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Hariharan Venkatesan
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San Diego, CA, US
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last 30 patents
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Patent Grant
Inhibitors of KEAP1-Nrf2 protein-protein interaction
Patent number
11,897,900
Issue date
Feb 13, 2024
JANSSEN PHARMACEUTICA NV
J. Kent Barbay
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzoimidazoles as prolyl hydroxylase inhibitors
Patent number
11,618,744
Issue date
Apr 4, 2023
JANSSEN PHARMACEUTICA NV
Frances Meredith Hocutt
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Inhibitors of KEAP1-Nrf2 protein-protein interaction
Patent number
11,427,601
Issue date
Aug 30, 2022
JANSSEN PHARMACEUTICA NV
J. Kent Barbay
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
4-aminoquinazolinyl compounds as prolyl hydroxylase inhibitors
Patent number
10,975,062
Issue date
Apr 13, 2021
Janssen Pharmaceutica NV
Michael H. Rabinowitz
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
6-aminopyridin-3-yl thiazoles as modulators of RORγT
Patent number
10,975,068
Issue date
Apr 13, 2021
JANSSEN PHARMACEUTICA NV
Steven Goldberg
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Inhibitors of KEAP1-Nrf2 protein-protein interaction
Patent number
10,947,252
Issue date
Mar 16, 2021
JANSSEN PHARMACEUTICA NV
J. Kent Barbay
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzoimidazoles as prolyl hydroxylase inhibitors
Patent number
10,851,083
Issue date
Dec 1, 2020
Janssen Pharmaceutica N.V.
Frances Meredith Hocutt
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Alkyl linked quinolinyl modulators of RORγt
Patent number
10,555,941
Issue date
Feb 11, 2020
JANSSEN PHARMACEUTICA NV
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Phenyl linked quinolinyl modulators of RORγt
Patent number
10,369,146
Issue date
Aug 6, 2019
JANSSEN PHARMACEUTICA NV
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
4-Aminoquinazolin compounds as prolyl hydroxylase inhibitors
Patent number
10,246,442
Issue date
Apr 2, 2019
Janssen Pharmaceutica N.V.
Michael H. Rabinowitz
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Quinolinyl modulators of RORγt
Patent number
10,201,546
Issue date
Feb 12, 2019
JANSSEN PHARMACEUTICA NV
Kristi A. Leonard
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Trifluoromethyl alcohols as modulators of RORγt
Patent number
10,150,762
Issue date
Dec 11, 2018
Janssen Pharmaceutica, N.V.
Steven Goldberg
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Trifluoromethyl alcohols as modulators of RORγt
Patent number
9,850,236
Issue date
Dec 26, 2017
JANSSEN PHARMACEUTICA NV
Steven Goldberg
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Amide substituted thiazoles as modulators of RORyt
Patent number
9,845,319
Issue date
Dec 19, 2017
Janssen Pharmaceutiuca NV
Steven Goldberg
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Quinolinyl modulators of RORγt
Patent number
9,624,225
Issue date
Apr 18, 2017
JANSSEN PHARMACEUTICA NV
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
4-aminoquinazolinyl-2-yl-1-pyrazole-4-carboxylic acid compounds as...
Patent number
9,573,940
Issue date
Feb 21, 2017
JANSSEN PHARMACEUTICA NV
Michael H. Rabinowitz
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Phenyl linked quinolinyl modulators of RORγt
Patent number
9,403,816
Issue date
Aug 2, 2016
JANSSEN PHARMACEUTICA NV
Kristi A. Leonard
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Alkyl linked quinolinyl modulators of RORγt
Patent number
9,346,782
Issue date
May 24, 2016
Janssen Pharmaceutica N.V.
Kristi A. Leonard
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heteroaryl linked quinolinyl modulators of RORgammat
Patent number
9,328,095
Issue date
May 3, 2016
Janssen Pharmaceutica NV
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Phenyl linked quinolinyl modulators of RORγt
Patent number
9,309,222
Issue date
Apr 12, 2016
Janssen Pharmaceutica N.V.
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Heteroaryl linked quinolinyl modulators of RORγt
Patent number
9,303,015
Issue date
Apr 5, 2016
Janssen Pharmaceutica N.V.
