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Lawrence Blas Perez
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Hakettstown, NJ, US
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Patents Grants
last 30 patents
Information
Patent Grant
N-azaspirocycloalkane substituted N-heteroaryl compounds and compos...
Patent number
11,952,386
Issue date
Apr 9, 2024
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds and compositions for inhibiting the activity of SHP2
Patent number
11,905,283
Issue date
Feb 20, 2024
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1-Pyridazin-/triazin-3-yl-piper(-azine)/idine/pyrolidine derivative...
Patent number
11,401,259
Issue date
Aug 2, 2022
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-azaspirocycloalkane substituted N-heteroaryl compounds and compos...
Patent number
10,968,235
Issue date
Apr 6, 2021
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds and compositions for inhibiting the activity of SHP2
Patent number
10,934,285
Issue date
Mar 2, 2021
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1-pyridazin-/triazin-3-yl-piper(-azine)/idine/pyrolidine derivative...
Patent number
10,774,065
Issue date
Sep 15, 2020
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-azaspirocycloalkane substituted N-heteroaryl compounds and compos...
Patent number
10,336,774
Issue date
Jul 2, 2019
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1-(triazin-3-yl/pyridazin-3-yl)-piper(-azine)idine derivatives and...
Patent number
10,301,278
Issue date
May 28, 2019
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds and compositions for inhibiting the activity of SHP2
Patent number
10,287,266
Issue date
May 14, 2019
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1-pyridazin-/triazin-3-yl-piper(-azine)/idine/pyrolidine derivative...
Patent number
10,093,646
Issue date
Oct 9, 2018
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-azaspirocycloalkane substituted N-heteroaryl compounds and compos...
Patent number
10,077,276
Issue date
Sep 18, 2018
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-azaspirocycloalkane substituted N-heteroaryl compounds and compos...
Patent number
9,938,295
Issue date
Apr 10, 2018
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1-(triazin-3-yl/pyridazin-3-yl)-piper(-azine)idine derivatives and...
Patent number
9,815,813
Issue date
Nov 14, 2017
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolopyrimidine compounds as inhibitors of CDK4/6
Patent number
9,309,252
Issue date
Apr 12, 2016
Novartis AG
Christopher Thomas Brain
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolopyrimidine compounds as inhibitors of CDK4/6
Patent number
8,957,074
Issue date
Feb 17, 2015
Novartis AG
Christopher Thomas Brain
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds and methods for inhibiting the interaction of BCL protein...
Patent number
8,609,706
Issue date
Dec 17, 2013
Infinity Discovery, Inc.
Alfredo C. Castro
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Imidazole derivatives and their use as modulators of cyclin depende...
Patent number
8,598,217
Issue date
Dec 3, 2013
Astex Therapeutics Ltd.
Steven Howard
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzyl and pyridinyl derivatives as modulators of the hedgehog sign...
Patent number
8,536,168
Issue date
Sep 17, 2013
Novartis AG
Miao Dai
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds and methods for inhibiting the interaction of BCL protein...
Patent number
8,178,690
Issue date
May 15, 2012
Infinity Pharmaceuticals, Inc.
Alfredo C. Castro
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds and methods for inhibiting the interaction of BCL protein...
Patent number
7,928,244
Issue date
Apr 19, 2011
Infinity Discovery, Inc.
Alfredo C. Castro
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bis-aromatic alkanols
Patent number
7,169,817
Issue date
Jan 30, 2007
IRM LLC
Shifeng Pan
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Deacetylase inhibitors
Patent number
7,067,551
Issue date
Jun 27, 2006
Novartis AG
Stacy W Remiszewski
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Deacetylase inhibitors
Patent number
6,833,384
Issue date
Dec 21, 2004
Novartis AG
Stacy William Remiszewski
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Deacetylase inhibitors
Patent number
6,552,065
Issue date
Apr 22, 2003
Novartis AG
Stacy William Remiszewski
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20220396585
Publication date
Dec 15, 2022
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1-PYRIDAZIN-/TRIAZIN-3-YL-PIPER(-AZINE)/IDINE/PYROLIDINE DERIVATIVE...
Publication number
20220348553
Publication date
Nov 3, 2022
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20220073537
Publication date
Mar 10, 2022
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20210371429
Publication date
Dec 2, 2021
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF SHP2
Publication number
20210300919
Publication date
Sep 30, 2021
Novartis AG
Zhuoliang CHEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
1-PYRIDAZIN-/TRIAZIN-3-YL-PIPER(-AZINE)/IDINE/PYROLIDINE DERIVATIVE...
Publication number
20200369643
Publication date
Nov 26, 2020
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20200181168
Publication date
Jun 11, 2020
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF SHP2
Publication number
20200002330
Publication date
Jan 2, 2020
Novartis AG
Zhuoliang CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1-PYRIDAZIN-/TRIAZIN-3-YL-PIPER(-AZINE)/IDINE/PYROLIDINE DERIVATIVE...
Publication number
20180362496
Publication date
Dec 20, 2018
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20180201623
Publication date
Jul 19, 2018
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF SHP2
Publication number
20180186770
Publication date
Jul 5, 2018
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1-(TRIAZIN-3-YL/PYRIDAZIN-3-YL)-PIPER(-AZINE)IDINE DERIVATIVES AND...
Publication number
20180065949
Publication date
Mar 8, 2018
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1-PYRIDAZIN-/TRIAZIN-3-YL-PIPER(-AZINE)/IDINE/PYROLIDINE DERIVATIVE...
Publication number
20170204080
Publication date
Jul 20, 2017
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20170015680
Publication date
Jan 19, 2017
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1-(TRIAZIN-3-YL/PYRIDAZIN-3-YL)-PIPER(-AZINE)IDINE DERIVATIVES AND...
Publication number
20170001975
Publication date
Jan 5, 2017
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOPYRIMIDINE COMPOUNDS AS INHIBITORS OF CDK4/6
Publication number
20150099737
Publication date
Apr 9, 2015
Novartis AG
Christopher Thomas BRAIN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DEUTERATED PYRROLOPYRIMIDINE COMPOUNDS AS INHIBITORS OF CDK4/6
Publication number
20130203765
Publication date
Aug 8, 2013
Novartis AG
Christopher Thomas Brain
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOPYRIMIDINE COMPOUNDS AS INHIBITORS OF CDK4/6
Publication number
20130150342
Publication date
Jun 13, 2013
Novartis AG
Christopher Thomas Brain
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Compounds and Methods for Inhibiting the Interaction of BCL Protein...
Publication number
20130131063
Publication date
May 23, 2013
Infinity Pharmaceuticals, Inc.
Alfredo C. Castro
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMIDAZOLE DERIVATIVES AND THEIR USE AS MODULATORS OF CYCLIN DEPENDE...
Publication number
20120101064
Publication date
Apr 26, 2012
ASTEX THERAPEUTICS LIMITED
Steven Howard
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Compounds and Methods for Inhibiting the Interaction of BCL Protein...
Publication number
20110213145
Publication date
Sep 1, 2011
Infinity Discovery, Inc.
Alfredo C. Castro
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Organic Compounds and Their Uses
Publication number
20100069368
Publication date
Mar 18, 2010
Miao Dai
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS
Publication number
20100048539
Publication date
Feb 25, 2010
IRM LLC
Donatella Chianelli
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Organic Compounds
Publication number
20090306107
Publication date
Dec 10, 2009
Novartis AG
Lawrence Blas Perez
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DEACETYLASE INHIBITORS
Publication number
20080176849
Publication date
Jul 24, 2008
Stacy William Remiszewski
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Compounds and Methods for Inhibiting the Interaction of BCL Protein...
Publication number
20080114167
Publication date
May 15, 2008
Infinity Discovery, Inc.
Alfredo C. CASTRO
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Trifluoromethyl substituted benzamides as kinase inhibitors
Publication number
20080096883
Publication date
Apr 24, 2008
Giorgio Caravatti
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1,4-Disubstituted isoquinilone derivatives as raf-kinase inhibitors...
Publication number
20070060582
Publication date
Mar 15, 2007
Cynthia Anne Fink
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Deacetylase inhibitors
Publication number
20060189674
Publication date
Aug 24, 2006
Stacy William Remiszewski
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Trifluoromethyl substituted benzamides as kinase inhibitors
Publication number
20060035897
Publication date
Feb 16, 2006
Giorgio Caravatti
C07 - ORGANIC CHEMISTRY