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Matthew J. LaMarche
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Philadelphia, PA, US
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Patents Grants
last 30 patents
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Patent Grant
N-azaspirocycloalkane substituted N-heteroaryl compounds and compos...
Patent number
12,209,098
Issue date
Jan 28, 2025
Novartis AG
Christine Hiu-Tung Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pharmaceutical combination comprising an ALK inhibitor and a SHP2 i...
Patent number
12,053,470
Issue date
Aug 6, 2024
Novartis AG
Leila Dardaei Alghalandis
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
N-azaspirocycloalkane substituted N-heteroaryl compounds and compos...
Patent number
11,952,386
Issue date
Apr 9, 2024
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds and compositions for inhibiting the activity of SHP2
Patent number
11,905,283
Issue date
Feb 20, 2024
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1-Pyridazin-/triazin-3-yl-piper(-azine)/idine/pyrolidine derivative...
Patent number
11,401,259
Issue date
Aug 2, 2022
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds and compositions for inhibiting the activity of SHP2
Patent number
10,975,080
Issue date
Apr 13, 2021
Novartis AG
Jeffrey T. Bagdanoff
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
N-azaspirocycloalkane substituted N-heteroaryl compounds and compos...
Patent number
10,968,235
Issue date
Apr 6, 2021
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds and compositions for inhibiting the activity of SHP2
Patent number
10,934,285
Issue date
Mar 2, 2021
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1-pyridazin-/triazin-3-yl-piper(-azine)/idine/pyrolidine derivative...
Patent number
10,774,065
Issue date
Sep 15, 2020
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-azaspirocycloalkane substituted N-heteroaryl compounds and compos...
Patent number
10,336,774
Issue date
Jul 2, 2019
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds and compositions for inhibiting the activity of SHP2
Patent number
10,308,660
Issue date
Jun 4, 2019
Novartis AG
Zhuoliang Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1-(triazin-3-yl/pyridazin-3-yl)-piper(-azine)idine derivatives and...
Patent number
10,301,278
Issue date
May 28, 2019
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds and compositions for inhibiting the activity of SHP2
Patent number
10,287,266
Issue date
May 14, 2019
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pharmaceutical combinations
Patent number
10,130,629
Issue date
Nov 20, 2018
Novartis AG
Nicole Buschmann
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1-pyridazin-/triazin-3-yl-piper(-azine)/idine/pyrolidine derivative...
Patent number
10,093,646
Issue date
Oct 9, 2018
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-azaspirocycloalkane substituted N-heteroaryl compounds and compos...
Patent number
10,077,276
Issue date
Sep 18, 2018
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-azaspirocycloalkane substituted N-heteroaryl compounds and compos...
Patent number
9,938,295
Issue date
Apr 10, 2018
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1-(triazin-3-yl/pyridazin-3-yl)-piper(-azine)idine derivatives and...
Patent number
9,815,813
Issue date
Nov 14, 2017
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aminothiazoles and their uses
Patent number
9,492,496
Issue date
Nov 15, 2016
Novartis AG
Simon Bushell
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocycles and their uses
Patent number
8,691,756
Issue date
Apr 8, 2014
Novartis AG
Roger Aki Fujimoto
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocycles and their uses
Patent number
8,476,224
Issue date
Jul 2, 2013
Novartis AG
Roger Aki Fujimoto
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Aminothiazoles and their uses
Patent number
8,426,356
Issue date
Apr 23, 2013
Novartis AG
Simon Bushell
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Antibacterial compounds and processes for its production
Patent number
8,183,341
Issue date
May 22, 2012
Novartis AG
Matthew J. Lamarche
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic compounds with kinase inhibitory activity
Patent number
8,110,687
Issue date
Feb 7, 2012
Millennium Pharmaceuticals, Inc.
Emily F. Calderwood
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
EFTU inhibitors or aminothiazoles and their uses
Patent number
7,851,439
Issue date
Dec 14, 2010
Novartis AG
Simon Bushell
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Synthetic techniques and intermediates for polyhydroxy dienyl lacto...
Patent number
7,723,536
Issue date
May 25, 2010
The Trustees of the University of Pennsylvania
Amos B. Smith, III
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cinnamide and hydrocinnamide derivatives with kinase inhibitory act...
Patent number
7,652,041
Issue date
Jan 26, 2010
Millennium Pharmaceuticals, Inc.
Ruth S. Adams
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds which mimic the chemical and biological properties of dis...
Patent number
7,652,031
Issue date
Jan 26, 2010
The Trustees of the University of Pennsylvania
Amos B Smith, III
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Synthetic techniques and intermediates for polyhydroxy dienyl lacto...
