H

Cl

OCOC

6

H

5

4595

CH

2

CH

3

CH

2

CH

3

H

Cl

OCOC

6

H

5

4596

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Cl

OCOC

6

H

5

4597

OCH

3

OCH

3

H

Cl

OCOC

6

H

5

4598

OCH

2

CH

3

OCH

2

CH

3

H

Cl

OCOC

6

H

5

4599

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Cl

OCOC

6

H

5

4600

SCH

3

SCH

3

H

Cl

OCOC

6

H

5

4601

SCH

2

CH

3

SCH

2

CH

3

H

Cl

OCOC

6

H

5

4602

N(CH

3

)

2

N(CH

3

)

2

H

Cl

OCOC

6

H

5

4603

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Cl

OCOC

6

H

5

4604

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Cl

OCOC

6

H

5

4605

O—(CH

2

CH

2

)—O

H

Cl

OCOC

6

H

5

4606

O—(CH

2

CH

2

CH

2

)—O

H

Cl

OCOC

6

H

5

4607

S—(CH

2

CH

2

)—S

H

Cl

OCOC

6

H

5

4608

S—(CH

2

CH

2

CH

2

)—S

H

Cl

OCOC

6

H

5

4609

—(CH

2

)

4

—

H

Cl

OCOC

6

H

5

4610

—(CH

2

)

5

—

H

Cl

OCOC

6

H

5

4611

H

H

NO

2

Cl

OCOC

6

H

5

4612

CH

3

CH

3

NO

2

Cl

OCOC

6

H

5

4613

CH

2

CH

3

CH

2

CH

3

NO

2

Cl

OCOC

6

H

5

4614

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Cl

OCOC

6

H

5

4615

OCH

3

OCH

3

NO

2

Cl

OCOC

6

H

5

4616

OCH

2

CH

3

OCH

2

CH

3

NO

2

Cl

OCOC

6

H

5

4617

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Cl

OCOC

6

H

5

4618

SCH

3

SCH

3

NO

2

Cl

OCOC

6

H

5

4619

SCH

2

CH

3

SCH

2

CH

3

NO

2

Cl

OCOC

6

H

5

4620

N(CH

3

)

2

N(CH

3

)

2

NO

2

Cl

OCOC

6

H

5

4621

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Cl

OCOC

6

H

5

4622

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Cl

OCOC

6

H

5

4623

O—(CH

2

CH

2

)—O

NO

2

Cl

OCOC

6

H

5

4624

O—(CH

2

CH

2

CH

2

)—O

NO

2

Cl

OCOC

6

H

5

4625

S—(CH

2

CH

2

)—S

NO

2

Cl

OCOC

6

H

5

4626

S—(CH

2

CH

2

CH

2

)—S

NO

2

Cl

OCOC

6

H

5

4627

—(CH

2

)

4

—

NO

2

Cl

OCOC

6

H

5

4628

—(CH

2

)

5

—

NO

2

Cl

OCOC

6

H

5

4629

H

H

CN

Cl

OCOC

6

H

5

4630

CH

3

CH

3

CN

Cl

OCOC

6

H

5

4631

CH

2

CH

3

CH

2

CH

3

CN

Cl

OCOC

6

H

5

4632

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Cl

OCOC

6

H

5

4633

OCH

3

OCH

3

CN

Cl

OCOC

6

H

5

4634

OCH

2

CH

3

OCH

2

CH

3

CN

Cl

OCOC

6

H

5

4635

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Cl

OCOC

6

H

5

4636

SCH

3

SCH

3

CN

Cl

OCOC

6

H

5

4637

SCH

2

CH

3

SCH

2

CH

3

CN

Cl

OCOC

6

H

5

4638

N(CH

3

)

2

N(CH

3

)

2

CN

Cl

OCOC

6

H

5

4639

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Cl

OCOC

6

H

5

4640

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Cl

OCOC

6

H

5

4641

O—(CH

2

CH

2

)—O

CN

Cl

OCOC

6

H

5

4642

O—(CH

2

CH

2

CH

2

)—O

CN

Cl

OCOC

6

H

5

4643

S—(CH

2

CH

2

)—S

CN

Cl

OCOC

6

H

5

4644

S—(CH

2

CH

2

CH

2

)—S

CN

Cl

OCOC

6

H

5

4645

—(CH

2

)

4

—

CN

Cl

OCOC

6

H

5

4646

—(CH

2

)

5

—

CN

Cl

OCOC

6

H

5

4647

H

H

F

Cl

OCOC

6

H

5

4648

CH

3

CH

3

F

Cl

OCOC

6

H

5

4649

CH

2

CH

3

CH

2

CH

3

F

Cl

OCOC

6

H

5

4650

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Cl

OCOC

6

H

5

4651

OCH

3

OCH

3

F

Cl

OCOC

6

H

5

4652

OCH

2

CH

3

OCH

2

CH

3

F

Cl

OCOC

6

H

5

4653

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Cl

OCOC

6

H

5

4654

SCH

3

SCH

3

F

Cl

OCOC

6

H

5

4655

SCH

2

CH

3

SCH

2

CH

3

F

Cl

OCOC

6

H

5

4656

N(CH

3

)

2

N(CH

3

)

2

F

Cl

OCOC

6

H

5

4657

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Cl

OCOC

6

H

5

4658

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Cl

OCOC

6

H

5

4659

O—(CH

2

CH

2

)—O

F

Cl

OCOC

6

H

5

4660

O—(CH

2

CH

2

CH

2

)—O

F

Cl

OCOC

6

H

5

4661

S—(CH

2

CH

2

)—S

F

Cl

OCOC

6

H

5

4662

S—(CH

2

CH

2

CH

2

)—S

F

Cl

OCOC

6

H

5

4663

—(CH

2

)

4

—

F

Cl

OCOC

6

H

5

4664

—(CH

2

)

5

—

F

Cl

OCOC

6

H

5

4665

H

H

Cl

Cl

OCOC

6

H

5

4666

CH

3

CH

3

Cl

Cl

OCOC

6

H

5

4667

CH

2

CH

3

CH

2

CH

3

Cl

Cl

OCOC

6

H

5

4668

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Cl

OCOC

6

H

5

4669

OCH

3

OCH

3

Cl

Cl

OCOC

6

H

5

4670

OCH

2

CH

3

OCH

2

CH

3

Cl

Cl

OCOC

6

H

5

4671

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Cl

OCOC

6

H

5

4672

SCH

3

SCH

3

Cl

Cl

OCOC

6

H

5

4673

SCH

2

CH

3

SCH

2

CH

3

Cl

Cl

OCOC

6

H

5

4674

N(CH

3

)

2

N(CH

3

)

2

Cl

Cl

OCOC

6

H

5

4675

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Cl

OCOC

6

H

5

4676

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Cl

OCOC

6

H

5

4677

O—(CH

2

CH

2

)—O

Cl

Cl

OCOC

6

H

5

4678

O—(CH

2

CH

2

CH

2

)—O

Cl

Cl

OCOC

6

H

5

4679

S—(CH

2

CH

2

)—S

Cl

Cl

OCOC

6

H

5

4680

S—(CH

2

CH

2

CH

2

)—S

Cl

Cl

OCOC

6

H

5

4681

—(CH

2

)

4

—

Cl

Cl

OCOC

6

H

5

4682

—(CH

2

)

5

—

Cl

Cl

OCOC

6

H

5

4683

H

H

Br

Cl

OCOC

6

H

5

4684

CH

3

CH

3

Br

Cl

OCOC

6

H

5

4685

CH

2

CH

3

CH

2

CH

3

Br

Cl

OCOC

6

H

5

4686

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Cl

OCOC

6

H

5

4687

OCH

3

OCH

3

Br

Cl

OCOC

6

H

5

4688

OCH

2

CH

3

OCH

2

CH

3

Br

Cl

OCOC

6

H

5

4689

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Cl

OCOC

6

H

5

4690

SCH

3

SCH

3

Br

Cl

OCOC

6

H

5

4691

SCH

2

CH

3

SCH

2

CH

3

Br

Cl

OCOC

6

H

5

4692

N(CH

3

)

2

N(CH

3

)

2

Br

Cl

OCOC

6

H

5

4693

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Cl

OCOC

6

H

5

4694

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Cl

OCOC

6

H

5

4695

O—(CH

2

CH

2

)—O

Br

Cl

OCOC

6

H

5

4696

O—(CH

2

CH

2

CH

2

)—O

Br

Cl

OCOC

6

H

5

4697

S—(CH

2

CH

2

)—S

Br

Cl

OCOC

6

H

5

4698

S—(CH

2

CH

2

CH

2

)—S

Br

Cl

OCOC

6

H

5

4699

—(CH

2

)

4

—

Br

Cl

OCOC

6

H

5

4700

—(CH

2

)

5

—

Br

Cl

OCOC

6

H

5

4701

H

H

CH

3

Cl

OCOC

6

H

5

4702

CH

3

CH

3

CH

3

Cl

OCOC

6

H

5

4703

CH

2

CH

3

CH

2

CH

3

CH

3

Cl

OCOC

6

H

5

4704

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Cl

OCOC

6

H

5

4705

OCH

3

OCH

3

CH

3

Cl

OCOC

6

H

5

4706

OCH

2

CH

3

OCH

2

CH

3

CH

3

Cl

OCOC

6

H

5

4707

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Cl

OCOC

6

H

5

4708

SCH

3

SCH

3

CH

3

Cl

OCOC

6

H

5

4709

SCH

2

CH

3

SCH

2

CH

3

CH

3

Cl

OCOC

6

H

5

4710

N(CH

3

)

2

N(CH

3

)

2

CH

3

Cl

OCOC

6

H

5

4711

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Cl

OCOC

6

H

5

4712

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Cl

OCOC

6

H

5

4713

O—(CH

2

CH

2

)—O

CH

3

Cl

OCOC

6

H

5

4714

O—(CH

2

CH

2

CH

2

)—O

CH

3

Cl

OCOC

6

H

5

4715

S—(CH

2

CH

2

)—S

CH

3

Cl

OCOC

6

H

5

4716

S—(CH

2

CH

2

CH

2

)—S

CH

3

Cl

OCOC

6

H

5

4717

—(CH

2

)

4

—

CH

3

Cl

OCOC

6

H

5

4718

—(CH

2

)

5

—

CH

3

Cl

OCOC

6

H

5

4719

H

H

CH

2

CH

3

Cl

OCOC

6

H

5

4720

CH

3

CH

3

CH

2

CH

3

Cl

OCOC

6

H

5

4721

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Cl

OCOC

6

H

5

4722

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Cl

OCOC

6

H

5

4723

OCH

3

OCH

3

CH

2

CH

3

Cl

OCOC

6

H

5

4724

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Cl

OCOC

6

H

5

4725

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Cl

OCOC

6

H

5

4726

SCH

3

SCH

3

CH

2

CH

3

Cl

OCOC

6

H

5

4727

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Cl

OCOC

6

H

5

4728

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Cl

OCOC

6

H

5

4729

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Cl

OCOC

6

H

5

4730

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Cl

OCOC

6

H

5

4731

O—(CH

2

CH

2

)—O

CH

2

CH

3

Cl

OCOC

6

H

5

4732

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Cl

OCOC

6

H

5

4733

S—(CH

2

CH

2

)—S

CH

2

CH

3

Cl

OCOC

6

H

5

4734

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Cl

OCOC

6

H

5

4735

—(CH

2

)

4

—

CH

2

CH

3

Cl

OCOC

6

H

5

4736

—(CH

2

)

5

—

CH

2

CH

3

Cl

OCOC

6

H

5

4737

H

H

CF

3

Cl

OCOC

6

H

5

4738

CH

3

CH

3

CF

3

Cl

OCOC

6

H

5

4739

CH

2

CH

3

CH

2

CH

3

CF

3

Cl

OCOC

6

H

5

4740

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Cl

OCOC

6

H

5

4741

OCH

3

OCH

3

CF

3

Cl

OCOC

6

H

5

4742

OCH

2

CH

3

OCH

2

CH

3

CF

3

Cl

OCOC

6

H

5

4743

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Cl

OCOC

6

H

5

4744

SCH

3

SCH

3

CF

3

Cl

OCOC

6

H

5

4745

SCH

2

CH

3

SCH

2

CH

3

CF

3

Cl

OCOC

6

H

5

4746

N(CH

3

)

2

N(CH

3

)

2

CF

3

Cl

OCOC

6

H

5

4747

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Cl

OCOC

6

H

5

4748

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Cl

OCOC

6

H

5

4749

O—(CH

2

CH

2

)—O

CF

3

Cl

OCOC

6

H

5

4750

O—(CH

2

CH

2

CH

2

)—O

CF

3

Cl

OCOC

6

H

5

4751

S—(CH

2

CH

2

)—S

CF

3

Cl

OCOC

6

H

5

4752

S—(CH

2

CH

2

CH

2

)—S

CF

3

Cl

OCOC

6

H

5

4753

—(CH

2

)

4

—

CF

3

Cl

OCOC

6

H

5

4754

—(CH

2

)

5

—

CF

3

Cl

OCOC

6

H

5

4755

H

H

OCH

3

Cl

OCOC

6

H

5

4756

CH

3

CH

3

OCH

3

Cl

OCOC

6

H

5

4757

CH

2

CH

3

CH

2

CH

3

OCH

3

Cl

OCOC

6

H

5

4758

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Cl

OCOC

6

H

5

4759

OCH

3

OCH

3

OCH

3

Cl

OCOC

6

H

5

4760

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Cl

OCOC

6

H

5

4761

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Cl

OCOC

6

H

5

4762

SCH

3

SCH

3

OCH

3

Cl

OCOC

6

H

5

4763

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Cl

OCOC

6

H

5

4764

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Cl

OCOC

6

H

5

4765

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Cl

OCOC

6

H

5

4766

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Cl

OCOC

6

H

5

4767

O—(CH

2

CH

2

)—O

OCH

3

Cl

OCOC

6

H

5

4768

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Cl

OCOC

6

H

5

4769

S—(CH

2

CH

2

)—S

OCH

3

Cl

OCOC

6

H

5

4770

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Cl

OCOC

6

H

5

4771

—(CH

2

)

4

—

OCH

3

Cl

OCOC

6

H

5

4772

—(CH

2

)

5

—

OCH

3

Cl

OCOC

6

H

5

4773

H

H

OCH

2

CH

3

Cl

OCOC

6

H

5

4774

CH

3

CH

3

OCH

2

CH

3

Cl

OCOC

6

H

5

4775

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Cl

OCOC

6

H

5

4776

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Cl

OCOC

6

H

5

4777

OCH

3

OCH

3

OCH

2

CH

3

Cl

OCOC

6

H

5

4778

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Cl

OCOC

6

H

5

4779

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Cl

OCOC

6

H

5

4780

SCH

3

SCH

3

OCH

2

CH

3

Cl

OCOC

6

H

5

4781

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Cl

OCOC

6

H

5

4782

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Cl

OCOC

6

H

5

4783

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Cl

OCOC

6

H

5

4784

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Cl

OCOC

6

H

5

4785

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Cl

OCOC

6

H

5

4786

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Cl

OCOC

6

H

5

4787

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Cl

OCOC

6

H

5

4788

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Cl

OCOC

6

H

5

4789

—(CH

2

)

4

—

OCH

2

CH

3

Cl

OCOC

6

H

5

4790

—(CH

2

)

5

—

OCH

2

CH

3

Cl

OCOC

6

H

5

4791

H

H

SCH

3

Cl

OCOC

6

H

5

4792

CH

3

CH

3

SCH

3

Cl

OCOC

6

H

5

4793

CH

2

CH

3

CH

2

CH

3

SCH

3

Cl

OCOC

6

H

5

4794

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Cl

OCOC

6

H

5

4795

OCH

3

OCH

3

SCH

3

Cl

OCOC

6

H

5

4796

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Cl

OCOC

6

H

5

4797

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Cl

OCOC

6

H

5

4798

SCH

3

SCH

3

SCH

3

Cl

OCOC

6

H

5

4799

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Cl

OCOC

6

H

5

4800

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Cl

OCOC

6

H

5

4801

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Cl

OCOC

6

H

5

4802

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Cl

OCOC

6

H

5

4803

O—(CH

2

CH

2

)—O

SCH

3

Cl

OCOC

6

H

5

4804

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Cl

OCOC

6

H

5

4805

S—(CH

2

CH

2

)—S

SCH

3

Cl

OCOC

6

H

5

4806

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Cl

OCOC

6

H

5

4807

—(CH

2

)

4

—

SCH

3

Cl

OCOC

6

H

5

4808

—(CH

2

)

5

—

SCH

3

Cl

OCOC

6

H

5

4809

H

H

SO

2

CH

3

Cl

OCOC

6

H

5

4810

CH

3

CH

3

SO

2

CH

3

Cl

OCOC

6

H

5

4811

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Cl

OCOC

6

H

5

4812

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Cl

OCOC

6

H

5

4813

OCH

3

OCH

3

SO

2

CH

3

Cl

OCOC

6

H

5

4814

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Cl

OCOC

6

H

5

4815

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Cl

OCOC

6

H

5

4816

SCH

3

SCH

3

SO

2

CH

3

Cl

OCOC

6

H

5

4817

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Cl

OCOC

6

H

5

4818

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Cl

OCOC

6

H

5

4819

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Cl

OCOC

6

H

5

4820

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Cl

OCOC

6

H

5

4821

O—(CH

2

CH

2

)—O

SO

2

CH

3

Cl

OCOC

6

H

5

4822

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Cl

OCOC

6

H

5

4823

S—(CH

2

CH

2

)—S

SO

2

CH

3

Cl

OCOC

6

H

5

4824

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Cl

OCOC

6

H

5

4825

—(CH

2

)

4

—

SO

2

CH

3

Cl

OCOC

6

H

5

4826

—(CH

2

)

5

—

SO

2

CH

3

Cl

OCOC

6

H

5

4827

H

H

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4828

CH

3

CH

3

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4829

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4830

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4831

OCH

3

OCH

3

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4832

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4833

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4834

SCH

3

SCH

3

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4835

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4836

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4837

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4838

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4839

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4840

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4841

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4842

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4843

—(CH

2

)

4

—

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4844

—(CH

2

)

5

—

PO(OCH

3

)

2

Cl

OCOC

6

H

5

4845

H

H

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4846

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4847

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4848

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4849

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4850

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4851

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4852

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4853

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4854

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4855

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4856

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4857

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4858

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4859

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4860

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4861

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4862

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Cl

OCOC

6

H

5

4863

H

H

PO(CH

3

)

2

Cl

OCOC

6

H

5

4864

CH

3

CH

3

PO(CH

3

)

2

Cl

OCOC

6

H

5

4865

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Cl

OCOC

6

H

5

4866

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

OCOC

6

H

5

4867

OCH

3

OCH

3

PO(CH

3

)

2

Cl

OCOC

6

H

5

4868

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Cl

OCOC

6

H

5

4869

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

OCOC

6

H

5

4870

SCH

3

SCH

3

PO(CH

3

)

2

Cl

OCOC

6

H

5

4871

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Cl

OCOC

6

H

5

4872

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Cl

OCOC

6

H

5

4873

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Cl

OCOC

6

H

5

4874

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Cl

OCOC

6

H

5

4875

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

OCOC

6

H

5

4876

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

OCOC

6

H

5

4877

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

OCOC

6

H

5

4878

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

OCOC

6

H

5

4879

—(CH

2

)

4

—

PO(CH

3

)

2

Cl

OCOC

6

H

5

4880

—(CH

2

)

5

—

PO(CH

3

)

2

Cl

OCOC

6

H

5

4881

H

H

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4882

CH

3

CH

3

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4883

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4884

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4885

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4886

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4887

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4888

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4889

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4890

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4891

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4892

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4893

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4894

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4895

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4896

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4897

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4898

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

Cl

OCOC

6

H

5

4899

H

H

H

Cl

SCH

3

4900

CH

3

CH

3

H

Cl

SCH

3

4901

CH

2

CH

3

CH

2

CH

3

H

Cl

SCH

3

4902

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Cl

SCH

3

4903

OCH

3

OCH

3

H

Cl

SCH

3

4904

OCH

2

CH

3

OCH

2

CH

3

H

Cl

SCH

3

4905

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Cl

SCH

3

4906

SCH

3

SCH

3

H

Cl

SCH

3

4907

SCH

2

CH

3

SCH

2

CH

3

H

Cl

SCH

3

4908

N(CH

3

)

2

N(CH

3

)

2

H

Cl

SCH

3

4909

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Cl

SCH

3

4910

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Cl

SCH

3

4911

O—(CH

2

CH

2

)—O

H

Cl

SCH

3

4912

O—(CH

2

CH

2

CH

2

)—O

H

Cl

SCH

3

4913

S—(CH

2

CH

2

)—S

H

Cl

SCH

3

4914

S—(CH

2

CH

2

CH

2

)—S

H

Cl

SCH

3

4915

—(CH

2

)

4

—

H

Cl

SCH

3

4916

—(CH

2

)

5

—

H

Cl

SCH

3

4917

H

H

NO

2

Cl

SCH

3

4918

CH

3

CH

3

NO

2

Cl

SCH

3

4919

CH

2

CH

3

CH

2

CH

3

NO

2

Cl

SCH

3

4920

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Cl

SCH

3

4921

OCH

3

OCH

3

NO

2

Cl

SCH

3

4922

OCH

2

CH

3

OCH

2

CH

3

NO

2

Cl

SCH

3

4923

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Cl

SCH

3

4924

SCH

3

SCH

3

NO

2

Cl

SCH

3

4925

SCH

2

CH

3

SCH

2

CH

3

NO

2

Cl

SCH

3

4926

N(CH

3

)

2

N(CH

3

)

2

NO

2

Cl

SCH

3

4927

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Cl

SCH

3

4928

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Cl

SCH

3

4929

O—(CH

2

CH

2

)—O

NO

2

Cl

SCH

3

4930

O—(CH

2

CH

2

CH

2

)—O

NO

2

Cl

SCH

3

4931

S—(CH

2

CH

2

)—S

NO

2

Cl

SCH

3

4932

S—(CH

2

CH

2

CH

2

)—S

NO

2

Cl

SCH

3

4933

—(CH

2

)

4

—

NO

2

Cl

SCH

3

4934

—(CH

2

)

5

—

NO

2

Cl

SCH

3

4935

H

H

CN

Cl

SCH

3

4936

CH

3

CH

3

CN

Cl

SCH

3

4937

CH

2

CH

3

CH

2

CH

3

CN

Cl

SCH

3

4938

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Cl

SCH

3

4939

OCH

3

OCH

3

CN

Cl

SCH

3

4940

OCH

2

CH

3

OCH

2

CH

3

CN

Cl

SCH

3

4941

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Cl

SCH

3

4942

SCH

3

SCH

3

CN

Cl

SCH

3

4943

SCH

2

CH

3

SCH

2

CH

3

CN

Cl

SCH

3

4944

N(CH

3

)

2

N(CH

3

)

2

CN

Cl

SCH

3

4945

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Cl

SCH

3

4946

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Cl

SCH

3

4947

O—(CH

2

CH

2

)—O

CN

Cl

SCH

3

4948

O—(CH

2

CH

2

CH

2

)—O

CN

Cl

SCH

3

4949

S—(CH

2

CH

2

)—S

CN

Cl

SCH

3

4950

S—(CH

2

CH

2

CH

2

)—S

CN

Cl

SCH

3

4951

—(CH

2

)

4

—

CN

Cl

SCH

3

4952

—(CH

2

)

5

—

CN

Cl

SCH

3

4953

H

H

F

Cl

SCH

3

4954

CH

3

CH

3

F

Cl

SCH

3

4955

CH

2

CH

3

CH

2

CH

3

F

Cl

SCH

3

4956

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Cl

SCH

3

4957

OCH

3

OCH

3

F

Cl

SCH

3

4958

OCH

2

CH

3

OCH

2

CH

3

F

Cl

SCH

3

4959

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Cl

SCH

3

4960

SCH

3

SCH

3

F

Cl

SCH

3

4961

SCH

2

CH

3

SCH

2

CH

3

F

Cl

SCH

3

4962

N(CH

3

)

2

N(CH

3

)

2

F

Cl

SCH

3

4963

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Cl

SCH

3

4964

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Cl

SCH

3

4965

O—(CH

2

CH

2

)—O

F

Cl

SCH

3

4966

O—(CH

2

CH

2

CH

2

)—O

F

Cl

SCH

3

4967

S—(CH

2

CH

2

)—S

F

Cl

SCH

3

4968

S—(CH

2

CH

2

CH

2

)—S

F

Cl

SCH

3

4969

—(CH

2

)

4

—

F

Cl

SCH

3

4970

—(CH

2

)

5

—

F

Cl

SCH

3

4971

H

H

Cl

Cl

SCH

3

4972

CH

3

CH

3

Cl

Cl

SCH

3

4973

CH

2

CH

3

CH

2

CH

3

Cl

Cl

SCH

3

4974

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Cl

SCH

3

4975

OCH

3

OCH

3

Cl

Cl

SCH

3

4976

OCH

2

CH

3

OCH

2

CH

3

Cl

Cl

SCH

3

4977

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Cl

SCH

3

4978

SCH

3

SCH

3

Cl

Cl

SCH

3

4979

SCH

2

CH

3

SCH

2

CH

3

Cl

Cl

SCH

3

4980

N(CH

3

)

2

N(CH

3

)

2

Cl

Cl

SCH

3

4981

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Cl

SCH

3

4982

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Cl

SCH

3

4983

O—(CH

2

CH

2

)—O

Cl

Cl

SCH

3

4984

O—(CH

2

CH

2

CH

2

)—O

Cl

Cl

SCH

3

4985

S—(CH

2

CH

2

)—S

Cl

Cl

SCH

3

4986

S—(CH

2

CH

2

CH

2

)—S

Cl

Cl

SCH

3

4987

—(CH

2

)

4

—

Cl

Cl

SCH

3

4988

—(CH

2

)

5

—

Cl

Cl

SCH

3

4989

H

H

Br

Cl

SCH

3

4990

CH

3

CH

3

Br

Cl

SCH

3

4991

CH

2

CH

3

CH

2

CH

3

Br

Cl

SCH

3

4992

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Cl

SCH

3

4993

OCH

3

OCH

3

Br

Cl

SCH

3

4994

OCH

2

CH

3

OCH

2

CH

3

Br

Cl

SCH

3

4995

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Cl

SCH

3

4996

SCH

3

SCH

3

Br

Cl

SCH

3

4997

SCH

2

CH

3

SCH

2

CH

3

Br

Cl

SCH

3

4998

N(CH

3

)

2

N(CH

3

)

2

Br

Cl

SCH

3

4999

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Cl

SCH

3

5000

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Cl

SCH

3

5001

O—(CH

2

CH

2

)—O

Br

Cl

SCH

3

5002

O—(CH

2

CH

2

CH

2

)—O

Br

Cl

SCH

3

5003

S—(CH

2

CH

2

)—S

Br

Cl

SCH

3

5004

S—(CH

2

CH

2

CH

2

)—S

Br

Cl

SCH

3

5005

—(CH

2

)

4

—

Br

Cl

SCH

3

5006

—(CH

2

)

5

—

Br

Cl

SCH

3

5007

H

H

CH

3

Cl

SCH

3

5008

CH

3

CH

3

CH

3

Cl

SCH

3

5009

CH

2

CH

3

CH

2

CH

3

CH

3

Cl

SCH

3

5010

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Cl

SCH

3

5011

OCH

3

OCH

3

CH

3

Cl

SCH

3

5012

OCH

2

CH

3

OCH

2

CH

3

CH

3

Cl

SCH

3

5013

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Cl

SCH

3

5014

SCH

3

SCH

3

CH

3

Cl

SCH

3

5015

SCH

2

CH

3

SCH

2

CH

3

CH

3

Cl

SCH

3

5016

N(CH

3

)

2

N(CH

3

)

2

CH

3

Cl

SCH

3

5017

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Cl

SCH

3

5018

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Cl

SCH

3

5019

O—(CH

2

CH

2

)—O

CH

3

Cl

SCH

3

5020

O—(CH

2

CH

2

CH

2

)—O

CH

3

Cl

SCH

3

5021

S—(CH

2

CH

2

)—S

CH

3

Cl

SCH

3

5022

S—(CH

2

CH

2

CH

2

)—S

CH

3

Cl

SCH

3

5023

—(CH

2

)

4

—

CH

3

Cl

SCH

3

5024

—(CH

2

)

5

—

CH

3

Cl

SCH

3

5025

H

H

CH

2

CH

3

Cl

SCH

3

5026

CH

3

CH

3

CH

2

CH

3

Cl

SCH

3

5027

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Cl

SCH

3

5028

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Cl

SCH

3

5029

OCH

3

OCH

3

CH

2

CH

3

Cl

SCH

3

5030

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Cl

SCH

3

5031

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Cl

SCH

3

5032

SCH

3

SCH

3

CH

2

CH

3

Cl

SCH

3

5033

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Cl

SCH

3

5034

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Cl

SCH

3

5035

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Cl

SCH

3

5036

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Cl

SCH

3

5037

O—(CH

2

CH

2

)—O

CH

2

CH

3

Cl

SCH

3

5038

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Cl

SCH

3

5039

S—(CH

2

CH

2

)—S

CH

2

CH

3

Cl

SCH

3

5040

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Cl

SCH

3

5041

—(CH

2

)

4

—

CH

2

CH

3

Cl

SCH

3

5042

—(CH

2

)

5

—

CH

2

CH

3

Cl

SCH

3

5043

H

H

CF

3

Cl

SCH

3

5044

CH

3

CH

3

CF

3

Cl

SCH

3

5045

CH

2

CH

3

CH

2

CH

3

CF

3

Cl

SCH

3

5046

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Cl

SCH

3

5047

OCH

3

OCH

3

CF

3

Cl

SCH

3

5048

OCH

2

CH

3

OCH

2

CH

3

CF

3

Cl

SCH

3

5049

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Cl

SCH

3

5050

SCH

3

SCH

3

CF

3

Cl

SCH

3

5051

SCH

2

CH

3

SCH

2

CH

3

CF

3

Cl

SCH

3

5052

N(CH

3

)

2

N(CH

3

)

2

CF

3

Cl

SCH

3

5053

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Cl

SCH

3

5054

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Cl

SCH

3

5055

O—(CH

2

CH

2

)—O

CF

3

Cl

SCH

3

5056

O—(CH

2

CH

2

CH

2

)—O

CF

3

Cl

SCH

3

5057

S—(CH

2

CH

2

)—S

CF

3

Cl

SCH

3

5058

S—(CH

2

CH

2

CH

2

)—S

CF

3

Cl

SCH

3

5059

—(CH

2

)

4

—

CF

3

Cl

SCH

3

5060

—(CH

2

)

5

—

CF

3

Cl

SCH

3

5061

H

H

OCH

3

Cl

SCH

3

5062

CH

3

CH

3

OCH

3

Cl

SCH

3

5063

CH

2

CH

3

CH

2

CH

3

OCH

3

Cl

SCH

3

5064

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Cl

SCH

3

5065

OCH

3

OCH

3

OCH

3

Cl

SCH

3

5066

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Cl

SCH

3

5067

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Cl

SCH

3

5068

SCH

3

SCH

3

OCH

3

Cl

SCH

3

5069

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Cl

SCH

3

5070

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Cl

SCH

3

5071

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Cl

SCH

3

5072

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Cl

SCH

3

5073

O—(CH

2

CH

2

)—O

OCH

3

Cl

SCH

3

5074

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Cl

SCH

3

5075

S—(CH

2

CH

2

)—S

OCH

3

Cl

SCH

3

5076

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Cl

SCH

3

5077

—(CH

2

)

4

—

OCH

3

Cl

SCH

3

5078

—(CH

2

)

5

—

OCH

3

Cl

SCH

3

5079

H

H

OCH

2

CH

3

Cl

SCH

3

5080

CH

3

CH

3

OCH

2

CH

3

Cl

SCH

3

5081

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Cl

SCH

3

5082

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Cl

SCH

3

5083

OCH

3

OCH

3

OCH

2

CH

3

Cl

SCH

3

5084

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Cl

SCH

3

5085

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Cl

SCH

3

5086

SCH

3

SCH

3

OCH

2

CH

3

Cl

SCH

3

5087

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Cl

SCH

3

5088

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Cl

SCH

3

5089

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Cl

SCH

3

5090

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Cl

SCH

3

5091

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Cl

SCH

3

5092

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Cl

SCH

3

5093

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Cl

SCH

3

5094

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Cl

SCH

3

5095

—(CH

2

)

4

—

OCH

2

CH

3

Cl

SCH

3

5096

—(CH

2

)

5

—

OCH

2

CH

3

Cl

SCH

3

5097

H

H

SCH

3

Cl

SCH

3

5098

CH

3

CH

3

SCH

3

Cl

SCH

3

5099

CH

2

CH

3

CH

2

CH

3

SCH

3

Cl

SCH

3

5100

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Cl

SCH

3

5101

OCH

3

OCH

3

SCH

3

Cl

SCH

3

5102

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Cl

SCH

3

5103

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Cl

SCH

3

5104

SCH

3

SCH

3

SCH

3

Cl

SCH

3

5105

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Cl

SCH

3

5106

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Cl

SCH

3

5107

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Cl

SCH

3

5108

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Cl

SCH

3

5109

O—(CH

2

CH

2

)—O

SCH

3

Cl

SCH

3

5110

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Cl

SCH

3

5111

S—(CH

2

CH

2

)—S

SCH

3

Cl

SCH

3

5112

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Cl

SCH

3

5113

—(CH

2

)

4

—

SCH

3

Cl

SCH

3

5114

—(CH

2

)

5

—

SCH

3

Cl

SCH

3

5115

H

H

SO

2

CH

3

Cl

SCH

3

5116

CH

3

CH

3

SO

2

CH

3

Cl

SCH

3

5117

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Cl

SCH

3

5118

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Cl

SCH

3

5119

OCH

3

OCH

3

SO

2

CH

3

Cl

SCH

3

5120

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Cl

SCH

3

5121

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Cl

SCH

3

5122

SCH

3

SCH

3

SO

2

CH

3

Cl

SCH

3

5123

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Cl

SCH

3

5124

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Cl

SCH

3

5125

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Cl

SCH

3

5126

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Cl

SCH

3

5127

O—(CH

2

CH

2

)—O

SO

2

CH

3

Cl

SCH

3

5128

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Cl

SCH

3

5129

S—(CH

2

CH

2

)—S

SO

2

CH

3

Cl

SCH

3

5130

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Cl

SCH

3

5131

—(CH

2

)

4

—

SO

2

CH

3

Cl

SCH

3

5132

—(CH

2

)

5

—

SO

2

CH

3

Cl

SCH

3

5133

H

H

PO(OCH

3

)

2

Cl

SCH

3

5134

CH

3

CH

3

PO(OCH

3

)

2

Cl

SCH

3

5135

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Cl

SCH

3

5136

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

SCH

3

5137

OCH

3

OCH

3

PO(OCH

3

)

2

Cl

SCH

3

5138

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Cl

SCH

3

5139

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

SCH

3

5140

SCH

3

SCH

3

PO(OCH

3

)

2

Cl

SCH

3

5141

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Cl

SCH

3

5142

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Cl

SCH

3

5143

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Cl

SCH

3

5144

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Cl

SCH

3

5145

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

SCH

3

5146

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

SCH

3

5147

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

SCH

3

5148

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

SCH

3

5149

—(CH

2

)

4

—

PO(OCH

3

)

2

Cl

SCH

3

5150

—(CH

2

)

5

—

PO(OCH

3

)

2

Cl

SCH

3

5151

H

H

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5152

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5153

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5154

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5155

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5156

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5157

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5158

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5159

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5160

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5161

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5162

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5163

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5164

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5165

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5166

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5167

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5168

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Cl

SCH

3

5169

H

H

PO(CH

3

)

2

Cl

SCH

3

5170

CH

3

CH

3

PO(CH

3

)

2

Cl

SCH

3

5171

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Cl

SCH

3

5172

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

SCH

3

5173

OCH

3

OCH

3

PO(CH

3

)

2

Cl

SCH

3

5174

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Cl

SCH

3

5175

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

SCH

3

5176

SCH

3

SCH

3

PO(CH

3

)

2

Cl

SCH

3

5177

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Cl

SCH

3

5178

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Cl

SCH

3

5179

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Cl

SCH

3

5180

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Cl

SCH

3

5181

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

SCH

3

5182

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

SCH

3

5183

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

SCH

3

5184

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

SCH

3

5185

—(CH

2

)

4

—

PO(CH

3

)

2

Cl

SCH

3

5186

—(CH

2

)

5

—

PO(CH

3

)

2

Cl

SCH

3

5187

H

H

PO(CH

2

CH

3

)

2

Cl

SCH

3

5188

CH

3

CH

3

PO(CH

2

CH

3

)

2

Cl

SCH

3

5189

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

SCH

3

5190

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

SCH

3

5191

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

Cl

SCH

3

5192

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

SCH

3

5193

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

SCH

3

5194

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

Cl

SCH

3

5195

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

Cl

SCH

3

5196

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

Cl

SCH

3

5197

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

Cl

SCH

3

5198

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

Cl

SCH

3

5199

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

Cl

SCH

3

5200

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

Cl

SCH

3

5201

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

Cl

SCH

3

5202

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

Cl

SCH

3

5203

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

Cl

SCH

3

5204

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

Cl

SCH

3

5205

H

H

H

Cl

SC

6

H

5

5206

CH

3

CH

3

H

Cl

SC

6

H

5

5207

CH

2

CH

3

CH

2

CH

3

H

Cl

SC

6

H

5

5208

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Cl

SC

6

H

5

5209

OCH

3

OCH

3

H

Cl

SC

6

H

5

5210

OCH

2

CH

3

OCH

2

CH

3

H

Cl

SC

6

H

5

5211

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Cl

SC

6

H

5

5212

SCH

3

SCH

3

H

Cl

SC

6

H

5

5213

SCH

2

CH

3

SCH

2

CH

3

H

Cl

SC

6

H

5

5214

N(CH

3

)

2

N(CH

3

)

2

H

Cl

SC

6

H

5

5215

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Cl

SC

6

H

5

5216

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Cl

SC

6

H

5

5217

O—(CH

2

CH

2

)—O

H

Cl

SC

6

H

5

5218

O—(CH

2

CH

2

CH

2

)—O

H

Cl

SC

6

H

5

5219

S—(CH

2

CH

2

)—S

H

Cl

SC

6

H

5

5220

S—(CH

2

CH

2

CH

2

)—S

H

Cl

SC

6

H

5

5221

—(CH

2

)

4

—

H

Cl

SC

6

H

5

5222

—(CH

2

)

5

—

H

Cl

SC

6

H

5

5223

H

H

NO

2

Cl

SC

6

H

5

5224

CH

3

CH

3

NO

2

Cl

SC

6

H

5

5225

CH

2

CH

3

CH

2

CH

3

NO

2

Cl

SC

6

H

5

5226

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Cl

SC

6

H

5

5227

OCH

3

OCH

3

NO

2

Cl

SC

6

H

5

5228

OCH

2

CH

3

OCH

2

CH

3

NO

2

Cl

SC

6

H

5

5229

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Cl

SC

6

H

5

5230

SCH

3

SCH

3

NO

2

Cl

SC

6

H

5

5231

SCH

2

CH

3

SCH

2

CH

3

NO

2

Cl

SC

6

H

5

5232

N(CH

3

)

2

N(CH

3

)

2

NO

2

Cl

SC

6

H

5

5233

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Cl

SC

6

H

5

5234

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Cl

SC

6

H

5

5235

O—(CH

2

CH

2

)—O

NO

2

Cl

SC

6

H

5

5236

O—(CH

2

CH

2

CH

2

)—O

NO

2

Cl

SC

6

H

5

5237

S—(CH

2

CH

2

)—S

NO

2

Cl

SC

6

H

5

5238

S—(CH

2

CH

2

CH

2

)—S

NO

2

Cl

SC

6

H

5

5239

—(CH

2

)

4

—

NO

2

Cl

SC

6

H

5

5240

—(CH

2

)

5

—

NO

2

Cl

SC

6

H

5

5241

H

H

CN

Cl

SC

6

H

5

5242

CH

3

CH

3

CN

Cl

SC

6

H

5

5243

CH

2

CH

3

CH

2

CH

3

CN

Cl

SC

6

H

5

5244

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Cl

SC

6

H

5

5245

OCH

3

OCH

3

CN

Cl

SC

6

H

5

5246

OCH

2

CH

3

OCH

2

CH

3

CN

Cl

SC

6

H

5

5247

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Cl

SC

6

H

5

5248

SCH

3

SCH

3

CN

Cl

SC

6

H

5

5249

SCH

2

CH

3

SCH

2

CH

3

CN

Cl

SC

6

H

5

5250

N(CH

3

)

2

N(CH

3

)

