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Maria G. Brasca
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Milan, IT
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last 30 patents
Information
Patent Grant
Substituted pyrroles active as kinases inhibitors
Patent number
10,479,778
Issue date
Nov 19, 2019
Nerviano Medical Sciences S.r.l.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrroles active as kinases inhibitors
Patent number
10,479,779
Issue date
Nov 19, 2019
Nerviano Medical Sciences S.r.l.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolo-quinazoline derivatives, process for their preparation and...
Patent number
10,280,176
Issue date
May 7, 2019
Nerviano Medical Sciences S.r.l.
Gabriella Traquandi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrroles active as kinases inhibitors
Patent number
10,071,986
Issue date
Sep 11, 2018
Nerviano Medical Sciences S.r.l.
Maria Gabriella Brasca
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrroles active as kinases inhibitors
Patent number
9,688,661
Issue date
Jun 27, 2017
Nerviano Medical Sciences S.r.l.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolo-quinazoline derivatives, process for their preparation and...
Patent number
9,637,497
Issue date
May 2, 2017
Nerviano Medical Sciences, S.R.L.
Gabriella Traquandi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolo-quinazoline derivatives, process for their preparation and...
Patent number
9,464,090
Issue date
Oct 11, 2016
Nerviano Medical Sciences S.R.L.
Gabriella Traquandi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Tricyclic pyrrolo derivatives, process for their preparation and th...
Patent number
9,309,253
Issue date
Apr 12, 2016
Nerviano Medical Sciences S.r.l.
Marina Caldarelli
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolyl-pyrimidine derivatives as kinase inhibitors
Patent number
9,284,298
Issue date
Mar 15, 2016
Nerviano Medical Sciences S.r.l.
Francesco Casuscelli
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrimidinyl-pyrroles active as kinase inhibitors
Patent number
9,283,224
Issue date
Mar 15, 2016
Nerviano Medical Sciences S.r.l.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Resorcinol derivatives as HSP90 inhibitors
Patent number
8,993,556
Issue date
Mar 31, 2015
Nerviano Medical Sciences S.r.l.
Maria Gabriella Brasca
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolo-quinazoline derivatives, process for their preparation and...
Patent number
8,981,089
Issue date
Mar 17, 2015
Nerviano Medical Sciences S.R.L.
Gabriella Traquandi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tricyclic pyrrolo derivatives, process for their preparation and th...
Patent number
8,975,267
Issue date
Mar 10, 2015
Nerviano Medical Sciences S.r.l.
Marina Caldarelli
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Alkynyl substituted pyrimidinyl-pyrroles active as kinases inhibitors
Patent number
8,912,200
Issue date
Dec 16, 2014
Nerviano Medical Sciences S.r.l.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrrolo-pyrazole derivatives as kinase inhibitors
Patent number
8,785,448
Issue date
Jul 22, 2014
Nerviano Medical Sciences S.r.l.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrrolo-pyrazole derivatives as kinase inhibitors
Patent number
8,623,876
Issue date
Jan 7, 2014
Nerviano Medical Sciences S.r.l.
Michele Caruso
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrazolo-quinazoline derivatives, process for their pre...
Patent number
8,614,220
Issue date
Dec 24, 2013
Nerviano Medical Sciences S.r.l.
Michele Caruso
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted dihydropteridin-6-one derivatives, process for their pr...
Patent number
8,598,172
Issue date
Dec 3, 2013
Nerviano Medical Sciences S.r.l.
Michele Caruso
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
CDK inhibitor salts
Patent number
8,586,598
Issue date
Nov 19, 2013
Nerviano Medical Sciences S.r.l.
Massimo Zampieri
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrrolo-pyrazole derivatives as kinase inhibitors
Patent number
8,557,857
Issue date
Oct 15, 2013
Nerviano Medical Sciences S.r.l.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrrolo-pyrazole derivatives as kinase inhibitors
Patent number
8,557,845
Issue date
Oct 15, 2013
Nerviano Medical Sciences S.r.l.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolo quinazoline derivatives, process for their preparation and...