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Methylene linked quinolinyl modulators of RORγt
Patent number
9,290,476
Issue date
Mar 22, 2016
JANSSEN PHARMACEUTICA NV
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Methylene linked quinolinyl modulators of RORγt
Patent number
9,284,308
Issue date
Mar 15, 2016
Janssen Pharmaceutica NV
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Secondary alcohol quinolinyl modulators of RORγt
Patent number
9,221,804
Issue date
Dec 29, 2015
Janssen Pharmaceutica N.V.
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzoimidazoles as prolyl hydroxylase inhibitors
Patent number
9,073,923
Issue date
Jul 7, 2015
JANSSEN PHARMACEUTICA NV
Frances Meredith Hocutt
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
4-aminoquinazolin-2-yl-1-pyrrazole-4-carboxylic acid compounds as p...
Patent number
9,006,251
Issue date
Apr 14, 2015
Janssen Pharamceutica NV
Michael H. Rabinowitz
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Quinazolinones as prolyl hydroxylase inhibitors
Patent number
8,937,078
Issue date
Jan 20, 2015
JANSSEN PHARMACEUTICA NV
Scott D. Bembenek
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzoimidazoles as prolyl hydroxylase inhibitors
Patent number
8,865,713
Issue date
Oct 21, 2014
JANSSEN PHARMACEUTICA NV
Frances Meredith Hocutt
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
4-aminoquinazolin-2-yl-1-pyrrazole-4-carboxylic acid compounds as p...
Patent number
8,796,263
Issue date
Aug 5, 2014
JANSSEN PHARMACEUTICA NV
Michael H. Rabinowitz
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzoimidazoles as prolyl hydroxylase inhibitors
Patent number
8,759,345
Issue date
Jun 24, 2014
JANSSEN PHARMACEUTICA NV
Frances Meredith Hocutt
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
INHIBITORS OF KEAP1-Nrf2 PROTEIN-PROTEIN INTERACTION
Publication number
20220315604
Publication date
Oct 6, 2022
Janssen Pharmaceutica N.V.
J. Kent Barbay
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZIMIDAZOLE DERIVATIVE FOR USE IN THE TREATMENT OF INFLAMMATORY D...
Publication number
20210369678
Publication date
Dec 2, 2021
Michael Rabinowitz
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
6-AMINOPYRIDIN-3-YL THIAZOLES AS MODULATORS OF RORyT
Publication number
20210221804
Publication date
Jul 22, 2021
Janssen Pharmaceutica N.V.
Steven Goldberg
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-AMINOPYRIDIN-3-YL THIAZOLES AS MODULATORS OF RORyT
Publication number
20210198251
Publication date
Jul 1, 2021
Janssen Pharmaceutica N.V.
Steven Goldberg
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-AMINOPYRIDIN-3-YL THIAZOLES AS MODULATORS OF RORyT
Publication number
20210188836
Publication date
Jun 24, 2021
Janssen Pharmaceutica N.V.
Steven Goldberg
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZOIMIDAZOLES AS PROLYL HYDROXYLASE INHIBITORS
Publication number
20210078978
Publication date
Mar 18, 2021
Janssen Pharmaceutica N.V.
Frances Meredith Hocutt
C07 - ORGANIC CHEMISTRY
Information
Patent Application
4-AMINOQUINAZOLINYL COMPOUNDS AS PROLYL HYDROXYLASE INHIBITORS
Publication number
20200095234
Publication date
Mar 26, 2020
Janssen Pharmaceutica N.V.
Michael H. RABINOWITZ
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INHIBITORS OF KEAP1-Nrf2 PROTEIN-PROTEIN INTERACTION
Publication number
20200055874
Publication date
Feb 20, 2020
Janssen Pharmaceutica N.V.
J. Kent Barbay
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZOIMIDAZOLES AS PROLYL HYDROXYLASE INHIBITORS
Publication number
20190367486
Publication date
Dec 5, 2019
Janssen Pharmaceutica N.V.
Frances Meredith Hocutt
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZOIMIDAZOLES AS PROLYL HYDROXYLASE INHIBITORS
Publication number
20180215732
Publication date
Aug 2, 2018
Janssen Pharmaceutica N.V.
Frances Meredith Hocutt
C07 - ORGANIC CHEMISTRY
Information
Patent Application
4-AMINOQUINAZOLIN COMPOUNDS AS PROLYL HYDROXYLASE INHIBITORS
Publication number
20180148435
Publication date
May 31, 2018
Janssen Pharmaceutica N.V.
Michael H. RABINOWITZ
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZOIMIDAZOLES AS PROLYL HYDROXYLASE INHIBITORS
Publication number
20180022733
Publication date
Jan 25, 2018
Janssen Pharmaceutica N.V.
Frances Meredith Hocutt
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TRIFLUOROMETHYL ALCOHOLS AS MODULATORS OF RORyt
Publication number
20170327492
Publication date
Nov 16, 2017
Janssen Pharmaceutica N.V.
Steven Goldberg
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
4-AMINOQUINAZOLIN COMPOUNDS AS PROLYL HYDROXYLASE INHIBITORS
Publication number
20170320859
Publication date
Nov 9, 2017
Janssen Pharmaceutica N.V.
Michael H. RABINOWITZ
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
6-AMINOPYRIDIN-3-YL THIAZOLES AS MODULATORS OF RORyT
Publication number
20170313691
Publication date
Nov 2, 2017
Janssen Pharmaceutica N.V.
Steven Goldberg
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ALKYL LINKED QUINOLINYL MODULATORS OF RORγt
Publication number
20170258782
Publication date
Sep 14, 2017
Janssen Pharmaceutica N.V.
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
QUINOLINYL MODULATORS OF RORyt
Publication number
20170182056
Publication date
Jun 29, 2017
Janssen Pharmaceutica N.V.
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PHENYL LINKED QUINOLINYL MODULATORS OF RORgammat
Publication number
20160279122
Publication date
Sep 29, 2016
Janssen Pharmaceutica N.V.
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZOIMIDAZOLES AS PROLYL HYDROXYLASE INHIBITORS
Publication number
20160168127
Publication date
Jun 16, 2016
Janssen Pharmaceutica N.V.
Frances Meredith Hocutt
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROARYL LINKED QUINOLINYL MODULATORS OF RORyt
Publication number
20160136149
Publication date
May 19, 2016
Janssen Pharmaceutica NV
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TRIFLUOROMETHYL ALCOHOLS AS MODULATORS OF RORyt
Publication number
20160122336
Publication date
May 5, 2016
Janssen Pharmaceutica NV
Steven Goldberg
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMIDE SUBSTITUTED THIAZOLES AS MODULATORS OF RORyt
Publication number
20160122335
Publication date
May 5, 2016
Janssen Pharmaceutica NV
Steven Goldberg
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Benzoimidazoles as prolyl hydroxylase inhibitors
Publication number
20150284335
Publication date
Oct 8, 2015
Janssen Pharmaceutica N.V.
Frances Meredith Hocutt
C07 - ORGANIC CHEMISTRY
Information
Patent Application
4-Aminoquinazolinyl compounds as prolyl hydroxylase inhibitors
Publication number
20150197507
Publication date
Jul 16, 2015
Janssen Pharmaceutica N.V.
Michael H. Rabinowitz
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINOLINYL MODULATORS OF RORyt
Publication number
20150111870
Publication date
Apr 23, 2015
JOHNSON & JOHNSON
KRISTI A. LEONARD
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PHENYL LINKED QUINOLINYL MODULATORS OF RORyt
Publication number
20150105404
Publication date
Apr 16, 2015
Janssen Pharmaceutica N.V.
KRISTI A. LEONARD
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHYLENE LINKED QUINOLINYL MODULATORS OF RORyt
Publication number
20150105366
Publication date
Apr 16, 2015
Janssen Pharmaceutica N.V.
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SECONDARY ALCOHOL QUINOLINYL MODULATORS OF RORyt
Publication number
20150105372
Publication date
Apr 16, 2015
Janssen Pharmaceutica N.V.
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ALKYL LINKED QUINOLINYL MODULATORS OF RORyt
Publication number
20150105369
Publication date
Apr 16, 2015
Janssen Pharmaceutica N.V.
KRISTI A. LEONARD
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROARYL LINKED QUINOLINYL MODULATORS OF RORgammat
Publication number
20150105365
Publication date
Apr 16, 2015
Janssen Pharmaceutica N.V.
Kristi A. Leonard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE