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Fabrizio Giordanetto
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New York, NY, US
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Patents Grants
last 30 patents
Information
Patent Grant
Pyrazolo[3,4-b]pyrazine derivatives as SHP2 phosphatase inhibitors
Patent number
11,701,354
Issue date
Jul 18, 2023
D. E. Shaw Research, LLC
Alexander M. Taylor
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
SHP2 phosphatase inhibitors and methods of use thereof
Patent number
11,629,145
Issue date
Apr 18, 2023
D. E. Shaw Research, LLC
Fabrizio Giordanetto
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrazolo[3,4-b]pyrazines as SHP2 phosphatase inhibitors
Patent number
11,591,336
Issue date
Feb 28, 2023
D. E. Shaw Research, LLC
Alexander M. Taylor
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolo[3,4-b]pyrazine derivatives as SHP2 phosphatase inhibitors
Patent number
11,529,348
Issue date
Dec 20, 2022
D. E. Shaw Research, LLC
Alexander M. Taylor
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
SHP2 phosphatase inhibitors and methods of use thereof
Patent number
11,529,347
Issue date
Dec 20, 2022
Relay Therapeutics, Inc.
Brian K. Albrecht
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
SHP2 phosphatase inhibitors and methods of use thereof
Patent number
10,934,302
Issue date
Mar 2, 2021
Relay Therapeutics, Inc.
Alexander M. Taylor
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
LACTAM COMPOUNDS AS Kv1.3 POTASSIUM SHAKER CHANNEL BLOCKERS
Publication number
20230373952
Publication date
Nov 23, 2023
D.E. Shaw Research, LLC
Fabrizio GIORDANETTO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PI3K-ALPHA INHIBITORS AND METHODS OF USE THEREOF
Publication number
20230353959
Publication date
Nov 2, 2023
Relay Therapeutics, Inc.
Lucian V. DIPIETRO
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF
Publication number
20230234958
Publication date
Jul 27, 2023
Relay Therapeutics, Inc.
Alexander M. Taylor
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FGFR INHIBITORS AND METHODS OF USE THEREOF
Publication number
20230192709
Publication date
Jun 22, 2023
Relay Therapeutics, Inc.
Bakary-Barry TOURÉ
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ARYLMETHYLENE AROMATIC COMPOUNDS AS Kv1.3 POTASSIUM SHAKER CHANNEL...
Publication number
20230131535
Publication date
Apr 27, 2023
D. E. Shaw Research, LLC
Fabrizio GIORDANETTO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FGFR INHIBITORS AND METHODS OF USE THEREOF
Publication number
20230104574
Publication date
Apr 6, 2023
Relay Therapeutics, Inc.
Bakary-Barry TOURÉ
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ARYL HETEROBICYCLIC COMPOUNDS AS Kv1.3 POTASSIUM SHAKER CHANNEL BLO...
Publication number
20230049231
Publication date
Feb 16, 2023
D. E. Shaw Research, LLC
Fabrizio GIORDANETTO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ARYL HETEROBICYCLIC COMPOUNDS AS Kv1.3 POTASSIUM SHAKER CHANNEL BLO...
Publication number
20230040182
Publication date
Feb 9, 2023
D. E. Shaw Research, LLC
Fabrizio GIORDANETTO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ARYL HETEROCYCLIC COMPOUNDS AS Kv1.3 POTASSIUM SHAKER CHANNEL BLOCKERS
Publication number
20230026611
Publication date
Jan 26, 2023
D. E. Shaw Research, LLC
Fabrizio GIORDANETTO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ARYLMETHYLENE HETEROCYCLIC COMPOUNDS AS KV1.3 POTASSIUM SHAKER CHAN...
Publication number
20230023559
Publication date
Jan 26, 2023
D. E. Shaw Research, LLC
Fabrizio GIORDANETTO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ARYLMETHYLENE HETEROCYCLIC COMPOUNDS AS KV1.3 POTASSIUM SHAKER CHAN...
Publication number
20220411367
Publication date
Dec 29, 2022
D. E. Shaw Research, LLC
Fabrizio GIORDANETTO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF
Publication number
20220340576
Publication date
Oct 27, 2022
Relay Therapeutics, Inc.
Alexander M. Taylor
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF
Publication number
20220315586
Publication date
Oct 6, 2022
Relay Therapeutics, Inc.
Alexander M. Taylor
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLIC COMPOUNDS AND THEIR USE IN THE TREATMENT OF AMYLOID-RE...
Publication number
20220144840
Publication date
May 12, 2022
D. E. Shaw Research, LLC
Fabrizio GIORDANETTO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLO[3,4-B]PYRAZINE SHP2 PHOSPHATASE INHIBITORS AND METHODS OF...
Publication number
20210069188
Publication date
Mar 11, 2021
Relay Therapeutics, Inc.
Alexander M. Taylor
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF
Publication number
20200392161
Publication date
Dec 17, 2020
Relay Therapeutics, Inc.
W. Patrick Walters
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Compounds as Ras Inhibitors and Use Thereof
Publication number
20200308165
Publication date
Oct 1, 2020
D. E. Shaw Research, LLC
Yibing SHAN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLO[3,4-B]PYRAZINE DERIVATIVES AS SHP2 PHOSPHATASE INHIBITORS
Publication number
20200253969
Publication date
Aug 13, 2020
Relay Therapeutics, Inc.
Alexander M. Taylor
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLO[3,4-B]PYRAZINE DERIVATIVES AS SHP2 PHOSPHATASE INHIBITORS
Publication number
20200172546
Publication date
Jun 4, 2020
Relay Therapeutics, Inc.
Alexander M. Taylor
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF
Publication number
20200062760
Publication date
Feb 27, 2020
Relay Therapeutics, Inc.
Fabrizio Giordanetto
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF
Publication number
20190307745
Publication date
Oct 10, 2019
Relay Therapeutics, Inc.
Brian K. Albrecht
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE