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Harold Mastalerz
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Guilford, CT, US
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Patents Grants
last 30 patents
Information
Patent Grant
Isofuranone compounds useful as HPK1 inhibitors
Patent number
11,166,959
Issue date
Nov 9, 2021
Bristol-Myers Squibb Company
Erika M. V. Araujo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-ones as RIPK3 in...
Patent number
10,301,306
Issue date
May 28, 2019
Bristol-Myers Squibb Company
Amy C. Hart
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazotriazinecarbonitriles useful as kinase inhibitors
Patent number
9,556,178
Issue date
Jan 31, 2017
Bristol-Myers Squibb Company
Ashok Vinayak Purandare
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Imidazotriazinecarbonitriles useful as kinase inhibitors
Patent number
9,273,057
Issue date
Mar 1, 2016
Bristol-Myers Squibb Company
Ashok Vinayak Purandare
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Imidazotriazinecarbonitriles useful as kinase inhibitors
Patent number
8,940,736
Issue date
Jan 27, 2015
Bristol-Myers Squibb Company
Ashok Vinayak Purandare
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Carbazole and carboline kinase inhibitors
Patent number
8,815,840
Issue date
Aug 26, 2014
Bristol-Myers Squibb Company
Ashok Vinayak Purandare
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolotriazine kinase inhibitors
Patent number
8,592,579
Issue date
Nov 26, 2013
Bristol-Myers Squibb Company
Mark D. Wittman
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolotriazine kinase inhibitors
Patent number
7,879,855
Issue date
Feb 1, 2011
Bristol-Myers Squibb Company
Mark D. Wittman
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolotriazine compounds as kinase inhibitors
Patent number
7,846,931
Issue date
Dec 7, 2010
Bristol-Myers Squibb Company
Brian E. Fink
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Intermediates useful in preparing certain pyrrolotriazine compounds...
Patent number
7,619,083
Issue date
Nov 17, 2009
Bristol-Myers Squibb Company
Harold Mastalerz
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolotriazine kinase inhibitors
Patent number
7,534,792
Issue date
May 19, 2009
Bristol-Myers Squibb Company
Mark D. Wittman
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolotriazine compounds useful as kinase inhibitors and methods o...
Patent number
7,442,700
Issue date
Oct 28, 2008
Bristol-Myers Squibb Company
Harold Mastalerz
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolotriazine compounds as kinase inhibitors
Patent number
7,297,695
Issue date
Nov 20, 2007
Bristol-Myers Squibb Company
Brian E. Fink
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Intermediates useful in preparing certain pyrrolotriazine compounds...
Patent number
7,232,901
Issue date
Jun 19, 2007
Bristol-Myers Squibb Company
Harold Mastalerz
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
C-6 modified indazolylpyrrolotriazines
Patent number
7,148,220
Issue date
Dec 12, 2006
Bristol-Myers Squibb Company
Gregory D. Vite
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolotriazine compounds as kinase inhibitors
Patent number
7,141,571
Issue date
Nov 28, 2006
Bristol-Myers Squibb Company
Brian E. Fink
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolotriazine compounds
Patent number
7,102,003
Issue date
Sep 5, 2006
Bristol-Myers Squibb Company
Ashvinikumar V. Gavai
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Di-substituted pyrrolotriazine compounds
Patent number
7,064,203
Issue date
Jun 20, 2006
Bristol-Myers Squibb Company
Ashvinikumar V. Gavai
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
C-6 modified indazolylpyrrolotriazines
Patent number
6,916,815
Issue date
Jul 12, 2005
Bristol-Myers Squibb Company
Gregory D. Vite
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Process for the preparation of C-4 carbonate taxanes
Patent number
6,916,942
Issue date
Jul 12, 2005
Bristol-Myers Squibb Company
John F. Kadow
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
C-5 modified indazolylpyrrolotriazines
Patent number
6,908,916
Issue date
Jun 21, 2005
Bristol-Myers Squibb Company
Harold Mastalerz
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
C-4 carbonate taxanes
Patent number
6,750,246
Issue date
Jun 15, 2004
Bristol-Myers Squibb Company
John F. Kadow
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
7-sulfur substituted paclitaxels
Patent number
6,017,935
Issue date
Jan 25, 2000
Bristol-Myers Squibb Company
Harold Mastalerz
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-thio-substituted paclitaxels
Patent number
5,977,386
Issue date
Nov 2, 1999
Bristol-Myers Squibb Company
Andrew J. Staab
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
ISOFURANONE COMPOUNDS USEFUL AS HPK1 INHIBITORS
Publication number
20200390776
Publication date
Dec 17, 2020
Bristol-Myers Squibb Company
Erika M.V. Araujo
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED DIHYDRO-1H-PYRROLO[3,2-C]PYRIDIN-4(5H)-ONES AS RIPK3 IN...
Publication number
20170362219
Publication date
Dec 21, 2017
Bristol-Myers Squibb Company
Amy C. HART
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDAZOTRIAZINECARBONITRILES USEFUL AS KINASE INHIBITORS
Publication number
20160108050
Publication date
Apr 21, 2016
Bristol-Myers Squibb Company
Ashok Vinayak Purandare
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDAZOTRIAZINECARBONITRILES USEFUL AS KINASE INHIBITORS
Publication number
20150210697
Publication date
Jul 30, 2015
Bristol-Myers Squibb Company
Ashok Vinayak Purandare
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDAZOTRIAZINECARBONITRILES USEFUL AS KINASE INHIBITORS
Publication number
20150065465
Publication date
Mar 5, 2015
Bristol-Myers Squibb Company
Ashok Vinayak Purandare
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMIDAZOTRIAZINECARBONITRILES USEFUL AS KINASE INHIBITORS
Publication number
20140018319
Publication date
Jan 16, 2014
Ashok Vinayak Purandare
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRROLOTRIAZINE KINASE INHIBITORS
Publication number
20120302747
Publication date
Nov 29, 2012
Bristol -Myers Squibb Company
Mark D. Wittman
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CARBAZOLE AND CARBOLINE KINASE INHIBITORS
Publication number
20120058988
Publication date
Mar 8, 2012
Bristol -Myers Squibb Company
Ashok Vinayak Purandare
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOTRIAZINE KINASE INHIBITORS
Publication number
20110124623
Publication date
May 26, 2011
Bristol -Myers Squibb Company
Mark D. Wittman
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOTRIAZINE COMPOUNDS AS KINASE INHIBITORS
Publication number
20110039838
Publication date
Feb 17, 2011
Bristol -Myers Squibb Company
Brian E. Fink
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOTRIAZINE COMPOUNDS USEFUL AS KINASE INHIBITORS AND METHODS O...
Publication number
20100137319
Publication date
Jun 3, 2010
Bristol -Myers Squibb Company
Harold Mastalerz
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOTRIAZINE KINASE INHIBITORS
Publication number
20090239838
Publication date
Sep 24, 2009
Bristol -Myers Squibb Company
Mark D. Wittman
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOTRIAZINE COMPOUNDS USEFUL AS KINASE INHIBITORS AND METHODS O...
Publication number
20090062288
Publication date
Mar 5, 2009
Harold Mastalerz
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOTRIAZINE COMPOUNDS AS KINASE INHIBITORS
Publication number
20090048244
Publication date
Feb 19, 2009
Bristol -Myers Squibb Company
Brian E. Fink
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOTRIAZINE KINASE INHIBITORS
Publication number
20080009497
Publication date
Jan 10, 2008
Bristol -Myers Squibb Company
Mark D. Wittman
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INTERMEDIATES USEFUL IN PREPARING CERTAIN PYRROLOTRIAZINE COMPOUNDS...
Publication number
20070015760
Publication date
Jan 18, 2007
Bristol -Myers Squibb Company
Harold Mastalerz
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOTRIAZINE COMPOUNDS USEFUL AS KINASE INHIBITORS AND METHODS O...
Publication number
20070004731
Publication date
Jan 4, 2007
Bristol-Myers Squibb Company
Harold Mastalerz
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Intermediates useful in preparing certain pyrrolotriazine compounds...
Publication number
20070004734
Publication date
Jan 4, 2007
Bristol -Myers Squibb Company
Harold Mastalerz
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOTRIAZINE COMPOUNDS AS KINASE INHIBITORS
Publication number
20060264438
Publication date
Nov 23, 2006
Bristol-Myers Squibb Company
Brian E. Fink
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrrolotriazine compounds
Publication number
20060014745
Publication date
Jan 19, 2006
Ashvinikumar V. Gavai
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Methods of treating cancer using C-4 carbonate taxanes
Publication number
20050250844
Publication date
Nov 10, 2005
John F. Kadow
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
C-6 modified indazolylpyrrolotriazines
Publication number
20050222153
Publication date
Oct 6, 2005
Gregory D. Vite
C07 - ORGANIC CHEMISTRY
Information
Patent Application
C-5 Modified indazolylpyrrolotriazines
Publication number
20050209235
Publication date
Sep 22, 2005
Harold Mastalerz
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Di-substituted pyrrolotrizine compounds
Publication number
20050197339
Publication date
Sep 8, 2005
Ashvinikumar V. Gavai
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrrolotriazine compounds as kinase inhibitors
Publication number
20050182058
Publication date
Aug 18, 2005
Brian E. Fink
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Process for the preparation of C-4 carbonate taxanes
Publication number
20040225009
Publication date
Nov 11, 2004
John F. Kadow
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
C-6 modified indazolylpyrrolotriazines
Publication number
20040142931
Publication date
Jul 22, 2004
Gregory D. Vite
C07 - ORGANIC CHEMISTRY
Information
Patent Application
C-5 Modified indazolylpyrrolotriazines
Publication number
20030186983
Publication date
Oct 2, 2003
Harold Mastalerz
C07 - ORGANIC CHEMISTRY