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Cornelis G. Kruse
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CP Weesp, NL
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Patents Grants
last 30 patents
Information
Patent Grant
Arylsulfonyl pyrazoline carboxamidine derivatives as 5-HT6 antagonists
Patent number
9,126,942
Issue date
Sep 8, 2015
ABBVIE BAHAMAS LIMITED
Arnold van Loevezijn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Arylsulfonyl pyrazoline carboxamidine derivatives as 5-HT6 antagonists
Patent number
8,901,108
Issue date
Dec 2, 2014
AbbVie Bahamas Limited
Arnold Van Loevezijn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Heterocyclic compounds with affinity to muscarinic receptors
Patent number
8,735,388
Issue date
May 27, 2014
AbbVie B.V.
Axel Stoit
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1H-imidazole derivative having CB1, agonistic, CB1 partial agonisti...
Patent number
8,729,101
Issue date
May 20, 2014
Solvay Pharmaceuticals, B.V.
Cornelis G. Kruse
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Sulfonylpyrazole and sulfonylpyrazoline carboxamidine derivatives a...
Patent number
8,722,887
Issue date
May 13, 2014
Abbvie Bahamas, Ltd.
Arnold Van Loevezijn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Heterocyclic compounds with affinity to muscarinic receptors
Patent number
8,586,606
Issue date
Nov 19, 2013
AbbVie B.V.
Axel Stoit
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Arylsulfonyl pyrazoline carboxamidine derivatives as 5-HT6 antagonists
Patent number
8,563,723
Issue date
Oct 22, 2013
Abbott Healthcare Products, B.V.
Arnold Van Loevezijn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Sulphur containing pyrazole derivatives as selective cannabinoid CB...
Patent number
8,461,184
Issue date
Jun 11, 2013
Solvay Pharmaceuticals B.V.
Josephus H. M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Azaindole derivatives with a combination of partial nicotinic acety...
Patent number
8,252,930
Issue date
Aug 28, 2012
Solvay Pharmaceuticals B.V.
Axel Stoit
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds with a combination of cannabinoid CB1 antagonism and sero...
Patent number
8,138,174
Issue date
Mar 20, 2012
Solvay Pharmaceuticals B.V.
Josephus H. M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Phenylpiperazine derivatives with a combination of partial dopamine...
Patent number
8,101,619
Issue date
Jan 24, 2012
Solvay Pharmaceuticals B.V.
Roelof W. Feenstra
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic compounds with affinity to muscarinic receptors
Patent number
8,084,473
Issue date
Dec 27, 2011
Solvay Pharmaceuticals B.V.
Axel Stoit
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds with a combination of cannabinoid-CB1 antagonism and acet...
Patent number
8,063,062
Issue date
Nov 22, 2011
Solvay Pharmaceuticals B.V.
Josephus H. M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Azaindole derivatives with a combination of partial nicotinic acety...
Patent number
7,964,728
Issue date
Jun 21, 2011
Solvay Pharmaceuticals B.V.
Axel Stoit
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Sulphur containing pyrazole derivatives as selective cannabinoid CB...
Patent number
7,786,144
Issue date
Aug 31, 2010
Solvay Pharmaceuticals B.V.
Josephus H. M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperazine and piperidine compounds
Patent number
RE41425
Issue date
Jul 6, 2010
Duphar International Research B.V.
Roelof Willem Feenstra
544 - Organic compounds
Information
Patent Grant
1,3,5-trisubstituted 4,5-dihydro-1H-pyrazole derivatives having CB1...
Patent number
7,745,476
Issue date
Jun 29, 2010
Solvay Pharmaceuticals B.V.
Josephus H. M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Sulfonylpyrazole and sulfonylpyrazoline carboxamidine derivatives a...
Patent number
7,728,018
Issue date
Jun 1, 2010
Solvay Pharmaceuticals B.V.
Arnold Van Loevezijn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
N-oxides of venlafaxine and o-desmethylvenlafaxine as prodrugs
Patent number
7,696,383
Issue date
Apr 13, 2010
Solvay Pharmaceuticals B.V.
Lechoslaw A. Turski
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
4,5-dihydro-1H-pyrazole derivatives having potent CB1-antagonistic...
Patent number
7,608,718
Issue date
Oct 27, 2009
Solvay Pharmaceuticals B.V.
Josephus H. M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Phenylpiperazine
Patent number
7,605,162
Issue date
Oct 20, 2009
Solvay Pharmaceuticals
Roelof Van Hes
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity
Patent number
7,528,162
Issue date
May 5, 2009
Solvay Pharmaceuticals, B.V.
Cornelis G. Kruse
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tetrasubstituted imidazole derivatives as cannabinoid CB1 receptor...
Patent number
7,524,867
Issue date
Apr 28, 2009
Solvay Pharmaceuticals, B.V.
Josephus H. M Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1 H-imidazole derivatives as cannabinoid receptor modulators
Patent number
7,498,348
Issue date
Mar 3, 2009
Solvay Pharmaceuticals, Inc.
Josephus H. M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazoline derivatives having CB1-antagonistic activity
Patent number
7,495,108
Issue date
Feb 24, 2009
Solvay Pharmaceuticals, B.V.
Josephus H. M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Phenylpiperazines
Patent number
7,456,182
Issue date
Nov 25, 2008
Solvay Pharmaceuticals, Inc.
Roelof Van Hes
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tetrahydropyridin-4-yl indoles with a combination of affinity for d...
Patent number
7,371,769
Issue date
May 13, 2008
Solvay Pharmaceuticals B.V.
Roelof van Hes
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Thiazole derivatives having CB1-antagonistic, agonistic or partial...
Patent number
7,342,032
Issue date
Mar 11, 2008
Solvay Pharmaceuticals, Inc.
Josephus H. M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1H-1,2,4-triazole-3-carboxamide derivatives having cannabinoid-CB1...
Patent number
7,319,110
Issue date
Jan 15, 2008
Solvay Pharmaceuticals B.V.
Josephus H. M. Lange
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Piperazine and piperidine compounds
Patent number
7,297,699
Issue date
Nov 20, 2007
Solvay Pharmaceuticals, Inc.
Roelof W. Feenstra
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
SULFONYLPYRAZOLE AND SULFONYLPYRAZOLINE CARBOXAMIDINE DERIVATIVES A...
Publication number
20140303372
Publication date
Oct 9, 2014
ABBVIE BHAMAS LTD.
Arnold Van Loevezijn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETEROCYCLIC COMPOUNDS IWTH AFFINITY TO MUSCARINIC RECEPTORS
Publication number
20140080861
Publication date
Mar 20, 2014
ABBVIE B.V.A
Axel Stoit
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ARYLSULFONYL PYRAZOLINE CARBOXAMIDINE DERIVATIVES AS 5-HT6 ANTAGONISTS
Publication number
20140011775
Publication date
Jan 9, 2014
ABBOTT HEALTHCARE PRODUCTS B.V.
Arnold van Loevezijn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETEROCYCLIC COMPOUNDS WITH AFFINITY TO MUSCARINIC RECEPTORS
Publication number
20120095039
Publication date
Apr 19, 2012
Solvay Pharmaceuticals B.V.
Axel Stoit
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AZAINDOLE DERIVATIVES WITH A COMBINATION OF PARTIAL NICOTINIC ACETY...
Publication number
20110053962
Publication date
Mar 3, 2011
Solvay Pharmaceuticals B.V.
Axel Stoit
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ARYLSULFONYL PYRAZOLINE CARBOXAMIDINE DERIVATIVES AS 5-HT6 ANTAGONISTS
Publication number
20110046171
Publication date
Feb 24, 2011
Arnold Van Loevezijn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SULPHUR CONTAINING PYRAZOLE DERIVATIVES AS SELECTIVE CANNABINOID CB...
Publication number
20100292204
Publication date
Nov 18, 2010
Solvay Pharmaceuticals, B.V.
Josephus H.M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SULFONYLPYRAZOLE AND SULFONYLPYRAZOLINE CARBOXAMIDINE DERIVATIVES A...
Publication number
20100145042
Publication date
Jun 10, 2010
Solvay Pharmaceuticals B.V.
Arnold Van Loevezijn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MUSCARINIC AGONISTS TO TREAT IMPULSE CONTROL DISORDERS
Publication number
20100120752
Publication date
May 13, 2010
Solvay Pharmaceuticals, B.V.
Natasja M.W.J. De Bruin
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
1H-IMIDAZOLE DERIVATIVE HAVING CB1, AGONISTIC, CB1 PARTIAL AGONISTI...
Publication number
20090181949
Publication date
Jul 16, 2009
Solvay Pharmaceuticals B.V.
Cornelis G. KRUSE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
New Phenylpiperazine
Publication number
20090143406
Publication date
Jun 4, 2009
Solvay Pharmaceuticals, Inc.
Roelof Van Hes
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Heterocyclic Compounds with Affinity to Muscarinic Receptors
Publication number
20090018160
Publication date
Jan 15, 2009
Axel Stoit
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
N-OXIDES OF VENLAFAXINE AND O-DESMETHYLVENLAFAXINE AS PRODRUGS
Publication number
20090005455
Publication date
Jan 1, 2009
Solvay Pharmaceuticals, B.V.
Lechoslaw A. Turski
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SILDENAFIL N-OXIDE AS PRODRUG
Publication number
20090005395
Publication date
Jan 1, 2009
Solvay Pharmaceuticals, B.V.
Lechoslaw A. Turski
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SULFONYLPYRAZOLE AND SULFONYLPYRAZOLINE CARBOXAMIDINE DERIVATIVES A...
Publication number
20080311179
Publication date
Dec 18, 2008
Arnold Van Loevezijn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS WITH A COMBINATION OF CANNABINOID CB1 ANTAGONISM AND SERO...
Publication number
20080214559
Publication date
Sep 4, 2008
Solvay Pharmaceuticals B.V.
Josephus H.M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Application
USE OF 5-HT6 ANTAGONISTS TO PREVENT RELAPSE INTO ADDICTION
Publication number
20080171779
Publication date
Jul 17, 2008
Solvay Pharmaceuticals B.V.
Natasja M.W.J. De Bruin
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS WITH A COMBINATION OF CANNABINOID-CB1 ANTAGONISM AND ACET...
Publication number
20080153867
Publication date
Jun 26, 2008
Solvay Pharmaceuticals B.V.
Josephus H.M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Selective inhibitors of neurotensin degrading enzymes
Publication number
20080146524
Publication date
Jun 19, 2008
Solvay Pharmaceuticals B.V.
Pieter Smid
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AZAINDOLE DERIVATIVES WITH A COMBINATION OF PARTIAL NICOTINIC ACETY...
Publication number
20080009514
Publication date
Jan 10, 2008
Axel STOIT
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SULPHUR CONTAINING PYRAZOLE DERIVATIVES AS SELECTIVE CANNABINOID CB...
Publication number
20070281973
Publication date
Dec 6, 2007
Josephus H.M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1 H-IMIDAZOLE DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS
Publication number
20070281974
Publication date
Dec 6, 2007
Solvay Pharmaceuticals, Inc.
Josephus H.M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MUSCARINIC AGONISTS TO TREAT IMPULSE CONTROL DISORDERS
Publication number
20070259859
Publication date
Nov 8, 2007
Natasja M.W.J. De Bruin
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
4,5-Dihydro-1H-pyrazole derivatives having potent CB1-antagonistic...
Publication number
20070259884
Publication date
Nov 8, 2007
Solvay Pharmaceuticals B.V.
Josephus H.M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHENYPIPERAZINE DERIVATIVES WITH A COMBINATION OF PARTIAL DOPAMINE-...
Publication number
20070142397
Publication date
Jun 21, 2007
SOLVAY PHARMECEUTICALS B.V.
Roelof W. Feenstra
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Imidazoline derivatives having CB1-antagonistic activity
Publication number
20070135492
Publication date
Jun 14, 2007
Solvay Pharmaceuticals, B.V,.
Josephus H.M. Lange
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHENYLPIPERAZINE DERIVATIVES WITH A COMBINATION OF PARTIAL DOPAMINE...
Publication number
20070072870
Publication date
Mar 29, 2007
SOLVAY PHARMECEUTICALS B.V.
Roelof Feenstra
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TETRAHYDROPYRIDIN-4-YL INDOLES WITH A COMBINATION OF AFFINITY FOR D...
Publication number
20070066634
Publication date
Mar 22, 2007
SOLVAY PHARMECEUTICALS B.V.
Roelof van Hes
C07 - ORGANIC CHEMISTRY
Information
Patent Application
New phenylpiperazines
Publication number
20060293313
Publication date
Dec 28, 2006
Solvay Pharmaceuticals, B.V.
Roelof Van Hes
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Phenylpiperazine derivatives with a combination of partial dopamine...
Publication number
20060247256
Publication date
Nov 2, 2006
Solvay Pharmaceuticals B.V.
Roelof W. Feenstra
C07 - ORGANIC CHEMISTRY