Joseph A. Kozlowski

Person

Princeton, NJ, US

People

Patents Grantslast 30 patents

Information Patent Grant
Inhibitors of histone deacetylase useful for the treatment or preve...
- Patent number 11,976,069
- Issue date May 7, 2024
- Merck Sharp & Dohme LLC
- Wensheng Yu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Substituted N′-hydroxycarbamimidoyl-1,2,5-oxadiazole compounds as i...
- Patent number 11,034,661
- Issue date Jun 15, 2021
- Merck Sharp & Dohme Corp.
- Liangqin Guo
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Substituted n′-hydroxycarbamimidoyl-1,2,5-oxadiazole compounds as i...
- Patent number 10,988,487
- Issue date Apr 27, 2021
- Merck Sharp & Dohme Corp.
- Kun Liu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Azabicyclo[4.1.0]heptane allosteric modulators of the M4 muscarinic...
- Patent number 10,945,771
- Issue date Mar 16, 2021
- Merck Sharp & Dohme Corp.
- Dane James Clausen
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Substituted sulfoximine compounds as indoleamine 2,3-dioxygenase (I...
- Patent number 10,927,086
- Issue date Feb 23, 2021
- Merck Sharp & Dohme Corp.
- Kun Liu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Hepatitis C virus inhibitors
- Patent number 10,787,441
- Issue date Sep 29, 2020
- Merck Sharp & Dohme Corp.
- Joseph A. Kozlowski
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Compounds that are ERK inhibitors
- Patent number 10,759,805
- Issue date Sep 1, 2020
- Merck Sharp & Dohme Corp.
- Jongwon Lim
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Chromane-substituted tetracyclic compounds and uses thereof for the...
- Patent number 10,738,062
- Issue date Aug 11, 2020
- Merck Sharp & Dohme Corp.
- Wensheng Yu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Heterocycle-substituted tetracyclic compounds and methods of use th...
- Patent number 10,646,494
- Issue date May 12, 2020
- Merck Sharp & Dohme Corp.
- Wensheng Yu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Compounds as indoleamine 2,3-dioxygenase inhibitors
- Patent number 10,538,497
- Issue date Jan 21, 2020
- Merck Sharp & Dohme Corp.
- Yongxin Han
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Indazole and azaindazole Btk inhibitors
- Patent number 10,246,457
- Issue date Apr 2, 2019
- Merck Sharp & Dohme Corp.
- Tony Siu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Btk inhibitors
- Patent number 10,214,546
- Issue date Feb 26, 2019
- Merck Sharp & Dohme Corp.
- Jian Liu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Tertiary alcohol imidazopyrazine BTK inhibitors
- Patent number 10,208,047
- Issue date Feb 19, 2019
- Merck Sharp & Dohme Corp.
- Jian Liu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
BTK inhibitors
- Patent number 10,130,630
- Issue date Nov 20, 2018
- Merck Sharp & Dohme Corp.
- Jian Liu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Benzamide imidazopyrazine Btk inhibitors
- Patent number 10,087,188
- Issue date Oct 2, 2018
- Merck Sharp & Dohme Corp.
- Jian Liu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Compounds that are ERK inhibitors
- Patent number 10,065,967
- Issue date Sep 4, 2018
- Merck, Sharp & Dohme Corp.
- Jongwon Lim
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Substituted imidazo[1,5-a]pyrazines as Btk inhibitors
- Patent number 10,040,805
- Issue date Aug 7, 2018
- Merck Sharp & Dohme Corp.
- Jian Liu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
ERK inhibitors
- Patent number 9,988,397
- Issue date Jun 5, 2018
- Merck Sharp & Dohme Corp.
- Phieng Siliphaivanh
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
BTK inhibitors
- Patent number 9,834,554
- Issue date Dec 5, 2017
- Merck Sharp & Dohme Corp.
- Jian Liu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Fused tetracyclic heterocyclic compounds and methods of use thereof...
- Patent number 9,828,365
- Issue date Nov 28, 2017
- Merck Sharp & Dohme Corp.
- Joseph Kozlowski
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Fused tricyclic compounds and methods of use thereof for the treatm...
- Patent number 9,796,705
- Issue date Oct 24, 2017
- Merck Sharp & Dohme Corp.
- Kevin X. Chen
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Compounds that are ERK inhibitors
- Patent number 9,745,307
- Issue date Aug 29, 2017
- Merck Sharp & Dohme Corp.
- Jongwon Lim
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Btk inhibitors
- Patent number 9,637,486
- Issue date May 2, 2017
- Merck Sharp & Dohme Corp.
- Jian Liu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Inhibitors of IRAK4 activity
- Patent number 9,598,440
- Issue date Mar 21, 2017
- Merck Sharp & Dohme Corp.
- W. Michael Seganish
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Heterocycle-substituted tetracyclic compounds and methods of use th...
- Patent number 9,555,038
- Issue date Jan 31, 2017
- Merck Sharp & Dohme Corp.
- Wensheng Yu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Tetracyclic xanthene derivatives and methods of use thereof for the...
- Patent number 9,504,690
- Issue date Nov 29, 2016
- Merck Sharp & Dohme Corp.
- Craig A. Coburn
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Substituted benzamides and substituted pyridinecarboxamides as Btk...
- Patent number 9,481,682
- Issue date Nov 1, 2016
- Merck Sharp & Dohme Corp.
- Ronald M. Kim
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Substituted pyridine and pyrimidine derivatives and their use in tr...
- Patent number 9,433,621
- Issue date Sep 6, 2016
- Merck Sharp & Dohme Corp.
- Ashok Arasappan
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Fused tetracycle derivatives and methods of use thereof for the tre...
- Patent number 9,254,292
- Issue date Feb 9, 2016
- Merck Sharp & Dohme Corp.
- Craig A. Coburn
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Compounds that are ERK inhibitors
- Patent number 9,233,979
- Issue date Jan 12, 2016
- Merck Sharp & Dohme Corp.
- Kevin J. Wilson
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE

Patents Applicationslast 30 patents

Information Patent Application
NOVEL SUBSTITUTED PIPERAZINE AMIDE COMPOUNDS AS INDOLEAMINE 2,3-DIO...
- Publication number 20230008022
- Publication date Jan 12, 2023
- MERCK SHARP & DOHME CORP.
- Dane Clausen
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
INHIBITORS OF HISTONE DEACETYLASE-3 USEFUL FOR THE TREATMENT OF CAN...
- Publication number 20220177465
- Publication date Jun 9, 2022
- MERCK SHARP & DOHME CORP.
- Jian LIU
- C07 - ORGANIC CHEMISTRY
Information Patent Application
INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVE...
- Publication number 20220144837
- Publication date May 12, 2022
- MERCK SHARP & DOHME CORP.
- Wensheng Yu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVE...
- Publication number 20220089585
- Publication date Mar 24, 2022
- MERCK SHARP & DOHME CORP.
- Dane James Clausen
- C07 - ORGANIC CHEMISTRY
Information Patent Application
OXAZOLIDINONE COMPOUNDS AND METHODS OF USE THEREOF AS ANTIBACTERIAL...
- Publication number 20220081403
- Publication date Mar 17, 2022
- MERCK SHARP & DOHME CORP.
- Randall R. Miller
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVE...
- Publication number 20210403479
- Publication date Dec 30, 2021
- MERCK SHARP & DOHME CORP.
- Wensheng Yu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
NOVEL SUBSTITUTED PYRAZOLE COMPOUNDS AS INDOLEAMINE 2,3-DIOXYGENASE...
- Publication number 20210395240
- Publication date Dec 23, 2021
- MERCK SHARP & DOHME CORP.
- Dane Clausen
- C07 - ORGANIC CHEMISTRY
Information Patent Application
NOVEL ARYLOXYPIPERIDINE PYRAZOLE COMPOUNDS AS INDOLEAMINE 2,3-DIOXY...
- Publication number 20210330676
- Publication date Oct 28, 2021
- MERCK SHARP & DOHME CORP.
- Dane Clausen
- C07 - ORGANIC CHEMISTRY
Information Patent Application
INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVE...
- Publication number 20210276992
- Publication date Sep 9, 2021
- MERCK SHARP & DOHME CORP.
- Jian Liu
- C07 - ORGANIC CHEMISTRY
Information Patent Application
NOVEL SUBSTITUTED N'-HYDROXYCARBAMIMIDOYL-1,2,5-OXADIAZOLE COMPOUND...
- Publication number 20200231606
- Publication date Jul 23, 2020
- MERCK SHARP & DOHME CORP.
- Kun Liu
- C07 - ORGANIC CHEMISTRY
Information Patent Application
NOVEL SUBSTITUTED N'-HYDROXYCARBAMIMIDOYL-1,2,5-OXADIAZOLE COMPOUND...
- Publication number 20200102278
- Publication date Apr 2, 2020
- MERCK SHARP & DOHME CORP.
- Liangqin Guo
- C07 - ORGANIC CHEMISTRY
Information Patent Application
AZABICYCLO[4.1.0]HEPTANE ALLOSTERIC MODULATORS OF THE M4 MUSCARINI...
- Publication number 20200095262
- Publication date Mar 26, 2020
- MERCK SHARP & DOHME CORP.
- Dane James CLAUSEN
- C07 - ORGANIC CHEMISTRY
Information Patent Application
NOVEL SUBSTITUTED SULFOXIMINE COMPOUNDS AS INDOLEAMINE 2,3-DIOXYGEN...
- Publication number 20200095212
- Publication date Mar 26, 2020
- MERCK SHARP & DOHME CORP.
- Kun Liu
- C07 - ORGANIC CHEMISTRY
Information Patent Application
CHROMANE-SUBSTITUTED TETRACYCLIC COMPOUNDS AND USES THEREOF FOR THE...
- Publication number 20190185486
- Publication date Jun 20, 2019
- MERCK SHARP & DOHME CORP.
- Wensheng Yu
- C07 - ORGANIC CHEMISTRY
Information Patent Application
HEPATITIS C VIRUS INHIBITORS
