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Mark J. Macielag
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Gwynedd Valley, PA, US
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Patents Grants
last 30 patents
Information
Patent Grant
Immunoglobulins and uses thereof
Patent number
12,134,636
Issue date
Nov 5, 2024
JANSSEN PHARMACEUTICA NV
Mark Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyridine N-oxide derivatives useful as factor XIa inhibitors
Patent number
11,814,364
Issue date
Nov 14, 2023
JANSSEN PHARMACEUTICA NV
Guozhang Xu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modu...
Patent number
11,767,354
Issue date
Sep 26, 2023
JANSSEN PHARMACEUTICA NV
Mark Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cyclic peptide tyrosine tyrosine compounds as modulators of neurope...
Patent number
11,732,019
Issue date
Aug 22, 2023
JANSSEN PHARMACEUTICA NV
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modu...
Patent number
11,591,379
Issue date
Feb 28, 2023
JANSSEN PHARMACEUTICA NV
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Immunoglobulins and uses thereof
Patent number
11,401,315
Issue date
Aug 2, 2022
JANSSEN PHARMACEUTICA NV
Mark Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cylcoalkenyl derivatives useful as agonists of the GPR120 and/or GP...
Patent number
11,230,526
Issue date
Jan 25, 2022
JANSSEN PHARMACEUTICA NV
James C. Lanter
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modu...
Patent number
10,968,265
Issue date
Apr 6, 2021
JANSSEN PHARMACEUTICA NV
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Cyclic peptide tyrosine tyrosine compounds as modulators of neurope...
Patent number
10,968,264
Issue date
Apr 6, 2021
JANSSEN PHARMACEUTICA NV
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Cyclic peptide tyrosine tyrosine compounds as modulators of neurope...
Patent number
10,961,293
Issue date
Mar 30, 2021
Janssen Pharmaceutics N.V.
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Immunoglobulins and uses thereof
Patent number
10,858,413
Issue date
Dec 8, 2020
JANSSEN PHARMACEUTICA NV
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Immunoglobulins and uses thereof
Patent number
10,787,495
Issue date
Sep 29, 2020
JANSSEN PHARMACEUTICA NV
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modu...
Patent number
10,640,544
Issue date
May 5, 2020
JANSSEN PHARMACEUTICA NV
Mark Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyridin-2-one derivatives of formula (I) useful as EP3 receptor ant...
Patent number
10,590,083
Issue date
Mar 17, 2020
JANSSEN PHARMACEUTICA NV
Xuqing Zhang
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Immunoglobulins and uses thereof
Patent number
10,428,134
Issue date
Oct 1, 2019
JANSSEN PHARMACEUTICA NV
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyridin-2-one derivatives of formula (III) useful as EP3 receptor a...
Patent number
10,399,944
Issue date
Sep 3, 2019
JANSSEN PHARMACEUTICA NV
Xuqing Zhang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyridin-2-one derivatives of formula (II) useful as EP3 receptor an...
Patent number
10,336,701
Issue date
Jul 2, 2019
JANSSEN PHARMACEUTICA NV
Xuqing Zhang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzimidazole derivatives useful as CB-1 inverse agonists
Patent number
10,118,900
Issue date
Nov 6, 2018
JANSSEN PHARMACEUTICA NV
Mark J. Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Chemically modified quinoline and quinolone derivatives useful as C...
Patent number
9,815,790
Issue date
Nov 14, 2017
JANSSEN PHARMACEUTICA NV
Mark J. Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cinnoline derivatives useful as CB-1 receptor inverse agonists
Patent number
9,732,061
Issue date
Aug 15, 2017
JANSSEN PHARMACEUTICA NV
Mark Joseph Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Quinazoline derivatives useful as CB-1 inverse agonists
Patent number
9,682,955
Issue date
Jun 20, 2017
JANSSEN PHARMACEUTICA NV
Mark Joseph Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Indazole derivatives useful as CB-1 inverse agonists
Patent number
9,682,940
Issue date
Jun 20, 2017
JANSSEN PHARMACEUTICA NV
Mark J. Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzimidazole derivatives useful TRPM8 channel modulators
Patent number
9,636,345
Issue date
May 2, 2017
JANSSEN PHARMACEUTICA NV
Mark J. Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Quinoline derivatives useful as CB-1 inverse agonists
Patent number
9,464,055
Issue date
Oct 11, 2016
JANSSEN PHARMACEUTICA NV
Bart DeCorte
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Sulfonamides as TRPM8 modulators
Patent number
9,434,711
Issue date
Sep 6, 2016
Janssen Pharmaceutica, N.V.
