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David S. Weinstein
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East Windsor, NJ, US
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Patents Grants
last 30 patents
Information
Patent Grant
Sulfone pyridine alkyl amide-substituted heteroaryl compounds
Patent number
11,787,779
Issue date
Oct 17, 2023
Bristol-Myers Squibb Company
Chunjian Liu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cereblon modulators and uses thereof
Patent number
11,771,689
Issue date
Oct 3, 2023
VIVIDION THERAPEUTICS, INC.
Benjamin F. Cravatt
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Heterocyclic compounds comprising pyridine useful as modulators of...
Patent number
11,597,721
Issue date
Mar 7, 2023
Bristol-Myers Squibb Company
Zili Xiao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted imidazo[1,2-b]pyridazines as interleukin-23 and interfe...
Patent number
11,299,494
Issue date
Apr 12, 2022
Bristol-Myers Squibb Company
David S. Weinstein
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Sulfone pyridine alkyl amide-substituted heteroaryl compounds
Patent number
11,021,462
Issue date
Jun 1, 2021
Bristol-Myers Squibb Company
Chunjian Liu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Amide-substituted heterocyclic compounds useful as modulators of IL...
Patent number
11,021,475
Issue date
Jun 1, 2021
Bristol-Myers Squibb Company
Ryan M. Moslin
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cereblon modulators and uses thereof
Patent number
10,869,860
Issue date
Dec 22, 2020
VIVIDION THERAPEUTICS, INC.
Benjamin F. Cravatt
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
In vivo engineered cereblon protein
Patent number
10,781,239
Issue date
Sep 22, 2020
VIVIDION THERAPEUTICS, INC.
David Weinstein
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterobicyclic compounds useful as modulators of IL-12, IL-23 and/o...
Patent number
10,781,215
Issue date
Sep 22, 2020
Bristol-Myers Squibb Company
Stephen T. Wrobleski
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Amide-substituted heterocyclic compounds useful as modulators of IL...
Patent number
RE47929
Issue date
Apr 7, 2020
Bristol-Myers Squibb Company
Ryan M. Moslin
Information
Patent Grant
Imidazopyridazine compounds useful as modulators of IL-12, IL-23 an...
Patent number
10,479,793
Issue date
Nov 19, 2019
Bristol-Myers Squibb Company
David S. Weinstein
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Phosphine oxide alkyl amide substituted heteroaryl compounds as mod...
Patent number
10,294,256
Issue date
May 21, 2019
Bristol-Myers Squibb Company
Michael G. Yang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazopyridazine compounds useful as modulators of IL-12, IL-23 an...
Patent number
10,273,237
Issue date
Apr 30, 2019
Bristol-Myers Squibb Company
Chunjian Liu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Amide-substituted heterocyclic compounds useful as modulators of IL...
Patent number
10,000,480
Issue date
Jun 19, 2018
Bristol-Myers Squibb Company
Ryan M. Moslin
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Alkyl-amide-substituted pyridyl compounds useful as modulators of I...
Patent number
9,987,266
Issue date
Jun 5, 2018
Bristol-Myers Squibb Company
Ryan M. Moslin
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Imidazole-derived modulators of the glucocorticoid receptor
Patent number
9,796,720
Issue date
Oct 24, 2017
Bristol-Myers Squibb Company
Michael G. Yang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
RORγ modulators
Patent number
9,725,443
Issue date
Aug 8, 2017
Bristol-Myers Squibb Company
T. G. Murali Dhar
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
RORγ modulators
Patent number
9,663,469
Issue date
May 30, 2017
Bristol-Myers Squibb Company
T. G. Murali Dhar
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Alkyl-amide-substituted pyridyl compounds useful as modulators of I...
Patent number
9,663,467
Issue date
May 30, 2017
Bristol-Myers Squibb Company
Ryan M. Moslin
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imide and acylurea derivatives as modulators of the glucocorticoid...
Patent number
9,593,113
Issue date
Mar 14, 2017
Bristol-Myers Squibb Company
David S. Weinstein
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Alkyl amide-substituted pyrimidine compounds useful in the modulati...
Patent number
9,540,333
Issue date
Jan 10, 2017
Bristol-Myers Squibb Company
Joseph B. Santella
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Amide-substituted heterocyclic compounds useful as modulators of IL...
