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Joseph E. Leenaerts
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Hoogstraten, BE
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Patents Grants
last 30 patents
Information
Patent Grant
Tau PET imaging ligands
Patent number
11,168,068
Issue date
Nov 9, 2021
JANSSEN PHARMACEUTICA NV
José Ignacio Andrés-Gil
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Morpholinothiazoles as alpha 7 positive allosteric modulators
Patent number
8,637,510
Issue date
Jan 28, 2014
JANSSEN PHARMACEUTICA NV
Gregor James Macdonald
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Quinoline or isoquinoline substituted P2X7 antagonists
Patent number
8,431,704
Issue date
Apr 30, 2013
JANSSEN PHARMACEUTICA NV
Christopher John Love
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 1-piperidin-4-yl-4-pyrrolidin-3-yl-piperazine derivativ...
Patent number
7,795,261
Issue date
Sep 14, 2010
Janssen Pharmaceutica N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Use of anti-histaminics for acute reduction of elevated intracrania...
Patent number
7,732,437
Issue date
Jun 8, 2010
Janssen Pharmaceutica, N.V.
Frank Tegtmeier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 1-piperidin-3-yl-4-piperidin-4-yl-piperazine derivative...
Patent number
7,572,786
Issue date
Aug 11, 2009
Janssen Pharmaceutica, N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 4-(4-piperidin-4-yl-piperazin-1-yl)-azepane derivatives...
Patent number
7,514,424
Issue date
Apr 7, 2009
JANSSEN PHARMACEUTICA NV
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted tetracyclic imidazole derivatives, processes for their...
Patent number
7,476,662
Issue date
Jan 13, 2009
Janssen Pharmaceutica N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 1-piperidin-4-yl-4-azetidin-3-yl-piperazine derivatives...
Patent number
7,435,736
Issue date
Oct 14, 2008
Janssen Pharmaceutica, N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 1,4,-di-piperidin-4-yl-piperazine derivatives and their...
Patent number
7,410,970
Issue date
Aug 12, 2008
Janssen Pharmaceutica, N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 4-phenyl-4-[1H-imidazol-2-yl]-piperidine derivatives fo...
Patent number
7,390,822
Issue date
Jun 24, 2008
Janssen Pharmaceutica, N.V.
Frans Eduard Janssens
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted 4-phenyl-4-(1H-imidazol-2-yl)-piperidine derivatives an...
Patent number
7,282,508
Issue date
Oct 16, 2007
Janssen Pharmaceutica N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Antihistaminic spiro compounds
Patent number
7,148,214
Issue date
Dec 12, 2006
Janssen Pharmaceutica, N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Antihistaminic spiro compounds
Patent number
7,087,595
Issue date
Aug 8, 2006
Janssen Pharmaceutica, N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1-(1,2-disubstituted piperidinyl)-4-substituted piperazine derivatives
Patent number
6,521,621
Issue date
Feb 18, 2003
Janssen Pharmaceutica N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Fused imidazole derivatives as multidrug resistance modulators
Patent number
6,476,018
Issue date
Nov 5, 2002
JANSSEN PHARMACEUTICA NV
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1-(1,2-Disubstituted piperidinyl)-4-substituted piperazine derivatives
Patent number
RE37886
Issue date
Oct 15, 2002
Janssen Pharmaceuticals, N.V.
Frans E. Janssens
514 - Drug, bio-affecting and body treating compositions
Information
Patent Grant
1-(1,2-disubstituted piperidinyl)-4 (fused imidazole)-piperidine de...
Patent number
6,251,894
Issue date
Jun 26, 2001
Janssen Pharmaceuticals N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Fused imidazole derivatives as multidrug resistance modulators
Patent number
6,218,381
Issue date
Apr 17, 2001
Janssen Pharmaceutica N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1- (1,2-disubstituted piperidinyl) -4-substituted piperazine deriva...
Patent number
6,197,772
Issue date
Mar 6, 2001
Janssen Pharmaceutica N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
(Benzimidazolyl- and imidazopyridinyl) containing 1-(1,2-disubstitu...
Patent number
6,110,939
Issue date
Aug 29, 2000
Janssen Pharmaceutica N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Antiallergic imidazoazepines
Patent number
5,674,866
Issue date
Oct 7, 1997
Janssen Pharmaceutica N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazo [1,2-A] (pyrrolo, thieno or furano) [2,3-D] azepine derivat...
Patent number
5,629,308
Issue date
May 13, 1997
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazo[2,1-b]benzazepine derivatives, compositions and method of use
Patent number
5,468,743
Issue date
Nov 21, 1995
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazo[1,2-a](pyrrolo, thieno or furano) [3,2a-d]azepine derivativ...
Patent number
5,461,050
Issue date
Oct 24, 1995
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Hydroxyalkylfuranyl derivatives
Patent number
5,272,150
Issue date
Dec 21, 1993
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
COMPOUNDS
Publication number
20230202989
Publication date
Jun 29, 2023
Janssen Pharmaceutica N.V.
