Membership
Tour
Register
Log in
Mark Edward Zak
Follow
Person
San Mateo, CA, US
People
Overview
Industries
Organizations
People
Information
Impact
Patents Grants
last 30 patents
Information
Patent Grant
Therapeutic compounds, compositions and methods of use thereof
Patent number
11,795,170
Issue date
Oct 24, 2023
Genentech, Inc.
Mark Zak
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Therapeutic compounds, compositions and methods of use thereof
Patent number
11,731,943
Issue date
Aug 22, 2023
Genentech, Inc.
James John Crawford
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolochlorophenyl compounds, compositions and methods of use the...
Patent number
11,649,241
Issue date
May 16, 2023
Genentech, Inc.
Mark Zak
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Amido spirocyclic amide and sulfonamide derivatives
Patent number
11,485,745
Issue date
Nov 1, 2022
Valo Health, Inc.
Kenneth W. Bair
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolopyrimidine inhibitors of JAK kinases and uses thereof
Patent number
11,453,671
Issue date
Sep 27, 2022
Genentech, Inc.
Mark Edward Zak
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolopyrimidine compounds and methods of use thereof
Patent number
11,155,557
Issue date
Oct 26, 2021
Genentech, Inc.
F. Anthony Romero
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Amido spirocyclic amide and sulfonamide derivatives
Patent number
10,730,889
Issue date
Aug 4, 2020
Forma TM, LLC
Kenneth W. Bair
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Amido-benzyl sulfone and sulfoxide derivates
Patent number
10,696,692
Issue date
Jun 30, 2020
Kenneth W Bair
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Therapeutic compounds and compositions, and methods of use thereof
Patent number
10,307,426
Issue date
Jun 4, 2019
Genentech, Inc.
Mark Zak
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Therapeutic compounds, compositions and methods of use thereof
Patent number
10,189,836
Issue date
Jan 29, 2019
Genentech, Inc.
Yun-Xing Cheng
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Triazolopyridine compounds, compositions and methods of use thereof
Patent number
9,873,709
Issue date
Jan 23, 2018
Genentech, Inc.
Nicholas C. Ray
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Amido spirocyclic amide and sulfonamide derivatives
Patent number
9,822,129
Issue date
Nov 21, 2017
Genentech, Inc.
Kenneth W Bair
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
5-chloro-2-difluoromethoxyphenyl pyrazolopyrimidine compounds, comp...
Patent number
9,604,984
Issue date
Mar 28, 2017
Genentech, Inc.
Mark Edward Zak
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyridinyl and pyrimidinyl sulfoxide and sulfone derivatives
Patent number
9,458,172
Issue date
Oct 4, 2016
Kenneth W Bair
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
5-chloro-2-difluoromethoxyphenyl pyrazolopyrimidine compounds, comp...
Patent number
9,346,815
Issue date
May 24, 2016
Genentech, Inc.
Mark Edward Zak
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolopyrimidine JAK inhibitor compounds and methods
Patent number
8,999,998
Issue date
Apr 7, 2015
Genentech, Inc.
Paul Gibbons
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolopyrimidone and pyrrolopyridone inhibitors of tankyrase
Patent number
8,722,661
Issue date
May 13, 2014
Hoffmann-La Roche Inc.
Nancy-Ellen Haynes
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tricyclic heterocyclic compounds, compositions and methods of use t...
Patent number
8,461,328
Issue date
Jun 11, 2013
Genentech, Inc.
Srinivasan Babu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
5-anilinoimidazopyridines and methods of use
Patent number
8,288,408
Issue date
Oct 16, 2012
Genentech, Inc.
Stephen Price
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
5-anilinoimidazo[1,5-a]-pyridines inhibitors of MEK kinase
Patent number
7,923,456
Issue date
Apr 12, 2011
Genentech, Inc.
Stephen Price
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
PYRAZOLOPYRIMIDINE JAK INHIBITOR COMPOUNDS AND METHODS
Publication number
20240150364
Publication date
May 9, 2024
Genentech, Inc.
Paul Gibbons
C07 - ORGANIC CHEMISTRY
Information
Patent Application
8-(AZETIDIN-1-YL)-[1,2,4]TRIAZOLO[1,5-A]PYRIDINYL COMPOUNDS, COMPOS...
Publication number
20230242530
Publication date
Aug 3, 2023
Genentech, Inc.
Simon Charles GOODACRE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLOPYRIMIDINE COMPOUNDS AS JAK INHIBITORS
Publication number
20230206644
Publication date
Jun 29, 2023
Genentech, Inc.
Mark ZAK
G06 - COMPUTING CALCULATING COUNTING
Information
Patent Application
TETRAZOLE-SUBSTITUTED PYRAZOLOPYRIMIDINE INHIBITORS OF JAK KINASES...
Publication number
20230167123
Publication date
Jun 1, 2023
Genentech, Inc.
Mark Edward Zak
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INHALABLE DRY POWDER AND AEROSOL FORMULATIONS OF JAK INHIBITORS
Publication number
20230016791
Publication date
Jan 19, 2023
Genentech, Inc.
Mark Edward Zak
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLOPYRIMIDINE JAK INHIBITOR COMPOUNDS AND METHODS
Publication number
20220389020
Publication date
Dec 8, 2022
Genentech, Inc.
