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Patents Grants
last 30 patents
Information
Patent Grant
C5A receptor modulators
Patent number
11,739,070
Issue date
Aug 29, 2023
IDORSIA PHARMACEUTICALS LTD
Sylvie Froidevaux
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted tetrahydropyrazolo[3,4-d]pyrimidines and tetrahydropyra...
Patent number
11,608,341
Issue date
Mar 21, 2023
IDORSIA PHARMACEUTICALS LTD
Sylvie Froidevaux
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Indole carboxamide derivatives as P2X7 receptor antagonist
Patent number
9,718,774
Issue date
Aug 1, 2017
IDORSIA PHARMACEUTICALS LTD
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Indole carboxamide derivatives as P2X7 receptor antagonists
Patent number
9,556,117
Issue date
Jan 31, 2017
Actelion Pharmaceuticals Ltd.
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic amide derivatives as P2X7 receptor antagonists
Patent number
9,409,917
Issue date
Aug 9, 2016
Actelion Pharmaceuticals Ltd.
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic amide derivatives as P2X7 receptor antagonists
Patent number
9,388,197
Issue date
Jul 12, 2016
Actelion Pharmaceuticals Ltd.
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic amide derivatives as P2X7 receptor antagonists
Patent number
9,388,198
Issue date
Jul 12, 2016
Actelion Pharmaceuticals Ltd.
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic amide derivatives as P2X7 receptor antagonists
Patent number
9,221,832
Issue date
Dec 29, 2015
Actelion Pharmaceuticals Ltd.
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Thiazole derivatives and their use as P2Y12 receptor antagonists
Patent number
8,664,203
Issue date
Mar 4, 2014
Actelion Pharmaceuticals Ltd.
Eva Caroff
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Alternative heterocycles for DNA recognition
Patent number
8,524,899
Issue date
Sep 3, 2013
California Institute of Technology
Peter B. Dervan
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Phosphonic acid derivates and their use as P2Y12 receptor antagonists
Patent number
8,518,912
Issue date
Aug 27, 2013
Actelion Pharmaceuticals Ltd.
Eva Caroff
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Salts of isobutyric acid (1 R*, 2R*, 4R*)-2-(2-{[3-(4,7-dimethoxy-1...
Patent number
8,492,555
Issue date
Jul 23, 2013
Actelion Pharmaceuticals Ltd.
Stefan Abele
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tetrahydronaphthalene compounds
Patent number
8,436,205
Issue date
May 7, 2013
Actelion Pharmaceuticals Ltd.
Kurt Hilpert
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bridged tetrahydronaphthalene derivatives
Patent number
8,314,253
Issue date
Nov 20, 2012
Actelion Pharmaceuticals Ltd.
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-(3-aza-bicyclo[3.1.0]hex-3-yl)-2-phenyl-pyrimidines
Patent number
8,288,385
Issue date
Oct 16, 2012
Actelion Pharmaceuticals Ltd.
Eva Caroff
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bridged six-membered ring compounds
Patent number
8,202,885
Issue date
Jun 19, 2012
Actelion Pharmaceuticals Ltd.
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 2-phenyl-pyridine derivatives
Patent number
8,058,263
Issue date
Nov 15, 2011
Actelion Pharmaceuticals Ltd.
Eva Caroff
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
2,4,6,7-TETRAHYDRO-PYRAZOLO[4,3-D]PYRIMIDIN-5-ONE DERIVATIVES AND R...
Publication number
20230192708
Publication date
Jun 22, 2023
IDORSIA PHARMACEUTICALS LTD
Sylvie FROIDEVAUX
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHARMACEUTICAL COMPOSITION COMPRISING A TETRAHYDROPYRAZOLOPYRIMIDIN...
Publication number
20220265658
Publication date
Aug 25, 2022
IDORSIA PHARMACEUTICALS LTD
Michael AMBUEHL
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2,4,6,7-TETRAHYDRO-PYRAZOLO[4,3-D]PYRIMIDIN-5-ONE DERIVATIVES AND R...
Publication number
20200369672
Publication date
Nov 26, 2020
IDORSIA PHARMACEUTICALS LTD
Sylvie FROIDEVAUX
C07 - ORGANIC CHEMISTRY
Information
Patent Application
C5A RECEPTOR MODULATORS
Publication number
20200347029
Publication date
Nov 5, 2020
IDORSIA PHARMACEUTICALS LTD
Sylvie FROIDEVAUX
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC AMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS
Publication number
20150361096
Publication date
Dec 17, 2015
Actelion Pharmaceutical Ltd.
KURT HILPERT
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC AMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS
Publication number
20150361097
Publication date
Dec 17, 2015
Actelion Pharmaceuticals LTD
KURT HILPERT
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INDOLE CARBOXAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS
Publication number
20150344425
Publication date
Dec 3, 2015
Actelion Pharmaceuticals LTD
KURT HILPERT
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INDOLE CARBOXAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONIST
Publication number
20150322008
Publication date
Nov 12, 2015
Actelion Pharmaceuticals LTD
KURT HILPERT
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC AMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS
Publication number
20150025075
Publication date
Jan 22, 2015
Actelion Pharmaceuticals LTD
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC AMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS
Publication number
20140163035
Publication date
Jun 12, 2014
Actelion Pharmaceuticals LTD
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS
Publication number
20140073651
Publication date
Mar 13, 2014
Actelion Pharmaceuticals LTD
Kurt Hilpert
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
THIAZOLE DERIVATIVES AND THEIR USE AS P2Y12 RECEPTOR ANTAGONISTS
Publication number
20130281406
Publication date
Oct 24, 2013
Actelion Pharmaceuticals LTD
Eva CAROFF
C07 - ORGANIC CHEMISTRY
Information
Patent Application
THIAZOLE DERIVATIVES AND THEIR USE AS P2Y12 RECEPTOR ANTAGONISTS
Publication number
20120053149
Publication date
Mar 1, 2012
Eva Caroff
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-(3-AZA-BICYCLO[3.1.0]HEX-3-YL)-2-PHENYL-PYRIMIDINES
Publication number
20120028989
Publication date
Feb 2, 2012
Eva Caroff
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BRIDGED TETRAHYDRONAPHTHALENE DERIVATIVES
Publication number
20110263648
Publication date
Oct 27, 2011
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SALTS OF ISOBUTYRIC ACID (1 R*,2R*,4R*) -2- (2- - ETHYL)-5-PHENYL-B...
Publication number
20110263667
Publication date
Oct 27, 2011
Stefan Abele
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TETRAHYDRONAPHTHALENE COMPOUNDS
Publication number
20110207815
Publication date
Aug 25, 2011
Kurt Hilpert
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 2-PHENYL-PYRIDINE DERIVATIVES
Publication number
20110046089
Publication date
Feb 24, 2011
Eva Caroff
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZIMIDAZOLE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS
Publication number
20110039905
Publication date
Feb 17, 2011
Francis Hubler
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHOSPHONIC ACID DERIVATES AD THEIR USE AS P2Y12 RECEPTOR ANTAGONISTS
Publication number
20100261678
Publication date
Oct 14, 2010
Eva Caroff
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BRIDGED SIX-MEMBERED RING COMPOUNDS
Publication number
20100130545
Publication date
May 27, 2010
Kurt Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Alternative heterocycles for DNA recognition
Publication number
20050026174
Publication date
Feb 3, 2005
California Institute of Technology
Peter B. Dervan
C07 - ORGANIC CHEMISTRY