- Publication number 20190127355
- Publication date May 2, 2019
- MERCK SHARP & DOHME CORP.
- Joseph A. Kozlowski
- C07 - ORGANIC CHEMISTRY
Information Patent Application
Silane-Containing Heterocyclic Compounds and Methods of Use Thereof...
- Publication number 20190002480
- Publication date Jan 3, 2019
- MERCK SHARP & DOHME CORP.
- Joseph A. Kozlowski
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
NOVEL COMPOUNDS AS INDOLEAMINE 2,3-DIOXYGENASE INHIBITORS
- Publication number 20180362482
- Publication date Dec 20, 2018
- MERCK SHARP & DOHME CORP.
- Yongxin Han
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
NOVEL COMPOUNDS THAT ARE ERK INHIBITORS
- Publication number 20180319804
- Publication date Nov 8, 2018
- MERCK SHARP & DOHME CORP.
- Jongwon Lim
- C07 - ORGANIC CHEMISTRY
Information Patent Application
AZACARBAZOLE BTK INHIBITORS
- Publication number 20180141962
- Publication date May 24, 2018
- MERCK SHARP & DOHME CORP.
- JIAN LIU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
INDAZOLE AND AZAINDAZOLE BTK INHIBITORS
- Publication number 20180127411
- Publication date May 10, 2018
- MERCK SHARP & DOHME CORP.
- Tony SIU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
BTK INHIBITORS
- Publication number 20180118766
- Publication date May 3, 2018
- MERCK SHARP & DOHME CORP.
- JIAN LIU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
BTK INHIBITORS
- Publication number 20180079752
- Publication date Mar 22, 2018
- MERCK SHARP & DOHME CORP.
- ADRIANUS PETRUS ANTONIUS DE MAN
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
IMIDAZOPYRAZINE ANALOGS WITH 3-TERTIARY CARBON SUBSTITUTIONS AS BTK...
- Publication number 20180009828
- Publication date Jan 11, 2018
- MERCK SHARP & DOHME CORP.
- JIAN LIU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
BIARYLETHER IMIDAZOPYRAZINE BTK INHIBITORS
- Publication number 20170362243
- Publication date Dec 21, 2017
- MERCK SHARP & DOHME CORP.
- JIAN LIU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
BENZAMIDE IMIDAZOPYRAZINE BTK INHIBITORS
- Publication number 20170362242
- Publication date Dec 21, 2017
- MERCK SHARP & DOHME CORP.
- JIAN LIU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
BTK INHIBITORS
- Publication number 20170349593
- Publication date Dec 7, 2017
- MERCK SHARP & DOHME CORP.
- JIAN LIU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
BTK INHIBITORS
- Publication number 20170340631
- Publication date Nov 30, 2017
- MERCK SHARP & DOHME CORP.
- JIAN LIU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
TERTIARY ALCOHOL IMIDAZOPYRAZINE BTK INHIBITORS
- Publication number 20170342076
- Publication date Nov 30, 2017
- MERCK SHARP & DOHME CORP.
- JIAN LIU
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
NOVEL COMPOUNDS THAT ARE ERK INHIBITORS
- Publication number 20170320882
- Publication date Nov 9, 2017
- MERCK SHARP & DOHME CORP.
- Jongwon Lim
- C07 - ORGANIC CHEMISTRY
Information Patent Application
ERK INHIBITORS
- Publication number 20170267695
- Publication date Sep 21, 2017
- MERCK SHARP & DOHME CORP.
- Phieng Siliphaivanh
- C07 - ORGANIC CHEMISTRY

Joseph A. Kozlowski

Person

Patents Grantslast 30 patents

Inhibitors of histone deacetylase useful for the treatment or preve...

Substituted N′-hydroxycarbamimidoyl-1,2,5-oxadiazole compounds as i...

Substituted n′-hydroxycarbamimidoyl-1,2,5-oxadiazole compounds as i...

Azabicyclo[4.1.0]heptane allosteric modulators of the M4 muscarinic...

Substituted sulfoximine compounds as indoleamine 2,3-dioxygenase (I...

Hepatitis C virus inhibitors

Compounds that are ERK inhibitors

Chromane-substituted tetracyclic compounds and uses thereof for the...

Heterocycle-substituted tetracyclic compounds and methods of use th...

Compounds as indoleamine 2,3-dioxygenase inhibitors

Indazole and azaindazole Btk inhibitors

Btk inhibitors

Tertiary alcohol imidazopyrazine BTK inhibitors

BTK inhibitors

Benzamide imidazopyrazine Btk inhibitors

Compounds that are ERK inhibitors

Substituted imidazo[1,5-a]pyrazines as Btk inhibitors

ERK inhibitors

BTK inhibitors

Fused tetracyclic heterocyclic compounds and methods of use thereof...

Fused tricyclic compounds and methods of use thereof for the treatm...

Compounds that are ERK inhibitors

Btk inhibitors

Inhibitors of IRAK4 activity

Heterocycle-substituted tetracyclic compounds and methods of use th...

Tetracyclic xanthene derivatives and methods of use thereof for the...

Substituted benzamides and substituted pyridinecarboxamides as Btk...

Substituted pyridine and pyrimidine derivatives and their use in tr...

Fused tetracycle derivatives and methods of use thereof for the tre...

Compounds that are ERK inhibitors

Patents Applicationslast 30 patents

NOVEL SUBSTITUTED PIPERAZINE AMIDE COMPOUNDS AS INDOLEAMINE 2,3-DIO...

INHIBITORS OF HISTONE DEACETYLASE-3 USEFUL FOR THE TREATMENT OF CAN...

INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVE...

INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVE...

OXAZOLIDINONE COMPOUNDS AND METHODS OF USE THEREOF AS ANTIBACTERIAL...

INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVE...

NOVEL SUBSTITUTED PYRAZOLE COMPOUNDS AS INDOLEAMINE 2,3-DIOXYGENASE...

NOVEL ARYLOXYPIPERIDINE PYRAZOLE COMPOUNDS AS INDOLEAMINE 2,3-DIOXY...

INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVE...

NOVEL SUBSTITUTED N'-HYDROXYCARBAMIMIDOYL-1,2,5-OXADIAZOLE COMPOUND...

NOVEL SUBSTITUTED N'-HYDROXYCARBAMIMIDOYL-1,2,5-OXADIAZOLE COMPOUND...

AZABICYCLO[4.1.0]HEPTANE ALLOSTERIC MODULATORS OF THE M4 MUSCARINI...

NOVEL SUBSTITUTED SULFOXIMINE COMPOUNDS AS INDOLEAMINE 2,3-DIOXYGEN...

CHROMANE-SUBSTITUTED TETRACYCLIC COMPOUNDS AND USES THEREOF FOR THE...

HEPATITIS C VIRUS INHIBITORS

Silane-Containing Heterocyclic Compounds and Methods of Use Thereof...

NOVEL COMPOUNDS AS INDOLEAMINE 2,3-DIOXYGENASE INHIBITORS

NOVEL COMPOUNDS THAT ARE ERK INHIBITORS

AZACARBAZOLE BTK INHIBITORS

INDAZOLE AND AZAINDAZOLE BTK INHIBITORS

BTK INHIBITORS

BTK INHIBITORS

IMIDAZOPYRAZINE ANALOGS WITH 3-TERTIARY CARBON SUBSTITUTIONS AS BTK...

BIARYLETHER IMIDAZOPYRAZINE BTK INHIBITORS

BENZAMIDE IMIDAZOPYRAZINE BTK INHIBITORS

BTK INHIBITORS

BTK INHIBITORS

TERTIARY ALCOHOL IMIDAZOPYRAZINE BTK INHIBITORS

NOVEL COMPOUNDS THAT ARE ERK INHIBITORS

ERK INHIBITORS