Paul Gibbons
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INHALED POWDER FORMULATIONS
Publication number
20220204517
Publication date
Jun 30, 2022
Genentech, Inc.
Yun-Xing Cheng
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLOPYRIMIDINE ARYL ETHER INHIBITORS OF JAK KINASES AND USES TH...
Publication number
20220106322
Publication date
Apr 7, 2022
Genentech, Inc.
Mark Edward Zak
C07 - ORGANIC CHEMISTRY
Information
Patent Application
THERAPEUTIC COMPOUNDS AND COMPOSITIONS, AND METHODS OF USE THEREOF
Publication number
20220024945
Publication date
Jan 27, 2022
Genentech, Inc.
Mark ZAK
C07 - ORGANIC CHEMISTRY
Information
Patent Application
THERAPEUTIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF
Publication number
20210179564
Publication date
Jun 17, 2021
Genentech, Inc.
James John Crawford
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLOCHLOROPHENYL COMPOUNDS, COMPOSITIONS AND METHODS OF USE THE...
Publication number
20210179626
Publication date
Jun 17, 2021
Genentech, Inc.
Mark ZAK
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMIDO SPIROCYCLIC AMIDE AND SULFONAMIDE DERIVATIVES
Publication number
20210171545
Publication date
Jun 10, 2021
Integral Early Discovery, Inc.
Kenneth W. Bair
C07 - ORGANIC CHEMISTRY
Information
Patent Application
THERAPEUTIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF
Publication number
20210009599
Publication date
Jan 14, 2021
Genentech, Inc.
Mark Zak
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLOPYRIMIDINE SULFONE INHIBITORS OF JAK KINASES AND USES THEREOF
Publication number
20200399275
Publication date
Dec 24, 2020
Genentech, Inc.
Mark Edward Zak
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TETRAZOLE-SUBSTITUTED PYRAZOLOPYRIMIDINE INHIBITORS OF JAK KINASES...
Publication number
20200399274
Publication date
Dec 24, 2020
Genentech, Inc.
Mark Edward Zak
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
THERAPEUTIC COMPOUNDS AND COMPOSITIONS, AND METHODS OF USE THEREOF
Publication number
20200352951
Publication date
Nov 12, 2020
Genentech, Inc.
Mark ZAK
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLOPYRIMIDINE COMPOUNDS AS JAK INHIBITORS
Publication number
20200339604
Publication date
Oct 29, 2020
Genentech, Inc.
Mark ZAK
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
8-(AZETIDIN-1-YL)-[1,2,4]TRIAZOLO[1,5-A]PYRIDINYL COMPOUNDS, COMPOS...
Publication number
20200270248
Publication date
Aug 27, 2020
Genentech, Inc.
Simon Charles GOODACRE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INHALED POWDER FORMULATIONS
Publication number
20200165260
Publication date
May 28, 2020
Genentech, Inc.
Yun-Xing Cheng
C07 - ORGANIC CHEMISTRY
Information
Patent Application
THERAPEUTIC COMPOUNDS AND COMPOSITIONS, AND METHODS OF USE THEREOF
Publication number
20200062779
Publication date
Feb 27, 2020
Genentech, Inc.
Mark ZAK
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLOPYRIMIDINE JAK INHIBITOR COMPOUNDS AND METHODS
Publication number
20200002345
Publication date
Jan 2, 2020
Genentech, Inc.
Paul Gibbons
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLOCHLOROPHENYL COMPOUNDS, COMPOSITIONS AND METHODS OF USE THE...
Publication number
20200002346
Publication date
Jan 2, 2020
Genentech, Inc.
Mark ZAK
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLOPYRIMIDINE COMPOUNDS AND METHODS OF USE THEREOF
Publication number
20190345165
Publication date
Nov 14, 2019
Genentech, Inc.
F. Anthony ROMERO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TRIAZOLOPYRIDINE COMPOUNDS AND METHODS OF USE THEREOF
Publication number
20190337946
Publication date
Nov 7, 2019
Genentech, Inc.
Simon Charles Goodacre
C07 - ORGANIC CHEMISTRY
Information
Patent Application
5-CHLORO-2-DIFLUOROMETHOXYPHENYL PYRAZOLOPYRIMIDINE COMPOUNDS,COMPO...
Publication number
20190322661
Publication date
Oct 24, 2019
Genentech, Inc.
Mark Edward Zak
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
THERAPEUTIC COMPOUNDS AND COMPOSITIONS, AND METHODS OF USE THEREOF
Publication number
20190240227
Publication date
Aug 8, 2019
Genentech, Inc.
Mark ZAK
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF
Publication number
20190233441
Publication date
Aug 1, 2019
Genentech, Inc.
Nicholas C. RAY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
8-(AZETIDIN-1-YL)-[1,2,4]TRIAZOLO[1,5-A]PYRIDINYL COMPOUNDS, COMPOS...
Publication number
20190202822
Publication date
Jul 4, 2019
Genentech, Inc.
Simon Charles GOODACRE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
THERAPEUTIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF
Publication number
20190071404
Publication date
Mar 7, 2019
Genentech, Inc.
James John Crawford
C07 - ORGANIC CHEMISTRY
Information
Patent Application
THERAPEUTIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF
Publication number
20180354959
Publication date
Dec 13, 2018
Genentech, Inc.
Mark Zak
C07 - ORGANIC CHEMISTRY