Shawn T Branum
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Monoacylglycerol lipase inhibitors for the treatment of metabolic d...
Patent number
9,375,430
Issue date
Jun 28, 2016
JANSSEN PHARMACEUTICA NV
Margery Connelly
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Quinoline derivatives useful as CB-1 inverse agonists
Patent number
9,266,835
Issue date
Feb 23, 2016
JANSSEN PHARMACEUTICA NV
Bart DeCorte
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazo[1,2-α]pyridine sulfonamides as TRPM8 modulators
Patent number
9,067,935
Issue date
Jun 30, 2015
Janssen Pharmaceutica, N.V.
Mark J Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Monoacylglycerol lipase inhibitors for the treatment of metabolic d...
Patent number
8,987,247
Issue date
Mar 24, 2015
JANSSEN PHARMACEUTICA NV
Margery Connelly
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzimidazole derivatives useful as TRPM8 channel modulators
Patent number
8,981,113
Issue date
Mar 17, 2015
JANSSEN PHARMACEUTICA NV
Mark J Macielag
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
IMMUNOGLOBULINS AND USES THEREOF
Publication number
20250026803
Publication date
Jan 23, 2025
Janssen Pharmaceutica N.V.
Mark MACIELAG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODULATORS OF NEUROPE...
Publication number
20240018208
Publication date
Jan 18, 2024
Janssen Pharmaceutica N.V.
Mark MACIELAG
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ANTIBODY-COUPLED CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODU...
Publication number
20230365644
Publication date
Nov 16, 2023
Janssen Pharmaceutica N.V.
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS USEFUL AS FACTOR XIA INHIBITORS
Publication number
20230312560
Publication date
Oct 5, 2023
Janssen Pharmaceutica N.V.
Guozhang XU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
3-(1H-IMIDAZOL-2-YL)-2,3,8,8A-TETRAHYDROINDOLIZIN-5(1H)-ONE DERIVAT...
Publication number
20230295157
Publication date
Sep 21, 2023
Janssen Pharmaceutica N.V.
Guozhang XU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic Pyridin-2-one and pyrimidin-4-one Derivatives Useful As a...
Publication number
20230183233
Publication date
Jun 15, 2023
Janssen Pharmaceutica N.V.
Guozhang Xu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic Pyridin-2-one and pyrimidin-4-one Derivatives Useful As a...
Publication number
20230097157
Publication date
Mar 30, 2023
Janssen Pharmaceutica N.V.
Guozhang Xu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDINE N-OXIDE DERIVATIVES USEFUL AS FACTOR XIA INHIBITORS
Publication number
20230091768
Publication date
Mar 23, 2023
Janssen Pharmaceutica N.V.
Guozhang Xu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
5-oxo-1,2,3,5,8,8a-hexahydroindolizine-3-carboxamide Derivatives Us...
Publication number
20230064443
Publication date
Mar 2, 2023
Janssen Pharmaceutica N.V.
Guozhang Xu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ACYLSUFONAMIDE COMPOUNDS USEFUL AS EP3 RECEPTOR ANTAGONISTS
Publication number
20210253562
Publication date
Aug 19, 2021
Janssen Pharmaceutica N.V.
Bin Zhu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Cyclic Peptide Tyrosine Tyrosine Compounds as Modulators of Neurope...
Publication number
20210206822
Publication date
Jul 8, 2021
Janssen Pharmaceutica N.V.