2

CN

Cl

SC

6

H

5

5251

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Cl

SC

6

H

5

5252

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Cl

SC

6

H

5

5253

O—(CH

2

CH

2

)—O

CN

Cl

SC

6

H

5

5254

O—(CH

2

CH

2

CH

2

)—O

CN

Cl

SC

6

H

5

5255

S—(CH

2

CH

2

)—S

CN

Cl

SC

6

H

5

5256

S—(CH

2

CH

2

CH

2

)—S

CN

Cl

SC

6

H

5

5257

—(CH

2

)

4

—

CN

Cl

SC

6

H

5

5258

—(CH

2

)

5

—

CN

Cl

SC

6

H

5

5259

H

H

F

Cl

SC

6

H

5

5260

CH

3

CH

3

F

Cl

SC

6

H

5

5261

CH

2

CH

3

CH

2

CH

3

F

Cl

SC

6

H

5

5262

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Cl

SC

6

H

5

5263

OCH

3

OCH

3

F

Cl

SC

6

H

5

5264

OCH

2

CH

3

OCH

2

CH

3

F

Cl

SC

6

H

5

5265

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Cl

SC

6

H

5

5266

SCH

3

SCH

3

F

Cl

SC

6

H

5

5267

SCH

2

CH

3

SCH

2

CH

3

F

Cl

SC

6

H

5

5268

N(CH

3

)

2

N(CH

3

)

2

F

Cl

SC

6

H

5

5269

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Cl

SC

6

H

5

5270

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Cl

SC

6

H

5

5271

O—(CH

2

CH

2

)—O

F

Cl

SC

6

H

5

5272

O—(CH

2

CH

2

CH

2

)—O

F

Cl

SC

6

H

5

5273

S—(CH

2

CH

2

)—S

F

Cl

SC

6

H

5

5274

S—(CH

2

CH

2

CH

2

)—S

F

Cl

SC

6

H

5

5275

—(CH

2

)

4

—

F

Cl

SC

6

H

5

5276

—(CH

2

)

5

—

F

Cl

SC

6

H

5

5277

H

H

Cl

Cl

SC

6

H

5

5278

CH

3

CH

3

Cl

Cl

SC

6

H

5

5279

CH

2

CH

3

CH

2

CH

3

Cl

Cl

SC

6

H

5

5280

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Cl

SC

6

H

5

5281

OCH

3

OCH

3

Cl

Cl

SC

6

H

5

5282

OCH

2

CH

3

OCH

2

CH

3

Cl

Cl

SC

6

H

5

5283

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Cl

SC

6

H

5

5284

SCH

3

SCH

3

Cl

Cl

SC

6

H

5

5285

SCH

2

CH

3

SCH

2

CH

3

Cl

Cl

SC

6

H

5

5286

N(CH

3

)

2

N(CH

3

)

2

Cl

Cl

SC

6

H

5

5287

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Cl

SC

6

H

5

5288

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Cl

SC

6

H

5

5289

O—(CH

2

CH

2

)—O

Cl

Cl

SC

6

H

5

5290

O—(CH

2

CH

2

CH

2

)—O

Cl

Cl

SC

6

H

5

5291

S—(CH

2

CH

2

)—S

Cl

Cl

SC

6

H

5

5292

S—(CH

2

CH

2

CH

2

)—S

Cl

Cl

SC

6

H

5

5293

—(CH

2

)

4

—

Cl

Cl

SC

6

H

5

5294

—(CH

2

)

5

—

Cl

Cl

SC

6

H

5

5295

H

H

Br

Cl

SC

6

H

5

5296

CH

3

CH

3

Br

Cl

SC

6

H

5

5297

CH

2

CH

3

CH

2

CH

3

Br

Cl

SC

6

H

5

5298

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Cl

SC

6

H

5

5299

OCH

3

OCH

3

Br

Cl

SC

6

H

5

5300

OCH

2

CH

3

OCH

2

CH

3

Br

Cl

SC

6

H

5

5301

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Cl

SC

6

H

5

5302

SCH

3

SCH

3

Br

Cl

SC

6

H

5

5303

SCH

2

CH

3

SCH

2

CH

3

Br

Cl

SC

6

H

5

5304

N(CH

3

)

2

N(CH

3

)

2

Br

Cl

SC

6

H

5

5305

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Cl

SC

6

H

5

5306

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Cl

SC

6

H

5

5307

O—(CH

2

CH

2

)—O

Br

Cl

SC

6

H

5

5308

O—(CH

2

CH

2

CH

2

)—O

Br

Cl

SC

6

H

5

5309

S—(CH

2

CH

2

)—S

Br

Cl

SC

6

H

5

5310

S—(CH

2

CH

2

CH

2

)—S

Br

Cl

SC

6

H

5

5311

—(CH

2

)

4

—

Br

Cl

SC

6

H

5

5312

—(CH

2

)

5

—

Br

Cl

SC

6

H

5

5313

H

H

CH

3

Cl

SC

6

H

5

5314

CH

3

CH

3

CH

3

Cl

SC

6

H

5

5315

CH

2

CH

3

CH

2

CH

3

CH

3

Cl

SC

6

H

5

5316

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Cl

SC

6

H

5

5317

OCH

3

OCH

3

CH

3

Cl

SC

6

H

5

5318

OCH

2

CH

3

OCH

2

CH

3

CH

3

Cl

SC

6

H

5

5319

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Cl

SC

6

H

5

5320

SCH

3

SCH

3

CH

3

Cl

SC

6

H

5

5321

SCH

2

CH

3

SCH

2

CH

3

CH

3

Cl

SC

6

H

5

5322

N(CH

3

)

2

N(CH

3

)

2

CH

3

Cl

SC

6

H

5

5323

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Cl

SC

6

H

5

5324

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Cl

SC

6

H

5

5325

O—(CH

2

CH

2

)—O

CH

3

Cl

SC

6

H

5

5326

O—(CH

2

CH

2

CH

2

)—O

CH

3

Cl

SC

6

H

5

5327

S—(CH

2

CH

2

)—S

CH

3

Cl

SC

6

H

5

5328

S—(CH

2

CH

2

CH

2

)—S

CH

3

Cl

SC

6

H

5

5329

—(CH

2

)

4

—

CH

3

Cl

SC

6

H

5

5330

—(CH

2

)

5

—

CH

3

Cl

SC

6

H

5

5331

H

H

CH

2

CH

3

Cl

SC

6

H

5

5332

CH

3

CH

3

CH

2

CH

3

Cl

SC

6

H

5

5333

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Cl

SC

6

H

5

5334

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Cl

SC

6

H

5

5335

OCH

3

OCH

3

CH

2

CH

3

Cl

SC

6

H

5

5336

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Cl

SC

6

H

5

5337

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Cl

SC

6

H

5

5338

SCH

3

SCH

3

CH

2

CH

3

Cl

SC

6

H

5

5339

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Cl

SC

6

H

5

5340

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Cl

SC

6

H

5

5341

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Cl

SC

6

H

5

5342

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Cl

SC

6

H

5

5343

O—(CH

2

CH

2

)—O

CH

2

CH

3

Cl

SC

6

H

5

5344

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Cl

SC

6

H

5

5345

S—(CH

2

CH

2

)—S

CH

2

CH

3

Cl

SC

6

H

5

5346

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Cl

SC

6

H

5

5347

—(CH

2

)

4

—

CH

2

CH

3

Cl

SC

6

H

5

5348

—(CH

2

)

5

—

CH

2

CH

3

Cl

SC

6

H

5

5349

H

H

CF

3

Cl

SC

6

H

5

5350

CH

3

CH

3

CF

3

Cl

SC

6

H

5

5351

CH

2

CH

3

CH

2

CH

3

CF

3

Cl

SC

6

H

5

5352

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Cl

SC

6

H

5

5353

OCH

3

OCH

3

CF

3

Cl

SC

6

H

5

5354

OCH

2

CH

3

OCH

2

CH

3

CF

3

Cl

SC

6

H

5

5355

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Cl

SC

6

H

5

5356

SCH

3

SCH

3

CF

3

Cl

SC

6

H

5

5357

SCH

2

CH

3

SCH

2

CH

3

CF

3

Cl

SC

6

H

5

5358

N(CH

3

)

2

N(CH

3

)

2

CF

3

Cl

SC

6

H

5

5359

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Cl

SC

6

H

5

5360

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Cl

SC

6

H

5

5361

O—(CH

2

CH

2

)—O

CF

3

Cl

SC

6

H

5

5362

O—(CH

2

CH

2

CH

2

)—O

CF

3

Cl

SC

6

H

5

5363

S—(CH

2

CH

2

)—S

CF

3

Cl

SC

6

H

5

5364

S—(CH

2

CH

2

CH

2

)—S

CF

3

Cl

SC

6

H

5

5365

—(CH

2

)

4

—

CF

3

Cl

SC

6

H

5

5366

—(CH

2

)

5

—

CF

3

Cl

SC

6

H

5

5367

H

H

OCH

3

Cl

SC

6

H

5

5368

CH

3

CH

3

OCH

3

Cl

SC

6

H

5

5369

CH

2

CH

3

CH

2

CH

3

OCH

3

Cl

SC

6

H

5

5370

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Cl

SC

6

H

5

5371

OCH

3

OCH

3

OCH

3

Cl

SC

6

H

5

5372

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Cl

SC

6

H

5

5373

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Cl

SC

6

H

5

5374

SCH

3

SCH

3

OCH

3

Cl

SC

6

H

5

5375

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Cl

SC

6

H

5

5376

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Cl

SC

6

H

5

5377

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Cl

SC

6

H

5

5378

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Cl

SC

6

H

5

5379

O—(CH

2

CH

2

)—O

OCH

3

Cl

SC

6

H

5

5380

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Cl

SC

6

H

5

5381

S—(CH

2

CH

2

)—S

OCH

3

Cl

SC

6

H

5

5382

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Cl

SC

6

H

5

5383

—(CH

2

)

4

—

OCH

3

Cl

SC

6

H

5

5384

—(CH

2

)

5

—

OCH

3

Cl

SC

6

H

5

5385

H

H

OCH

2

CH

3

Cl

SC

6

H

5

5386

CH

3

CH

3

OCH

2

CH

3

Cl

SC

6

H

5

5387

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Cl

SC

6

H

5

5388

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Cl

SC

6

H

5

5389

OCH

3

OCH

3

OCH

2

CH

3

Cl

SC

6

H

5

5390

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Cl

SC

6

H

5

5391

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Cl

SC

6

H

5

5392

SCH

3

SCH

3

OCH

2

CH

3

Cl

SC

6

H

5

5393

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Cl

SC

6

H

5

5394

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Cl

SC

6

H

5

5395

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Cl

SC

6

H

5

5396

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Cl

SC

6

H

5

5397

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Cl

SC

6

H

5

5398

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Cl

SC

6

H

5

5399

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Cl

SC

6

H

5

5400

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Cl

SC

6

H

5

5401

—(CH

2

)

4

—

OCH

2

CH

3

Cl

SC

6

H

5

5402

—(CH

2

)

5

—

OCH

2

CH

3

Cl

SC

6

H

5

5403

H

H

SCH

3

Cl

SC

6

H

5

5404

CH

3

CH

3

SCH

3

Cl

SC

6

H

5

5405

CH

2

CH

3

CH

2

CH

3

SCH

3

Cl

SC

6

H

5

5406

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Cl

SC

6

H

5

5407

OCH

3

OCH

3

SCH

3

Cl

SC

6

H

5

5408

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Cl

SC

6

H

5

5409

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Cl

SC

6

H

5

5410

SCH

3

SCH

3

SCH

3

Cl

SC

6

H

5

5411

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Cl

SC

6

H

5

5412

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Cl

SC

6

H

5

5413

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Cl

SC

6

H

5

5414

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Cl

SC

6

H

5

5415

O—(CH

2

CH

2

)—O

SCH

3

Cl

SC

6

H

5

5416

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Cl

SC

6

H

5

5417

S—(CH

2

CH

2

)—S

SCH

3

Cl

SC

6

H

5

5418

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Cl

SC

6

H

5

5419

—(CH

2

)

4

—

SCH

3

Cl

SC

6

H

5

5420

—(CH

2

)

5

—

SCH

3

Cl

SC

6

H

5

5421

H

H

SO

2

CH

3

Cl

SC

6

H

5

5422

CH

3

CH

3

SO

2

CH

3

Cl

SC

6

H

5

5423

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Cl

SC

6

H

5

5424

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Cl

SC

6

H

5

5425

OCH

3

OCH

3

SO

2

CH

3

Cl

SC

6

H

5

5426

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Cl

SC

6

H

5

5427

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Cl

SC

6

H

5

5428

SCH

3

SCH

3

SO

2

CH

3

Cl

SC

6

H

5

5429

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Cl

SC

6

H

5

5430

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Cl

SC

6

H

5

5431

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Cl

SC

6

H

5

5432

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Cl

SC

6

H

5

5433

O—(CH

2

CH

2

)—O

SO

2

CH

3

Cl

SC

6

H

5

5434

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Cl

SC

6

H

5

5435

S—(CH

2

CH

2

)—S

SO

2

CH

3

Cl

SC

6

H

5

5436

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Cl

SC

6

H

5

5437

—(CH

2

)

4

—

SO

2

CH

3

Cl

SC

6

H

5

5438

—(CH

2

)

5

—

SO

2

CH

3

Cl

SC

6

H

5

5439

H

H

PO(OCH

3

)

2

Cl

SC

6

H

5

5440

CH

3

CH

3

PO(OCH

3

)

2

Cl

SC

6

H

5

5441

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Cl

SC

6

H

5

5442

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

SC

6

H

5

5443

OCH

3

OCH

3

PO(OCH

3

)

2

Cl

SC

6

H

5

5444

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Cl

SC

6

H

5

5445

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

SC

6

H

5

5446

SCH

3

SCH

3

PO(OCH

3

)

2

Cl

SC

6

H

5

5447

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Cl

SC

6

H

5

5448

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Cl

SC

6

H

5

5449

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Cl

SC

6

H

5

5450

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Cl

SC

6

H

5

5451

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

SC

6

H

5

5452

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

SC

6

H

5

5453

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

SC

6

H

5

5454

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

SC

6

H

5

5455

—(CH

2

)

4

—

PO(OCH

3

)

2

Cl

SC

6

H

5

5456

—(CH

2

)

5

—

PO(OCH

3

)

2

Cl

SC

6

H

5

5457

H

H

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5458

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5459

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5460

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5461

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5462

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5463

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5464

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5465

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5466

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5467

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5468

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5469

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5470

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5471

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5472

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5473

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5474

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Cl

SC

6

H

5

5475

H

H

PO(CH

3

)

2

Cl

SC

6

H

5

5476

CH

3

CH

3

PO(CH

3

)

2

Cl

SC

6

H

5

5477

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Cl

SC

6

H

5

5478

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

SC

6

H

5

5479

OCH

3

OCH

3

PO(CH

3

)

2

Cl

SC

6

H

5

5480

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Cl

SC

6

H

5

5481

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

SC

6

H

5

5482

SCH

3

SCH

3

PO(CH

3

)

2

Cl

SC

6

H

5

5483

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Cl

SC

6

H

5

5484

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Cl

SC

6

H

5

5485

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Cl

SC

6

H

5

5486

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Cl

SC

6

H

5

5487

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

SC

6

H

5

5488

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

SC

6

H

5

5489

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

SC

6

H

5

5490

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

SC

6

H

5

5491

—(CH

2

)

4

—

PO(CH

3

)

2

Cl

SC

6

H

5

5492

—(CH

2

)

5

—

PO(CH

3

)

2

Cl

SC

6

H

5

5493

H

H

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5494

CH

3

CH

3

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5495

CH

2

CH

3

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5496

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5497

OCH

3

OCH

3

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5498

OCH

2

CH

3

OCH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5499

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5500

SCH

3

SCH

3

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5501

SCH

2

CH

3

SCH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5502

N(CH

3

)

2

N(CH

3

)

2

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5503

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5504

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5505

O—(CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5506

O—(CH

2

CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5507

S—(CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5508

S—(CH

2

CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5509

—(CH

2

)

4

—

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5510

—(CH

2

)

5

—

PC(CH

2

CH

3

)

2

Cl

SC

6

H

5

5511

H

H

H

Cl

Het1

5512

CH

3

CH

3

H

Cl

Het1

5513

CH

2

CH

3

CH

2

CH

3

H

Cl

Het1

5514

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Cl

Het1

5515

OCH

3

OCH

3

H

Cl

Het1

5516

OCH

2

CH

3

OCH

2

CH

3

H

Cl

Het1

5517

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Cl

Het1

5518

SCH

3

SCH

3

H

Cl

Het1

5519

SCH

2

CH

3

SCH

2

CH

3

H

Cl

Het1

5520

N(CH

3

)

2

N(CH

3

)

2

H

Cl

Het1

5521

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Cl

Het1

5522

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Cl

Het1

5523

O—(CH

2

CH

2

)—O

H

Cl

Het1

5524

O—(CH

2

CH

2

CH

2

)—O

H

Cl

Het1

5525

S—(CH

2

CH

2

)—S

H

Cl

Het1

5526

S—(CH

2

CH

2

CH

2

)—S

H

Cl

Het1

5527

—(CH

2

)

4

—

H

Cl

Het1

5528

—(CH

2

)

5

—

H

Cl

Het1

5529

H

H

NO

2

Cl

Het1

5530

CH

3

CH

3

NO

2

Cl

Het1

5531

CH

2

CH

3

CH

2

CH

3

NO

2

Cl

Het1

5532

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Cl

Het1

5533

OCH

3

OCH

3

NO

2

Cl

Het1

5534

OCH

2

CH

3

OCH

2

CH

3

NO

2

Cl

Het1

5535

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Cl

Het1

5536

SCH

3

SCH

3

NO

2

Cl

Het1

5537

SCH

2

CH

3

SCH

2

CH

3

NO

2

Cl

Het1

5538

N(CH

3

)

2

N(CH

3

)

2

NO

2

Cl

Het1

5539

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Cl

Het1

5540

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Cl

Het1

5541

O—(CH

2

CH

2

)—O

NO

2

Cl

Het1

5542

O—(CH

2

CH

2

CH

2

)—O

NO

2

Cl

Het1

5543

S—(CH

2

CH

2

)—S

NO

2

Cl

Het1

5544

S—(CH

2

CH

2

CH

2

)—S

NO

2

Cl

Het1

5545

—(CH

2

)

4

—

NO

2

Cl

Het1

5546

—(CH

2

)

5

—

NO

2

Cl

Het1

5547

H

H

CN

Cl

Het1

5548

CH

3

CH

3

CN

Cl

Het1

5549

CH

2

CH

3

CH

2

CH

3

CN

Cl

Het1

5550

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Cl

Het1

5551

OCH

3

OCH

3

CN

Cl

Het1

5552

OCH

2

CH

3

OCH

2

CH

3

CN

Cl

Het1

5553

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Cl

Het1

5554

SCH

3

SCH

3

CN

Cl

Het1

5555

SCH

2

CH

3

SCH

2

CH

3

CN

Cl

Het1

5556

N(CH

3

)

2

N(CH

3

)

2

CN

Cl

Het1

5557

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Cl

Het1

5558

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Cl

Het1

5559

O—(CH

2

CH

2

)—O

CN

Cl

Het1

5560

O—(CH

2

CH

2

CH

2

)—O

CN

Cl

Het1

5561

S—(CH

2

CH

2

)—S

CN

Cl

Het1

5562

S—(CH

2

CH

2

CH

2

)—S

CN

Cl

Het1

5563

—(CH

2

)

4

—

CN

Cl

Het1

5564

—(CH

2

)

5

—

CN

Cl

Het1

5565

H

H

F

Cl

Het1

5566

CH

3

CH

3

F

Cl

Het1

5567

CH

2

CH

3

CH

2

CH

3

F

Cl

Het1

5568

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Cl

Het1

5569

OCH

3

OCH

3

F

Cl

Het1

5570

OCH

2

CH

3

OCH

2

CH

3

F

Cl

Het1

5571

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Cl

Het1

5572

SCH

3

SCH

3

F

Cl

Het1

5573

SCH

2

CH

3

SCH

2

CH

3

F

Cl

Het1

5574

N(CH

3

)

2

N(CH

3

)

2

F

Cl

Het1

5575

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Cl

Het1

5576

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Cl

Het1

5577

O—(CH

2

CH

2

)—O

F

Cl

Het1

5578

O—(CH

2

CH

2

CH

2

)—O

F

Cl

Het1

5579

S—(CH

2

CH

2

)—S

F

Cl

Het1

5580

S—(CH

2

CH

2

CH

2

)—S

F

Cl

Het1

5581

—(CH

2

)

4

—

F

Cl

Het1

5582

—(CH

2

)

5

—

F

Cl

Het1

5583

H

H

Cl

Cl

Het1

5584

CH

3

CH

3

Cl

Cl

Het1

5585

CH

2

CH

3

CH

2

CH

3

Cl

Cl

Het1

5586

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Cl

Het1

5587

OCH

3

OCH

3

Cl

Cl

Het1

5588

OCH

2

CH

3

OCH

2

CH

3

Cl

Cl

Het1

5589

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Cl

Het1

5590

SCH

3

SCH

3

Cl

Cl

Het1

5591

SCH

2

CH

3

SCH

2

CH

3

Cl

Cl

Het1

5592

N(CH

3

)

2

N(CH

3

)

2

Cl

Cl

Het1

5593

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Cl

Het1

5594

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Cl

Het1

5595

O—(CH

2

CH

2

)—O

Cl

Cl

Het1

5596

O—(CH

2

CH

2

CH

2

)—O

Cl

Cl

Het1

5597

S—(CH

2

CH

2

)—S

Cl

Cl

Het1

5598

S—(CH

2

CH

2

CH

2

)—S

Cl

Cl

Het1

5599

—(CH

2

)

4

—

Cl

Cl

Het1

5600

—(CH

2

)

5

—

Cl

Cl

Het1

5601

H

H

Br

Cl

Het1

5602

CH

3

CH

3

Br

Cl

Het1

5603

CH

2

CH

3

CH

2

CH

3

Br

Cl

Het1

5604

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Cl

Het1

5605

OCH

3

OCH

3

Br

Cl

Het1

5606

OCH

2

CH

3

OCH

2

CH

3

Br

Cl

Het1

5607

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Cl

Het1

5608

SCH

3

SCH

3

Br

Cl

Het1

5609

SCH

2

CH

3

SCH

2

CH

3

Br

Cl

Het1

5610

N(CH

3

)

2

N(CH

3

)

2

Br

Cl

Het1

5611

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Cl

Het1

5612

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Cl

Het1

5613

O—(CH

2

CH

2

)—O

Br

Cl

Het1

5614

O—(CH

2

CH

2

CH

2

)—O

Br

Cl

Het1

5615

S—(CH

2

CH

2

)—S

Br

Cl

Het1

5616

S—(CH

2

CH

2

CH

2

)—S

Br

Cl

Het1

5617

—(CH

2

)

4

—

Br

Cl

Het1

5618

—(CH

2

)

5

—

Br

Cl

Het1

5619

H

H

CH

3

Cl

Het1

5620

CH

3

CH

3

CH

3

Cl

Het1

5621

CH

2

CH

3

CH

2

CH

3

CH

3

Cl

Het1

5622

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Cl

Het1

5623

OCH

3

OCH

3

CH

3

Cl

Het1

5624

OCH

2

CH

3

OCH

2

CH

3

CH

3

Cl

Het1

5625

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Cl

Het1

5626

SCH

3

SCH

3

CH

3

Cl

Het1

5627

SCH

2

CH

3

SCH

2

CH

3

CH

3

Cl

Het1

5628

N(CH

3

)

2

N(CH

3

)

2

CH

3

Cl

Het1

5629

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Cl

Het1

5630

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Cl

Het1

5631

O—(CH

2

CH

2

)—O

CH

3

Cl

Het1

5632

O—(CH

2

CH

2

CH

2

)—O

CH

3

Cl

Het1

5633

S—(CH

2

CH

2

)—S

CH

3

Cl

Het1

5634

S—(CH

2

CH

2

CH

2

)—S

CH

3

Cl

Het1

5635

—(CH

2

)

4

—

CH

3

Cl

Het1

5636

—(CH

2

)

5

—

CH

3

Cl

Het1

5637

H

H

CH

2

CH

3

Cl

Het1

5638

CH

3

CH

3

CH

2

CH

3

Cl

Het1

5639

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Cl

Het1

5640

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Cl

Het1

5641

OCH

3

OCH

3

CH

2

CH

3

Cl

Het1

5642

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Cl

Het1

5643

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Cl

Het1

5644

SCH

3

SCH

3

CH

2

CH

3

Cl

Het1

5645

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Cl

Het1

5646

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Cl

Het1

5647

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Cl

Het1

5648

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Cl

Het1

5649

O—(CH

2

CH

2

)—O

CH

2

CH

3

Cl

Het1

5650

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Cl

Het1

5651

S—(CH

2

CH

2

)—S

CH

2

CH

3

Cl

Het1

5652

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Cl

Het1

5653

—(CH

2

)

4

—

CH

2

CH

3

Cl

Het1

5654

—(CH

2

)

5

—

CH

2

CH

3

Cl

Het1

5655

H

H

CF

3

Cl

Het1

5656

CH

3

CH

3

CF

3

Cl

Het1

5657

CH

2

CH

3

CH

2

CH

3

CF

3

Cl

Het1

5658

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Cl

Het1

5659

OCH

3

OCH

3

CF

3

Cl

Het1

5660

OCH

2

CH

3

OCH

2

CH

3

CF

3

Cl

Het1

5661

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Cl

Het1

5662

SCH

3

SCH

3

CF

3

Cl

Het1

5663

SCH

2

CH

3

SCH

2

CH

3

CF

3

Cl

Het1

5664

N(CH

3

)

2

N(CH

3

)

2

CF

3

Cl

Het1

5665

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Cl

Het1

5666

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Cl

Het1

5667

O—(CH

2

CH

2

)—O

CF

3

Cl

Het1

5668

O—(CH

2

CH

2

CH

2

)—O

CF

3

Cl

Het1

5669

S—(CH

2

CH

2

)—S

CF

3

Cl

Het1

5670

S—(CH

2

CH

2

CH

2

)—S

CF

3

Cl

Het1

5671

—(CH

2

)

4

—

CF

3

Cl

Het1

5672

—(CH

2

)

5

—

CF

3

Cl

Het1

5673

H

H

OCH

3

Cl

Het1

5674

CH

3

CH

3

OCH

3

Cl

Het1

5675

CH

2

CH

3

CH

2

CH

3

OCH

3

Cl

Het1

5676

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Cl

Het1

5677

OCH

3

OCH

3

OCH

3

Cl

Het1

5678

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Cl

Het1

5679

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Cl

Het1

5680

SCH

3

SCH

3

OCH

3

Cl

Het1

5681

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Cl

Het1

5682

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Cl

Het1

5683

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Cl

Het1

5684

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Cl

Het1

5685

O—(CH

2

CH

2

)—O

OCH

3

Cl

Het1

5686

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Cl

Het1

5687

S—(CH

2

CH

2

)—S

OCH

3

Cl

Het1

5688

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Cl

Het1

5689

—(CH

2

)

4

—

OCH

3

Cl

Het1

5690

—(CH

2

)

5

—

OCH

3

Cl

Het1

5691

H

H

OCH

2

CH

3

Cl

Het1

5692

CH

3

CH

3

OCH

2

CH

3

Cl

Het1

5693

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Cl

Het1

5694

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Cl

Het1

5695

OCH

3

OCH

3

OCH

2

CH

3

Cl

Het1

5696

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Cl

Het1

5697

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Cl

Het1

5698

SCH

3

SCH

3

OCH

2

CH

3

Cl

Het1

5699

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Cl

Het1

5700

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Cl

Het1

5701

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Cl

Het1

5702

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Cl

Het1

5703

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Cl

Het1

5704

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Cl

Het1

5705

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Cl

Het1

5706

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Cl

Het1

5707

—(CH

2

)

4

—

OCH

2

CH

3

Cl

Het1

5708

—(CH

2

)

5

—

OCH

2

CH

3

Cl

Het1

5709

H

H

SCH

3

Cl

Het1

5710

CH

3

CH

3

SCH

3

Cl

Het1

5711

CH

2

CH

3

CH

2

CH

3

SCH

3

Cl

Het1

5712

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Cl

Het1

5713

OCH

3

OCH

3

SCH

3

Cl

Het1

5714

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Cl

Het1

5715

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Cl

Het1

5716

SCH

3

SCH

3

SCH

3

Cl

Het1

5717

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Cl

Het1

5718

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Cl

Het1

5719

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Cl

Het1

5720

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Cl

Het1

5721

O—(CH

2

CH

2

)—O

SCH

3

Cl

Het1

5722

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Cl

Het1

5723

S—(CH

2

CH

2

)—S

SCH

3

Cl

Het1

5724

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Cl

Het1

5725

—(CH

2

)

4

—

SCH

3

Cl

Het1

5726

—(CH

2

)

5

—

SCH

3

Cl

Het1

5727

H

H

SO

2

CH

3

Cl

Het1

5728

CH

3

CH

3

SO

2

CH

3

Cl

Het1

5729

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Cl

Het1

5730

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Cl

Het1

5731

OCH

3

OCH

3

SO

2

CH

3

Cl

Het1

5732

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Cl

Het1

5733

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Cl

Het1

5734

SCH

3

SCH

3

SO

2

CH

3

Cl

Het1

5735

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Cl

Het1

5736

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Cl

Het1

5737

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Cl

Het1

5738

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Cl

Het1

5739

O—(CH

2

CH

2

)—O

SO

2

CH

3

Cl

Het1

5740

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Cl

Het1

5741

S—(CH

2

CH

2

)—S

SO

2

CH

3

Cl

Het1

5742

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Cl

Het1

5743

—(CH

2

)

4

—

SO

2

CH

3

Cl

Het1

5744

—(CH

2

)

5

—

SO

2

CH

3

Cl

Het1

5745

H

H

PO(OCH

3

)

2

Cl

Het1

5746

CH

3

CH

3

PO(OCH

3

)

2

Cl

Het1

5747

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Cl

Het1

5748

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

Het1

5749

OCH

3

OCH

3

PO(OCH

3

)

2

Cl

Het1

5750

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Cl

Het1

5751

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

Het1

5752

SCH

3

SCH

3

PO(OCH

3

)

2

Cl

Het1

5753

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Cl

Het1

5754

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Cl

Het1

5755

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Cl

Het1

5756

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Cl

Het1

5757

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

Het1

5758

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

Het1

5759

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

Het1

5760

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

Het1

5761

—(CH

2

)

4

—

PO(OCH

3

)

2

Cl

Het1

5762

—(CH

2

)

5

—

PO(OCH

3

)

2

Cl

Het1

5763

H

H

PO(OCH

2

CH

3

)

2

Cl

Het1

5764

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het1

5765

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het1

5766

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het1

5767

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Cl

Het1

5768

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het1

5769

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het1

5770

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Cl

Het1

5771

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het1

5772

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

Het1

5773

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

Het1

5774

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Cl

Het1

5775

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

Het1

5776

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

Het1

5777

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

Het1

5778

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

Het1

5779

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Cl

Het1

5780

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Cl

Het1

5781

H

H

PO(CH

3

)

2

Cl

Het1

5782

CH

3

CH

3

PO(CH

3

)

2

Cl

Het1

5783

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Cl

Het1

5784

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

Het1

5785

OCH

3

OCH

3

PO(CH

3

)

2

Cl

Het1

5786

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Cl

Het1

5787

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

Het1

5788

SCH

3

SCH

3

PO(CH

3

)

2

Cl

Het1

5789

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Cl

Het1

5790

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Cl

Het1

5791

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Cl

Het1

5792

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Cl

Het1

5793

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

Het1

5794

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

Het1

5795

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

Het1

5796

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

Het1

5797

—(CH

2

)

4

—

PO(CH

3

)

2

Cl

Het1

5798

—(CH

2

)

5

—

PO(CH

3

)

2

Cl

Het1

5799

H

H

PC(CH

2

CH

3

)

2

Cl

Het1

5800

CH

3

CH

3

PC(CH

2

CH

3

)

2

Cl

Het1

5801

CH

2

CH

3

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het1

5802

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het1

5803

OCH

3

OCH

3

PC(CH

2

CH

3

)

2

Cl

Het1

5804

OCH

2

CH

3

OCH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het1

5805

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het1

5806

SCH

3

SCH

3

PC(CH

2

CH

3

)

2

Cl

Het1

5807

SCH

2

CH

3

SCH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het1

5808

N(CH

3

)

2

N(CH

3

)

2

PC(CH

2

CH

3

)

2

Cl

Het1

5809

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PC(CH

2

CH

3

)

2

Cl

Het1

5810

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PC(CH

2

CH

3

)

2

Cl

Het1

5811

O—(CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Cl

Het1

5812

O—(CH

2

CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Cl

Het1

5813

S—(CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Cl

Het1

5814

S—(CH

2

CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Cl

Het1

5815

—(CH

2

)

4

—

PC(CH

2

CH

3

)

2

Cl

Het1

5816

—(CH

2

)

5

—

PC(CH

2

CH

3

)

2

Cl

Het1

5817

H

H

H

Cl

Het2

5818

CH

3

CH

3

H

Cl

Het2

5819

CH

2

CH

3

CH

2

CH

3

H

Cl

Het2

5820

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Cl

Het2

5821

OCH

3

OCH

3

H

Cl

Het2

5822

OCH

2

CH

3

OCH

2

CH

3

H

Cl

Het2

5823

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Cl

Het2

5824

SCH

3

SCH

3

H

Cl

Het2

5825

SCH

2

CH

3

SCH

2

CH

3

H

Cl

Het2

5826

N(CH

3

)

2

N(CH

3

)

2

H

Cl

Het2

5827

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Cl

Het2

5828

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Cl

Het2

5829

O—(CH

2

CH

2

)—O

H

Cl

Het2

5830

O—(CH

2

CH

2

CH

2

)—O

H

Cl

Het2

5831

S—(CH

2

CH

2

)—S

H

Cl

Het2

5832

S—(CH

2

CH

2

CH

2

)—S

H

Cl

Het2

5833

—(CH

2

)

4

—

H

Cl

Het2

5834

—(CH

2

)

5

—

H

Cl

Het2

5835

H

H

NO

2

Cl

Het2

5836

CH

3

CH

3

NO

2

Cl

Het2

5837

CH

2

CH

3

CH

2

CH

3

NO

2

Cl

Het2

5838

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Cl

Het2

5839

OCH

3

OCH

3

NO

2

Cl

Het2

5840

OCH

2

CH

3

OCH

2

CH

3

NO

2

Cl

Het2

5841

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Cl

Het2

5842

SCH

3

SCH

3

NO

2

Cl

Het2

5843

SCH

2

CH

3

SCH

2

CH

3

NO

2

Cl

Het2

5844

N(CH

3

)

2

N(CH

3

)

2

NO

2

Cl

Het2

5845

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Cl

Het2

5846

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Cl

Het2

5847

O—(CH

2

CH

2

)—O

NO

2

Cl

Het2

5848

O—(CH

2

CH

2

CH

2

)—O

NO

2

Cl

Het2

5849

S—(CH

2

CH

2

)—S

NO

2

Cl

Het2

5850

S—(CH

2

CH

2

CH

2

)—S

NO

2

Cl

Het2

5851

—(CH

2

)

4

—

NO

2

Cl

Het2

5852

—(CH

2

)

5

—

NO

2

Cl

Het2

5853

H

H

CN

Cl

Het2

5854

CH

3

CH

3

CN

Cl

Het2

5855

CH

2

CH

3

CH

2

CH

3

CN

Cl

Het2

5856

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Cl

Het2

5857

OCH

3

OCH

3

CN

Cl

Het2

5858

OCH

2

CH

3

OCH

2

CH

3

CN

Cl

Het2

5859

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Cl

Het2

5860

SCH

3

SCH

3

CN

Cl

Het2

5861

SCH

2

CH

3

SCH

2

CH

3

CN

Cl

Het2

5862

N(CH

3

)

2

N(CH

3

)

2

CN

Cl

Het2

5863

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Cl

Het2

5864

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Cl

Het2

5865

O—(CH

2

CH

2

)—O

CN

Cl

Het2

5866

O—(CH

2

CH

2

CH

2

)—O

CN

Cl

Het2

5867

S—(CH

2

CH

2

)—S

CN

Cl

Het2

5868

S—(CH

2

CH

2

CH

2

)—S

CN

Cl

Het2

5869

—(CH

2

)

4

—

CN

Cl

Het2

5870

—(CH

2

)

5

—

CN

Cl

Het2

5871

H

H

F

Cl

Het2

5872

CH

3

CH

3

F

Cl

Het2

5873

CH

2

CH

3

CH

2

CH

3

F

Cl

Het2

5874

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Cl

Het2

5875

OCH

3

OCH

3

F

Cl

Het2

5876

OCH

2

CH

3

OCH

2

CH

3

F

Cl

Het2

5877

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Cl

Het2

5878

SCH

3

SCH

3

F

Cl

Het2

5879

SCH

2

CH

3

SCH

2

CH

3

F

Cl

Het2

5880

N(CH

3

)

2

N(CH

3

)

2

F

Cl

Het2

5881

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Cl

Het2

5882

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Cl

Het2

5883

O—(CH

2

CH

2

)—O

F

Cl

Het2

5884

O—(CH

2

CH

2

CH

2

)—O

F

Cl

Het2

5885

S—(CH

2

CH

2

)—S

F

Cl

Het2

5886

S—(CH

2

CH

2

CH

2

)—S

F

Cl

Het2

5887

—(CH

2

)

4

—

F

Cl

Het2

5888

—(CH

2

)

5

—

F

Cl

Het2

5889

H

H

Cl

Cl

Het2

5890

CH

3

CH

3

Cl

Cl

Het2

5891

CH

2

CH

3

CH

2

CH

3

Cl

Cl

Het2

5892

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Cl

Het2

5893

OCH

3

OCH

3

Cl

Cl

Het2

5894

OCH

2

CH

3

OCH

2

CH

3

Cl

Cl

Het2

5895

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Cl

Het2

5896

SCH

3

SCH

3

Cl

Cl

Het2

5897

SCH

2

CH

3

SCH

2

CH

3

Cl

Cl

Het2

5898

N(CH

3

)

2

N(CH

3

)

2

Cl

Cl

Het2

5899

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Cl

Het2

5900

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Cl

Het2

5901

O—(CH

2

CH

2

)—O

Cl

Cl

Het2

5902

O—(CH

2

CH

2

CH

2

)—O

Cl

Cl

Het2

5903

S—(CH

2

CH

2

)—S

Cl

Cl

Het2

5904

S—(CH

2

CH

2

CH

2

)—S

Cl

Cl

Het2

5905

—(CH

2

)

4

—

Cl

Cl

Het2

5906

—(CH

2

)

5

—

Cl

Cl

Het2

5907

H

H

Br

Cl

Het2

5908

CH

3

CH

3

Br

Cl

Het2

5909

CH

2

CH

3

CH

2

CH

3

Br

Cl

Het2

5910

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Cl

Het2

5911

OCH

3

OCH

3

Br

Cl

Het2

5912

OCH

2

CH

3

OCH

2

CH

3

Br

Cl

Het2

5913

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Cl

Het2

5914

SCH

3

SCH

3

Br

Cl

Het2

5915

SCH

2

CH

3

SCH

2

CH

3

Br

Cl

Het2

5916

N(CH

3

)

2

N(CH

3

)

2

Br

Cl

Het2

5917

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Cl

Het2

5918

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Cl

Het2

5919

O—(CH

2

CH

2

)—O

Br

Cl

Het2

5920

O—(CH

2

CH

2

CH

2

)—O

Br

Cl

Het2

5921

S—(CH

2

CH

2

)—S

Br

Cl

Het2

5922

S—(CH

2

CH

2

CH

2

)—S

Br

Cl

Het2

5923

—(CH

2

)

4

—

Br

Cl

Het2

5924

—(CH

2

)

5

—

Br

Cl

Het2

5925

H

H

CH

3

Cl

Het2

5926

CH

3

CH

3

CH

3

Cl

Het2

5927

CH

2

CH

3

CH

2

CH

3

CH

3

Cl

Het2

5928

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Cl

Het2

5929

OCH

3

OCH

3

CH

3

Cl

Het2

5930

OCH

2

CH

3

OCH

2

CH

3

CH

3

Cl

Het2

5931

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Cl

Het2

5932

SCH

3

SCH

3

CH

3

Cl

Het2

5933

SCH

2

CH

3

SCH

2

CH

3

CH

3

Cl

Het2

5934

N(CH

3

)

2

N(CH

3

)

2

CH

3

Cl

Het2

5935

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Cl

Het2

5936

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Cl

Het2

5937

O—(CH

2

CH

2

)—O

CH

3

Cl

Het2

5938

O—(CH

2

CH

2

CH

2

)—O

CH

3

Cl

Het2

5939

S—(CH

2

CH

2

)—S

CH

3

Cl

Het2

5940

S—(CH

2

CH

2

CH

2

)—S

CH

3

Cl

Het2

5941

—(CH

2

)

4

—

CH

3

Cl

Het2

5942

—(CH

2

)

5

—

CH

3

Cl

Het2

5943

H

H

CH

2

CH

3

Cl

Het2

5944

CH

3

CH

3

CH

2

CH

3

Cl

Het2

5945

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Cl

Het2

5946

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Cl

Het2

5947

OCH

3

OCH

3

CH

2

CH

3

Cl

Het2

5948

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Cl

Het2

5949

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Cl

Het2

5950

SCH

3

SCH

3

CH

2

CH

3

Cl

Het2

5951

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Cl

Het2

5952

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Cl

Het2

5953

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Cl

Het2

5954

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Cl

Het2

5955

O—(CH

2

CH

2

)—O

CH

2

CH

3

Cl

Het2

5956

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Cl

Het2

5957

S—(CH

2

CH

2

)—S

CH

2

CH

3

Cl

Het2

5958

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Cl

Het2

5959

—(CH

2

)

4

—

CH

2

CH

3

Cl

Het2

5960

—(CH

2

)

5

—

CH

2

CH

3

Cl

Het2

5961

H

H

CF

3

Cl

Het2

5962

CH

3

CH

3

CF

3

Cl

Het2

5963

CH

2

CH

3

CH

2

CH

3

CF

3

Cl

Het2

5964

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Cl

Het2

5965

OCH

3

OCH

3

CF

3

Cl

Het2

5966

OCH

2

CH

3

OCH

2

CH

3

CF

3

Cl

Het2

5967

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Cl

Het2

5968

SCH

3

SCH

3

CF

3

Cl

Het2

5969

SCH

2

CH

3

SCH

2

CH

3

CF

3

Cl

Het2

5970

N(CH

3

)

2

N(CH

3

)

2

CF

3

Cl

Het2

5971

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Cl

Het2

5972

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Cl

Het2

5973

O—(CH

2

CH

2

)—O

CF

3

Cl

Het2

5974

O—(CH

2

CH

2

CH

2

)—O

CF

3

Cl

Het2

5975

S—(CH

2

CH

2

)—S

CF

3

Cl

Het2

5976

S—(CH

2

CH

2

CH

2

)—S

CF

3

Cl

Het2

5977

—(CH

2

)

4

—

CF

3

Cl

Het2

5978

—(CH

2

)

5

—

CF

3

Cl

Het2

5979

H

H

OCH

3

Cl

Het2

5980

CH

3

CH

3

OCH

3

Cl

Het2

5981

CH

2

CH

3

CH

2

CH

3

OCH

3

Cl

Het2

5982

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Cl

Het2

5983

OCH

3

OCH

3

OCH

3

Cl

Het2

5984

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Cl

Het2

5985

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Cl

Het2

5986

SCH

3

SCH

3

OCH

3

Cl

Het2

5987

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Cl

Het2

5988

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Cl

Het2

5989

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Cl

Het2

5990

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Cl

Het2

5991

O—(CH

2

CH

2

)—O

OCH

3

Cl

Het2

5992

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Cl

Het2

5993

S—(CH

2

CH

2

)—S

OCH

3

Cl

Het2

5994

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Cl

Het2

5995

—(CH

2

)

4

—

OCH

3

Cl

Het2

5996

—(CH

2

)

5

—

OCH

3

Cl

Het2

5997

H

H

OCH

2

CH

3

Cl

Het2

5998

CH

3

CH

3

OCH

2

CH

3

Cl

Het2

5999

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Cl

Het2

6000

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Cl

Het2

6001

OCH

3

OCH

3

OCH

2

CH

3

Cl

Het2

6002

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Cl

Het2

6003

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Cl

Het2

6004

SCH

3

SCH

3

OCH

2

CH

3

Cl

Het2

6005

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Cl

Het2

6006

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Cl

Het2

6007

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Cl

Het2

6008

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Cl

Het2

6009

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Cl

Het2

6010

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Cl

Het2

6011

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Cl

Het2

6012

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Cl

Het2

6013

—(CH

2

)

4

—

OCH

2

CH

3

Cl

Het2

6014

—(CH

2

)

5

—

OCH

2

CH

3

Cl

Het2

6015

H

H

SCH

3

Cl

Het2

6016

CH

3

CH

3

SCH

3

Cl

Het2

6017

CH

2

CH

3

CH

2

CH

3

SCH

3

Cl

Het2

6018

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Cl

Het2

6019

OCH

3

OCH

3

SCH

3

Cl

Het2

6020

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Cl

Het2

6021

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Cl

Het2

6022

SCH

3

SCH

3

SCH

3

Cl

Het2

6023

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Cl

Het2

6024

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Cl

Het2

6025

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Cl

Het2

6026

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Cl

Het2

6027

O—(CH

2

CH

2

)—O

SCH

3

Cl

Het2

6028

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Cl

Het2

6029

S—(CH

2

CH

2

)—S

SCH

3

Cl

Het2

6030

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Cl

Het2

6031

—(CH

2

)

4

—

SCH

3

Cl

Het2

6032

—(CH

2

)

5

—

SCH

3

Cl

Het2

6033

H

H

SO

2

CH

3

Cl

Het2

6034

CH

3

CH

3

SO

2

CH

3

Cl

Het2

6035

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Cl

Het2

6036

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Cl

Het2

6037

OCH

3

OCH

3

SO

2

CH

3

Cl

Het2

6038

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Cl

Het2

6039

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Cl

Het2

6040

SCH

3

SCH

3

SO

2

CH

3

Cl

Het2

6041

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Cl

Het2

6042

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Cl

Het2

6043

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Cl

Het2

6044

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Cl

Het2

6045

O—(CH

2

CH

2

)—O

SO

2

CH

3

Cl

Het2

6046

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Cl

Het2

6047

S—(CH

2

CH

2

)—S

SO

2

CH

3

Cl

Het2

6048

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Cl

Het2

6049

—(CH

2

)

4

—

SO

2

CH

3

Cl

Het2

6050

—(CH

2

)

5

—

SO

2

CH

3

Cl

Het2

6051

H

H

PO(OCH

3

)

2

Cl

Het2

6052

CH

3

CH

3

PO(OCH

3

)

2

Cl

Het2

6053

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Cl

Het2

6054

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

Het2

6055

OCH

3

OCH

3

PO(OCH

3

)

2

Cl

Het2

6056

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Cl

Het2

6057

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

Het2

6058

SCH

3

SCH

3

PO(OCH

3

)

2

Cl

Het2

6059

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Cl

Het2

6060

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Cl

Het2

6061

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Cl

Het2

6062

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Cl

Het2

6063

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

Het2

6064

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

Het2

6065

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

Het2

6066

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

Het2

6067

—(CH

2

)

4

—

PO(OCH

3

)

2

Cl

Het2

6068

—(CH

2

)

5

—

PO(OCH

3

)

2

Cl

Het2

6069

H

H

PO(OCH

2

CH

3

)

2

Cl

Het2

6070

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het2

6071

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het2

6072

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het2

6073

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Cl

Het2

6074

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het2

6075

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het2

6076

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Cl

Het2

6077

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het2

6078

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

Het2

6079

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

Het2

6080

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Cl

Het2

6081

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

Het2

6082

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

Het2

6083

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

Het2

6084

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

Het2

6085

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Cl

Het2

6086

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Cl

Het2

6087

H

H

PO(CH

3

)

2

Cl

Het2

6088

CH

3

CH

3

PO(CH

3

)

2

Cl

Het2

6089

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Cl

Het2

6090

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

Het2

6091

OCH

3

OCH

3

PO(CH

3

)

2

Cl

Het2

6092

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Cl

Het2

6093

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

Het2

6094

SCH

3

SCH

3

PO(CH

3

)

2

Cl

Het2

6095

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Cl

Het2

6096

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Cl

Het2

6097

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Cl

Het2

6098

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Cl

Het2

6099

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

Het2

6100

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

Het2

6101

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

Het2

6102

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

Het2

6103

—(CH

2

)

4

—

PO(CH

3

)

2

Cl

Het2

6104

—(CH

2

)

5

—

PO(CH

3

)

2

Cl

Het2

6105

H

H

PC(CH

2

CH

3

)

2

Cl

Het2

6106

CH

3

CH

3

PC(CH

2

CH

3

)

2

Cl

Het2

6107

CH

2

CH

3

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het2

6108

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het2

6109

OCH

3

OCH

3

PC(CH

2

CH

3

)

2

Cl

Het2

6110

OCH

2

CH

3

OCH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het2

6111

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het2

6112

SCH

3

SCH

3

PC(CH

2

CH

3

)

2

Cl

Het2

6113

SCH

2

CH

3

SCH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het2

6114

N(CH

3

)

2

N(CH

3

)

2

PC(CH

2

CH

3

)

2

Cl

Het2

6115

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PC(CH

2

CH

3

)

2

Cl

Het2

6116

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PC(CH

2

CH

3

)

2

Cl

Het2

6117

O—(CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Cl

Het2

6118

O—(CH

2

CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Cl

Het2

6119

S—(CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Cl

Het2

6120

S—(CH

2

CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Cl

Het2

6121

—(CH

2

)

4

—

PC(CH

2

CH

3

)

2

Cl

Het2

6122

—(CH

2

)

5

—

PC(CH

2

CH

3

)

2

Cl

Het2

6123

H

H

H

Cl

Het3

6124

CH

3

CH

3

H

Cl

Het3

6125

CH

2

CH

3

CH

2

CH

3

H

Cl

Het3

6126

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Cl

Het3

6127

OCH

3

OCH

3

H

Cl

Het3

6128

OCH

2

CH

3

OCH

2

CH

3

H

Cl

Het3

6129

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Cl

Het3

6130

SCH

3

SCH

3

H

Cl

Het3

6131

SCH

2

CH

3

SCH

2

CH

3

H

Cl

Het3

6132

N(CH

3

)

2

N(CH

3

)

2

H

Cl

Het3

6133

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Cl

Het3

6134

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Cl

Het3

6135

O—(CH

2

CH

2

)—O

H

Cl

Het3

6136

O—(CH

2

CH

2

CH

2

)—O

H

Cl

Het3

6137

S—(CH

2

CH

2

)—S

H

Cl

Het3

6138

S—(CH

2

CH

2

CH

2

)—S

H

Cl

Het3

6139

—(CH

2

)

4

—

H

Cl

Het3

6140

—(CH

2

)

5

—

H

Cl

Het3

6141

H

H

NO

2

Cl

Het3

6142

CH

3

CH

3

NO

2

Cl

Het3

6143

CH

2

CH

3

CH

2

CH

3

NO

2

Cl

Het3

6144

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Cl

Het3

6145

OCH

3

OCH

3

NO

2

Cl

Het3

6146

OCH

2

CH

3

OCH

2

CH

3

NO

2

Cl

Het3

6147

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Cl

Het3

6148

SCH

3

SCH

3

NO

2

Cl

Het3

6149

SCH

2

CH

3

SCH

2

CH

3

NO

2

Cl

Het3

6150

N(CH

3

)

2

N(CH

3

)

2

NO

2

Cl

Het3

6151

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Cl

Het3

6152

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Cl

Het3

6153

O—(CH

2

CH

2

)—O

NO

2

Cl

Het3

6154

O—(CH

2

CH

2

CH

2

)—O

NO

2

Cl

Het3

6155

S—(CH

2

CH

2

)—S

NO

2

Cl

Het3

6156

S—(CH

2

CH

2

CH

2

)—S

NO

2

Cl

Het3

6157

—(CH

2

)

4

—

NO

2

Cl

Het3

6158

—(CH

2

)

5

—

NO

2

Cl

Het3

6159

H

H

CN

Cl

Het3

6160

CH

3

CH

3

CN

Cl

Het3

6161

CH

2

CH

3

CH

2

CH

3

CN

Cl

Het3

6162

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Cl

Het3

6163

OCH

3

OCH

3

CN

Cl

Het3

6164

OCH

2

CH

3

OCH

2

CH

3

CN

Cl

Het3

6165

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Cl

Het3

6166

SCH

3

SCH

3

CN

Cl

Het3

6167

SCH

2

CH

3

SCH

2

CH

3

CN

Cl

Het3

6168

N(CH

3

)

2

N(CH

3

)

2

CN

Cl

Het3

6169

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Cl

Het3

6170

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Cl

Het3

6171

O—(CH

2

CH

2

)—O

CN

Cl

Het3

6172

O—(CH

2

CH

2

CH

2

)—O

CN

Cl

Het3

6173

S—(CH

2

CH

2

)—S

CN

Cl

Het3

6174

S—(CH

2

CH

2

CH

2

)—S

CN

Cl

Het3

6175

—(CH

2

)

4

—

CN

Cl

Het3

6176

—(CH

2

)

5

—

CN

Cl

Het3

6177

H

H

F

Cl

Het3

6178

CH

3

CH

3

F

Cl

Het3

6179

CH

2

CH

3

CH

2

CH

3

F

Cl

Het3

6180

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Cl

Het3

6181

OCH

3

OCH

3

F

Cl

Het3

6182

OCH

2

CH

3

OCH

2

CH

3

F

Cl

Het3

6183

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Cl

Het3

6184

SCH

3

SCH

3

F

Cl

Het3

6185

SCH

2

CH

3

SCH

2

CH

3

F

Cl

Het3

6186

N(CH

3

)

2

N(CH

3

)

2

F

Cl

Het3

6187

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Cl

Het3

6188

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Cl

Het3

6189

O—(CH

2

CH

2

)—O

F

Cl

Het3

6190

O—(CH

2

CH

2

CH

2

)—O

F

Cl

Het3

6191

S—(CH

2

CH

2

)—S

F

Cl

Het3

6192

S—(CH

2

CH

2

CH

2

)—S

F

Cl

Het3

6193

—(CH

2

)

4

—

F

Cl

Het3

6194

—(CH

2

)

5

—

F

Cl

Het3

6195

H

H

Cl

Cl

Het3

6196

CH

3

CH

3

Cl

Cl

Het3

6197

CH

2

CH

3

CH

2

CH

3

Cl

Cl

Het3

6198

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Cl

Het3

6199

OCH

3

OCH

3

Cl

Cl

Het3

6200

OCH

2

CH

3

OCH

2

CH

3

Cl

Cl

Het3

6201

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Cl

Het3

6202

SCH

3

SCH

3

Cl

Cl

Het3

6203

SCH

2

CH

3

SCH

2

CH

3

Cl

Cl

Het3

6204

N(CH

3

)

2

N(CH

3

)

2

Cl

Cl

Het3

6205

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Cl

Het3

6206

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Cl

Het3

6207

O—(CH

2

CH

2

)—O

Cl

Cl

Het3

6208

O—(CH

2

CH

2

CH

2

)—O

Cl

Cl

Het3

6209

S—(CH

2

CH

2

)—S

Cl

Cl

Het3

6210

S—(CH

2

CH

2

CH

2

)—S

Cl

Cl

Het3

6211

—(CH

2

)

4

—

Cl

Cl

Het3

6212

—(CH

2

)

5

—

Cl

Cl

Het3

6213

H

H

Br

Cl

Het3

6214

CH

3

CH

3

Br

Cl

Het3

6215

CH

2

CH

3

CH

2

CH

3

Br

Cl

Het3

6216

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Cl

Het3

6217

OCH

3

OCH

3

Br

Cl

Het3

6218

OCH

2

CH

3

OCH

2

CH

3

Br

Cl

Het3

6219

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Cl

Het3

6220

SCH

3

SCH

3

Br

Cl

Het3

6221

SCH

2

CH

3

SCH

2

CH

3

Br

Cl

Het3

6222

N(CH

3

)

2

N(CH

3

)

2

Br

Cl

Het3

6223

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Cl

Het3

6224

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Cl

Het3

6225

O—(CH

2

CH

2

)—O

Br

Cl

Het3

6226

O—(CH

2

CH

2

CH

2

)—O

Br

Cl

Het3

6227

S—(CH

2

CH

2

)—S

Br

Cl

Het3

6228

S—(CH

2

CH

2

CH

2

)—S

Br

Cl

Het3

6229

—(CH

2

)

4

—

Br

Cl

Het3

6230

—(CH

2

)

5

—

Br

Cl

Het3

6231

H

H

CH

3

Cl

Het3

6232

CH

3

CH

3

CH

3

Cl

Het3

6233

CH

2

CH

3

CH

2

CH

3

CH

3

Cl

Het3

6234

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Cl

Het3

6235

OCH

3

OCH

3

CH

3

Cl

Het3

6236

OCH

2

CH

3

OCH

2

CH

3

CH

3

Cl

Het3

6237

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Cl

Het3

6238

SCH

3

SCH

3

CH

3

Cl

Het3

6239

SCH

2

CH

3

SCH

2

CH

3

CH

3

Cl

Het3

6240

N(CH

3

)

2

N(CH

3

)

2

CH

3

Cl

Het3

6241

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Cl

Het3

6242

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Cl

Het3

6243

O—(CH

2

CH

2

)—O

CH

3

Cl

Het3

6244

O—(CH

2

CH

2

CH

2

)—O

CH

3

Cl

Het3

6245

S—(CH

2

CH

2

)—S

CH

3

Cl

Het3

6246

S—(CH

2

CH

2

CH

2

)—S

CH

3

Cl

Het3

6247

—(CH

2

)

4

—

CH

3

Cl

Het3

6248

—(CH

2

)

5

—

CH

3

Cl

Het3

6249

H

H

CH

2

CH

3

Cl

Het3

6250

CH

3

CH

3

CH

2

CH

3

Cl

Het3

6251

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Cl

Het3

6252

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Cl

Het3

6253

OCH

3

OCH

3

CH

2

CH

3

Cl

Het3

6254

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Cl

Het3

6255

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Cl

Het3

6256

SCH

3

SCH

3

CH

2

CH

3

Cl

Het3

6257

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Cl

Het3

6258

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Cl

Het3

6259

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Cl

Het3

6260

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Cl

Het3

6261

O—(CH

2

CH

2

)—O

CH

2

CH

3

Cl

Het3

6262

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Cl

Het3

6263

S—(CH

2

CH

2

)—S

CH

2

CH

3

Cl

Het3

6264

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Cl

Het3

6265

—(CH

2

)

4

—

CH

2

CH

3

Cl

Het3

6266

—(CH

2

)

5

—

CH

2

CH

3

Cl

Het3

6267

H

H

CF

3

Cl

Het3

6268

CH

3

CH

3

CF

3

Cl

Het3

6269

CH

2

CH

3

CH

2

CH

3

CF

3

Cl

Het3

6270

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Cl

Het3

6271

OCH

3

OCH

3

CF

3

Cl

Het3

6272

OCH

2

CH

3

OCH

2

CH

3

CF

3

Cl

Het3

6273

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Cl

Het3

6274

SCH

3

SCH

3

CF

3

Cl

Het3

6275

SCH

2

CH

3

SCH

2

CH

3

CF

3

Cl

Het3

6276

N(CH

3

)

2

N(CH

3

)

2

CF

3

Cl

Het3

6277

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Cl

Het3

6278

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Cl

Het3

6279

O—(CH

2

CH

2

)—O

CF

3

Cl

Het3

6280

O—(CH

2

CH

2

CH

2

)—O

CF

3

Cl

Het3

6281

S—(CH

2

CH

2

)—S

CF

3

Cl

Het3

6282

S—(CH

2

CH

2

CH

2

)—S

CF

3

Cl

Het3

6283

—(CH

2

)

4

—

CF

3

Cl

Het3

6284

—(CH

2

)

5

—

CF

3

Cl

Het3

6285

H

H

OCH

3

Cl

Het3

6286

CH

3

CH

3

OCH

3

Cl

Het3

6287

CH

2

CH

3

CH

2

CH

3

OCH

3

Cl

Het3

6288

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Cl

Het3

6289

OCH

3

OCH

3

OCH

3

Cl

Het3

6290

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Cl

Het3

6291

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Cl

Het3

6292

SCH

3

SCH

3

OCH

3

Cl

Het3

6293

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Cl

Het3

6294

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Cl

Het3

6295

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Cl

Het3

6296

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Cl

Het3

6297

O—(CH

2

CH

2

)—O

OCH

3

Cl

Het3

6298

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Cl

Het3

6299

S—(CH

2

CH

2

)—S

OCH

3

Cl

Het3

6300

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Cl

Het3

6301

—(CH

2

)

4

—

OCH

3

Cl

Het3

6302

—(CH

2

)

5

—

OCH

3

Cl

Het3

6303

H

H

OCH

2

CH

3

Cl

Het3

6304

CH

3

CH

3

OCH

2

CH

3

Cl

Het3

6305

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Cl

Het3

6306

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Cl

Het3

6307

OCH

3

OCH

3

OCH

2

CH

3

Cl

Het3

6308

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Cl

Het3

6309

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Cl

Het3

6310

SCH

3

SCH

3

OCH

2

CH

3

Cl

Het3

6311

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Cl

Het3

6312

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Cl

Het3

6313

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Cl

Het3

6314

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Cl

Het3

6315

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Cl

Het3

6316

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Cl

Het3

6317

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Cl

Het3

6318

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Cl

Het3

6319

—(CH

2

)

4

—

OCH

2

CH

3

Cl

Het3

6320

—(CH

2

)

5

—

OCH

2

CH

3

Cl

Het3

6331

H

H

SCH

3

Cl

Het3

6332

CH

3

CH

3

SCH

3

Cl

Het3

6333

CH

2

CH

3

CH

2

CH

3

SCH

3

Cl

Het3

6334

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Cl

Het3

6335

OCH

3

OCH

3

SCH

3

Cl

Het3

6336

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Cl

Het3

6337

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Cl

Het3

6338

SCH

3

SCH

3

SCH

3

Cl

Het3

6339

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Cl

Het3

6340

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Cl

Het3

6341

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Cl

Het3

6342

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Cl

Het3

6343

O—(CH

2

CH

2

)—O

SCH

3

Cl

Het3

6344

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Cl

Het3

6345

S—(CH

2

CH

2

)—S

SCH

3

Cl

Het3

6346

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Cl

Het3

6347

—(CH

2

)

4

—

SCH

3

Cl

Het3

6348

—(CH

2

)

5

—

SCH

3

Cl

Het3

6349

H

H

SO

2

CH

3

Cl

Het3

6350

CH

3

CH

3

SO

2

CH

3

Cl

Het3

6351

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Cl

Het3

6352

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Cl

Het3

6353

OCH

3

OCH

3

SO

2

CH

3

Cl

Het3

6354

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Cl

Het3

6355

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Cl

Het3

6356

SCH

3

SCH

3

SO

2

CH

3

Cl

Het3

6357

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Cl

Het3

6358

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Cl

Het3

6359

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Cl

Het3

6360

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Cl

Het3

6361

O—(CH

2

CH

2

)—O

SO

2

CH

3

Cl

Het3

6362

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Cl

Het3

6363

S—(CH

2

CH

2

)—S

SO

2

CH

3

Cl

Het3

6364

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Cl

Het3

6365

—(CH

2

)

4

—

SO

2

CH

3

Cl

Het3

6366

—(CH

2

)

5

—

SO

2

CH

3

Cl

Het3

6367

H

H

PO(OCH

3

)

2

Cl

Het3

6368

CH

3

CH

3

PO(OCH

3

)

2

Cl

Het3

6369

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Cl

Het3

6370

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

Het3

6371

OCH

3

OCH

3

PO(OCH

3

)

2

Cl

Het3

6372

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Cl

Het3

6373

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Cl

Het3

6374

SCH

3

SCH

3

PO(OCH

3

)

2

Cl

Het3

6375

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Cl

Het3

6376

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Cl

Het3

6377

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Cl

Het3

6378

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Cl

Het3

6379

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

Het3

6380

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Cl

Het3

6381

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

Het3

6382

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Cl

Het3

6383

—(CH

2

)

4

—

PO(OCH

3

)

2

Cl

Het3

6384

—(CH

2

)

5

—

PO(OCH

3

)

2

Cl

Het3

6385

H

H

PO(OCH

2

CH

3

)

2

Cl

Het3

6386

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het3

6387

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het3

6388

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het3

6389

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Cl

Het3

6390

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het3

6391

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het3

6392

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Cl

Het3

6393

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Cl

Het3

6394

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

Het3

6395

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Cl

Het3

6396

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Cl

Het3

6397

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

Het3

6398

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Cl

Het3

6399

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

Het3

6400

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Cl

Het3

6401

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Cl

Het3

6402

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Cl

Het3

6403

H

H

PO(CH

3

)

2

Cl

Het3

6404

CH

3

CH

3

PO(CH

3

)

2

Cl

Het3

6405

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Cl

Het3

6406

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

Het3

6407

OCH

3

OCH

3

PO(CH

3

)

2

Cl

Het3

6408

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Cl

Het3

6409

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Cl

Het3

6410

SCH

3

SCH

3

PO(CH

3

)

2

Cl

Het3

6411

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Cl

Het3

6412

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Cl

Het3

6413

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Cl

Het3

6414

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Cl

Het3

6415

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

Het3

6416

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Cl

Het3

6417

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

Het3

6418

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Cl

Het3

6419

—(CH

2

)

4

—

PO(CH

3

)

2

Cl

Het3

6420

—(CH

2

)

5

—

PO(CH

3

)

2

Cl

Het3

6421

H

H

PC(CH

2

CH

3

)

2

Cl

Het3

6422

CH

3

CH

3

PC(CH

2

CH

3

)

2

Cl

Het3

6423

CH

2

CH

3

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het3

6424

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het3

6425

OCH

3

OCH

3

PC(CH

2

CH

3

)

2

Cl

Het3

6426

OCH

2

CH

3

OCH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het3

6427

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het3

6428

SCH

3

SCH

3

PC(CH

2

CH

3

)

2

Cl

Het3

6429

SCH

2

CH

3

SCH

2

CH

3

PC(CH

2

CH

3

)

2

Cl

Het3

6430

N(CH

3

)

2

N(CH

3

)

2

PC(CH

2

CH

3

)

2

Cl

Het3

6431

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PC(CH

2

CH

3

)

2

Cl

Het3

6432

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PC(CH

2

CH

3

)

2

Cl

Het3

6433

O—(CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Cl

Het3

6434

O—(CH

2

CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Cl

Het3

6435

S—(CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Cl

Het3

6436

S—(CH

2

CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Cl

Het3

6437

—(CH

2

)

4

—

PC(CH

2

CH

3

)

2

Cl

Het3

6438

—(CH

2

)

5

—

PC(CH

2

CH

3

)

2

Cl

Het3

6439

H

H

H

Br

OH

6440

CH

3

CH

3

H

Br

OH

6441

CH

2

CH

3

CH

2

CH

3

H

Br

OH

6442

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Br

OH

6443

OCH

3

OCH

3

H

Br

OH

6444

OCH

2

CH

3

OCH

2

CH

3

H

Br

OH

6445

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Br

OH

6446

SCH

3

SCH

3

H

Br

OH

6447

SCH

2

CH

3

SCH

2

CH

3

H

Br

OH

6448

N(CH

3

)

2

N(CH

3

)

2

H

Br

OH

6449

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Br

OH

6450

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Br

OH

6451

O—(CH

2

CH

2

)—O

H

Br

OH

6452

O—(CH

2

CH

2

CH

2

)—O

H

Br

OH

6453

S—(CH

2

CH

2

)—S

H

Br

OH

6454

S—(CH

2

CH

2

CH

2

)—S

H

Br

OH

6455

—(CH

2

)

4

—

H

Br

OH

6456

—(CH

2

)

5

—

H

Br

OH

6457

H

H

NO

2

Br

OH

6458

CH

3

CH

3

NO

2

Br

OH

6459

CH

2

CH

3

CH

2

CH

3

NO

2

Br

OH

6460

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Br

OH

6461

OCH

3

OCH

3

NO

2

Br

OH

6462

OCH

2

CH

3

OCH

2

CH

3

NO

2

Br

OH

6463

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Br

OH

6464

SCH

3

SCH

3

NO

2

Br

OH

6465

SCH

2

CH

3

SCH

2

CH

3

NO

2

Br

OH

6466

N(CH

3

)

2

N(CH

3

)

2

NO

2

Br

OH

6467

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Br

OH

6468

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Br

OH

6469

O—(CH

2

CH

2

)—O

NO

2

Br

OH

6470

O—(CH

2

CH

2

CH

2

)—O

NO

2

Br

OH

6471

S—(CH

2

CH

2

)—S

NO

2

Br

OH

6472

S—(CH

2

CH

2

CH

2

)—S

NO

2

Br

OH

6473

—(CH

2

)

4

—

NO

2

Br

OH

6474

—(CH

2

)

5

—

NO

2

Br

OH

6475

H

H

CN

Br

OH

6476

CH

3

CH

3

CN

Br

OH

6477

CH

2

CH

3

CH

2

CH

3

CN

Br

OH

6478

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Br

OH

6479

OCH

3

OCH

3

CN

Br

OH

6480

OCH

2

CH

3

OCH

2

CH

3

CN

Br

OH

6481

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Br

OH

6482

SCH

3

SCH

3

CN

Br

OH

6483

SCH

2

CH

3

SCH

2

CH

3

CN

Br

OH

6484

N(CH

3

)

2

N(CH

3

)

2

CN

Br

OH

6485

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Br

OH

6486

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Br

OH

6487

O—(CH

2

CH

2

)—O

CN

Br

OH

6488

O—(CH

2

CH

2

CH

2

)—O

CN

Br

OH

6489

S—(CH

2

CH

2

)—S

CN

Br

OH

6490

S—(CH

2

CH

2

CH

2

)—S

CN

Br

OH

6491

—(CH

2

)

4

—

CN

Br

OH

6492

—(CH

2

)

5

—

CN

Br

OH

6493

H

H

F

Br

OH

6494

CH

3

CH

3

F

Br

OH

6495

CH

2

CH

3

CH

2

CH

3

F

Br

OH

6496

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Br

OH

6497

OCH

3

OCH

3

F

Br

OH

6498

OCH

2

CH

3

OCH

2

CH

3

F

Br

OH

6499

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Br

OH

6500

SCH

3

SCH

3

F

Br

OH

6501

SCH

2

CH

3

SCH

2

CH

3

F

Br

OH

6502

N(CH

3

)

2

N(CH

3

)

2

F

Br

OH

6503

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Br

OH

6504

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Br

OH

6505

O—(CH

2

CH

2

)—O

F

Br

OH

6506

O—(CH

2

CH

2

CH

2

)—O

F

Br

OH

6507

S—(CH

2

CH

2

)—S

F

Br

OH

6508

S—(CH

2

CH

2

CH

2

)—S

F

Br

OH

6509

—(CH

2

)

4

—

F

Br

OH

6510

—(CH

2

)

5

—

F

Br

OH

6511

H

H

Cl

Br

OH

6512

CH

3

CH

3

Cl

Br

OH

6513

CH

2

CH

3

CH

2

CH

3

Cl

Br

OH

6514

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Br

OH

6515

OCH

3

OCH

3

Cl

Br

OH

6516

OCH

2

CH

3

OCH

2

CH

3

Cl

Br

OH

6517

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Br

OH

6518

SCH

3

SCH

3

Cl

Br

OH

6519

SCH

2

CH

3

SCH

2

CH

3

Cl

Br

OH

6520

N(CH

3

)

2

N(CH

3

)

2

Cl

Br

OH

6521

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Br

OH

6522

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Br

OH

6523

O—(CH

2

CH

2

)—O

Cl

Br

OH

6524

O—(CH

2

CH

2

CH

2

)—O

Cl

Br

OH

6525

S—(CH

2

CH

2

)—S

Cl

Br

OH

6526

S—(CH

2

CH

2

CH

2

)—S

Cl

Br

OH

6527

—(CH

2

)

4

—

Cl

Br

OH

6528

—(CH

2

)

5

—

Cl

Br

OH

6529

H

H

Br

Br

OH

6530

CH

3

CH

3

Br

Br

OH

6531

CH

2

CH

3

CH

2

CH

3

Br

Br

OH

6532

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Br

OH

6533

OCH

3

OCH

3

Br

Br

OH

6534

OCH

2

CH

3

OCH

2

CH

3

Br

Br

OH

6535

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Br

OH

6536

SCH

3

SCH

3

Br

Br

OH

6537

SCH

2

CH

3

SCH

2

CH

3

Br

Br

OH

6538

N(CH

3

)

2

N(CH

3

)

2

Br

Br

OH

6539

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Br

OH

6540

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Br

OH

6541

O—(CH

2

CH

2

)—O

Br

Br

OH

6542

O—(CH

2

CH

2

CH

2

)—O

Br

Br

OH

6543

S—(CH

2

CH

2

)—S

Br

Br

OH

6544

S—(CH

2

CH

2

CH

2

)—S

Br

Br

OH

6545

—(CH

2

)

4

—

Br

Br

OH

6546

—(CH

2

)

5

—

Br

Br

OH

6547

H

H

CH

3

Br

OH

6548

CH

3

CH

3

CH

3

Br

OH

6549

CH

2

CH

3

CH

2

CH

3

CH

3

Br

OH

6550

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Br

OH

6551

OCH

3

OCH

3

CH

3

Br

OH

6552

OCH

2

CH

3

OCH

2

CH

3

CH

3

Br

OH

6553

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Br

OH

6554

SCH

3

SCH

3

CH

3

Br

OH

6555

SCH

2

CH

3

SCH

2

CH

3

CH

3

Br

OH

6556

N(CH

3

)

2

N(CH

3

)

2

CH

3

Br

OH

6557

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Br

OH

6558

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Br

OH

6559

O—(CH

2

CH

2

)—O

CH

3

Br

OH

6560

O—(CH

2

CH

2

CH

2

)—O

CH

3

Br

OH

6561

S—(CH

2

CH

2

)—S

CH

3

Br

OH

6562

S—(CH

2

CH

2

CH

2

)—S

CH

3

Br

OH

6563

—(CH

2

)

4

—

CH

3

Br

OH

6564

—(CH

2

)

5

—

CH

3

Br

OH

6565

H

H

CH

2

CH

3

Br

OH

6566

CH

3

CH

3

CH

2

CH

3

Br

OH

6567

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Br

OH

6568

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Br

OH

6569

OCH

3

OCH

3

CH

2

CH

3

Br

OH

6570

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Br

OH

6571

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Br

OH

6572

SCH

3

SCH

3

CH

2

CH

3

Br

OH

6573

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Br

OH

6574

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Br

OH

6575

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Br

OH

6576

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Br

OH

6577

O—(CH

2

CH

2

)—O

CH

2

CH

3

Br

OH

6578

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Br

OH

6579

S—(CH

2

CH

2

)—S

CH

2

CH

3

Br

OH

6580

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Br

OH

6581

—(CH

2

)

4

—

CH

2

CH

3

Br

OH

6582

—(CH

2

)

5

—

CH

2

CH

3

Br

OH

6583

H

H

CF

3

Br

OH

6584

CH

3

CH

3

CF

3

Br

OH

6585

CH

2

CH

3

CH

2

CH

3

CF

3

Br

OH

6586

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Br

OH

6587

OCH

3

OCH

3

CF

3

Br

OH

6588

OCH

2

CH

3

OCH

2

CH

3

CF

3

Br

OH

6589

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Br

OH

6590

SCH

3

SCH

3

CF

3

Br

OH

6591

SCH

2

CH

3

SCH

2

CH

3

CF

3

Br

OH

6592

N(CH

3

)

2

N(CH

3

)

2

CF

3

Br

OH

6593

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Br

OH

6594

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Br

OH

6595

O—(CH

2

CH

2

)—O

CF

3

Br

OH

6596

O—(CH

2

CH

2

CH

2

)—O

CF

3

Br

OH

6597

S—(CH

2

CH

2

)—S

CF

3

Br

OH

6598

S—(CH

2

CH

2

CH

2

)—S

CF

3

Br

OH

6599

—(CH

2

)

4

—

CF

3

Br

OH

6600

—(CH

2

)

5

—

CF

3

Br

OH

6601

H

H

OCH

3

Br

OH

6602

CH

3

CH

3

OCH

3

Br

OH

6603

CH

2

CH

3

CH

2

CH

3

OCH

3

Br

OH

6604

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Br

OH

6605

OCH

3

OCH

3

OCH

3

Br

OH

6606

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Br

OH

6607

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Br

OH

6608

SCH

3

SCH

3

OCH

3

Br

OH

6609

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Br

OH

6610

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Br

OH

6611

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Br

OH

6612

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Br

OH

6613

O—(CH

2

CH

2

)—O

OCH

3

Br

OH

6614

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Br

OH

6615

S—(CH

2

CH

2

)—S

OCH

3

Br

OH

6616

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Br

OH

6617

—(CH

2

)

4

—

OCH

3

Br

OH

6618

—(CH

2

)

5

—

OCH

3

Br

OH

6619

H

H

OCH

2

CH

3

Br

OH

6620

CH

3

CH

3

OCH

2

CH

3

Br

OH

6621

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Br

OH

6622

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Br

OH

6623

OCH

3

OCH

3

OCH

2

CH

3

Br

OH

6624

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Br

OH

6625

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Br

OH

6626

SCH

3

SCH

3

OCH

2

CH

3

Br

OH

6627

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Br

OH

6628

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Br

OH

6629

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Br

OH

6630

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Br

OH

6631

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Br

OH

6632

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Br

OH

6633

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Br

OH

6634

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Br

OH

6635

—(CH

2

)

4

—

OCH

2

CH

3

Br

OH

6636

—(CH

2

)

5

—

OCH

2

CH

3

Br

OH

6637

H

H

SCH

3

Br

OH

6638

CH

3

CH

3

SCH

3

Br

OH

6639

CH

2

CH

3

CH

2

CH

3

SCH

3

Br

OH

6640

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Br

OH

6641

OCH

3

OCH

3

SCH

3

Br

OH

6642

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Br

OH

6643

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Br

OH

6644

SCH

3

SCH

3

SCH

3

Br

OH

6645

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Br

OH

6646

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Br

OH

6647

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Br

OH

6648

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Br

OH

6649

O—(CH

2

CH

2

)—O

SCH

3

Br

OH

6650

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Br

OH

6651

S—(CH

2

CH

2

)—S

SCH

3

Br

OH

6652

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Br

OH

6653

—(CH

2

)

4

—

SCH

3

Br

OH

6654

—(CH

2

)

5

—

SCH

3

Br

OH

6655

H

H

SO

2

CH

3

Br

OH

6656

CH

3

CH

3

SO

2

CH

3

Br

OH

6657

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Br

OH

6658

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Br

OH

6659

OCH

3

OCH

3

SO

2

CH

3

Br

OH

6660

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Br

OH

6661

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Br

OH

6662

SCH

3

SCH

3

SO

2

CH

3

Br

OH

6663

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Br

OH

6664

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Br

OH

6665

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Br

OH

6666

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Br

OH

6667

O—(CH

2

CH

2

)—O

SO

2

CH

3

Br

OH

6668

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Br

OH

6669

S—(CH

2

CH

2

)—S

SO

2

CH

3

Br

OH

6670

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Br

OH

6671

—(CH

2

)

4

—

SO

2

CH

3

Br

OH

6672

—(CH

2

)

5

—

SO

2

CH

3

Br

OH

6673

H

H

PO(OCH

3

)

2

Br

OH

6674

CH

3

CH

3

PO(OCH

3

)

2

Br

OH

6675

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Br

OH

6676

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

OH

6677

OCH

3

OCH

3

PO(OCH

3

)

2

Br

OH

6678

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Br

OH

6679

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

OH

6680

SCH

3

SCH

3

PO(OCH

3

)

2

Br

OH

6681

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Br

OH

6682

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Br

OH

6683

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Br

OH

6684

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Br

OH

6685

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

OH

6686

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

OH

6687

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

OH

6688

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

OH

6689

—(CH

2

)

4

—

PO(OCH

3

)

2

Br

OH

6690

—(CH

2

)

5

—

PO(OCH

3

)

2

Br

OH

6691

H

H

PO(OCH

2

CH

3

)

2

Br

OH

6692

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Br

OH

6693

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

OH

6694

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

OH

6695

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Br

OH

6696

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

OH

6697

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

OH

6698

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Br

OH

6699

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

OH

6700

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

OH

6701

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

OH

6702

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Br

OH

6703

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

OH

6704

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

OH

6705

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

OH

6706

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

OH

6707

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Br

OH

6708

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Br

OH

6709

H

H

PO(CH

3

)

2

Br

OH

6710

CH

3

CH

3

PO(CH

3

)

2

Br

OH

6711

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Br

OH

6712

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Br

OH

6713

OCH

3

OCH

3

PO(CH

3

)

2

Br

OH

6714

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Br

OH

6715

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Br

OH

6716

SCH

3

SCH

3

PO(CH

3

)

2

Br

OH

6717

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Br

OH

6718

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Br

OH

6719

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Br

OH

6720

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Br

OH

6721

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Br

OH

6722

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Br

OH

6723

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Br

OH

6724

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Br

OH

6725

—(CH

2

)

4

—

PO(CH

3

)

2

Br

OH

6726

—(CH

2

)

5

—

PO(CH

3

)

2

Br

OH

6727

H

H

PC(CH

2

CH

3

)

2

Br

OH

6728

CH

3

CH

3

PC(CH

2

CH

3

)

2

Br

OH

6729

CH

2

CH

3

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

OH

6730

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

OH

6731

OCH

3

OCH

3

PC(CH

2

CH

3

)

2

Br

OH

6732

OCH

2

CH

3

OCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

OH

6733

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

OH

6734

SCH

3

SCH

3

PC(CH

2

CH

3

)

2

Br

OH

6735

SCH

2

CH

3

SCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

OH

6736

N(CH

3

)

2

N(CH

3

)

2

PC(CH

2

CH

3

)

2

Br

OH

6737

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PC(CH

2

CH

3

)

2

Br

OH

6738

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PC(CH

2

CH

3

)

2

Br

OH

6739

O—(CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

OH

6740

O—(CH

2

CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

OH

6741

S—(CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

OH

6742

S—(CH

2

CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

OH

6743

—(CH

2

)

4

—

PC(CH

2

CH

3

)

2

Br

OH

6744

—(CH

2

)

5

—

PC(CH

2

CH

3

)

2

Br

OH

6745

H

H

H

Br

OCOC

6

H

5

6746

CH

3

CH

3

H

Br

OCOC

6

H

5

6747

CH

2

CH

3

CH

2

CH

3

H

Br

OCOC

6

H

5

6748

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Br

OCOC

6

H

5

6749

OCH

3

OCH

3

H

Br

OCOC

6

H

5

6750

OCH

2

CH

3

OCH

2

CH

3

H

Br

OCOC

6

H

5

6751

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Br

OCOC

6

H

5

6752

SCH

3

SCH

3

H

Br

OCOC

6

H

5

6753

SCH

2

CH

3

SCH

2

CH

3

H

Br

OCOC

6

H

5

6754

N(CH

3

)

2

N(CH

3

)

2

H

Br

OCOC

6

H

5

6755

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Br

OCOC

6

H

5

6756

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Br

OCOC

6

H

5

6757

O—(CH

2

CH

2

)—O

H

Br

OCOC

6

H

5

6758

O—(CH

2

CH

2

CH

2

)—O

H

Br

OCOC

6

H

5

6759

S—(CH

2

CH

2

)—S

H

Br

OCOC

6

H

5

6760

S—(CH

2

CH

2

CH

2

)—S

H

Br

OCOC

6

H

5

6761

—(CH

2

)

4

—

H

Br

OCOC

6

H

5

6762

—(CH

2

)

5

—

H

Br

OCOC

6

H

5

6763

H

H

NO

2

Br

OCOC

6

H

5

6764

CH

3

CH

3

NO

2

Br

OCOC

6

H

5

6765

CH

2

CH

3

CH

2

CH

3

NO

2

Br

OCOC

6

H

5

6766

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Br

OCOC

6

H

5

6767

OCH

3

OCH

3

NO

2

Br

OCOC

6

H

5

6768

OCH

2

CH

3

OCH

2

CH

3

NO

2

Br

OCOC

6

H

5

6769

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Br

OCOC

6

H

5

6770

SCH

3

SCH

3

NO

2

Br

OCOC

6

H

5

6771

SCH

2

CH

3

SCH

2

CH

3

NO

2

Br

OCOC

6

H

5

6772

N(CH

3

)

2

N(CH

3

)

2

NO

2

Br

OCOC

6

H

5

6773

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Br

OCOC

6

H

5

6774

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Br

OCOC

6

H

5

6775

O—(CH

2

CH

2

)—O

NO

2

Br

OCOC

6

H

5

6776

O—(CH

2

CH

2

CH

2

)—O

NO

2

Br

OCOC

6

H

5

6777

S—(CH

2

CH

2

)—S

NO

2

Br

OCOC

6

H

5

6778

S—(CH

2

CH

2

CH

2

)—S

NO

2

Br

OCOC

6

H

5

6779

—(CH

2

)

4

—

NO

2

Br

OCOC

6

H

5

6780

—(CH

2

)

5

—

NO

2

Br

OCOC

6

H

5

6781

H

H

CN

Br

OCOC

6

H

5

6782

CH

3

CH

3

CN

Br

OCOC

6

H

5

6783

CH

2

CH

3

CH

2

CH

3

CN

Br

OCOC

6

H

5

6784

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Br

OCOC

6

H

5

6785

OCH

3

OCH

3

CN

Br

OCOC

6

H

5

6786

OCH

2

CH

3

OCH

2

CH

3

CN

Br

OCOC

6

H

5

6787

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Br

OCOC

6

H

5

6788

SCH

3

SCH

3

CN

Br

OCOC

6

H

5

6789

SCH

2

CH

3

SCH

2

CH

3

CN

Br

OCOC

6

H

5

6790

N(CH

3

)

2

N(CH

3

)

2

CN

Br

OCOC

6

H

5

6791

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Br

OCOC

6

H

5

6792

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Br

OCOC

6

H

5

6793

O—(CH

2

CH

2

)—O

CN

Br

OCOC

6

H

5

6794

O—(CH

2

CH

2

CH

2

)—O

CN

Br

OCOC

6

H

5

6795

S—(CH

2

CH

2

)—S

CN

Br

OCOC

6

H

5

6796

S—(CH

2

CH

2

CH

2

)—S

CN

Br

OCOC

6

H

5

6797

—(CH

2

)

4

—

CN

Br

OCOC

6

H

5

6798

—(CH

2

)

5

—

CN

Br

OCOC

6

H

5

6799

H

H

F

Br

OCOC

6

H

5

6800

CH

3

CH

3

F

Br

OCOC

6

H

5

6801

CH

2

CH

3

CH

2

CH

3

F

Br

OCOC

6

H

5

6802

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Br

OCOC

6

H

5

6803

OCH

3

OCH

3

F

Br

OCOC

6

H

5

6804

OCH

2

CH

3

OCH

2

CH

3

F

Br

OCOC

6

H

5

6805

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Br

OCOC

6

H

5

6806

SCH

3

SCH

3

F

Br

OCOC

6

H

5

6807

SCH

2

CH

3

SCH

2

CH

3

F

Br

OCOC

6

H

5

6808

N(CH

3

)

2

N(CH

3

)

2

F

Br

OCOC

6

H

5

6809

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Br

OCOC

6

H

5

6810

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Br

OCOC

6

H

5

6811

O—(CH

2

CH

2

)—O

F

Br

OCOC

6

H

5

6812

O—(CH

2

CH

2

CH

2

)—O

F

Br

OCOC

6

H

5

6813

S—(CH

2

CH

2

)—S

F

Br

OCOC

6

H

5

6814

S—(CH

2

CH

2

CH

2

)—S

F

Br

OCOC

6

H

5

6815

—(CH

2

)

4

—

F

Br

OCOC

6

H

5

6816

—(CH

2

)

5

—

F

Br

OCOC

6

H

5

6817

H

H

Cl

Br

OCOC

6

H

5

6818

CH

3

CH

3

Cl

Br

OCOC

6

H

5

6819

CH

2

CH

3

CH

2

CH

3

Cl

Br

OCOC

6

H

5

6820

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Br

OCOC

6

H

5

6821

OCH

3

OCH

3

Cl

Br

OCOC

6

H

5

6822

OCH

2

CH

3

OCH

2

CH

3

Cl

Br

OCOC

6

H

5

6823

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Br

OCOC

6

H

5

6824

SCH

3

SCH

3

Cl

Br

OCOC

6

H

5

6825

SCH

2

CH

3

SCH

2

CH

3

Cl

Br

OCOC

6

H

5

6826

N(CH

3

)

2

N(CH

3

)

2

Cl

Br

OCOC

6

H

5

6827

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Br

OCOC

6

H

5

6828

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Br

OCOC

6

H

5

6829

O—(CH

2

CH

2

)—O

Cl

Br

OCOC

6

H

5

6830

O—(CH

2

CH

2

CH

2

)—O

Cl

Br

OCOC

6

H

5

6831

S—(CH

2

CH

2

)—S

Cl

Br

OCOC

6

H

5

6832

S—(CH

2

CH

2

CH

2

)—S

Cl

Br

OCOC

6

H

5

6833

—(CH

2

)

4

—

Cl

Br

OCOC

6

H

5

6834

—(CH

2

)

5

—

Cl

Br

OCOC

6

H

5

6835

H

H

Br

Br

OCOC

6

H

5

6836

CH

3

CH

3

Br

Br

OCOC

6

H

5

6837

CH

2

CH

3

CH

2

CH

3

Br

Br

OCOC

6

H

5

6838

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Br

OCOC

6

H

5

6839

OCH

3

OCH

3

Br

Br

OCOC

6

H

5

6840

OCH

2

CH

3

OCH

2

CH

3

Br

Br

OCOC

6

H

5

6841

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Br

OCOC

6

H

5

6842

SCH

3

SCH

3

Br

Br

OCOC

6

H

5

6843

SCH

2

CH

3

SCH

2

CH

3

Br

Br

OCOC

6

H

5

6844

N(CH

3

)

2

N(CH

3

)

2

Br

Br

OCOC

6

H

5

6845

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Br

OCOC

6

H

5

6846

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Br

OCOC

6

H

5

6847

O—(CH

2

CH

2

)—O

Br

Br

OCOC

6

H

5

6848

O—(CH

2

CH

2

CH

2

)—O

Br

Br

OCOC

6

H

5

6849

S—(CH

2

CH

2

)—S

Br

Br

OCOC

6

H

5

6850

S—(CH

2

CH

2

CH

2

)—S

Br

Br

OCOC

6

H

5

6851

—(CH

2

)

4

—

Br

Br

OCOC

6

H

5

6852

—(CH

2

)

5

—

Br

Br

OCOC

6

H

5

6853

H

H

CH

3

Br

OCOC

6

H

5

6854

CH

3

CH

3

CH

3

Br

OCOC

6

H

5

6855

CH

2

CH

3

CH

2

CH

3

CH

3

Br

OCOC

6

H

5

6856

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Br

OCOC

6

H

5

6857

OCH

3

OCH

3

CH

3

Br

OCOC

6

H

5

6858

OCH

2

CH

3

OCH

2

CH

3

CH

3

Br

OCOC

6

H

5

6859

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Br

OCOC

6

H

5

6860

SCH

3

SCH

3

CH

3

Br

OCOC

6

H

5

6861

SCH

2

CH

3

SCH

2

CH

3

CH

3

Br

OCOC

6

H

5

6862

N(CH

3

)

2

N(CH

3

)

2

CH

3

Br

OCOC

6

H

5

6863

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Br

OCOC

6

H

5

6864

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Br

OCOC

6

H

5

6865

O—(CH

2

CH

2

)—O

CH

3

Br

OCOC

6

H

5

6866

O—(CH

2

CH

2

CH

2

)—O

CH

3

Br

OCOC

6

H

5

6867

S—(CH

2

CH

2

)—S

CH

3

Br

OCOC

6

H

5

6868

S—(CH

2

CH

2

CH

2

)—S

CH

3

Br

OCOC

6

H

5

6869

—(CH

2

)

4

—

CH

3

Br

OCOC

6

H

5

6870

—(CH

2

)

5

—

CH

3

Br

OCOC

6

H

5

6871

H

H

CH

2

CH

3

Br

OCOC

6

H

5

6872

CH

3

CH

3

CH

2

CH

3

Br

OCOC

6

H

5

6873

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Br

OCOC

6

H

5

6874

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Br

OCOC

6

H

5

6875

OCH

3

OCH

3

CH

2

CH

3

Br

OCOC

6

H

5

6876

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Br

OCOC

6

H

5

6877

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Br

OCOC

6

H

5

6878

SCH

3

SCH

3

CH

2

CH

3

Br

OCOC

6

H

5

6879

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Br

OCOC

6

H

5

6880

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Br

OCOC

6

H

5

6881

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Br

OCOC

6

H

5

6882

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Br

OCOC

6

H

5

6883

O—(CH

2

CH

2

)—O

CH

2

CH

3

Br

OCOC

6

H

5

6884

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Br

OCOC

6

H

5

6885

S—(CH

2

CH

2

)—S

CH

2

CH

3

Br

OCOC

6

H

5

6886

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Br

OCOC

6

H

5

6887

—(CH

2

)

4

—

CH

2

CH

3

Br

OCOC

6

H

5

6888

—(CH

2

)

5

—

CH

2

CH

3

Br

OCOC

6

H

5

6889

H

H

CF

3

Br

OCOC

6

H

5

6890

CH

3

CH

3

CF

3

Br

OCOC

6

H

5

6891

CH

2

CH

3

CH

2

CH

3

CF

3

Br

OCOC

6

H

5

6892

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Br

OCOC

6

H

5

6893

OCH

3

OCH

3

CF

3

Br

OCOC

6

H

5

6894

OCH

2

CH

3

OCH

2

CH

3

CF

3

Br

OCOC

6

H

5

6895

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Br

OCOC

6

H

5

6896

SCH

3

SCH

3

CF

3

Br

OCOC

6

H

5

6897

SCH

2

CH

3

SCH

2

CH

3

CF

3

Br

OCOC

6

H

5

6898

N(CH

3

)

2

N(CH

3

)

2

CF

3

Br

OCOC

6

H

5

6899

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Br

OCOC

6

H

5

6900

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Br

OCOC

6

H

5

6901

O—(CH

2

CH

2

)—O

CF

3

Br

OCOC

6

H

5

6902

O—(CH

2

CH

2

CH

2

)—O

CF

3

Br

OCOC

6

H

5

6903

S—(CH

2

CH

2

)—S

CF

3

Br

OCOC

6

H

5

6904

S—(CH

2

CH

2

CH

2

)—S

CF

3

Br

OCOC

6

H

5

6905

—(CH

2

)

4

—

CF

3

Br

OCOC

6

H

5

6906

—(CH

2

)

5

—

CF

3

Br

OCOC

6

H

5

6907

H

H

OCH

3

Br

OCOC

6

H

5

6908

CH

3

CH

3

OCH

3

Br

OCOC

6

H

5

6909

CH

2

CH

3

CH

2

CH

3

OCH

3

Br

OCOC

6

H

5

6910

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Br

OCOC

6

H

5

6911

OCH

3

OCH

3

OCH

3

Br

OCOC

6

H

5

6912

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Br

OCOC

6

H

5

6913

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Br

OCOC

6

H

5

6914

SCH

3

SCH

3

OCH

3

Br

OCOC

6

H

5

6915

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Br

OCOC

6

H

5

6916

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Br

OCOC

6

H

5

6917

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Br

OCOC

6

H

5

6918

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Br

OCOC

6

H

5

6919

O—(CH

2

CH

2

)—O

OCH

3

Br

OCOC

6

H

5

6920

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Br

OCOC

6

H

5

6921

S—(CH

2

CH

2

)—S

OCH

3

Br

OCOC

6

H

5

6922

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Br

OCOC

6

H

5

6923

—(CH

2

)

4

—

OCH

3

Br

OCOC

6

H

5

6924

—(CH

2

)

5

—

OCH

3

Br

OCOC

6

H

5

6925

H

H

OCH

2

CH

3

Br

OCOC

6

H

5

6926

CH

3

CH

3

OCH

2

CH

3

Br

OCOC

6

H

5

6927

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Br

OCOC

6

H

5

6928

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Br

OCOC

6

H

5

6929

OCH

3

OCH

3

OCH

2

CH

3

Br

OCOC

6

H

5

6930

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Br

OCOC

6

H

5

6931

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Br

OCOC

6

H

5

6932

SCH

3

SCH

3

OCH

2

CH

3

Br

OCOC

6

H

5

6933

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Br

OCOC

6

H

5

6934

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Br

OCOC

6

H

5

6935

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Br

OCOC

6

H

5

6936

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Br

OCOC

6

H

5

6937

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Br

OCOC

6

H

5

6938

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Br

OCOC

6

H

5

6939

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Br

OCOC

6

H

5

6940

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Br

OCOC

6

H

5

6941

—(CH

2

)

4

—

OCH

2

CH

3

Br

OCOC

6

H

5

6942

—(CH

2

)

5

—

OCH

2

CH

3

Br

OCOC

6

H

5

6943

H

H

SCH

3

Br

OCOC

6

H

5

6944

CH

3

CH

3

SCH

3

Br

OCOC

6

H

5

6945

CH

2

CH

3

CH

2

CH

3

SCH

3

Br

OCOC

6

H

5

6946

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Br

OCOC

6

H

5

6947

OCH

3

OCH

3

SCH

3

Br

OCOC

6

H

5

6948

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Br

OCOC

6

H

5

6949

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Br

OCOC

6

H

5

6950

SCH

3

SCH

3

SCH

3

Br

OCOC

6

H

5

6951

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Br

OCOC

6

H

5

6952

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Br

OCOC

6

H

5

6953

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Br

OCOC

6

H

5

6954

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Br

OCOC

6

H

5

6955

O—(CH

2

CH

2

)—O

SCH

3

Br

OCOC

6

H

5

6956

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Br

OCOC

6

H

5

6957

S—(CH

2

CH

2

)—S

SCH

3

Br

OCOC

6

H

5

6958

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Br

OCOC

6

H

5

6959

—(CH

2

)

4

—

SCH

3

Br

OCOC

6

H

5

6960

—(CH

2

)

5

—

SCH

3

Br

OCOC

6

H

5

6961

H

H

SO

2

CH

3

Br

OCOC

6

H

5

6962

CH

3

CH

3

SO

2

CH

3

Br

OCOC

6

H

5

6963

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Br

OCOC

6

H

5

6964

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Br

OCOC

6

H

5

6965

OCH

3

OCH

3

SO

2

CH

3

Br

OCOC

6

H

5

6966

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Br

OCOC

6

H

5

6967

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Br

OCOC

6

H

5

6968

SCH

3

SCH

3

SO

2

CH

3

Br

OCOC

6

H

5

6969

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Br

OCOC

6

H

5

6970

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Br

OCOC

6

H

5

6971

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Br

OCOC

6

H

5

6972

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Br

OCOC

6

H

5

6973

O—(CH

2

CH

2

)—O

SO

2

CH

3

Br

OCOC

6

H

5

6974

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Br

OCOC

6

H

5

6975

S—(CH

2

CH

2

)—S

SO

2

CH

3

Br

OCOC

6

H

5

6976

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Br

OCOC

6

H

5

6977

—(CH

2

)

4

—

SO

2

CH

3

Br

OCOC

6

H

5

6978

—(CH

2

)

5

—

SO

2

CH

3

Br

OCOC

6

H

5

6979

H

H

PO(OCH

3

)

2

Br

OCOC

6

H

5

6980

CH

3

CH

3

PO(OCH

3

)

2

Br

OCOC

6

H

5

6981

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Br

OCOC

6

H

5

6982

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

OCOC

6

H

5

6983

OCH

3

OCH

3

PO(OCH

3

)

2

Br

OCOC

6

H

5

6984

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Br

OCOC

6

H

5

6985

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

OCOC

6

H

5

6986

SCH

3

SCH

3

PO(OCH

3

)

2

Br

OCOC

6

H

5

6987

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Br

OCOC

6

H

5

6988

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Br

OCOC

6

H

5

6989

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Br

OCOC

6

H

5

6990

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Br

OCOC

6

H

5

6991

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

OCOC

6

H

5

6992

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

OCOC

6

H

5

6993

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

OCOC

6

H

5

6994

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

OCOC

6

H

5

6995

—(CH

2

)

4

—

PO(OCH

3

)

2

Br

OCOC

6

H

5

6996

—(CH

2

)

5

—

PO(OCH

3

)

2

Br

OCOC

6

H

5

6997

H

H

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

6998

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

6999

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7000

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7001

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7002

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7003

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7004

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7005

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7006

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7007

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7008

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7009

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7010

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7011

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7012

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7013

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7014

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Br

OCOC

6

H

5

7015

H

H

PO(CH

3

)

2

Br

OCOC

6

H

5

7016

CH

3

CH

3

PO(CH

3

)

2

Br

OCOC

6

H

5

7017

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Br

OCOC

6

H

5

7018

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Br

OCOC

6

H

5

7019

OCH

3

OCH

3

PO(CH

3

)

2

Br

OCOC

6

H

5

7020

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Br

OCOC

6

H

5

7021

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Br

OCOC

6

H

5

7022

SCH

3

SCH

3

PO(CH

3

)

2

Br

OCOC

6

H

5

7023

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Br

OCOC

6

H

5

7024

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Br

OCOC

6

H

5

7025

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Br

OCOC

6

H

5

7026

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Br

OCOC

6

H

5

7027

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Br

OCOC

6

H

5

7028

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Br

OCOC

6

H

5

7029

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Br

OCOC

6

H

5

7030

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Br

OCOC

6

H

5

7031

—(CH

2

)

4

—

PO(CH

3

)

2

Br

OCOC

6

H

5

7032

—(CH

2

)

5

—

PO(CH

3

)

2

Br

OCOC

6

H

5

7033

H

H

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7034

CH

3

CH

3

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7035

CH

2

CH

3

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7036

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7037

OCH

3

OCH

3

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7038

OCH

2

CH

3

OCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7039

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7040

SCH

3

SCH

3

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7041

SCH

2

CH

3

SCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7042

N(CH

3

)

2

N(CH

3

)

2

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7043

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7044

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7045

O—(CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7046

O—(CH

2

CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7047

S—(CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7048

S—(CH

2

CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7049

—(CH

2

)

4

—

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7050

—(CH

2

)

5

—

PC(CH

2

CH

3

)

2

Br

OCOC

6

H

5

7051

H

H

H

Br

SCH

3

7052

CH

3

CH

3

H

Br

SCH

3

7053

CH

2

CH

3

CH

2

CH

3

H

Br

SCH

3

7054

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Br

SCH

3

7055

OCH

3

OCH

3

H

Br

SCH

3

7056

OCH

2

CH

3

OCH

2

CH

3

H

Br

SCH

3

7057

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Br

SCH

3

7058

SCH

3

SCH

3

H

Br

SCH

3

7059

SCH

2

CH

3

SCH

2

CH

3

H

Br

SCH

3

7060

N(CH

3

)

2

N(CH

3

)

2

H

Br

SCH

3

7061

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Br

SCH

3

7062

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Br

SCH

3

7063

O—(CH

2

CH

2

)—O

H

Br

SCH

3

7064

O—(CH

2

CH

2

CH

2

)—O

H

Br

SCH

3

7065

S—(CH

2

CH

2

)—S

H

Br

SCH

3

7066

S—(CH

2

CH

2

CH

2

)—S

H

Br

SCH

3

7067

—(CH

2

)

4

—

H

Br

SCH

3

7068

—(CH

2

)

5

—

H

Br

SCH

3

7069

H

H

NO

2

Br

SCH

3

7070

CH

3

CH

3

NO

2

Br

SCH

3

7071

CH

2

CH

3

CH

2

CH

3

NO

2

Br

SCH

3

7072

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Br

SCH

3

7073

OCH

3

OCH

3

NO

2

Br

SCH

3

7074

OCH

2

CH

3

OCH

2

CH

3

NO

2

Br

SCH

3

7075

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Br

SCH

3

7076

SCH

3

SCH

3

NO

2

Br

SCH

3

7077

SCH

2

CH

3

SCH

2

CH

3

NO

2

Br

SCH

3

7078

N(CH

3

)

2

N(CH

3

)

2

NO

2

Br

SCH

3

7079

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Br

SCH

3

7080

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Br

SCH

3

7081

O—(CH

2

CH

2

)—O

NO

2

Br

SCH

3

7082

O—(CH

2

CH

2

CH

2

)—O

NO

2

Br

SCH

3

7083

S—(CH

2

CH

2

)—S

NO

2

Br

SCH

3

7084

S—(CH

2

CH

2

CH

2

)—S

NO

2

Br

SCH

3

7085

—(CH

2

)

4

—

NO

2

Br

SCH

3

7086

—(CH

2

)

5

—

NO

2

Br

SCH

3

7087

H

H

CN

Br

SCH

3

7088

CH

3

CH

3

CN

Br

SCH

3

7089

CH

2

CH

3

CH

2

CH

3

CN

Br

SCH

3

7090

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Br

SCH

3

7091

OCH

3

OCH

3

CN

Br

SCH

3

7092

OCH

2

CH

3

OCH

2

CH

3

CN

Br

SCH

3

7093

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Br

SCH

3

7094

SCH

3

SCH

3

CN

Br

SCH

3

7095

SCH

2

CH

3

SCH

2

CH

3

CN

Br

SCH

3

7096

N(CH

3

)

2

N(CH

3

)

2

CN

Br

SCH

3

7097

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Br

SCH

3

7098

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Br

SCH

3

7099

O—(CH

2

CH

2

)—O

CN

Br

SCH

3

7100

O—(CH

2

CH

2

CH

2

)—O

CN

Br

SCH

3

7101

S—(CH

2

CH

2

)—S

CN

Br

SCH

3

7102

S—(CH

2

CH

2

CH

2

)—S

CN

Br

SCH

3

7103

—(CH

2

)

4

—

CN

Br

SCH

3

7104

—(CH

2

)

5

—

CN

Br

SCH

3

7105

H

H

F

Br

SCH

3

7106

CH

3

CH

3

F

Br

SCH

3

7107

CH

2

CH

3

CH

2

CH

3

F

Br

SCH

3

7108

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Br

SCH

3

7109

OCH

3

OCH

3

F

Br

SCH

3

7110

OCH

2

CH

3

OCH

2

CH

3

F

Br

SCH

3

7111

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Br

SCH

3

7112

SCH

3

SCH

3

F

Br

SCH

3

7113

SCH

2

CH

3

SCH

2

CH

3

F

Br

SCH

3

7114

N(CH

3

)

2

N(CH

3

)

2

F

Br

SCH

3

7115

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Br

SCH

3

7116

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Br

SCH

3

7117

O—(CH

2

CH

2

)—O

F

Br

SCH

3

7118

O—(CH

2

CH

2

CH

2

)—O

F

Br

SCH

3

7119

S—(CH

2

CH

2

)—S

F

Br

SCH

3

7120

S—(CH

2

CH

2

CH

2

)—S

F

Br

SCH

3

7121

—(CH

2

)

4

—

F

Br

SCH

3

7122

—(CH

2

)

5

—

F

Br

SCH

3

7123

H

H

Cl

Br

SCH

3

7124

CH

3

CH

3

Cl

Br

SCH

3

7125

CH

2

CH

3

CH

2

CH

3

Cl

Br

SCH

3

7126

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Br

SCH

3

7127

OCH

3

OCH

3

Cl

Br

SCH

3

7128

OCH

2

CH

3

OCH

2

CH

3

Cl

Br

SCH

3

7129

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Br

SCH

3

7130

SCH

3

SCH

3

Cl

Br

SCH

3

7131

SCH

2

CH

3

SCH

2

CH

3

Cl

Br

SCH

3

7132

N(CH

3

)

2

N(CH

3

)

2

Cl

Br

SCH

3

7133

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Br

SCH

3

7134

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Br

SCH

3

7135

O—(CH

2

CH

2

)—O

Cl

Br

SCH

3

7136

O—(CH

2

CH

2

CH

2

)—O

Cl

Br

SCH

3

7137

S—(CH

2

CH

2

)—S

Cl

Br

SCH

3

7138

S—(CH

2

CH

2

CH

2

)—S

Cl

Br

SCH

3

7139

—(CH

2

)

4

—

Cl

Br

SCH

3

7140

—(CH

2

)

5

—

Cl

Br

SCH

3

7141

H

H

Br

Br

SCH

3

7142

CH

3

CH

3

Br

Br

SCH

3

7143

CH

2

CH

3

CH

2

CH

3

Br

Br

SCH

3

7144

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Br

SCH

3

7145

OCH

3

OCH

3

Br

Br

SCH

3

7146

OCH

2

CH

3

OCH

2

CH

3

Br

Br

SCH

3

7147

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Br

SCH

3

7148

SCH

3

SCH

3

Br

Br

SCH

3

7149

SCH

2

CH

3

SCH

2

CH

3

Br

Br

SCH

3

7150

N(CH

3

)

2

N(CH

3

)

2

Br

Br

SCH

3

7151

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Br

SCH

3

7152

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Br

SCH

3

7153

O—(CH

2

CH

2

)—O

Br

Br

SCH

3

7154

O—(CH

2

CH

2

CH

2

)—O

Br

Br

SCH

3

7155

S—(CH

2

CH

2

)—S

Br

Br

SCH

3

7156

S—(CH

2

CH

2

CH

2

)—S

Br

Br

SCH

3

7157

—(CH

2

)

4

—

Br

Br

SCH

3

7158

—(CH

2

)

5

—

Br

Br

SCH

3

7159

H

H

CH

3

Br

SCH

3

7160

CH

3

CH

3

CH

3

Br

SCH

3

7161

CH

2

CH

3

CH

2

CH

3

CH

3

Br

SCH

3

7162

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Br

SCH

3

7163

OCH

3

OCH

3

CH

3

Br

SCH

3

7164

OCH

2

CH

3

OCH

2

CH

3

CH

3

Br

SCH

3

7165

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Br

SCH

3

7166

SCH

3

SCH

3

CH

3

Br

SCH

3

7167

SCH

2

CH

3

SCH

2

CH

3

CH

3

Br

SCH

3

7168

N(CH

3

)

2

N(CH

3

)

2

CH

3

Br

SCH

3

7169

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Br

SCH

3

7170

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Br

SCH

3

7171

O—(CH

2

CH

2

)—O

CH

3

Br

SCH

3

7172

O—(CH

2

CH

2

CH

2

)—O

CH

3

Br

SCH

3

7173

S—(CH

2

CH

2

)—S

CH

3

Br

SCH

3

7174

S—(CH

2

CH

2

CH

2

)—S

CH

3

Br

SCH

3

7175

—(CH

2

)

4

—

CH

3

Br

SCH

3

7176

—(CH

2

)

5

—

CH

3

Br

SCH

3

7177

H

H

CH

2

CH

3

Br

SCH

3

7178

CH

3

CH

3

CH

2

CH

3

Br

SCH

3

7179

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Br

SCH

3

7180

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Br

SCH

3

7181

OCH

3

OCH

3

CH

2

CH

3

Br

SCH

3

7182

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Br

SCH

3

7183

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Br

SCH

3

7184

SCH

3

SCH

3

CH

2

CH

3

Br

SCH

3

7185

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Br

SCH

3

7186

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Br

SCH

3

7187

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Br

SCH

3

7188

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Br

SCH

3

7189

O—(CH

2

CH

2

)—O

CH

2

CH

3

Br

SCH

3

7190

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Br

SCH

3

7191

S—(CH

2

CH

2

)—S

CH

2

CH

3

Br

SCH

3

7192

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Br

SCH

3

7193

—(CH

2

)

4

—

CH

2

CH

3

Br

SCH

3

7194

—(CH

2

)

5

—

CH

2

CH

3

Br

SCH

3

7195

H

H

CF

3

Br

SCH

3

7196

CH

3

CH

3

CF

3

Br

SCH

3

7197

CH

2

CH

3

CH

2

CH

3

CF

3

Br

SCH

3

7198

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Br

SCH

3

7199

OCH

3

OCH

3

CF

3

Br

SCH

3

7200

OCH

2

CH

3

OCH

2

CH

3

CF

3

Br

SCH

3

7201

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Br

SCH

3

7202

SCH

3

SCH

3

CF

3

Br

SCH

3

7203

SCH

2

CH

3

SCH

2

CH

3

CF

3

Br

SCH

3

7204

N(CH

3

)

2

N(CH

3

)

2

CF

3

Br

SCH

3

7205

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Br

SCH

3

7206

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Br

SCH

3

7207

O—(CH

2

CH

2

)—O

CF

3

Br

SCH

3

7208

O—(CH

2

CH

2

CH

2

)—O

CF

3

Br

SCH

3

7209

S—(CH

2

CH

2

)—S

CF

3

Br

SCH

3

7210

S—(CH

2

CH

2

CH

2

)—S

CF

3

Br

SCH

3

7211

—(CH

2

)

4

—

CF

3

Br

SCH

3

7212

—(CH

2

)

5

—

CF

3

Br

SCH

3

7213

H

H

OCH

3

Br

SCH

3

7214

CH

3

CH

3

OCH

3

Br

SCH

3

7215

CH

2

CH

3

CH

2

CH

3

OCH

3

Br

SCH

3

7216

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Br

SCH

3

7217

OCH

3

OCH

3

OCH

3

Br

SCH

3

7218

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Br

SCH

3

7219

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Br

SCH

3

7220

SCH

3

SCH

3

OCH

3

Br

SCH

3

7221

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Br

SCH

3

7222

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Br

SCH

3

7223

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Br

SCH

3

7224

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Br

SCH

3

7225

O—(CH

2

CH

2

)—O

OCH

3

Br

SCH

3

7226

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Br

SCH

3

7227

S—(CH

2

CH

2

)—S

OCH

3

Br

SCH

3

7228

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Br

SCH

3

7229

—(CH

2

)

4

—

OCH

3

Br

SCH

3

7230

—(CH

2

)

5

—

OCH

3

Br

SCH

3

7231

H

H

OCH

2

CH

3

Br

SCH

3

7232

CH

3

CH

3

OCH

2

CH

3

Br

SCH

3

7233

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Br

SCH

3

7234

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Br

SCH

3

7235

OCH

3

OCH

3

OCH

2

CH

3

Br

SCH

3

7236

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Br

SCH

3

7237

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Br

SCH

3

7238

SCH

3

SCH

3

OCH

2

CH

3

Br

SCH

3

7239

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Br

SCH

3

7240

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Br

SCH

3

7241

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Br

SCH

3

7242

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Br

SCH

3

7243

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Br

SCH

3

7244

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Br

SCH

3

7245

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Br

SCH

3

7246

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Br

SCH

3

7247

—(CH

2

)

4

—

OCH

2

CH

3

Br

SCH

3

7248

—(CH

2

)

5

—

OCH

2

CH

3

Br

SCH

3

7249

H

H

SCH

3

Br

SCH

3

7250

CH

3

CH

3

SCH

3

Br

SCH

3

7251

CH

2

CH

3

CH

2

CH

3

SCH

3

Br

SCH

3

7252

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Br

SCH

3

7253

OCH

3

OCH

3

SCH

3

Br

SCH

3

7254

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Br

SCH

3

7255

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Br

SCH

3

7256

SCH

3

SCH

3

SCH

3

Br

SCH

3

7257

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Br

SCH

3

7258

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Br

SCH

3

7259

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Br

SCH

3

7260

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Br

SCH

3

7261

O—(CH

2

CH

2

)—O

SCH

3

Br

SCH

3

7262

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Br

SCH

3

7263

S—(CH

2

CH

2

)—S

SCH

3

Br

SCH

3

7264

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Br

SCH

3

7265

—(CH

2

)

4

—

SCH

3

Br

SCH

3

7266

—(CH

2

)

5

—

SCH

3

Br

SCH

3

7267

H

H

SO

2

CH

3

Br

SCH

3

7268

CH

3

CH

3

SO

2

CH

3

Br

SCH

3

7269

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Br

SCH

3

7270

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Br

SCH

3

7271

OCH

3

OCH

3

SO

2

CH

3

Br

SCH

3

7272

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Br

SCH

3

7273

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Br

SCH

3

7274

SCH

3

SCH

3

SO

2

CH

3

Br

SCH

3

7275

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Br

SCH

3

7276

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Br

SCH

3

7277

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Br

SCH

3

7278

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Br

SCH

3

7279

O—(CH

2

CH

2

)—O

SO

2

CH

3

Br

SCH

3

7280

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Br

SCH

3

7281

S—(CH

2

CH

2

)—S

SO

2

CH

3

Br

SCH

3

7282

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Br

SCH

3

7283

—(CH

2

)

4

—

SO

2

CH

3

Br

SCH

3

7284

—(CH

2

)

5

—

SO

2

CH

3

Br

SCH

3

7285

H

H

PO(OCH

3

)

2

Br

SCH

3

7286

CH

3

CH

3

PO(OCH

3

)

2

Br

SCH

3

7287

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Br

SCH

3

7288

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

SCH

3

7289

OCH

3

OCH

3

PO(OCH

3

)

2

Br

SCH

3

7290

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Br

SCH

3

7291

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

SCH

3

7292

SCH

3

SCH

3

PO(OCH

3

)

2

Br

SCH

3

7293

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Br

SCH

3

7294

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Br

SCH

3

7295

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Br

SCH

3

7296

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Br

SCH

3

7297

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

SCH

3

7298

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

SCH

3

7299

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

SCH

3

7300

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

SCH

3

7301

—(CH

2

)

4

—

PO(OCH

3

)

2

Br

SCH

3

7302

—(CH

2

)

5

—

PO(OCH

3

)

2

Br

SCH

3

7303

H

H

PO(OCH

2

CH

3

)

2

Br

SCH

3

7304

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Br

SCH

3

7305

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

SCH

3

7306

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

SCH

3

7307

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Br

SCH

3

7308

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

SCH

3

7309

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

SCH

3

7310

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Br

SCH

3

7311

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

SCH

3

7312

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

SCH

3

7313

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

SCH

3

7314

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Br

SCH

3

7315

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

SCH

3

7316

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

SCH

3

7317

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

SCH

3

7318

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

SCH

3

7319

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Br

SCH

3

7320

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Br

SCH

3

7321

H

H

PO(CH

3

)

2

Br

SCH

3

7322

CH

3

CH

3

PO(CH

3

)

2

Br

SCH

3

7323

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Br

SCH

3

7324

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Br

SCH

3

7325

OCH

3

OCH

3

PO(CH

3

)

2

Br

SCH

3

7326

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Br

SCH

3

7327

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Br

SCH

3

7328

SCH

3

SCH

3

PO(CH

3

)

2

Br

SCH

3

7329

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Br

SCH

3

7330

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Br

SCH

3

7331

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Br

SCH

3

7332

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Br

SCH

3

7333

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Br

SCH

3

7334

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Br

SCH

3

7335

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Br

SCH

3

7336

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Br

SCH

3

7337

—(CH

2

)

4

—

PO(CH

3

)

2

Br

SCH

3

7338

—(CH

2

)

5

—

PO(CH

3

)

2

Br

SCH

3

7339

H

H

PC(CH

2

CH

3

)

2

Br

SCH

3

7340

CH

3

CH

3

PC(CH

2

CH

3

)

2

Br

SCH

3

7341

CH

2

CH

3

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

SCH

3

7342

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

SCH

3

7343

OCH

3

OCH

3

PC(CH

2

CH

3

)

2

Br

SCH

3

7344

OCH

2

CH

3

OCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

SCH

3

7345

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

SCH

3

7346

SCH

3

SCH

3

PC(CH

2

CH

3

)

2

Br

SCH

3

7347

SCH

2

CH

3

SCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

SCH

3

7348

N(CH

3

)

2

N(CH

3

)

2

PC(CH

2

CH

3

)

2

Br

SCH

3

7349

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PC(CH

2

CH

3

)

2

Br

SCH

3

7350

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PC(CH

2

CH

3

)

2

Br

SCH

3

7351

O—(CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

SCH

3

7352

O—(CH

2

CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

SCH

3

7353

S—(CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

SCH

3

7354

S—(CH

2

CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

SCH

3

7355

—(CH

2

)

4

—

PC(CH

2

CH

3

)

2

Br

SCH

3

7356

—(CH

2

)

5

—

PC(CH

2

CH

3

)

2

Br

SCH

3

7357

H

H

H

Br

SC

6

H

5

7358

CH

3

CH

3

H

Br

SC

6

H

5

7359

CH

2

CH

3

CH

2

CH

3

H

Br

SC

6

H

5

7360

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Br

SC

6

H

5

7361

OCH

3

OCH

3

H

Br

SC

6

H

5

7362

OCH

2

CH

3

OCH

2

CH

3

H

Br

SC

6

H

5

7363

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Br

SC

6

H

5

7364

SCH

3

SCH

3

H

Br

SC

6

H

5

7365

SCH

2

CH

3

SCH

2

CH

3

H

Br

SC

6

H

5

7366

N(CH

3

)

2

N(CH

3

)

2

H

Br

SC

6

H

5

7367

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Br

SC

6

H

5

7368

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Br

SC

6

H

5

7369

O—(CH

2

CH

2

)—O

H

Br

SC

6

H

5

7370

O—(CH

2

CH

2

CH

2

)—O

H

Br

SC

6

H

5

7371

S—(CH

2

CH

2

)—S

H

Br

SC

6

H

5

7372

S—(CH

2

CH

2

CH

2

)—S

H

Br

SC

6

H

5

7373

—(CH

2

)

4

—

H

Br

SC

6

H

5

7374

—(CH

2

)

5

—

H

Br

SC

6

H

5

7375

H

H

NO

2

Br

SC

6

H

5

7376

CH

3

CH

3

NO

2

Br

SC

6

H

5

7377

CH

2

CH

3

CH

2

CH

3

NO

2

Br

SC

6

H

5

7378

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Br

SC

6

H

5

7379

OCH

3

OCH

3

NO

2

Br

SC

6

H

5

7380

OCH

2

CH

3

OCH

2

CH

3

NO

2

Br

SC

6

H

5

7381

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Br

SC

6

H

5

7382

SCH

3

SCH

3

NO

2

Br

SC

6

H

5

7383

SCH

2

CH

3

SCH

2

CH

3

NO

2

Br

SC

6

H

5

7384

N(CH

3

)

2

N(CH

3

)

2

NO

2

Br

SC

6

H

5

7385

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Br

SC

6

H

5

7386

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Br

SC

6

H

5

7387

O—(CH

2

CH

2

)—O

NO

2

Br

SC

6

H

5

7388

O—(CH

2

CH

2

CH

2

)—O

NO

2

Br

SC

6

H

5

7389

S—(CH

2

CH

2

)—S

NO

2

Br

SC

6

H

5

7390

S—(CH

2

CH

2

CH

2

)—S

NO

2

Br

SC

6

H

5

7391

—(CH

2

)

4

—

NO

2

Br

SC

6

H

5

7392

—(CH

2

)

5

—

NO

2

Br

SC

6

H

5

7393

H

H

CN

Br

SC

6

H

5

7394

CH

3

CH

3

CN

Br

SC

6

H

5

7395

CH

2

CH

3

CH

2

CH

3

CN

Br

SC

6

H

5

7396

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Br

SC

6

H

5

7397

OCH

3

OCH

3

CN

Br

SC

6

H

5

7398

OCH

2

CH

3

OCH

2

CH

3

CN

Br

SC

6

H

5

7399

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Br

SC

6

H

5

7400

SCH

3

SCH

3

CN

Br

SC

6

H

5

7401

SCH

2

CH

3

SCH

2

CH

3

CN

Br

SC

6

H

5

7402

N(CH

3

)

2

N(CH

3

)

2

CN

Br

SC

6

H

5

7403

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Br

SC

6

H

5

7404

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Br

SC

6

H

5

7405

O—(CH

2

CH

2

)—O

CN

Br

SC

6

H

5

7406

O—(CH

2

CH

2

CH

2

)—O

CN

Br

SC

6

H

5

7407

S—(CH

2

CH

2

)—S

CN

Br

SC

6

H

5

7408

S—(CH

2

CH

2

CH

2

)—S

CN

Br

SC

6

H

5

7409

—(CH

2

)

4

—

CN

Br

SC

6

H

5

7410

—(CH

2

)

5

—

CN

Br

SC

6

H

5

7411

H

H

F

Br

SC

6

H

5

7412

CH

3

CH

3

F

Br

SC

6

H

5

7413

CH

2

CH

3

CH

2

CH

3

F

Br

SC

6

H

5

7414

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Br

SC

6

H

5

7415

OCH

3

OCH

3

F

Br

SC

6

H

5

7416

OCH

2

CH

3

OCH

2

CH

3

F

Br

SC

6

H

5

7417

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Br

SC

6

H

5

7418

SCH

3

SCH

3

F

Br

SC

6

H

5

7419

SCH

2

CH

3

SCH

2

CH

3

F

Br

SC

6

H

5

7420

N(CH

3

)

2

N(CH

3

)

2

F

Br

SC

6

H

5

7421

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Br

SC

6

H

5

7422

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Br

SC

6

H

5

7423

O—(CH

2

CH

2

)—O

F

Br

SC

6

H

5

7424

O—(CH

2

CH

2

CH

2

)—O

F

Br

SC

6

H

5

7425

S—(CH

2

CH

2

)—S

F

Br

SC

6

H

5

7426

S—(CH

2

CH

2

CH

2

)—S

F

Br

SC

6

H

5

7427

—(CH

2

)

4

—

F

Br

SC

6

H

5

7428

—(CH

2

)

5

—

F

Br

SC

6

H

5

7429

H

H

Cl

Br

SC

6

H

5

7430

CH

3

CH

3

Cl

Br

SC

6

H

5

7431

CH

2

CH

3

CH

2

CH

3

Cl

Br

SC

6

H

5

7432

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Br

SC

6

H

5

7433

OCH

3

OCH

3

Cl

Br

SC

6

H

5

7434

OCH

2

CH

3

OCH

2

CH

3

Cl

Br

SC

6

H

5

7435

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Br

SC

6

H

5

7436

SCH

3

SCH

3

Cl

Br

SC

6

H

5

7437

SCH

2

CH

3

SCH

2

CH

3

Cl

Br

SC

6

H

5

7438

N(CH

3

)

2

N(CH

3

)

2

Cl

Br

SC

6

H

5

7439

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Br

SC

6

H

5

7440

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Br

SC

6

H

5

7441

O—(CH

2

CH

2

)—O

Cl

Br

SC

6

H

5

7442

O—(CH

2

CH

2

CH

2

)—O

Cl

Br

SC

6

H

5

7443

S—(CH

2

CH

2

)—S

Cl

Br

SC

6

H

5

7444

S—(CH

2

CH

2

CH

2

)—S

Cl

Br

SC

6

H

5

7445

—(CH

2

)

4

—

Cl

Br

SC

6

H

5

7446

—(CH

2

)

5

—

Cl

Br

SC

6

H

5

7447

H

H

Br

Br

SC

6

H

5

7448

CH

3

CH

3

Br

Br

SC

6

H

5

7449

CH

2

CH

3

CH

2

CH

3

Br

Br

SC

6

H

5

7450

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Br

SC

6

H

5

7451

OCH

3

OCH

3

Br

Br

SC

6

H

5

7452

OCH

2

CH

3

OCH

2

CH

3

Br

Br

SC

6

H

5

7453

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Br

SC

6

H

5

7454

SCH

3

SCH

3

Br

Br

SC

6

H

5

7455

SCH

2

CH

3

SCH

2

CH

3

Br

Br

SC

6

H

5

7456

N(CH

3

)

2

N(CH

3

)

2

Br

Br

SC

6

H

5

7457

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Br

SC

6

H

5

7458

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Br

SC

6

H

5

7459

O—(CH

2

CH

2

)—O

Br

Br

SC

6

H

5

7460

O—(CH

2

CH

2

CH

2

)—O

Br

Br

SC

6

H

5

7461

S—(CH

2

CH

2

)—S

Br

Br

SC

6

H

5

7462

S—(CH

2

CH

2

CH

2

)—S

Br

Br

SC

6

H

5

7463

—(CH

2

)

4

—

Br

Br

SC

6

H

5

7464

—(CH

2

)

5

—

Br

Br

SC

6

H

5

7465

H

H

CH

3

Br

SC

6

H

5

7466

CH

3

CH

3

CH

3

Br

SC

6

H

5

7467

CH

2

CH

3

CH

2

CH

3

CH

3

Br

SC

6

H

5

7468

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Br

SC

6

H

5

7469

OCH

3

OCH

3

CH

3

Br

SC

6

H

5

7470

OCH

2

CH

3

OCH

2

CH

3

CH

3

Br

SC

6

H

5

7471

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Br

SC

6

H

5

7472

SCH

3

SCH

3

CH

3

Br

SC

6

H

5

7473

SCH

2

CH

3

SCH

2

CH

3

CH

3

Br

SC

6

H

5

7474

N(CH

3

)

2

N(CH

3

)

2

CH

3

Br

SC

6

H

5

7475

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Br

SC

6

H

5

7476

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Br

SC

6

H

5

7477

O—(CH

2

CH

2

)—O

CH

3

Br

SC

6

H

5

7478

O—(CH

2

CH

2

CH

2

)—O

CH

3

Br

SC

6

H

5

7479

S—(CH

2

CH

2

)—S

CH

3

Br

SC

6

H

5

7480

S—(CH

2

CH

2

CH

2

)—S

CH

3

Br

SC

6

H

5

7481

—(CH

2

)

4

—

CH

3

Br

SC

6

H

5

7482

—(CH

2

)

5

—

CH

3

Br

SC

6

H

5

7483

H

H

CH

2

CH

3

Br

SC

6

H

5

7484

CH

3

CH

3

CH

2

CH

3

Br

SC

6

H

5

7485

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Br

SC

6

H

5

7486

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Br

SC

6

H

5

7487

OCH

3

OCH

3

CH

2

CH

3

Br

SC

6

H

5

7488

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Br

SC

6

H

5

7489

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Br

SC

6

H

5

7490

SCH

3

SCH

3

CH

2

CH

3

Br

SC

6

H

5

7491

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Br

SC

6

H

5

7492

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Br

SC

6

H

5

7493

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Br

SC

6

H

5

7494

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Br

SC

6

H

5

7495

O—(CH

2

CH

2

)—O

CH

2

CH

3

Br

SC

6

H

5

7496

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Br

SC

6

H

5

7497

S—(CH

2

CH

2

)—S

CH

2

CH

3

Br

SC

6

H

5

7498

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Br

SC

6

H

5

7499

—(CH

2

)

4

—

CH

2

CH

3

Br

SC

6

H

5

7500

—(CH

2

)

5

—

CH

2

CH

3

Br

SC

6

H

5

7501

H

H

CF

3

Br

SC

6

H

5

7502

CH

3

CH

3

CF

3

Br

SC

6

H

5

7503

CH

2

CH

3

CH

2

CH

3

CF

3

Br

SC

6

H

5

7504

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Br

SC

6

H

5

7505

OCH

3

OCH

3

CF

3

Br

SC

6

H

5

7506

OCH

2

CH

3

OCH

2

CH

3

CF

3

Br

SC

6

H

5

7507

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Br

SC

6

H

5

7508

SCH

3

SCH

3

CF

3

Br

SC

6

H

5

7509

SCH

2

CH

3

SCH

2

CH

3

CF

3

Br

SC

6

H

5

7510

N(CH

3

)

2

N(CH

3

)

2

CF

3

Br

SC

6

H

5

7511

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Br

SC

6

H

5

7512

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Br

SC

6

H

5

7513

O—(CH

2

CH

2

)—O

CF

3

Br

SC

6

H

5

7514

O—(CH

2

CH

2

CH

2

)—O

CF

3

Br

SC

6

H

5

7515

S—(CH

2

CH

2

)—S

CF

3

Br

SC

6

H

5

7516

S—(CH

2

CH

2

CH

2

)—S

CF

3

Br

SC

6

H

5

7517

—(CH

2

)

4

—

CF

3

Br

SC

6

H

5

7518

—(CH

2

)

5

—

CF

3

Br

SC

6

H

5

7519

H

H

OCH

3

Br

SC

6

H

5

7520

CH

3

CH

3

OCH

3

Br

SC

6

H

5

7521

CH

2

CH

3

CH

2

CH

3

OCH

3

Br

SC

6

H

5

7522

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Br

SC

6

H

5

7523

OCH

3

OCH

3

OCH

3

Br

SC

6

H

5

7524

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Br

SC

6

H

5

7525

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Br

SC

6

H

5

7526

SCH

3

SCH

3

OCH

3

Br

SC

6

H

5

7527

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Br

SC

6

H

5

7528

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Br

SC

6

H

5

7529

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Br

SC

6

H

5

7530

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Br

SC

6

H

5

7531

O—(CH

2

CH

2

)—O

OCH

3

Br

SC

6

H

5

7532

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Br

SC

6

H

5

7533

S—(CH

2

CH

2

)—S

OCH

3

Br

SC

6

H

5

7534

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Br

SC

6

H

5

7535

—(CH

2

)

4

—

OCH

3

Br

SC

6

H

5

7536

—(CH

2

)

5

—

OCH

3

Br

SC

6

H

5

7537

H

H

OCH

2

CH

3

Br

SC

6

H

5

7538

CH

3

CH

3

OCH

2

CH

3

Br

SC

6

H

5

7539

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Br

SC

6

H

5

7540

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Br

SC

6

H

5

7541

OCH

3

OCH

3

OCH

2

CH

3

Br

SC

6

H

5

7542

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Br

SC

6

H

5

7543

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Br

SC

6

H

5

7544

SCH

3

SCH

3

OCH

2

CH

3

Br

SC

6

H

5

7545

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Br

SC

6

H

5

7546

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Br

SC

6

H

5

7547

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Br

SC

6

H

5

7548

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Br

SC

6

H

5

7549

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Br

SC

6

H

5

7550

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Br

SC

6

H

5

7551

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Br

SC

6

H

5

7552

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Br

SC

6

H

5

7553

—(CH

2

)

4

—

OCH

2

CH

3

Br

SC

6

H

5

7554

—(CH

2

)

5

—

OCH

2

CH

3

Br

SC

6

H

5

7555

H

H

SCH

3

Br

SC

6

H

5

7556

CH

3

CH

3

SCH

3

Br

SC

6

H

5

7557

CH

2

CH

3

CH

2

CH

3

SCH

3

Br

SC

6

H

5

7558

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Br

SC

6

H

5

7559

OCH

3

OCH

3

SCH

3

Br

SC

6

H

5

7560

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Br

SC

6

H

5

7561

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Br

SC

6

H

5

7562

SCH

3

SCH

3

SCH

3

Br

SC

6

H

5

7563

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Br

SC

6

H

5

7564

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Br

SC

6

H

5

7565

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Br

SC

6

H

5

7566

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Br

SC

6

H

5

7567

O—(CH

2

CH

2

)—O

SCH

3

Br

SC

6

H

5

7568

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Br

SC

6

H

5

7569

S—(CH

2

CH

2

)—S

SCH

3

Br

SC

6

H

5

7570

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Br

SC

6

H

5

7571

—(CH

2

)

4

—

SCH

3

Br

SC

6

H

5

7572

—(CH

2

)

5

—

SCH

3

Br

SC

6

H

5

7573

H

H

SO

2

CH

3

Br

SC

6

H

5

7574

CH

3

CH

3

SO

2

CH

3

Br

SC

6

H

5

7575

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Br

SC

6

H

5

7576

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Br

SC

6

H

5

7577

OCH

3

OCH

3

SO

2

CH

3

Br

SC

6

H

5

7578

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Br

SC

6

H

5

7579

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Br

SC

6

H

5

7580

SCH

3

SCH

3

SO

2

CH

3

Br

SC

6

H

5

7581

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Br

SC

6

H

5

7582

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Br

SC

6

H

5

7583

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Br

SC

6

H

5

7584

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Br

SC

6

H

5

7585

O—(CH

2

CH

2

)—O

SO

2

CH

3

Br

SC

6

H

5

7586

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Br

SC

6

H

5

7587

S—(CH

2

CH

2

)—S

SO

2

CH

3

Br

SC

6

H

5

7588

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Br

SC

6

H

5

7589

—(CH

2

)

4

—

SO

2

CH

3

Br

SC

6

H

5

7590

—(CH

2

)

5

—

SO

2

CH

3

Br

SC

6

H

5

7591

H

H

PO(OCH

3

)

2

Br

SC

6

H

5

7592

CH

3

CH

3

PO(OCH

3

)

2

Br

SC

6

H

5

7593

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Br

SC

6

H

5

7594

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

SC

6

H

5

7595

OCH

3

OCH

3

PO(OCH

3

)

2

Br

SC

6

H

5

7596

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Br

SC

6

H

5

7597

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

SC

6

H

5

7598

SCH

3

SCH

3

PO(OCH

3

)

2

Br

SC

6

H

5

7599

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Br

SC

6

H

5

7600

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Br

SC

6

H

5

7601

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Br

SC

6

H

5

7602

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Br

SC

6

H

5

7603

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

SC

6

H

5

7604

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

SC

6

H

5

7605

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

SC

6

H

5

7606

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

SC

6

H

5

7607

—(CH

2

)

4

—

PO(OCH

3

)

2

Br

SC

6

H

5

7608

—(CH

2

)

5

—

PO(OCH

3

)

2

Br

SC

6

H

5

7609

H

H

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7610

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7611

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7612

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7613

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7614

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7615

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7616

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7617

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7618

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7619

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7620

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7621

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7622

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7623

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7624

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7625

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7626

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Br

SC

6

H

5

7627

H

H

PO(CH

3

)

2

Br

SC

6

H

5

7628

CH

3

CH

3

PO(CH

3

)

2

Br

SC

6

H

5

7629

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Br

SC

6

H

5

7630

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Br

SC

6

H

5

7631

OCH

3

OCH

3

PO(CH

3

)

2

Br

SC

6

H

5

7632

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Br

SC

6

H

5

7633

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Br

SC

6

H

5

7634

SCH

3

SCH

3

PO(CH

3

)

2

Br

SC

6

H

5

7635

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Br

SC

6

H

5

7636

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Br

SC

6

H

5

7637

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Br

SC

6

H

5

7638

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Br

SC

6

H

5

7639

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Br

SC

6

H

5

7640

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Br

SC

6

H

5

7641

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Br

SC

6

H

5

7642

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Br

SC

6

H

5

7643

—(CH

2

)

4

—

PO(CH

3

)

2

Br

SC

6

H

5

7644

—(CH

2

)

5

—

PO(CH

3

)

2

Br

SC

6

H

5

7645

H

H

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7646

CH

3

CH

3

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7647

CH

2

CH

3

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7648

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7649

OCH

3

OCH

3

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7650

OCH

2

CH

3

OCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7651

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7652

SCH

3

SCH

3

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7653

SCH

2

CH

3

SCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7654

N(CH

3

)

2

N(CH

3

)

2

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7655

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7656

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7657

O—(CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7658

O—(CH

2

CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7659

S—(CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7660

S—(CH

2

CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7661

—(CH

2

)

4

—

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7662

—(CH

2

)

5

—

PC(CH

2

CH

3

)

2

Br

SC

6

H

5

7663

H

H

H

Br

Het1

7664

CH

3

CH

3

H

Br

Het1

7665

CH

2

CH

3

CH

2

CH

3

H

Br

Het1

7666

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Br

Het1

7667

OCH

3

OCH

3

H

Br

Het1

7668

OCH

2

CH

3

OCH

2

CH

3

H

Br

Het1

7669

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Br

Het1

7670

SCH

3

SCH

3

H

Br

Het1

7671

SCH

2

CH

3

SCH

2

CH

3

H

Br

Het1

7672

N(CH

3

)

2

N(CH

3

)

2

H

Br

Het1

7673

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Br

Het1

7674

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Br

Het1

7675

O—(CH

2

CH

2

)—O

H

Br

Het1

7676

O—(CH

2

CH

2

CH

2

)—O

H

Br

Het1

7677

S—(CH

2

CH

2

)—S

H

Br

Het1

7678

S—(CH

2

CH

2

CH

2

)—S

H

Br

Het1

7679

—(CH

2

)

4

—

H

Br

Het1

7680

—(CH

2

)

5

—

H

Br

Het1

7681

H

H

NO

2

Br

Het1

7682

CH

3

CH

3

NO

2

Br

Het1

7683

CH

2

CH

3

CH

2

CH

3

NO

2

Br

Het1

7684

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Br

Het1

7685

OCH

3

OCH

3

NO

2

Br

Het1

7686

OCH

2

CH

3

OCH

2

CH

3

NO

2

Br

Het1

7687

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Br

Het1

7688

SCH

3

SCH

3

NO

2

Br

Het1

7689

SCH

2

CH

3

SCH

2

CH

3

NO

2

Br

Het1

7690

N(CH

3

)

2

N(CH

3

)

2

NO

2

Br

Het1

7691

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Br

Het1

7692

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Br

Het1

7693

O—(CH

2

CH

2

)—O

NO

2

Br

Het1

7694

O—(CH

2

CH

2

CH

2

)—O

NO

2

Br

Het1

7695

S—(CH

2

CH

2

)—S

NO

2

Br

Het1

7696

S—(CH

2

CH

2

CH

2

)—S

NO

2

Br

Het1

7697

—(CH

2

)

4

—

NO

2

Br

Het1

7698

—(CH

2

)

5

—

NO

2

Br

Het1

7699

H

H

CN

Br

Het1

7700

CH

3

CH

3

CN

Br

Het1

7701

CH

2

CH

3

CH

2

CH

3

CN

Br

Het1

7702

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Br

Het1

7703

OCH

3

OCH

3

CN

Br

Het1

7704

OCH

2

CH

3

OCH

2

CH

3

CN

Br

Het1

7705

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Br

Het1

7706

SCH

3

SCH

3

CN

Br

Het1

7707

SCH

2

CH

3

SCH

2

CH

3

CN

Br

Het1

7708

N(CH

3

)

2

N(CH

3

)

2

CN

Br

Het1

7709

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Br

Het1

7710

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Br

Het1

7711

O—(CH

2

CH

2

)—O

CN

Br

Het1

7712

O—(CH

2

CH

2

CH

2

)—O

CN

Br

Het1

7713

S—(CH

2

CH

2

)—S

CN

Br

Het1

7714

S—(CH

2

CH

2

CH

2

)—S

CN

Br

Het1

7715

—(CH

2

)

4

—

CN

Br

Het1

7716

—(CH

2

)

5

—

CN

Br

Het1

7717

H

H

F

Br

Het1

7718

CH

3

CH

3

F

Br

Het1

7719

CH

2

CH

3

CH

2

CH

3

F

Br

Het1

7720

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Br

Het1

7721

OCH

3

OCH

3

F

Br

Het1

7722

OCH

2

CH

3

OCH

2

CH

3

F

Br

Het1

7723

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Br

Het1

7724

SCH

3

SCH

3

F

Br

Het1

7725

SCH

2

CH

3

SCH

2

CH

3

F

Br

Het1

7726

N(CH

3

)

2

N(CH

3

)

2

F

Br

Het1

7727

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Br

Het1

7728

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Br

Het1

7729

O—(CH

2

CH

2

)—O

F

Br

Het1

7730

O—(CH

2

CH

2

CH

2

)—O

F

Br

Het1

7731

S—(CH

2

CH

2

)—S

F

Br

Het1

7732

S—(CH

2

CH

2

CH

2

)—S

F

Br

Het1

7733

—(CH

2

)

4

—

F

Br

Het1

7734

—(CH

2

)

5

—

F

Br

Het1

7735

H

H

Cl

Br

Het1

7736

CH

3

CH

3

Cl

Br

Het1

7737

CH

2

CH

3

CH

2

CH

3

Cl

Br

Het1

7738

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Br

Het1

7739

OCH

3

OCH

3

Cl

Br

Het1

7740

OCH

2

CH

3

OCH

2

CH

3

Cl

Br

Het1

7741

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Br

Het1

7742

SCH

3

SCH

3

Cl

Br

Het1

7743

SCH

2

CH

3

SCH

2

CH

3

Cl

Br

Het1

7744

N(CH

3

)

2

N(CH

3

)

2

Cl

Br

Het1

7745

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Br

Het1

7746

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Br

Het1

7747

O—(CH

2

CH

2

)—O

Cl

Br

Het1

7748

O—(CH

2

CH

2

CH

2

)—O

Cl

Br

Het1

7749

S—(CH

2

CH

2

)—S

Cl

Br

Het1

7750

S—(CH

2

CH

2

CH

2

)—S

Cl

Br

Het1

7751

—(CH

2

)

4

—

Cl

Br

Het1

7752

—(CH

2

)

5

—

Cl

Br

Het1

7753

H

H

Br

Br

Het1

7754

CH

3

CH

3

Br

Br

Het1

7755

CH

2

CH

3

CH

2

CH

3

Br

Br

Het1

7756

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Br

Het1

7757

OCH

3

OCH

3

Br

Br

Het1

7758

OCH

2

CH

3

OCH

2

CH

3

Br

Br

Het1

7759

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Br

Het1

7760

SCH

3

SCH

3

Br

Br

Het1

7761

SCH

2

CH

3

SCH

2

CH

3

Br

Br

Het1

7762

N(CH

3

)

2

N(CH

3

)

2

Br

Br

Het1

7763

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Br

Het1

7764

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Br

Het1

7765

O—(CH

2

CH

2

)—O

Br

Br

Het1

7766

O—(CH

2

CH

2

CH

2

)—O

Br

Br

Het1

7767

S—(CH

2

CH

2

)—S

Br

Br

Het1

7768

S—(CH

2

CH

2

CH

2

)—S

Br

Br

Het1

7769

—(CH

2

)

4

—

Br

Br

Het1

7770

—(CH

2

)

5

—

Br

Br

Het1

7771

H

H

CH

3

Br

Het1

7772

CH

3

CH

3

CH

3

Br

Het1

7773

CH

2

CH

3

CH

2

CH

3

CH

3

Br

Het1

7774

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Br

Het1

7775

OCH

3

OCH

3

CH

3

Br

Het1

7776

OCH

2

CH

3

OCH

2

CH

3

CH

3

Br

Het1

7777

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Br

Het1

7778

SCH

3

SCH

3

CH

3

Br

Het1

7779

SCH

2

CH

3

SCH

2

CH

3

CH

3

Br

Het1

7780

N(CH

3

)

2

N(CH

3

)

2

CH

3

Br

Het1

7781

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Br

Het1

7782

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Br

Het1

7783

O—(CH

2

CH

2

)—O

CH

3

Br

Het1

7784

O—(CH

2

CH

2

CH

2

)—O

CH

3

Br

Het1

7785

S—(CH

2

CH

2

)—S

CH

3

Br

Het1

7786

S—(CH

2

CH

2

CH

2

)—S

CH

3

Br

Het1

7787

—(CH

2

)

4

—

CH

3

Br

Het1

7788

—(CH

2

)

5

—

CH

3

Br

Het1

7789

H

H

CH

2

CH

3

Br

Het1

7790

CH

3

CH

3

CH

2

CH

3

Br

Het1

7791

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Br

Het1

7792

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Br

Het1

7793

OCH

3

OCH

3

CH

2

CH

3

Br

Het1

7794

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Br

Het1

7795

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Br

Het1

7796

SCH

3

SCH

3

CH

2

CH

3

Br

Het1

7797

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Br

Het1

7798

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Br

Het1

7799

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Br

Het1

7800

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Br

Het1

7801

O—(CH

2

CH

2

)—O

CH

2

CH

3

Br

Het1

7802

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Br

Het1

7803

S—(CH

2

CH

2

)—S

CH

2

CH

3

Br

Het1

7804

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Br

Het1

7805

—(CH

2

)

4

—

CH

2

CH

3

Br

Het1

7806

—(CH

2

)

5

—

CH

2

CH

3

Br

Het1

7807

H

H

CF

3

Br

Het1

7808

CH

3

CH

3

CF

3

Br

Het1

7809

CH

2

CH

3

CH

2

CH

3

CF

3

Br

Het1

7810

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Br

Het1

7811

OCH

3

OCH

3

CF

3

Br

Het1

7812

OCH

2

CH

3

OCH

2

CH

3

CF

3

Br

Het1

7813

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Br

Het1

7814

SCH

3

SCH

3

CF

3

Br

Het1

7815

SCH

2

CH

3

SCH

2

CH

3

CF

3

Br

Het1

7816

N(CH

3

)

2

N(CH

3

)

2

CF

3

Br

Het1

7817

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Br

Het1

7818

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Br

Het1

7819

O—(CH

2

CH

2

)—O

CF

3

Br

Het1

7820

O—(CH

2

CH

2

CH

2

)—O

CF

3

Br

Het1

7821

S—(CH

2

CH

2

)—S

CF

3

Br

Het1

7822

S—(CH

2

CH

2

CH

2

)—S

CF

3

Br

Het1

7823

—(CH

2

)

4

—

CF

3

Br

Het1

7824

—(CH

2

)

5

—

CF

3

Br

Het1

7825

H

H

OCH

3

Br

Het1

7826

CH

3

CH

3

OCH

3

Br

Het1

7827

CH

2

CH

3

CH

2

CH

3

OCH

3

Br

Het1

7828

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Br

Het1

7829

OCH

3

OCH

3

OCH

3

Br

Het1

7830

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Br

Het1

7831

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Br

Het1

7832

SCH

3

SCH

3

OCH

3

Br

Het1

7833

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Br

Het1

7834

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Br

Het1

7835

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Br

Het1

7836

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Br

Het1

7837

O—(CH

2

CH

2

)—O

OCH

3

Br

Het1

7838

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Br

Het1

7839

S—(CH

2

CH

2

)—S

OCH

3

Br

Het1

7840

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Br

Het1

7841

—(CH

2

)

4

—

OCH

3

Br

Het1

7842

—(CH

2

)

5

—

OCH

3

Br

Het1

7843

H

H

OCH

2

CH

3

Br

Het1

7844

CH

3

CH

3

OCH

2

CH

3

Br

Het1

7845

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Br

Het1

7846

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Br

Het1

7847

OCH

3

OCH

3

OCH

2

CH

3

Br

Het1

7848

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Br

Het1

7849

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Br

Het1

7850

SCH

3

SCH

3

OCH

2

CH

3

Br

Het1

7851

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Br

Het1

7852

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Br

Het1

7853

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Br

Het1

7854

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Br

Het1

7855

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Br

Het1

7856

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Br

Het1

7857

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Br

Het1

7858

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Br

Het1

7859

—(CH

2

)

4

—

OCH

2

CH

3

Br

Het1

7860

—(CH

2

)

5

—

OCH

2

CH

3

Br

Het1

7861

H

H

SCH

3

Br

Het1

7862

CH

3

CH

3

SCH

3

Br

Het1

7863

CH

2

CH

3

CH

2

CH

3

SCH

3

Br

Het1

7864

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Br

Het1

7865

OCH

3

OCH

3

SCH

3

Br

Het1

7866

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Br

Het1

7867

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Br

Het1

7868

SCH

3

SCH

3

SCH

3

Br

Het1

7869

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Br

Het1

7870

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Br

Het1

7871

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Br

Het1

7872

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Br

Het1

7873

O—(CH

2

CH

2

)—O

SCH

3

Br

Het1

7874

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Br

Het1

7875

S—(CH

2

CH

2

)—S

SCH

3

Br

Het1

7876

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Br

Het1

7877

—(CH

2

)

4

—

SCH

3

Br

Het1

7878

—(CH

2

)

5

—

SCH

3

Br

Het1

7879

H

H

SO

2

CH

3

Br

Het1

7880

CH

3

CH

3

SO

2

CH

3

Br

Het1

7881

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Br

Het1

7882

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Br

Het1

7883

OCH

3

OCH

3

SO

2

CH

3

Br

Het1

7884

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Br

Het1

7885

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Br

Het1

7886

SCH

3

SCH

3

SO

2

CH

3

Br

Het1

7887

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Br

Het1

7888

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Br

Het1

7889

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Br

Het1

7890

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Br

Het1

7891

O—(CH

2

CH

2

)—O

SO

2

CH

3

Br

Het1

7892

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Br

Het1

7893

S—(CH

2

CH

2

)—S

SO

2

CH

3

Br

Het1

7894

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Br

Het1

7895

—(CH

2

)

4

—

SO

2

CH

3

Br

Het1

7896

—(CH

2

)

5

—

SO

2

CH

3

Br

Het1

7897

H

H

PO(OCH

3

)

2

Br

Het1

7898

CH

3

CH

3

PO(OCH

3

)

2

Br

Het1

7899

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Br

Het1

7900

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

Het1

7901

OCH

3

OCH

3

PO(OCH

3

)

2

Br

Het1

7902

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Br

Het1

7903

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

Het1

7904

SCH

3

SCH

3

PO(OCH

3

)

2

Br

Het1

7905

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Br

Het1

7906

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Br

Het1

7907

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Br

Het1

7908

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Br

Het1

7909

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

Het1

7910

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

Het1

7911

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

Het1

7912

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

Het1

7913

—(CH

2

)

4

—

PO(OCH

3

)

2

Br

Het1

7914

—(CH

2

)

5

—

PO(OCH

3

)

2

Br

Het1

7915

H

H

PO(OCH

2

CH

3

)

2

Br

Het1

7916

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Br

Het1

7917

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het1

7918

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het1

7919

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Br

Het1

7920

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het1

7921

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het1

7922

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Br

Het1

7923

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het1

7924

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

Het1

7925

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

Het1

7926

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Br

Het1

7927

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

Het1

7928

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

Het1

7929

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

Het1

7930

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

Het1

7931

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Br

Het1

7932

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Br

Het1

7933

H

H

PO(CH

3

)

2

Br

Het1

7934

CH

3

CH

3

PO(CH

3

)

2

Br

Het1

7935

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Br

Het1

7936

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Br

Het1

7937

OCH

3

OCH

3

PO(CH

3

)

2

Br

Het1

7938

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Br

Het1

7939

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Br

Het1

7940

SCH

3

SCH

3

PO(CH

3

)

2

Br

Het1

7941

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Br

Het1

7942

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Br

Het1

7943

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Br

Het1

7944

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Br

Het1

7945

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Br

Het1

7946

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Br

Het1

7947

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Br

Het1

7948

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Br

Het1

7949

—(CH

2

)

4

—

PO(CH

3

)

2

Br

Het1

7950

—(CH

2

)

5

—

PO(CH

3

)

2

Br

Het1

7951

H

H

PC(CH

2

CH

3

)

2

Br

Het1

7952

CH

3

CH

3

PC(CH

2

CH

3

)

2

Br

Het1

7953

CH

2

CH

3

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het1

7954

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het1

7955

OCH

3

OCH

3

PC(CH

2

CH

3

)

2

Br

Het1

7956

OCH

2

CH

3

OCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het1

7957

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het1

7958

SCH

3

SCH

3

PC(CH

2

CH

3

)

2

Br

Het1

7959

SCH

2

CH

3

SCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het1

7960

N(CH

3

)

2

N(CH

3

)

2

PC(CH

2

CH

3

)

2

Br

Het1

7961

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PC(CH

2

CH

3

)

2

Br

Het1

7962

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PC(CH

2

CH

3

)

2

Br

Het1

7963

O—(CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

Het1

7964

O—(CH

2

CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

Het1

7965

S—(CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

Het1

7966

S—(CH

2

CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

Het1

7967

—(CH

2

)

4

—

PC(CH

2

CH

3

)

2

Br

Het1

7968

—(CH

2

)

5

—

PC(CH

2

CH

3

)

2

Br

Het1

7969

H

H

H

Br

Het2

7970

CH

3

CH

3

H

Br

Het2

7971

CH

2

CH

3

CH

2

CH

3

H

Br

Het2

7972

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Br

Het2

7973

OCH

3

OCH

3

H

Br

Het2

7974

OCH

2

CH

3

OCH

2

CH

3

H

Br

Het2

7975

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Br

Het2

7976

SCH

3

SCH

3

H

Br

Het2

7977

SCH

2

CH

3

SCH

2

CH

3

H

Br

Het2

7978

N(CH

3

)

2

N(CH

3

)

2

H

Br

Het2

7979

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Br

Het2

7980

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Br

Het2

7981

O—(CH

2

CH

2

)—O

H

Br

Het2

7982

O—(CH

2

CH

2

CH

2

)—O

H

Br

Het2

7983

S—(CH

2

CH

2

)—S

H

Br

Het2

7984

S—(CH

2

CH

2

CH

2

)—S

H

Br

Het2

7985

—(CH

2

)

4

—

H

Br

Het2

7986

—(CH

2

)

5

—

H

Br

Het2

7987

H

H

NO

2

Br

Het2

7988

CH

3

CH

3

NO

2

Br

Het2

7989

CH

2

CH

3

CH

2

CH

3

NO

2

Br

Het2

7990

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Br

Het2

7991

OCH

3

OCH

3

NO

2

Br

Het2

7992

OCH

2

CH

3

OCH

2

CH

3

NO

2

Br

Het2

7993

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Br

Het2

7994

SCH

3

SCH

3

NO

2

Br

Het2

7995

SCH

2

CH

3

SCH

2

CH

3

NO

2

Br

Het2

7996

N(CH

3

)

2

N(CH

3

)

2

NO

2

Br

Het2

7997

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Br

Het2

7998

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Br

Het2

7999

O—(CH

2

CH

2

)—O

NO

2

Br

Het2

8000

O—(CH

2

CH

2

CH

2

)—O

NO

2

Br

Het2

8001

S—(CH

2

CH

2

)—S

NO

2

Br

Het2

8002

S—(CH

2

CH

2

CH

2

)—S

NO

2

Br

Het2

8003

—(CH

2

)

4

—

NO

2

Br

Het2

8004

—(CH

2

)

5

—

NO

2

Br

Het2

8005

H

H

CN

Br

Het2

8006

CH

3

CH

3

CN

Br

Het2

8007

CH

2

CH

3

CH

2

CH

3

CN

Br

Het2

8008

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Br

Het2

8009

OCH

3

OCH

3

CN

Br

Het2

8010

OCH

2

CH

3

OCH

2

CH

3

CN

Br

Het2

8011

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Br

Het2

8012

SCH

3

SCH

3

CN

Br

Het2

8013

SCH

2

CH

3

SCH

2

CH

3

CN

Br

Het2

8014

N(CH

3

)

2

N(CH

3

)

2

CN

Br

Het2

8015

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Br

Het2

8016

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Br

Het2

8017

O—(CH

2

CH

2

)—O

CN

Br

Het2

8018

O—(CH

2

CH

2

CH

2

)—O

CN

Br

Het2

8019

S—(CH

2

CH

2

)—S

CN

Br

Het2

8020

S—(CH

2

CH

2

CH

2

)—S

CN

Br

Het2

8021

—(CH

2

)

4

—

CN

Br

Het2

8022

—(CH

2

)

5

—

CN

Br

Het2

8023

H

H

F

Br

Het2

8024

CH

3

CH

3

F

Br

Het2

8025

CH

2

CH

3

CH

2

CH

3

F

Br

Het2

8026

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Br

Het2

8027

OCH

3

OCH

3

F

Br

Het2

8028

OCH

2

CH

3

OCH

2

CH

3

F

Br

Het2

8029

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Br

Het2

8030

SCH

3

SCH

3

F

Br

Het2

8031

SCH

2

CH

3

SCH

2

CH

3

F

Br

Het2

8032

N(CH

3

)

2

N(CH

3

)

2

F

Br

Het2

8033

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Br

Het2

8034

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Br

Het2

8035

O—(CH

2

CH

2

)—O

F

Br

Het2

8036

O—(CH

2

CH

2

CH

2

)—O

F

Br

Het2

8037

S—(CH

2

CH

2

)—S

F

Br

Het2

8038

S—(CH

2

CH

2

CH

2

)—S

F

Br

Het2

8039

—(CH

2

)

4

—

F

Br

Het2

8040

—(CH

2

)

5

—

F

Br

Het2

8041

H

H

Cl

Br

Het2

8042

CH

3

CH

3

Cl

Br

Het2

8043

CH

2

CH

3

CH

2

CH

3

Cl

Br

Het2

8044

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Br

Het2

8045

OCH

3

OCH

3

Cl

Br

Het2

8046

OCH

2

CH

3

OCH

2

CH

3

Cl

Br

Het2

8047

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Br

Het2

8048

SCH

3

SCH

3

Cl

Br

Het2

8049

SCH

2

CH

3

SCH

2

CH

3

Cl

Br

Het2

8050

N(CH

3

)

2

N(CH

3

)

2

Cl

Br

Het2

8051

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Br

Het2

8052

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Br

Het2

8053

O—(CH

2

CH

2

)—O

Cl

Br

Het2

8054

O—(CH

2

CH

2

CH

2

)—O

Cl

Br

Het2

8055

S—(CH

2

CH

2

)—S

Cl

Br

Het2

8056

S—(CH

2

CH

2

CH

2

)—S

Cl

Br

Het2

8057

—(CH

2

)

4

—

Cl

Br

Het2

8058

—(CH

2

)

5

—

Cl

Br

Het2

8059

H

H

Br

Br

Het2

8060

CH

3

CH

3

Br

Br

Het2

8061

CH

2

CH

3

CH

2

CH

3

Br

Br

Het2

8062

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Br

Het2

8063

OCH

3

OCH

3

Br

Br

Het2

8064

OCH

2

CH

3

OCH

2

CH

3

Br

Br

Het2

8065

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Br

Het2

8066

SCH

3

SCH

3

Br

Br

Het2

8067

SCH

2

CH

3

SCH

2

CH

3

Br

Br

Het2

8068

N(CH

3

)

2

N(CH

3

)

2

Br

Br

Het2

8069

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Br

Het2

8070

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Br

Het2

8071

O—(CH

2

CH

2

)—O

Br

Br

Het2

8072

O—(CH

2

CH

2

CH

2

)—O

Br

Br

Het2

8073

S—(CH

2

CH

2

)—S

Br

Br

Het2

8074

S—(CH

2

CH

2

CH

2

)—S

Br

Br

Het2

8075

—(CH

2

)

4

—

Br

Br

Het2

8076

—(CH

2

)

5

—

Br

Br

Het2

8077

H

H

CH

3

Br

Het2

8078

CH

3

CH

3

CH

3

Br

Het2

8079

CH

2

CH

3

CH

2

CH

3

CH

3

Br

Het2

8080

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Br

Het2

8081

OCH

3

OCH

3

CH

3

Br

Het2

8082

OCH

2

CH

3

OCH

2

CH

3

CH

3

Br

Het2

8083

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Br

Het2

8084

SCH

3

SCH

3

CH

3

Br

Het2

8085

SCH

2

CH

3

SCH

2

CH

3

CH

3

Br

Het2

8086

N(CH

3

)

