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Douglas Walsh Hobbs
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Yardley, PA, US
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Patents Grants
last 30 patents
Information
Patent Grant
Cyclic amide BACE-1 inhibitors having a benzamide substituent
Patent number
9,062,007
Issue date
Jun 23, 2015
Merck Sharp & Dohme Corp.
Jared N. Cumming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrazolo[1,5-a]pyrimidines as cyclin dependent kinase i...
Patent number
8,673,924
Issue date
Mar 18, 2014
Merck Sharp & Dohme Corp.
Timothy J. Guzi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Cyclic amine BACE-1 inhibitors having a benzamide substituent
Patent number
8,623,867
Issue date
Jan 7, 2014
Merck Sharp & Dohme Corp.
Jared N. Cumming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cyclic amine BACE-1 inhibitors having a benzamide substituent
Patent number
8,278,334
Issue date
Oct 2, 2012
Merck, Sharp & Dohme Corp.
Jared N. Cumming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic substituted piperazines with CXCR3 antagonist activity
Patent number
8,207,170
Issue date
Jun 26, 2012
Schering Corporation
Seong Heon Kim
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic substituted pyridine compounds with CXCR3 antagonist a...
Patent number
8,017,616
Issue date
Sep 13, 2011
Schering Corporation
Stuart B. Rosenblum
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic substituted piperazine compounds with CXCR3 antagonist...
Patent number
7,902,199
Issue date
Mar 8, 2011
Schering Corporation
Stuart B. Rosenblum
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic substituted piperazines with CXCR3 antagonist activity
Patent number
7,868,006
Issue date
Jan 11, 2011
Schering Corporation
Seong Heon Kim
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazinyl substituted piperazine-piperidines with CXCR3 antagonist...
Patent number
7,868,005
Issue date
Jan 11, 2011
Schering Corporation
Stuart B. Rosenblum
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-heteroaryl pyrazolopyrimidines as cyclin dependent kinase inhibitors
Patent number
7,807,683
Issue date
Oct 5, 2010
Schering Corporation
Timothy J. Guzi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic substituted pyridine or phenyl compounds with CXCR3 an...
Patent number
7,799,789
Issue date
Sep 21, 2010
Schering Corporation
Gopinadhan N. Anilkumar
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic substituted pyridine compounds with CXCR3 antagonist a...
Patent number
7,786,124
Issue date
Aug 31, 2010
Schering Corporation
Stuart B. Rosenblum
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyridyl and phenyl substituted piperazine-piperidines with CXCR3 an...
Patent number
7,776,862
Issue date
Aug 17, 2010
Schering Corporation
Brian F. McGuinness
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperazine-piperidines with CXCR3 antagonist activity
Patent number
7,763,616
Issue date
Jul 27, 2010
Schering Corporation
Wensheng Yu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cyclic amine BACE-1 inhibitors having a benzamide substituent
Patent number
7,662,816
Issue date
Feb 16, 2010
Schering Corporation
Jared N. Cumming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cyclic amine BACE-1 inhibitors having a heterocyclic substituent
Patent number
7,598,250
Issue date
Oct 6, 2009
Schering Corporation
Jared N. Cumming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Amine-linked pyridyl and phenyl substituted piperazine-piperidines...
Patent number
7,566,718
Issue date
Jul 28, 2009
Schering Corporation
Michael K. C. Wong
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic compounds as selective melanin concentrating hormone recep...
Patent number
7,550,467
Issue date
Jun 23, 2009
Schering Corporation
Tao Guo
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic substituted pyridine or phenyl compounds with CXCR3 an...
