Related Application This application is a division of U.S. application Ser. No. 07/279,194, filed Dec. 6, 1988, which is a continuation-in-part of U.S. application Ser. No. 07/142,580, filed Jan. 7, 1988, now abandoned, which is a continuation-in-part of U.S. application Ser. No. 050,341, filed May 22, 1987, now abandoned, which is a continuation-in-part of U.S. application Ser. No. 884,920, filed Jul. 11, 1986, now abandoned.
Number | Name | Date | Kind |
---|---|---|---|
3772315 | Regel et al. | Nov 1973 | |
4207324 | Matsumura et al. | Jun 1980 | |
4226878 | Iizuka et al. | Oct 1980 | |
4301169 | Yamanaka et al. | Nov 1981 | |
4328349 | Grayboyes et al. | May 1982 | |
4340598 | Furukawa et al. | Jul 1982 | |
4347364 | Walser et al. | Aug 1982 | |
4347365 | Walser et al. | Aug 1982 | |
4355040 | Furukawa et al. | Oct 1982 | |
4379927 | Vorbruggen et al. | Apr 1983 | |
4402966 | Yamanaka et al. | Sep 1983 | |
4435395 | Loev et al. | Mar 1984 | |
4448781 | Cross et al. | May 1984 | |
4463011 | Ogata | Jul 1984 | |
4532331 | Frazee et al. | Jul 1985 | |
4533669 | Yamanaka et al. | Aug 1985 | |
4539322 | Campbell et al. | Sep 1985 | |
4602031 | Yamanaka et al. | Jul 1986 | |
4689182 | Rafferty | Aug 1987 | |
4755518 | Rafferty | Jul 1988 |
Number | Date | Country |
---|---|---|
028834 | May 1981 | EPX |
90978 | Oct 1983 | EPX |
103647 | Mar 1984 | EPX |
125003 | Nov 1984 | EPX |
125033 | Nov 1984 | EPX |
142754 | May 1985 | EPX |
146228 | Jun 1985 | EPX |
0253310A2 | Jan 1988 | EPX |
3426081 | Jan 1986 | DEX |
3426195 | Jan 1986 | DEX |
8298270 | Jun 1982 | JPX |
Entry |
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Wong et al., Abstract No. 30, Hypertension, p. 340, vol. 12, No. 3, Sep. 1988, High Blood Pressure Council Mtg., San Francisco, Calif., Sep. 28-Oct. 1, 1988, "X-6803 Methyl-2-N-Butyl-1-(4-(2-Carboxybenzamido)Benzyl-4-Chloroimidazole-5-Acetate, Sodium Salt): A Novel Noneptide Angiotensin II Receptor Antagonist". |
Chiu et al., Abstract No. 118.11, The Pharmacologist, vol. 30, p. A165, 1988, for ASPET Mtg., Montreal, Canada, Oct. 9-13, 1988: "Nonpeptide Angiotensin II (AII) Receptor Antagonists: Structure Function Studies". |
Wong et al., Nonpeptide Angiotensin II Receptor Antagonists, I Pharmacological Characterization of 2-n-Butyl-Chloro-1(2-chlorobenzyl)imidazole-5-acetic Acid, Sodium Salt (S-8307), "J. Pharmacology and Experimental Therapeutics," vol. 247, No. 1, pp. 1-7 (1988). |
Chiu et al., "Non-Peptide Angiotensin II Receptor Antagonists, II, Pharmacology of S-8303," European Journal of Pharmacology, vol. 157, pp. 13-21 (1988). |
Lindgren et al., Eur. J. Pharmacol., 135:383, 1987. |
Schmidt et al., J. Cardiovascular Pharmacology, vol. 8, pp. S100-105, 1986. |
H. Torii, Takeda Kenkyusshoho, 40, No. 3/4, 180-191 (1982). |
Pals et al., Circulation Research, 29, 673 (1971). |
Streeten and Anderson, Handbook of Hypertension, vol. 5, Clinical Pharmogy of Antihypertensive Drugs, A. E. Doyle (Editor), Elsevier Science Publishers B. V., p. 246 (1984). |
Satoh et al., Cir. Res., 36/37 & Suppl. I: I-89, 1975. |
Number | Date | Country | |
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Parent | 279194 | Dec 1988 |
Number | Date | Country | |
---|---|---|---|
Parent | 142580 | Jan 1988 | |
Parent | 50341 | May 1987 | |
Parent | 884920 | Jul 1986 |