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last 30 patents
Information
Patent Grant
Solid forms of [(1S)-1-[(2S,4R,5R)-5-(5-amino-2-oxo-thiazolo[4,5-d]...
Patent number
12,012,420
Issue date
Jun 18, 2024
Hoffmann-La Roche, Inc.
Katja Grosse-Sender
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Solid forms of [(1S)-1-[(2S,4R,5R)-5-(5-amino-2-oxo-thiazolo[4,5-d]...
Patent number
12,012,421
Issue date
Jun 18, 2024
HOFFMANN-LA ROCHE INC.
Katja Grosse-Sender
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Solid forms of a compound of HBV core protein allosteric modifier
Patent number
11,873,302
Issue date
Jan 16, 2024
HOFFMANN-LA ROCHE INC.
Jing Xiong
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Solid forms of [(1 S)-1 -[(2S,4R,5R)-5-(5-amino-2-oxo-thiazolo[4,5-...
Patent number
11,230,559
Issue date
Jan 25, 2022
HOFFMANN-LA ROCHE INC.
Katja Grosse-Sender
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Process for the preparation of 3-substituted 5-amino-6H-thiazolo[4,...
Patent number
11,142,534
Issue date
Oct 12, 2021
HOFFMANN-LA ROCHE INC.
Junli Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Use of ring-fused bicyclic pyridyl derivatives as FGFR4 inhibitors
Patent number
10,507,201
Issue date
Dec 17, 2019
Novartis AG
Nicole Buschmann
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Use of ring-fused bicyclic pyridyl derivatives as FGFR4 inhibitors
Patent number
10,463,653
Issue date
Nov 5, 2019
Novartis AG
Lv Liao
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pharmaceutical combinations
Patent number
10,130,629
Issue date
Nov 20, 2018
Novartis AG
Nicole Buschmann
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Ring-fused bicyclic pyridyl derivatives as FGFR4 inhibitors
Patent number
9,896,449
Issue date
Feb 20, 2018
Novartis AG
Nicole Buschmann
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Particles of N-(5-cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-7-fo...
Patent number
9,802,917
Issue date
Oct 31, 2017
Novartis AG
Nicole Buschmann
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Ring-fused bicyclic pyridyl derivatives as FGFR4 inhibitors
Patent number
9,533,988
Issue date
Jan 3, 2017
Novartis AG
Nicole Buschmann
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Ring-fused bicyclic pyridyl derivatives as FGFR4 inhibitors
Patent number
9,266,883
Issue date
Feb 23, 2016
Novartis AG
Nicole Buschmann
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
SOLID FORMS OF A HBV CORE PROTEIN ALLOSTERIC MODIFIER
Publication number
20240116941
Publication date
Apr 11, 2024
HOFFMANN-LA ROCHE INC.
Jing Xiong
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SOLID FORMS OF [(1S)-1-[(2S,4R,5R)-5-(5-AMINO-2-OXO-THIAZOLO[4,5-D]...
Publication number
20220119414
Publication date
Apr 21, 2022
HOFFMANN-LA ROCHE INC.
Katja GROSSE-SENDER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SOLID FORMS OF [(1S)-1-[(2S,4R,5R)-5-(5-AMINO-2-OXO-THIAZOLO[4,5-D]...
Publication number
20220119415
Publication date
Apr 21, 2022
HOFFMANN-LA ROCHE INC.
Katja GROSSE-SENDER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SOLID FORMS OF A COMPOUND OF HBV CORE PROTEIN ALLOSTERIC MODIFIER
Publication number
20200308178
Publication date
Oct 1, 2020
HOFFMANN-LA ROCHE INC.
Jing Xiong
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SOLID FORMS OF [(1 S)-1 -[(2S,4R,5R)-5-(5-AMINO-2-OXO-THIAZOLO[4,5-...
Publication number
20200024288
Publication date
Jan 23, 2020
HOFFMANN-LA ROCHE INC.
Katja GROSSE-SENDER
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESS FOR THE PREPARATION OF 3-SUBSTITUTED 5-AMINO-6H-THIAZOLO[4,...
Publication number
20200024287
Publication date
Jan 23, 2020
HOFFMANN-LA ROCHE INC.
Junli CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
USE OF RING-FUSED BICYCLIC PYRIDYL DERIVATIVES AS FGFR4 INHIBITORS
Publication number
20190231760
Publication date
Aug 1, 2019
Novartis AG
Nicole BUSCHMANN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
USE OF RING-FUSED BICYCLIC PYRIDYL DERIVATIVES AS FGFR4 INHIBITORS
Publication number
20190076412
Publication date
Mar 14, 2019
Novartis AG
Nicole BUSCHMANN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
USE OF RING-FUSED BICYCLIC PYRIDYL DERIVATIVES AS FGFR4 INHIBITORS
Publication number
20180185341
Publication date
Jul 5, 2018
Novartis AG
Nicole BUSCHMANN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Ring-fused bicyclic pyridyl derivatives as FGFR4 inhibitors
Publication number
20170066766
Publication date
Mar 9, 2017
Novartis AG
Nicole Buschmann
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Particles of N-(5-cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-7-fo...
Publication number
20160304489
Publication date
Oct 20, 2016
Novartis AG
Nicole BUSCHMANN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Ring-fused bicyclic pyridyl derivatives as FGFR4 inhibitors
Publication number
20160102092
Publication date
Apr 14, 2016
Novartis AG
Nicole Buschmann
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Ring-fused bicyclic pyridyl derivatives as FGFR4 inhibitors
Publication number
20150119385
Publication date
Apr 30, 2015
Novartis AG
Nicole Buschmann
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE