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Patents Grants
last 30 patents
Information
Patent Grant
Heterocyclic compounds as monoacylglycerol lipase inhibitors
Patent number
11,802,133
Issue date
Oct 31, 2023
HOFFMANN-LA ROCHE INC.
Charles Bell
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Difluoroketamide derivatives as HTRA1 inhibitors
Patent number
11,001,555
Issue date
May 11, 2021
Hoffman-La Roche Inc.
Benoit Hornsperger
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Trifluoromethylpropanamide derivatives as HTRA1 inhibitors
Patent number
10,870,623
Issue date
Dec 22, 2020
HOFFMANN-LA ROCHE INC.
Benoit Hornsperger
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Difluoroketamide derivatives as HtrA1 inhibitors
Patent number
10,865,182
Issue date
Dec 15, 2020
HOFFMANN-LA ROCHE INC.
Hans P. Maerki
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Difluoroketamide derivatives
Patent number
10,428,108
Issue date
Oct 1, 2019
HOFFMANN-LA ROCHE INC.
Benoit Hornsperger
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Spirodiamine derivatives as aldosterone synthase inhibitors
Patent number
10,035,804
Issue date
Jul 31, 2018
Hoffman-La Roche Inc.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Trifluoromethylpropanamide derivatives
Patent number
9,980,929
Issue date
May 29, 2018
Hoffman-La Roche Inc.
Benoit Hornsperger
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Dihydroquinoline pyrazolyl compounds
Patent number
9,796,702
Issue date
Oct 24, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dihydroquinoline pyrazolyl compounds
Patent number
9,796,726
Issue date
Oct 24, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Dihydroquinoline pyrazolyl compounds
Patent number
9,790,200
Issue date
Oct 17, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyridinyloxy- and phenyloxy-pyrazolyl compounds
Patent number
9,790,217
Issue date
Oct 17, 2017
Hoffmann-La Roche Inc.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3,4-dihydro-2H-isoquinoline-1-one and 2,3-dihydro-isoindol-1-one co...
Patent number
9,695,152
Issue date
Jul 4, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3,4-dihydro-2H-isoquinoline-1-one and 2,3-dihydro-isoindol-1-one co...
Patent number
9,695,151
Issue date
Jul 4, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Phenyl-dihydropyridine derivatives as inhibitors of aldosterone syn...
Patent number
9,636,338
Issue date
May 2, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Phenyl-dihydropyridine derivatives as aldosterone synthase inhibitors
Patent number
9,636,339
Issue date
May 2, 2017
Hoffman-La Roche Inc.
Johannes Aebi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Dihydroquinoline-2-one derivatives
Patent number
9,593,107
Issue date
Mar 14, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3,4-dihydro-2H-isoquinoline-1-one and 2,3-dihydro-isoindol-1-one co...
Patent number
9,505,742
Issue date
Nov 29, 2016
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazolylketone derivatives
Patent number
9,464,058
Issue date
Oct 11, 2016
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dihydroquinoline-2-one derivatives
Patent number
9,458,135
Issue date
Oct 4, 2016
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic dihydroquinoline-2-one derivatives
Patent number
9,353,081
Issue date
May 31, 2016
Hoffmann-La Roche Inc.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dihydroquinoline-2-one derivatives
Patent number
9,260,408
Issue date
Feb 16, 2016
Hoffmann-La Roche Inc.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Phenyl-tetrahydroisoquinoline derivatives
Patent number
9,187,429
Issue date
Nov 17, 2015
Hoffmann-La Roche Inc.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic dihydroisoquinoline-1-one derivatives
Patent number
9,133,158
Issue date
Sep 15, 2015
Hoffman-La Roche Inc.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,4,5,6-tetrahydro-pyrimidin-2-ylamine compounds
Patent number
8,815,881
Issue date
Aug 26, 2014
Hoffmann-La Roche Inc.
David Banner
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Organic compounds
Patent number
8,367,662
Issue date
Feb 5, 2013
Novartis AG
Duncan Shaw
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
HETEROCYCLIC COMPOUNDS AS MONOACYLGLYCEROL LIPASE INHIBITORS
Publication number
20240150373
Publication date
May 9, 2024
HOFFMANN-LA ROCHE INC.
Charles BELL
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MODIFIED IL-18 POLYPEPTIDES
Publication number
20230357342
Publication date
Nov 9, 2023
Bright Peak Therapeutics AG
Vijaya Raghavan PATTABIRAMAN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC COMPOUNDS
Publication number
20230203056
Publication date
Jun 29, 2023
HOFFMANN-LA ROCHE INC.
Joerg BENZ
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BEZOXAZINE DERIVATIVES USEFUL AS MONOACYLGLYCEROL LIPASE INHIBITORS
Publication number
20230183224
Publication date
Jun 15, 2023
HOFFMANN-LA ROCHE INC.
Charles BELL
C07 - ORGANIC CHEMISTRY
Information
Patent Application
OXAZINE MONOACYLGLYCEROL LIPASE (MAGL) INHIBITORS
Publication number
20230117324
Publication date
Apr 20, 2023
HOFFMANN-LA ROCHE INC.
Charles BELL
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETEROCYCLIC COMPOUNDS AS MONOACYLGLYCEROL LIPASE INHIBITORS
Publication number
20230050901
Publication date
Feb 16, 2023
HOFFMANN-LA ROCHE INC.
Charles BELL
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC COMPOUNDS
Publication number
20220275005
Publication date
Sep 1, 2022
HOFFMANN-LA ROCHE INC.
Uwe GRETHER
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC COMPOUNDS
Publication number
20220267349
Publication date
Aug 25, 2022
HOFFMANN-LA ROCHE INC.
Joerg BENZ
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC COMPOUNDS
Publication number
20220242876
Publication date
Aug 4, 2022
HOFFMANN-LA ROCHE INC.
Carsten KROLL
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FLUORESCENT PROBES FOR MONOACYLGLYCEROL LIPASE (MAGL)
Publication number
20220220373
Publication date
Jul 14, 2022
HOFFMANN-LA ROCHE INC.
Joerg BENZ
G01 - MEASURING TESTING
Information
Patent Application
HETEROCYCLIC MONOACYLGLYCEROL LIPASE (MAGL) INHIBITORS
Publication number
20220213093
Publication date
Jul 7, 2022
HOFFMANN-LA ROCHE INC.
Joerg BENZ
C07 - ORGANIC CHEMISTRY
Information
Patent Application
RADIOLABELED COMPOUNDS
Publication number
20220202963
Publication date
Jun 30, 2022
HOFFMANN-LA ROCHE INC.
Ludovic COLLIN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETEROCYCLIC COMPOUNDS AS INHIBITORS OF MONOACYLGLYCEROL LIPASE (MAGL)
Publication number
20220135591
Publication date
May 5, 2022
HOFFMANN-LA ROCHE INC.
Joerg BENZ
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC COMPOUNDS
Publication number
20220106328
Publication date
Apr 7, 2022
HOFFMANN-LA ROCHE INC.
Joerg BENZ
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MODIFIED IL-18 POLYPEPTIDES AND USES THEREOF
Publication number
20220056091
Publication date
Feb 24, 2022
Bright Peak Therapeutics AG
Vijaya Raghavan PATTABIRAMAN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NEW TRIFLUOROMETHYLPROPANAMIDE DERIVATIVES AS HTRA1 INHIBITORS
Publication number
20190185426
Publication date
Jun 20, 2019
HOFFMANN-LA ROCHE INC.
Benoit HORNSPERGER
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DIFLUOROKETAMIDE DERIVATIVES AS HTRA1 INHIBITORS
Publication number
20190185427
Publication date
Jun 20, 2019
HOFFMANN-LA ROCHE INC.
Benoit Hornsperger
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW DIFLUOROKETAMIDE DERIVATIVES AS HTRAl INHIBITORS
Publication number
20190152895
Publication date
May 23, 2019
HOFFMANN-LA ROCHE INC.
Hans P. MAERKI
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW DIFLUOROKETAMIDE DERIVATIVES
Publication number
20180057526
Publication date
Mar 1, 2018
HOFFMANN-LA ROCHE INC.
Benoit HORNSPERGER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NEW TRIFLUOROMETHYLPROPANAMIDE DERIVATIVES
Publication number
20170348257
Publication date
Dec 7, 2017
HOFFMANN-LA ROCHE INC.
Benoit Hornsperger
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
DIHYDROQUINOLINE PYRAZOLYL COMPOUNDS
Publication number
20170226079
Publication date
Aug 10, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDINYLOXY- AND PHENYLOXY-PYRAZOLYL COMPOUNDS
Publication number
20170226097
Publication date
Aug 10, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DIHYDROQUINOLINE PYRAZOLYL COMPOUNDS
Publication number
20170226085
Publication date
Aug 10, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW DIHYDROQUINOLINE PYRAZOLYL COMPOUNDS
Publication number
20170226116
Publication date
Aug 10, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SPIRODIAMINE DERIVATIVES AS ALDOSTERONE SYNTHASE INHIBITORS
Publication number
20170204107
Publication date
Jul 20, 2017
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW PHENYL-DIHYDROPYRIDINE DERIVATIVES AS ALDOSTERONE SYNTHASE INHI...
Publication number
20160229807
Publication date
Aug 11, 2016
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHENYL-DIHYDROPYRIDINE DERIVATIVES AS INHIBITORS OF ALDOSTERONE SYN...
Publication number
20160221954
Publication date
Aug 4, 2016
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW 3,4-DIHYDRO-2H-ISOQUINOLINE-1-ONE AND 2,3-DIHYDRO-ISOINDOL-1-ON...
Publication number
20160075686
Publication date
Mar 17, 2016
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW 3,4-DIHYDRO-2H-ISOQUINOLINE-1-ONE AND 2,3-DIHYDRO-ISOINDOL-1-O...
Publication number
20160075688
Publication date
Mar 17, 2016
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW 3,4-DIHYDRO-2H-ISOQUINOLINE-1-ONE AND 2,3-DIHYDRO-ISOINDOL-1-O...
Publication number
20160075687
Publication date
Mar 17, 2016
HOFFMANN-LA ROCHE INC.
Johannes Aebi
C07 - ORGANIC CHEMISTRY