Michael Eric MURATORE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLO[1,2-D][1,2,4]TRIAZINE-2-YL-ACETAMIDES AS INHIBITORS OF THE...
Publication number
20230183248
Publication date
Jun 15, 2023
Janssen Pharmaceutica N.V.
Daniel OEHLRICH
C07 - ORGANIC CHEMISTRY
Information
Patent Application
OGA INHIBITOR COMPOUNDS
Publication number
20230099293
Publication date
Mar 30, 2023
Janssen Pharmaceutica N.V.
José Manuel BARTOLOMÉ-NEBREDA
C07 - ORGANIC CHEMISTRY
Information
Patent Application
OGA INHIBITOR COMPOUNDS
Publication number
20230058733
Publication date
Feb 23, 2023
Janssen Pharmaceutica N.V.
José Manuel BARTOLOMÉ-NEBREDA
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TAU PET IMAGING LIGANDS
Publication number
20220024896
Publication date
Jan 27, 2022
Janssen Pharmaceutica N.V.
José Ignacio Andrés-Gil
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TAU PET IMAGING LIGANDS
Publication number
20210283277
Publication date
Sep 16, 2021
Diederik Willem Elisabeth MOECHARS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
OGA INHIBITOR COMPOUNDS
Publication number
20210277003
Publication date
Sep 9, 2021
Janssen Pharmaceutica N.V.
José Manuel Bartolomé-Nebreda
C07 - ORGANIC CHEMISTRY
Information
Patent Application
OGA INHIBITOR COMPOUNDS
Publication number
20210130352
Publication date
May 6, 2021
Janssen Pharmaceutica N.V.
José Manuel Bartolomé-Nebreda
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TAU PET IMAGING LIGANDS
Publication number
20190284165
Publication date
Sep 19, 2019
Janssen Pharnaceutica NV
Jos ANDRéS-GIL Andres-Gil
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TAU PET IMAGING LIGANDS
Publication number
20190038784
Publication date
Feb 7, 2019
Diederik Willem Elisabeth MOECHARS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MORPHOLINOTHIAZOLES AS ALPHA 7 POSITIVE ALLOSTERIC MODULATORS
Publication number
20120238561
Publication date
Sep 20, 2012
Gregor James Macdonald
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINOLINE OR ISOQUINOLINE SUBSTITUTED P2X7 ANTAGONISTS
Publication number
20110092481
Publication date
Apr 21, 2011
Janssen Pharmaceutica N.V.
Christopher John Love
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel Substituted 4-Phenyl-4[H-Imidazol-2-YL]-Piperidine Derivative...
Publication number
20080096925
Publication date
Apr 24, 2008
Janssen Pharmaceutica N.V.
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel Formulations For Opioid-Based Treatments Of Pain Comprising 1...
Publication number
20080070924
Publication date
Mar 20, 2008
Frans Eduard Janssens
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Substituted 4-Alkyl-And 4-Alkanoyl-Piperidine Derivatives And Their...
Publication number
20070213346
Publication date
Sep 13, 2007
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Substituted 4-phenyl-4-[1h-imidazol-2-yl]-piperidine derivatives as...
Publication number
20060287345
Publication date
Dec 21, 2006
Thomas Horst Wolfgang Steckler
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Substitituted 1-piperidin-3-yl-piperidin 4-yl-piperazine derivative...
Publication number
20060252747
Publication date
Nov 9, 2006
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Substituted 1,4,-di-piperidin-4-yl-piperazine derivatives and their...
Publication number
20060167008
Publication date
Jul 27, 2006
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel formulations of opioid-based treatments of pain comprising su...
Publication number
20060128721
Publication date
Jun 15, 2006
Frans Eduard Janssens
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Substituted 1-piperidin-4-yl-4-azetidin-3-yl-piperazine derivatives...
Publication number
20060074069
Publication date
Apr 6, 2006
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Substituted 4-(4-piperidin-4-yl-piperazin-1-yl)-azepane derivatives...
Publication number
20060058285
Publication date
Mar 16, 2006
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Substituted 1-piperidin-4-yl-4-pyrrolidin-3-yl-piperazine derivativ...
Publication number
20060040950
Publication date
Feb 23, 2006
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Use of anti-histaminics for acute reduction of elevated intracrania...
Publication number
20050070525
Publication date
Mar 31, 2005
Frank Tegtmeier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Antihistaminic spiro compounds
Publication number
20050026901
Publication date
Feb 3, 2005
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Substituted 4-phenyl-4-[1h-imidazol-2-yl]-piperidine derivatives fo...
Publication number
20050004170
Publication date
Jan 6, 2005
Frans Eduard Janssens
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Novel substituted 4-phenyl-4-{1h-imidazol-2-yl}-piperidine derivati...
Publication number
20040260096
Publication date
Dec 23, 2004
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel substituted tetracyclic imidazole derivatives, processes for...
Publication number
20040167138
Publication date
Aug 26, 2004
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Fused imidazole derivatives as multidrug resistance modulators
Publication number
20030087895
Publication date
May 8, 2003
Frans Eduard Janssens
C07 - ORGANIC CHEMISTRY