2

N(CH

3

)

2

CH

3

Br

Het2

8087

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Br

Het2

8088

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Br

Het2

8089

O—(CH

2

CH

2

)—O

CH

3

Br

Het2

8090

O—(CH

2

CH

2

CH

2

)—O

CH

3

Br

Het2

8091

S—(CH

2

CH

2

)—S

CH

3

Br

Het2

8092

S—(CH

2

CH

2

CH

2

)—S

CH

3

Br

Het2

8093

—(CH

2

)

4

—

CH

3

Br

Het2

8094

—(CH

2

)

5

—

CH

3

Br

Het2

8095

H

H

CH

2

CH

3

Br

Het2

8096

CH

3

CH

3

CH

2

CH

3

Br

Het2

8097

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Br

Het2

8098

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Br

Het2

8099

OCH

3

OCH

3

CH

2

CH

3

Br

Het2

8100

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Br

Het2

8101

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Br

Het2

8102

SCH

3

SCH

3

CH

2

CH

3

Br

Het2

8103

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Br

Het2

8104

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Br

Het2

8105

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Br

Het2

8106

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Br

Het2

8107

O—(CH

2

CH

2

)—O

CH

2

CH

3

Br

Het2

8108

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Br

Het2

8109

S—(CH

2

CH

2

)—S

CH

2

CH

3

Br

Het2

8110

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Br

Het2

8111

—(CH

2

)

4

—

CH

2

CH

3

Br

Het2

8112

—(CH

2

)

5

—

CH

2

CH

3

Br

Het2

8113

H

H

CF

3

Br

Het2

8114

CH

3

CH

3

CF

3

Br

Het2

8115

CH

2

CH

3

CH

2

CH

3

CF

3

Br

Het2

8116

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Br

Het2

8117

OCH

3

OCH

3

CF

3

Br

Het2

8118

OCH

2

CH

3

OCH

2

CH

3

CF

3

Br

Het2

8119

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Br

Het2

8120

SCH

3

SCH

3

CF

3

Br

Het2

8121

SCH

2

CH

3

SCH

2

CH

3

CF

3

Br

Het2

8122

N(CH

3

)

2

N(CH

3

)

2

CF

3

Br

Het2

8123

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Br

Het2

8124

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Br

Het2

8125

O—(CH

2

CH

2

)—O

CF

3

Br

Het2

8126

O—(CH

2

CH

2

CH

2

)—O

CF

3

Br

Het2

8127

S—(CH

2

CH

2

)—S

CF

3

Br

Het2

8128

S—(CH

2

CH

2

CH

2

)—S

CF

3

Br

Het2

8129

—(CH

2

)

4

—

CF

3

Br

Het2

8130

—(CH

2

)

5

—

CF

3

Br

Het2

8131

H

H

OCH

3

Br

Het2

8132

CH

3

CH

3

OCH

3

Br

Het2

8133

CH

2

CH

3

CH

2

CH

3

OCH

3

Br

Het2

8134

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Br

Het2

8135

OCH

3

OCH

3

OCH

3

Br

Het2

8136

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Br

Het2

8137

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Br

Het2

8138

SCH

3

SCH

3

OCH

3

Br

Het2

8139

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Br

Het2

8140

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Br

Het2

8141

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Br

Het2

8142

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Br

Het2

8143

O—(CH

2

CH

2

)—O

OCH

3

Br

Het2

8144

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Br

Het2

8145

S—(CH

2

CH

2

)—S

OCH

3

Br

Het2

8146

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Br

Het2

8147

—(CH

2

)

4

—

OCH

3

Br

Het2

8148

—(CH

2

)

5

—

OCH

3

Br

Het2

8149

H

H

OCH

2

CH

3

Br

Het2

8150

CH

3

CH

3

OCH

2

CH

3

Br

Het2

8151

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Br

Het2

8152

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Br

Het2

8153

OCH

3

OCH

3

OCH

2

CH

3

Br

Het2

8154

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Br

Het2

8155

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Br

Het2

8156

SCH

3

SCH

3

OCH

2

CH

3

Br

Het2

8157

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Br

Het2

8158

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Br

Het2

8159

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Br

Het2

8160

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Br

Het2

8161

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Br

Het2

8162

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Br

Het2

8163

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Br

Het2

8164

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Br

Het2

8165

—(CH

2

)

4

—

OCH

2

CH

3

Br

Het2

8166

—(CH

2

)

5

—

OCH

2

CH

3

Br

Het2

8167

H

H

SCH

3

Br

Het2

8168

CH

3

CH

3

SCH

3

Br

Het2

8169

CH

2

CH

3

CH

2

CH

3

SCH

3

Br

Het2

8170

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Br

Het2

8171

OCH

3

OCH

3

SCH

3

Br

Het2

8172

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Br

Het2

8173

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Br

Het2

8174

SCH

3

SCH

3

SCH

3

Br

Het2

8175

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Br

Het2

8176

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Br

Het2

8177

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Br

Het2

8178

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Br

Het2

8179

O—(CH

2

CH

2

)—O

SCH

3

Br

Het2

8180

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Br

Het2

8181

S—(CH

2

CH

2

)—S

SCH

3

Br

Het2

8182

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Br

Het2

8183

—(CH

2

)

4

—

SCH

3

Br

Het2

8184

—(CH

2

)

5

—

SCH

3

Br

Het2

8185

H

H

SO

2

CH

3

Br

Het2

8186

CH

3

CH

3

SO

2

CH

3

Br

Het2

8187

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Br

Het2

8188

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Br

Het2

8189

OCH

3

OCH

3

SO

2

CH

3

Br

Het2

8190

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Br

Het2

8191

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Br

Het2

8192

SCH

3

SCH

3

SO

2

CH

3

Br

Het2

8193

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Br

Het2

8194

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Br

Het2

8195

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Br

Het2

8196

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Br

Het2

8197

O—(CH

2

CH

2

)—O

SO

2

CH

3

Br

Het2

8198

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Br

Het2

8199

S—(CH

2

CH

2

)—S

SO

2

CH

3

Br

Het2

8200

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Br

Het2

8201

—(CH

2

)

4

—

SO

2

CH

3

Br

Het2

8202

—(CH

2

)

5

—

SO

2

CH

3

Br

Het2

8203

H

H

PO(OCH

3

)

2

Br

Het2

8204

CH

3

CH

3

PO(OCH

3

)

2

Br

Het2

8205

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Br

Het2

8206

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

Het2

8207

OCH

3

OCH

3

PO(OCH

3

)

2

Br

Het2

8208

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Br

Het2

8209

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

Het2

8210

SCH

3

SCH

3

PO(OCH

3

)

2

Br

Het2

8211

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Br

Het2

8212

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Br

Het2

8213

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Br

Het2

8214

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Br

Het2

8215

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

Het2

8216

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

Het2

8217

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

Het2

8218

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

Het2

8219

—(CH

2

)

4

—

PO(OCH

3

)

2

Br

Het2

8220

—(CH

2

)

5

—

PO(OCH

3

)

2

Br

Het2

8221

H

H

PO(OCH

2

CH

3

)

2

Br

Het2

8222

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Br

Het2

8223

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het2

8224

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het2

8225

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Br

Het2

8226

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het2

8227

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het2

8228

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Br

Het2

8229

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het2

8230

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

Het2

8231

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

Het2

8232

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Br

Het2

8233

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

Het2

8234

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

Het2

8235

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

Het2

8236

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

Het2

8237

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Br

Het2

8238

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Br

Het2

8239

H

H

PO(CH

3

)

2

Br

Het2

8240

CH

3

CH

3

PO(CH

3

)

2

Br

Het2

8241

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Br

Het2

8242

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Br

Het2

8243

OCH

3

OCH

3

PO(CH

3

)

2

Br

Het2

8244

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Br

Het2

8245

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Br

Het2

8246

SCH

3

SCH

3

PO(CH

3

)

2

Br

Het2

8247

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Br

Het2

8248

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Br

Het2

8249

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Br

Het2

8250

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Br

Het2

8251

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Br

Het2

8252

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Br

Het2

8253

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Br

Het2

8254

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Br

Het2

8255

—(CH

2

)

4

—

PO(CH

3

)

2

Br

Het2

8256

—(CH

2

)

5

—

PO(CH

3

)

2

Br

Het2

8257

H

H

PC(CH

2

CH

3

)

2

Br

Het2

8258

CH

3

CH

3

PC(CH

2

CH

3

)

2

Br

Het2

8259

CH

2

CH

3

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het2

8260

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het2

8261

OCH

3

OCH

3

PC(CH

2

CH

3

)

2

Br

Het2

8262

OCH

2

CH

3

OCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het2

8263

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het2

8264

SCH

3

SCH

3

PC(CH

2

CH

3

)

2

Br

Het2

8265

SCH

2

CH

3

SCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het2

8266

N(CH

3

)

2

N(CH

3

)

2

PC(CH

2

CH

3

)

2

Br

Het2

8267

N(CH

2CH

3

)

2

N(CH

2

CH

3

)

2

PC(CH

2

CH

3

)

2

Br

Het2

8268

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PC(CH

2

CH

3

)

2

Br

Het2

8269

O—(CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

Het2

8270

O—(CH

2

CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

Het2

8271

S—(CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

Het2

8272

S—(CH

2

CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

Het2

8273

—(CH

2

)

4

—

PC(CH

2

CH

3

)

2

Br

Het2

8274

—(CH

2

)

5

—

PC(CH

2

CH

3

)

2

Br

Het2

8275

H

H

H

Br

Het3

8276

CH

3

CH

3

H

Br

Het3

8277

CH

2

CH

3

CH

2

CH

3

H

Br

Het3

8278

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

Br

Het3

8279

OCH

3

OCH

3

H

Br

Het3

8280

OCH

2

CH

3

OCH

2

CH

3

H

Br

Het3

8281

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

Br

Het3

8282

SCH

3

SCH

3

H

Br

Het3

8283

SCH

2

CH

3

SCH

2

CH

3

H

Br

Het3

8284

N(CH

3

)

2

N(CH

3

)

2

H

Br

Het3

8285

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

Br

Het3

8286

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

Br

Het3

8287

O—(CH

2

CH

2

)—O

H

Br

Het3

8288

O—(CH

2

CH

2

CH

2

)—O

H

Br

Het3

8289

S—(CH

2

CH

2

)—S

H

Br

Het3

8290

S—(CH

2

CH

2

CH

2

)—S

H

Br

Het3

8291

—(CH

2

)

4

—

H

Br

Het3

8292

—(CH

2

)

5

—

H

Br

Het3

8293

H

H

NO

2

Br

Het3

8294

CH

3

CH

3

NO

2

Br

Het3

8295

CH

2

CH

3

CH

2

CH

3

NO

2

Br

Het3

8296

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

Br

Het3

8297

OCH

3

OCH

3

NO

2

Br

Het3

8298

OCH

2

CH

3

OCH

2

CH

3

NO

2

Br

Het3

8299

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

Br

Het3

8300

SCH

3

SCH

3

NO

2

Br

Het3

8301

SCH

2

CH

3

SCH

2

CH

3

NO

2

Br

Het3

8302

N(CH

3

)

2

N(CH

3

)

2

NO

2

Br

Het3

8303

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

Br

Het3

8304

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

Br

Het3

8305

O—(CH

2

CH

2

)—O

NO

2

Br

Het3

8306

O—(CH

2

CH

2

CH

2

)—O

NO

2

Br

Het3

8307

S—(CH

2

CH

2

)—S

NO

2

Br

Het3

8308

S—(CH

2

CH

2

CH

2

)—S

NO

2

Br

Het3

8309

—(CH

2

)

4

—

NO

2

Br

Het3

8310

—(CH

2

)

5

—

NO

2

Br

Het3

8311

H

H

CN

Br

Het3

8312

CH

3

CH

3

CN

Br

Het3

8313

CH

2

CH

3

CH

2

CH

3

CN

Br

Het3

8314

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

Br

Het3

8315

OCH

3

OCH

3

CN

Br

Het3

8316

OCH

2

CH

3

OCH

2

CH

3

CN

Br

Het3

8317

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

Br

Het3

8318

SCH

3

SCH

3

CN

Br

Het3

8319

SCH

2

CH

3

SCH

2

CH

3

CN

Br

Het3

8320

N(CH

3

)

2

N(CH

3

)

2

CN

Br

Het3

8321

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

Br

Het3

8322

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

Br

Het3

8323

O—(CH

2

CH

2

)—O

CN

Br

Het3

8324

O—(CH

2

CH

2

CH

2

)—O

CN

Br

Het3

8325

S—(CH

2

CH

2

)—S

CN

Br

Het3

8326

S—(CH

2

CH

2

CH

2

)—S

CN

Br

Het3

8327

—(CH

2

)

4

—

CN

Br

Het3

8328

—(CH

2

)

5

—

CN

Br

Het3

8329

H

H

F

Br

Het3

8330

CH

3

CH

3

F

Br

Het3

8331

CH

2

CH

3

CH

2

CH

3

F

Br

Het3

8332

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

Br

Het3

8333

OCH

3

OCH

3

F

Br

Het3

8334

OCH

2

CH

3

OCH

2

CH

3

F

Br

Het3

8335

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

Br

Het3

8336

SCH

3

SCH

3

F

Br

Het3

8337

SCH

2

CH

3

SCH

2

CH

3

F

Br

Het3

8338

N(CH

3

)

2

N(CH

3

)

2

F

Br

Het3

8339

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

Br

Het3

8340

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

Br

Het3

8341

O—(CH

2

CH

2

)—O

F

Br

Het3

8342

O—(CH

2

CH

2

CH

2

)—O

F

Br

Het3

8343

S—(CH

2

CH

2

)—S

F

Br

Het3

8344

S—(CH

2

CH

2

CH

2

)—S

F

Br

Het3

8345

—(CH

2

)

4

—

F

Br

Het3

8346

—(CH

2

)

5

—

F

Br

Het3

8347

H

H

Cl

Br

Het3

8348

CH

3

CH

3

Cl

Br

Het3

8349

CH

2

CH

3

CH

2

CH

3

Cl

Br

Het3

8350

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

Br

Het3

8351

OCH

3

OCH

3

Cl

Br

Het3

8352

OCH

2

CH

3

OCH

2

CH

3

Cl

Br

Het3

8353

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

Br

Het3

8354

SCH

3

SCH

3

Cl

Br

Het3

8355

SCH

2

CH

3

SCH

2

CH

3

Cl

Br

Het3

8356

N(CH

3

)

2

N(CH

3

)

2

Cl

Br

Het3

8357

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

Br

Het3

8358

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

Br

Het3

8359

O—(CH

2

CH

2

)—O

Cl

Br

Het3

8360

O—(CH

2

CH

2

CH

2

)—O

Cl

Br

Het3

8361

S—(CH

2

CH

2

)—S

Cl

Br

Het3

8362

S—(CH

2

CH

2

CH

2

)—S

Cl

Br

Het3

8363

—(CH

2

)

4

—

Cl

Br

Het3

8364

—(CH

2

)

5

—

Cl

Br

Het3

8365

H

H

Br

Br

Het3

8366

CH

3

CH

3

Br

Br

Het3

8367

CH

2

CH

3

CH

2

CH

3

Br

Br

Het3

8368

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

Br

Het3

8369

OCH

3

OCH

3

Br

Br

Het3

8370

OCH

2

CH

3

OCH

2

CH

3

Br

Br

Het3

8371

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

Br

Het3

8372

SCH

3

SCH

3

Br

Br

Het3

8373

SCH

2

CH

3

SCH

2

CH

3

Br

Br

Het3

8374

N(CH

3

)

2

N(CH

3

)

2

Br

Br

Het3

8375

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

Br

Het3

8376

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

Br

Het3

8377

O—(CH

2

CH

2

)—O

Br

Br

Het3

8378

O—(CH

2

CH

2

CH

2

)—O

Br

Br

Het3

8379

S—(CH

2

CH

2

)—S

Br

Br

Het3

8380

S—(CH

2

CH

2

CH

2

)—S

Br

Br

Het3

8381

—(CH

2

)

4

—

Br

Br

Het3

8382

—(CH

2

)

5

—

Br

Br

Het3

8383

H

H

CH

3

Br

Het3

8384

CH

3

CH

3

CH

3

Br

Het3

8385

CH

2

CH

3

CH

2

CH

3

CH

3

Br

Het3

8386

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

Br

Het3

8387

OCH

3

OCH

3

CH

3

Br

Het3

8388

OCH

2

CH

3

OCH

2

CH

3

CH

3

Br

Het3

8389

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

Br

Het3

8390

SCH

3

SCH

3

CH

3

Br

Het3

8391

SCH

2

CH

3

SCH

2

CH

3

CH

3

Br

Het3

8392

N(CH

3

)

2

N(CH

3

)

2

CH

3

Br

Het3

8393

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

Br

Het3

8394

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

Br

Het3

8395

O—(CH

2

CH

2

)—O

CH

3

Br

Het3

8396

O—(CH

2

CH

2

CH

2

)—O

CH

3

Br

Het3

8397

S—(CH

2

CH

2

)—S

CH

3

Br

Het3

8398

S—(CH

2

CH

2

CH

2

)—S

CH

3

Br

Het3

8399

—(CH

2

)

4

—

CH

3

Br

Het3

8400

—(CH

2

)

5

—

CH

3

Br

Het3

8401

H

H

CH

2

CH

3

Br

Het3

8402

CH

3

CH

3

CH

2

CH

3

Br

Het3

8403

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

Br

Het3

8404

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

Br

Het3

8405

OCH

3

OCH

3

CH

2

CH

3

Br

Het3

8406

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

Br

Het3

8407

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

Br

Het3

8408

SCH

3

SCH

3

CH

2

CH

3

Br

Het3

8409

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

Br

Het3

8410

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

Br

Het3

8411

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

Br

Het3

8412

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

Br

Het3

8413

O—(CH

2

CH

2

)—O

CH

2

CH

3

Br

Het3

8414

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

Br

Het3

8415

S—(CH

2

CH

2

)—S

CH

2

CH

3

Br

Het3

8416

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

Br

Het3

8417

—(CH

2

)

4

—

CH

2

CH

3

Br

Het3

8418

—(CH

2

)

5

—

CH

2

CH

3

Br

Het3

8419

H

H

CF

3

Br

Het3

8420

CH

3

CH

3

CF

3

Br

Het3

8421

CH

2

CH

3

CH

2

CH

3

CF

3

Br

Het3

8422

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

Br

Het3

8423

OCH

3

OCH

3

CF

3

Br

Het3

8424

OCH

2

CH

3

OCH

2

CH

3

CF

3

Br

Het3

8425

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

Br

Het3

8426

SCH

3

SCH

3

CF

3

Br

Het3

8427

SCH

2

CH

3

SCH

2

CH

3

CF

3

Br

Het3

8428

N(CH

3

)

2

N(CH

3

)

2

CF

3

Br

Het3

8429

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

Br

Het3

8430

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

Br

Het3

8431

O—(CH

2

CH

2

)—O

CF

3

Br

Het3

8432

O—(CH

2

CH

2

CH

2

)—O

CF

3

Br

Het3

8433

S—(CH

2

CH

2

)—S

CF

3

Br

Het3

8434

S—(CH

2

CH

2

CH

2

)—S

CF

3

Br

Het3

8435

—(CH

2

)

4

—

CF

3

Br

Het3

8436

—(CH

2

)

5

—

CF

3

Br

Het3

8437

H

H

OCH

3

Br

Het3

8438

CH

3

CH

3

OCH

3

Br

Het3

8439

CH

2

CH

3

CH

2

CH

3

OCH

3

Br

Het3

8440

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

Br

Het3

8441

OCH

3

OCH

3

OCH

3

Br

Het3

8442

OCH

2

CH

3

OCH

2

CH

3

OCH

3

Br

Het3

8443

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

Br

Het3

8444

SCH

3

SCH

3

OCH

3

Br

Het3

8445

SCH

2

CH

3

SCH

2

CH

3

OCH

3

Br

Het3

8446

N(CH

3

)

2

N(CH

3

)

2

OCH

3

Br

Het3

8447

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

Br

Het3

8448

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

Br

Het3

8449

O—(CH

2

CH

2

)—O

OCH

3

Br

Het3

8450

O—(CH

2

CH

2

CH

2

)—O

OCH

3

Br

Het3

8451

S—(CH

2

CH

2

)—S

OCH

3

Br

Het3

8452

S—(CH

2

CH

2

CH

2

)—S

OCH

3

Br

Het3

8453

—(CH

2

)

4

—

OCH

3

Br

Het3

8454

—(CH

2

)

5

—

OCH

3

Br

Het3

8455

H

H

OCH

2

CH

3

Br

Het3

8456

CH

3

CH

3

OCH

2

CH

3

Br

Het3

8457

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

Br

Het3

8458

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

Br

Het3

8459

OCH

3

OCH

3

OCH

2

CH

3

Br

Het3

8460

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

Br

Het3

8461

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

Br

Het3

8462

SCH

3

SCH

3

OCH

2

CH

3

Br

Het3

8463

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

Br

Het3

8464

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

Br

Het3

8465

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

Br

Het3

8466

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

Br

Het3

8467

O—(CH

2

CH

2

)—O

OCH

2

CH

3

Br

Het3

8468

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

Br

Het3

8469

S—(CH

2

CH

2

)—S

OCH

2

CH

3

Br

Het3

8470

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

Br

Het3

8471

—(CH

2

)

4

—

OCH

2

CH

3

Br

Het3

8472

—(CH

2

)

5

—

OCH

2

CH

3

Br

Het3

8473

H

H

SCH

3

Br

Het3

8474

CH

3

CH

3

SCH

3

Br

Het3

8475

CH

2

CH

3

CH

2

CH

3

SCH

3

Br

Het3

8476

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

Br

Het3

8477

OCH

3

OCH

3

SCH

3

Br

Het3

8478

OCH

2

CH

3

OCH

2

CH

3

SCH

3

Br

Het3

8479

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

Br

Het3

8480

SCH

3

SCH

3

SCH

3

Br

Het3

8481

SCH

2

CH

3

SCH

2

CH

3

SCH

3

Br

Het3

8482

N(CH

3

)

2

N(CH

3

)

2

SCH

3

Br

Het3

8483

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

Br

Het3

8484

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

Br

Het3

8485

O—(CH

2

CH

2

)—O

SCH

3

Br

Het3

8486

O—(CH

2

CH

2

CH

2

)—O

SCH

3

Br

Het3

8487

S—(CH

2

CH

2

)—S

SCH

3

Br

Het3

8488

S—(CH

2

CH

2

CH

2

)—S

SCH

3

Br

Het3

8489

—(CH

2

)

4

—

SCH

3

Br

Het3

8490

—(CH

2

)

5

—

SCH

3

Br

Het3

8491

H

H

SO

2

CH

3

Br

Het3

8492

CH

3

CH

3

SO

2

CH

3

Br

Het3

8493

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

Br

Het3

8494

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

Br

Het3

8495

OCH

3

OCH

3

SO

2

CH

3

Br

Het3

8496

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

Br

Het3

8497

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

Br

Het3

8498

SCH

3

SCH

3

SO

2

CH

3

Br

Het3

8499

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

Br

Het3

8500

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

Br

Het3

8501

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

Br

Het3

8502

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

Br

Het3

8503

O—(CH

2

CH

2

)—O

SO

2

CH

3

Br

Het3

8504

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

Br

Het3

8505

S—(CH

2

CH

2

)—S

SO

2

CH

3

Br

Het3

8506

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

Br

Het3

8507

—(CH

2

)

4

—

SO

2

CH

3

Br

Het3

8508

—(CH

2

)

5

—

SO

2

CH

3

Br

Het3

8509

H

H

PO(OCH

3

)

2

Br

Het3

8510

CH

3

CH

3

PO(OCH

3

)

2

Br

Het3

8511

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

Br

Het3

8512

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

Het3

8513

OCH

3

OCH

3

PO(OCH

3

)

2

Br

Het3

8514

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

Br

Het3

8515

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

Br

Het3

8516

SCH

3

SCH

3

PO(OCH

3

)

2

Br

Het3

8517

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

Br

Het3

8518

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

Br

Het3

8519

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

Br

Het3

8520

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

Br

Het3

8521

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

Het3

8522

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

Br

Het3

8523

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

Het3

8524

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

Br

Het3

8525

—(CH

2

)

4

—

PO(OCH

3

)

2

Br

Het3

8526

—(CH

2

)

5

—

PO(OCH

3

)

2

Br

Het3

8527

H

H

PO(OCH

2

CH

3

)

2

Br

Het3

8528

CH

3

CH

3

PO(OCH

2

CH

3

)

2

Br

Het3

8529

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het3

8530

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het3

8531

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

Br

Het3

8532

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het3

8533

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het3

8534

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

Br

Het3

8535

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

Br

Het3

8536

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

Het3

8537

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

Br

Het3

8538

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

Br

Het3

8539

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

Het3

8540

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

Br

Het3

8541

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

Het3

8542

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

Br

Het3

8543

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

Br

Het3

8544

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

Br

Het3

8545

H

H

PO(CH

3

)

2

Br

Het3

8546

CH

3

CH

3

PO(CH

3

)

2

Br

Het3

8547

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

Br

Het3

8548

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

Br

Het3

8549

OCH

3

OCH

3

PO(CH

3

)

2

Br

Het3

8550

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

Br

Het3

8551

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

Br

Het3

8552

SCH

3

SCH

3

PO(CH

3

)

2

Br

Het3

8553

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

Br

Het3

8554

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

Br

Het3

8555

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

Br

Het3

8556

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

Br

Het3

8557

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

Br

Het3

8558

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

Br

Het3

8559

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

Br

Het3

8560

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

Br

Het3

8561

—(CH

2

)

4

—

PO(CH

3

)

2

Br

Het3

8562

—(CH

2

)

5

—

PO(CH

3

)

2

Br

Het3

8563

H

H

PC(CH

2

CH

3

)

2

Br

Het3

8564

CH

3

CH

3

PC(CH

2

CH

3

)

2

Br

Het3

8565

CH

2

CH

3

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het3

8566

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het3

8567

OCH

3

OCH

3

PC(CH

2

CH

3

)

2

Br

Het3

8568

OCH

2

CH

3

OCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het3

8569

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het3

8570

SCH

3

SCH

3

PC(CH

2

CH

3

)

2

Br

Het3

8571

SCH

2

CH

3

SCH

2

CH

3

PC(CH

2

CH

3

)

2

Br

Het3

8572

N(CH

3

)

2

N(CH

3

)

2

PC(CH

2

CH

3

)

2

Br

Het3

8573

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PC(CH

2

CH

3

)

2

Br

Het3

8574

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PC(CH

2

CH

3

)

2

Br

Het3

8575

O—(CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

Het3

8576

O—(CH

2

CH

2

CH

2

)—O

PC(CH

2

CH

3

)

2

Br

Het3

8577

S—(CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

Het3

8578

S—(CH

2

CH

2

CH

2

)—S

PC(CH

2

CH

3

)

2

Br

Het3

8579

—(CH

2

)

4

—

PC(CH

2

CH

3

)

2

Br

Het3

8580

—(CH

2

)

5

—

PC(CH

2

CH

3

)

2

Br

Het3

where:

Het1 is 1-methoxy-N-methylamino;

Het2 is 1-tetrahydropyrrolyl;

Het3 is 1-tetrahydroisoxazolyl.

Extraordinary preference is also given to the compounds I1a2 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

1

; R

7

, R

8

, R

9

, R

11

, R

12

=H and R

10

=CH

3

), in particular to the compounds I1a2.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I1a3 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

1

; R

8

, R

9

, R

10

, R

11

, R

12

=H and R

7

=CH

3

), in particular to the compounds I1a3.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I1a4 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

1

; R

7

, R

8

, R

11

, R

12

=H and R

9

, R

10

=CH

3

), in particular to the compounds I1a4.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I1a5 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

1

; R

7

, R

8

=CH

3

and R

9

, R

10

, R

11

, R

12

=H), in particular to the compounds I1a5.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I1a6 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

1

; R

7

, R

8

, R

9

, R

10

=H and R

11

, R

12

=CH

3

), in particular to the compounds I1a6.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I1a7 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

1

; R

7

, R

8

, R

11

, R

12

=H and R

9

and R

10

together with the carbon to which they are attached form a carbonyl group), in particular to the compounds I1a7.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I1a8 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

1

; R

7

, R

8

, R

11

, R

12

=CH

3

and R

9

and R

10

together with the carbon to which they are attached form a carbonyl group), in particular to the compounds I1a8.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I1a9 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

1

; R

7

and R

11

together form a —CH

2

—CH

2

— chain and R

8

, R

9

, R

10

, R

12

=H), in particular to the compounds I1a9.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I2a1 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

1

; R

7

, R

8

, R

9

, R

10

, R

11

, R

12

=H), in particular to the compounds I2a1.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I2a2 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

1

; R

7

, R

8

, R

9

, R

11

, R

12

=H and R

10

=CH

3

), in particular to the compounds I2a2.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I2a3 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

1

; R

8

, R

9

, R

10

, R

11

, R

12

=H and R

7

=CH

3

), in particular to the compounds I2a3.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I2a4 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

1

; R

7

, R

8

, R

11

, R

12

=H and R

9

, R

10

=CH

3

), in particular to the compounds I2a4.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I2a5 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

1

; R

7

, R

8

=CH

3

, R

9

, R

10

, R

11

, R

12

=H), in particular to the compounds I2a5.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I2a6 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

1

; R

7

, R

8

, R

9

, R

10

=H and R

11

, R

12

=CH

3

), in particular to the compounds I2a6.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I2a7 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

1

; R

7

, R

8

, R

11

, R

12

=H and R

9

and R

10

together with the carbon to which they are attached form a carbonyl group), in particular to the compounds I2a7.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I2a8 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

1

; R

7

, R

8

, R

11

, R

12

=CH

3

and R

9

and R

10

together with the carbon to which they are attached form a carbonyl group), in particular to the compounds I2a8.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I2a9 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

1

; R

7

and R

11

together form a —CH

2

—CH

2

— chain and R

8

, R

9

, R

10

, R

12

=H), in particular to the compounds I2a9.n, where the variables R

1

to R

4

and R

6

are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b1 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=CH

3

and R

22

=H), in particular to the compounds I1b1.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b2 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=CH

2

CH

3

and R

22

=H), in particular to the compounds I1b2.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b3 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=CH(CH

3

)

2

and R

22

=H), in particular to the compounds I1b3.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b4 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=C(CH

3

)

3

and R

22

=H), in particular to the compounds I1b4.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b5 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=CH

2

CF

3

and R

22

=H), in particular to the compounds I1b5.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b6 (≡where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=CH

3

and R

22

=CH

3

), in particular to the compounds I1b6.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b7 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

7

” is attached in the 2-position; Q=Q

2

; R

21

=CH

2

CH

3

and R

22

=CH

3

), in particular to the compounds I1b7.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b8 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=CH(CH

3

)

2

and R

22

=CH

3

), in particular to the compounds I1b8.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b9 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=C(CH

3

)

3

and R

22

=CH

3

), in particular to the compounds I1b9.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b10 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=CH

2

CH

3

and R

22

=CH

3

), in particular to the compounds I1b10.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b11 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=CH

3

and R

22

=CH

3

), in particular to the compounds I1b11.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b12 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=CH

2

CH

3

and R

22

=CF

3

), in particular to the compounds I1b12.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b13 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=CH(CH

3

)

2

and R

22

=CF

3

), in particular to the compounds I1b13.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b14 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=C(CH

3

)

3

and R

22

=CF

3

), in particular to the compounds I1b14.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b15 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

2

; R

21

=CH

2

CF

3

and R

22

=CF

3

), in particular to the compounds I1b15.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b1 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=CH

3

and R

22

=H), in particular to the compounds I2b1.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b2 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=CH

2

CH

3

and R

22

=H), in particular to the compounds I2b2.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b3 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=CH(CH

3

)

2

and R

22

=H), in particular to the compounds I2b3.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b4 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=C(CH

3

)

3

and R

22

=H), in particular to the compounds I2b4.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b5 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=CH

2

CF

3

and R

22

=H), in particular to the compounds I2b5.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b6 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=CH

3

and R

22

=CH

3

), in particular to the compounds I2b6.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b7 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

7

” is attached in the 24-position; Q=Q

2

; R

21

=CH

2

CH

3

and R

22

=CH

3

), in particular to the compounds I2b7.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b8 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=CH(CH

3

)

2

and R

22

=CH

3

), in particular to the compounds I2b8.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b9 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=C(CH

3

)

3

and R

22

=CH

3

), in particular to the compounds I2b9.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b10 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=CH

2

CF

3

and R

22

=CH

3

), in particular to the compounds I2b10.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b11 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=CH

3

and R

22

=CF

3

), in particular to the compounds I2b11.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b12 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=CH

2

CH

3

and R

22

=CF

3

), in particular to the compounds I2b12.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b13(≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=CH(CH

3

)

2

and R

22

=CF

3

), in particular to the compounds I2b13.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1b14 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=C(CH

3

)

3

and R

22

=CF

3

), in particular to the compounds I2b14.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I2b15 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

2

; R

21

=CH

2

CF

3

and R

22

=CF

3

), in particular to the compounds I2b15.n, where the variables R

1

to R

4

and R

20

(which in this case corresponds to R

6

) are as defined in Table 1.

Extraordinary preference is also given to the compounds I1c1 (≡I where X=O; R

3

is attached in the 4-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

3

; 1=0, R

23

=cyclopropyl and R

24

=H), in particular to the compounds Ic1.n, where the variables R

1

to R

3

are as defined in Table 2.

TABLE 2

n

R

1

R

2

R

3

1

H

H

H

2

CH

3

CH

3

H

3

CH

2

CH

3

CH

2

CH

3

H

4

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

H

5

OCH

3

OCH

3

H

6

OCH

2

CH

3

OCH

2

CH

3

H

7

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

H

8

SCH

3

SCH

3

H

9

SCH

2

CH

3

SCH

2

CH

3

H

10

N(CH

3

)

2

N(CH

3

)

2

H

11

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

H

12

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

H

13

O—(CH

2

CH

2

)—O

H

14

O—(CH

2

CH

2

CH

2

)—O

H

15

S—(CH

2

CH

2

)—S

H

16

S—(CH

2

CH

2

CH

2

)—S

H

17

—(CH

2

)

4

—

H

18

—(CH

2

)

5

—

H

19

H

H

NO

2

20

CH

3

CH

3

NO

2

21

CH

2

CH

3

CH

2

CH

3

NO

2

22

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

NO

2

23

OCH

3

OCH

3

NO

2

24

OCH

2

CH

3

OCH

2

CH

3

NO

2

25

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

NO

2

26

SCH

3

SCH

3

NO

2

27

SCH

2

CH

3

SCH

2

CH

3

NO

2

28

N(CH

3

)

2

N(CH

3

)

2

NO

2

29

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

NO

2

30

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

NO

2

31

O—(CH

2

CH

2

)—O

NO

2

32

O—(CH

2

CH

2

CH

2

)—O

NO

2

33

S—(CH

2

CH

2

)—S

NO

2

34

S—(CH

2

CH

2

CH

2

)—S

NO

2

35

—(CH

2

)

4

—

NO

2

36

—(CH

2

)

5

—

NO

2

37

H

H

CN

38

CH

3

CH

3

CN

39

CH

2

CH

3

CH

2

CH

3

CN

40

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CN

41

OCH

3

OCH

3

CN

42

OCH

2

CH

3

OCH

2

CH

3

CN

43

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CN

44

SCH

3

SCH

3

CN

45

SCH

2

CH

3

SCH

2

CH

3

CN

46

N(CH

3

)

2

N(CH

3

)

2

CN

47

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CN

48

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CN

49

O—(CH

2

CH

2

)—O

CN

50

O—(CH

2

CH

2

CH

2

)—O

CN

51

S—(CH

2

CH

2

)—S

CN

52

S—(CH

2

CH

2

CH

2

)—S

CN

53

—(CH

2

)

4

—

CN

54

—(CH

2

)

5

—

CN

55

H

H

F

56

CH

3

CH

3

F

57

CH

2

CH

3

CH

2

CH

3

F

58

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

F

59

OCH

3

OCH

3

F

60

OCH

2

CH

3

OCH

2

CH

3

F

61

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

F

62

SCH

3

SCH

3

F

63

SCH

2

CH

3

SCH

2

CH

3

F

64

N(CH

3

)

2

N(CH

3

)

2

F

65

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

F

66

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

F

67

O—(CH

2

CH

2

)—O

F

68

O—(CH

2

CH

2

CH

2

)—O

F

69

S—(CH

2

CH

2

)—S

F

70

S—(CH

2

CH

2

CH

2

)—S

F

71

—(CH

2

)

4

—

F

72

—(CH

2

)

5

—

F

73

H

H

Cl

74

CH

3

CH

3

Cl

75

CH

2

CH

3

CH

2

CH

3

Cl

76

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Cl

77

OCH

3

OCH

3

Cl

78

OCH

2

CH

3

OCH

2

CH

3

Cl

79

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Cl

80

SCH

3

SCH

3

Cl

81

SCH

2

CH

3

SCH

2

CH

3

Cl

82

N(CH

3

)

2

N(CH

3

)

2

Cl

83

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Cl

84

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Cl

85

O—(CH

2

CH

2

)—O

Cl

86

O—(CH

2

CH

2

CH

2

)—O

Cl

87

S—(CH

2

CH

2

)—S

Cl

88

S—(CH

2

CH

2

CH

2

)—S

Cl

89

—(CH

2

)

4

—

Cl

90

—(CH

2

)

5

—

Cl

91

H

H

Br

92

CH

3

CH

3

Br

93

CH

2

CH

3

CH

2

CH

3

Br

94

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

Br

95

OCH

3

OCH

3

Br

96

OCH

2

CH

3

OCH

2

CH

3

Br

97

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

Br

98

SCH

3

SCH

3

Br

99

SCH

2

CH

3

SCH

2

CH

3

Br

100

N(CH

3

)

2

N(CH

3

)

2

Br

101

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

Br

102

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

Br

103

O—(CH

2

CH

2

)—O

Br

104

O—(CH

2

CH

2

CH

2

)—O

Br

105

S—(CH

2

CH

2

)—S

Br

106

S—(CH

2

CH

2

CH

2

)—S

Br

107

—(CH

2

)

4

—

Br

108

—(CH

2

)

5

—

Br

109

H

H

CH

3

110

CH

3

CH

3

CH

3

111

CH

2

CH

3

CH

2

CH

3

CH

3

112

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

3

113

OCH

3

OCH

3

CH

3

114

OCH

2

CH

3

OCH

2

CH

3

CH

3

115

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

3

116

SCH

3

SCH

3

CH

3

117

SCH

2

CH

3

SCH

2

CH

3

CH

3

118

N(CH

3

)

2

N(CH

3

)

2

CH

3

119

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

3

120

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

3

121

O—(CH

2

CH

2

)—O

CH

3

122

O—(CH

2

CH

2

CH

2

)—O

CH

3

123

S—(CH

2

CH

2

)—S

CH

3

124

S—(CH

2

CH

2

CH

2

)—S

CH

3

125

—(CH

2

)

4

—

CH

3

126

—(CH

2

)

5

—

CH

3

127

H

H

CH

2

CH

3

128

CH

3

CH

3

CH

2

CH

3

129

CH

2

CH

3

CH

2

CH

3

CH

2

CH

3

130

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CH

2

CH

3

131

OCH

3

OCH

3

CH

2

CH

3

132

OCH

2

CH

3

OCH

2

CH

3

CH

2

CH

3

133

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CH

2

CH

3

134

SCH

3

SCH

3

CH

2

CH

3

135

SCH

2

CH

3

SCH

2

CH

3

CH

2

CH

3

136

N(CH

3

)

2

N(CH

3

)

2

CH

2

CH

3

137

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CH

2

CH

3

138

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CH

2

CH

3

139

O—(CH

2

CH

2

)—O

CH

2

CH

3

140

O—(CH

2

CH

2

CH

2

)—O

CH

2

CH

3

141

S—(CH

2

CH

2

)—S

CH

2

CH

3

142

S—(CH

2

CH

2

CH

2

)—S

CH

2

CH

3

143

—(CH

2

)

4

—

CH

2

CH

3

144

—(CH

2

)

5

—

CH

2

CH

3

145

H

H

CF

3

146

CH

3

CH

3

CF

3

147

CH

2

CH

3

CH

2

CH

3

CF

3

148

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

CF

3

149

OCH

3

OCH

3

CF

3

150

OCH

2

CH

3

OCH

2

CH

3

CF

3

151

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

CF

3

152

SCH

3

SCH

3

CF

3

153

SCH

2

CH

3

SCH

2

CH

3

CF

3

154

N(CH

3

)

2

N(CH

3

)

