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2340 Beerse, BE
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Patents Grants
last 30 patents
Information
Patent Grant
Macrocyclic quinazole derivatives and their use as MTKI
Patent number
10,208,062
Issue date
Feb 19, 2019
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Macrocylic pyrimidine derivatives
Patent number
10,017,509
Issue date
Jul 10, 2018
JANSSEN PHARMACEUTICA NV
Gaston Stanislas Marcella Diels
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Macrocyclic quinazole derivatives and their use as MTKI
Patent number
9,688,691
Issue date
Jun 27, 2017
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Quinazoline derivatives
Patent number
9,273,013
Issue date
Mar 1, 2016
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrido and pyrimidopyrimidine derivatives as anti-profilerative agents
Patent number
8,933,067
Issue date
Jan 13, 2015
JANSSEN PHARMACEUTICA NV
Eddy Jean Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrido-and pyrimidopyrimidine derivatives as anti-proliferative agents
Patent number
8,772,272
Issue date
Jul 8, 2014
Janssen Pharmaceutica N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
MTKI quinazoline derivatives
Patent number
8,492,377
Issue date
Jul 23, 2013
JANSSEN PHARMACEUTICA NV
Alexandra Papanikos
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Quinazoline derivatives
Patent number
8,394,786
Issue date
Mar 12, 2013
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2,4 (4,6) pyrimidine derivatives
Patent number
8,394,955
Issue date
Mar 12, 2013
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2,4 (4,6) pyrimidine derivatives
Patent number
8,148,388
Issue date
Apr 3, 2012
Janssen Pharmaceutica, N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Macrocyclic quinazoline derivatives as antiproliferative agents
Patent number
7,648,975
Issue date
Jan 19, 2010
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibi...
Patent number
7,560,458
Issue date
Jul 14, 2009
Janssen Pharmaceutica, N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heteroaryl amines as glycogen synthase kinase 3β inhibitors (GSK3...
Patent number
7,514,445
Issue date
Apr 7, 2009
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibi...
Patent number
7,449,465
Issue date
Nov 11, 2008
Janssen Pharmaceutica, N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Angiogenesis inhibiting 5-substituted-1,2,4-thiadiazolyl derivatives
Patent number
7,208,503
Issue date
Apr 24, 2007
Janssen Pharmaceutica N.V.
Raymond Antoine Stokbroekx
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Amide derivatives as glycogen synthase kinase 3-β inhibitors
Patent number
7,183,288
Issue date
Feb 27, 2007
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Angiogenesis inhibiting 5-substituted-1,2,4,-thiadiazolyl derivatives
Patent number
6,833,369
Issue date
Dec 21, 2004
Janssen Pharmaceutica, N.V.
Raymond Antoine Stokbroekx
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Angiogenesis inhibiting thiadiazolyl pyridazine derivatives
Patent number
6,602,873
Issue date
Aug 5, 2003
Janssen Pharamaceutica, N.V.
Raymond Antoine Stokbroekx
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Angiogenesis inhibiting thiadiazolyl pyridazine derivatives
Patent number
6,265,407
Issue date
Jul 24, 2001
Janssen Pharmaceutica N.V.
Raymond Antoine Stokbroekx
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Angiogenesis inhibiting pyridazinamines
Patent number
5,985,878
Issue date
Nov 16, 1999
Janssen Pharmaceuticals, N.V.
Raymond Antoine Stokbroekx
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Urea and thiourea derivatives of azolones
Patent number
5,811,426
Issue date
Sep 22, 1998
Janssen Pharmaceutica, N.V.
Jan Heeres
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Urea and thiourea derivatives of azolones
Patent number
5,639,754
Issue date
Jun 17, 1997
Janssen Pharmaceutica N.V.
Jan Heeres
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic derivatives of azolones
Patent number
5,607,932
Issue date
Mar 4, 1997
Janssen Pharmaceutica N.V.
Jan Heeres
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
MACROCYCLIC QUINAZOLE DERIVATIVES AND THEIR USE AS MTKI
Publication number
20170320894
Publication date
Nov 9, 2017
Janssen Pharmaceutica N.V.
