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Hans Hilpert
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Muenchenstein, CH
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Patents Grants
last 30 patents
Information
Patent Grant
Peptide macrocycles against Acinetobacter baumannii
Patent number
12,012,466
Issue date
Jun 18, 2024
HOFFMANN-LA ROCHE INC.
Alexander Alanine
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
BACE1 inhibitors
Patent number
11,447,478
Issue date
Sep 20, 2022
Hoffmann-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Peptide macrocycles against Acinetobacter baumannii
Patent number
11,098,080
Issue date
Aug 24, 2021
HOFFMANN-LA ROCHE INC.
Alexander Alanine
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Anti-bacterial peptide macrocycles and use thereof
Patent number
11,066,443
Issue date
Jul 20, 2021
HOFFMANN-LA ROCHE INC.
Alexander Alanine
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Indolin-2-one derivatives
Patent number
10,457,667
Issue date
Oct 29, 2019
HOFFMANN-LA ROCHE INC.
Delphine Gaufreteau
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Indolin-2-one and 1,3-dihydro-pyrrolo[3,2-c]pyridin-2-one derivatives
Patent number
10,385,050
Issue date
Aug 20, 2019
HOFFMANN-LA ROCHE INC.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Indolin-2-one derivatives
Patent number
10,377,746
Issue date
Aug 13, 2019
HOFFMANN-LA ROCHE INC.
Delphine Gaufreteau
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Indolin-2-one and 1,3-dihydro-pyrrolo[3,2-c]pyridin-2-one derivatives
Patent number
10,112,938
Issue date
Oct 30, 2018
Hoffman-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Peptide macrocycles against acinetobacter baumannii
Patent number
10,030,047
Issue date
Jul 24, 2018
HOFFMANN-LA ROCHE INC.
Alexander Alanine
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrimidone derivatives and their use in the treatment, amelioration...
Patent number
9,988,390
Issue date
Jun 5, 2018
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Indolin-2-one or pyrrolo-pyridin/pyrimidin-2-one derivatives
Patent number
9,616,053
Issue date
Apr 11, 2017
HOFFMANN-LA ROCHE INC.
Daniela Brunner
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
5-amino[1,4]thiazines as BACE 1 inhibitors
Patent number
9,273,042
Issue date
Mar 1, 2016
Hoffmann-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,4 oxazines as BACE1 and/or BACE2 inhibitors
Patent number
9,242,943
Issue date
Jan 26, 2016
Siena Biotech S.p.A.
Matteo Andreini
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Difluoro-hexahydro-cyclopentaoxazinyls and difluoro-hexahydro-benzo...
Patent number
9,181,232
Issue date
Nov 10, 2015
Hoffmann-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,3-oxazines as BACE1 and/or BACE2 inhibitors
Patent number
9,115,098
Issue date
Aug 25, 2015
Hoffman-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
[1,3]oxazines
Patent number
9,073,909
Issue date
Jul 7, 2015
Hoffmann-La Roche Inc.
Edilio Boroni
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,4 thiazepines/sulfones as BACE1 and/or BACE2 inhibitors
Patent number
9,067,924
Issue date
Jun 30, 2015
Hoffmann-La Roche Inc.
Hans Hilpert
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Fluoromethyl-5,6-dihydro-4H-[1,3]OXAZINES
Patent number
9,067,926
Issue date
Jun 30, 2015
HOFFMANN-LA ROCHE INC.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,4,5,6-tetrahydro-pyrimidin-2-ylamine compounds
Patent number
8,815,881
Issue date
Aug 26, 2014
Hoffmann-La Roche Inc.
David Banner
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1,4-Oxazepines as BACE1 and/or BACE2 inhibitors
Patent number
8,815,841
Issue date
Aug 26, 2014
Hoffmann-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,3-oxazines as BACE 1 and/or BACE2 inhibitors
Patent number
8,785,436
Issue date
Jul 22, 2014
Hoffmann-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,3-oxazines as BACE1 and/or BACE2 inhibitors
Patent number
8,754,075
Issue date
Jun 17, 2014
Hoffmann-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,4-oxazepines as BACE1 and/or BACE2 inhibitors
Patent number
8,748,418
Issue date
Jun 10, 2014
Hoffmann-La Roche Inc.
Emanuele Gabellieri
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2,5,6,7-tetrahydro-[1,4]oxazepin-3-ylamine or 2,3,6,7-tetrahydro-[1...
Patent number
8,673,894
Issue date
Mar 18, 2014
Hoffmann-La Roche Inc.
David Banner
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-(3-(2-amino-6,6-difluoro-4,4A,5,6,7,7A-hexahydro-cyclopenta[E][1,...
Patent number
8,476,264
Issue date
Jul 2, 2013
Hoffmann-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dihydropyrimidinones
Patent number
8,461,160
Issue date
Jun 11, 2013
Hoffmann-La Roche, Inc.
David Banner
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-[3-(5-amino-3,3a,7,7a-tetrahydro-1H-2,4-dioxa-6-aza-inden-7-yl)-p...
Patent number
8,404,680
Issue date
Mar 26, 2013
Hoffmann-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2-amino-5,5-difluoro-5,6-dihydro-4H-[1,3]oxazin-4-yl)-phenyl]-amides
Patent number
8,389,513
Issue date
Mar 5, 2013
Hoffmann-La Roche Inc.
David Banner
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3-amino-5-phenyl-5,6-dihydro-2H-[1,4]oxazines
Patent number
8,188,079
Issue date
May 29, 2012
Hoffman-La Roche Inc.
Matteo Andreini
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Proline derivatives
Patent number
8,163,793
Issue date
Apr 24, 2012
Hoffman-La Roche Inc.
Rubén Alvarez Sánchez
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
INDOLIN-2-ONE OR PYRROLO -PYRIDIN -2 -ONE DERIVATIVES
Publication number
20230391778
Publication date
Dec 7, 2023
HOFFMANN-LA ROCHE INC.
Hans HILPERT
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PEPTIDE MACROCYCLES AGAINST ACINETOBACTER BAUMANNII
Publication number
20220411468
Publication date
Dec 29, 2022
HOFFMANN-LA ROCHE INC.
Alexander Alanine
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INDOLIN-2-ONE OR PYRROLO -PYRIDIN -2 -ONE DERIVATIVES
Publication number
20220033395
Publication date
Feb 3, 2022
HOFFMANN-LA ROCHE INC.
Hans Hilpert
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INDOLIN-2-ONE OR PYRROLO -PYRIDIN -2 -ONE DERIVATIVES
Publication number
20210246133
Publication date
Aug 12, 2021
HOFFMANN-LA ROCHE INC.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ANTI-BACTERIAL PEPTIDE MACROCYCLES AND USE THEREOF
Publication number
20200040031
Publication date
Feb 6, 2020
Alexander Alanine
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INDOLIN-2-ONE OR PYRROLO-PYRIDIN-2-ONE DERIVATIVES
Publication number
20200010466
Publication date
Jan 9, 2020
HOFFMANN-LA ROCHE INC.
Hans Hilpert
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INDOLIN-2-ONE AND 1,3-DIHYDRO-PYRROLO[3,2-c]PYRIDIN-2-ONE DERIVATIVES
Publication number
20190016719
Publication date
Jan 17, 2019
HOFFMANN-LA ROCHE INC.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PEPTIDE MACROCYCLES AGAINST ACINETOBACTER BAUMANNII
Publication number
20180362578
Publication date
Dec 20, 2018
HOFFMANN-LA ROCHE INC.
Alexander Alanine
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INDOLIN-2-ONE DERIVATIVES
Publication number
20180251451
Publication date
Sep 6, 2018
HOFFMANN-LA ROCHE INC.
Delphine Gaufreteau
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INDOLIN-2-ONE DERIVATIVES
Publication number
20180251455
Publication date
Sep 6, 2018
HOFFMANN-LA ROCHE INC.
Delphine Gaufreteau
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Pyrimidone derivatives and their use in the treatment, amelioration...
Publication number
20170267680
Publication date
Sep 21, 2017
F. Hoffmann-La Roche AG
Hans HILPERT
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PEPTIDE MACROCYCLES AGAINST ACINETOBACTER BAUMANNII
Publication number
20170233437
Publication date
Aug 17, 2017
HOFFMANN-LA ROCHE INC.
Alexander Alanine
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INDOLIN-2-ONE OR PYRROLO-PYRIDIN-2-ONE DERIVATIVES
Publication number
20170101409
Publication date
Apr 13, 2017
HOFFMANN-LA ROCHE INC.
Hans Hilpert
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INDOLIN-2-ONE AND 1,3-DIHYDRO-PYRROLO[3,2-c]PYRIDIN-2-ONE DERIVATIVES
Publication number
20170057960
Publication date
Mar 2, 2017
HOFFMANN-LA ROCHE INC.
Hans Hilpert
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INDOLIN-2-ONE OR PYRROLO-PYRIDIN/PYRIMIDIN-2-ONE DERIVATIVES
Publication number
20160095844
Publication date
Apr 7, 2016
HOFFMANN-LA ROCHE INC.
Daniela Brunner
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BACE1 INHIBITORS
Publication number
20160052920
Publication date
Feb 25, 2016
Hoffmann-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FLUORO-[1,3]OXAZINES AS BACE1 INHIBITORS
Publication number
20150376172
Publication date
Dec 31, 2015
Hoffmann-La Roche Inc.
Wolfgang Guba
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1,3-Oxazines As Bace1 And/Or Bace2 Inhibitors
Publication number
20150322054
Publication date
Nov 12, 2015
HOFFMANN-LA ROCHE INC.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
5-AMINO[1,4]THIAZINES AS BACE 1 INHIBITORS
Publication number
20150141413
Publication date
May 21, 2015
Hoffmnn-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DIFLUORO-HEXAHYDRO-CYCLOPENTAOXAZINYLS AND DIFLUORO-HEXAHYDRO-BENZO...
Publication number
20150133440
Publication date
May 14, 2015
Hoffmann-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FLUOROMETHYL-5,6-DIHYDRO-4H-[1,3]OXAZINES
Publication number
20150031690
Publication date
Jan 29, 2015
F. Hoffmann-La Roche AG
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1,4,5,6-TETRAHYDRO-PYRIMIDIN-2-YLAMINE COMPOUNDS
Publication number
20140336208
Publication date
Nov 13, 2014
David Banner
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
1,4 OXAZEPINES AS BACE1 AND/OR BACE2 INHIBITORS
Publication number
20140323469
Publication date
Oct 30, 2014
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1,3-Oxazines as Bace1 and/or Bace2 Inhibitors
Publication number
20140243325
Publication date
Aug 28, 2014
Hoffmann-La Roche Inc.
Hans Hilpert
C07 - ORGANIC CHEMISTRY
Information
Patent Application
USE OF AMINODIHYDROTHIAZINES FOR THE TREATMENT OR PREVENTION OF DIA...
Publication number
20140221360
Publication date
Aug 7, 2014
Hoffmann-La Roche Inc.
Jeremy Beauchamp
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
[1,3]OXAZINES
Publication number
20140112867
Publication date
Apr 24, 2014
Edilio Borroni
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2,5,6,7-Tetrahydro-[1,4]oxazepin-3-ylamine or 2,3,6,7-tetrahydro-[1...
Publication number
20140045820
Publication date
Feb 13, 2014
Hoffmann-La Roche Inc.
David Banner
C07 - ORGANIC CHEMISTRY
Information
Patent Application
3-AMINO-5-PHENYL-56-DIHYDRO-2H-[1,4]OXAZINES
Publication number
20130196984
Publication date
Aug 1, 2013
Siena Biotech S.p.A.
Matteo Andreini
C07 - ORGANIC CHEMISTRY
Information
Patent Application
USE OF AMINODIHYDROTHIAZINES FOR THE TREATMENT OR PREVENTION OF DIA...
Publication number
20130096107
Publication date
Apr 18, 2013
Hoffmann-La Roche Inc.
Jeremy Beauchamp
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
N-(3-(2-AMINO-6,6-DIFLUORO-4,4A,5,6,7,7A-HEXAHYDRO-CYCLOPENTA[E][1,...
Publication number
20130072478
Publication date
Mar 21, 2013
Hans Hilpert
C07 - ORGANIC CHEMISTRY