Claims
- 1. An N-substituted N-arylcyanamide derivative of the general formula: ##STR17## wherein R.sup.3, R.sup.4 and R.sup.5 are the same or different, each of which is hydrogen, optionally substituted alkyl or optionally substituted aryl; R.sup.12 is optionally substituted aryl; and X is halogen, with the exception of N-phenyl-N-(2-bromo-2-propenyl)cyanamide.
- 2. A compound of the formula: ##STR18##
- 3. The derivative of claim 1, wherein R.sup.3, R.sup.4 and R.sup.5 are the same or different, and each is hydrogen, C.sub.1-8 alkyl optionally substituted with at least one substituent elected from the group consisting of C.sub.1-8 alkoxy, aryl, and C.sub.3-8 cycloalkyl; and aryl optionally substituted with at least one substituent selected from the group consisting of C.sub.1-8 alkyl, C.sub.1-8 alkoxy, aryl, nitro and halogen.
- 4. The derivative of claim 1, wherein R.sup.12 is aryl optionally substituted with at least one substituent selected from the group consisting of C.sub.1-8 alkyl optionally substituted with at least one halogen; C.sub.1-8 alkoxy optionally substituted with at least one halogen; aryl; nitro; and halogen.
- 5. The derivative of claim 1 which is selected from the group consisting of:
- N-(3-trifluoromethyl)phenyl)-N-(2-chloro-2-propenyl)cyanamide;
- N-(3-trifluoromethyl)phenyl)-N-(2-chloro-1-methyl-2-propenyl)cyanamide;
- N-(3-trifluoromethyl)phenyl)-N-(2-chloro-2-butenyl)cyanamide;
- N-(3-trifluoromethyl)phenyl)-N-(2-chloro-3-methyl-2-butenyl)cyanamide;
- N-(3-trifluoromethyl)phenyl)-N-(2-bromo-2-propenyl)cyanamide;
- N-(3-trifluoromethoxy)phenyl)-N-(2-chloro-2-propenyl)cyanamide;
- N-(3-trifluoromethoxy)phenyl)-N-(2-chloro-1-methyl-2-propenyl)cyanamide;
- N-(3-trifluoromethoxy)phenyl)-N-(2-chloro -2-butenyl)cyanamide;
- N-(3-trifluoromethoxy)phenyl)-N-(2-chloro-3-methyl-2-butenyl)cycanmide;
- N-(4-fluoro-3-(trifluoromethyl)phenyl)-N-(2-chloro-2-propenyl)cyanamide;
- N-(4-fluoro-3-(trifluoromethyl)phenyl)-N-(2-chloro-1-methyl-2-propenyl)-cyanamide;
- N-(4-fluoro-3-(trifluoromethyl)phenyl)-N-(2-chloro-2-butenyl)cyanamide;
- N-(4-fluoro-3-(trifluoromethyl)phenyl)-N-(2-chloro-3-methyl-2-butenyl)-cyanamide;
- N-(3,5-dichlorophenyl)-N-(2-chloro-2-propenyl)cyanamide;
- N-(4-methoxyphenyl)-N-(2-chloro-2-propenyl)cyanamide; and
- N-(2-chlorophenyl)-N-(2-chloro-2-propenyl)cyanamide.
Priority Claims (2)
Number |
Date |
Country |
Kind |
4-325259 |
Apr 1992 |
JPX |
|
5-018609 |
May 1993 |
JPX |
|
Parent Case Info
This application is a divisional of copending application Ser. No. 08/434,589, filed on May 4, 1995, the entire contents of which are hereby incorporated by reference; which was a divisional of application Ser. No. 08/160,261, filed on Dec. 2, 1993, now U.S. Pat. No. 5,463,069 the entire contents of which are hereby incorporated by reference.
US Referenced Citations (4)
Foreign Referenced Citations (4)
Number |
Date |
Country |
529482A1 |
Mar 1993 |
EPX |
529481A1 |
Mar 1993 |
EPX |
1511325 |
Dec 1967 |
FRX |
53-90222 |
Aug 1978 |
JPX |
Non-Patent Literature Citations (3)
Entry |
Johnson et al., J. Org. Chem., Jan. 1964, vol. 20, pp. 153-157. |
Bramley et al., J. Chem. Soc. Perkin Trans. I, 1987, pp. 639-643. |
Sugiyama et al., Chem. Pharm. Bull., 37(8), 1989, pp. 2122-2131. |
Divisions (2)
|
Number |
Date |
Country |
Parent |
434589 |
May 1995 |
|
Parent |
160261 |
Dec 1993 |
|