2

CF

3

155

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

CF

3

156

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

CF

3

157

O—(CH

2

CH

2

)—O

CF

3

158

O—(CH

2

CH

2

CH

2

)—O

CF

3

159

S—(CH

2

CH

2

)—S

CF

3

160

S—(CH

2

CH

2

CH

2

)—S

CF

3

161

—(CH

2

)

4

—

CF

3

162

—(CH

2

)

5

—

CF

3

163

H

H

OCH

3

164

CH

3

CH

3

OCH

3

165

CH

2

CH

3

CH

2

CH

3

OCH

3

166

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

3

167

OCH

3

OCH

3

OCH

3

168

OCH

2

CH

3

OCH

2

CH

3

OCH

3

169

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

3

170

SCH

3

SCH

3

OCH

3

171

SCH

2

CH

3

SCH

2

CH

3

OCH

3

172

N(CH

3

)

2

N(CH

3

)

2

OCH

3

173

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

3

174

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

3

175

O—(CH

2

CH

2

)—O

OCH

3

176

O—(CH

2

CH

2

CH

2

)—O

OCH

3

177

S—(CH

2

CH

2

)—S

OCH

3

178

S—(CH

2

CH

2

CH

2

)—S

OCH

3

179

—(CH

2

)

4

—

OCH

3

180

—(CH

2

)

5

—

OCH

3

181

H

H

OCH

2

CH

3

182

CH

3

CH

3

OCH

2

CH

3

183

CH

2

CH

3

CH

2

CH

3

OCH

2

CH

3

184

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

OCH

2

CH

3

185

OCH

3

OCH

3

OCH

2

CH

3

186

OCH

2

CH

3

OCH

2

CH

3

OCH

2

CH

3

187

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

OCH

2

CH

3

188

SCH

3

SCH

3

OCH

2

CH

3

189

SCH

2

CH

3

SCH

2

CH

3

OCH

2

CH

3

190

N(CH

3

)

2

N(CH

3

)

2

OCH

2

CH

3

191

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

OCH

2

CH

3

192

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

OCH

2

CH

3

193

O—(CH

2

CH

2

)—O

OCH

2

CH

3

194

O—(CH

2

CH

2

CH

2

)—O

OCH

2

CH

3

195

S—(CH

2

CH

2

)—S

OCH

2

CH

3

196

S—(CH

2

CH

2

CH

2

)—S

OCH

2

CH

3

197

—(CH

2

)

4

—

OCH

2

CH

3

198

—(CH

2

)

5

—

OCH

2

CH

3

199

H

H

SCH

3

200

CH

3

CH

3

SCH

3

201

CH

2

CH

3

CH

2

CH

3

SCH

3

202

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SCH

3

203

OCH

3

OCH

3

SCH

3

204

OCH

2

CH

3

OCH

2

CH

3

SCH

3

205

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SCH

3

206

SCH

3

SCH

3

SCH

3

207

SCH

2

CH

3

SCH

2

CH

3

SCH

3

208

N(CH

3

)

2

N(CH

3

)

2

SCH

3

209

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SCH

3

210

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SCH

3

211

O—(CH

2

CH

2

)—O

SCH

3

212

O—(CH

2

CH

2

CH

2

)—O

SCH

3

213

S—(CH

2

CH

2

)—S

SCH

3

214

S—(CH

2

CH

2

CH

2

)—S

SCH

3

215

—(CH

2

)

4

—

SCH

3

216

—(CH

2

)

5

—

SCH

3

217

H

H

SO

2

CH

3

218

CH

3

CH

3

SO

2

CH

3

219

CH

2

CH

3

CH

2

CH

3

SO

2

CH

3

220

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

SO

2

CH

3

221

OCH

3

OCH

3

SO

2

CH

3

222

OCH

2

CH

3

OCH

2

CH

3

SO

2

CH

3

223

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

SO

2

CH

3

224

SCH

3

SCH

3

SO

2

CH

3

225

SCH

2

CH

3

SCH

2

CH

3

SO

2

CH

3

226

N(CH

3

)

2

N(CH

3

)

2

SO

2

CH

3

227

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

SO

2

CH

3

228

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

SO

2

CH

3

229

O—(CH

2

CH

2

)—O

SO

2

CH

3

230

O—(CH

2

CH

2

CH

2

)—O

SO

2

CH

3

231

S—(CH

2

CH

2

)—S

SO

2

CH

3

232

S—(CH

2

CH

2

CH

2

)—S

SO

2

CH

3

233

—(CH

2

)

4

—

SO

2

CH

3

234

—(CH

2

)

5

—

SO

2

CH

3

235

H

H

PO(OCH

3

)

2

236

CH

3

CH

3

PO(OCH

3

)

2

237

CH

2

CH

3

CH

2

CH

3

PO(OCH

3

)

2

238

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

3

)

2

239

OCH

3

OCH

3

PO(OCH

3

)

2

240

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

3

)

2

241

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

3

)

2

242

SCH

3

SCH

3

PO(OCH

3

)

2

243

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

3

)

2

244

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

3

)

2

245

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

3

)

2

246

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

3

)

2

247

O—(CH

2

CH

2

)—O

PO(OCH

3

)

2

248

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

3

)

2

249

S—(CH

2

CH

2

)—S

PO(OCH

3

)

2

250

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

3

)

2

251

—(CH

2

)

4

—

PO(OCH

3

)

2

252

—(CH

2

)

5

—

PO(OCH

3

)

2

253

H

H

PO(OCH

2

CH

3

)

2

254

CH

3

CH

3

PO(OCH

2

CH

3

)

2

255

CH

2

CH

3

CH

2

CH

3

PO(OCH

2

CH

3

)

2

256

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

257

OCH

3

OCH

3

PO(OCH

2

CH

3

)

2

258

OCH

2

CH

3

OCH

2

CH

3

PO(OCH

2

CH

3

)

2

259

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(OCH

2

CH

3

)

2

260

SCH

3

SCH

3

PO(OCH

2

CH

3

)

2

261

SCH

2

CH

3

SCH

2

CH

3

PO(OCH

2

CH

3

)

2

262

N(CH

3

)

2

N(CH

3

)

2

PO(OCH

2

CH

3

)

2

263

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(OCH

2

CH

3

)

2

264

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(OCH

2

CH

3

)

2

265

O—(CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

266

O—(CH

2

CH

2

CH

2

)—O

PO(OCH

2

CH

3

)

2

267

S—(CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

268

S—(CH

2

CH

2

CH

2

)—S

PO(OCH

2

CH

3

)

2

269

—(CH

2

)

4

—

PO(OCH

2

CH

3

)

2

270

—(CH

2

)

5

—

PO(OCH

2

CH

3

)

2

271

H

H

PO(CH

3

)

2

272

CH

3

CH

3

PO(CH

3

)

2

273

CH

2

CH

3

CH

2

CH

3

PO(CH

3

)

2

274

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

3

)

2

275

OCH

3

OCH

3

PO(CH

3

)

2

276

OCH

2

CH

3

OCH

2

CH

3

PO(CH

3

)

2

277

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

3

)

2

278

SCH

3

SCH

3

PO(CH

3

)

2

279

SCH

2

CH

3

SCH

2

CH

3

PO(CH

3

)

2

280

N(CH

3

)

2

N(CH

3

)

2

PO(CH

3

)

2

281

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

3

)

2

282

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

3

)

2

283

O—(CH

2

CH

2

)—O

PO(CH

3

)

2

284

O—(CH

2

CH

2

CH

2

)—O

PO(CH

3

)

2

285

S—(CH

2

CH

2

)—S

PO(CH

3

)

2

286

S—(CH

2

CH

2

CH

2

)—S

PO(CH

3

)

2

287

—(CH

2

)

4

—

PO(CH

3

)

2

288

—(CH

2

)

5

—

PO(CH

3

)

2

289

H

H

PO(CH

2

CH

3

)

2

290

CH

3

CH

3

PO(CH

2

CH

3

)

2

291

CH

2

CH

3

CH

2

CH

3

PO(CH

2

CH

3

)

2

292

CH

2

CH

2

CH

3

CH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

293

OCH

3

OCH

3

PO(CH

2

CH

3

)

2

294

OCH

2

CH

3

OCH

2

CH

3

PO(CH

2

CH

3

)

2

295

OCH

2

CH

2

CH

3

OCH

2

CH

2

CH

3

PO(CH

2

CH

3

)

2

296

SCH

3

SCH

3

PO(CH

2

CH

3

)

2

297

SCH

2

CH

3

SCH

2

CH

3

PO(CH

2

CH

3

)

2

298

N(CH

3

)

2

N(CH

3

)

2

PO(CH

2

CH

3

)

2

299

N(CH

2

CH

3

)

2

N(CH

2

CH

3

)

2

PO(CH

2

CH

3

)

2

300

N(CH

3

)(CH

2

CH

3

)

N(CH

3

)(CH

2

CH

3

)

PO(CH

2

CH

3

)

2

301

O—(CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

302

O—(CH

2

CH

2

CH

2

)—O

PO(CH

2

CH

3

)

2

303

S—(CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

304

S—(CH

2

CH

2

CH

2

)—S

PO(CH

2

CH

3

)

2

305

—(CH

2

)

4

—

PO(CH

2

CH

3

)

2

306

—(CH

2

)

5

—

PO(CH

2

CH

3

)

2

Extraordinary preference is also given to the compounds I1c2 (≡I where X=O; R

3

is attached in the 4-position, R

4

in the 5-position and “P(═X)R

1

R

2

” in the 2-position; Q=Q

3

; R

4

=CH

3

, R

23

=cyclopropyl and R

24

=H), in particular to the compounds I1c2.n, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I1c3 (≡I where X=O; R

3

is attached in the 4-position, R

4

in the 5-position and “P(═X)R

1

R

2

” in the 2-position; Q=Q

3

; R

4

=Cl, R

23

=cyclopropyl and R

24

=H), in particular to the compounds I1c3.n, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I1c4 (≡I where X=O; R

3

is attached in the 4-position, R

4

in the 5-position and “P(═X)R

1

R

2

” in the 2-position; Q=Q

3

; R

4

=Br, R

23

=cyclopropyl and R

24

=H), in particular to the compounds I1c4, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I2cl (≡I where X=O; R

3

is attached in the 2-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

3

; 1=0; R

23

=cyclopropyl and R

24

=H), in particular to the compounds I2c1.n, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I2c2 (≡I where X=O; R

3

is attached in the 2-position, R

4

in the 5-position and “P(═X)R

1

R

2

” in the 4-position; Q=Q

3

; R

4

=CH

3

, R

23

=cyclopropyl and R

24

=H), in particular to the compounds I2c2.n, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I2c3 (≡I where X=O; R

3

is attached in the 2-position, R

4

in the 5-position and “P(═X)R

1

R

2

” in the 2-position; Q=Q

3

; R

4

=Cl, R

23

=cyclopropyl and R

24

=H), in particular to the compounds I2c3.n, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I2c4 (≡I where X=O; R

3

is attached in the 2-position, R

4

in the 5-position and “P(═X)R

1

R

2

” in the 4-position; Q=Q

3

; R

4

=Br, R

23

=cyclopropyl and R

24

=H), in particular to the compounds I2c4, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I1d1 (≡I where X=O; R

3

is attached in the 4-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

4

; 1=0; R

25

=cyclopropyl), in particular to the compounds I1d1.n, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I1d2 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

4

; R

4

=CH

3

, R

25

=cyclopropyl), in particular to the compounds I1d2.n, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I1d3 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

4

; R

4

=Cl, R

25

=cyclopropyl), in particular to the compounds I1d3.n, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I1d4 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

4

; R

4

=Br, R

25

=cyclopropyl), in particular to the compounds I1d4, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I2d1 (≡I where X=O; R

3

is attached in the 2-position and “P(═X)R

1

R

2

” is attached in the 4-position; Q=Q

4

; 1=0; R

25

=cyclopropyl), in particular to the compounds I2d1.n, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I2d2 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

4

; R

4

=CH

3

, R

25

=cyclopropyl), in particular to the compounds I2a2.n, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I2d3 (≡I where X=O; R

3

is attached in the 2-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

4

; R

4

=Cl, R

25

=cyclopropyl), in particular to the compounds I2d3.n, where the variables R

1

to R

3

are as defined in Table 2.

Extraordinary preference is also given to the compounds I2d4 (≡I where X=O; R

3

is attached in the 4-position, R

4

is attached in the 5-position and “P(═X)R

1

R

2

” is attached in the 2-position; Q=Q

4

; R

4

=Br, R

25

=cyclopropyl), in particular to the compounds I2d4, where the variables R

1

to R

3

are as defined in Table 2.

The phosphorus-containing benzoyl derivatives of the formula I can be obtained by different routes, for example by the following processes:

A. Preparation of compounds of the formula Ia where R

6

=halogen by reaction of compounds of the formula Ia (≡I where Q=Q

1

) where R

6

=hydroxyl with halogenating agents:

Suitable halogenating agents are, for example, phosgene, diphosgene, triphosgene, thionyl chloride, oxalyl chloride, phosphorus oxychloride, phosphorus pentachloride, mesyl chloride, chloromethylene-N,N-dimethylammonium chloride, oxalyl bromide, phosphorus oxybromide, etc.

The starting materials are generally employed in equimolar amounts. However, it may also be advantageous to employ an excess of one or the other component.

Suitable solvents are, for example, chlorinated hydrocarbons, such as methylene chloride or 1,2-dichloroethane, aromatic hydrocarbons, for example toluene, xylene or chlorobenzene, polar aprotic solvents, such as acetonitrile, dimethylformamide or dimethyl sulfoxide, or mixtures of these. However, it is also possible to carry out the reaction without a solvent.

In general, the reaction temperature is in the range from 0° C. to the boiling point of the reaction mixture.

Work-up can be carried out in a manner known per se to afford the product.

B. Preparation of compounds of the formula Ia (≡I where Q=Q

1

) where R

6

=OR

13

, OSO

2

R

14

, OPR

15

R

16

, OPOR

15

R

16

or OPSR

15

R

16

by reaction of compounds of the formula Ia (≡I where Q=Q

1

) where R

6

=hydroxyl with alkylating, sulfonylating or phosphonylating agents IIα, IIβ, IIγ, IIδ or IIε.

L

1

is a nucleophilically replaceable leaving group, such as halogen, for example chlorine or bromine, hetaryl, for example imidazolyl, carboxylate, for example acetate, or sulfonate, for example mesylate or triflate, etc.

The compounds of the formula IIα, IIβ, IIγ, IIδ or IIε can be employed directly, such as in the case of the carbonyl halides, or generated in situ, for example activated carboxylic acids (using carboxylic acid and dicyclohexylcarbodiimide, etc.).

The starting materials are generally employed in equimolar amounts. However, it may also be advantageous to employ an excess of one or the other component.

If appropriate, it may also be advantageous to carry out the reaction in the presence of a base. The reactants and the base are advantageously employed in equimolar amounts. In certain cases, an excess of base of, for example, 1.5 to 3 molar equivalents may be advantageous.

Suitable bases are tertiary alkylamines, such as triethylamine, aromatic amines, such as pyridine, alkali metal carbonates, for example sodium carbonate or potassium carbonate, alkali metal bicarbonates, such as sodium bicarbonate and potassium bicarbonate, alkali metal alkoxides, such as sodium methoxide, sodium ethoxide, potassium tert-butoxide, or alkali metal hydrides, for example sodium hydride. Preference is given to using triethylamine or pyridine.

Suitable solvents are, for example, chlorinated hydrocarbons, such as methylene chloride or 1,2-dichloroethane, aromatic hydrocarbons, for example toluene, xylene or chlorobenzene, ethers, such as diethyl ether, methyl tert-butyl ether, tetrahydrofuran or dioxane, polar aprotic solvents, such as acetonitrile, dimethylformamide or dimethyl sulfoxide, or esters, such as ethyl acetate, or mixtures of these.

The reaction temperature is generally in the range from 0° C. to the boiling point of the reaction mixture.

Work-up can be carried out in a manner known per se to afford the product.

C. Preparation of compounds of the formula Ia (≡I where Q=Q

1

) where R

6

=OR

13

, SR

13

, POR

15

R

16

, NR

17

R

18

, ONR

18

R

19

, N-bonded heterocyclyl or O-(N-bonded heterocyclyl) by reaction of compounds of the formula Ia (≡I where Q=Q

1

) where R

6

=halogen, OSO

2

R

14

with compounds of the formula IIIα, IIIβ, IIIγ, IIIδ, IIIε, IIIη or IIIΘ, if appropriate in the presence of a base or with prior salt formation.

The starting materials are employed in equimolar amounts. However, it may also be advantageous to employ an excess of one or the other component.

If appropriate, it may also be advantageous to carry out the reaction in the presence of a base. The reactants and the base are advantageously employed in equimolar amounts. An excess of base of, for example, from 1.5 to 3 molar equivalents, based on Ia (≡I where Q=Q

1

) where R

6

=halogen, OSO

2

R

14

, may be advantageous in certain cases.

Suitable bases are tertiary alkylamines, such as triethylamine, aromatic amines, such as pyridine, alkali metal carbonates, for example sodium carbonate or potassium carbonate, alkali metal bicarbonates, such as sodium bicarbonate and potassium bicarbonate, alkali metal alkoxides, such as sodium methoxide, sodium ethoxide, potassium tert-butoxide, or alkali metal hydrides, for example sodium hydride. Preference is given to using sodium hydride or potassium tert-butoxide.

Suitable solvents are, for example, chlorinated hydrocarbons, such as methylene chloride or 1,2-dichloroethane, aromatic hydrocarbons, for example toluene, xylene or chlorobenzene, ethers, such as diethyl ether, methyl tert-butyl ether, tetrahydrofuran or dioxane, polar aprotic solvents, such as acetonitrile, dimethylformamide or dimethyl sulfoxide, or mixtures of these.

In general, the reaction temperature is in the range from 0° C. to the boiling point of the reaction mixture.

Work-up can be carried out in a manner known per se to afford the product.

D. Preparation of compounds of the formula Ia (≡I where Q=Q

1

) where R

6

=SOR

14

, SO

2

R

14

by reaction of compounds of the formula Ia (≡I where Q=Q

1

) where R

6

=SR

14

with an oxidizing agent.

Suitable oxidizing agents are, for example, m-chloroperbenzoic acid, peroxyacetic acid, trifluoroperoxyacetic acid, hydrogen peroxide, if appropriate in the presence of a catalyst, such as tungstate.

The starting materials are generally employed in equimolar amounts. However, it may also be advantageous to employ an excess of one or the other component.

Suitable solvents are, for example, chlorinated hydrocarbons, such as methylene chloride or 1,2-dichloroethane, aromatic hydrocarbons, for example toluene, xylene or chlorobenzene, ethers, such as diethyl ether, methyl tert-butyl ether, tetrahydrofuran or dioxane, polar aprotic solvents, such as acetonitrile or dimethylformamide, or esters, such as ethyl acetate, or mixtures of these.

In general, the reaction temperature is in the range from 0° C. to the boiling point of the reaction mixture.

Work-up can be carried out in a manner known per se to afford the product.

E. Preparation of compounds of the formula Ia (≡I where Q=Q

1

) where R

6

=OH by reaction of an activated phosphorus-containing benzoic acid of the formula IVα or a phosphorus-containing benzoic acid IVβ, which is preferably activated in situ, with a cyclohexanedione of the formula V to give the acylation product, followed by rearrangement.

L

2

is a nucleophilically replaceable leaving group, such as halogen, for example bromine or chlorine, hetaryl, for example imidazolyl or pyridyl, carboxylate, for example acetate or trifluoroacetate, etc.

The activated benzoic acid IV can be employed directly, such as in the case of the benzoyl halides, or generated in situ, for example using dicyclohexylcarbodiimide, triphenylphosphine/azodicarboxylic acid ester, 2-pyridine disulfide/triphenylphosphine, carbonyldiimidazole, etc.

If appropriate, it may be advantageous to carry out the acylation reaction in the presence of a base. The reactants and the auxiliary base are advantageously employed in equimolar amounts. A slight excess of auxiliary base, for example from 1. to 1.5 molar equivalents, based on IVα or IVβ, may be advantageous in certain cases.

Suitable auxiliary bases are tertiary alkylamines, pyridine or alkali metal carbonates. Suitable solvents are, for example, chlorinated hydrocarbons, such as methylene chloride or 1,2-dichloroethane, aromatic hydrocarbons, such as toluene, xylene or chlorobenzene, ethers, such as diethyl ether, methyl tert-butyl ether, tetrahydrofuran or dioxane, polar aprotic solvents, such as acetonitrile, dimethylformamide or dimethyl sulfoxide, or esters, such as ethyl acetate, or mixtures of these.

If the activated carboxylic acid component used is a phosphorus-containing benzoyl halide, it may be advantageous to cool the reaction mixture to 0-10° C. when adding this reaction partner. The mixture is subsequently stirred at 20-100° C., preferably at 25-50° C., until the reaction has gone to completion. Work-up is carried out in a customary manner, for example by pouring the reaction mixture into water and extracting the product of value. Solvents which are suitable for this purpose are, in particular, methylene chloride, diethyl ether and ethyl acetate. The organic phase is dried and the solvent is removed, and the crude ester can then be employed for the rearrangement without further purification.

The rearrangement of the esters VI to the compounds of the formula Ia is advantageously carried out at 20-100° C. in a solvent and in the presence of a base and, if appropriate, using a cyano compound as catalyst.

Suitable solvents are, for example, acetonitrile, methylene chloride, 1,2-dichloroethane, dioxane, ethyl acetate, toluene or mixtures of these. Preferred solvents are acetonitrile and dioxane.

Suitable bases are tertiary amines, such as triethylamine, aromatic amines, such as pyridine, or alkali metal carbonates, such as sodium carbonate or potassium carbonate, which are preferably employed in equimolar amounts or in up to four-fold excess, based on the ester. Preference is given to using triethylamine or alkali metal carbonate, preferably in twice the equimolar amount, based on the ester.

Suitable cyano compounds are inorganic cyanides, such as sodium cyanide or potassium cyanide, and organic cyano compounds, such as acetone cyanohydrin or trimethylsilyl cyanide. They are employed in an amount of from 1 to 50 mol percent, based on the ester. Preference is given to using acetone cyanohydrin or trimethylsilyl cyanide, for example in an amount of from 5 to 15, preferably 10, mol percent, based on the ester.

Work-up can be carried out in a manner known per se. The reaction mixture is, for example, acidified with dilute mineral acid, such as 5% strength hydrochloric acid or sulfuric acid, and extracted with an organic solvent, for example methylene chloride or ethyl acetate. The organic extract can be extracted with 5-10% strength alkali metal carbonate solution, for example sodium carbonate or potassium carbonate solution. The aqueous phase is acidified and the resulting precipitate is filtered off with suction and/or the mixture is extracted with methylene chloride or ethyl acetate and the extract is dried and concentrated.

F. Preparation of compounds of the formula Ib (≡I where Q=Q

2

) where R

20

=halogen by reaction of compounds of the formula Ib (≡I where Q=Q

2

) where R

20

=hydroxyl with halogenating agents:

What has been said in section A applies analogously.

G. Preparation of compounds of the formula Ib (≡I where Q=Q

2

) where R

20

=OR

13

, OSO

2

R

14

, OPR

15

R

16

, OPOR

15

R

16

or OPSR

15

R

16

by reaction of compounds of the formula Ib (≡I where Q=Q

2

) where R

6

=hydroxyl with alkylating, sulfonylating or phosphonylating agents IIα, IIβ, IIγ, IIδ or IIε.

What has been said in section B applies analogously.

H. Preparation of compounds of the formula Ib (≡I where Q=Q

2

) where R

6

=OR

13

, SR

13

, POR

15

R

16

, NR

17

R

18

, ONR

18

R

19

, N-bonded heterocyclyl or O—(N-bonded heterocyclyl) by reaction of compounds of the formula Ib (≡I where Q=Q

2

) where R

20

=halogen, OSO

2

R

14

with compounds of the formula IIIα, IIIβ, IIIγ, IIIδ, IIIε, IIIη or IIIΘ, if appropriate in the presence of a base or with prior salt formation.

What has been said in section C applies analogously.

I. Preparation of compounds of the formula Ib (≡I where Q=Q

2

) where R

20

=SOR

14

, SO

2

R

14

by reaction of compounds of the formula Ib (≡I where Q=Q

2

) where R

20

=SR

14

with an oxidizing agent.

What has been said in section D applies analogously.

K. Preparation of compounds of the formula Ib (≡I where Q=Q

2

) where R

20

≠hydroxyl by reaction of a metallated pyrazole derivative of the formula VII with a phosphorus-containing benzoic acid derivative of the formula VIγ:

M is a metal, in particular an alkali metal, such as lithium or sodium, an alkaline earth metal, such as magnesium, or a transition metal, such as palladium, nickel, etc., and L

3

is a nucleophilically replaceable leaving group, such as halogen, for example chlorine or bromine, alkylsulfonate, such as mesylate, haloalkylsulfonate, such as triflate, or cyanide.

The reaction is generally carried out at temperatures from −100° C. to the reflux temperature of the reaction mixture. Suitable solvents are inert aprotic solvents, such as ethers, such as diethyl ether, tetrahydrofuran. The compounds of the formula Ivγ are generally employed in excess; however, it may also be advantageous to employ them in equimolar amounts or substoichiometric amounts. Work-up is carried out to afford the product.

The metallated pyrazole derivatives of the formula VII can be generated in a manner known per se by reacting pyrazoles halogenated in the 4-position with metals such as lithium, sodium, magnesium etc., or with organometallic compounds, for example butyllithium. However, it is also possible to metallate pyrazoles which are linked to hydrogen in the 4-position directly, for example using the abovementioned metals or organometallic compounds. The reactions are generally carried out in an inert aprotic solvent, preferably in ether, such as diethyl ether, tetrahydrofuran, etc. The reaction temperature is in the range from −100° C. to the boiling point of the reaction mixture. The compounds of the formula VII are generally directly reacted further or generated in situ.

L. Preparation of compounds of the formula Ib (≡I where Q=Q

2

) where R

20

=hydroxyl by reaction of an activated phosphorus-containing benzoic acid of the formula IVα or a phosphorus-containing benzoic acid IVβ, which is preferably activated in situ, with a pyrazole of the formula VIII to give the acylating product, followed by rearrangement.

What has been said in section E applies analogously.

However, it is also possible to generate the ester IX in situ by reacting a pyrazole of the formula VIII, or an alkali metal salt thereof, with a phosphorus-containing benzene derivative of the formula X in the presence of carbon monoxide, a catalyst and a base.

L

4

is a leaving group, such as halogen, for example chlorine, bromine or iodine, or sulfonate, such as mesylate or triflate; preference is given to bromine or triflate.

If appropriate, the ester IX reacts directly to give the phosphorus-containing benzoyl derivative of the formula Ib.

Suitable catalysts are palladium-ligand complexes in which the palladium is present in oxidation state 0, metallic palladium, which has optionally been absorbed on a carrier, and preferably palladium(II) salts. The reaction with palladium(II) salts and metallic palladium is preferably carried out in the presence of complex ligands.

An example of a suitable palladium(0)-ligand complex is tetrakis(triphenylphosphine)palladium.

Metallic palladium is preferably absorbed on an inert carrier such as, for example, active carbon, silica, alumina, barium sulfate or calcium carbonate. The reaction is preferably carried out in the presence of complex ligands such as, for example, triphenylphosphine.

Examples of suitable palladium(II) salts are palladium acetate and palladium chloride. The presence of complex ligands such as, for example, triphenylphosphine is preferred.

Suitable complex ligands for the palladium-ligand complexes, or in whose presence the reaction is preferably carried out with metallic palladium or palladium(II) salts, are tertiary phosphines whose structure is represented by the following formulae:

where z is from 1 to 4 and the radicals R

a

to R

g

are C

1

-C

6

-alkyl, aryl-C

1

-C

2

-alkyl or preferably aryl. Aryl is, for example, naphthyl and unsubstituted or substituted phenyl, such as, for example, 2-tolyl and, in particular, unsubstituted phenyl.

The complex palladium salts can be prepared in a manner known per se starting from commercially obtainable palladium salts such as palladium chloride or palladium acetate and the appropriate phosphines, such as, for example, triphenylphosphine or 1,2-bis(diphenylphosphino)ethane. Many of the complex palladium salts are commercially available. Preferred palladium salts are [(R)(+)-2,2′-bis(diphenylphosphino)-1,1′-binaphthyl]palladium(II) chloride, bis(triphenylphosphine)palladium(II) acetate and, in particular, bis(triphenylphosphine)palladium(II) chloride.

The palladium catalyst is generally employed in a concentration of from 0.05 to 5 mol %, and preferably 1-3 mol %.

Suitable bases are tertiary amines, such as, for example, N-methylpiperidine, ethyldiisopropylamine, 1,8-bisdimethylaminonaphthalene or, in particular, triethylamine. Also suitable are alkali metal carbonates, such as sodium carbonate or potassium carbonate. However, mixtures of potassium carbonate and triethylamine are also suitable.

In general, from 2 to 4 molar equivalents, in particular 2 molar equivalents, of the alkali metal carbonate and from 1 to 4 molar equivalents, in particular 2 molar equivalents, of the tertiary amine are employed, based on the phosphorus-containing benzene derivative of the formula X.

Suitable solvents are nitrites, such as benzonitrile and acetonitrile, amides, such as dimethylformamide, dimethylacetamide, tetra-C

1

-C

4

-alkylureas or N-methylpyrrolidone and, preferably, ethers such as tetrahydrofuran, methyl tert-butyl ether. Particularly preferred solvents are ethers such as 1,4-dioxane and dimethoxyethane.

M. Preparation of compounds of the formula Ic (≡I where Q=Q

3

) where R

24

=H by reaction of a 1,3-dicarbonyl compound of the formula XI with hydroxylamine.

L

5

is an O—C

1

-C

6

-alkyl or N(C

1

-C

6

-alkyl)

2

group. The 1,3-dicarbonyl compound of the formula XI is reacted with hydroxylamine which is generated in situ, for example from hydroxylamine salt using a base or an acid acceptor, such as triethylamine or sodium acetate.

The starting material of the formula XI is obtained by reacting the β-keto esters of the formula XII, which are known per se, with an activated phosphorus-containing benzoic acid IVα. The acylation product XIII is subsequently converted into the 1,3-diketone XIV using, for example, p-toluenesulfonic acid as catalyst in an inert solvent, such as toluene. The 1,3-diketone XIV is subsequently reacted with an orthoester or dimethylformamide dialkyl acetal to give the 1,3-dicarbonyl compound of the formula XI.

N. Preparation of compounds of the formula Ic (≡I where Q=Q

3

) by cycloaddition of the α,β-unsaturated benzoyl derivative XV with a nitrile oxide of the formula XVI

The α,β-unsaturated benzoyl derivative XV is obtained by ethynylation of the activated phosphorus-containing benzoic acid of the formula IVα.

Z is a metal such as lithium, an organotin radical such as Sn(C

4

H

9

)

3

or a zinc radical such as ZnCl or ZnBr.

O. Preparation of compounds of the formula Id (≡I where Q=Q

4

) by reaction of the cyanoketone XVII with an activated phosphorus-containing benzoic acid of the formula IVα in the presence of a base such as triethylamine, sodium carbonate, sodium hydride or magnesium ethoxide in an inert organic solvent such as diethyl ether, tetrahydrofuran, N,N-diethylformamide, dichloromethane or acetonitrile.

The phosphorus-containing benzoyl halides of the formula IVα where L

2

=halogen can be prepared in a manner known per se by reacting the benzoic acids of the formula IVβ with halogenating agents such as thionyl chloride, thionyl bromide, phosgene, diphosgene, triphosgene, oxalyl chloride, oxalyl bromide.

The phosphorus-containing benzoic acids of the formula IVβ can be prepared in a manner known per se by acidic or basic hydrolysis from the corresponding phosphorus-containing benzoic esters IVδ (cf. J. March, “Advanced Organic Chemistry”, 4

th

edition, Wiley, New York, p. 378 ff.)

where T is C

1

-C

6

-alkoxy.

The phosphorus-containing benzoic esters IVδ are obtainable by different routes:

They can be obtained by electrophilic or nucleophilic aromatic substitution of benzoic esters of the formula XVIII and, if appropriate, further functionalization of the group thus introduced.

For example, the ester of the formula XVIII can be nitrated analogously to known methods (R

3

=NO

2

; cf. J. March, “Advanced Organic Chemistry”, 4

th

edition, p. 522 ff.), brominated or chlorinated (R

3

=Cl, Br; cf. J. March, “Advanced Organic Chemistry”, 4

th

edition, p. 531 ff.).

The abovementioned electrophilic aromatic substitution reaction may result in mixtures of isomers, which can be separated or purified by distillation, crystallization or chromatographic methods.

Phosphorus-containing benzoic esters of the formula IVδ where R

3

=NH

2

can be obtained by reduction of the corresponding nitro compounds of the formula IVδ where R

3

=NO

2

.

Suitable reducing agents are, inter alia, metals such as iron or zinc in the presence of hydrochloric acid and catalytically activated hydrogen (cf. J. March, “Advanced Organic Chemistry”, 4

th

edition, p. 1216 ff.)

Phosphorus-containing benzoic esters of the formula IVδ where R

3

=(C

1

-C

6

-alkylsulfonyl)amino, (C

1

-C

6

-haloalkylsulfonyl)amino can be obtained by reaction of the corresponding amino compounds with appropriately substituted sulfonyl chlorides in the presence of a base (cf.

T. W. Green et al., “Protective Groups in Organic Synthesis”, p. 379 f.)

The latter can be converted into the corresponding N-alkyl derivatives by alkylation in the presence of a base.

Suitable bases are, inter alia, sodium hydride, potassium hydride, potassium tert-butoxide, and suitable alkyl halides are alkyl bromides and alkyl iodides (cf. J. P. Dunn et al., J. Med. Chem. 1981, 24, p. 1097).

Phosphorus-containing benzoic esters of the formula IVδ where R

3

=halogen, cyano, C

1

-C

6

-alkyl, C

1

-C

6

-alkylthio or C

1

-C

6

-haloalkylthio can be obtained from the corresponding amino compounds by Sandmeyer reaction or related reactions (cf. J. March, “Advanced Organic Chemistry”, 4

th

edition, pp. 723-724, pp. 669-671)

If appropriate, it may be advantageous to carry out the reactions in the presence of metal catalysts such as, for example, copper(I) or palladium(II) (cf., for example, Kikukawa et al., J. Org. Chem. 1983, 48, 1333).

Phosphorus-containing benzoic esters of the formula IVδ where R

3

=S(O)

1,2

—C

1

-C

6

-alkyl or S(O)

1,2

—C

1

-C

6

-haloalkyl can be obtained by reaction of the corresponding sulfur compounds with an oxidizing agent such as bromine, peroxyacetic acid, m-chloroperbenzoic acid and hydrogen peroxide, if appropriate in the presence of a catalyst such as tungstate.

Phosphorus-containing benzoic esters of the formula IVδ here R

3

=aminosulfonyl, C

1

-C

6

-alkylaminosulfonyl or di(C

1

-C

6

-alkyl)aminosulfonyl can be obtained by reaction of the corresponding sulfonyl chloride with ammonia or suitable amines. If appropriate, it may be useful to operate in the presence of a base such as triethylamine, sodium carbonate, potassium carbonate, sodium bicarbonate, potassium bicarbonate or pyridine (cf. J. March, “Advanced Organic Chemistry”, 4

th

edition, p. 499). The sulfonyl chloride is obtained by sulfochlorination of the corresponding diazonium salt.

Phosphorus-containing benzoic esters of the formula IVδ where R

3

=C

1

-C

6

-alkoxy or C

1

-C

6

-haloalkoxy can be obtained by alkylation of the corresponding phenols in the presence of a base. Suitable bases are, in addition to the customary bases, in particular sodium carbonate, potassium carbonate, sodium hydride or potassium tert-butoxide. Preferred alkylating agents are appropriate halogenated or non-halogenated alkyl bromides or chlorides (cf., for example, H. Fener et al., “The Chemistry of the Ether Linkage”, Wiley, New York, 1967, pp. 445-498.)

The phenols can be obtained by boiling down of corresponding diazonium compounds.

Phosphorus-containing benzoic esters of the formula IVδ where R

3

=PXR

1

R

2

can be obtained by reaction of compounds of the formula IVδ where R

3

=Br, I, OSO

2

CF

3

etc., with suitable phosphonous acids or phosphorous acids in the presence of a transition metal catalyst such as nickel or palladium and, if appropriate, of a base (cf., for example, T. Hirao et al., Synthesis 1981, 56).

Phosphorus-containing benzoic esters of the formula IVδ where R

3

=phenyl can be prepared by reaction of a corresponding bromide or iodide of the formula IVδ where R

3

=Br or I with a phenyl bromide or phenyl iodide, which may be substituted, in the presence of copper (cf. Ranta et al., Synthesis 1974, 9; Goshaer et al., Russ. Chem. Rev. 1972, 41, 1046)

Phosphorus-containing benzoic esters of the formula IVδ where R

3

=unsub. or sub. phenyl, unsub. or sub. heterocyclyl can be obtained by reaction of compounds of the formula IVδ where R

3

=a leaving group such as bromine, iodine, triflate, fluorosulfonyloxy, etc., with an unsub. or sub. phenyl or heterocyclyl stannane (Stille coupling), an unsub. or sub. phenyl or heterocyclyl boron compound (Suzuki coupling) or an unsub. or sub. phenyl or heterocyclyl zinc compound (Negishi coupling) in a manner known per se (cf. Tetrahedron Lett. 1986, 27, 5265) in the presence of a palladium or nickel catalyst and, if appropriate, a base.

Ar′=unsub. or sub. phenyl or heterocyclyl

Met=Sn(C

1

-C

4

-alkyl)

3

, B(OH)

2

, ZnBr, ZnCl

Phosphorus-containing benzoic esters of the formula IVδ where R

3

=unsub. or sub. heterocyclyl can also be obtained by constructing the heterocycle from suitable precursors.

1,2,4-Oxadiazoline derivatives, for example, can be prepared from aldoximes of the formula XIX by condensation with aldehydes of the ketones (cf., for example, Arch. Pharm. 1993, 326, 383-389).

The thioamides of the formula XX are suitable precursors for 2-thiazolinyl derivatives (cf., for example, Tetrahedron 1986, 42, 1449-1460) and for 2-thiazolyl derivatives (cf., for example, Houben-Weyl, “Methoden der organischen Chemie”[Methods of Organic Chemistry], 4

th

edition, Vol. E5, p. 1268 ff. (1985)).

2-Oxazolinyl, 2-thiazolinyl and 2-imidazolinyl derivatives are obtainable from the carboxylic acids of the formula XXI (cf., for example, Tetrahedron Lett. 1981, 22, 4471-4474).

According to processes known from the literature, it is possible to prepare 1,3-thiazole-5(4H)-thion-2-yl or 5-oxo-2-imidazolin-2-yl derivatives from carbonyl halides of the formula XXII where Hal is halogen, in particular from carbonyl chlorides (cf., for example, Helv. Chim. Acta, 1986, 69, 374-388; Heterocycles 1989, 29, 1185-1189).

Furthermore, it is possible to prepare 2-oxazolyl derivatives from the carboxylic acids of the formula XXI or the carbonyl halides of the formula XXII (cf., for example, Heterocyclic Chem. 1991, 28, 17-28).

The conversion of oximes of the formula XXIV into 4,5-dihydroisoxazol-3-yl or isoxazol-3-yl derivatives can be carried out in a manner known per se via the intermediate of the hydroxamoyl chlorides or bromides. Using the latter, nitrile oxides are generated in situ which react with alkenes or alkynes to give the desired products (cf., for example, Chem. Ber. 1973, 106, 3258-3274). 1,3-Dipolar cycloaddition with chlorosulfonyl isocyanate to the nitrile oxide formed in situ affords 1,2,4-oxadiazolin-5-on-3-yl derivatives (cf., for example, Heterocycles 1988, 27, 683-685).

The aldehydes of the formula XXV can be converted into 2,4-dihydro-1,2,4-triazol-3-on-5-yl derivatives via the intermediate of the semicarbazones (cf., for example, J. Heterocyclic Chem. 1986, 23, 881-883).

2-Imidazolinyl derivatives are preparable from benzonitriles of the formula XXVI by known methods (cf., for example, J. Org. Chem. 1987, 52, 1017-1021).

It is also possible to prepare 1,2,4-triazol-3-yl derivatives by known processes from the benzonitriles of the formula XXVI (cf., for example, J. Chem. Soc. 1954, 3461-3464).

The aldehydes XXV can be reacted in a manner known per se by Wittig reaction with phosphonium salts (Ph)

3

P

+

CH

2

COR*X

−

(J. March, “Advanced Organic Chemistry”, 3

rd

edition, p. 864 ff., Wiley-Interscience Publication, 1985) to give α,β-unsaturated ketones XXVII. By reaction with hydroxylamine, these give the corresponding oximes which can be converted into the 5-isoxazolyl derivatives by oxidative cyclization (J. Am. Chem. Soc. 1972, 94, 9128) (the meaning of R* thus corresponds to the meaning of a radical by which the heterocyclyl may be substituted).

It is also possible to convert the aldehydes XXV with alkoxymethylphosphonium salts in a manner known per se (J. March, “Advanced Organic Chemistry”, 3

rd

edition, p. 864 ff., Wiley-Interscience Publication, 1985) into the corresponding enol ethers. Cleavage of these enol ethers analogously to processes known from the literature yield the acetaldehyde derivatives XXVIII. By bromination in the α-position these can be converted into the α-bromoacetaldehyde derivatives (Tetrahedron Lett. 1988, 29, 5893), which afford, by cyclization with amides, thioamides and amidines, oxazoles, thiazoles and imidazoles. Furthermore, the acetaldehyde derivatives XXVIII can be converted with dimethylformamide dimethyl acetal into corresponding enamines which can then be converted into isoxazoles or pyrazoles using hydroxylamines and hydrazines, respectively.

Furthermore, the aldehydes XXV can be converted into hydroxyketone derivatives by Aldol reaction with ketones. Subsequent oxidation leads to 1,3-diketones which can be converted into isoxazoles, pyrazoles or pyrimidines using hydroxylamine, hydrazines or amidines.

The aldehydes XXV can also be converted by methods known from the literature (Houben-Weyl, “Methoden der organischen Chemie”[Methods of Organic Chemistry], 4

th

edition, Vol. E14b) into the corresponding diazo compounds XXIX. 1,3-dipolar cycloaddition to alkenes or alkynes and subsequent isomerization leads to pyrazolines or pyrazoles.

The aldehyde XXV can be prepared analogously to processes known from the literature, for example from the corresponding methyl compound XXX, by bromination, for example with N-bromosuccinimide or 1,3-dibromo-5,5-dimethylhydantoin, and subsequent oxidation (cf. Synth. Commun. 1992, 22, 1967-1971).

The oximes of the formula XXIV are advantageously obtained by reacting, in a manner known per se, aldehydes of the formula XXV with hydroxylamine (cf. J. March, “Advanced Organic Chemistry”, 3

rd

edition, pp. 805-806, Wiley, New York, 1985).

The conversion of the oximes XXIV into the nitrites XXVI can also be carried out by processes known per se (cf. J. March, “Advanced Organic Chemistry”, 3

rd

edition, pp. 931-932, Wiley, New York, 1985).

The nitrites of the formula XXVI can be converted in a manner known per se with hydroxylamine into the corresponding aldoximes XIX, converted with hydrogen sulfide into the thioamides XX or hydrolyzed to give the carboxylic acids XXI. The latter can also be obtained from the aldehydes XXV by oxidation (cf. J. March, “Advanced Organic Chemistry”, 3

rd

edition, p. 629 ff., Wiley, New York, 1985).

The acyl halides XXII can be obtained analogously to standard processes from the corresponding carboxylic acids of the formula XXI.

The phosphorus-containing compounds of the formula IVδ are obtainable by reaction of compounds of the formula XXXII where L

5

=bromine, iodine, triflate and a corresponding substituted phosphorous acid or phosphonous acid in the presence of a transition metal catalyst, such as nickel or palladium, and, if appropriate, a base (cf., for example, T. Hirao et al., Synthesis 1981, 56.)

The compounds of the formula XXXII where L

5

=Br, I are obtained from the corresponding nitro compounds by reaction of the nitro group and subsequent Sandmeyer reaction. The compounds of the formula XXXII where L

5

=OSO

2

CF

3

can be obtained by reacting the corresponding phenol with trifluoromethylsulfonyl chloride or trifluoromethylsulfonic anhydride.

The compounds of the formula IVδ where R

1

, R

2

=C

1

-C

6

-alkoxy, C

1

-C

6

-alkylthio, C

1

-C

6

-alkylamino etc., can also be obtained by reaction of nucleophilically substitutable phosphorus compounds of the formula IVδ where L′, L″=a leaving group, such as halogen, C

1

-C

6

-alkoxy, etc., with suitable alcohols, amines or mercaptans, if appropriate in the presence of a base, (cf., for example, L. J. Kaplan, J.Org. Chem. 1979, 44, 2226; Houben-Weyl, “Methoden der organischen Chemie”[Methods of Organic Chemistry], Vol. XII/1, p. 423 ff.; R. Z. Greenley et al., J. Org. Chem. 1964, 29, 1009).

Compounds of the formula IVδ where L′, L″=halogen can be obtained by reaction of compounds of the formula IVδ where R

1

, R

2

=OCH

3

with halogenating agents (cf. z. B. W. Althoff et al., Chem. Ber. 1978, 111, 1845).

Suitable halogenating agents are, inter alia, phosgene, thionyl chloride and thionyl bromide.

Compounds of the formula IVβ are furthermore obtainable by oxidation of compounds of the formula XXXIII.

Suitable oxidizing agents are, for example, potassium permanganate (cf., for example, Houben Weyl, “Methoden der Organischen Chemie”[Methods of Organic Chemistry], Vol. IV/1a, 1981, and Vol. VIII, 1952; E. I. Bengtsson, Acta Chem. Scand. 1953, 7, 774), chromium(VI) compounds (cf., for example, A. W. Singer et al., Org. Synth. Coll. Vol. III 1955, 740) or atmospheric oxygen in the presence of a catalyst such as, for example, cobalt or manganese (cf., for example, A. S. Hay et al., Can. J. Chem. 1965, 43, 1306).

The compounds of the formula XXXIII are obtainable by reaction of organometallic compounds of the formula XXXIV (where Met′=Li, Mg) with phosphorus compounds carrying nucleophilically replaceable groups (L=halogen, such as Cl, Br, alkoxy, etc.) (cf., for example, A. Berger et al., J. Org. Chem. 1951, 16, 1250; M. Sander, Chem. Ber. 1960, 93, 1220).

These compounds can also be obtained by oxidation of the corresponding phosphorus(III) compounds, which can be prepared analogously to the reaction shown above.

Suitable oxidizing agents are, for example, hydrogen peroxide, peroxyacetic acid, etc.

The compounds of the formula XXXIII (where R

2

=C

1

-C

6

-alkoxy, C

1

-C

6

-alkyl, C

2

-C

6

-alkenyl, C

2

-C

6

-alkynyl, etc.) can furthermore be obtained by reacting a phosphorus compound of the formula XXXV with an alkyl halide (Arbuzov reaction).

Preferred alkyl halides are the corresponding bromides and iodides (cf., for example, B. A. Arbuzov, Pure Appl. Chem. 1964, 9, 307; G. M. Kosolapoff, Org. React. 1951, 6, 273).

In general, it is possible to introduce or synthesize the radical R

3

at a suitable stage of the reaction sequence of the preparation of compounds of the formula I, where these reactions are described above or can be prepared analogously to known processes.

It may also be feasible to change the order of the reaction steps.

Furthermore, it is possible to modify the substituents R

1

and R

2

at a suitable stage of the reaction sequence. For example, the radicals R

1

, R

2

=C

1

-C

6

-alkoxy can be converted by reaction with organometallic compounds into R

1

, R

2

=C

1

-C

6

-alkyl, C

2

-C

6

-alkenyl, C

2

-C

6

-alkynyl etc. Organometallic reagents which are suitable for this purpose are appropriate organolithium or organomagnesium compounds (cf., for example, Houben-Weyl, “Methoden der Organischen Chemie”[Methods of Organic Chemistry], Vol. E. 2, p. 38 ff., Wiley, New York).

Novel are the phosphorus-containing benzoic acid derivatives of the formula IV

where:

X is oxygen or sulfur;

R

1

,R

2

are hydrogen, C

1

-C

6

-alkyl, C

2

-C

6

-alkenyl, C

2

-C

6

-alkynyl, C

1

-C

6

-alkoxy, C

3

-C

6

-alkenyloxy, C

3

-C

6

-alkynyloxy, mercapto, C

1

-C

6

-alkylthio, C

3

-C

6

-alkenylthio, C

3

-C

6

-alkynylthio, amino, C

1

-C

6

-alkylamino, di(C

1

-C

6

-alkyl)amino, (C

1

-C

6

-alkoxy)(C

1

-C

6

-alkyl)amino, (C

3

-C

6

-alkenyl)(C

1

-C

6

-alkyl)amino, (C

3

-C

6

-alkynyl)(C

1

-C

6

-alkyl)amino, di(C

3

-C

6

-alkenyl)amino or di(C

3

-C

6

-alkynyl)amino, where the abovementioned alkyl, alkenyl or alkynyl radicals may be partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio, C

1

-C

4

-alkylsulfinyl, C

1

-C

4

-alkylsulfonyl, di(C

1

-C

4

-alkyl)amino, C

1

-C

4

-alkylcarbonyl, C

1

-C

4

-alkoxycarbonyl,

are phenyl or heterocyclyl, where the two last-mentioned radicals for their part may be partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl;

are phenoxy which may by partially or fully halogenated and/or may carry one to three of the following groups: nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl; or

R

1

and R

2

together form a —O—(CH

2

)

m

—O—, —O—(CH

2

)

m

—S—, —S—(CH

2

)

m

—S—, —NR

5

—(CH

2

)

m

—NR

5

—, —O—(CH

2

)

m

—NR

5

—, —S—(CH

2

)

m

—NR

5

—, —(CH

2

)

n

—O—, —(CH

2

)

n

—S— or —(CH

2

)

n

—NR

5

chain which may carry one to three radicals from the following group:

halogen, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

l

-C

4

-alkoxy, C

1

-C

4

-alkoxycarbonyl or phenyl which is unsubstituted or partially or fully halogenated and/or may carry one to three of the following groups: nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl; or

R

1

and R

2

together form —(CH

2

)

p

chain which may be interrupted by oxygen, sulfur or NR

5

and/or may carry one to three radicals from the following group:

halogen, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-alkoxycarbonyl or phenyl which is unsubstituted or partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl;

R

3

is cyano, halogen, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, C

1

-C

6

-alkoxy-C

1

-C

6

-alkyl, C

1

-C

6

-haloalkoxy-C

1

-C

6

-alkyl, C

1

-C

6

-alkylthio-C

1

-C

6

-alkyl, C

1

-C

6

-alkylsulfinyl-C

1

-C

6

-alkyl, C

1

-C

6

-alkylsulfonyl-C

1

-C

6

-alkyl, C

1

-C

6

-alkylcarbonyl, C

1

-C

6

-alkoxy, C

1

-C

6

-haloalkoxy, C

1

-C

6

-alkylthio, C

1

-C

6

-haloalkylthio, C

1

-C

6

-alkylsulfinyl, C

1

-C

6

-haloalkylsulfinyl, C

1

-C

6

-alkylsulfonyl, C

1

-C

6

-haloalkylsulfonyl, aminosulfonyl, C

1

-C

6

-alkylaminosulfonyl, di(C

1

-C

6

-alkyl)aminosulfonyl, (C

1

-C

6

-alkylsulfonyl)amino, (C

1

-C

6

-haloalkylsulfonyl)amino, N—(C

1

-C

6

-alkyl)—N—(C

1

-C

6

-alkylsulfonyl)amino, N—(C

1

-C

6

-alkyl)—N—(C

1

-C

6

-haloalkylsulfonyl)amino, —P(═X)R

1

R

2

, phenyl or heterocyclyl, where the two last-mentioned radicals may be partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl;

R

4

is nitro, cyano, halogen, C

1

-C

6

-alkyl, C

1

-C

6

-alkoxy, C

1

-C

6

-alkylthio, C

1

-C

6

-alkylsulfinyl or C

1

-C

6

-alkylsulfonyl;

R

5

is hydrogen, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl or C

1

-C

6

-alkoxy;

l is 0, 1 or 2;

m is 2, 3 or 4;

n is 3, 4 or 5;

p is 4, 5 or 6;

R

26

is a radical which can be removed by hydrolysis.

Examples of radicals which can be removed by hydrolysis are alkoxy, phenoxy, alkylthio and phenylthio radicals, which may be unsubstituted or substituted; halides, heteroaryl radicals attached via nitrogen; amino and imino radicals which may be unsubstituted or substituted, etc.

Preference is given to phosphorus-containing benzoic acid derivatives of the formula IVα where L

2

=halogen (≡IV where R

26

=halogen),

where the variables X, R

1

to R

4

and l are as defined under the compounds of the formula IV. Hal is halogen, in particular chlorine or bromine.

Preference is also given to the phosphorus-containing benzoic derivatives of the formula IVβ (≡IV where R

26

=hydroxyl),

where the variables X, R

1

to R

4

and l are as defined under the compounds of the formula IV.

Preference is also given to the phosphorus-containing benzoic acid derivatives of the formula IVδ (≡IV where R

26

=C

1

-C

6

-alkoxy),

where the variables X, R

1

to R

4

and l are as defined under the compounds of the formula IV and

T is C

1

-C

6

-alkoxy.

The particularly preferred embodiments of the phosphorus-containing benzoic acid derivatives of the formulae IV, IVα where L

2

=halogen, IVβ and IVδ with respect to the variables X, R

1

to R

4

and 1 correspond to those of the phosphorus-containing benzoyl derivatives of the formula I.

Particular preference is also given to the compounds of the formula IV where the variables have the following meanings:

R

1

,R

2

are hydrogen, C

1

-C

6

-alkyl, C

2

-C

6

-alkenyl, C

2

-C

6

-alkynyl, C

1

-C

6

-alkoxy, C

3

-C

6

-alkenyloxy, C

3

-C

6

-alkynyloxy, mercapto, C

1

-C

6

-alkylthio, C

3

-C

6

-alkenylthio, C

3

-C

6

-alkynylthio, amino, C

1

-C

6

-alkylamino or di-(C

1

-C

6

-alkyl)amino, where the alkyl, alkenyl or alkynyl radicals mentioned may be partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio, C

1

-C

4

-alkylsulfonyl, di(C

1

-C

4

-alkyl)-amino, C

1

-C

4

-alkylcarbonyl, C

1

-C

4

-alkoxycarbonyl, phenyl or heterocyclyl, where the two lastmentioned radicals for their part may be partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

—C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl;

are phenoxy which may be partially or fully halogenated and/or may carry one to three of the following groups: nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl; or

R

1

and R

2

together form a —O—(CH

2

)

m

—O—, —O—(CH

2

)

m

—S—, —S—(CH

2

)

m

—S—, —NR

5

—(CH

2

)

m

—NR

5

—, —O—(CH

2

)

m

—NR

5

— or —S—(CH

2

)

m

—NR

5

— chain which may carry one to three radicals from the following group:

halogen, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-alkoxycarbonyl or phenyl, which is unsubstituted or partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

—C

4

-alkyl, C

1

—C

4

-haloalkyl, C

1

—C

4

-alkoxy, C

1

—C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl;

R

3

is cyano, halogen, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, C

1

-C

6

-alkylcarbonyl, C

1

-C

6

-alkoxy, C

1

-C

6

-haloalkoxy, C

1

-C

6

-alkylthio, C

1

-C

6

-haloalkylthio, C

1

-C

6

-alkylsulfinyl, C

1

-C

6

-haloalkylsulfinyl, C

1

-C

6

-alkylsulfonyl, C

1

-C

6

-haloalkylsulfonyl, —P(═X)R

1

R

2

, phenyl or heterocyclyl, where the two lastmentioned radicals may be partially or fully halogenated and/or may carry one to three of the following groups:

nitro, cyano, C

1

-C

4

-alkyl, C

1

-C

4

-haloalkyl, C

1

-C

4

-alkoxy, C

1

-C

4

-haloalkoxy or C

1

-C

4

-alkoxycarbonyl;

R

4

is nitro, cyano, halogen, C

1

-C

6

-alkyl, C

1

-C

6

-alkoxy, C

1

-C

6

-alkylthio, C

1

-C

6

-alkylsulfinyl or C

1

-C

6

-alkylsulfonyl;

R

5

is hydrogen, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl or C

1

-C

6

-alkoxy;

l is 0, 1 or 2;

m is 2, 3 or 4;

R

26

is a radical which can be removed by hydrolysis.

Especially preferred are the compounds of the formula IV where the variables have the following meanings:

R

1

, R

2

are hydrogen, C

1

-C

6

-alkyl, C

1

-C

6

-alkoxy or C

1

-C

6

-alkylthio, where the alkyl radicals mentioned may be partially or fully halogenated and/or may carry one to three of the following groups: nitro, cyano, C

1

-C

4

-alkoxy, C

1

-C

4

-alkylthio, di-(C

1

-C

4

-alkyl)amino, C

1

-C

4

-alkylcarbonyl or C

1

-C

4

-alkoxycarbonyl;

R

3

is cyano, halogen, C

1

-C

6

-alkyl, C

1

-C

6

-haloalkyl, C

1

-C

6

-alkoxy, C

1

-C

6

-haloalkoxy, C

1

-C

6

-alkylthio, C

1

-C

6

-haloalkylthio, C

1

-C

6

-alkylsulfinyl, C

1

-C

6

-haloalkylsulfinyl, C

1

-C

6

-alkylsulfonyl or C

1

-C

6

-haloalkylsulfonyl;

l is 0.

PREPARATION EXAMPLES

1. Synthesis of diethyl{3-chloro-4-[(2-hydroxy-4,4-dimethyl-6-oxocyclohex-1-en-1-yl)carbonyl]phenyl}phosphonate (Compound 3.1)

Step a) Diethyl(3-chloro-4-methylphenyl)phosphonate

A mixture of 32.0 g (0.127 mol) of 2-chloro-4-iodotoluene, 17.5 g (0.127 mol) of diethyl phosphite, 12.8 g (0.127 mol) of triethylamine and 14.7 g (0.0127 mol) of tetrakis(triphenylphosphine)palladium (0) in 200 ml of acetonitrile was refluxed for 5 hours. After cooling, the mixture was stirred into water and extracted with ethyl acetate. The organic phase was dried and concentrated and the residue was then distilled.

Yield: 23.4 g (70%); colorless oil

1

H NMR (CDCl

3

): δ=7.88 (m,1H); 7.60 (m,1H); 7,52 (m,1H); 4.10 (m,4H); 2.40 (s,3H); 1.34 (t, 6H)

Step b) Diethyl(3-chloro-4-hydroxycarbonylphenyl)phosphonate (Compound 6.1)

At 80° C., a solution of 1.76 g (11 mmol) of potassium permanganate in 10 ml of water was added a little at a time to a solution of 1.0 g (3.81 mmol) of the product from step a) in 5 ml of pyridine. The mixture was stirred at room temperature for 6 hours, sodium carbonate solution was added and the precipitate was filtered off. The filtrate was acidified using hydrochloric acid and extracted with ethyl acetate.

Yield: 0.75 g (67%); colorless solid

1

H NMR (d

6

-DMSO) δ=13.8 (brd s, 1H); 7.90 (m,1H); 7.75 (m,2H); 4.06 (m,4H); 1.25 (t,6H)

Step c) Diethyl {3-chloro-4-[(2-hydroxy-4,4-dimethyl-6-oxo-cyclohex-1-en-1-yl)carbonyl]phenyl}phosphonate

A mixture of 0.65 g (2.2 mmol) of the product from step b), 0.45 g (2.2 mmol) of N,N-dicyclohexylcarbodiimide and 0.31 g of dimedone in 30 ml of acetonitrile was stirred at room temperature overnight. 0.45 g (4.4 mmol) of triethylamine and 0.2 ml of trimethylsilyl cyanide were then added, and the mixture was stirred at room temperature for a further 18 hours. The reaction mixture was poured into 50 ml each of ethyl acetate and 2% strength sodium carbonate solution and filtered. The aqueous phase was washed with diethyl ether and subsequently adjusted to a pH of 4-5 using hydrochloric acid. The mixture was extracted with ethyl acetate, the organic phase was dried and the solvent was removed.

Yield: 0.36 g (39%); red oil

1

H NMR (CDCl

3

): δ=7.78 (m,2H); 7.28 (m,1H); 4.12 (m,4H); 2.65 (m,2H); 2.32 (m,2H); 1.32 (t,6H); 1.14 (s,6H).

2. Synthesis of diethyl {3-chloro-4-[(1-ethyl-5-hydroxy-1H-pyrazol-4-ylcarbonyl]phenyl}phosphonate (Compound 5.1)

At room temperature, a mixture of 1.0 g (3.4 mmol) of the product from Synthesis 1 step b), 0.71 g (3.4 mmol) of N,N-dicyclohexylcarbodiimide and 0.38 g (3.4 mmol) of 5-hydroxy-1-ethylpyrazole was stirred for 36 hours. The reaction mixture was poured into 50 ml each of ethyl acetate and 2% strength sodium carbonate solution, the organic phase was dried and the solvent was removed. The residue was chromatographed over silica gel using cyclohexane/ethyl acetate. The resulting O-acylated product (0.36 g) in 1,4-dioxane was then admixed with potassium carbonate and refluxed for 4 hours. The reaction mixture was poured into water and extracted with ethyl acetate. The aqueous phase was washed once with diethyl ether, adjusted to pH 4 using hydrochloric acid and extracted with ethyl acetate. The organic phase was dried and the solvent was removed.

Yield: 0.17 g; red oil

1

H NMR (CDCl

3

): δ=7.95 (m,1H); 7.78 (m,1H); 7.55 (m,1H); 7.38 (s,1H); 4.40 (m,2H); 4.13 (m,4H); 1.44 (t,3H); 1.36 (t,6H)

In addition to the compounds of the formula I or IV described above, Tables 3 to 7 list other compounds which were prepared or are preparable in a similar manner:

TABLE 3

physical data mp [° C.].

No.

R

1

R

2

R

3

R

4

l

R

6

R

7

R

8

R

9

R

10

R

11

R

12

1

H NMR [δppm]

3.1

OCH

2

CH

3

OCH

2

CH

3

Cl

H(1 = O)

OH

H

H

CH

3

CH

3

H

H

7.78(m.2H); 7.28(m.1H);

4.12(m.4H); 2.65(m.2H);

2.32(m.2H); 1.32(t.6H);

1.14(s.6H)

3.2

OCH

2

CH

3

OCH

2

CH

3

Cl

H(1 = O)

OH

H

H

H

H

H

H

97-98

3.3

CH

3

CH

3

Cl

H(1 = O)

OH

H

H

CH

3

CH

3

H

H

7.70(m.2H); 7.35(m.1H);

2.68(s.2H); 2.35(s.2H);

1.78(d.6H); 1.12(s.6H)

3.4

CH

3

CH

3

Cl

H(1 = O)

OH

H

H

H

H

H

H

60-62

3.5

CH

3

CH

3

Cl

H(1 = O)

OH

CH

3

CH

3

═O

CH

3

CH

3

99-100

3.6

OCH

2

CH

3

OCH

2

CH

3

Cl

H(1 = O)

OH

CH

3

CH

3

═O

CH

3

CH

3

121-122

TABLE 4

physical data mp [° C.],

No.

R

1

R

2

R

3

R

4

l

R

6

1

H NMR [δppm]

4.1

OCH

2

CH

3

OCH

2

CH

3

Cl

H(1 = O)

SC

6

H

5

7.78(m.2H); 7.52(m.6H); 4.10(m.4H);

3.07(t.1H); 2.90(t.1H); 2.05(m.2H);

1.84(m.2H); 1.55(m.2H); 1.38(t.6H)

4.2

OCH

2

CH

3

OCH

2

CH

3

Cl

H(1 = O)

OH

150

4.3

CH

3

CH

3

Cl

H(1 = O)

OH

178-179

TABLE 5

physical data mp [° C.],

No.

R

1

R

2

R

3

R

4

l

R

20

R

21

R

22

1

H NMR [δppm]

5.1

OCH

2

CH

3

OCH

2

CH

3

Cl

H(1 = O)

OH

CH

2

CH

3

H

7.95(m.1H); 7.78(m.1H); 7.55(m.1H);

7.38(s.1H); 4.40(m.2H); 4.13(m.4H);

1.44(t.3H); 1.36(t.6H)

5.2

OCH

2

CH

3

OCH

2

CH

3

Cl

H(1 = O)

OH

CH

3

H

7.90(d.1H); 7.80(m.1H); 7.54(m.1H);

7.38(s.1H); 4.16(m.4H); 3.70(s.3H);

1.38(t.6H)

TABLE 6

physical data mp [° C.],

No.

R

1

R

2

R

3

R

4

l

R

6

R

7

R

8

R

9

R

10

R

11

R

12

1

H NMR [δppm]

6.1

CH

3

CH

3

Cl

H(1 = O)

OH

H

H

H

H

H

H

200-201

6.2

CH

3

CH

3

Cl

H(1 = O)

OH

H

H

CH

3

CH

3

H

H

161-162

TABLE 7

IV2

physical data mp [° C.],

No.

R

1

R

2

R

3

R

4

l

R

26

1

H NMR [δ ppm]

7.1

OCH

2

CH

3

OCH

2

CH

3

Cl

H(l═O)

OH

13.8 (bs. 1H); 7.90 (m.1H);7.75 (m.2H);

4.06 (m.4H); 1.25 (t.6H)

7.2

CH

3

CH

3

Cl

H(l═O)

OH

7.84 (m.3H); 1.68 (d.6H)

The compounds of the formula I and their agriculturally useful salts are suitable, both in the form of isomer mixtures and in the form of the pure isomers, as herbicides. The herbicidal compositions comprising compounds of the formula I control vegetation on non-crop areas very efficiently, especially at high rates of application. They act against broad-leaved weeds and grass weeds in crops such as wheat, rice, maize, soya and cotton without causing any significant damage to the crop plants. This effect is mainly observed at low rates of application.

Depending on the application method in question, the compounds of the formula I, or herbicidal compositions comprising them, can additionally be employed in a further number of crop plants for eliminating undesirable plants. Examples of suitable crops are the following:

Allium cepa, Ananas comosus, Arachis hypogaea, Asparagus officinalis, Beta vulgaris

spec.

altissima, Beta vulgaris

spec.

rapa, Brassica napus

var.

napus, Brassica napus

var.

napobrassica, Brassica rapa

var.

silvestris, Camellia sinensis, Carthamus tinctorius, Carya illinoinensis, Citrus limon, Citrus sinensis, Coffea arabica

(

Coffea canephora, Coffea liberica

),

Cucumis sativus, Cynodon dactylon, Daucus carota, Elaeis guineensis, Fragaria vesca, Glycine max, Gossypium hirsutum

, (

Gossypium arboreum, Gossypium herbaceum, Gossypium vitifolium

),

Helianthus annuus, Hevea brasiliensis, Hordeum vulgare, Humulus lupulus, Ipomoea batatas, Juglans regia, Lens culinaris, Linum usitatissimum, Lycopersicon lycopersicum

, Malus spec.,

Manihot esculenta, Medicago sativa

, Musa spec.,

Nicotiana tabacum

(

N.rustica

),

Olea europaea, Oryza sativa, Phaseolus lunatus, Phaseolus vulgaris, Picea abies

, Pinus spec.,

Pisum sativum, Prunus avium, Prunus persica, Pyrus communis, Ribes sylvestre, Ricinus communis, Saccharum officinarum, Secale cereale, Solanum tuberosum, Sorghum bicolor

(

s. vulgare

),

Theobroma cacao, Trifolium pratense, Triticum aestivum, Triticum durum, Vicia faba, Vitis vinifera

and

Zea mays.

In addition, the compounds of the formula I may also be used in crops which tolerate the action of herbicides owing to breeding, including genetic engineering methods.

The compounds of the formula I, or the compositions comprising them, can be used for example in the form of ready-to-spray aqueous solutions, powders, suspensions, also highly-concentrated aqueous, oily or other suspensions or dispersions, emulsions, oil dispersions, pastes, dusts, materials for broadcasting, or granules, by means of spraying, atomizing, dusting, spreading or watering. The use forms depend on the intended purpose; in any case, they should guarantee the finest possible distribution of the active ingredients according to the invention.

The herbicidal compositions comprise a herbicidally effective amount of at least one compound of the formula I or an agriculturally useful salt of I, and auxiliaries which are customary for the formulation of crop protection agents.

Suitable as inert auxiliaries are essentially the following:

mineral oil fractions of medium to high boiling point, such as kerosene and diesel oil, furthermore coal tar oils and oils of vegetable or animal origin, aliphatic, cyclic and aromatic hydrocarbons, e.g. paraffin, tetrahydronaphthalene, alkylated naphthalenes and their derivatives, alkylated benzenes and their derivatives, alcohols such as methanol, ethanol, propanol, butanol and cyclohexanol, ketones such as cyclohexanone, strongly polar solvents, e.g. amines such as N-methylpyrrolidone, and water.

Aqueous use forms can be prepared from emulsion concentrates, Asuspensions, pastes, wettable powders or water-dispersible granules by adding water. To prepare emulsions, pastes or oil dispersions, the phosphorus-containing benzoyl derivatives of the formula I, either as such or dissolved in an oil or solvent, can be homogenized in water by means of a wetting agent, tackifier, dispersant or emulsifier. Alternatively, it is also possible to prepare concentrates comprising active ingredient, wetting agent, tackifier, dispersant or emulsifier and, if desired, solvent or oil, which are suitable for dilution with water.

Suitable surfactants are the alkali metal salts, alkaline earth metal salts and ammonium salts of aromatic sulfonic acids, e.g. ligno-, phenol-, naphthalene- and dibutylnaphthalenesulfonic acid, and of fatty acids, alkyl- and alkylarylsulfonates, alkyl sulfates, lauryl ether sulfates and fatty alcohol sulfates, and salts of sulfated hexa-, hepta- and octadecanols, and also of fatty alcohol glycol ethers, condensates of sulfonated naphthalene and its derivatives with formaldehyde, condensates of naphthalene or of the naphthalenesulfonic acids with phenol and formaldehyde, polyoxyethylene octylphenol ether, ethoxylated isooctyl-, octyl- or nonylphenol, alkylphenyl or tributylphenyl polyglycol ether, alkylaryl polyether alcohols, isotridecyl alcohol, fatty alcohol/ethylene oxide condensates, ethoxylated castor oil, polyoxyethylene alkyl ethers or polyoxypropylene alkyl ethers, lauryl alcohol polyglycol ether acetate, sorbitol esters, lignin-sulfite waste liquors or methylcellulose.

Powders, materials for scattering and dusts can be prepared by mixing or grinding the active ingredients together with a solid carrier.

Granules, e.g. coated granules, impregnated granules and homogeneous granules, can be prepared by binding the active ingredients to solid carriers. Solid carriers are mineral earths such as silicas, silica gels, silicates, talc, kaolin, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate, magnesium sulfate and magnesium oxide, ground synthetic materials, fertilizers such as ammonium sulfate, ammonium phosphate, ammonium nitrate and ureas, and products of vegetable origin, such as cereal meal, tree bark meal, wood meal and nutshell meal, cellulose powders, or other solid carriers.

The concentrations of the compounds of the formula I in the ready-to-use preparations can be varied within wide ranges. In general, the formulations comprise approximately from 0.001 to 98% by weight, preferably 0.01 to 95% by weight of at least one active ingredient. The active ingredients are employed in a purity of from 90% to 100%, preferably 95% to 100% (according to NMR spectrum).

The formulation examples below illustrate the preparation of such compositions:

I. 20 parts by weight of the compound No. 3.3 are dissolved in a mixture composed of 80 parts by weight of alkylated benzene, 10 parts by weight of the adduct of from 8 to 10 mol of ethylene oxide to 1 mol of oleic acid N-monoethanol-amide, 5 parts by weight of calcium dodecylbenzenesulfonate and 5 parts by weight of the adduct of 40 mol of ethylene oxide to 1 mol of castor oil. Pouring the solution into 100,000 parts by weight of water and finely distributing it therein gives an aqueous dispersion which comprises 0.02% by weight of the active ingredient.

iii. 20 parts by weight of the compound No. 3.3 are dissolved in a mixture composed of 40 parts by weight of cyclohexanone, 30 parts by weight of isobutanol, 20 parts by weight of the adduct of 7 mol of ethylene oxide to 1 mol of isooctyl-phenol and 10 parts by weight of the adduct of 40 mol of ethylene oxide to 1 mol of castor oil. Pouring the solution into 100,000 parts by weight of water and finely distributing it therein gives an aqueous dispersion which comprises 0.02% by weight of the active ingredient.

II. 20 parts by weight of the compound No. 3.3 are dissolved in a mixture composed of 25 parts by weight of cyclohexanone, 65 parts by weight of a mineral oil fraction of boiling point 210 to 280° C. and 10 parts by weight of the adduct of 40 mol of ethylene oxide to 1 mol of castor oil. Pouring the solution into 100,000 parts by weight of water and finely distributing it therein gives an aqueous dispersion which comprises 0.02% by weight of the active ingredient.

IV. 20 parts by weight of the compound No. 3.3 are mixed thoroughly with 3 parts by weight of sodium diisobutylnaphthalenesulfonate, 17 parts by weight of the sodium salt of a lignosulfonic acid from a sulfite waste liquor and 60 parts by weight of pulverulent silica gel, and the mixture is ground in a hammer mill. Finely distributing the mixture in 20,000 parts by weight of water gives a spray mixture which comprises 0.1% by weight of the active ingredient.

V. 3 parts by weight of the compound No. 3.3 are mixed with 97 parts by weight of finely divided kaolin. This gives a dust which comprises 3% by weight of the active ingredient.

VI. 20 parts by weight of the compound No. 3.3 are mixed intimately with 2 parts by weight of calcium dodecylbenzenesulfonate, 8 parts by weight of fatty alcohol polyglycol ether, 2 parts by weight of the sodium salt of a phenol/urea/formaldehyde condensate and 68 parts by weight of a paraffinic mineral oil. This gives a stable oily dispersion.

VII. 1 part by weight of the compound No. 3.3 is dissolved in a mixture composed of 70 parts by weight of cyclohexanone, 20 parts by weight of ethoxylated isooctylphenol and 10 parts by weight of ethoxylated castor oil. This gives a stable emulsion concentrate.

VIII. 1 part by weight of the compound No. 3.3 is dissolved in a mixture composed of 80 parts by weight of cyclohexanone and 20 parts by weight of Wettol® EM 31 (=nonionic emulsifier based on ethoxylated castor oil). This gives a stable emulsion concentrate.

The compounds of the formula I or the herbicidal compositions can be appled pre- or post-emergence. If the active ingredients are less well tolerated by certain crop plants, application techniques may be used in which the herbicidal compositions are sprayed, with the aid of the spraying equipment, in such a way that as far as possible they do not come into contact with the leaves of the sensitive crop plants, while the active ingredients reach the leaves of undesirable plants growing underneath, or the bare soil surface (post-directed, lay-by).

The rates of application of the compound of the formula I are from 0.001 to 3.0, preferably 0.01 to 1.0, kg/ha of active substance (a.s.), depending on the control target, the season, the target plants and the growth stage.

To widen the spectrum of action and to achieve synergistic effects, the phosphorus-containing benzoyl derivatives of the formula I may be mixed with a large number of representatives of other herbicidal or growth-regulating active ingredient groups and then applied concomitantly. Suitable components for mixtures are, for example, 1,2,4-thiadiazoles, 1,3,4-thiadiazoles, amides, amino-phosphoric acid and its derivatives, aminotriazoles, anilides, aryloxy-/heteroaryloxyalkanoic acids and their derivatives, benzoic acid and its derivatives, benzothiadiazinones, 2-aroyl-1,3-cyclohexanediones, hetaryl aryl ketones, benzylisoxazolidinones, meta-CF

3

-phenyl derivatives, carbamates, quinolinecarboxylic acid and its derivatives, chloroacetanilides, cyclohexenone oxime ether derivatives, diazines, dichloropropionic acid and its derivatives, dihydrobenzofurans, dihydrofuran-3-ones, dinitroanilines, dinitrophenols, diphenyl ethers, dipyridyls, halocarboxylic acids and their derivatives, ureas, 3-phenyluracils, imidazoles, imidazolinones, N-phenyl-3,4,5,6-tetrahydro-phthalimides, oxadiazoles, oxiranes, phenols, aryloxy- and hetaryloxyphenoxypropionic esters, phenylacetic acid and its derivatives, phenylpropionic acid and its derivatives, pyrazoles, phenylpyrazoles, pyridazines, pyridinecarboxylic acid and its derivatives, pyrimidyl ethers, sulfonamides, sulfonylureas, triazines, triazinones, triazolinones, triazolecarboxamides and uracils.

It may furthermore be advantageous to apply the compounds of the formula I, alone or in combination with other herbicides, or in the form of a mixture with other crop protection agents, for example together with agents for controlling pests or phytopathogenic fungi or bacteria. Also of interest is the miscibility with mineral salt solutions, which are employed for treating nutritional and trace element deficiencies.

Non-phytotoxic oils and oil concentrates may also be added.

USE EXAMPLES

The herbicidal activity of the phosphorus-containing benzoyl derivatives of the formula I was demonstrated by the following greenhouse experiments:

The culture containers used were plastic flowerpots containing loamy sand with approximately 3.0% of humus as the substrate. The seeds of the test plants were sown separately for each species.

For the pre-emergence treatment, the active ingredients, which had been suspended or emulsified in water, were applied directly after sowing by means of finely distributing nozzles. The containers were irrigated gently to promote germination and growth and subsequently covered with transparent plastic hoods until the plants had rooted. This cover causes uniform germination of the test plants, unless this was adversely affected by the active ingredients.

For the post-emergence treatment, the test plants were first grown to a height of 3 to 15 cm, depending on the plant habit, and only then treated with the active compounds which had been suspended or emulsified in water. For this purpose, the test plants were either sown directly and grown in the same containers, or they were first grown separately as seedlings and transplanted into the test containers a few days prior to treatment. The rate of application for the post-emergence treatment was 0.5 or 0.25 kg/ha of a.s. (active substance).

Depending on the species, the plants were kept at 10-25° C. or 20-35° C. The test period extended over 2 to 4 weeks. During this time, the plants were tended, and their response to the individual treatments was evaluated.

Evaluation was carried out using a scale from 0 to 100. 100 means no emergence of the plants, or complete destruction of at least the aerial parts, and 0 means no damage, or normal course of growth.

The plants used in the greenhouse experiments belonged to the following species:

338

Scientific name

English name

Chenopodium album

lambsquarters

(goosefoot)

Echinochloa crus-galli

barnyardgrass

Setaria faberi

giant foxtail

Setaria viridis

green foxtail

Solanum nigrum

black nightshade

The compounds 3.4, applied post-emergence, showed very good activity against the abovementioned harmful plants at rates of application of 0.5 and 0.25 kg/ha, respectively.

Number	Name	Date	Kind
3775057	Redmore	Nov 1973	A
3882202	Aya et al.	May 1975	A
3936433	Satomi et al.	Feb 1976	A
3974243	Kleiner	Aug 1976	A
4780127	Michaely et al.	Oct 1988	A
5834402	von Deyn et al.	Nov 1998	A
5846907	von Deyn et al.	Dec 1998	A
6165944	von Deyn et al.	Dec 2000	A

Number	Date	Country
2289114	Nov 1998	CA
203 428	Dec 1986	EP
315 975	May 1989	EP
418 175	Mar 1991	EP
609 797	Aug 1994	EP
625 505	Nov 1994	EP
1 200 273	Jul 1970	GB
49 011418	Mar 1974	JP
WO 9850337	Nov 1998	WO

Phosphoric benzoyl derivatives and their use as herbicides

Information

Patent Number

Date Filed

Date Issued

Inventors

Original Assignees

Examiners

Agents

CPC

US Classifications

Field of Search

US

International Classifications

Abstract

Description

Claims

Priority Claims (1)

Parent Case Info

PCT Information

US Referenced Citations (8)

Foreign Referenced Citations (9)

Non-Patent Literature Citations (6)

Entry
Hawkins et al. “An In-depth Study of the Azidobenzophenone-Anthranil-Acridone Transformation”Chem. Soc. Perkins Trans. (1983) pp. 2077-2087.
Kluger et al. “Amide Phosphate Interactions: Acid Catalysts in Amide-Assisted Hydrolysis of Phosphonate Esters” Jour. Am. Chem. Soc. vol. 98, No. 16, (1976) pp. 4913-4917.
Petrakis et al. “Palladium Catalyzed Substitutions of Triflates Derived from Tyrosine-Containing Peptides and Simpler Hydroxyarenes Forming 4-(Diethoxyphosphinyl) pheylzlanines and Diethyl Arylphosphonates” Jour. Am. Chem. SOc. vol. 109 No. 9 (1987) pp. 2831-2833.
El-Deek et al. “Synthesis and reaction of p-(diphenylophosphino)benzoic acid” J. Indian Chem. Soc. vol. 58 No. 2 (1981) pp. 197-199.
Petrovxkii et al. “Amidophosphinylbenzoic acids” Izv. Akad. Nunk. SSSR Ser. Khim. vol. 9 (1974) pp. 2090-2093.
Hall et al. “The Preparation and Diels-Alder Reactivity of Ethyl (Diethoxyphosphinyl) Propynoate” Tetrahedron Letters vol. 23 No. 25 (1982) pp. 2603-2604.