Patent number
7,417,045
Issue date
Aug 26, 2008
Schering Corporation
Gopinadhan N. Anilkumar
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Gamma secretase inhibitors
Patent number
7,256,186
Issue date
Aug 14, 2007
Schering Corporation
Dimitri A. Pissarntiski
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Gamma secretase inhibitors
Patent number
7,208,602
Issue date
Apr 24, 2007
Schering Corporation
Dmitri A. Pissarnitski
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolopyrimidines as cyclin dependent kinase inhibitors
Patent number
7,161,003
Issue date
Jan 9, 2007
Schering Corporation
Timothy J. Guzi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolopyrimidines as cyclin dependent kinase inhibitors
Patent number
7,119,200
Issue date
Oct 10, 2006
Schering Corporation
Timothy J. Guzi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Aryl and biaryl compounds having MCH modulatory activity
Patent number
7,034,056
Issue date
Apr 25, 2006
Pharmacopeia Drug Discovery, Inc.
Douglas Walsh Hobbs
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aryl and biaryl piperdines with MCH modulatory activity
Patent number
6,887,889
Issue date
May 3, 2005
Pharmacopeia Drug Discovery, Inc.
Douglas W. Hobbs
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Method and apparatus for controlled photoelution
Patent number
6,468,787
Issue date
Oct 22, 2002
Pharmacopeia, Inc.
Rhett L. Affleck
C40 - COMBINATORIAL CHEMISTRY
Information
Patent Grant
Method and apparatus for controlled photoelution
Patent number
6,410,342
Issue date
Jun 25, 2002
Pharmacopeia, Inc.
Rhett L. Affleck
C40 - COMBINATORIAL CHEMISTRY
Information
Patent Grant
Hydantoin and succinimide-substituted derivatives of spiroindanylca...
Patent number
5,693,643
Issue date
Dec 2, 1997
Merck & Co., Inc.
Kevin Gilbert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Camphorcarbonyl
Patent number
5,686,454
Issue date
Nov 11, 1997
Merck & Co., Inc.
Mark G. Bock
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tocolytic oxytocin receptor antagonists
Patent number
5,670,509
Issue date
Sep 23, 1997
Merck & Co., Inc.
Ben E. Evans
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
CYCLIC AMIDE BACE-1 INHIBITORS HAVING A BENZAMIDE SUBSTITUENT
Publication number
20140128361
Publication date
May 8, 2014
Pharmacopeia Drug Discovery, Inc.
Jared N. Cumming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CYCLIC AMINE BACE-1 INHIBITORS HAVING A BENZAMIDE SUBSTITUENT
Publication number
20130004518
Publication date
Jan 3, 2013
Merck, Sharp & Dohme Corp.
Jared N. Cumming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC COMPOUNDS WITH CXCR3 ANTAGONIST ACTIVITY
Publication number
20120157466
Publication date
Jun 21, 2012
Qingbei Zeng
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC SUBSTITUTED PIPERAZINES WITH CXCR3 ANTAGONIST ACTIVITY
Publication number
20110065651
Publication date
Mar 17, 2011
Schering Corporation
Seong Heon Kim
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL HETEROCYCLIC SUBSTITUTED PYRIDINE COMPOUNDS WITH CXCR3 ANTAGO...
Publication number
20100168124
Publication date
Jul 1, 2010
Schering Corporation
Stuart B. Rosenblum
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CYCLIC AMINE BACE-1 INHIBITORS HAVING A BENZAMIDE SUBSTITUENT
Publication number
20100152138
Publication date
Jun 17, 2010
Schering Corp.
Jared N. Cumming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CYCLIC AMINE BACE-1 INHIBITORS HAVING A HETEROCYCLIC SUBSTITUENT
Publication number
20090312341
Publication date
Dec 17, 2009
Schering Corporation
Jared N. Cumming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL HETEROCYCLIC SUBSTITUTED PYRIDINE OR PHENYL COMPOUNDS WITH CX...
Publication number
20080292589
Publication date
Nov 27, 2008
Schering Corporation
Gopinadhan N. Anilkumar
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC SUBSTITUTED PIPERAZINE COMPOUNDS WITH CXCR3 ANTAGONIST...
Publication number
20080058343
Publication date
Mar 6, 2008
Schering Corporation and Pharmacopeia, Inc.
Stuart B. Rosenblum
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors
Publication number
20080050384
Publication date
Feb 28, 2008
Shering Corporation and Pharmacopeia, Inc.
Timothy J. Guzi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL HETEROCYCLIC SUBSTITUTED PYRIDINE COMPOUNDS WITH CXCR3 ANTAGO...
Publication number
20080039474
Publication date
Feb 14, 2008
Schering Corporation
STUART B. ROSENBLUM
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrazinyl substituted piperazine-piperidines with CXCR3 antagonist...
Publication number
20070054919
Publication date
Mar 8, 2007
Schering Corporation
Stuart B. Rosenblum
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors
Publication number
20070054925
Publication date
Mar 8, 2007
Schering Corporation
Timothy J. Guzi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors
Publication number
20070054906
Publication date
Mar 8, 2007
Schering Corporation
Timothy J. Guzi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors
Publication number
20070037824
Publication date
Feb 15, 2007
Schering Corporation
Timothy J. Guzi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyridyl and phenyl substituted piperazine-piperidines with CXCR3 an...
Publication number
20070021611
Publication date
Jan 25, 2007
Schering Corporation
Brian F. McGuinness
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Heterocyclic substituted piperazines with CXCR3 antagonist activity
Publication number
20060276479
Publication date
Dec 7, 2006
Schering Corporation and
Seong Heon Kim
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Piperazine-piperidines with CXCR3 antagonist activity
Publication number
20060276457
Publication date
Dec 7, 2006
Schering Corporation and Pharmacopeia Drug Discovery, Inc.
Wensheng Yu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Amine-linked pyridyl and phenyl substituted piperazine-piperidines...
Publication number
20060276480
Publication date
Dec 7, 2006
Schering Corporation and
Michael K. C. Wong
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel heterocyclic substituted pyridine or phenyl compounds with CX...
Publication number
20060217392
Publication date
Sep 28, 2006
Schering Corporation and
Gopinadhan N. Anilkumar
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic compounds as selective melanin concentrating hormone recep...
Publication number
20060111360
Publication date
May 25, 2006
Tao Guo
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel Gamma Secretase inhibitors
Publication number
20060100427
Publication date
May 11, 2006
Schering Corporation and Pharmacopeia, Inc.
Dmitri Pissarnitski
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Cyclic amine bace-1 inhibitors having a benzamide substituent
Publication number
20050119227
Publication date
Jun 2, 2005
Schering Corporation
Jared N. Cumming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel gamma secretase inhibitors
Publication number
20050085506
Publication date
Apr 21, 2005
Schering-Plough Corporation and Pharmacopeia, Inc.
Dmitri A. Pissarnitski
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Cyclic amine BACE-1 inhibitors having a heterocyclic substituent
Publication number
20050043290
Publication date
Feb 24, 2005
Schering Corporation and Pharmacopeia Drug Discovery Inc.
Jared N. Cumming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel pyrazolopyrimidines as cyclin dependent kinase inhibitors
Publication number
20040209878
Publication date
Oct 21, 2004
Schering Corporation and Pharmacopeia, Inc.
Timothy J. Guzi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Novel gamma secretase inhibitors
Publication number
20040171614
Publication date
Sep 2, 2004
Schering-Plough Corporation
Dmitri A. Pissarnitski
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel gamma secretase inhibitors
Publication number
20040048848
Publication date
Mar 11, 2004
Schering-Plough Corporation and Pharmacopeia, Inc.
Dmitri A. Pissarnitski
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Aryl and biaryl compounds having MCH modulatory activity
Publication number
20030092715
Publication date
May 15, 2003
Schering Corporation
Douglas Walsh Hobbs
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Aryl and biaryl piperidines with MCH modulatory activity
Publication number
20030013720
Publication date
Jan 16, 2003
PHARMACOPEIA, INC.
Douglas W. Hobbs
C07 - ORGANIC CHEMISTRY