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Janusz Josef Kulagowski
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Harlow Essex, GB
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Patents Grants
last 30 patents
Information
Patent Grant
Substituted azaindoline derivatives as NIK inhibitors
Patent number
11,236,084
Issue date
Feb 1, 2022
JANSSEN PHARMACEUTICA NV
George Hynd
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cyanoindoline derivatives as NIK inhibitors
Patent number
11,186,589
Issue date
Nov 30, 2021
JANSSEN PHARMACEUTICA NV
Ian Stansfield
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted cyanoindoline derivatives as NIK inhibitors
Patent number
11,180,487
Issue date
Nov 23, 2021
JANSSEN PHARMACEUTICA NV
Ian Stansfield
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heteroaromatic derivatives as NIK inhibitors
Patent number
11,136,311
Issue date
Oct 5, 2021
JANSSEN PHARMACEUTICA NV
Ian Stansfield
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-membered heteroaromatic substituted cyanoindoline derivatives as...
Patent number
11,001,569
Issue date
May 11, 2021
JANSSEN PHARMACEUTICA NV
Ian Stansfield
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1-(4-pyrimidinyl)-1H-pyrrolo[3,2-c]pyridine derivatives as NIK inhi...
Patent number
10,005,773
Issue date
Jun 26, 2018
JANSSEN PHARMACEUTICA NV
George Hynd
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds as NIK inhibitors
Patent number
10,005,776
Issue date
Jun 26, 2018
JANSSEN PHARMACEUTICA NV
George Hynd
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazole derivatives as NIK inhibitors
Patent number
9,981,962
Issue date
May 29, 2018
JANSSEN PHARMACEUTICA NV
George Hynd
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3-(1H-pyrazol-4-yl)-1H-pyrrolo[2,3-c]pyridine derivatives as NIK in...
Patent number
9,981,963
Issue date
May 29, 2018
JANSSEN PHARMACEUTICA NV
George Hynd
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3-(2-aminopyrimidin-4-yl)-5-(3-hydroxypropynyl)-1H-pyrrolo[2,3-C]py...
Patent number
9,643,964
Issue date
May 9, 2017
JANSSEN PHARMACEUTICA NV
George Hynd
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrimidine derivatives and their use in the treatment of respirator...
Patent number
9,156,844
Issue date
Oct 13, 2015
CHIESI FARMACEUTICI S.P.A.
Christine Edwards
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrimidine derivatives and their use in the treatment of respirator...
Patent number
9,120,802
Issue date
Sep 1, 2015
CHIESI FARMACEUTICI S.P.A.
Christine Edwards
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Sulphone compounds and methods of making and using same
Patent number
9,067,905
Issue date
Jun 30, 2015
Zafgen, Inc.
Hazel J. Dyke
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds
Patent number
9,023,855
Issue date
May 5, 2015
CHIESI FARMACEUTICI S.P.A.
Toby Jonathan Blench
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds
Patent number
8,691,826
Issue date
Apr 8, 2014
CHIESI FARMACEUTICI S.P.A.
Toby Jonathan Blench
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Adenine inhibitors of HSP90
Patent number
8,669,248
Issue date
Mar 11, 2014
John Montana
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tricyclic heterocyclic compounds, compositions and methods of use t...
Patent number
8,461,328
Issue date
Jun 11, 2013
Genentech, Inc.
Srinivasan Babu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperidines and related compounds for the treatment of Alzheimer's...
Patent number
8,389,547
Issue date
Mar 5, 2013
Yudith Garcia
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperidine derivatives for treatment of Alzheimer's disease
Patent number
7,985,758
Issue date
Jul 26, 2011
Merck, Sharp & Dohme Limited
Andrew Madin
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Thiazolopyrimidines and their use as inhibitors of phosphatidylinos...
Patent number
7,893,060
Issue date
Feb 22, 2011
F. Hoffmann-La Roche AG
Timothy Colin Hancox
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperidines and related compounds for treatment of alzheimer's disease
Patent number
7,638,629
Issue date
Dec 29, 2009
Merck Sharp & Dohme Ltd,
Joanne Clare Hannam
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tetrahydropyran compounds as tachykinin antagonists
Patent number
7,393,858
Issue date
Jul 1, 2008
Merck Sharp & Dohme Ltd.
Olivier Dirat
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
5-HT7 receptor antagonists
Patent number
7,276,607
Issue date
Oct 2, 2007
Merck Sharp & Dohme Limited
Neil Roy Curtis
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Sulfone derivatives as 5-HT7 receptor ligands
Patent number
7,101,892
Issue date
Sep 5, 2006
Merck Sharp & Dohme Ltd
Sylvie Bourrain
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Azabicyclic ether derivatives and their use as therapeutic agents
Patent number
6,727,249
Issue date
Apr 27, 2004
Merck Sharp & Dohme Ltd.
Neil Roy Curtis
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Use of NK-1 receptor antagonists for treating major depressive diso...
Patent number
6,613,765
Issue date
Sep 2, 2003
Merck Sharp & Dohme Limited
Raymond Baker
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pentaaza-cyclopental[a]naphthalene derivatives as l...
Patent number
6,613,766
Issue date
Sep 2, 2003
Merck Sharp & Dohme Ltd.
Neil Roy Curtis
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Azabicyclic amine derivatives and their use as therapeutic agents
Patent number
6,555,552
Issue date
Apr 29, 2003
Merck Sharp & Dohme Ltd.
Janusz Jozef Kulagowski
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Azabicyclic spiroether derivatives and their use as therapeutic agents
Patent number
6,479,486
Issue date
Nov 12, 2002
Merck Sharp & Dohme Ltd.
Ian Thomas Huscroft
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,4 substituted piperidinyl NMDA/NR2B antagonists
Patent number
6,476,041
Issue date
Nov 5, 2002
Merck & Co., Inc.
Wayne Thompson
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
NEW SUBSTITUTED AZAINDOLINE DERIVATIVES AS NIK INHIBITORS
Publication number
20210188840
Publication date
Jun 24, 2021
Janssen Pharmaceutica N.V.
George HYND
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW SUBSTITUTED CYANOINDOLINE DERIVATIVES AS NIK INHIBITORS
Publication number
20210087182
Publication date
Mar 25, 2021
Janssen Pharmaceutica N.V.
Ian STANSFIELD
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CYANOINDOLINE DERIVATIVES AS NIK INHIBITORS
Publication number
20210032267
Publication date
Feb 4, 2021
Janssen Pharmaceutica N.V.
Ian Stansfield
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NEW 6-MEMBERED HETEROAROMATIC SUBSTITUTED CYANOINDOLINE DERIVATIVES...
Publication number
20200109129
Publication date
Apr 9, 2020
Janssen Pharmaceutica N.V.
Ian STANSFIELD
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROAROMATIC DERIVATIVES AS NIK INHIBITORS
Publication number
20190359598
Publication date
Nov 28, 2019
Janssen Pharmaceutica N.V.
Ian Stansfield
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CYANOINDOLINE DERIVATIVES AS NIK INHIBITORS
Publication number
20190119299
Publication date
Apr 25, 2019
Janssen Pharmaceutica N.V.
Ian Stansfield
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NEW PYRAZOLE DERIVATIVES AS NIK INHIBITORS
Publication number
20170334900
Publication date
Nov 23, 2017
Janssen Pharmaceutica N.V.
George HYND
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW COMPOUNDS AS NIK INHIBITORS
Publication number
20170334906
Publication date
Nov 23, 2017
Janssen Pharmaceutica N.V.
George HYND
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW 1-(4-PYRIMIDINYL)-1H-PYRROLO[3,2-c]PYRIDINE DERIVATIVES AS NIK...
Publication number
20160257679
Publication date
Sep 8, 2016
Janssen Pharmaceutica N.V.
George HYND
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NEW 3-(1H-PYRAZOL-4-YL)-1H-PYRROLO[2,3-c]PYRIDINE DERIVATIVES AS NI...
Publication number
20160229851
Publication date
Aug 11, 2016
George HYND
C07 - ORGANIC CHEMISTRY
Information
Patent Application
3-(2-AMINOPYRIMIDIN-4-YL)-5-(3-HYDROXYPROPYNYL)-1H-PYRROLO[2,3-C]PY...
Publication number
20160075699
Publication date
Mar 17, 2016
Janssen Pharmaceutica N.V.
George HYND
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SULPHONE COMPOUNDS AND METHODS OF MAKING AND USING SAME
Publication number
20160051531
Publication date
Feb 25, 2016
Zafgen, Inc.
Hazel J. Dyke
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL COMPOUNDS
Publication number
20140179714
Publication date
Jun 26, 2014
Chiesi Farmaceutici s.p.A.
Toby Jonathan Blench
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIMIDINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF RESPIRATOR...
Publication number
20130150380
Publication date
Jun 13, 2013
Chiesi Farmaceutici s.p.A.
Christine Edwards
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIMIDINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF RESPIRATOR...
Publication number
20130123278
Publication date
May 16, 2013
Chiesi Farmaceutici s.p.A.
Christine Edwards
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL COMPOUNDS
Publication number
20130065913
Publication date
Mar 14, 2013
Chiesi Farmaceutici s.p.A.
Toby Jonathan Blench
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Sulphone Compounds and Methods of Making and Using Same
Publication number
20130053364
Publication date
Feb 28, 2013
Hazel J. Dyke
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PURINE DERIVATIVES USEFUL AS P13 KINASE INHIBITORS
Publication number
20110230464
Publication date
Sep 22, 2011
Paul Goldsmith
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TRICYCLIC HETEROCYCLIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE T...
Publication number
20110201593
Publication date
Aug 18, 2011
Genentech, Inc.
Srinivasan Babu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
THIAZOLOPYRIMIDINES AND THEIR USE AS INHIBITORS OF PHOSPHATIDYLINOS...
Publication number
20100190769
Publication date
Jul 29, 2010
Timothy Colin Hancox
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Indolizineacetic Acids and Their Therapeutic Use as Ligands of the...
Publication number
20100093751
Publication date
Apr 15, 2010
George Hynd
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PIPERIDINES AND RELATED COMPOUNDS FOR THE TREATMENT OF ALZHEIMER'S...
Publication number
20100048623
Publication date
Feb 25, 2010
Yudith Garcia
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PIPERIDINE DERIVATIVES FOR TREATMENT OF ALZHEIMER'S DISEASE
Publication number
20090186919
Publication date
Jul 23, 2009
MERCK SHARP & DOHME LIMITED
Andrew Madin
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Piperidines and Related Compounds for Treatment of Alzheimer's Disease
Publication number
20080021043
Publication date
Jan 24, 2008
MERCK SHARP & DOHME LTD.
Joanne Clare Hannam
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Tetrahydropyran compounds as tachykinin antagonists
Publication number
20060172999
Publication date
Aug 3, 2006
Olivier Dirat
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Tetrahydropyran derivatives and their use as therapeutic agents
Publication number
20050261285
Publication date
Nov 24, 2005
Olivier Dirat
C07 - ORGANIC CHEMISTRY
Information
Patent Application
5-ht7 receptor antagonists
Publication number
20050080077
Publication date
Apr 14, 2005
Neil Roy Curtis
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Sulfone derivatives as 5-HT7 receptor ligands
Publication number
20040229864
Publication date
Nov 18, 2004
Sylvie Bourrain
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Amidine derivatives as selective antagonists of ndma receptors
Publication number
20030119871
Publication date
Jun 26, 2003
Neil Roy Curtis
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1,4 substituted piperidinyl NMDA/NR2B antagonists
Publication number
20030018038
Publication date
Jan 23, 2003
MERCK & CO., Inc.
Wayne Thompson
C07 - ORGANIC CHEMISTRY