Patent number
7,368,585
Issue date
May 6, 2008
The Trustees of the University of Pennsylvania
Amos B. Smith, III
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Antagonists of melanin concentrating hormone receptor
Patent number
6,921,821
Issue date
Jul 26, 2005
Abbott Laboratories
Christopher Blackburn
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF SHP2
Publication number
20240199609
Publication date
Jun 20, 2024
Novartis AG
Zhuoliang CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20220396585
Publication date
Dec 15, 2022
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1-PYRIDAZIN-/TRIAZIN-3-YL-PIPER(-AZINE)/IDINE/PYROLIDINE DERIVATIVE...
Publication number
20220348553
Publication date
Nov 3, 2022
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHARMACEUTICAL COMBINATION COMPRISING AN ALK INHIBITOR AND A SHP2 I...
Publication number
20220241277
Publication date
Aug 4, 2022
Novartis AG
Leila DARDAEI ALGHALANDIS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS AND COMPOSITIONS FOR INHBITING THE ACTIVITY OF SHP2
Publication number
20220089597
Publication date
Mar 24, 2022
Novartis AG
Jeffrey T. Bagdanoff
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20220073537
Publication date
Mar 10, 2022
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20210371429
Publication date
Dec 2, 2021
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS AND COMPOSITIONS FOR INHBITING THE ACTIVITY OF SHP2
Publication number
20210309663
Publication date
Oct 7, 2021
Novartis AG
Jeffrey T. Bagdanoff
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF SHP2
Publication number
20210300919
Publication date
Sep 30, 2021
Novartis AG
Zhuoliang CHEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
1-PYRIDAZIN-/TRIAZIN-3-YL-PIPER(-AZINE)/IDINE/PYROLIDINE DERIVATIVE...
Publication number
20200369643
Publication date
Nov 26, 2020
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20200181168
Publication date
Jun 11, 2020
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF SHP2
Publication number
20200002330
Publication date
Jan 2, 2020
Novartis AG
Zhuoliang CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHARMACEUTICAL COMBINATION COMPRISING AN ALK INHIBITOR AND A SHP2 I...
Publication number
20190343836
Publication date
Nov 14, 2019
Novartis AG
Leila DARDAEI ALGHALANDIS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS AND COMPOSITIONS FOR INHBITING THE ACTIVITY OF SHP2
Publication number
20190185475
Publication date
Jun 20, 2019
Novartis AG
Jeffrey T. Bagdanoff
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1-PYRIDAZIN-/TRIAZIN-3-YL-PIPER(-AZINE)/IDINE/PYROLIDINE DERIVATIVE...
Publication number
20180362496
Publication date
Dec 20, 2018
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF SHP2
Publication number
20180251471
Publication date
Sep 6, 2018
Zhuoliang Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20180201623
Publication date
Jul 19, 2018
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF SHP2
Publication number
20180186770
Publication date
Jul 5, 2018
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1-(TRIAZIN-3-YL/PYRIDAZIN-3-YL)-PIPER(-AZINE)IDINE DERIVATIVES AND...
Publication number
20180065949
Publication date
Mar 8, 2018
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHARMACEUTICAL COMBINATIONS
Publication number
20180064709
Publication date
Mar 8, 2018
Nicole Buschmann
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
1-PYRIDAZIN-/TRIAZIN-3-YL-PIPER(-AZINE)/IDINE/PYROLIDINE DERIVATIVE...
Publication number
20170204080
Publication date
Jul 20, 2017
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-AZASPIROCYCLOALKANE SUBSTITUTED N-HETEROARYL COMPOUNDS AND COMPOS...
Publication number
20170015680
Publication date
Jan 19, 2017
Novartis AG
Christine Hiu-Tung Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMINOTHIAZOLES AND THEIR USES
Publication number
20170015704
Publication date
Jan 19, 2017
Novartis AG
Simon Bushell
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
1-(TRIAZIN-3-YL/PYRIDAZIN-3-YL)-PIPER(-AZINE)IDINE DERIVATIVES AND...
Publication number
20170001975
Publication date
Jan 5, 2017
Novartis AG
Zhuoliang Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMINOTHIAZOLES AND THEIR USES
Publication number
20140315790
Publication date
Oct 23, 2014
Simon Bushell
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMINOTHIAZOLES AND THEIR USES
Publication number
20140274878
Publication date
Sep 18, 2014
Novartis AG
Simon Bushell
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Macrocycles and Their Uses
Publication number
20130252883
Publication date
Sep 26, 2013
Roger Aki Fujimoto
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMINIOTHIAZOLES AND THEIR USES
Publication number
20130231275
Publication date
Sep 5, 2013
Novartis AG
Simon Bushell
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMINOTHIAZOLES AND THEIR USES
Publication number
20100267757
Publication date
Oct 21, 2010
Matthew J. LaMarche
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ANTIBACTERIAL COMPOUNDS AND PROCESSES FOR ITS PRODUCTION
Publication number
20100093615
Publication date
Apr 15, 2010
Matthew J. Lamarche
C07 - ORGANIC CHEMISTRY