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Eddy Jean Edgard Freyne
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Patents Grants
last 30 patents
Information
Patent Grant
Pyrazolyl quinoxaline kinase inhibitors
Patent number
10,519,137
Issue date
Dec 31, 2019
Astex Therapeutics Ltd.
Gordon Saxty
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Macrocyclic quinazole derivatives and their use as MTKI
Patent number
10,208,062
Issue date
Feb 19, 2019
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolyl quinoxaline kinase inhibitors
Patent number
9,850,228
Issue date
Dec 26, 2017
Astex Therapeutics Ltd.
Gordon Saxty
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocyclic quinazole derivatives and their use as MTKI
Patent number
9,688,691
Issue date
Jun 27, 2017
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolyl quinoxaline kinase inhibitors
Patent number
9,464,071
Issue date
Oct 11, 2016
Astex Therapeutics Ltd.
Gordon Saxty
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
3-cyano-quinoline derivatives with antiproliferative activity
Patent number
9,365,517
Issue date
Jun 14, 2016
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Quinazoline derivatives
Patent number
9,273,013
Issue date
Mar 1, 2016
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3-cyano-quinoline derivatives with antiproliferative activity
Patent number
9,040,511
Issue date
May 26, 2015
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrido and pyrimidopyrimidine derivatives as anti-profilerative agents
Patent number
8,933,067
Issue date
Jan 13, 2015
JANSSEN PHARMACEUTICA NV
Eddy Jean Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolyl quinoxaline kinase inhibitors
Patent number
8,895,601
Issue date
Nov 25, 2014
Astex Therapeutics Ltd.
Gordon Saxty
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases
Patent number
8,796,244
Issue date
Aug 5, 2014
Astex Therapeutics Ltd.
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3-cyano-quinoline derivatives with antiproliferative activity
Patent number
8,778,920
Issue date
Jul 15, 2014
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Quinolinone derivatives as PARP and tank inhibitors
Patent number
8,778,966
Issue date
Jul 15, 2014
Janssen Pharmaceutica, N.V.
Jorge Eduardo Vialard
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrido-and pyrimidopyrimidine derivatives as anti-proliferative agents
Patent number
8,772,272
Issue date
Jul 8, 2014
Janssen Pharmaceutica N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazo [1,2-A]pyridine derivatives as FGFR kinase inhibitors for u...
Patent number
8,722,687
Issue date
May 13, 2014
Astex Therapeutics Ltd.
Gordon Saxty
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
MTKI quinazoline derivatives
Patent number
8,492,377
Issue date
Jul 23, 2013
JANSSEN PHARMACEUTICA NV
Alexandra Papanikos
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic heterocyclyl derivatives as FGFR kinase inhibitors for the...
Patent number
8,481,531
Issue date
Jul 9, 2013
Astex Therapeutics Ltd.
Gordon Saxty
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aza-bicyclohexyl substituted indolyl alkyl amino derivatives as nov...
Patent number
8,476,289
Issue date
Jul 2, 2013
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Quinazoline derivatives
Patent number
8,394,786
Issue date
Mar 12, 2013
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2,4 (4,6) pyrimidine derivatives
Patent number
8,394,955
Issue date
Mar 12, 2013
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Il-5 inhibiting 6-azauracil derivatives
Patent number
6,803,364
Issue date
Oct 12, 2004
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-azauracil derivatives as IL-5 inhibitors
Patent number
6,743,792
Issue date
Jun 1, 2004
Janssen Pharmaceutica N.V.
Eddy Jean Edgard Freyne
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
PDE IV inhibiting pyridine derivatives
Patent number
6,656,959
Issue date
Dec 2, 2003
JANSSEN PHARMACEUTICA NV
Eddy Jean Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
4,5-dihydro-isoxazole derivatives and their pharmaceutical use
Patent number
6,583,141
Issue date
Jun 24, 2003
Janssen Pharmaceutica, N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Il-5 inhibiting 6-azauracil derivatives
Patent number
6,498,158
Issue date
Dec 24, 2002
Janssen Pharmaceutica N.V.
Jean Fernand Armand Lacrampe
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
IL-5 inhibiting 6-azauracil derivatives
Patent number
6,469,001
Issue date
Oct 22, 2002
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,3-dihydro-1-(phenylalkyl)-2H-imidazol-2-one derivatves
Patent number
6,403,805
Issue date
Jun 11, 2002
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Farnesyltransferase inhibiting quinazolinones
Patent number
6,358,961
Issue date
Mar 19, 2002
Jannsen-Cilag S.A.
Patrick René Angibaud
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Farnesyltransferase inhibiting quinazolinones
Patent number
6,177,432
Issue date
Jan 23, 2001
Janssen-Cilag S.A.
Patrick Rene Angibaud
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
PDE IV inhibiting 2-cyanoiminoimidazole derivatives
Patent number
6,051,718
Issue date
Apr 18, 2000
Janssen Pharmaceutica, N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
PYRAZOLYL QUINOXALINE KINASE INHIBITORS
Publication number
20220135544
Publication date
May 5, 2022
Astex Therapeutics Ltd.
Gordon SAXTY
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLYL QUINOXALINE KINASE INHIBITORS
Publication number
20200131153
Publication date
Apr 30, 2020
Astex Therapeutics Ltd.
Gordon SAXTY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLYL QUINOXALINE KINASE INHIBITORS
Publication number
20180127397
Publication date
May 10, 2018
Astex Therapeutics Ltd.
Gordon SAXTY
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYCLIC QUINAZOLE DERIVATIVES AND THEIR USE AS MTKI
Publication number
20170320894
Publication date
Nov 9, 2017
Janssen Pharmaceutica N.V.
Eddy Jean Edgard FREYNE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLYL QUINOXALINE KINASE INHIBITORS
Publication number
20160311800
Publication date
Oct 27, 2016
Astex Therapeutics Ltd.
Gordon SAXTY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINAZOLINE DERIVATIVES
Publication number
20160207938
Publication date
Jul 21, 2016
Janssen Pharmaceutica N.V.
Eddy Jean Edgard FREYNE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLYL QUINOXALINE KINASE INHIBITORS
Publication number
20150105368
Publication date
Apr 16, 2015
Astex Therapeutics Ltd.
Gordon SAXTY
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3-CYANO-QUINOLINE DERIVATIVES WITH ANTIPROLIFERATIVE ACTIVITY
Publication number
20140256948
Publication date
Sep 11, 2014
Janssen Pharmaceutica N.V.
Eddy Jean Edgard FREYNE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYCLIC QUINAZOLE DERIVATIVES AND THEIR USE AS MTKI
Publication number
20140256714
Publication date
Sep 11, 2014
Janssen Pharmaceutica N.V.
Eddy Jean Edgard FREYNE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDO- AND PYRIMIDOPYRIMIDINE DERIVATIVES AS ANTI-PROFILERATIVE AG...
Publication number
20130231353
Publication date
Sep 5, 2013
Janssen Pharmaceutica N.V.
Eddy Jean Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
3-CYANO-QUINOLINE DERIVATIVES WITH ANTIPROLIFERATIVE ACTIVITY
Publication number
20130197022
Publication date
Aug 1, 2013
Janssen Pharmaceutica N.V.
Eddy Jean Edgard Freyne
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
QUINAZOLINE DERIVATIVES
Publication number
20130178624
Publication date
Jul 11, 2013
Janssen Pharmaceutica N.V.
Eddy Jean Edgard FREYNE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLYL QUINAZOLINE KINASE INHIBITORS
Publication number
20130072457
Publication date
Mar 21, 2013
ASTEX THERAPEUTICS LIMITED
Gordon Saxty
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
QUINOLINONE DERIVATIVES AS PARP AND TANK INHIBITORS
Publication number
20130018017
Publication date
Jan 17, 2013
Jorge Eduardo VIALARD
C07 - ORGANIC CHEMISTRY
Information
Patent Application
5-Membered Annelated Heterocyclic Pyrimidines As Kinase Inhibitors
Publication number
20080070914
Publication date
Mar 20, 2008
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrazolopyrimidines as Cell Cycle Kinase Inhibitors
Publication number
20080039477
Publication date
Feb 14, 2008
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrido-and pyrimidopyrimidine derivatives as anti-profilerative agents
Publication number
20070078132
Publication date
Apr 5, 2007
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibi...
Publication number
20060183747
Publication date
Aug 17, 2006
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
3-Furanyl analogs of toxoflavine as kinase inhibitors
Publication number
20060040943
Publication date
Feb 23, 2006
Jean Fernand Armand LaCrampe
C07 - ORGANIC CHEMISTRY
Information
Patent Application
3-Phenyl analogs of toxoflavine as kinase inhibitors
Publication number
20050239784
Publication date
Oct 27, 2005
Jean Fernand Armand LaCrampe
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel IL-5 inhibiting 6-azauracil derivatives for marking and ident...
Publication number
20050090495
Publication date
Apr 28, 2005
Jean Fernand Armand Lacrampe
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel IL-5 inhibiting 6-azauracil derivatives for marking and ident...
Publication number
20040167333
Publication date
Aug 26, 2004
Jean Fernand Armand Lacrampe
C07 - ORGANIC CHEMISTRY
Information
Patent Application
4,5-Dihydro-isoxazole derivatives and their pharmaceutical use
Publication number
20040019059
Publication date
Jan 29, 2004
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-Azauracil derivatives as IL-5 inhibitors
Publication number
20030220331
Publication date
Nov 27, 2003
Eddy Jean Edgard Freyne
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Non-steroidal IL-5 inhibitors, processes and intermediates for thei...
Publication number
20030114453
Publication date
Jun 19, 2003
Jean Fernand Armand Lacrampe
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Novel IL-5 inhibiting 6-azauracil derivatives
Publication number
20020072603
Publication date
Jun 13, 2002
Jean Fernand Armand Lacrampe
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-azauracil derivatives as IL-5 inhibitors
Publication number
20020042416
Publication date
Apr 11, 2002
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IL-5 inhibiting 6-azauracil derivatives
Publication number
20020010177
Publication date
Jan 24, 2002
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY