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Alexander J. Pickrell
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Westlake Village, CA, US
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Patents Grants
last 30 patents
Information
Patent Grant
Substituted piperazines as KRAS G12C inhibitors
Patent number
12,083,121
Issue date
Sep 10, 2024
Amgen Inc.
John Gordon Allen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Apelin polypeptides
Patent number
11,807,693
Issue date
Nov 7, 2023
Amgen Inc.
Jerry Ryan Holder
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
KRAS G12C inhibitors and methods of using the same
Patent number
11,766,436
Issue date
Sep 26, 2023
Amgen Inc.
John Gordon Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted piperazines as KRAS G12C inhibitors
Patent number
11,285,156
Issue date
Mar 29, 2022
Amgen Inc.
John Gordon Allen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
KRAS G12C inhibitors and methods of using the same
Patent number
11,285,135
Issue date
Mar 29, 2022
Amgen Inc.
Brian Alan Lanman
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds that inhibits MCL-1 protein
Patent number
11,224,601
Issue date
Jan 18, 2022
Amgen Inc.
Paul E. Harrington
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
KRAS G12C inhibitors and methods of using the same
Patent number
11,090,304
Issue date
Aug 17, 2021
Amgen Inc.
John Gordon Allen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Apelin polypeptides
Patent number
10,941,182
Issue date
Mar 9, 2021
Amgen Inc.
Jerry Ryan Holder
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Cyclopropyl fused thiazine derivatives as beta-secretase inhibitors...
Patent number
10,889,581
Issue date
Jan 12, 2021
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds that inhibit Mcl-1 protein
Patent number
10,821,115
Issue date
Nov 3, 2020
Amgen Inc.
Paul E. Harrington
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds that inhibit Mcl-1 protein
Patent number
10,632,128
Issue date
Apr 28, 2020
Amgen Inc.
Paul E. Harrington
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
KRAS G12C inhibitors and methods of using the same
Patent number
10,532,042
Issue date
Jan 14, 2020
Amgen Inc.
Brian Alan Lanman
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Unsaturated nitrogen heterocyclic compounds useful as PDE10 inhibitors
Patent number
9,718,803
Issue date
Aug 1, 2017
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cyclopropyl fused thiazin-2-amine compounds as beta-secretase inhib...
Patent number
9,550,762
Issue date
Jan 24, 2017
Amgen, Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Azetidine and piperidine compounds useful as PDE10 inhibitors
Patent number
9,493,459
Issue date
Nov 15, 2016
Amgen Inc.
Jennifer R. Allen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Carbohydrate phosphonate derivatives as modulators of glycosylation
Patent number
9,328,134
Issue date
May 3, 2016
Amgen Inc.
John Gordon Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Azetidine and piperidine compounds useful as PDE10 inhibitors
Patent number
9,303,028
Issue date
Apr 5, 2016
Amgen Inc.
Jennifer R. Allen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Heterobicyclic compounds
Patent number
9,174,992
Issue date
Nov 3, 2015
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Unsaturated nitrogen heterocyclic compounds useful as PDE10 inhibitors
Patent number
8,957,073
Issue date
Feb 17, 2015
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heteroaryloxycarbocyclyl compounds as PDE10 inhibitors
Patent number
8,952,037
Issue date
Feb 10, 2015
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aryl- and heteroaryl- nitrogen-heterocyclic compounds as PDE10 inhi...
Patent number
8,946,230
Issue date
Feb 3, 2015
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors
Patent number
8,759,532
Issue date
Jun 24, 2014
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Azetidine and piperidine compounds useful as PDE10 inhibitors
Patent number
8,691,986
Issue date
Apr 8, 2014
Amgen Inc.
Jennifer R. Allen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Aminopyridine and carboxypyridine compounds as phosphodiesterase 10...
Patent number
8,637,500
Issue date
Jan 28, 2014
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors
Patent number
8,318,718
Issue date
Nov 27, 2012
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory ac...
Patent number
7,928,139
Issue date
Apr 19, 2011
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory ac...
Patent number
7,635,715
Issue date
Dec 22, 2009
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
5,6-FUSED AND 6,6-FUSED BICYCLIC ALCOHOLS AND ETHERS AND COMPOSITIO...
Publication number
20240409557
Publication date
Dec 12, 2024
Amgen Inc.
Kevin Lloyd GREENMAN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
APELIN POLYPEPTIDES
Publication number
20240327461
Publication date
Oct 3, 2024
Amgen Inc.
Jerry Ryan HOLDER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETEROCYCLIC SPIRO COMPOUNDS AND METHODS OF USE
Publication number
20240059703
Publication date
Feb 22, 2024
Amgen Inc.
BRIAN ALAN LANMAN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
KRAS G12C INHIBITORS AND METHODS OF USING THE SAME
Publication number
20240050430
Publication date
Feb 15, 2024
Amgen Inc.
John Gordon Allen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETEROCYCLIC SPIRO COMPOUNDS AND METHODS OF USE
Publication number
20230406860
Publication date
Dec 21, 2023
Amgen Inc.
BRIAN ALAN LANMAN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL PRMT5 INHIBITORS
Publication number
20230159510
Publication date
May 25, 2023
Amgen Inc.
Jennifer Rebecca ALLEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
KRAS G12C INHIBITORS AND METHODS OF USING THE SAME
Publication number
20220395504
Publication date
Dec 15, 2022
Amgen Inc.
John Gordon Allen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
KRAS G12C INHIBITORS AND METHODS OF USING THE SAME
Publication number
20220175782
Publication date
Jun 9, 2022
Amgen Inc.
John Gordon ALLEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
KRAS G12C INHIBITORS AND METHODS OF USING THE SAME
Publication number
20220168280
Publication date
Jun 2, 2022
Amgen Inc.
Brian Alan LANMAN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
APELIN POLYPEPTIDES
Publication number
20210261619
Publication date
Aug 26, 2021
Amgen Inc.
Jerry Ryan HOLDER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CYCLOPROPYL FUSED THIAZINE DERIVATIVES AS BETA-SECRETASE INHIBITORS...
Publication number
20200231585
Publication date
Jul 23, 2020
Amgen Inc.
Jennifer R. ALLEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS THAT INHIBIT MCL-1 PROTEIN
Publication number
20200171043
Publication date
Jun 4, 2020
Amgen Inc.
Paul E. HARRINGTON
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
KRAS G12C INHIBITORS AND METHODS OF USING THE SAME
Publication number
20200069657
Publication date
Mar 5, 2020
Amgen Inc.
Brian Alan LANMAN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS THAT INHIBIT MCL-1 PROTEIN
Publication number
20190381064
Publication date
Dec 19, 2019
Amgen Inc.
Paul E. HARRINGTON
C07 - ORGANIC CHEMISTRY
Information
Patent Application
KRAS G12C INHIBITORS AND METHODS OF USING THE SAME
Publication number
20190374542
Publication date
Dec 12, 2019
Amgen Inc.
John Gordon ALLEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
KRAS G12C INHIBITORS AND METHODS OF USING THE SAME
Publication number
20190343838
Publication date
Nov 14, 2019
Amgen Inc.
John Gordon Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS THAT INHIBIT MCL-1 PROTEIN
Publication number
20180289720
Publication date
Oct 11, 2018
Amgen Inc.
Paul E. Harrington
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
KRAS G12C INHIBITORS AND METHODS OF USING THE SAME
Publication number
20180177767
Publication date
Jun 28, 2018
Amgen Inc.
Brian Alan LANMAN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CYCLOPROPYL FUSED THIAZIN-2-AMINE COMPOUNDS AS BETA-SECRETASE INHIB...
Publication number
20170267673
Publication date
Sep 21, 2017
Amgen Inc.
Jennifer R. ALLEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
APELIN POLYPEPTIDES
Publication number
20170107255
Publication date
Apr 20, 2017
Amgen Inc.
Jerry Ryan HOLDER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Heteroaryloxycarbocyclyl Compounds as PDE 10 Inhibitors
Publication number
20160280703
Publication date
Sep 29, 2016
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AZETIDINE AND PIPERIDINE COMPOUNDS USEFUL AS PDE10 INHIBITORS
Publication number
20160176874
Publication date
Jun 23, 2016
Amgen Inc.
Jennifer R. ALLEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
UNSATURATED NITROGEN HETEROCYCLIC COMPOUNDS USEFUL AS PDE10 INHIBITORS
Publication number
20160102075
Publication date
Apr 14, 2016
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Cyclopropyl Fused Thiazin-2-Amine Compounds as Beta-Secretase Inhib...
Publication number
20160046618
Publication date
Feb 18, 2016
Amgen Inc.
Jennifer R. ALLEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Carbohydrate Phosphonate Derivatives as Modulators of Glycosylation
Publication number
20150376221
Publication date
Dec 31, 2015
Amgen Inc.
John Gordon Allen
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Application
UNSATURATED NITROGEN HETEROCYCLIC COMPOUNDS USEFUL AS PDE10 INHIBITORS
Publication number
20140213572
Publication date
Jul 31, 2014
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AZETIDINE AND PIPERIDINE COMPOUNDS USEFUL AS PDE10 INHIBITORS
Publication number
20140148435
Publication date
May 29, 2014
Amgen Inc.
Jennifer R. Allen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AZETIDINE AND PIPERIDINE COMPOUNDS USEFUL AS PDE10 INHIBITORS
Publication number
20130338138
Publication date
Dec 19, 2013
Jennifer R. Allen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETEROBICYCLIC COMPOUNDS
Publication number
20130225552
Publication date
Aug 29, 2013
Amgen Inc.
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDINE AND PYRIMIDINE DERIVATIVES AS PHOSPHODIESTERASE 10 INHIBITORS
Publication number
20130079325
Publication date
Mar 28, 2013
Jennifer R. Allen
C07 - ORGANIC CHEMISTRY