Mark MACIELAG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Antibody-Coupled Cyclic Peptide Tyrosine Tyrosine Compounds as Modu...
Publication number
20210163566
Publication date
Jun 3, 2021
Janssen Pharmaceutica N.V.
Mark MACIELAG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMMUNOGLOBULINS AND USES THEREOF
Publication number
20210094998
Publication date
Apr 1, 2021
Janssen Pharmaceutica N.V.
Mark MACIELAG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMMUNOGLOBULINS AND USES THEREOF
Publication number
20200385439
Publication date
Dec 10, 2020
Janssen Pharmaceutica N.V.
Mark MACIELAG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ANTIBODY-COUPLED CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODU...
Publication number
20200283491
Publication date
Sep 10, 2020
Janssen Pharmaceutica N.V.
Mark MACIELAG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMMUNOGLOBULINS AND USES THEREOF
Publication number
20190367577
Publication date
Dec 5, 2019
Janssen Pharmaceutica N.V.
Mark MACIELAG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODULATORS OF NEUROPE...
Publication number
20190345214
Publication date
Nov 14, 2019
Janssen Pharmaceutica N.V.
Mark MACIELAG
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ANTIBODY-COUPLED CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODU...
Publication number
20190298849
Publication date
Oct 3, 2019
Janssen Pharmaceutica N.V.
Mark MACIELAG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMMUNOGLOBULINS AND USES THEREOF
Publication number
20190263879
Publication date
Aug 29, 2019
Janssen Pharmaceutica N.V.
Mark MACIELAG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRIDIN-2-ONE DERIVATIVES OF FORMULA (II) USEFUL AS EP3 RECEPTOR AN...
Publication number
20190047960
Publication date
Feb 14, 2019
Janssen Pharmaceutica N.V.
Xuqing Zhang
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRIDIN-2-ONE DERIVATIVES OF FORMULA (I) USEFUL AS EP3 RECEPTOR ANT...
Publication number
20190047959
Publication date
Feb 14, 2019
Janssen Pharmaceutica N.V.
Xuqing Zhang
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRIDIN-2-ONE DERIVATIVES OF FORMULA (III) USEFUL AS EP3 RECEPTOR A...
Publication number
20190047961
Publication date
Feb 14, 2019
Janssen Pharmaceutica N.V.
Xuqing Zhang
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZIMIDAZOLE DERIVATIVES USEFUL AS CB-1 INVERSE AGONISTS
Publication number
20190031618
Publication date
Jan 31, 2019
Janssen Pharmaceutica N.V.
Mark J. Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMMUNOGLOBULINS AND USES THEREOF
Publication number
20180125998
Publication date
May 10, 2018
Janssen Pharmaceutica N.V.
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODULATORS OF NEUROPE...
Publication number
20180127476
Publication date
May 10, 2018
Janssen Pharmaceutica N.V.
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ANTIBODY-COUPLED CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODU...
Publication number
20180117170
Publication date
May 3, 2018
Janssen Pharmaceutica N.V.
Mark Macielag
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZIMIDAZOLE DERIVATIVES USEFUL AS CB-1 INVERSE AGONISTS
Publication number
20170057929
Publication date
Mar 2, 2017
Janssen Pharmaceutica N.V.
Mark J. Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CHEMICALLY MODIFIED QUINOLINE AND QUINOLONE DERIVATIVES USEFUL AS C...
Publication number
20170057922
Publication date
Mar 2, 2017
Janssen Pharmaceutica N.V.
Mark J. Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INDAZOLE DERIVATIVES USEFUL AS CB-1 INVERSE AGONISTS
Publication number
20170057925
Publication date
Mar 2, 2017
Janssen Pharmaceutica N.V.
Mark J. Macielag
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CINNOLINE DERIVATIVES USEFUL AS CB-1 RECEPTOR INVERSE AGONISTS
Publication number
20160200719
Publication date
Jul 14, 2016
Janssen Pharmaceutica N.V.
Mark Joseph Macielag
C07 - ORGANIC CHEMISTRY