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last 30 patents
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Patent Grant
P2X7 modulators
Patent number
12,247,027
Issue date
Mar 11, 2025
JANSSEN PHARMACEUTICA NV
Manuel Jesus Alcazar Vaca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrazolo-pyridine amides and their use as GluN2B recept...
Patent number
12,172,997
Issue date
Dec 24, 2024
JANSSEN PHARMACEUTICA NV
Afton Hiscox
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
P2X7 modulators
Patent number
11,820,770
Issue date
Nov 21, 2023
JANSSEN PHARMACEUTICA NV
Manuel Jesus Alcazar Vaca
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 1H-imidazo[4,5-b]pyridin-2(3H)-ones and their use as GL...
Patent number
11,759,455
Issue date
Sep 19, 2023
JANSSEN PHARMACEUTICA NV
Christa C Chrovian
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrazolo-pyridine amides and their use as GluN2B recept...
Patent number
11,618,750
Issue date
Apr 4, 2023
JANSSEN PHARMACEUTICA NV
Afton Hiscox
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
P2X7 modulators
Patent number
11,225,478
Issue date
Jan 18, 2022
JANSSEN PHARMACEUTICA NV
Manuel Jesus Alcazar Vaca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted 1H-imidazo[4,5-b]pyridin-2(3H)-ones and their use as GL...
Patent number
11,207,298
Issue date
Dec 28, 2021
JANSSEN PHARMACEUTICA NV
Christa C Chrovian
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Disubstituted octahydropyrrolo[3,4-c]pyrroles as orexin receptor mo...
Patent number
RE48841
Issue date
Dec 7, 2021
JANSSEN PHARMACEUTICA NV
Wenying Chai
Information
Patent Grant
Substituted 1,2,3-triazoles as NR2B-selective NMDA modulators
Patent number
10,766,880
Issue date
Sep 8, 2020
JANSSEN PHARMACEUTICA NV
Gang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
P2X7 modulators
Patent number
10,703,749
Issue date
Jul 7, 2020
JANSSEN PHARMACEUTICA NV
Manuel Jesus Alcazar Vaca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted 1H-imidazo[4,5-b]pyridin-2(3H)-ones and their use as Gl...
Patent number
10,617,676
Issue date
Apr 14, 2020
JANSSEN PHARMACEUTICA NV
Christa C Chrovian
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted 4-azaindoles and their use as GluN2B receptor modulators
Patent number
10,377,753
Issue date
Aug 13, 2019
JANSSEN PHARMACEUTICA NV
Christa C. Chrovian
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 1,2,3-triazoles as NR2B-selective NMDA modulators
Patent number
10,233,173
Issue date
Mar 19, 2019
JANSSEN PHARMACEUTICA NV
Gang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
P2X7 modulators
Patent number
10,150,765
Issue date
Dec 11, 2018
JANSSEN PHARMACEUTICA NV
Manuel Jesus Alcazar Vaca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
P2X7 modulators and methods of use
Patent number
10,112,937
Issue date
Oct 30, 2018
JANSSEN PHARMACEUTICA NV
Manuel Jesus Alcazar Vaca
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 1,2,3-triazoles as NR2B-selective NMDA modulators
Patent number
10,071,988
Issue date
Sep 11, 2018
JANSSEN PHARMACEUTICA NV
Gang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 4-azaindoles and their use as GluN2B receptor modulators
Patent number
9,963,447
Issue date
May 8, 2018
Janssen Pharmaceutica N.V.
Christa C. Chrovian
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
P2X7 modulators
Patent number
9,464,084
Issue date
Oct 11, 2016
Janssen Pharmaceutica N.V.
Manuel Jesus Alcazar Vaca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
P2X7 modulators
Patent number
9,066,946
Issue date
Jun 30, 2015
JANSSEN PHARMACEUTICA NV
Manuel Jesus Alcazar Vaca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Disubstituted octahydropyrrolo[3,4-c]pyrroles as orexin receptor mo...
Patent number
8,653,263
Issue date
Feb 18, 2014
Janssen Pharmaceutica
Wenying Chai
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrrolidine amides as modulators of the histamine H3 re...
Patent number
8,236,792
Issue date
Aug 7, 2012
JANSSEN PHARMACEUTICA NV
Nicholas I Carruthers
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
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Patent Application
P2X7 MODULATORS
Publication number
20240116930
Publication date
Apr 11, 2024
Janssen Pharmaceutica N.V.
Manuel Jesus ALCAZAR VACA
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 1H-IMIDAZO[4,5-b]PYRIDIN-2(3H)-ONES AND THEIR USE AS GL...
Publication number
20230338341
Publication date
Oct 26, 2023
Janssen Pharmaceutica N.V.
Christa C. Chrovian
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRAZOLO-PYRIDINE AMIDES AND THEIR USE AS GLUN2B RECEPTOR
Publication number
20230151006
Publication date
May 18, 2023
Janssen Pharmaceutica N.V.
Afton HISCOX
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 1H-IMIDAZO[4,5-b]PYRIDIN-2(3H)-ONES AND THEIR USE AS GL...
Publication number
20230000833
Publication date
Jan 5, 2023
Janssen Pharmaceutica N.V.
Christa C. Chrovian
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
P2X7 MODULATORS
Publication number
20220235062
Publication date
Jul 28, 2022
Janssen Pharmaceutica N.V.
Jose Ignacio ANDRES GIL
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
P2X7 MODULATORS
Publication number
20220213095
Publication date
Jul 7, 2022
Janssen Pharmaceutica N.V.
Manuel Jesus Alcazar Vaca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 1H-IMIDAZO[4,5-B]PYRIDIN-2(3H)-ONES AND THEIR USE AS GL...
Publication number
20210069155
Publication date
Mar 11, 2021
Janssen Pharmaceutica N.V.
Christa C. Chrovian
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRAZOLO-PYRIDINE AMIDES AND THEIR USE AS GLUN2B RECEPT...
Publication number
20210017168
Publication date
Jan 21, 2021
Janssen Pharmaceutica N.V.
Afton HISCOX
C07 - ORGANIC CHEMISTRY
Information
Patent Application
P2X7 Modulators
Publication number
20200325138
Publication date
Oct 15, 2020
Janssen Pharmaceutica N.V.
Manuel Jesus Alcazar Vaca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 1,2,3-TRIAZOLES AS NR2B-SELECTIVE NMDA MODULATORS
Publication number
20190135791
Publication date
May 9, 2019
Janssen Pharmaceutica N.V.
Gang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
P2X7 Modulators
Publication number
20190092770
Publication date
Mar 28, 2019
Janssen Pharmaceutica N.V.
Manuel Jesus Alcazar Vaca
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 1,2,3-TRIAZOLES AS NR2B-SELECTIVE NMDA MODULATORS
Publication number
20180334451
Publication date
Nov 22, 2018
Janssen Pharmaceutica N.V.
Gang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 4-AZAINDOLES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS
Publication number
20180208595
Publication date
Jul 26, 2018
Janssen Pharmaceutica N.V.
Christa C. Chrovian
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 1H-IMIDAZO[4,5-b]PYRIDIN-2(3H)-ONES AND THEIR USE AS GL...
Publication number
20180125826
Publication date
May 10, 2018
JANSSEN PHARMACEUTICA NV
Christa C. Chrovian
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 1,2,3-TRIAZOLES AS NR2B-SELECTIVE NMDA MODULATORS
Publication number
20170226089
Publication date
Aug 10, 2017
Janssen Pharmaceutica N.V.
Gang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 4-AZAINDOLES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS
Publication number
20170008890
Publication date
Jan 12, 2017
Janssen Pharmaceutica N.V.
Christa C. CHROVIAN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
P2X7 MODULATORS
Publication number
20160376271
Publication date
Dec 29, 2016
Janssen Pharmaceutica N.V.
Manuel Jesus Alcazar Vaca
C07 - ORGANIC CHEMISTRY
Information
Patent Application
P2X7 MODULATORS
Publication number
20160039809
Publication date
Feb 11, 2016
Janssen Pharmaceutica N.V.
Manuel Jesus ALCAZAR VACA
C07 - ORGANIC CHEMISTRY
Information
Patent Application
P2X7 MODULATORS
Publication number
20150322062
Publication date
Nov 12, 2015
Janssen Pharmaceutica N.V.
Manuel Jesus Alcazar Vaca
C07 - ORGANIC CHEMISTRY
Information
Patent Application
P2X7 MODULATORS
Publication number
20140275015
Publication date
Sep 18, 2014
Janssen Pharmaceutica N.V.
Manuel Jesus Alcazar Vaca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
DISUBSTITUTED OCTAHYDROPYRROLO[3,4-c]PYRROLES AS OREXIN RECEPTOR MO...
Publication number
20120208812
Publication date
Aug 16, 2012
Janssen Pharmaceutica N.V.
Wenying Chai
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRROLIDINE AMIDES AS MODULATORS OF THE HISTAMINE H3 RE...
Publication number
20090291903
Publication date
Nov 26, 2009
Nicholas I. Carruthers
C07 - ORGANIC CHEMISTRY