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Bruce J. Melancon
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Nashville, TN, US
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Patents Grants
last 30 patents
Information
Patent Grant
Substituted 2-(4-heterocyclylbenzyl)isoindolin-1-one analogs as pos...
Patent number
10,654,847
Issue date
May 19, 2020
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Positive allosteric modulators of the muscarinic acetylcholine rece...
Patent number
10,189,857
Issue date
Jan 29, 2019
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 5-aminothieno[2,3-C]pyridazine-6-carboxamide analogs as...
Patent number
9,868,746
Issue date
Jan 16, 2018
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted thieno[2,3-C]pyridazine-6-carboxamide analogs as positi...
Patent number
9,637,498
Issue date
May 2, 2017
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 2-(4-heterocyclylbenzyl)isoindolin-1-one analogs as pos...
Patent number
9,586,964
Issue date
Mar 7, 2017
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 5-aminothieno[2,3—C]pyridazine-6-carboxamide analogs as...
Patent number
9,493,481
Issue date
Nov 15, 2016
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted benzylspiroindolin-2-one analogs as positive allosteric...
Patent number
9,073,935
Issue date
Jul 7, 2015
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 1H-pyrazolo[3′,4′,4,5]thieno[2,3-b]pyridin-3-amine anal...
Patent number
9,056,876
Issue date
Jun 16, 2015
Vanderbilt University
Jeffrey P. Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 1-benzylindolin-2-one analogs as positive allosteric mo...
Patent number
9,029,563
Issue date
May 12, 2015
Vanderbilt University
Craig W. Lindsley
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted 4-(1H-pyrazol-4-yl)benzyl analogues as positive alloste...
Patent number
9,012,445
Issue date
Apr 21, 2015
Vanderbilt University
Craig W. Lindsley
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted (1-(methylsulfonyl)azetidin-3-yl)(heterocycloalkyl)meth...
Patent number
8,697,888
Issue date
Apr 15, 2014
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Alkyl 3-((2-amidoethyl)amino)-8-azabicyclo[3.2.1]octane-8-carboxyla...
Patent number
8,697,691
Issue date
Apr 15, 2014
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
SUBSTITUTED 2-(4-HETEROCYCLYLBENZYL)ISOINDOLIN-1-ONE ANALOGS AS POS...
Publication number
20200231592
Publication date
Jul 23, 2020
Vanderbilt Unversity
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 2-(4-HETEROCYCLYLBENZYL)ISOINDOLIN-1-ONE ANALOGS AS POS...
Publication number
20180179205
Publication date
Jun 28, 2018
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECE...
Publication number
20180086776
Publication date
Mar 29, 2018
Vanderbilt University
Craig W. Lindsley
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 2-(4-HETEROCYCLYLBENZYL)ISOINDOLIN-1-ONE ANALOGS AS POS...
Publication number
20170129889
Publication date
May 11, 2017
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 5-AMINOTHIENO[2,3-C]PYRIDAZINE-6-CARBOXAMIDE ANALOGS AS...
Publication number
20170022216
Publication date
Jan 26, 2017
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED THIENO[2,3-C]PYRIDAZINE-6-CARBOXAMIDE ANALOGS AS POSITI...
Publication number
20160207935
Publication date
Jul 21, 2016
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED THIENO[2,3-B]PYRIDINE-2-CARBOXAMIDE ANALOGS AS POSITIVE...
Publication number
20160200733
Publication date
Jul 14, 2016
Vanderbilt University
Craig W. LINDSLEY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 5-AMINOTHIENO[2,3-C]PYRIDAZINE-6-CARBOXAMIDE ANALOGS AS...
Publication number
20150018309
Publication date
Jan 15, 2015
Craig W Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 1H-PYRAZOLO[3',4',4,5]THIENO[2,3-B]PYRIDIN-3-AMINE ANAL...
Publication number
20140357615
Publication date
Dec 4, 2014
Jeffrey P. Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 2-(4-HETEROCYCLYLBENZYL)ISOINDOLIN-1-ONE ANALOGS AS POS...
Publication number
20140288084
Publication date
Sep 25, 2014
VANDERBILT UNIVERSITY
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 4-(1H-PYRAZOL-4-YL)BENZYL ANALOGUES AS POSITIVE ALLOSTE...
Publication number
20140206676
Publication date
Jul 24, 2014
Vanderbilt University
Craig W. Lindsley
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 1-BENZYLINDOLIN-2-ONE ANALOGS AS POSITIVE ALLOSTERIC MO...
Publication number
20140194471
Publication date
Jul 10, 2014
Vanderbilt University
Craig W. Lindlsley
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED (1-(METHYLSULFONYL)AZETIDIN-3-YL)(HETEROCYCLOALKYL)METH...
Publication number
20130178458
Publication date
Jul 11, 2013
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BENZYLSPIROINDOLIN-2-ONE ANALOGS AS POSITIVE ALLOSTERIC...
Publication number
20130123236
Publication date
May 16, 2013
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ALKYL 3-((2-AMIDOETHYL)AMINO)-8-AZABICYCLO[3.2.1]OCTANE-8-CARBOXYLA...
Publication number
20110172227
Publication date
Jul 14, 2011
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY