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Giuseppe Cecere
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Patents Grants
last 30 patents
Information
Patent Grant
Isoxazolyl ether derivatives as GABAA α5 PAM
Patent number
11,840,528
Issue date
Dec 12, 2023
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepines as GABA A...
Patent number
11,739,095
Issue date
Aug 29, 2023
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Isoxazolyl ether derivatives as GABAA α5 PAM
Patent number
11,091,471
Issue date
Aug 17, 2021
HOFFMANN-LA ROCHE INC.
Bernd Buettelmann
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrazino[2,2-a]isoquinoline derivatives
Patent number
10,316,036
Issue date
Jun 11, 2019
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted azetidine derivatives
Patent number
10,023,559
Issue date
Jul 17, 2018
Hoffman-La Roche Inc.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-amino-5,6,7,8-tetrahydronaphthalen-2-yl or 3-aminochroman-7-yl de...
Patent number
9,957,261
Issue date
May 1, 2018
Hoffman-La Roche Inc.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Morpholin-pyridine derivatives
Patent number
9,840,501
Issue date
Dec 12, 2017
HOFFMANN-LA ROCHE INC.
Guido Galley
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrazino[2,2-a]isoquinoline derivatives
Patent number
9,828,374
Issue date
Nov 28, 2017
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperazine thiazole derivatives useful in the treatment of tauopath...
Patent number
9,808,456
Issue date
Nov 7, 2017
REMYND NV
Gerard Griffioen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
2-oxa-5-azabicyclo[2.2.1]heptan-3-yl derivatives
Patent number
9,790,230
Issue date
Oct 17, 2017
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
5-oxa-2-azabicyclo[2.2.2]OCTAN-4-yl and 5-oxa-2-azabicyclo[2.2.1]he...
Patent number
9,663,530
Issue date
May 30, 2017
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperazine thiazole derivatives useful in the treatment of tauopath...
Patent number
9,187,440
Issue date
Nov 17, 2015
REMYND NV
Gerard Griffioen
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
PET TRACERS FOR VISUALIZING GABAA GAMMA1 RECEPTORS
Publication number
20250049967
Publication date
Feb 13, 2025
HOFFMANN-LA ROCHE INC.
Giuseppe CECERE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CYCLOHEPTA-THIENO-DIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAM
Publication number
20240294543
Publication date
Sep 5, 2024
HOFFMANN-LA ROCHE INC.
Bjoern BARTELS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAM
Publication number
20240287082
Publication date
Aug 29, 2024
HOFFMANN-LA ROCHE INC.
Giuseppe CECERE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ISOXAZOLYL ETHER DERIVATIVES AS GABA A ALPHA5 PAM
Publication number
20240279218
Publication date
Aug 22, 2024
HOFFMANN-LA ROCHE INC.
Bernd BUETTELMANN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW PYRIDO DIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAM
Publication number
20240270744
Publication date
Aug 15, 2024
HOFFMANN-LA ROCHE INC.
Giuseppe CECERE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NEW CYCLOPENTA-THIENO-DIAZEPINE DERIVATIVES AS GABA A GAMMA1 POSITI...
Publication number
20240190889
Publication date
Jun 13, 2024
HOFFMANN-LA ROCHE INC.
Giuseppe CECERE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BENZO[f][l ,2,4JTRIAZOL0[4,3-a][l ,4JDIAZEPINES AS GABA...
Publication number
20240002393
Publication date
Jan 4, 2024
HOFFMANN-LA ROCHE INC.
Giuseppe CECERE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAM
Publication number
20230141603
Publication date
May 11, 2023
HOFFMANN-LA ROCHE INC.
Giuseppe CECERE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAM
Publication number
20230142171
Publication date
May 11, 2023
HOFFMANN-LA ROCHE INC.
Bjoern BARTELS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA 1 PAM
Publication number
20230136326
Publication date
May 4, 2023
HOFFMANN-LA ROCHE INC.
Bjoern BARTELS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TRIAZOLYL DERIVATIVES AS GABA A ALPHA5 PAM
Publication number
20230135093
Publication date
May 4, 2023
HOFFMANN-LA ROCHE INC.
Giuseppe CECERE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW PYRIDO DIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAM
Publication number
20230109111
Publication date
Apr 6, 2023
HOFFMANN-LA ROCHE INC.
Giuseppe CECERE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ISOXAZOLYL ETHER DERIVATIVES AS GABA A ALPHA5 PAM
Publication number
20220411415
Publication date
Dec 29, 2022
HOFFMANN-LA ROCHE INC.
Bernd BUETTELMANN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAM
Publication number
20210309664
Publication date
Oct 7, 2021
HOFFMANN-LA ROCHE INC.
Giuseppe CECERE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW ISOXAZOLYL ETHER DERIVATIVES AS GABA A ALPHA5 PAM
Publication number
20210094945
Publication date
Apr 1, 2021
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ISOXAZOLYL ETHER DERIVATIVES AS GABA A ALPHA5 PAM
Publication number
20190300516
Publication date
Oct 3, 2019
HOFFMANN-LA ROCHE INC.
Bernd BUETTELMANN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PYRAZINO[2,2-a]ISOQUINOLINE DERIVATIVES
Publication number
20180037582
Publication date
Feb 8, 2018
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PYRAZINO[2,2-a]ISOQUINOLINE DERIVATIVES
Publication number
20170145010
Publication date
May 25, 2017
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED AZETIDINE DERIVATIVES
Publication number
20170144994
Publication date
May 25, 2017
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2-OXA-5-AZABICYCLO[2.2.1]HEPTAN-3-YL DERIVATIVES
Publication number
20170137435
Publication date
May 18, 2017
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-AMINO-5,6,7,8-TETRAHYDRONAPHTHALEN-2-YL OR 3-AMINOCHROMAN-7-YL DE...
Publication number
20170137416
Publication date
May 18, 2017
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Application
5-OXA-2-AZABICYCLO[2.2.2]OCTAN-4-YL AND 5-OXA-2-AZABICYCLO[2.2.1]HE...
Publication number
20170066775
Publication date
Mar 9, 2017
HOFFMANN-LA ROCHE INC.
Giuseppe Cecere
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MORPHOLIN-PYRIDINE DERIVATIVES
Publication number
20170044145
Publication date
Feb 16, 2017
HOFFMANN-LA ROCHE INC.
Guido Galley
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PIPERAZINE THIAZOLE DERIVATIVES USEFUL IN THE TREATMENT OF TAUOPATH...
Publication number
20160101102
Publication date
Apr 14, 2016
REMYND NV
Gerard Griffioen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PIPERAZINE THIAZOLE DERIVATIVES USEFUL IN THE TREATMENT OF TAUOPATH...
Publication number
20140206699
Publication date
Jul 24, 2014
REMYND NV
Gerard Griffioen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE