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Patents Grants
last 30 patents
Information
Patent Grant
Salt of LSD1 inhibitor and a polymorph thereof
Patent number
12,024,494
Issue date
Jul 2, 2024
CSPC Zhongqi Pharmaceutical Technology (Shijiazhuang) Co., Ltd.
Lele Zhao
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzo 2-azaspiro[4.4]nonane compound and use thereof
Patent number
11,760,751
Issue date
Sep 19, 2023
Helioeast Science & Technology Co., Ltd.
Lingyun Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Salt types, crystal forms, and preparation methods for benzopyrazol...
Patent number
11,702,400
Issue date
Jul 18, 2023
Medshine Discovery Inc.
Lingyun Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cyclopropylamine compound as LSD1 inhibitor and use thereof
Patent number
11,649,245
Issue date
May 16, 2023
HELIOEAST PHARMACEUTICAL CO., LTD.
Lingyun Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazole compounds as LSD1 inhibitors and applications thereof
Patent number
11,524,941
Issue date
Dec 13, 2022
Medshine Discovery Inc.
Lingyun Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Crystal and salt forms of tricyclic compound and preparation proces...
Patent number
11,465,995
Issue date
Oct 11, 2022
Medshine Discovery Inc.
Peng Zhang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
LSD1 inhibitor and preparation method and application thereof
Patent number
11,433,053
Issue date
Sep 6, 2022
Medshine Discovery Inc.
Lingyun Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Aryl-phosphorus-oxygen compound as EGFR kinase inhibitor
Patent number
11,390,625
Issue date
Jul 19, 2022
Chia Tai Tianqing Pharmaceutical Group Co., Ltd.
Lingyun Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Hydroxyl purine compounds and applications thereof
Patent number
RE49128
Issue date
Jul 12, 2022
GUANGDONG RAYNOVENT BIOTECH CO., LTD.
Lingyun Wu
Information
Patent Grant
Benzopyrazole compound used as RHO kinase inhibitor
Patent number
11,345,678
Issue date
May 31, 2022
Medshine Discovery Inc.
Lingyun Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
S1P1 agonist and application thereof
Patent number
11,192,886
Issue date
Dec 7, 2021
MEDSHINE DISCOVERY INC.
Lingyun Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Sulfonyl-substituted isoquinolines as inhibitors of RHO kinase and...
Patent number
11,155,559
Issue date
Oct 26, 2021
CHINA RESOURCES PHARMACEUTICAL HOLDINGS COMPANY LIMITED
Yuanshan Yao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dimethylphosphine oxide compound
Patent number
11,046,720
Issue date
Jun 29, 2021
GUIZHOU INOCHINI TECHNOLOGY CO., LTD
Lingyun Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Quinazoline compound for EGFR inhibition
Patent number
11,040,984
Issue date
Jun 22, 2021
Medshine Discovery Inc.
Xile Liu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Spiro compound and use thereof
Patent number
10,981,900
Issue date
Apr 20, 2021
MEDSHINE DISCOVERY INC.
Peng Zhang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Crystal form A of 7-(cyclopropylmethyl)-1-(((cis )-4-hydroxy-4-meth...
Patent number
10,399,981
Issue date
Sep 3, 2019
GUANGDONG RAYNOVENT BIOTECH CO., LTD.
Lingyun Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Hydroxyl purine compounds and use thereof
Patent number
10,278,973
Issue date
May 7, 2019
GUANGDONG RAYNOVENT BIOTECH CO., LTD.
Lingyun Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Hydroxyl purine compounds and applications thereof
Patent number
10,098,885
Issue date
Oct 16, 2018
GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD
Lingyun Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Isoquinolinesulfonyl derivative as RHO kinase inhibitor
Patent number
9,856,264
Issue date
Jan 2, 2018
Medshine Discovery Inc.
Lingyun Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Triazolyl derivatives as Syk inhibitors
Patent number
9,586,931
Issue date
Mar 7, 2017
Merck Sharp & Dohme Corp.
Michelle R. Machacek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
BENZOXAZINONE DERIVATIVES
Publication number
20250034099
Publication date
Jan 30, 2025
CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD
Lingyun WU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
5-SUBSTITUTED PYRIDINE-2(1H)-KETONE COMPOUND AND USE THEREOF
Publication number
20240383906
Publication date
Nov 21, 2024
JIANGSU KANION PHARMACEUTICAL CO., LTD.
Xiongbin XU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SALT FORM OF PYRROLOTRIAZINE COMPOUND, CRYSTAL FORM THEREOF, AND PR...
Publication number
20240254144
Publication date
Aug 1, 2024
JUMBO DRUG BANK CO., LTD
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-CARBAMATE SUBSTITUTED HETEROARYL RING DERIVATIVES
Publication number
20240208945
Publication date
Jun 27, 2024
MEDSHINE DISCOVERY INC.
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
THIOPHENE COMPOUND AND APPLICATION THEREOF
Publication number
20240199571
Publication date
Jun 20, 2024
MEDSHINE DISCOVERY INC.
Lingyun WU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
OXADIAZOLE-SUBSTITUTED SPIROCYCLIC COMPOUND AND APPLICATION THEREOF
Publication number
20240182457
Publication date
Jun 6, 2024
HELIOEAST PHARMACEUTICAL CO., LTD.
Lingyun WU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRIDAZINE PHENOL DERIVATIVES
Publication number
20240166610
Publication date
May 23, 2024
MEDSHINE DISCOVERY INC.
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FUSED RING DERIVATIVES CONTAINING 1,4-OXAZEPANE
Publication number
20240150335
Publication date
May 9, 2024
MEDSHINE DISCOVERY INC.
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SALT FORM OF ISOQUINOLINONE TYPE COMPOUND AS ROCK INHIBITOR AND PRE...
Publication number
20230331696
Publication date
Oct 19, 2023
GUANGZHOU OCUSUN OPHTHALMIC BIOTECHNOLOGY CO., LTD.
Jian GE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ACETOPHENONE OXIME COMPOUND AND APPLICATION THEREOF
Publication number
20230295076
Publication date
Sep 21, 2023
MEDSHINE DISCOVERY INC.
Lingyun Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZO 2-AZASPIRO[4.4]NONANE COMPOUND AND USE THEREOF
Publication number
20230126480
Publication date
Apr 27, 2023
HELIOEAST PHARMACEUTICAL CO., LTD.
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TRICYCLIC COMPOUNDS AND USE THEREOF
Publication number
20230124301
Publication date
Apr 20, 2023
HELIOEAST PHARMACEUTICAL CO., LTD.
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ISOQUINOLINONE DERIVATIVES SERVING AS ROCK PROTEIN KINASE INHIBITOR...
Publication number
20230024516
Publication date
Jan 26, 2023
GUANGZHOU OCUSUN OPHTHALMIC BIOTECHNOLOGY CO., LTD.
Yizhi Liu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUND AS SMALL MOLECULE INHIBITOR PD-1/PD-L1 AND APPLICATION THE...
Publication number
20220402917
Publication date
Dec 22, 2022
MEDSHINE DISCOVERY INC.
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SALT TYPES, CRYSTAL FORMS, AND PREPARATION METHODS FOR BENZOPYRAZOL...
Publication number
20220380336
Publication date
Dec 1, 2022
MEDSHINE DISCOVERY INC.
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUND AS PORCUPINE INHIBITOR AND USE THEREOF
Publication number
20220281873
Publication date
Sep 8, 2022
MEDSHINE DISCOVERY INC.
Xiongbin XU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLOTRIAZINE COMPOUNDS ACTING AS MNK INHIBITOR
Publication number
20220281895
Publication date
Sep 8, 2022
JUMBO DRUG BANK CO., LTD.
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SALT OF EGFR INHIBITOR, CRYSTAL FORM, AND PREPARATION METHOD THEREFOR
Publication number
20220119431
Publication date
Apr 21, 2022
CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD.
Lingyun WU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CYCLOPROPYLAMINE COMPOUND AS LSD1 INHIBITOR AND USE THEREOF
Publication number
20220119401
Publication date
Apr 21, 2022
MEDSHINE DISCOVERY INC.
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrazole Compounds As LSD1 Inhibitors And Applications Thereof
Publication number
20220064126
Publication date
Mar 3, 2022
MEDSHINE DISCOVERY INC.
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZOPYRAZOLE COMPOUND USED AS RHO KINASE INHIBITOR
Publication number
20210371393
Publication date
Dec 2, 2021
MEDSHINE DISCOVERY INC.
Lingyun WU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SALT OF LSD1 INHIBITOR AND A POLYMORPH THEREOF
Publication number
20210317096
Publication date
Oct 14, 2021
CSPC ZHONGQI PHARMACEUTICAL TECHNOLOGY (SHIJIAZHUANG) CO., LTD.
Lele ZHAO
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
S1P1 AGONIST AND APPLICATION THEREOF
Publication number
20210300908
Publication date
Sep 30, 2021
SHIJIAZHUANG SAGACITY NEW DRUG DEVELOPMENT CO., LTD.
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DIMETHYLPHOSPHINE OXIDE COMPOUND
Publication number
20210147453
Publication date
May 20, 2021
GUIZHOU INOCHINI TECHNOLOGY CO., LTD
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
LSD1 INHIBITOR AND PREPARATION METHOD AND APPLICATION THEREOF
Publication number
20200345700
Publication date
Nov 5, 2020
MEDSHINE DISCOVERY INC.
Lingyun WU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CRYSTAL AND SALT FORMS OF TRICYCLIC COMPOUND AND PREPARATION PROCES...
Publication number
20200339553
Publication date
Oct 29, 2020
Peng ZHANG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Aryl-Phosphorus-Oxygen Compound As EGFR Kinase Inhibitor
Publication number
20200207768
Publication date
Jul 2, 2020
CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD.
Lingyun WU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ISOQUINOLINYLSULFONYL DERIVATIVE AND USE THEREOF
Publication number
20200207772
Publication date
Jul 2, 2020
CHINA RESOURCES PHARMACEUTICAL HOLDINGS COMPANY LIMITED
Yuanshan YAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINAZOLINE COMPOUND FOR EGFR INHIBITION
Publication number
20200190107
Publication date
Jun 18, 2020
MEDSHINE DISCOVERY INC.
Xile LIU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SPIRO COMPOUND AND USE THEREOF
Publication number
20200048235
Publication date
Feb 13, 2020
MEDSHINE DISCOVERY INC.
Peng ZHANG
C07 - ORGANIC CHEMISTRY