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Colleen M. Niswender
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Brentwood, TN, US
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Patents Grants
last 30 patents
Information
Patent Grant
Indazole compounds as MGLUR4 allosteric potentiators, compositions,...
Patent number
11,427,573
Issue date
Aug 30, 2022
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyridine quinoline compounds as MGLUR4 allosteric potentiators, com...
Patent number
11,319,304
Issue date
May 3, 2022
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Indazole and azaindazole substituted compounds as mGluR4 allosteric...
Patent number
10,526,323
Issue date
Jan 7, 2020
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Indazole compounds as mGluR4 allosteric potentiators, compositions,...
Patent number
10,508,105
Issue date
Dec 17, 2019
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Isoquiniline and napthalene-substituted compounds as mGluR4 alloste...
Patent number
10,227,343
Issue date
Mar 12, 2019
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzothiazole and benzisothiazole-substituted compounds as mGluR4 a...
Patent number
10,221,172
Issue date
Mar 5, 2019
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzoisoxazole-substituted compounds as MGLUR4 allosteric potentiat...
Patent number
9,980,945
Issue date
May 29, 2018
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Heterocyclic sulfone mGluR4 allosteric potentiators, compositions,...
Patent number
9,192,603
Issue date
Nov 24, 2015
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
mGluR4 allosteric potentiators, compositions, and methods of treati...
Patent number
9,180,192
Issue date
Nov 10, 2015
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolopyridine, pyrarolopyrazine, pyrazolopyrimidine, pyrazolothi...
Patent number
9,163,015
Issue date
Oct 20, 2015
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolopyridine, pyrazolopyrazine, pyrazolopyrimidine, pyrazolothi...
Patent number
9,108,963
Issue date
Aug 18, 2015
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzisoxazoles and azabenzisoxazoles as MGLUR4 allosteric potentiat...
Patent number
8,916,584
Issue date
Dec 23, 2014
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Aryl and heteroaryl sulfones as mGluR4 allosteric potentiators, com...
Patent number
8,912,336
Issue date
Dec 16, 2014
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzamide mGluR5 positive allosteric modulators and methods of maki...
Patent number
8,853,392
Issue date
Oct 7, 2014
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
MGLUR4 allosteric potentiators, compositions, and methods of treati...
Patent number
8,779,157
Issue date
Jul 15, 2014
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted dioxopiperidines and dioxopyrrolidines as MGLUR4 allost...
Patent number
8,759,377
Issue date
Jun 24, 2014
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Alkyl 3-((2-amidoethyl)amino)-8-azabicyclo[3.2.1]octane-8-carboxyla...
Patent number
8,697,691
Issue date
Apr 15, 2014
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 1,1,3,1-tetraoxidobenzo[D][1,3,2]dithiazoles as MGLUR4...
Patent number
8,658,650
Issue date
Feb 25, 2014
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic mGluR5 positive allosteric modulators and methods of makin...
Patent number
8,034,806
Issue date
Oct 11, 2011
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
INDAZOLE COMPOUNDS AS MGLUR4 ALLOSTERIC POTENTIATORS, COMPOSITIONS,...
Publication number
20220259190
Publication date
Aug 18, 2022
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INDAZOLE COMPOUNDS AS MGLUR4 ALLOSTERIC POTENTIATORS, COMPOSITIONS,...
Publication number
20200291019
Publication date
Sep 17, 2020
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDINE QUINOLINE COMPOUNDS AS MGLUR4 ALLOSTERIC POTENTIATORS, COM...
Publication number
20200165232
Publication date
May 28, 2020
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INDAZOLE COMPOUNDS AS MGLUR4 ALLOSTERIC POTENTIATORS, COMPOSITIONS,...
Publication number
20190055225
Publication date
Feb 21, 2019
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZOISOXAZOLE-SUBSTITUTED COMPOUNDS AS MGLUR4 ALLOSTERIC POTENTIAT...
Publication number
20180021312
Publication date
Jan 25, 2018
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZOTHIAZOLE AND BENZISOTHIAZOLE-SUBSTITUTED COMPOUNDS AS MGLUR4 A...
Publication number
20180022744
Publication date
Jan 25, 2018
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INDAZOLE AND AZAINDAZOLE SUBSTITUTED COMPOUNDS AS MGLUR4 ALLOSTERIC...
Publication number
20180022746
Publication date
Jan 25, 2018
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ISOQUINILINE AND NAPTHALENE-SUBSTITUTED COMPOUNDS AS MGLUR4 ALLOSTE...
Publication number
20180022745
Publication date
Jan 25, 2018
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MGLUR4 ALLOSTERIC POTENTIATORS, COMPOSITIONS, AND METHODS OF TREATI...
Publication number
20130338154
Publication date
Dec 19, 2013
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETEROCYCLYL-AZABICYCLO[3.2.1]OCTANE ANALOGS AS SELECTIVE M1 AGONI...
Publication number
20130197027
Publication date
Aug 1, 2013
Craig Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Heterocyclic Sulfone MGLUR4 Allosteric Potentiators, Compositions,...
Publication number
20130158078
Publication date
Jun 20, 2013
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Pyrazolopyridine, Pyrazolopyrazine, Pyrazolopyrimidine, Pyrazolothi...
Publication number
20130096110
Publication date
Apr 18, 2013
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Benzisoxazoles and Azabenzisoxazoles as MGLUR4 Allosteric Potentiat...
Publication number
20130079366
Publication date
Mar 28, 2013
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Pyrazolopyridine, Pyrazolopyrazine, Pyrazolopyrimidine, Pyrazolothi...
Publication number
20130065895
Publication date
Mar 14, 2013
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MGLUR4 ALLOSTERIC POTENTIATORS, COMPOSITIONS, AND METHODS OF TREATI...
Publication number
20130040944
Publication date
Feb 14, 2013
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MGLUR4 ALLOSTERIC POTENTIATORS, COMPOSITIONS, AND METHODS OF TREATI...
Publication number
20120245153
Publication date
Sep 27, 2012
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ARYL AND HETEROARYL SULFONES AS MGLUR4 ALLOSTERIC POTENTIATORS, COM...
Publication number
20120245185
Publication date
Sep 27, 2012
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED ENZOIMIDAZOLESULFONAMIDES AND SUBSTITUTED INDOLESULFONA...
Publication number
20120184556
Publication date
Jul 19, 2012
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMIDOBIPIPERIDINECARBOXYLATE M1 ALLOSTERIC AGONISTS, ANALOGS AND DE...
Publication number
20120088791
Publication date
Apr 12, 2012
Vanderbilt University
Craig W. Lindsley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKIN...
Publication number
20120028955
Publication date
Feb 2, 2012
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKIN...
Publication number
20120028956
Publication date
Feb 2, 2012
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 1,1,3,1-TETRAOXIDOBENZO[D][1,3,2]DITHIAZOLES AS MGLUR4...
Publication number
20110319429
Publication date
Dec 29, 2011
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ALKYL 3-((2-AMIDOETHYL)AMINO)-8-AZABICYCLO[3.2.1]OCTANE-8-CARBOXYLA...
Publication number
20110172227
Publication date
Jul 14, 2011
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED DIOXOPIPERIDINES AND DIOXOPYRROLIDINES AS MGLUR4 ALLOST...
Publication number
20110124663
Publication date
May 26, 2011
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKIN...
Publication number
20090270362
Publication date
Oct 29, 2009
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZAMIDE mGluR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKI...
Publication number
20090042855
Publication date
Feb 12, 2009
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE