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David Siesel
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San Diego, CA, US
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Patents Grants
last 30 patents
Information
Patent Grant
Process of making CFTR modulators
Patent number
12,122,788
Issue date
Oct 22, 2024
Vertex Pharmaceuticals Incorporated
Paul Angell
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Process of making CFTR modulators
Patent number
11,584,761
Issue date
Feb 21, 2023
Vertex Pharmaceuticals Incorporated
Paul Angell
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Processes for making modulators of cystic fibrosis transmembrane co...
Patent number
11,465,985
Issue date
Oct 11, 2022
Vertex Pharmaceuticals Incorporated
Paul T. Angell
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Modulator of the cystic fibrosis transmembrane conductance regulato...
Patent number
11,453,655
Issue date
Sep 27, 2022
Vertex Pharmaceuticals Incorporated
Alexander Russell Abela
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Processes for preparing ATR inhibitors
Patent number
10,822,331
Issue date
Nov 3, 2020
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Modulator of the cystic fibrosis transmembrane conductance regulato...
Patent number
10,793,547
Issue date
Oct 6, 2020
Vertex Pharmaceuticals Incorporated
Alexander Russell Abela
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Modulator of cystic fibrosis transmembrane conductance regulator, p...
Patent number
10,570,115
Issue date
Feb 25, 2020
Vertex Pharmaceuticals Incorporated
Timothy Alcacio
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Processes for preparing ATR inhibitors
Patent number
10,435,397
Issue date
Oct 8, 2019
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Processes for preparing ATR inhibitors
Patent number
10,208,027
Issue date
Feb 19, 2019
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Process of producing cycloalkylcarboxamido-indole compounds
Patent number
10,071,979
Issue date
Sep 11, 2018
Vertex Pharmaceuticals Incorporated
Gerald J. Tanoury
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Processes for making compounds useful as inhibitors of ATR kinase
Patent number
9,862,709
Issue date
Jan 9, 2018
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Processes for producing cycloalkylcarboxamido-pyridine benzoic acids
Patent number
9,776,968
Issue date
Oct 3, 2017
Vertex Pharmaceuticals Incorporated
David Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Processes for making compounds useful as inhibitors of ATR kinase
Patent number
9,035,053
Issue date
May 19, 2015
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Process of producing cycloalkylcarboxamido-indole compounds
Patent number
9,035,072
Issue date
May 19, 2015
Vertex Pharmaceuticals Incorporated
Daniel T. Belmont
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Processes for producing cycloalkylcarboxamido-pyridine benzoic acids
Patent number
9,012,652
Issue date
Apr 21, 2015
Vertex Pharmaceuticals Incorporated
David Andrew Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
8,846,686
Issue date
Sep 30, 2014
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Processes for producing cycloalkylcarboxamido-pyridine benzoic acids
Patent number
8,816,093
Issue date
Aug 26, 2014
Vertex Pharmaceuticals Incorporated
David Andrew Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Processes for producing cycloalkylcarboxamido-pyridine benzoic acids
Patent number
8,592,602
Issue date
Nov 26, 2013
Vertex Pharmaceuticals Incorporated
David Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Processes for producing cycloalkylcarboxamido-pyridine benzoic acids
Patent number
8,461,342
Issue date
Jun 11, 2013
Vertex Pharmaceuticals Incorporated
David Andrew Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Processes for producing cycloalkylcarboxamido-pyridine benzoic acids
Patent number
8,124,781
Issue date
Feb 28, 2012
Vertex Pharmaceuticals Incorporated
David Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted benzimidazoles and methods of preparation
Patent number
7,767,820
Issue date
Aug 3, 2010
Novartis Vaccines and Diagnostics, Inc.
Martin Dimitroff
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CO...
Publication number
20240025877
Publication date
Jan 25, 2024
VERTEX PHARMACEUTICALS INCORPORATED
Paul T. Angell
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESS OF MAKING CFTR MODULATORS
Publication number
20230399343
Publication date
Dec 14, 2023
VERTEX PHARMACEUTICALS INCORPORATED
Paul Angell
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MODULATOR OF THE CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATO...
Publication number
20230357191
Publication date
Nov 9, 2023
Vertex Pharmaceuticals Incorporated
Alexander Russell Abela
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CO...
Publication number
20210246117
Publication date
Aug 12, 2021
VERTEX PHARMACEUTICALS INCORPORATED
Paul T. Angell
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESS OF PRODUCING CYCLOALKYLCARBOXAMIDO-INDOLE COMPOUNDS
Publication number
20210238158
Publication date
Aug 5, 2021
VERTEX PHARMACEUTICALS INCORPORATED
Gerald J. Tanoury
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESS OF MAKING CFTR MODULATORS
Publication number
20210047345
Publication date
Feb 18, 2021
VERTEX PHARMACEUTICALS INCORPORATED
Paul Angell
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MODULATOR OF THE CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATO...
Publication number
20210047295
Publication date
Feb 18, 2021
VERTEX PHARMACEUTICALS INCORPORATED
Alexander Russell Abela
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PROCESS OF PRODUCING CYCLOALKYLCARBOXAMIDO-INDOLE COMPOUNDS
Publication number
20190210991
Publication date
Jul 11, 2019
VERTEX PHARMACEUTICALS INCORPORATED
Gerald J. Tanoury
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR PREPARING ATR INHIBITORS
Publication number
20190202818
Publication date
Jul 4, 2019
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR PREPARING ATR INHIBITORS
Publication number
20180244662
Publication date
Aug 30, 2018
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Modulator of the Cystic Fibrosis Transmembrane Conductance Regulato...
Publication number
20180162839
Publication date
Jun 14, 2018
VERTEX PHARMACEUTICALS INCORPORATED
Alexander Russell Abela
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Modulator of Cystic Fibrosis Transmembrane Conductance Regulator, P...
Publication number
20180093969
Publication date
Apr 5, 2018
Vertex Pharmaceuticals Incorporated
Timothy Alcacio
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
Publication number
20170158676
Publication date
Jun 8, 2017
VERTEX PHARMACEUTICALS INCORPORATED
David Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
Publication number
20160200712
Publication date
Jul 14, 2016
VERTEX PHARMACEUTICALS INCORPORATED
David Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR MAKING COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20150274710
Publication date
Oct 1, 2015
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Process of Producing Cycloalkylcarboxamido-indole Compounds
Publication number
20150218122
Publication date
Aug 6, 2015
VERTEX PHARMACEUTICALS INCORPORATED
Gerald J. Tanoury
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
Publication number
20140330023
Publication date
Nov 6, 2014
David Andrew Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
Publication number
20140121379
Publication date
May 1, 2014
Vertex Pharmaceuticals Incorporated.
David Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESS OF PRODUCING CYCLOALKYLCARBOXAMIDO-INDOLE COMPOUNDS
Publication number
20130324743
Publication date
Dec 5, 2013
Vertex Pharmaceuticals Incorporated.
Daniel T. Belmont
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
Publication number
20130274477
Publication date
Oct 17, 2013
Vertex Pharmaceuticals Incorporated.
David Andrew Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Processes for Making Compounds Useful as Inhibitors of ATR Kinase
Publication number
20130184292
Publication date
Jul 18, 2013
Vertex Pharmaceuticals Incorporated.
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Compounds Useful as Inhibitors of ATR Kinase
Publication number
20130089625
Publication date
Apr 11, 2013
Vertex Pharmaceuticals Incorporated.
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
Publication number
20120203006
Publication date
Aug 9, 2012
Vertex Pharmaceuticals Incorporated.
David Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
Publication number
20120190856
Publication date
Jul 26, 2012
Vertex Pharmaceuticals Incorporated.
David Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BENZIMIDAZOLES AND METHODS OF PREPARATION
Publication number
20100256375
Publication date
Oct 7, 2010
Novartis Vaccines and Diagnostics, Inc.
Martin Dimitroff
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
Publication number
20100036130
Publication date
Feb 11, 2010
Vertex Pharmaceuticals Incorporated.
David Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR PRODUCING CYCLOALKYLCARBOXAMIDO-PYRIDINE BENZOIC ACIDS
Publication number
20090176989
Publication date
Jul 9, 2009
David Siesel
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Substituted benzimidazoles and methods of preparation
Publication number
20080287682
Publication date
Nov 20, 2008
Novartis AG
Martin Dimitroff
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Substituted benzimidazoles and methods of preparation
Publication number
20070049622
Publication date
Mar 1, 2007
Novartis AG
Martin Dimitroff
C07 - ORGANIC CHEMISTRY