Patent number
8,541,429
Issue date
Sep 24, 2013
Nerviano Medical Sciences S.r.l.
Gabriella Traquandi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrrolo-pyrazole derivatives as kinase inhibitors
Patent number
8,481,585
Issue date
Jul 9, 2013
Nerviano Medical Sciences S.r.l.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrrolo-pyrimidine derivatives, process for their prepa...
Patent number
8,426,417
Issue date
Apr 23, 2013
Nerviano Medical Sciences S.r.l.
Michele Caruso
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic pyrazole and isoxazole derivatives as antitumor and antine...
Patent number
8,309,578
Issue date
Nov 13, 2012
Nerviano Medical Sciences S.r.l.
Sergio Mantegani
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrrolo-pyrazole derivatives as kinase inhibitors
Patent number
8,227,472
Issue date
Jul 24, 2012
Nerviano Medical Sciences S.r.l.
Michele Caruso
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolo[2,3-b]pyridine derivatives active as kinase inhibitors
Patent number
8,198,298
Issue date
Jun 12, 2012
Pfizer Italia S.R.L.
Barbara Salom
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolo[2,3-b]pyridine derivatives active as kinase inhibitors and...
Patent number
8,106,069
Issue date
Jan 31, 2012
Pfizer Italia S.R.L.
Barbara Salom
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolo[2,3-B]pyridine derivatives active as kinase inhibitors
Patent number
7,888,508
Issue date
Feb 15, 2011
Pfizer Italia S.R.L.
Barbara Salom
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolo[2,3-b]pyridine derivatives active as kinase inhibitors and...
Patent number
7,728,140
Issue date
Jun 1, 2010
Pfizer Italia S.R.L.
Barbara Salom
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
PYRAZOLO-QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND...
Publication number
20210300935
Publication date
Sep 30, 2021
Nerviano Medical Sciences S.R.L.
Gabriella Traquandi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLO-QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND...
Publication number
20190194214
Publication date
Jun 27, 2019
Nerviano Medical Sciences S.R.L.
Gabriella Traquandi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PYRROLES ACTIVE AS KINASES INHIBITORS
Publication number
20180339978
Publication date
Nov 29, 2018
NERVIANO MEDICAL SCIENCES S.R.L.
Maria Gabriella Brasca
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PYRROLES ACTIVE AS KINASES INHIBITORS
Publication number
20170253578
Publication date
Sep 7, 2017
NERVIANO MEDICAL SCIENCES S.R.L.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRROLES ACTIVE AS KINASES INHIBITORS
Publication number
20170253579
Publication date
Sep 7, 2017
NERVIANO MEDICAL SCIENCES S.R.L.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLO-QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND...
Publication number
20170190714
Publication date
Jul 6, 2017
Nerviano Medical Sciences S.R.L.
Gabriella Traquandi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLO-QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND...
Publication number
20170050972
Publication date
Feb 23, 2017
Nerviano Medical Sciences, S.R.L.
Gabriella Traquandi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PYRROLES ACTIVE AS KINASES INHIBITORS
Publication number
20150166512
Publication date
Jun 18, 2015
NERVIANO MEDICAL SCIENCES S.R.L.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLO-QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND...
Publication number
20150158876
Publication date
Jun 11, 2015
NERVIANO MEDICAL SCIENCES S.R.L.
Gabriella Traquandi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TRICYCLIC PYRROLO DERIVATIVES, PROCESS FOR THEIR PREPARATION AND TH...
Publication number
20150141408
Publication date
May 21, 2015
NERVIANO MEDICAL SCIENCES S.R.L.
Marina Caldarelli
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Application
ALKYNYL SUBSTITUTED PYRIMIDINYL-PYRROLES ACTIVE AS KINASES INHIBITORS
Publication number
20140194406
Publication date
Jul 10, 2014
NERVIANO MEDICAL SCIENCES S.R.L.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRIMIDINYL-PYRROLES ACTIVE AS KINASE INHIBITORS
Publication number
20140155421
Publication date
Jun 5, 2014
NERVIANO MEDICAL SCIENCES S.R.L.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLYL-PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS
Publication number
20140051708
Publication date
Feb 20, 2014
NERVIANO MEDICAL SCIENCES S.R.L.