Patent number
9,505,748
Issue date
Nov 29, 2016
Bristol-Myers Squibb Company
Ryan M. Moslin
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Alkyl-amide-substituted pyridyl compounds useful as modulators of I...
Patent number
9,315,494
Issue date
Apr 19, 2016
Bristol-Myers Squibb Company
Ryan M. Moslin
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Fused heteroaryl modulators of glucocorticoid receptor, AP-1, and/o...
Patent number
8,304,539
Issue date
Nov 6, 2012
Bristol-Myers Squibb Company
Jingwu Duan
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity...
Patent number
8,034,940
Issue date
Oct 11, 2011
Bristol-Myers Squibb Company
David S. Weinstein
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity,...
Patent number
7,888,381
Issue date
Feb 15, 2011
Bristol-Myers Squibb Company
Jingwu Duan
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic modulators of the glucocorticoid receptor, AP-1, and/o...
Patent number
7,605,264
Issue date
Oct 20, 2009
Bristol-Myers Squibb Company
David S. Weinstein
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tricyclic modulators of the glucocorticoid receptor, AP-1, and/or N...
Patent number
7,544,808
Issue date
Jun 9, 2009
Bristol-Myers Squibb Company
David S. Weinstein
A23 - FOODS OR FOODSTUFFS THEIR TREATMENT, NOT COVERED BY OTHER CLASSES
Information
Patent Grant
Benzoxazole inhibitors of 15-lipoxygenase
Patent number
7,534,804
Issue date
May 19, 2009
Bristol-Myers Squibb Company
David S. Weinstein
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolyl inhibitors of 15-lipoxygenase
Patent number
7,432,271
Issue date
Oct 7, 2008
Bristol-Myers Squibb Company
Khehyong Ngu
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
PHARMACEUTICAL COMPOSITIONS COMPRISING WRN HELICASE INHIBITORS
Publication number
20240140915
Publication date
May 2, 2024
Vividion Therapeutics, Inc.
Shota Kikuchi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PHARMACEUTICAL COMPOSITIONS COMPRISING WRN HELICASE INHIBITORS
Publication number
20240067612
Publication date
Feb 29, 2024
Vividion Therapeutics, Inc.
Shota Kikuchi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SULFONE PYRIDINE ALKYL AMIDE-SUBSTITUTED HETEROARYL COMPOUNDS
Publication number
20240002364
Publication date
Jan 4, 2024
Bristol-Myers Squibb Company
Chunjian Liu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PRODRUGS IN THE MODULATION OF INTERLEUKIN
Publication number
20230167082
Publication date
Jun 1, 2023
Bristol-Myers Squibb Company
Ryan M. Moslin
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-(METHYL-D3)PYRIDAZINE-3-CARBOXAMIDE OR N-(METHYL-D3)-...
Publication number
20230167092
Publication date
Jun 1, 2023
Bristol-Myers Squibb Company
Chunjian Liu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMIDE-SUBSTITUTED HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF IL...
Publication number
20220356180
Publication date
Nov 10, 2022
Bristol-Myers Squibb Company
Ryan M. Moslin
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IN VIVO ENGINEERED CEREBLON PROTEIN
Publication number
20220298213
Publication date
Sep 22, 2022
Vividion Therapeutics, Inc.
David WEINSTEIN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CEREBLON MODULATORS AND USES THEREOF
Publication number
20220062248
Publication date
Mar 3, 2022
Vividion Therapeutics, Inc.
Benjamin F. CRAVATT
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMIDAZOPYRIDAZINE COMPOUNDS
Publication number
20210323966
Publication date
Oct 21, 2021
Bristol-Myers Squibb Company
David S. WEINSTEIN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SULFONE PYRIDINE ALKYL AMIDE-SUBSTITUTED HETEROARYL COMPOUNDS
Publication number
20210253554
Publication date
Aug 19, 2021
Bristol-Myers Squibb Company
Chunjian Liu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETEROCYCLIC COMPOUNDS COMPRISING PYRIDINE USEFUL AS MODULATORS OF...
Publication number
20210032220
Publication date
Feb 4, 2021
Bristol-Myers Squibb Company
Zili Xiao
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IN VIVO ENGINEERED CEREBLON PROTEIN
Publication number
20210002337
Publication date
Jan 7, 2021
Vividion Therapeutics, Inc.
David WEINSTEIN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IN VIVO ENGINEERED CEREBLON PROTEIN
Publication number
20200216507
Publication date
Jul 9, 2020
Vividion Therapeutics, Inc.
David WEINSTEIN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CEREBLON MODULATORS AND USES THEREOF
Publication number
20200206201
Publication date
Jul 2, 2020
Vividion Therapeutics, Inc.
Benjamin F. CRAVATT
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMIDE-SUBSTITUTED HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF IL...
Publication number
20200071315
Publication date
Mar 5, 2020
Bristol-Myers Squibb Company
Ryan M. Moslin
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROBICYCLIC COMPOUNDS USEFUL AS MODULATORS OF IL-12, IL-23 AND/O...
Publication number
20190322672
Publication date
Oct 24, 2019
Bristol-Myers Squibb Company
Stephen T. Wrobleski
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SULFONE PYRIDINE ALKYL AMIDE-SUBSTITUTED HETEROARYL COMPOUNDS
Publication number
20190152948
Publication date
May 23, 2019
Bristol-Myers Squibb Company
Chunjian Liu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDAZOPYRIDAZINE COMPOUNDS USEFUL AS MODULATORS OF IL-12, IL-23 AN...
Publication number
20180325899
Publication date
Nov 15, 2018
Bristol-Myers Squibb Company
David S. Weinstein
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMIDE-SUBSTITUTED HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF IL...
Publication number
20180265504
Publication date
Sep 20, 2018
Bristol-Myers Squibb Company
Ryan M. Moslin
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHOSPHINE OXIDE ALKYL AMIDE SUBSTITUTED HETEROARYL COMPOUNDS AS MOD...
Publication number
20180162889
Publication date
Jun 14, 2018
Bristol-Myers Squibb Company
Michael G. YANG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ALKYL-AMIDE-SUBSTITUTED PYRIDYL COMPOUNDS USEFUL AS MODULATORS OF I...
Publication number
20170209426
Publication date
Jul 27, 2017
Bristol-Myers Squibb Company
Ryan M. Moslin
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMIDE-SUBSTITUTED HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF IL...
Publication number
20170022192
Publication date
Jan 26, 2017
Bristol-Myers Squibb Company
Ryan M. Moslin
C07 - ORGANIC CHEMISTRY
Information
Patent Application
RORy MODULATORS
Publication number
20160318870
Publication date
Nov 3, 2016
Bristol-Myers Squibb Company
T.G Murali Dhar
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDAZOPYRIDAZINE COMPOUNDS USEFUL AS MODULATORS OF IL-12, IL-23 AN...
Publication number
20160304524
Publication date
Oct 20, 2016
Bristol-Myers Squibb Company
Chunjian Liu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ALKYL-AMIDE-SUBSTITUTED PYRIDYL COMPOUNDS USEFUL AS MODULATORS OF I...
Publication number
20160280649
Publication date
Sep 29, 2016
Bristol-Myers Squibb Company
Ryan M. MOSLIN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
RORgamma MODULATORS
Publication number
20160229844
Publication date
Aug 11, 2016
Bristol-Myers Squibb Company
T. G. Murali Dhar
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDAZOLE-DERIVED MODULATORS OF THE GLUCOCORTICOID RECEPTOR
Publication number
20160200728
Publication date
Jul 14, 2016
Bristol-Myers Squibb Company
Michael G. Yang
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDE AND ACYLUREA DERIVATIVES AS MODULATORS OF THE GLUCOCORTICOID...
Publication number
20160185776
Publication date
Jun 30, 2016
Bristol-Myers Squibb Company
David S. Weinstein
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ALKYL-AMIDE-SUBSTITUTED PYRIDYL COMPOUNDS USEFUL AS MODULATORS OF I...
Publication number
20150307483
Publication date
Oct 29, 2015
Bristol-Myers Squibb Company
Ryan M. Moslin
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ALKYL AMIDE-SUBSTITUTED PYRIMIDINE COMPOUNDS USEFUL IN THE MODULATI...
Publication number
20150299139
Publication date
Oct 22, 2015
Bristol-Myers Squibb Company
Joseph B. Santella
C07 - ORGANIC CHEMISTRY