Eddy Jean Edgard FREYNE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINAZOLINE DERIVATIVES
Publication number
20160207938
Publication date
Jul 21, 2016
Janssen Pharmaceutica N.V.
Eddy Jean Edgard FREYNE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MACROCYCLIC QUINAZOLE DERIVATIVES AND THEIR USE AS MTKI
Publication number
20140256714
Publication date
Sep 11, 2014
Janssen Pharmaceutica N.V.
Eddy Jean Edgard FREYNE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDO- AND PYRIMIDOPYRIMIDINE DERIVATIVES AS ANTI-PROFILERATIVE AG...
Publication number
20130231353
Publication date
Sep 5, 2013
Janssen Pharmaceutica N.V.
Eddy Jean Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINAZOLINE DERIVATIVES
Publication number
20130178624
Publication date
Jul 11, 2013
Janssen Pharmaceutica N.V.
Eddy Jean Edgard FREYNE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2,4 (4,6) PYRIMIDINE DERIVATIVES
Publication number
20120065395
Publication date
Mar 15, 2012
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDO-AND PYRIMIDOPYRIMIDINE DERIVATIVES AS ANTI-PROLIFERATIVE AG...
Publication number
20100173913
Publication date
Jul 8, 2010
Janssen Pharmaceutica N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2,4 (4,6) PYRIMIDINE DERIVATIVES
Publication number
20100160310
Publication date
Jun 24, 2010
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MACROCYCLIC QUINAZOLE DERIVATIVES AND THEIR USE AS MTKI
Publication number
20100152174
Publication date
Jun 17, 2010
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Quinazoline derivatives
Publication number
20100105668
Publication date
Apr 29, 2010
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MTKI QUINAZOLINE DERIVATIVES
Publication number
20100029627
Publication date
Feb 4, 2010
Alexandra Papanikos
C08 - ORGANIC MACROMOLECULAR COMPOUNDS THEIR PREPARATION OR CHEMICAL WORKING-...
Information
Patent Application
Triazolopyrimidine Derivatives As Glycogen Synthase Kinase 3 Inhibi...
Publication number
20090036471
Publication date
Feb 5, 2009
Eddy Jean Edgard
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrido-and pyrimidopyrimidine derivatives as anti-profilerative agents
Publication number
20070078132
Publication date
Apr 5, 2007
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Macrocyclic quinazoline derivatives as antiproliferative agents
Publication number
20060247237
Publication date
Nov 2, 2006
Janssen Pharmaceutica N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibi...
Publication number
20060183747
Publication date
Aug 17, 2006
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Aminobenzamide derivatives as glycogen synthase kinase 3 beta inhib...
Publication number
20060063789
Publication date
Mar 23, 2006
Eddy Jean Edgard Freyne
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Amide derivatives as glycogen synthase kinase 3-beta inhibitors
Publication number
20050176713
Publication date
Aug 11, 2005
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Heteroaryl amines as glycogen synthase kinase 3beta inhibitors (gsk...
Publication number
20050004125
Publication date
Jan 6, 2005
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ANGIOGENESIS INHIBITING 5-SUBSTITUTED-1,2,4,-THIADIAZOLYL DERIVATIVES
Publication number
20040009987
Publication date
Jan 15, 2004
Raymond Antoine Stokbroekx
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Angiogenesis inhibiting 5-substituted-1,2,4-thiadiazolyl derivatives
Publication number
20030181460
Publication date
Sep 25, 2003
Raymond Antoine Stokbroekx
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Angiogenesis inhibiting 5-substituted-1,2,4,-thiadiazolyl derivatives
Publication number
20020061890
Publication date
May 23, 2002
Raymond Antoine Stokbroekx
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Angiogenesis inhibiting thiadiazolyl pyridazine derivatives
Publication number
20010046999
Publication date
Nov 29, 2001
Raymond Antoine Stokbroekx
C07 - ORGANIC CHEMISTRY