Francesco Casuscelli
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRROLO-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS
Publication number
20130344031
Publication date
Dec 26, 2013
NERVIANO MEDICAL SCIENCES S.R.L.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLO-QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND...
Publication number
20130338148
Publication date
Dec 19, 2013
Nerviano Medical Sciences S.r.l.
Gabriella Traquandi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TRICYCLIC PYRROLO DERIVATIVES, PROCESS FOR THEIR PREPARATION AND TH...
Publication number
20130296305
Publication date
Nov 7, 2013
NERVIANO MEDICAL SCIENCES S.R.L.
Marina Caldarelli
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Application
SUBSTITUTED PYRROLO-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS
Publication number
20130017170
Publication date
Jan 17, 2013
NERVIANO MEDICAL SCIENCES S.R.L.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRROLO-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS
Publication number
20130012507
Publication date
Jan 10, 2013
NERVIANO MEDICAL SCIENCES S.R.L.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRROLO-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS
Publication number
20120277248
Publication date
Nov 1, 2012
NERVIANO MEDICAL SCIENCES S.R.L.
Michele Caruso
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Substituted Pyrrolo-Pyrimidine Derivatives, Process for Their Prepa...
Publication number
20120122882
Publication date
May 17, 2012
NERVIANO MEDICAL SCIENCES S.R.L.
Michele Caruso
C07 - ORGANIC CHEMISTRY
Information
Patent Application
RESORCINOL DERIVATIVES AS HSP90 INHIBITORS
Publication number
20120046266
Publication date
Feb 23, 2012
NERVIANO MEDICAL SCIENCES S.R.L.
Maria Gabriella Brasca
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CDK INHIBITOR SALTS
Publication number
20120041007
Publication date
Feb 16, 2012
NERVIANO MEDICAL SCIENCES S.R.L.
Massimo Zampieri
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC PYRAZOLE AND ISOXAZOLE DERIVATIVES AS ANTITUMOR AND ANTINE...
Publication number
20110294790
Publication date
Dec 1, 2011
NERVIANO MEDICAL SCIENCES S.R.L.
Sergio Mantegani
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLE[2,3-B]PYRIDINE DERIVATIVES ACTIVE AS KINASE INHIBITORS
Publication number
20110136857
Publication date
Jun 9, 2011
Pfizer Italia S.r.l.
Barbara Salom
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED DIHYDROPTERIDIN-6-ONE DERIVATIVES, PROCESS FOR THEIR PR...
Publication number
20110053944
Publication date
Mar 3, 2011
NERVIANO MEDICAL SCIENCES S.R.L.
Michele Caruso
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PYRAZOLO-QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PRE...
Publication number
20100216808
Publication date
Aug 26, 2010
NERVIANO MEDICAL SCIENCES S.R.L.
Michele Caruso
C40 - COMBINATORIAL CHEMISTRY
Information
Patent Application
Pyrrolo[2,3-b]Pyridine Derivatives Active as Kinase Inhibitors and...
Publication number
20100210476
Publication date
Aug 19, 2010
Pfizer Italia S.r.l.
Barbara Salom
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PYRROLO-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS
Publication number
20100010008
Publication date
Jan 14, 2010
NERVIANO MEDICAL SCIENCES S.R.L.
Michele Caruso
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrazolo-Quinazoline Derivatives, Process for Their Preparation and...
Publication number
20090124605
Publication date
May 14, 2009
Nerviano Medical Sciences S.r.l.
Gabriella Traquandi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Substituted Pyrrolo-Pyrazole Derivatives as Kinase Inhibitors
Publication number
20090082346
Publication date
Mar 26, 2009
Pfizer Italia S.r.l.
Maria Gabriella Brasca
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE