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Michael Alan GREEN
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Easton, PA, US
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Patents Grants
last 30 patents
Information
Patent Grant
Organophosphorus-substituted compounds as c-MET inhibitors and ther...
Patent number
12,258,365
Issue date
Mar 25, 2025
Beta Pharma, Inc.
Don Zhang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pharmaceutical formulations of N-(2-(2-(dimethylamino)ethoxy)-4-met...
Patent number
12,187,707
Issue date
Jan 7, 2025
Beta Pharma, Inc.
Michael Nicholas Greco
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted 2-anilinopyrimidine derivatives as EGFR modulators
Patent number
11,414,401
Issue date
Aug 16, 2022
Beta Pharma Inc.
Jirong Peng
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pharmaceutical formulations of N-(2-(2-(dimethylamino) ethoxy)-4-me...
Patent number
11,180,478
Issue date
Nov 23, 2021
Beta Pharma, Inc.
Michael Nicholas Greco
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2-anilinopyrimidine derivatives as therapeutic agents for treatment...
Patent number
11,052,086
Issue date
Jul 6, 2021
Beta Pharma, Inc.
Michael Nicholas Greco
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pharmaceutical salts N-(2-(2-(dimethylamino)ethoxy)-4-methoxy-5-((4...
Patent number
10,844,045
Issue date
Nov 24, 2020
Beta Pharma, Inc.
Michael N. Greco
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 2-anilinopyrimidine derivatives as EGFR modulators
Patent number
10,590,111
Issue date
Mar 17, 2020
Beta Pharma, Inc.
Jirong Peng
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolo[1,5-a]pyrimidine-based compounds, compositions comprising...
Patent number
9,862,724
Issue date
Jan 9, 2018
Lexicon Pharmaceuticals, Inc.
Yingzhi Bi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolo[1,5-a]pyrimidine-based compounds, compositions comprising...
Patent number
9,403,832
Issue date
Aug 2, 2016
Lexicon Pharmaceuticals, Inc.
Yingzhi Bi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Imidazo[1,2-b]pyridazine-based compounds, compositions comprising t...
Patent number
8,969,565
Issue date
Mar 3, 2015
Lexicon Pharmaceuticals, Inc.
Yingzhi Bi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolo[1,5-a]pyrimidine-based compounds, compositions comprising...
Patent number
8,946,415
Issue date
Feb 3, 2015
Lexicon Pharmaceuticals, Inc.
Yingzhi Bi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Modulators of G protein-coupled receptor 88
Patent number
8,497,271
Issue date
Jul 30, 2013
Bristol-Myers Squibb Company
Yingzhi Bi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Modulators of G protein-coupled receptor 88
Patent number
8,426,414
Issue date
Apr 23, 2013
Bristol-Myers Squibb Company
Yingzhi Bi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Modulators of G protein-coupled receptor 88
Patent number
8,304,577
Issue date
Nov 6, 2012
Bristol-Myers Squibb Company
Carolyn Diane Dzierba
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Deacetylase inhibitors
Patent number
7,067,551
Issue date
Jun 27, 2006
Novartis AG
Stacy W Remiszewski
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Deacetylase inhibitors
Patent number
6,833,384
Issue date
Dec 21, 2004
Novartis AG
Stacy William Remiszewski
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Deacetylase inhibitors
Patent number
6,552,065
Issue date
Apr 22, 2003
Novartis AG
Stacy William Remiszewski
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
PYRIDOPYRIMIDINE DERIVATIVES AS KRAS INHIBITORS
Publication number
20240140948
Publication date
May 2, 2024
Beta Pharma, Inc.
Don Zhang
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDAZINE AND 1,2,4-TRIAZINE DERIVATIVES AS FGFR KINASE INHIBITORS
Publication number
20240002365
Publication date
Jan 4, 2024
Beta Pharma, Inc.
Don ZHANG
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDOPYRIMIDINE DERIVATIVES AS KRAS INHIBITORS
Publication number
20230099858
Publication date
Mar 30, 2023
Beta Pharma, Inc.
Don ZHANG
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TREATMENT OF EGFR MUTANT-RELATED CANCERS USING A COMBINATION OF EGF...
Publication number
20220347177
Publication date
Nov 3, 2022
Beta Pharma, Inc.
Michael Nicholas Greco
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PHARMACEUTICAL FORMULATIONS OF N-(2-(2-(DIMETHYLAMINO)ETHOXY)-4-MET...
Publication number
20220153726
Publication date
May 19, 2022
Beta Pharma, Inc.
Michael Nicholas Greco
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ORGANOPHOSPHORUS-SUBSTITUTED COMPOUNDS AS C-MET INHIBITORS AND THER...
Publication number
20220064194
Publication date
Mar 3, 2022
BETA PHARMA, INC.
Don ZHANG
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 2-ANILINOPYRIMIDINE DERIVATIVES AS EGFR MODULATORS
Publication number
20200216421
Publication date
Jul 9, 2020
Beta Pharma, Inc.
Jirong Peng
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHARMACEUTICAL FORMULATIONS OF N-(2-(2-(DIMETHYLAMINO) ETHOXY)-4-ME...
Publication number
20200131152
Publication date
Apr 30, 2020
Beta Pharma, Inc.
Michael Nicholas Greco
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2-ANILINOPYRIMIDINE DERIVATIVES AS THERAPEUTIC AGENTS FOR TREATMENT...
Publication number
20190365755
Publication date
Dec 5, 2019
Beta Pharma, Inc.
Michael Nicholas Greco
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PHARMACEUTICAL SALTS N-(2-(2-(DIMETHYLAMINO)ETHOXY)-4-METHOXY-5-((4...
Publication number
20190233399
Publication date
Aug 1, 2019
Beta Pharma, Inc.
Michael N. Greco
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 2-ANILINOPYRIMIDINE DERIVATIVES AS EGFR MODULATORS
Publication number
20170362203
Publication date
Dec 21, 2017
Beta Pharma, Inc.
Jirong Peng
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLO[1,5-a]PYRIMIDINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING...
Publication number
20170129896
Publication date
May 11, 2017
Lexion Pharmaceuticals, Inc.
Yingzhi BI
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLO[1,5-a]PYRIMIDINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING...
Publication number
20170081330
Publication date
Mar 23, 2017
Yingzhi BI
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDAZO[1,2-b]PYRIDAZINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING T...
Publication number
20170057964
Publication date
Mar 2, 2017
Yingzhi BI
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDAZO[1,2-b]PYRIDAZINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING T...
Publication number
20160024093
Publication date
Jan 28, 2016
Yingzhi BI
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLO[1,5-a]PYRIMIDINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING...
Publication number
20150183792
Publication date
Jul 2, 2015
Yingzhi BI
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDAZO[1,2-b]PYRIDAZINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING T...
Publication number
20150183791
Publication date
Jul 2, 2015
Yingzhi BI
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLO[1,5-a]PYRIMIDINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING...
Publication number
20150175610
Publication date
Jun 25, 2015
Yingzhi BI
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLO[1,5-a]PYRIMIDINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING...
Publication number
20130253194
Publication date
Sep 26, 2013
Yingzhi BI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMIDAZO[1,2-b]PYRIDAZINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING T...
Publication number
20130245021
Publication date
Sep 19, 2013
Yingzhi BI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Modulators of G Protein-Coupled Receptor 88
Publication number
20110251196
Publication date
Oct 13, 2011
Bristol-Myers Squibb Company and Lexicon Pharmaceuticals, Inc.
Carolyn Diane Dzierba
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Modulators of G Protein-Coupled Receptor 88
Publication number
20110251204
Publication date
Oct 13, 2011
Bristol-Myers Squibb Company and Lexicon Pharmaceuticals, Inc.
Yingzhi Bi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Modulators of G Protein-Coupled Receptor 88
Publication number
20110245264
Publication date
Oct 6, 2011
Bristol-Myers Squibb Company and Lexicon Pharmaceuticals, Inc.
Yingzhi Bi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
(R)-PHENYL(HETEROCYCLE)METHANOL-BASED COMPOUNDS, COMPOSITIONS COMPR...
Publication number
20090286820
Publication date
Nov 19, 2009
Joseph Barbosa
C07 - ORGANIC CHEMISTRY
Information
Patent Application
(S)-PHENYL(HETEROCYCLE)METHANOL-BASED COMPOUNDS, COMPOSITIONS COMPR...
Publication number
20090181992
Publication date
Jul 16, 2009
Joseph Barbosa
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DEACETYLASE INHIBITORS
Publication number
20080176849
Publication date
Jul 24, 2008
Stacy William Remiszewski
C07 - ORGANIC CHEMISTRY
Information
Patent Application
(R)-PHENYL(HETEROCYCLE)METHANOL-BASED COMPOUNDS, COMPOSITIONS COMPR...
Publication number
20080146596
Publication date
Jun 19, 2008
Joseph Barbosa
C07 - ORGANIC CHEMISTRY
Information
Patent Application
(S)-PHENYL(HETEROCYCLE)METHANOL-BASED COMPOUNDS, COMPOSITIONS COMPR...
Publication number
20080146600
Publication date
Jun 19, 2008
Joseph Barbosa
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SOLID FORMS OF (3'-CHLOROBIPHENYL-4-YL)(1-(PYRIMIDIN-2-YL)PIPERIDIN...
Publication number
20080076788
Publication date
Mar 27, 2008
Joseph BARBOSA
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Deacetylase inhibitors
Publication number
20060189674
Publication date
Aug 24, 2006
Stacy William Remiszewski
C07 - ORGANIC CHEMISTRY